97 SID26751614 148 SID26753737 173 SID26751593 250 SID26752101 273 SID29215044 322 SID26753729 323 8-Bromo-2,3,4,9-tetrahydro-1H-beta-carboline 324 8-Bromo-4,9-dihydro-3H-beta-carboline 325 (S)-2-{(S)-2-[(S)-2-({(R)-1-[6-Amino-2-(4-amino-butyl)-hexanoyl]-pyrrolidine-2-carbonyl}-amino)-3-(1H-indol-3-yl)-propionylamino]-3,3-dimethyl-butyrylamino}-4-methyl-pentanoic acid 343 5-Methoxy-4,9-dihydro-3H-beta-carboline 344 5-Methoxy-2,3,4,9-tetrahydro-1H-beta-carboline 351 7-Methoxy-2,3,4,9-tetrahydro-1H-beta-carboline 352 8-Methoxy-2,3,4,9-tetrahydro-1H-beta-carboline 364 (S)-2-{(S)-2-[(S)-2-({(R)-1-[(S)-6-Amino-2-((S)-2-amino-5-guanidino-pentylamino)-hexanoyl]-pyrrolidine-2-carbonyl}-amino)-3-(1H-indol-3-yl)-propionylamino]-3,3-dimethyl-butyrylamino}-4-methyl-pentanoic acid ethyl ester 365 (S)-2-{(S)-2-[(S)-2-({(R)-1-[(S)-6-Amino-2-((S)-2,6-diamino-hexylamino)-hexanoyl]-pyrrolidine-2-carbonyl}-amino)-3-(1H-indol-3-yl)-propionylamino]-3,3-dimethyl-butyrylamino}-4-methyl-pentanoic acid ethyl ester 382 (S)-2-{(S)-2-[(S)-2-{[(S)-1-((S)-2,6-Diamino-hexanoyl)-pyrrolidine-2-carbonyl]-amino}-3-(1H-indol-3-yl)-propionylamino]-3,3-dimethyl-butyrylamino}-4-methyl-pentanoic acid 388 5-Bromo-2,3,4,9-tetrahydro-1H-beta-carboline 390 (S)-2-{(S)-2-[(S)-2-({(R)-1-[5-Guanidino-2-(3-guanidino-propyl)-pentanoyl]-pyrrolidine-2-carbonyl}-amino)-3-(1H-indol-3-yl)-propionylamino]-3,3-dimethyl-butyrylamino}-4-methyl-pentanoic acid 391 2-{2-[(S)-2-({1-[(S)-6-Amino-2-((S)-(S)-2,6-diamino-hexylamino)-hexanoyl]-pyrrolidine-2-carbonyl}-amino)-3-(1H-indol-3-yl)-1-(S)-oxo-propylamino]-3-methyl-pentanoylamino}-4-methyl-pentanoic acid 392 (S)-2-{(S)-2-[(S)-2-({(R)-1-[(S)-6-Amino-2-(6-amino-hexylamino)-hexanoyl]-pyrrolidine-2-carbonyl}-amino)-3-(1H-indol-3-yl)-propionylamino]-3,3-dimethyl-butyrylamino}-4-methyl-pentanoic acid ethyl ester 416 (S)-2-{(S)-2-[(S)-2-({(R)-1-[5-Amino-2-(3-amino-propyl)-pentanoyl]-pyrrolidine-2-carbonyl}-amino)-3-(1H-indol-3-yl)-propionylamino]-3,3-dimethyl-butyrylamino}-4-methyl-pentanoic acid 417 Tryptoline 436 4-iodo-2,5-dimenthoxyamphetamine 448 (1S,2S,4S)-2-{2-[(S)-2-({1-[6-Amino-2-(2,6-diamino-hexylamino)-hexanoyl]-pyrrolidine-2-carbonyl}-amino)-3-(4-hydroxy-phenyl)-1-(S)-oxo-propylamino]-3,3-dimethyl-butyrylamino}-4-methyl-pentanoic acid 449 2-{2-[(S)-2-({1-[(S)-6-Amino-2-((S)-2,6-diamino-hexylamino)-hexanoyl]-pyrrolidine-2-carbonyl}-amino)-3-(1H-indol-3-yl)-1-(S)-oxo-propylamino]-3,3-dimethyl-butyrylamino}-4-methyl-pentanoic acid 450 (S)-2-{(S)-2-[(S)-2-({(R)-1-[(S)-6-Amino-2-((S)-2-amino-5-guanidino-pentylamino)-hexanoyl]-pyrrolidine-2-carbonyl}-amino)-3-(1H-indol-3-yl)-propionylamino]-3,3-dimethyl-butyrylamino}-4-methyl-pentanoic acid 452 8-Methoxy-4,9-dihydro-3H-beta-carboline 454 SID11110666 490 SID11114085 573 SID26752015 592 3,4-methylenedioxyamphetamine 601 Lysergic acid diethylamide 697 1,2,3,4-Tetrahydro-pyrazino[1,2-a]indole 699 7-Methoxy-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole 700 8-Methoxy-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole 789 Metoprolol 840 (R)-2-(2,5-Dimethoxy-phenyl)-1-methyl-ethylamine 892 SID26747465 923 Rapamycin 924 SID29216422 1011 8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-7-methoxy-1-methyl-1,4,5,6-tetrahydro-2H-benzo[e][1,4]diazocin-3-one 1022 SID26755647 1054 (2S,5S)-8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1-methyl-1,4,5,6-tetrahydro-2H-benzo[e][1,4]diazocin-3-one 1090 DOB 1279 SID26751696 1325 SID4252673 1333 Sulpiride 1370 SID26755283 1475 Cyclopentyl-(1-trifluoromethyl-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl)-amine 1564 SID26752115 1620 SID26751957 1847 [2-(5-Methoxy-1-methyl-1H-indol-3-yl)-ethyl]-dimethyl-amine 1924 N-formylmethionine-leucine-phenylalanine 1986 2-(2-ethyl-5-methoxy-1H-indol-3-yl)-N,N-dimethylethanamine 1994 SID26752240 2076 SID26732553 2150 3-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-1H-indole 2207 SID14719328 2214 SID26754232 2223 SID26755310 2232 SID11111436 2241 3,4-di(1H-indol-3-yl)-1H-pyrrole-2,5-dione 2246 SID11113847 2249 SID26751860 2261 SID26751524 2361 FAUC 113 2379 2-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b,e][1,4]diazepine 2384 10-methyl-3-phenyl-10H-benzo[4,5]imidazo[2,1-c][1,2,4]triazin-4-one 2395 2-(5-Bromo-furan-2-yl)-9-chloro-[1,2,4]triazolo[1,5-c]quinazolin-5-ylamine 2447 3-phenyl-10H-benzo[4,5]imidazo[2,1-c][1,2,4]triazin-4-one 2474 9-Chloro-2-furan-2-yl-6H-[1,2,4]triazolo[1,5-c]quinazolin-5-one 2488 8-chloro-5-methyl-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b,e][1,4]diazepine 2537 SID11111582 2557 (S)-2-[(S)-2-{3-[1-(2,6-Dichloro-benzyl)-3-pyrrolidin-1-ylmethyl-1H-indol-6-yl]-ureido}-3-(3,4-difluoro-phenyl)-propionylamino]-5-guanidino-pentanoic acid benzylamide 2569 3-(3,6,7,8,9,9a-Hexahydro-4H-quinolizin-1-yl)-phenol 2586 (S)-2-[(S)-2-{3-[1-(4-Fluoro-benzyl)-3-pyrrolidin-1-ylmethyl-1H-indol-6-yl]-ureido}-3-(4-methoxy-phenyl)-propionylamino]-5-guanidino-pentanoic acid benzylamide 2590 isomer-23-(Octahydro-indolizin-8-yl)-phenol 2591 3-(Octahydro-indolizin-8-yl)-phenol 2612 6-[Propyl-(2-thiophen-3-yl-ethyl)-amino]-5,6,7,8-tetrahydro-naphthalen-1-ol 2636 [3-(3-Chloro-phenyl)-5-hydroxy-7-methoxy-4-oxo-4H-quinolin-1-yl]-acetic acid methyl ester 2658 SID26752076 2687 3-(3-Chloro-phenyl)-5-hydroxy-7-methoxy-1-phenethyl-1H-quinolin-4-one 2693 3-(Octahydro-indolizin-8-yl)-phenol 2723 isomer-23-(Octahydro-quinolizin-1-yl)-phenol 2724 (S)-3-(1-propylpiperidin-3-yl)phenol 2725 L-158809 2728 1-(1-(2,6-dichlorobenzyl)-3-(pyrrolidin-1-ylmethyl)-1H-indol-6-yl)-3-((S)-1-((S)-1-(benzylamino)-5-guanidino-1-oxopentan-2-ylamino)-3-(4-methoxyphenyl)-1-oxopropan-2-yl)urea 2757 3-(3-Chloro-phenyl)-5-hydroxy-7-methoxy-chromen-4-one 2779 8-chloro-11-(4-methylpiperazin-1-yl)dibenzo[b,f][1,4]oxazepine 2782 SID29215546 2809 3-(3-Chloro-phenyl)-5,7-dihydroxy-1H-quinolin-4-one 2866 SID26752150 2867 3-(3-Chloro-phenyl)-5,7-dihydroxy-chromen-4-one 2915 5,6-Bis-p-tolylamino-isoindole-1,3-dione 2951 3-(3-Chloro-phenyl)-5-hydroxy-7-methoxy-1-methyl-1H-quinolin-4-one 2961 3-(3-Chloro-phenyl)-5-hydroxy-7-methoxy-1H-quinolin-4-one 2962 3'-Chloro-5,7-dimethoxyisoflavone 3012 SID26752764 3102 5-(4-Methoxy-phenylamino)-6-phenylamino-isoindole-1,3-dione 3372 1-[2-[1-[2-amino-2-(4-hydroxyphenyl)acetyl]-(2S)-tetrahydro-1H-2-pyrrolylcarboxamido]-3-phenyl-(2S)-propanoyl]-(2R)-tetrahydro-1H-2-pyrrolecarboxamide 3389 [Leu5]enkephalin 3485 1-(2,4,5-trimethoxyphenyl)propan-2-amine 3574 2-(4-Butyl-2,5-dimethoxy-phenyl)-1-methyl-ethylamine 3583 Racemic DOM 3587 SID11114236 3599 SID26751994 3635 3-(1-Propyl-piperidin-3-yl)-phenol 3666 SID26752086 3671 2-(2,5-Dimethoxy-4-propyl-phenyl)-1-methyl-ethylamine 3683 SID26755333 3700 1-(4-ethyl-2,5-dimethoxyphenyl)propan-2-amine 3702 2-(4-Ethoxy-2,5-dimethoxy-phenyl)-1-methyl-ethylamine 3710 1-(2,5-dimethoxyphenyl)propan-2-amine 3799 3-Ethyl-2-methyl-5-morpholin-4-ylmethyl-1,5,6,7-tetrahydro-indol-4-one 3854 SID26752261 3859 SID11113356 4149 SID26751756 4160 (S)-2-{(2S,3S)-2-[(S)-2-{N'-[2-((S)-1-{(S)-2-[(Adamantane-1-carbonyl)-amino]-6-amino-hexanoyl}-pyrrolidin-2-yl)-2-oxo-ethyl]-hydrazino}-3-(4-hydroxy-phenyl)-propionylamino]-3-methyl-pentanoylamino}-4-methyl-pentanoic acid 4181 SID26751769 4358 (S)-2-{(2S,3S)-2-[(S)-2-{(E)-3-[(S)-1-((S)-6-Amino-2-tert-butoxycarbonylamino-hexanoyl)-pyrrolidin-2-yl]-3-oxo-propenylamino}-3-(4-hydroxy-phenyl)-propionylamino]-3-methyl-pentanoylamino}-4-methyl-pentanoic acid 4392 (S)-2-{(S)-2-[(S)-2-{[1-((1S,6S)-2,6-Diamino-hexanoyl)-pyrrolidine-2-carbonyl]-amino}-3-(4-hydroxy-phenyl)-propionylamino]-3-methyl-pentanoylamino}-4-methyl-pentanoic acid 4393 (S)-2-{(S)-2-[(S)-2-({1-[(S)-5-Amino-2-((S)-tert-butoxycarbonylamino)-pentanoyl]-pyrrolidine-2-carbonyl}-amino)-3-(4-hydroxy-phenyl)-propionylamino]-3-methyl-pentanoylamino}-4-methyl-pentanoic acid 4394 (S)-2-{(S)-2-[(S)-2-{[1-((1S,3S)-6-Amino-2-tert-butoxycarbonylamino-hexanoyl)-pyrrolidine-2-carbonyl]-amino}-3-(4-hydroxy-phenyl)-propionylamino]-3-methyl-pentanoylamino}-4-methyl-pentanoic acid 4395 (S)-2-((2S,3S)-2-{N'-[(S)-3-[((S)-1-{(S)-2-[(Adamantane-1-carbonyl)-amino]-6-amino-hexanoyl}-pyrrolidine-2-carbonyl)-amino]-4-(4-hydroxy-phenyl)-2-oxo-butyl]-hydrazino}-3-methyl-pentanoylamino)-4-methyl-pentanoic acid 4407 (S)-2-((2S,3S)-2-{N'-[(S)-3-[((S)-1-{(S)-3-[(Adamantane-1-carbonyl)-amino]-7-amino-2-oxo-heptylamino}-pyrrolidine-2-carbonyl)-amino]-4-(4-hydroxy-phenyl)-2-oxo-butyl]-hydrazino}-3-methyl-pentanoylamino)-4-methyl-pentanoic acid 4408 (S)-2-{(2S,3S)-2-[(S)-2-(N'-{2-[(S)-1-((S)-5-Amino-2-tert-butoxycarbonylamino-pentanoyl)-pyrrolidin-2-yl]-2-oxo-ethyl}-hydrazino)-3-(4-hydroxy-phenyl)-propionylamino]-3-methyl-pentanoylamino}-4-methyl-pentanoic acid 4420 4-(1-Methyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)-benzenesulfonic acid 3-nitro-phenyl ester 4464 4-(1-Butyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)-benzenesulfonic acid 4465 4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-benzenesulfonic acid 3-nitro-phenyl ester 4472 4-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-benzenesulfonic acid 3-nitro-phenyl ester 4485 SID29217615 4486 4-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-benzenesulfonic acid 4496 Dronabinol 4542 SID11110671 4543 1-Butyl-8-phenyl-3,7-dihydro-purine-2,6-dione 4544 8-Phenyl-1-propyl-3,7-dihydro-purine-2,6-dione 4545 1-Methyl-8-phenyl-3,7-dihydro-purine-2,6-dione 4557 SID26753527 4581 4-(1-Methyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)-benzenesulfonic acid 4-nitro-phenyl ester 4584 SID26753787 4593 4-(1-Butyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)-benzenesulfonic acid 4-nitro-phenyl ester 4594 4-(1,3-Dimethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)-benzenesulfonic acid 4-nitro-phenyl ester 4601 4-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-benzenesulfonic acid 4-nitro-phenyl ester 4602 4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-benzenesulfonic acid 4-nitro-phenyl ester 4615 4-(1-Butyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)-benzenesulfonic acid 3-nitro-phenyl ester 4634 SID26751487 4671 SID11113767 4672 SID26719717 4686 SID26755017 4721 (-)-(S)-N-((1-ethylpyrrolidin-2-yl)methyl)-2-hydroxy-3-iodo-6-methoxybenzamide 4726 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-3-methyl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 4731 4-(1,3-Dimethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)-benzenesulfonic acid 3-nitro-phenyl ester 4750 (6aR,10aR)-6,6,9-trimethyl-3-pentyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol 4778 SID11113793 5183 1-(4-Bromo-phenyl)-3-{2-[3-(3-isopropoxy-phenyl)-4-oxo-3,4-dihydro-quinazolin-2-yl]-ethyl}-urea 5185 3-(benzo[d][1,3]dioxol-5-yl)-5-hydroxy-5-(4-methoxyphenyl)-4-(3,4,5-trimethoxybenzyl)furan-2(5H)-one 5195 1-(4-Bromo-phenyl)-3-[3-(3-isopropoxy-phenyl)-4-oxo-3,4-dihydro-quinazolin-2-ylmethyl]-urea 5306 1H-Indole-2-carboxylic acid (3-phenyl-allyl)-amide 5313 1H-Indole-2-carboxylic acid (3,3-diphenyl-propyl)-amide 5314 3,4-Dichloro-N-(3,3-diphenyl-allyl)-benzamide 5318 Naphthalene-2-carboxylic acid (3,3-diphenyl-allyl)-amide 5324 1H-Indole-2-carboxylic acid (3,3-diphenyl-allyl)-amide 5325 Quinoline-2-carboxylic acid (3,3-diphenyl-allyl)-amide 5341 Naphthalene-1-carboxylic acid (3,3-diphenyl-allyl)-amide 5353 1-(3,3-Diphenyl-allyl)-3-m-tolyl-urea 5359 1H-Indole-2-carboxylic acid [3,3-bis-(4-chloro-phenyl)-allyl]-amide 5371 (R)-1-(1-methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-m-tolylurea 5443 6-Oxo-heptanoic acid (2-{2-[4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetylamino}-ethyl)-amide 5459 7-(2-{2-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetylamino}-ethylcarbamoyl)-heptanoic acid 2,5-dioxo-pyrrolidin-1-yl ester 5480 1-(4-Chloro-phenyl)-3-(3-pentyl-oct-2-enyl)-urea 5495 1-(4-Chloro-phenyl)-3-(3,3-diphenyl-allyl)-urea 5508 2-(4-Amino-phenyl)-N-(2-{2-[4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetylamino}-ethyl)-acetamide 5511 1-(4-Chloro-phenyl)-3-(2-diphenylamino-ethyl)-urea 5526 1-(4-Chloro-phenyl)-3-(4,4-diphenyl-but-3-enyl)-urea 5535 SID29215529 5536 4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-butyric acid 5579 4-Bromomethyl-N-(2-{2-[4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetylamino}-ethyl)-benzamide 5653 2-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-N-[2-(3-pentafluorophenyl-thioureido)-ethyl]-acetamide 5654 4-(2,5-Dioxo-2,5-dihydro-pyrrol-1-yl)-N-[(2-{2-[4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetylamino}-ethylcarbamoyl)-methyl]-butyramide 5704 2-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-N-{2-[3-(4-isothiocyanato-phenyl)-thioureido]-ethyl}-acetamide 5712 2-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-N-(2-oxo-ethyl)-acetamide 5797 SID26751564 5884 SID26751928 5925 SID11111755 5931 2-Piperazin-1-yl-phenol 5970 SID26752322 6005 Morphine 6095 1-(2-Chloro-phenyl)-piperazine 6149 2-{2-[4-(5-Fluoro-2-oxo-2,3-dihydro-benzoimidazol-1-yl)-piperidin-1-yl]-ethyl}-2,3,4,5-tetrahydro-benzo[c]azepin-1-one 6182 SID26756537 6216 SID26751621 6291 (2-Benzofuran-6-yl-ethyl)-((R)-5-methoxy-1,2,3,4-tetrahydro-naphthalen-1-ylmethyl)-methyl-amine 6358 SID11111349 6446 (2-Benzo[1,3]dioxol-5-yl-ethyl)-(5-methoxy-1,2,3,4-tetrahydro-naphthalen-1-ylmethyl)-methyl-amine 6579 Chloroquine 6593 Rauwolscine 6641 3-Hydroxy-2-phenyl-quinoline-4-carboxylic acid ((R)-1-phenyl-propyl)-amide 6656 3-Dimethylaminomethyl-2-phenyl-quinoline-4-carboxylic acid ((R)-1-phenyl-propyl)-amide 6686 1-{4-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-benzyl}-piperidin-2-one 6706 SID26758000 6713 mazapertine 6720 1-{2-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-benzyl}-piperidin-2-one 6753 {2-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-phenyl}-piperidin-1-yl-methanone 6759 3-Amino-2-phenyl-quinoline-4-carboxylic acid ((R)-1-phenyl-propyl)-amide 6760 talnetant 6772 SID26751604 6837 2-Phenyl-quinoline-4-carboxylic acid ((R)-1-phenyl-propyl)-amide 6841 3-(2-Hydroxy-ethoxy)-2-phenyl-quinoline-4-carboxylic acid ((R)-1-phenyl-propyl)-amide 6870 1-{3-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-benzyl}-piperidin-2-one 6902 Naloxone 6964 3-Ethyl-2-phenyl-quinoline-4-carboxylic acid ((R)-1-phenyl-propyl)-amide 6965 3-Benzo[1,3]dioxol-5-yl-1-benzo[1,3]dioxol-5-ylmethyl-5-propoxy-1H-indole-2-carboxylic acid 7024 1-{5-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-1-methyl-1H-pyrrol-2-ylmethyl}-piperidin-2-one 7025 {4-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-phenyl}-piperidin-1-yl-methanone 7056 [2-Phenyl-4-((R)-1-phenyl-propylcarbamoyl)-quinolin-3-yloxy]-acetic acid 7065 SID26755307 7078 3-Methyl-2-phenyl-quinoline-4-carboxylic acid ((R)-1-phenyl-propyl)-amide 7159 3-Benzo[1,3]dioxol-5-yl-1-benzo[1,3]dioxol-5-ylmethyl-5,6-dimethoxy-1H-indole-2-carboxylic acid 7389 [3-((E)-6-Hydroxy-undec-4-enyl)-phenoxy]-acetic acid 7398 [6-((E)-4-Hydroxy-non-2-enyl)-5,6,7,8-tetrahydro-naphthalen-1-yloxy]-acetic acid 7452 [6-((E)-4-Hydroxy-5-phenyl-pent-2-enyl)-5,6,7,8-tetrahydro-naphthalen-1-yloxy]-acetic acid 7459 [6-((E)-5,5-Diphenyl-pent-2-enyl)-5,6,7,8-tetrahydro-naphthalen-1-yloxy]-acetic acid 7480 [3-(4-Benzhydryloxyimino-butyl)-phenoxy]-acetic acid 7493 [6-(2-Benzhydryloxyimino-ethyl)-5,6,7,8-tetrahydro-naphthalen-1-yloxy]-acetic acid 7494 (E)-5-((3aS,5R,6aS)-5-hydroxy-6-((3S,E)-3-hydroxy-4-methyloct-1-en-6-ynyl)-hexahydropentalen-2(1H)-ylidene)pentanoic acid 7512 [6-((Z)-5,5-Diphenyl-pent-2-enyl)-5,6,7,8-tetrahydro-naphthalen-1-yloxy]-acetic acid 7513 [6-((E)-5-Phenyl-pent-2-enyl)-5,6,7,8-tetrahydro-naphthalen-1-yloxy]-acetic acid 7530 [5-(3-Benzhydryloxyimino-propyl)-5,6,7,8-tetrahydro-naphthalen-1-yloxy]-acetic acid 7547 [5-((E)-5-Hydroxy-dec-3-enyl)-5,6,7,8-tetrahydro-naphthalen-1-yloxy]-acetic acid 7646 2,2-diphenylethanamine 7714 SID26753640 7736 SID26751627 7958 1-Allyl-3-methyl-8-phenyl-3,7-dihydro-purine-2,6-dione 7982 (R)-N-((S)-1-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)-3-methylbutan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 7988 [6-(2-Benzhydryloxyimino-pentyl)-5,6,7,8-tetrahydro-naphthalen-1-yloxy]-acetic acid 7995 N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethylamino}-butyl)-phenyl]-ethylaminosulfonamide 8045 3-(4-Hydroxy-phenyl)-N-{1-[4-(3-hydroxy-phenyl)-3,4-dimethyl-piperidin-1-ylmethyl]-2-methyl-propyl}-propionamide 8074 3-Benzo[1,3]dioxol-5-yl-4-benzyl-5-methoxy-5-(4-methoxy-phenyl)-5H-furan-2-one 8089 N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-2,3-dihydro-1H-indol-3-yl]-ethylamino}-butyl)-phenyl]-methanesulfonamide 8090 (3R)-7-Hydroxy-N-[(1S)-1-{[(3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl-1-piperidinyl]methyl}-2-methylpropyl)-1,2,3,4-tetrahydro-3-isoquinolinecarboxamide 8106 N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethylamino}-butyl)-phenyl]-benzenesulfonamide 8110 ((S)-6-{2-[(E)-Benzhydryloxyimino]-propyl}-5,6,7,8-tetrahydro-naphthalen-1-yloxy)-acetic acid 8118 (5-{3-[(E)-Benzhydryloxyimino]-hexyl}-5,6,7,8-tetrahydro-naphthalen-1-yloxy)-acetic acid 8122 N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethylamino}-butyl)-phenyl]-methylaminosulfonamide 8123 1-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethylamino}-butyl)-phenyl]-3-ethyl-urea 8130 Alprostadil 8134 Propane-2-sulfonic acid [4-(4-{2-[2-(3,5-dimethyl-phenyl)-1H-indol-3-yl]-ethylamino}-butyl)-phenyl]-amide 8137 (6-{2-[(E)-Benzhydryloxyimino]-propyl}-5,6,7,8-tetrahydro-naphthalen-1-yloxy)-acetic acid 8151 1-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohepta[1,2-b]pyridin-11-ylidene)-piperidin-1-yl]-ethanone 8152 4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethylamino}-butyl)-benzenesulfonamide 8160 1-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethylamino}-butyl)-phenyl]-3-methyl-urea 8169 4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethylamino}-butyl)-phenylamine 8170 ((R)-6-{2-[(E)-Benzhydryloxyimino]-propyl}-5,6,7,8-tetrahydro-naphthalen-1-yloxy)-acetic acid 8172 (6-{2-[(E)-Benzyloxyimino]-propyl}-5,6,7,8-tetrahydro-naphthalen-1-yloxy)-acetic acid 8173 Ethanesulfonic acid [4-(4-{2-[2-(3,5-dimethyl-phenyl)-1H-indol-3-yl]-ethylamino}-butyl)-phenyl]-amide 8205 {2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethyl}-[4-(4-fluoro-phenyl)-butyl]-amine 8209 Agomelatine 8232 4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethylamino}-butyl)-phenol 8239 8-(4-Amino-phenyl)-1,3-dimethyl-3,7-dihydro-purine-2,6-dione 8242 {2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethyl}-[4-(4-nitro-phenyl)-butyl]-amine 8243 4-(1,3-Dimethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)-benzoic acid 8248 N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethylamino}-butyl)-phenyl]-acetamide 8256 (6-{2-[(E)-Benzhydryloxyimino]-butyl}-5,6,7,8-tetrahydro-naphthalen-1-yloxy)-acetic acid 8284 3-(1,3-Dimethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)-benzoic acid 8328 N-Methyl-N-(4-pyrrolidin-1-yl-but-2-ynyl)-acetamide 8357 8-(2-Amino-phenyl)-1,3-dimethyl-3,7-dihydro-purine-2,6-dione 8407 1,3-Dimethyl-8-nitro-3,7-dihydro-purine-2,6-dione 8414 8-(3-Amino-phenyl)-1,3-dimethyl-3,7-dihydro-purine-2,6-dione 8531 SID11113334 8535 SID17401580 8543 SID26752014 8548 SID11110669 8556 8-(2-Amino-4-chloro-phenyl)-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8580 8-(3-Hydroxy-phenyl)-1,3-dimethyl-3,7-dihydro-purine-2,6-dione 8635 8-{4-[(5-Methoxy-chroman-3-yl)-propyl-amino]-butyl}-8-aza-spiro[4.5]decane-7,9-dione 8636 (+) 8-{4-[5-methoxyspiro[3,4-dihydro-2H-chromene-3,2'-(tetrahydro-1'H-pyrrole)]-1-yl]butyl}-8-azaspiro[4.5]decane-7,9-dione 8724 (3aR,9aS)-1-allyl-2,3,3a,4,9,9a-hexahydro-1H-benzo[f]indol-5-ol 8725 (3aS,9aR)-1-allyl-2,3,3a,4,9,9a-hexahydro-1H-benzo[f]indol-5-ol 8738 SID26747541 8786 (3aR,9aS)-1-propyl-2,3,3a,4,9,9a-hexahydro-1H-benzo[f]indol-5-ol 8787 (3aS,9aR)-1-propyl-2,3,3a,4,9,9a-hexahydro-1H-benzo[f]indol-5-ol 8828 (2 beta-methyl) 8-Methoxy-2-methyl-1-propyl-2,3,3a,4,9,9a-hexahydro-1H-benzo[f]indole 8910 SID26753352 8960 (3aS,9aR)-5-methoxy-1-propyl-2,3,3a,4,9,9a-hexahydro-1H-benzo[f]indole 9128 6-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-ol 9133 (8-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-dipropyl-amine 9203 (5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-dipropyl-amine 9277 SID26753571 9826 (2-Amino-3-methyl-phenyl)-{4-[4-(3-chloro-benzenesulfonyl)-benzyl]-[1,4']bipiperidinyl-1'-yl}-methanone 9879 (2-Amino-3-methyl-phenyl)-{4-[4-(propane-2-sulfonyl)-benzyl]-[1,4']bipiperidinyl-1'-yl}-methanone 9889 3-Amino-2-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]-propylsulfanyl}-3,5,6,7-tetrahydro-cyclopenta[4,5]thieno[2,3-d]pyrimidin-4-one 9894 1-{3-[5-(2-Ethoxy-phenyl)-[1,3,4]thiadiazol-2-ylsulfanyl]-propyl}-4-(2-methoxy-phenyl)-piperazine 9898 3-Amino-6-ethyl-2-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]-propylsulfanyl}-3H-thieno[2,3-d]pyrimidin-4-one 9919 [4-(4-Isopropylsulfanyl-benzyl)-[1,4']bipiperidinyl-1'-yl]-naphthalen-1-yl-methanone 9926 4'-(2-Butyl-4-oxo-1,3-diaza-spiro[4.4]non-1-en-3-ylmethyl)-2'-(3,3-dimethyl-2-oxo-pyrrolidin-1-ylmethyl)-biphenyl-2-sulfonic acid (3,4-dimethyl-isoxazol-5-yl)-amide 9931 2-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propylsulfanyl}-5,6-dimethyl-thieno[2,3-d]pyrimidin-4-ylamine 9932 3-Amino-2-[3-(4-pyrimidin-2-yl-piperazin-1-yl)-propylsulfanyl]-3H-thieno[2,3-d]pyrimidin-4-one 9938 3-Amino-5,6-dimethyl-2-{3-[4-(2-nitro-phenyl)-piperazin-1-yl]-propylsulfanyl}-3H-thieno[2,3-d]pyrimidin-4-one 9946 3-Amino-5,6-dimethyl-2-[3-(4-pyrimidin-2-yl-piperazin-1-yl)-propylsulfanyl]-3H-thieno[2,3-d]pyrimidin-4-one 9955 3-Amino-2-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]-propylsulfanyl}-5,6-dimethyl-3H-thieno[2,3-d]pyrimidin-4-one 9956 3-Amino-2-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]-propylsulfanyl}-6-propyl-3H-thieno[2,3-d]pyrimidin-4-one 9970 3-Amino-6-ethyl-2-[3-(4-pyrimidin-2-yl-piperazin-1-yl)-propylsulfanyl]-3H-thieno[2,3-d]pyrimidin-4-one 9994 3-Amino-2-{3-[4-(2-nitro-phenyl)-piperazin-1-yl]-propylsulfanyl}-3H-thieno[2,3-d]pyrimidin-4-one 9996 1-{3-[5-(2-Ethoxy-phenyl)-[1,3,4]thiadiazol-2-ylsulfanyl]-propyl}-4-(2-nitro-phenyl)-piperazine 10001 3-Amino-6-ethyl-2-{3-[4-(2-nitro-phenyl)-piperazin-1-yl]-propylsulfanyl}-3H-thieno[2,3-d]pyrimidin-4-one 10018 N-{3-[4-(2-Isopropoxy-phenyl)-piperazin-1-yl]-propyl}-2-(2-oxo-piperidin-1-yl)-acetamide 10028 N-{2-[4-(2-Isopropoxy-phenyl)-piperazin-1-yl]-ethyl}-N-methyl-2-(2-oxo-piperidin-1-yl)-acetamide 10030 1-[4-(2-Isopropoxy-phenyl)-piperazin-1-yl]-5-(2-oxo-piperidin-1-yl)-pentane-2,4-dione 10038 1-Methyl-4-((S)-8-methylsulfanyl-10,11-dihydro-dibenzo[b,f]thiepin-10-yl)-piperazine 10046 N-{2-[4-(4-Fluoro-2-isopropoxy-phenyl)-piperazin-1-yl]-ethyl}-2-(2-oxo-piperidin-1-yl)-acetamide 10085 3-Amino-2-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]-propylsulfanyl}-3H-thieno[2,3-d]pyrimidin-4-one 10116 1-{(E)-5-[4-(2-Isopropoxy-phenyl)-piperazin-1-yl]-2-oxo-pent-3-enyl}-piperidin-2-one 10124 1-{4-Hydroxy-5-[4-(2-isopropoxy-phenyl)-piperazin-1-yl]-2-oxo-pentyl}-piperidin-2-one 10184 1-Methyl-5-(3-methyl-[1,2,4]oxadiazol-5-yl)-1,2,3,6-tetrahydro-pyridine 10249 (2-Oxo-piperidin-1-yl)-acetic acid 2-[4-(2-isopropoxy-phenyl)-piperazin-1-yl]-ethyl ester 10261 N-(2-{4-[4-Fluoro-2-(2,2,2-trifluoro-ethoxy)-phenyl]-piperazin-1-yl}-ethyl)-2-(2-oxo-piperidin-1-yl)-acetamide 10311 N-{2-[4-(2-Isopropoxy-phenyl)-piperazin-1-yl]-ethyl}-2-(2-oxo-azepan-1-yl)-acetamide 10312 N-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyl}-2-(2-oxo-piperidin-1-yl)-acetamide 10313 N-{2-[4-(2-Isopropoxy-phenyl)-piperazin-1-yl]-ethyl}-2-(2-oxo-piperidin-1-yl)-acetamide 10340 1-({2-[4-(2-Isopropoxy-phenyl)-piperazin-1-yl]-ethylcarbamoyl}-methyl)-5-oxo-pyrrolidine-2-carboxylic acid ethyl ester 10346 N-[2-(1H-Imidazol-4-yl)-ethyl]-4-phenyl-butyramide 10347 N-[2-(1H-Imidazol-4-yl)-ethyl]-3-phenyl-propionamide 10348 N-[2-(1H-Imidazol-4-yl)-ethyl]-4,4-diphenyl-butyramide 10382 N-[2-(1H-Imidazol-4-yl)-ethyl]-2-phenyl-acetamide 10383 SID26751775 10454 1-[4-(1H-Imidazol-4-yl)-butyl]-3-methyl-thiourea 10469 4-(1H-Imidazol-4-yl)-N-[2-(1H-imidazol-4-yl)-ethyl]-butyramide 10488 5-Phenyl-pentanoic acid [2-(1H-imidazol-4-yl)-ethyl]-amide 10521 N-[2-(1H-Imidazol-4-yl)-ethyl]-4-pyridin-2-yl-butyramide 10584 SID26756614 10661 SID26751558 10686 4-Cyclohexyl-N-[2-(1H-imidazol-4-yl)-ethyl]-butyramide 10687 [2-(1H-Imidazol-4-yl)-ethyl]-(4-phenyl-butyl)-amine 10747 SID11111716 10755 3,4-Dichloro-N-methyl-N-[(R)-1-methyl-3-(4-methyl-piperidin-1-yl)-propyl]-benzenesulfonamide 10762 Naphthalene-1-sulfonic acid methyl-[(R)-1-methyl-3-(4-methyl-piperidin-1-yl)-propyl]-amide 10800 2a-[3-(4-Phenyl-piperazin-1-yl)-propyl]-2a,3,4,5-tetrahydro-1H-benzo[cd]indol-2-one 10801 4'-(2-Butyl-4-chloro-5-hydroxymethyl-imidazol-1-ylmethyl)-biphenyl-2-carboxylic acid 10841 3,N-Dimethyl-N-[(R)-1-methyl-3-(4-methyl-piperidin-1-yl)-propyl]-benzenesulfonamide 10842 4,5-Dibromo-thiophene-2-sulfonic acid methyl-[(R)-1-methyl-3-(4-methyl-piperidin-1-yl)-propyl]-amide 10846 Naphthalene-1-sulfonic acid methyl-[1-methyl-3-(3-methyl-piperidin-1-yl)-propyl]-amide 10876 Naphthalene-1-sulfonic acid methyl-[(S)-1-methyl-3-((R)-3-methyl-piperidin-1-yl)-propyl]-amide 10905 Naphthalene-1-sulfonic acid methyl-[(R)-1-methyl-3-((S)-3-methyl-piperidin-1-yl)-propyl]-amide 10912 Naphthalene-1-sulfonic acid methyl-[(R)-1-methyl-3-((R)-3-methyl-piperidin-1-yl)-propyl]-amide 10956 4-Methyl-1-{2-[(R)-1-(toluene-3-sulfonyl)-pyrrolidin-2-yl]-ethyl}-piperidine 10959 SID26756534 10969 (6aR,9R)-5-Bromo-7-methyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid diethylamide 11005 SID26751603 11015 SID11111401 11029 3,4-Dibromo-N-methyl-N-[(R)-1-methyl-3-(4-methyl-piperidin-1-yl)-propyl]-benzenesulfonamide 11248 Tetradecanoic acid (2S,3R)-2-hydroxymethyl-5-oxo-tetrahydro-furan-3-yl ester 11356 Hydroxy-diphenyl-acetic acid 1-aza-bicyclo[2.2.2]oct-3-yl ester (QNB) 11601 Acetic acid (2S,3R)-2-hydroxymethyl-5-oxo-4-tetradecylidene-tetrahydro-furan-3-yl ester 11740 Acetic acid (2S,3R)-2-hydroxymethyl-5-oxo-4-tetradecylidene-tetrahydro-furan-3-yl ester 11747 [2-Methyl-1-(2-morpholin-4-yl-ethyl)-1H-indol-3-yl]-naphthalen-1-yl-methanone 11748 [1-(2-Morpholin-4-yl-ethyl)-1H-indol-3-yl]-naphthalen-1-yl-methanone 11805 Dicarba-Closo-Dodecaborane analogue 11861 (4-Methoxy-phenyl)-[1-(2-morpholin-4-yl-ethyl)-1H-indol-3-yl]-methanone 11898 {1-[2-(2-Hydroxy-morpholin-4-yl)-ethyl]-2-methyl-1H-indol-3-yl}-naphthalen-1-yl-methanone 11911 Benzo[b]thiophen-3-yl-[2-methyl-1-(2-morpholin-4-yl-ethyl)-1H-indol-3-yl]-methanone 11929 Dicarba-Closo-Dodecaborane analogue 11985 SID26756872 12055 SID26753228 12118 (S)-4-[(S)-2-Acetylamino-3-(4-phosphonooxy-phenyl)-propionylamino]-4-[(3-cyclohexyl-propyl)-methyl-carbamoyl]-butyric acid 12225 SID26751883 12494 SID26754331 12837 3-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-1-methyl-5-phenyl-1H-thieno[2,3-d]pyrimidine-2,4-dione 12850 1-{[(2R)-3-(benzyloxy)-1-{1-methanesulfonyl-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}-1-oxopropan-2-yl]carbamoyl}-1-methylethan-1-aminium 12872 SID26752024 12878 5-(5-Bromo-2-oxo-1,2-dihydro-indol-3-ylidenemethyl)-2,4-dimethyl-1H-pyrrole-3-carboxylic acid (2-diethylamino-ethyl)-amide 12886 3-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-5-m-tolyl-1H-thieno[2,3-d]pyrimidine-2,4-dione 12902 3-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyl}-5-phenyl-1H-thieno[2,3-d]pyrimidine-2,4-dione 12911 3-((3,5-dimethyl-1H-pyrrol-2-yl)methylene)indolin-2-one 12912 3-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-1H-thieno[2,3-d]pyrimidine-2,4-dione 12922 3-(2,4-dimethyl-5-((2-oxoindolin-3-ylidene)methyl)-1H-pyrrol-3-yl)propanoic acid 12928 (S)-2-((2S,5S,11bR)-2-(benzyloxycarbonyl)-3-oxo-2,3,5,6,11,11b-hexahydro-1H-indolizino[8,7-b]indole-5-carboxamido)-3-phenylpropanoic acid 12930 3-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-6-methyl-5-phenyl-1H-thieno[2,3-d]pyrimidine-2,4-dione 12964 (S)-2-((2R,5R,11bS)-2-(benzyloxycarbonyl)-3-oxo-2,3,5,6,11,11b-hexahydro-1H-indolizino[8,7-b]indole-5-carboxamido)-3-phenylpropanoic acid 12987 5-(5-Fluoro-2-oxo-1,2-dihydro-indol-3-ylidenemethyl)-2,4-dimethyl-1H-pyrrole-3-carboxylic acid (1-methyl-piperidin-4-ylmethyl)-amide 12991 3-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-6-phenyl-1H-thieno[2,3-d]pyrimidine-2,4-dione 13013 4-Fluoro-N-[2-(5-methoxy-1,3,4,4a,9,9a-hexahydro-indeno[2,1-c]pyridin-2-yl)-ethyl]-benzamide 13036 (1R,2R)-2-(3H-Imidazol-4-yl)-cyclopropylamine 13037 (alphaS,betaR)(2-Chloro-4-{2-[2-hydroxy-2-(4-hydroxy-phenyl)-1-methyl-ethylamino]-ethyl}-phenoxy)-acetic acid 13048 SID26758053 13050 (1S,2S)-2-(3H-Imidazol-4-yl)-cyclopropylamine 13109 3-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-5-phenyl-1H-thieno[2,3-d]pyrimidine-2,4-dione 13118 2-[3-(5-Methoxy-1,3,4,4a,9,9a-hexahydro-indeno[2,1-c]pyridin-2-yl)-propyl]-1,1-dioxo-1,2-dihydro-1lambda*6*-benzo[d]isothiazol-3-one 13121 2-[4-(5-Methoxy-1,3,4,4a,9,9a-hexahydro-indeno[2,1-c]pyridin-2-yl)-butyl]-1,1-dioxo-1,2-dihydro-1lambda*6*-benzo[d]isothiazol-3-one 13139 2-(4-tert-Butyl-phenyl)-4,5-dihydro-1H-imidazole 13284 (7-Methyl-4,6,6a,7,8,9,10,10a-octahydro-indolo[4,3-fg]quinolin-9-ylmethyl)-carbamic acid benzyl ester 13364 1N-[1-benzyl-2-[5-carbamoyl-(5S)-dihydro-1H-1-pyrrolyl]-2-oxo-(1S)-ethylcarbamoylmethyl]-2-[1-amino-2-(4-hydroxyphenyl)-(1S)-ethylcarboxamido]-4-methylsulfanyl-(2S)-butanamide 13365 2-[1-[1-[1-amino-2-(4-hydroxyphenyl)-(1S)-ethylcarboxamido]-(1S)-ethylcarboxamidomethyl(methyl)carboxamido]-2-phenyl-(1S)-ethylcarboxamido]-4-methylsulfinyl-(2S)-butanoic acid 13431 2-Amino-N-(1-{[(1,3-dimethyl-butylcarbamoyl)-methyl]-carbamoyl}-ethyl)-3-(4-hydroxy-phenyl)-propionamide 13432 [Met5]-enkephalin 13433 2-(1-{1-[1-amino-2-(4-hydroxyphenyl)ethylcarboxamidomethylcarboxamidomethylcarboxamido]-2-phenylethylcarboxamido}-3-methylsulfanylpropylcarboxamido)-3-hydroxy-(3R)-butanoic acid 13434 2-[1-(1-{1-[1-amino-2-(4-hydroxyphenyl)ethylcarboxamido]-2-hydroxyethylcarboxamidomethylcarboxamido}-2-phenylethylcarboxamido)-3-methylbutylcarboxamido]-3-hydroxy-(3R)-butanoic acid 13559 2-{1-[1-{1-[1-amino-2-(4-hydroxyphenyl)ethylcarboxamido]ethylcarboxamidomethylcarboxamido}-2-phenyl-(1S)-ethylcarboxamido]-3-methylsulfanylpropylcarboxamido}-3-hydroxy-(3R)-butanoic acid 13560 1N-(1,3-dimethylbutylcarbamoylmethyl)-2-[1-amino-2-(4-hydroxyphenyl)-(1S)-ethylcarboxamido]-4-methylsulfanyl-(2S)-butanamide 13693 SID26756547 13739 N-[2-(7-{5-[8-(2-Acetylamino-ethyl)-naphthalen-2-yloxy]-pentyloxy}-naphthalen-1-yl)-ethyl]-acetamide 13775 N-[2-(7-{8-[8-(2-Acetylamino-ethyl)-naphthalen-2-yloxy]-octyloxy}-naphthalen-1-yl)-ethyl]-acetamide 13776 N-[2-(7-{6-[8-(2-Acetylamino-ethyl)-naphthalen-2-yloxy]-hexyloxy}-naphthalen-1-yl)-ethyl]-acetamide 13781 N,N'-(2,2'-(7,7'-(butane-1,4-diylbis(oxy))bis(naphthalene-7,1-diyl))bis(ethane-2,1-diyl))diacetamide 13784 N-[2-(7-{2-[8-(2-Acetylamino-ethyl)-naphthalen-2-yloxy]-ethoxy}-naphthalen-1-yl)-ethyl]-acetamide 13875 N,N'-(2,2'-(7,7'-(propane-1,3-diylbis(oxy))bis(naphthalene-7,1-diyl))bis(ethane-2,1-diyl))diacetamide 13956 1-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-butyl]-pyrrolidine-2,5-dione 13963 8-[2-(3,4-Dihydro-1H-isoquinolin-2-yl)-ethyl]-8-aza-spiro[4.5]decane-7,9-dione 13971 2-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-butyl]-isoindole-1,3-dione 13983 2-[2-(3,4-Dihydro-1H-isoquinolin-2-yl)-ethyl]-isoindole-1,3-dione 13984 8-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-butyl]-8-aza-spiro[4.5]decane-7,9-dione 14055 N-[2-(7-{10-[8-(2-Acetylamino-ethyl)-naphthalen-2-yloxy]-decyloxy}-naphthalen-1-yl)-ethyl]-acetamide 14090 SID26752153 14101 SID29215039 14108 5-Methylsulfanyl-6-trifluoromethyl-2,3-dihydro-indole-1-carboxylic acid (3-pyridin-4-yl-phenyl)-amide 14131 6-chloro-5-methyl-N-(6-(2-methylpyridin-3-yloxy)pyridin-3-yl)indoline-1-carboxamide 14132 5-methyl-N-(6-(2-methylpyridin-3-yloxy)pyridin-3-yl)-6-(trifluoromethyl)indoline-1-carboxamide 14138 SID11113800 14189 5-Methoxy-6-trifluoromethyl-2,3-dihydro-indole-1-carboxylic acid [5-(2,6-difluoro-phenyl)-pyridin-3-yl]-amide 14221 SID26753650 14223 5-Methoxy-6-trifluoromethyl-2,3-dihydro-indole-1-carboxylic acid [3,4']bipyridinyl-5-ylamide 14224 5-Methoxy-6-trifluoromethyl-2,3-dihydro-indole-1-carboxylic acid (4'-methyl-[3,3']bipyridinyl-5-yl)-amide 14232 5-Methylsulfanyl-6-trifluoromethyl-2,3-dihydro-indole-1-carboxylic acid (3-pyridin-3-yl-phenyl)-amide 14243 (2R,3R,4R,5R)-5-(6-Amino-purin-9-yl)-2-hydroxymethyl-4-mercapto-tetrahydro-furan-3-ol 14303 5-Methoxy-6-trifluoromethyl-2,3-dihydro-indole-1-carboxylic acid [5-(4-fluoro-phenyl)-pyridin-3-yl]-amide 14337 5-Methoxy-6-trifluoromethyl-2,3-dihydro-indole-1-carboxylic acid [2,3']bipyridinyl-5-ylamide 14366 Flavopiridol 14373 5-Methoxy-6-trifluoromethyl-2,3-dihydro-indole-1-carboxylic acid [3,3']bipyridinyl-5-ylamide 14411 3-(4-Chloro-benzyl)-5-[2-(1H-imidazol-4-yl)-ethyl]-[1,2,4]oxadiazole 14412 5-Cyclohexyl-1-[4-(1H-imidazol-4-yl)-piperidin-1-yl]-pentan-1-one 14442 4-(7-Methyl-oct-3-ynyl)-1H-imidazole 14443 4-Hex-3-ynyl-1H-imidazole 14444 2-(3-Methyl-3H-imidazol-4-yl)-ethylamine 14451 5-Methoxy-6-trifluoromethyl-2,3-dihydro-indole-1-carboxylic acid [5-(3,5-difluoro-phenyl)-pyridin-3-yl]-amide 14483 Verongamine 14491 5-Methoxy-6-trifluoromethyl-2,3-dihydro-indole-1-carboxylic acid (5-phenyl-pyridin-3-yl)-amide 14559 SID26751870 14595 4-Hept-3-ynyl-1H-imidazole 14596 4-(6-Cyclopentyl-hex-3-ynyl)-1H-imidazole 14603 4-(8-Phenyl-oct-3-ynyl)-1H-imidazole 14604 4-(7,7-Dimethyl-oct-3-ynyl)-1H-imidazole 14634 4-(6-Cyclohexyl-hex-3-ynyl)-1H-imidazole 14715 (7-Chloro-quinolin-4-yl)-[4-(3-piperidin-1-yl-propoxy)-phenyl]-amine oxalic acid 14718 Ciproxifan 14727 {3-[4-(3-Piperidin-1-yl-propoxy)-phenyl]-propyl}-(1,2,3,4-tetrahydro-acridin-9-yl)-amine oxalic acid 14734 {4-[4-(3-Piperidin-1-yl-propoxy)-phenyl]-butyl}-(1,2,3,4-tetrahydro-acridin-9-yl)-amine oxalic acid 14768 {4-[4-(3-Piperidin-1-yl-propoxy)-phenyl]-butyl}-quinolin-4-yl-amine oxalic acid 14776 {3-[4-(3-Piperidin-1-yl-propoxy)-phenyl]-propyl}-quinolin-4-yl-amine oxalic acid 14785 SID26757996 14789 7-Fluoro-2-methyl-10-(4-methyl-piperazin-1-yl)-4H-3-thia-4,9-diaza-benzo[f]azulene 14798 N-(4-(3-(piperidin-1-yl)propoxy)phenethyl)-5,6,7,8-tetrahydroacridin-9-amine 14805 Lapatinib 14825 (7-Chloro-quinolin-4-yl)-{2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-ethyl}-amine oxalic acid 14851 {2-[4-(3-Piperidin-1-yl-propoxy)-phenyl]-ethyl}-quinolin-4-yl-amine oxalic acid 14923 N-(4-(3-(piperidin-1-yl)propoxy)phenyl)quinolin-4-amine 15018 (S)-2-Amino-3-(4-hydroxy-phenyl)-N-((5S,8R,16aR)-5-naphthalen-1-ylmethyl-4,7,13,16-tetraoxo-hexadecahydro-3a,6,12,15-tetraaza-cyclopentacyclopentadecen-8-yl)-propionamide 15019 (S)-2-Amino-3-(4-hydroxy-phenyl)-N-((5S,8S,16aR)-5-naphthalen-2-ylmethyl-4,7,13,16-tetraoxo-hexadecahydro-3a,6,12,15-tetraaza-cyclopentacyclopentadecen-8-yl)-propionamide 15091 (S)-2-Amino-3-(4-hydroxy-phenyl)-N-((5S,8S,17aR)-5-naphthalen-2-ylmethyl-4,7,14,17-tetraoxo-hexadecahydro-3a,6,13,16-tetraaza-cyclopentacyclohexadecen-8-yl)-propionamide 15097 (S)-2-Amino-3-(4-hydroxy-phenyl)-N-((5R,8R,15aS)-5-naphthalen-2-ylmethyl-4,7,12,15-tetraoxo-tetradecahydro-3a,6,11,14-tetraaza-cyclopentacyclotetradecen-8-yl)-propionamide 15098 (S)-2-Amino-N-((5S,8S,16aR)-5-benzyl-4,7,13,16-tetraoxo-hexadecahydro-3a,6,12,15-tetraaza-cyclopentacyclopentadecen-8-yl)-3-(4-hydroxy-phenyl)-propionamide 15149 N-methyl-2-phenyl-N-((5S,7S,8S)-8-(pyrrolidin-1-yl)-1-oxaspiro[4.5]decan-7-yl)acetamide 15191 SID46501178 15227 (S)-2-Amino-3-(4-hydroxy-phenyl)-N-[(5S,8R,16aR)-5-(1H-indol-3-ylmethyl)-4,7,13,16-tetraoxo-hexadecahydro-3a,6,12,15-tetraaza-cyclopentacyclopentadecen-8-yl]-propionamide 15245 (S)-2-Amino-3-(4-hydroxy-phenyl)-N-((5S,8S,13aR)-5-naphthalen-2-ylmethyl-4,7,13-trioxo-tetradecahydro-3a,6,12-triaza-cyclopentacyclododecen-8-yl)-propionamide 15330 7-[3-(4-Acetyl-3-methoxy-2-propyl-phenoxy)-propoxy]-8-propyl-chroman-2-carboxylic acid 15670 2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-acetylamino}-acetylamino)-3-phenyl-propionylamino]-4-methyl-pentanoic acid 15945 6-{4-[4-(3,4-Dichloro-benzyl)-piperazin-1-yl]-butyl}-3-methyl-3H-benzothiazol-2-one 15995 3-Methyl-6-[2-(4-phenyl-piperidin-1-yl)-ethyl]-3H-benzothiazol-2-one 16038 6-[2-((3R,5S)-3,5-Dimethyl-piperazin-1-yl)-ethyl]-3-methyl-3H-benzothiazol-2-one 16088 SID26757994 16097 6-{2-[4-(3,4-Dichloro-benzyl)-piperazin-1-yl]-ethyl}-3-methyl-3H-benzothiazol-2-one 16103 SID26752202 16116 6-{2-[4-(2,4-Dichloro-benzyl)-piperazin-1-yl]-ethyl}-3-methyl-3H-benzothiazol-2-one 16137 6-[4-(4-Benzyl-piperidin-1-yl)-butyl]-3-methyl-3H-benzothiazol-2-one 16146 6-[2-(4-Benzyl-piperazin-1-yl)-ethyl]-3-methyl-3H-benzothiazol-2-one 16209 (5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid bis-(2-hydroxy-ethyl)-amide 16217 SID26754691 16224 [4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-2-propyl-phenoxy]-phenyl-acetic acid 16240 6-[4-(4-Benzyl-piperazin-1-yl)-butyl]-3-methyl-3H-benzothiazol-2-one 16241 6-{4-[4-(2,4-Dichloro-benzyl)-piperazin-1-yl]-butyl}-3-methyl-3H-benzothiazol-2-one 16275 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-(N-cyclohexylcarboxamide) 16295 1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-methyl-1H-imidazole-4-carboxylic acid (hexahydro-cyclopenta[c]pyrrol-2-yl)-amide 16314 SID26751933 16316 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-(N-cyclohexyl,N-methylcarboxamide) 16331 6-[2-(4-Benzyl-piperidin-1-yl)-ethyl]-3-methyl-3H-benzothiazol-2-one 16332 3-Methyl-6-[4-(4-phenyl-piperidin-1-yl)-butyl]-3H-benzothiazol-2-one 16344 1-(4-chlorophenyl)-N-cyclohexyl-2-(2,4-dichlorophenyl)-1H-imidazole-4-carboxamide 16396 SID11114099 16446 SID26755749 16451 1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-1H-imidazole-4-carboxylic acid piperidin-1-ylamide 16485 SID26732615 16505 SID26747080 16524 ((S)-2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2-methoxy-benzyl)-amine 16538 N-(2,3-Dihydro-1'-methylspiro[benzofuran-3,4'-piperidine]-5-yl)-2'-methyl-4'-(5-methyl-1,2,4-oxadiazol-3-yl)biphenylcarboxamide 16603 N-{2-Benzo[1,3]dioxol-5-yl-2-[4-(2-ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-2,6-dipropyl-phenoxy]-acetyl}-methanesulfonamide 16604 5-Isobutyl-thiophene-2-sulfonic acid {2-benzo[1,3]dioxol-5-yl-2-[4-(2-ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-2-propyl-phenoxy]-acetyl}-amide 16656 SID11112153 16659 5-Isobutyl-3H-1lambda*4*-thiophene-2-sulfonic acid {2-benzo[1,3]dioxol-5-yl-2-[4-(2-ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-2,6-dipropyl-phenoxy]-acetyl}-amide 16660 N-{2-Benzo[1,3]dioxol-5-yl-2-[4-(2-ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-2,6-dipropyl-phenoxy]-acetyl}-4-isopropyl-benzenesulfonamide 16661 N-{2-Benzo[1,3]dioxol-5-yl-2-[4-(2-ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-2,6-dipropyl-phenoxy]-acetyl}-benzenesulfonamide 16687 (2,5-Dibromo-3,4-dimethoxy-phenyl)-[4-(2-ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-2,6-dipropyl-phenoxy]-acetic acid 16725 N-{2-Benzo[1,3]dioxol-5-yl-2-[4-(2-ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-2-propyl-phenoxy]-acetyl}-4-isopropyl-benzenesulfonamide 16812 Benzo[1,3]dioxol-5-yl-[4-(2-ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-2,6-dipropyl-phenoxy]-acetic acid 16827 Propane-2-sulfonic acid {2-benzo[1,3]dioxol-5-yl-2-[4-(2-ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-2,6-dipropyl-phenoxy]-acetyl}-amide 16828 3H-1lambda*4*-Thiophene-2-sulfonic acid {2-benzo[1,3]dioxol-5-yl-2-[4-(2-ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-2,6-dipropyl-phenoxy]-acetyl}-amide 16829 Dicarba-Closo-Dodecaborane analogue 16863 Benzo[1,3]dioxol-5-yl-[4-(2-ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-2-propyl-phenoxy]-acetic acid 16879 SID11111017 17528 4-amino-2-(4-methoxyphenyl)-[1,2,4]triazolo[4,3-a]quinoxalin-1(2H)-one 17632 4-(2,2-Diphenyl-ethylamino)-2-phenyl-2H-[1,2,4]triazolo[4,3-a]quinoxalin-1-one 17736 N-(1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl)acetamide 17773 N-(1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl)benzamide 17853 SID26753723 18145 SID17389570 18321 2-(furan-2-yl)-7-(3-phenylpropyl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine 18353 2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine 18397 2,3,8,9-tetrahydro-1H-indolo[2,3-a]pyrrolo[3,4-c]carbazol-1-one 18398 4-phenyl-2,3-dihydropyrrolo[3,4-c]carbazol-1(6H)-one 18402 8-butyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine 18409 SID26752233 18414 2-(furan-2-yl)-8-phenethyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine 18511 SID26753254 18536 SID11111478 18542 N-(2-Acetyl-phenyl)-3-[4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenyl]-acrylamide 18558 N-(2-Acetyl-phenyl)-3-[4-(1,3-dibenzyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenyl]-acrylamide 18562 SID11114142 18569 [4-(1,3-Dibenzyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetic acid () 18596 N-(3-Acetyl-phenyl)-2-[4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetamide 18639 N-(4-chlorophenyl)-2-(4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)phenoxy)acetamide 18645 4-{2-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetylamino}-benzamide 18646 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(4-fluorophenyl)acetamide 18653 3-[4-(1,3-Dibenzyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenyl]-acrylic acid 18683 4-{2-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetylamino}-benzoic acid methyl ester 18684 2-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-N-(4-trifluoromethyl-phenyl)-acetamide 18690 3-[4-(1,3-Bis-cyclohexylmethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenyl]-acrylic acid 18691 (E)-3-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenyl]-acrylic acid 18693 [4-(1,3-Dibutyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetic acid 18694 SID17389545 18714 4-{2-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetylamino}-benzoic acid (0.60CH2CL2) 18721 2-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-N-(4-nitro-phenyl)-acetamide (0.43CH3OH) 18722 [4-(1,3-Diallyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetic acid 18726 SID26719787 18729 N-(3,4-Dimethyl-2,5-dioxo-2,5-dihydro-pyrrol-1-yl)-2-[4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetamide 18743 N-{4-[(2-Amino-ethylcarbamoyl)-methyl]-phenyl}-2-[4-(1,3-diethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetamide 18751 4-{2-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetylamino}-N-methyl-benzamide (1.8CH2CL2) 18756 N-(2-Acetyl-phenyl)-2-[4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetamide 18761 N-Benzhydryl-2-[4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetamide 18778 2-[4-(1,3-Diethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-N-p-tolyl-acetamide 18798 8-[4-(2-Oxo-1,4-dihydro-2H-benzo[d][1,3]oxazin-4-yl)-phenyl]-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 18809 N-benzyl-2-(4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)phenoxy)acetamide 18817 N,N-dibenzyl-2-(4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)phenoxy)acetamide 18821 2-(4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)phenoxy)-N-phenylacetamide 18829 2-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-N-methyl-N-phenyl-acetamide 18880 1-[2-(5-Chloro-2-oxo-benzothiazol-3-yl)-acetyl]-piperidine-4-carboxylic acid thiazol-2-ylamide 18959 Boc-Asn-Arg-D-Phe-Phe-D-Trp-Leu-Met-OMe 18967 2-(4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)phenoxy)-N-(4-iodophenyl)acetamide 18977 N-(4-bromophenyl)-2-(4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)phenoxy)acetamide 19008 N-(3,4-Dimethyl-2,5-dioxo-2,5-dihydro-pyrrol-1-yl)-3-[4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenyl]-acrylamide 19040 4-(2-Dipropylamino-ethyl)-7-hydroxy-1,3-dihydro-benzoimidazol-2-one 19048 7-(2-Amino-ethyl)-4-hydroxy-3H-benzothiazol-2-one 19081 SID26752146 19149 4-(2-Dipropylamino-ethyl)-7-hydroxy-1,3-dihydro-indol-2-one 19150 4-(2-Dipropylamino-ethyl)-7-hydroxy-1H-indole-2,3-dione 19157 7-(2-Dipropylamino-ethyl)-4-hydroxy-3H-benzooxazol-2-one 19207 7-(2-Dipropylamino-ethyl)-4-hydroxy-3H-benzothiazol-2-one 19220 7-(2-Dipropylamino-ethyl)-3H-benzothiazol-2-one 19278 SID26752227 19279 4-(2-Amino-ethyl)-7-hydroxy-1,3-dihydro-indol-2-one 19316 SID26750081 19320 SID29217718 19362 Phosphoric acid mono-[4-(2-[2-(7-hydroxy-2-oxo-2H-chromen-4-yl)-acetylamino]-2-{3-[4-(3-methyl-5-oxo-4,5-dihydro-pyrazol-1-yl)-benzoylamino]-propylcarbamoyl}-ethyl)-phenyl] ester 19363 Phosphoric acid mono-(4-{2-(3-acetylamino-propylcarbamoyl)-2-[2-(7-hydroxy-2-oxo-2H-chromen-4-yl)-acetylamino]-ethyl}-phenyl) ester 19453 Phosphoric acid mono-[4-(2-acetylamino-2-{3-[4-(3-methyl-5-oxo-4,5-dihydro-pyrazol-1-yl)-benzoylamino]-propylcarbamoyl}-ethyl)-phenyl] ester 19468 Phosphoric acid mono-(4-{2-{3-[(1,3-dihydroxy-acridine-9-carbonyl)-amino]-propylcarbamoyl}-2-[2-(7-hydroxy-2-oxo-2H-chromen-4-yl)-acetylamino]-ethyl}-phenyl) ester 19572 levorphanol 19627 2-(4-Butyl-[1,4]diazepan-1-yl)-1-(2-ethoxy-ethyl)-1H-benzoimidazole 19642 2-(4-Benzyl-piperazin-1-yl)-1-(2-ethoxy-ethyl)-1H-benzoimidazole 19668 1-(2-Ethoxy-ethyl)-2-(4-propyl-[1,4]diazepan-1-yl)-1H-benzoimidazole 19669 2-[1,4]Diazepan-1-yl-1-(2-ethoxy-ethyl)-1H-benzoimidazole 19684 2-{2-[2-(4-Methyl-piperazin-1-yl)-benzoimidazol-1-yl]-ethoxy}-ethanol 19685 2-(4-Methyl-piperazin-1-yl)-1-(2-vinyloxy-ethyl)-1H-benzoimidazole 19686 1-(2-Methoxy-ethyl)-2-(4-methyl-piperazin-1-yl)-1H-benzoimidazole 19700 3,1'-Dimethyl-1',2',3',6'-tetrahydro-[2,4']bipyridinyl 19701 1-Benzyl-2-(4-methyl-piperazin-1-yl)-1H-benzoimidazole 19702 2-(4-Methyl-piperazin-1-yl)-1-phenyl-1H-benzoimidazole 19703 1-(2-Methyl-pentyl)-2-(4-methyl-piperazin-1-yl)-1H-benzoimidazole 19711 1-(2-Ethoxy-ethyl)-2-(4-ethyl-[1,4]diazepan-1-yl)-1H-benzoimidazole 19712 1-(2-Ethoxy-ethyl)-2-(4-methyl-[1,4]diazepan-1-yl)-1H-benzoimidazole 19731 1-(2-Ethoxy-ethyl)-2-(4-pentyl-piperazin-1-yl)-1H-benzoimidazole 19732 1-(3-Ethylsulfanyl-propyl)-2-(4-methyl-piperazin-1-yl)-1H-benzoimidazole 19733 1-(2-Ethylsulfanyl-ethyl)-2-(4-methyl-piperazin-1-yl)-1H-benzoimidazole 19735 3-Fluoro-1'-methyl-1',2',3',6'-tetrahydro-[2,4']bipyridinyl 19742 1-(2-Ethoxy-ethyl)-2-piperazin-1-yl-1H-benzoimidazole 19743 1-(2-Benzyloxy-ethyl)-2-(4-methyl-piperazin-1-yl)-1H-benzoimidazole 19768 1-(2-Butoxy-ethyl)-2-(4-methyl-piperazin-1-yl)-1H-benzoimidazole 19770 2-(4-Methyl-piperazin-1-yl)-1-pentyl-1H-benzoimidazole 19771 1-(3-Methoxy-propyl)-2-(4-methyl-piperazin-1-yl)-1H-benzoimidazole 19772 1-(2-Ethoxy-ethyl)-2-(4-methyl-piperazin-1-yl)-1H-benzoimidazole 19773 2-(4-Methyl-piperazin-1-yl)-1-propoxymethyl-1H-benzoimidazole 19782 2-(4-Methyl-piperazin-1-yl)-1-(2-phenoxy-ethyl)-1H-benzoimidazole 19915 Fentanyl 19965 3'-Fluoro-1-methyl-1,2,3,6-tetrahydro-[4,4']bipyridinyl 19987 1-(2-Ethoxy-ethyl)-2-(4-hexyl-piperazin-1-yl)-1H-benzoimidazole 19991 1-(3-Fluoro-pyridin-2-yl)-4-methyl-piperazine 19996 1'-Methyl-1',2',3',6'-tetrahydro-[2,4']bipyridinyl 19999 1-(1-Methyl-butyl)-2-(4-methyl-piperazin-1-yl)-1H-benzoimidazole 20000 1-(3-Methyl-butyl)-2-(4-methyl-piperazin-1-yl)-1H-benzoimidazole 20001 1'-Methyl-1',2',3',4',5',6'-hexahydro-[2,4']bipyridinyl 20005 1-(2-Ethoxy-ethyl)-2-(4-phenethyl-piperazin-1-yl)-1H-benzoimidazole 20025 2-[2-(4-Methyl-piperazin-1-yl)-benzoimidazol-1-yl]-ethanol 20029 2-(4-Methyl-piperazin-1-yl)-1-(2-prop-2-ynyloxy-ethyl)-1H-benzoimidazole 20030 1-(pyridin-2-yl)piperazine 20032 1'-Methyl-1',2',3',6'-tetrahydro-[3,4']bipyridinyl 20034 2-(4-Methyl-piperazin-1-yl)-1-propylsulfanylmethyl-1H-benzoimidazole 20035 2-(4-Methyl-piperazin-1-yl)-1-phenethyl-1H-benzoimidazole 20042 1-(2-Ethoxy-ethyl)-2-(4-propyl-piperazin-1-yl)-1H-benzoimidazole 20043 2-(4-Methyl-piperazin-1-yl)-1-(2-propoxy-ethyl)-1H-benzoimidazole 20069 1-(2-Allyloxy-ethyl)-2-(4-methyl-piperazin-1-yl)-1H-benzoimidazole 20070 1-Heptyl-2-(4-methyl-piperazin-1-yl)-1H-benzoimidazole 20078 2-(4-Butyl-piperazin-1-yl)-1-(2-ethoxy-ethyl)-1H-benzoimidazole 20081 2-(4-Methyl-piperazin-1-yl)-1-propyl-1H-benzoimidazole 20082 1-Methyl-2-(4-methyl-piperazin-1-yl)-1H-benzoimidazole 20085 1-(2-Ethoxy-ethyl)-2-(4-ethyl-piperazin-1-yl)-1H-benzoimidazole 20111 Ethyl-{2-[2-(4-methyl-piperazin-1-yl)-benzoimidazol-1-yl]-ethyl}-amine 20131 SID26751466 20287 Boc-Tyr(SO3H)-Nle-Gly-Trp-Nle-Asp-Phe-NH2 20293 1-Butyl-2-(4-methyl-piperazin-1-yl)-1H-benzoimidazole 20299 1',2',3',6'-Tetrahydro-[2,4']bipyridinyl 20329 Boc-gama-D-Glu-Tyr(SO3H)-Nle-D-Lys-Trp-Nle-Asp-Phe-NH2 20332 1-Hexyl-2-(4-methyl-piperazin-1-yl)-1H-benzoimidazole 20424 3-Chloro-1'-methyl-1',2',3',6'-tetrahydro-[2,4']bipyridinyl 20432 1-Decyl-2-(4-methyl-piperazin-1-yl)-1H-benzoimidazole 20443 Zacopride 20461 2-(4-Methyl-[1,4]diazepan-1-yl)-1-(2-phenoxy-ethyl)-1H-benzoimidazole 20462 1-(2-Butoxy-ethyl)-2-(4-methyl-[1,4]diazepan-1-yl)-1H-benzoimidazole 20465 1-(2-Allyloxy-ethyl)-2-(4-methyl-[1,4]diazepan-1-yl)-1H-benzoimidazole 20466 2-(4-Methyl-[1,4]diazepan-1-yl)-1-(2-propoxy-ethyl)-1H-benzoimidazole 20467 2-(4-Benzyl-[1,4]diazepan-1-yl)-1-(2-ethoxy-ethyl)-1H-benzoimidazole 20468 1-(2-Ethoxy-ethyl)-2-(4-pentyl-[1,4]diazepan-1-yl)-1H-benzoimidazole 20500 2-(4-Methyl-[1,4]diazepan-1-yl)-1-(2-prop-2-ynyloxy-ethyl)-1H-benzoimidazole 20592 Boc-cyclo-(gama-D-Glu-Tyr(SO3H)-Nle-D-Lys)-Trp-Nle-Asp-Phe-NH2 20819 5-hydroxy-alpha-methyltryptamine 20844 Boc-cyclo-(D-Glu-Tyr(SO3H)-Nle-D-Lys)-Trp-Nle-Asp-Phe-NH2 20845 Boc-cyclo-(Glu-Tyr(SO3H)-Nle-D-Lys)-Trp-Nle-Asp-Phe-NH2 20890 Boc-cyclo-(Glu-Tyr-Nle-D-Lys)-Trp-Nle-Asp-Phe-NH2 20952 Boc-cyclo-(gama-D-Glu-Tyr-Nle-D-Lys)-Trp-Nle-Asp-Phe-NH2 20953 Boc-D-Glu-Tyr(SO3H)-Nle-D-Lys-Trp-Nle-Asp-Phe-NH2 20954 Boc-Glu-Tyr(SO3H)-Nle-D-Lys-Trp-Nle-Asp-Phe-NH2 20969 6-Chloro-1H-benzoimidazole-4-carboxylic acid (9-methyl-9-aza-bicyclo[3.3.1]non-3-yl)-amide 21025 1H-Benzoimidazole-4-carboxylic acid (1-methyl-piperidin-4-yl)-amide 21035 Boc-D-Glu-Tyr(SO3H)-Nle-D-Nle-Trp-Nle-Asp-Phe-NH2 21072 6-Chloro-1H-benzoimidazole-4-carboxylic acid (1-methyl-piperidin-4-yl)-amide 21258 SID26751806 21313 Boc-cyclo-(D-Glu-Tyr-Nle-D-Lys)-Trp-Nle-Asp-Phe-NH2 21325 SID11113509 21432 SID11111754 21459 Naltrexone 21481 SID26751964 21505 (6aR,10aR)-3-(hept-1-ynyl)-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol 21534 immepip 21620 6-Chloro-1H-benzoimidazole-4-carboxylic acid 1-aza-bicyclo[2.2.2]oct-3-yl ester 21650 SID26755246 21698 SID11111431 21731 6-Chloro-1H-benzoimidazole-4-carboxylic acid (1-aza-bicyclo[2.2.2]oct-3-yl)-amide 21798 1-Methyl-8-phenyl-3-propyl-3,7-dihydro-purine-2,6-dione 21802 SID26755679 21839 (R)-2-Bromo-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol 21917 Iodine radioligand 4-[3-(4-Iodo-benzyloxy)-propyl]-1H-imidazole 22012 (-)-2-(6a,7,10,10a-tetrahydro-6,6,9-trimethylhydroxy-6H-dibenzo[b,d]pyranyl)-2-hexyl-1,3-dithiolane 22043 proxifan 22135 (1R,2S)-2-(1H-Imidazol-4-yl)-1-methyl-propylamine 22264 SID11113546 22289 3-Methyl-8-phenyl-1-propyl-3,7-dihydro-purine-2,6-dione 22306 4-((2R,3S)-2-Methyl-pyrrolidin-3-yl)-1H-imidazole 22307 4-((2S,3R)-2-Methyl-pyrrolidin-3-yl)-1H-imidazole 22383 SID29215512 22388 (1-Phenethyl-piperidin-4-yl)-phenyl-methanone 22426 4-((1S,2S)-2-(5,5-dimethylhex-1-ynyl)cyclopropyl)-1H-imidazole 22470 (1-Phenethyl-piperidin-4-yl)-phenyl-methanol 22512 (4-Fluoro-phenyl)-[1-(4-phenyl-butyl)-piperidin-4-yl]-methanol 22540 (1H-Imidazo[4,5-c]quinolin-4-yl)-phenyl-amine HCl 22577 (6aR,10aR)-3-(1-hexylcyclopropyl)-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol 22636 3,4-dihydroxy-2-[10-hydroxy-4-methyl-(5R,13R,14S,17R)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10,15-tetraen-14-yloxy]-3,4-dihydro-2H-6-pyrancarboxylic acid 22763 SID29217579 22826 2,3-Dihydro-1H-indol-5-ol 22875 1-(4-Hydroxy-benzyl)-1,2,3,4-tetrahydro-isoquinoline-6,7-diol 22912 1H-Imidazo[4,5-c]quinolin-4-ylamine 22929 Cyclopentyl-(1H-imidazo[4,5-c]quinolin-4-yl)-amine HCl 23056 SID26756723 23093 Terazocin 23103 Cyclopentyl-(2-phenyl-1H-imidazo[4,5-c]quinolin-4-yl)-amine 23156 SID26756967 23157 1-(3,4-Dihydroxy-benzyl)-1,2,3,4-tetrahydro-isoquinoline-6,7-diol 23240 Phenyl-(2-phenyl-1H-imidazo[4,5-c]quinolin-4-yl)-amine 23241 2-Phenyl-1H-imidazo[4,5-c]quinolin-4-ylamine 23242 Cyclopentyl-(2-cyclopentyl-1H-imidazo[4,5-c]quinolin-4-yl)-amine 23244 N-phenyl-2-cyclopentyl-1H-imidazo[4,5-c]quinolin-4-amine 23245 2-Cyclopentyl-1H-imidazo[4,5-c]quinolin-4-ylamine 23425 3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiophene-2-carboxylic acid (2,4,6-trimethyl-phenyl)-amide 23715 1-methyl-6,7-dihydroxytetrahydroisoquinoline 23727 2-[10-hydroxy-4-methyl-(5R,13R,14S,17R)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10,15-tetraen-14-yloxy]-6-methyltetrahydro-2H-3,4,5-pyrantriol 23782 3-hydroxy-6-[10-hydroxy-4-methyl-(5R,13R,14S,17R)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10,15-tetraen-14-yloxy]-3,6-dihydro-2H-2-pyrancarboxylic acid 23907 6-[10-hydroxy-4-methyl-(5R,13R,14S,17R)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10,15-tetraen-14-yloxy]tetrahydro-2H-2-pyrancarboxylic acid 23932 8-Hydroxy-6,11-dimethyl-3-(tetrahydro-furan-2-ylmethyl)-3,4,5,6-tetrahydro-2H-2,6-methano-benzo[d]azocin-1-one 23966 7-{(1R,2R,5S)-2-Fluoro-5-[(4-fluoro-benzenesulfonylamino)-methyl]-cyclopentyl}-heptanoic acid 24134 (Z)-7-[(1R,2R,5S)-2-Fluoro-5-(toluene-4-sulfonylamino)-cyclopentyl]-hept-5-enoic acid 24135 {4-[(1R,2R,5S)-2-Fluoro-5-(4-fluoro-benzenesulfonylamino)-cyclopentyl]-butoxy}-acetic acid 24245 {4-[(S)-5-(3,4-Dichloro-benzenesulfonylamino)-cyclopent-1-enyl]-butoxy}-acetic acid 24275 3-Cyclopropylmethyl-6-ethyl-8-hydroxy-11-methyl-3,4,5,6-tetrahydro-2H-2,6-methano-benzo[d]azocin-1-one 24284 (Z)-6-{(1R,2R,5S)-2-Fluoro-5-[(4-fluoro-benzenesulfonylamino)-methyl]-cyclopentyl}-hex-4-enoic acid 24286 {4-[(S)-5-(2-Nitro-benzenesulfonylamino)-cyclopent-1-enyl]-butoxy}-acetic acid 24288 (5Z)-7-[(1R,2S,5R)-2-benzenesulfonamido-5-fluorocyclopentyl]hept-5-enoic acid 24318 (Z)-6-{(1R,2S,5S)-2-Fluoro-5-[(4-fluoro-benzenesulfonylamino)-methyl]-cyclopentyl}-hex-4-enoic acid 24320 {4-[(S)-5-(2,4-Difluoro-benzenesulfonylamino)-cyclopent-1-enyl]-butoxy}-acetic acid 24322 {4-[(1R,2R,5S)-2-Fluoro-5-(toluene-4-sulfonylamino)-cyclopentyl]-butoxy}-acetic acid 24381 (Z)-7-[(1R,2R,5S)-2-Fluoro-5-(naphthalene-2-sulfonylamino)-cyclopentyl]-hept-5-enoic acid 24382 (Z)-6-[(1R,2S,5R)-2-(3,4-Dichloro-benzenesulfonylamino)-5-fluoro-cyclopentyl]-hex-4-enoic acid 24383 {4-[(1R,2R,5S)-2-Fluoro-5-(2-nitro-benzenesulfonylamino)-cyclopentyl]-butoxy}-acetic acid 24409 (Z)-7-[(1R,2S,5R)-2-(3,4-Dichloro-benzenesulfonylamino)-5-fluoro-cyclopentyl]-hept-5-enoic acid 24410 (Z)-6-[(S)-5-(Toluene-4-sulfonylamino)-cyclopent-1-enyl]-hex-4-enoic acid 24411 {4-[(1R,2S,5R)-2-(2,4-Difluoro-benzenesulfonylamino)-5-fluoro-cyclopentyl]-butoxy}-acetic acid 24412 (Z)-7-[(1R,2S,5R)-2-(4-Chloro-benzenesulfonylamino)-5-fluoro-cyclopentyl]-hept-5-enoic acid 24420 SID26753288 24437 (4Z)-6-[(5S)-5-benzenesulfonamidocyclopent-1-en-1-yl]hex-4-enoic acid 24438 6-{(1R,2R,5S)-2-Fluoro-5-[(4-fluoro-benzenesulfonylamino)-methyl]-cyclopentyl}-hexanoic acid 24439 (E)-7-[(S)-5-(Quinoline-8-sulfonylamino)-cyclopent-1-enyl]-hept-5-enoic acid 24461 (Z)-7-[(S)-5-(Naphthalene-2-sulfonylamino)-cyclopent-1-enyl]-hept-5-enoic acid 24462 (4-{(1R,2R,5S)-2-Fluoro-5-[(4-fluoro-benzenesulfonylamino)-methyl]-cyclopentyl}-butoxy)-acetic acid 24464 Naltrexone semicarbazone 24473 (Z)-7-[(S)-5-(2-Nitro-benzenesulfonylamino)-cyclopent-1-enyl]-hept-5-enoic acid 24484 (5Z)-7-((5S)-5-{[(4-fluorophenyl)sulfonyl]amino}cyclopent-1-en-1-yl)hept-5-enoic acid 24487 (Z)-7-[(S)-5-(Toluene-4-sulfonylamino)-cyclopent-1-enyl]-hept-5-enoic acid 24511 (Z)-6-[(1R,2S,5R)-2-(4-Chloro-benzenesulfonylamino)-5-fluoro-cyclopentyl]-hex-4-enoic acid 24512 (Z)-6-[(1R,2R,5S)-2-Fluoro-5-(2-nitro-benzenesulfonylamino)-cyclopentyl]-hex-4-enoic acid 24513 (E)-6-[(1R,2S,5R)-2-(2,4-Difluoro-benzenesulfonylamino)-5-fluoro-cyclopentyl]-hex-4-enoic acid 24514 (Z)-6-[(1R,2R,5S)-2-Fluoro-5-(4-fluoro-benzenesulfonylamino)-cyclopentyl]-hex-4-enoic acid 24516 (Z)-6-[(1R,2R,5S)-2-Fluoro-5-(toluene-4-sulfonylamino)-cyclopentyl]-hex-4-enoic acid 24523 (5Z)-7-[(5S)-5-benzenesulfonamidocyclopent-1-en-1-yl]hept-5-enoic acid 24530 4-Bromo-N-[4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-3-methyl-benzamide 24546 (Z)-7-[(1R,2R,5S)-2-Fluoro-5-(2-nitro-benzenesulfonylamino)-cyclopentyl]-hept-5-enoic acid 24547 (Z)-6-[(S)-5-(3,4-Dichloro-benzenesulfonylamino)-cyclopent-1-enyl]-hex-4-enoic acid 24548 (Z)-6-[(S)-5-(4-Chloro-benzenesulfonylamino)-cyclopent-1-enyl]-hex-4-enoic acid 24551 (Z)-6-[(S)-5-(2-Nitro-benzenesulfonylamino)-cyclopent-1-enyl]-hex-4-enoic acid 24572 1-{3-[4-(3-Chloro-phenyl)-piperazin-1-yl]-propyl}-3-[1-pyridin-3-yl-meth-(Z)-ylidene]-1,3-dihydro-indol-2-one 24580 2-tert-butyl-9-fluoro-3H-benzo[h]imidazo[4,5-f]isoquinolin-7(6H)-one 24581 2-(Benzothiazol-2-ylsulfanyl)-N-(1-benzyl-piperidin-4-yl)-acetamide 24585 7-[(S)-5-(4-Fluoro-benzenesulfonylamino)-cyclopent-1-enyl]-heptanoic acid 24586 (Z)-6-{(S)-5-[(4-Fluoro-benzenesulfonylamino)-methyl]-cyclopent-1-enyl}-hex-4-enoic acid 24587 (4-{(S)-5-[(4-Fluoro-benzenesulfonylamino)-methyl]-cyclopent-1-enyl}-butoxy)-acetic acid 24588 (Z)-6-[(S)-5-(2,4-Difluoro-benzenesulfonylamino)-cyclopent-1-enyl]-hex-4-enoic acid 24589 (5Z)-7-[(5S)-5-[(4-fluorobenzene)sulfonamidomethyl]cyclopent-1-en-1-yl]hept-5-enoic acid 24629 2-(Benzothiazol-2-ylsulfanyl)-N-(1-benzyl-piperidin-3-ylmethyl)-acetamide 24640 7-[(1R,2R,5S)-2-Fluoro-5-(4-fluoro-benzenesulfonylamino)-cyclopentyl]-heptanoic acid 24641 (Z)-6-{(1R,2S,5R)-2-[(4-Chloro-benzenesulfonylamino)-methyl]-5-fluoro-cyclopentyl}-hex-4-enoic acid 24654 (4Z)-6-[(1R,2S,5R)-2-benzenesulfonamido-5-fluorocyclopentyl]hex-4-enoic acid 24687 (Z)-6-{(1R,2R,5S)-2-Fluoro-5-[(toluene-4-sulfonylamino)-methyl]-cyclopentyl}-hex-4-enoic acid 24700 (Z)-6-[(S)-5-(4-Fluoro-benzenesulfonylamino)-cyclopent-1-enyl]-hex-4-enoic acid 24726 N-[3-(4-Pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide 24776 4-Methyl-N-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide 24801 2-(Benzothiazol-2-ylsulfanyl)-N-(1-cyclohexylmethyl-piperidin-3-ylmethyl)-acetamide 24828 (3S)-3-[(2S)-2-[(2R)-2-[(2S)-2-[(2S)-2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]-4-(methylsulfanyl)butanamido]-3-phenylpropanamido]-3-(1H-imidazol-4-yl)propanamido]-4-methylpentanamido]-4-(methylsulfanyl)butanamido]-3-carbamoylpropanoic acid 24829 (3S)-3-[(2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]-4-(methylsulfanyl)butanamido]-3-phenylpropanamido]-4-methylpentanamido]-4-(methylsulfanyl)butanamido]-3-carbamoylpropanoic acid 24868 3-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-3-phenyl-propionylamino)-4-methyl-pentanoylamino]-4-methylsulfanyl-butyrylamino}-succinamic acid 24904 (3S)-3-[(2S)-2-[(2S)-2-[(2R)-2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]-4-(methylsulfanyl)butanamido]-3-phenylpropanamido]-4-methylpentanamido]-4-(methylsulfanyl)butanamido]-3-carbamoylpropanoic acid 24905 (3S)-3-[(2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-[(2R)-2-amino-3-(4-hydroxyphenyl)propanamido]-4-(methylsulfanyl)butanamido]-3-phenylpropanamido]-4-methylpentanamido]-4-(methylsulfanyl)butanamido]-3-carbamoylpropanoic acid 24939 (4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S)-6-amino-1-[(2S)-2-{[(1S)-1-carbamoyl-2-methylpropyl]carbamoyl}pyrrolidin-1-yl]-1-oxohexan-2-yl]carbamoyl}methyl)carbamoyl]-2-(1H-indol-3-yl)ethyl]carbamoyl}-4-carbamimidamidobutyl]carbamoyl}-2-phenylethyl]carbamoyl}-2-(1H-imidazol-5-yl)ethyl]carbamoyl}-4-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-acetamido-3-hydroxypropanamido]-3-(4-hydroxyphenyl)propanamido]-3-hydroxypropanamido]-4-(methylsulfanyl)butanamido]butanoic acid 24948 2-(Benzothiazol-2-ylsulfanyl)-N-[1-(4-chloro-benzyl)-piperidin-4-yl]-acetamide 24964 (3S)-3-[(2S)-2-[(2R)-2-[(2S)-2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]-4-(methylsulfanyl)butanamido]-3-phenylpropanamido]-4-methylpentanamido]-4-(methylsulfanyl)butanamido]-3-carbamoylpropanoic acid 24983 [4-((1R,2S,5R)-2-Benzenesulfonylamino-5-fluoro-cyclopentyl)-butoxy]-acetic acid 25015 (3R)-3-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]-4-(methylsulfanyl)butanamido]-3-phenylpropanamido]-3-(1H-imidazol-4-yl)propanamido]-4-methylpentanamido]-4-(methylsulfanyl)butanamido]-3-carbamoylpropanoic acid 25033 2-(6-Amino-benzothiazol-2-ylsulfanyl)-N-[1-(3,4-dichloro-benzyl)-piperidin-4-yl]-acetamide 25034 N-[1-(3,4-Dichloro-benzyl)-piperidin-4-yl]-2-(6-ethoxy-benzothiazol-2-ylsulfanyl)-acetamide 25035 2-{[1-(3,4-Dichloro-benzyl)-piperidin-4-ylcarbamoyl]-methylsulfanyl}-benzothiazole-6-carboxylic acid ethyl ester 25036 2-(Benzothiazol-2-ylsulfanyl)-N-[1-(3,4-dichloro-benzyl)-piperidin-4-yl]-acetamide 25058 1-Cyclooct-1-enylmethyl-4-[(2,7-dichloro-9H-xanthene-9-carbonyl)-amino]-1-ethyl-piperidinium iodide 25063 {4-[(S)-5-(4-Fluoro-benzenesulfonylamino)-cyclopent-1-enyl]-butoxy}-acetic acid 25065 {4-[(S)-5-(Toluene-4-sulfonylamino)-cyclopent-1-enyl]-butoxy}-acetic acid 25067 (Z)-7-[(1R,2R,5S)-2-Fluoro-5-(4-fluoro-benzenesulfonylamino)-cyclopentyl]-hept-5-enoic acid 25072 2-(Benzothiazol-2-ylsulfanyl)-N-[1-(3-chloro-benzyl)-piperidin-4-yl]-acetamide 25076 4-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-4-mercapto-butyrylamino}-3-phenyl-propionylamino)-4-{1-[1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propylcarbamoyl}-butyric acid 25078 (3R)-3-[(2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]-4-(methylsulfanyl)butanamido]-3-phenylpropanamido]-4-methylpentanamido]-4-(methylsulfanyl)butanamido]-3-carbamoylpropanoic acid 25079 (3S)-3-[(2R)-2-[(2S)-2-[(2S)-2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]-4-(methylsulfanyl)butanamido]-3-phenylpropanamido]-4-methylpentanamido]-4-(methylsulfanyl)butanamido]-3-carbamoylpropanoic acid 25101 (Z)-7-[(1R,2S,5R)-2-(2,4-Difluoro-benzenesulfonylamino)-5-fluoro-cyclopentyl]-hept-5-enoic acid 25107 [4-((S)-5-Benzenesulfonylamino-cyclopent-1-enyl)-butoxy]-acetic acid 25121 (Z)-7-{(1R,2R,5S)-2-Fluoro-5-[(4-fluoro-benzenesulfonylamino)-methyl]-cyclopentyl}-hept-5-enoic acid 25151 4-Amino-N-[2-(benzyl-methyl-amino)-ethyl]-5-chloro-2-methoxy-benzamide 25154 1-{3-[4-(3-Chloro-phenyl)-piperazin-1-yl]-propyl}-3-[1-phenyl-meth-(Z)-ylidene]-1,3-dihydro-indol-2-one 25185 1-Methyl-1,3-dihydro-indol-2-one 25241 1-{3-[4-(3-Chloro-phenyl)-piperazin-1-yl]-propyl}-3-[1-pyridin-3-yl-meth-(E)-ylidene]-1,3-dihydro-indol-2-one 25301 4-[3-Isobutyl-1-(3-methyl-butyl)-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl]-benzenesulfonic acid 25305 SID11111028 25310 3-[1-(4-Chloro-phenyl)-meth-(E)-ylidene]-1-{3-[4-(3-chloro-phenyl)-piperazin-1-yl]-propyl}-1,3-dihydro-indol-2-one 25341 1,3,7-trimethyl-8-phenyl-3,4,5,7-tetrahydro-1H-purine-2,6-dione 25382 1-{3-[4-(3-Chloro-phenyl)-piperazin-1-yl]-propyl}-3-[1-thiophen-2-yl-meth-(E)-ylidene]-1,3-dihydro-indol-2-one 25383 3-[1-(4-Chloro-phenyl)-meth-(Z)-ylidene]-1-{3-[4-(3-chloro-phenyl)-piperazin-1-yl]-propyl}-1,3-dihydro-indol-2-one 25409 4-Bromo-3-methyl-N-[4-methyl-3-(4-methyl-piperazin-1-yl)-phenyl]-benzamide 25527 (racemic)5'-(5-Ethanesulfonyl-2-methoxy-phenyl)-1-ethyl-2,3,4,5-tetrahydro-1H,1'H-[2,2']bipyrrolyl 25538 (3S)-3-[(2R)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]-4-(methylsulfanyl)butanamido]-3-phenylpropanamido]-3-(1H-imidazol-4-yl)propanamido]-4-methylpentanamido]-4-(methylsulfanyl)butanamido]-3-carbamoylpropanoic acid 25539 3-(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-4-methylsulfanyl-butyrylamino}-3-phenyl-propionylamino)-3-(3H-imidazol-4-yl)-propionylamino]-4-methyl-pentanoylamino}-4-methylsulfanyl-butyrylamino)-succinamic acid 25684 1-{3-[4-(3-Chloro-phenyl)-piperazin-1-yl]-propyl}-3-[1-(4-methoxy-phenyl)-meth-(E)-ylidene]-1,3-dihydro-indol-2-one 25728 1-{3-[4-(3-Chloro-phenyl)-piperazin-1-yl]-propyl}-3-[1-(4-methoxy-phenyl)-meth-(Z)-ylidene]-1,3-dihydro-indol-2-one 25729 1-{3-[4-(3-Chloro-phenyl)-piperazin-1-yl]-propyl}-3-[1-thiophen-2-yl-meth-(Z)-ylidene]-1,3-dihydro-indol-2-one 25730 1-{3-[4-(3-Chloro-phenyl)-piperazin-1-yl]-propyl}-3-[1-phenyl-meth-(E)-ylidene]-1,3-dihydro-indol-2-one 25739 (R)-3-Cyclobutyl-2-{(3S,4S)-3-phenyl-4-[4-(3-phenyl-propyl)-piperidin-1-ylmethyl]-pyrrolidin-1-yl}-propionic acid 25874 2-Furan-2-yl-8-methyl-9-(4-methyl-piperazin-1-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 25936 2-(furan-2-yl)-8-methyl-9-(propylthio)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine 25966 2-Furan-2-yl-8-methyl-9-methylsulfanyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 26085 [6-(2-Dimethylamino-ethoxy)-5-methoxy-2,3-dihydro-indol-1-yl]-[2'-methyl-4'-(5-methyl-[1,2,4]oxadiazol-3-yl)-biphenyl-4-yl]-methanone 26091 8-Cyclopentyl-7-methyl-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 26106 2'-Methyl-4'-(5-methyl-[1,2,4]oxadiazol-3-yl)-biphenyl-4-carboxylic acid [3-(2-dimethylamino-ethylamino)-4-methoxy-phenyl]-amide 26118 SID11113970 26126 8-Cyclohexyl-1,3,7-trimethyl-3,7-dihydro-purine-2,6-dione 26144 4-Bromo-3-methyl-N-[3-(4-methyl-piperazin-1-yl)-phenyl]-benzamide 26180 SID29215037 26237 SID11111643 26262 2'-Methyl-4'-(5-methyl-[1,2,4]oxadiazol-3-yl)-biphenyl-4-carboxylic acid [3-(3-dimethylamino-propyl)-4-methoxy-phenyl]-amide 26293 2'-Methyl-4'-(5-methyl-[1,2,4]oxadiazol-3-yl)-biphenyl-4-carboxylic acid [7-(2-dimethylamino-ethoxy)-2,3-dihydro-benzofuran-5-yl]-amide 26294 2'-Methyl-4'-(5-methyl-[1,2,4]oxadiazol-3-yl)-biphenyl-4-carboxylic acid [4-(2-dimethylamino-ethyl)-3,4-dihydro-2H-benzo[1,4]oxazin-6-yl]-amide 26348 N*9*-Ethyl-2-furan-2-yl-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine-5,9-diamine 26358 N-(2-(furan-2-yl)-8-methyl-9-(methylthio)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-2-(4-methoxyphenyl)acetamide 26389 1-(9-Ethylamino-2-furan-2-yl-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-methoxy-phenyl)-urea 26418 1-[2-Furan-2-yl-8-methyl-9-(4-methyl-piperazin-1-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl]-3-(4-methoxy-phenyl)-urea 26420 2-Furan-2-yl-9-methylsulfanyl-8-(3-phenyl-propyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 26470 1-(2-Furan-2-yl-8-methyl-9-methylsulfanyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-methoxy-phenyl)-urea 26537 (S)-3-((S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-3-phenyl-propionylamino)-N-{(S)-1-[(S)-1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-succinamic acid 26648 sufugolix 26653 Xanomeline 26665 5-(3-Methyl-[1,2,4]oxadiazol-5-yl)-1,4,5,6-tetrahydro-pyrimidine TFA 26735 N-(2-Furan-2-yl-8-methyl-9-methylsulfanyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-2-(4-isobutyl-phenyl)-acetamide 26749 1-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-{3-[methyl-(1H-tetrazol-5-yl)-amino]-phenyl}-urea 26803 2-Benzo[1,3]dioxol-5-yl-N-(9-ethylamino-2-furan-2-yl-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-acetamide 26809 1-(4-(1-(2,6-difluorobenzyl)-5-((benzyl(methyl)amino)methyl)-2,4-dioxo-3-phenyl-1,2,3,4-tetrahydrothieno[2,3-d]pyrimidin-6-yl)phenyl)-3-ethylurea 26832 2-Benzo[1,3]dioxol-5-yl-N-(2-furan-2-yl-8-methyl-9-methylsulfanyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-acetamide 26838 N-(4-(1-(2,6-difluorobenzyl)-5-((benzyl(methyl)amino)methyl)-2,4-dioxo-3-phenyl-1,2,3,4-tetrahydrothieno[2,3-d]pyrimidin-6-yl)phenyl)benzamide 27031 6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine-8-carboxylic acid ((S)-1-butyl-pyrrolidin-2-ylmethyl)-amide 27111 Sumatriptan 27151 6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine-8-carboxylic acid ((R)-1-butyl-pyrrolidin-2-ylmethyl)-amide 27177 3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester 27207 (E)-6-{4-[2-(4-Chloro-benzenesulfonylamino)-ethyl]-phenyl}-6-pyridin-3-yl-hex-5-enoic acid 27254 [2-{4-[3-(2-Chloro-phenyl)-ureido]-butylcarbamoyl}-1-(1H-indol-3-ylmethyl)-1-phenethylcarbamoyl-ethyl]-carbamic acid adamantan-2-yl ester 27302 6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine-8-carboxylic acid ((R)-1-phenethyl-pyrrolidin-2-ylmethyl)-amide 27304 6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine-8-carboxylic acid ((S)-1-phenethyl-pyrrolidin-2-ylmethyl)-amide 27336 5-(3-Pent-1-ynyl-[1,2,4]oxadiazol-5-yl)-1,4,5,6-tetrahydro-pyrimidine TFA 27419 Triazolam 27517 Diprenorphine 27531 3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid ethyl ester 27609 SID26751841 27610 SID11114267 27616 SID11113786 27624 oxycodone 27644 (1S,7R)-4-[4-(4-Pyrimidin-2-yl-piperazin-1-yl)-butyl]-4-aza-tricyclo[5.2.1.0*2,6*]decane-3,5-dione 27645 8-{2-[4-(4-Methoxy-phenyl)-butylamino]-ethoxy}-chroman-6-ol 27648 SID29215419 27715 2,2'-(4-(3-(5-amino-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)propyl)phenylazanediyl)diethanol 27906 2-(4-(2-(5-amino-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)ethyl)phenylsulfonamido)acetic acid 27937 (3S,3aR,4R,4aS,8aR,9aS)-4-[(E)-2-((2R,6S)-1,6-Dimethyl-piperidin-2-yl)-vinyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 27957 3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid isopropyl ester 27958 3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid benzyl ester 27981 4-[2-(3-Phenoxy-propylamino)-ethoxy]-phenol 28077 [4-(4-Methoxy-phenyl)-butyl]-[2-(6-methyl-chroman-8-yloxy)-ethyl]-amine 28080 [2-(6-Chloro-chroman-8-yloxy)-ethyl]-[4-(4-methoxy-phenyl)-butyl]-amine 28103 N-(4-(2-(5-amino-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)ethyl)phenyl)acetamide 28109 3-(4-{2-[4-(5-carbamoyl-1H-3-indolyl)-3-cyclohexenylamino]ethylamino}-1-cyclohexenyl)-1H-5-indolecarboxamide 28111 3-(4-{5-[4-(5-carbamoyl-1H-3-indolyl)-3-cyclohexenylamino]pentylamino}-1-cyclohexenyl)-1H-5-indolecarboxamide 28135 2-(furan-2-yl)-7-(3-(4-nitrophenyl)propyl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine 28136 5-[3-(5-Amino-2-furan-2-yl-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)-propyl]-benzo[1,3]dioxole-2-carboxylic acid 28137 5-[3-(5-Amino-2-furan-2-yl-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)-propyl]-benzo[1,3]dioxole-2-carboxylic acid ethyl ester 28143 1-(diaziridin-1-ylphosphoryl)aziridine 28150 2,2'-(4-(2-(5-amino-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)ethyl)phenylazanediyl)diethanol 28174 5-(3-(5-amino-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)propyl)benzo[d][1,3]dioxole-2,2-dicarboxylic acid 28190 disodium 5-[3-(5-Amino-2-furan-2-yl-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)-propyl]-benzo[1,3]dioxole-2,2-dicarboxylic acid 28343 3-(4-{6-[4-(5-carbamoyl-1H-3-indolyl)-3-cyclohexenylamino]hexylamino}-1-cyclohexenyl)-1H-5-indolecarboxamide 28344 3-(4-{4-[4-(5-carbamoyl-1H-3-indolyl)-3-cyclohexenylamino]butylamino}-1-cyclohexenyl)-1H-5-indolecarboxamide 28350 (3S,4S)-4-[(1H-Indole-2-carbonyl)-amino]-5-oxo-1-phenyl-pyrrolidine-3-carboxylic acid 28386 (3S,4R)-4-[(Naphthalene-2-carbonyl)-amino]-5-oxo-1-phenyl-pyrrolidine-3-carboxylic acid 28423 (3S,4S)-1-Benzyl-4-[(naphthalene-2-carbonyl)-amino]-5-oxo-pyrrolidine-3-carboxylic acid 28432 (3S,4R)-4-[(1H-Indole-2-carbonyl)-amino]-5-oxo-1-phenyl-pyrrolidine-3-carboxylic acid 28433 4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-butyric acid 28449 (3S,4S)-4-[(Naphthalene-2-carbonyl)-amino]-5-oxo-1-phenyl-pyrrolidine-3-carboxylic acid 28450 (3S,4S)-1-(2-Fluoro-phenyl)-4-[(naphthalene-2-carbonyl)-amino]-5-oxo-pyrrolidine-3-carboxylic acid 28451 (3S,4S)-1-(2-Fluoro-phenyl)-5-oxo-4-[(quinoline-3-carbonyl)-amino]-pyrrolidine-3-carboxylic acid 28462 (3S,4S)-1-Benzyl-4-[(1H-indole-2-carbonyl)-amino]-5-oxo-pyrrolidine-3-carboxylic acid 28538 [2-(6-Fluoro-chroman-8-yloxy)-ethyl]-[4-(4-methoxy-phenyl)-butyl]-amine 28553 SID11111941 28558 [2-(7-Fluoro-chroman-8-yloxy)-ethyl]-[4-(4-methoxy-phenyl)-butyl]-amine 28601 [2-(6-Methoxy-chroman-8-yloxy)-ethyl]-[4-(4-methoxy-phenyl)-butyl]-amine 28621 [2-(Chroman-8-yloxy)-ethyl]-[4-(4-methoxy-phenyl)-butyl]-amine 28623 [2-(5-Fluoro-chroman-8-yloxy)-ethyl]-[4-(4-methoxy-phenyl)-butyl]-amine 28629 4-(3-(5-amino-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)propyl)benzonitrile 28631 (5-(3-(5-amino-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)propyl)benzo[d][1,3]dioxole-2,2-diyl)dimethanol 28645 4-(2-(5-amino-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)ethyl)benzenesulfonic acid 28659 4-(3-(5-amino-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)propyl)benzoic acid 28677 4-(2-(5-amino-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)ethyl)-N,N-bis(2-hydroxyethyl)benzenesulfonamide 28691 7-(3-(4-aminophenyl)propyl)-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine 28692 {4-[2-(5-Amino-2-furan-2-yl-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)-ethyl]-phenoxy}-acetic acid ethyl ester 28693 4-[3-(5-Amino-2-furan-2-yl-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)-propyl]-benzoic acid ethyl ester 28706 7-(3-(4-(aminomethyl)phenyl)propyl)-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine 28707 4-(3-(5-amino-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)propyl)-N'-hydroxybenzimidamide 28730 3-(4-{10-[4-(5-carbamoyl-1H-3-indolyl)-3-cyclohexenylamino]decylamino}-1-cyclohexenyl)-1H-5-indolecarboxamide 28745 3-(4-{12-[4-(5-carbamoyl-1H-3-indolyl)-3-cyclohexenylamino]dodecylamino}-1-cyclohexenyl)-1H-5-indolecarboxamide 28746 3-(4-{8-[4-(5-carbamoyl-1H-3-indolyl)-3-cyclohexenylamino]octylamino}-1-cyclohexenyl)-1H-5-indolecarboxamide 28871 1-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-imidazol-2-yl]-cyclohexanol 28874 4-[4-(4-Fluoro-phenyl)-5-pyridin-4-yl-1H-imidazol-2-yl]-1-methyl-piperidin-4-ol 28875 4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-oxazol-2-yl]-1-methyl-piperidin-4-ol 28878 4-[4-(4-Fluoro-phenyl)-5-pyridin-4-yl-oxazol-2-yl]-1-methyl-piperidin-4-ol 28896 4-[4-(4-Fluoro-phenyl)-5-pyridin-4-yl-thiazol-2-yl]-1-methyl-piperidin-4-ol 28898 4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-1-methyl-piperidin-4-ol 28926 1-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-imidazol-2-yl]-cycloheptanol 28928 1-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-imidazol-2-yl]-cyclopentanol 28952 SID26751906 28976 SID26754420 29061 SID26756673 29084 2-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-imidazol-2-yl]-propan-2-ol 29101 4-(3-(5-amino-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)propyl)benzimidamide 29115 1-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-imidazol-2-yl]-cyclopropanol 29116 2-(furan-2-yl)-7-(4-(4-methylpiperazin-1-ylsulfonyl)phenethyl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine 29117 1-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-imidazol-2-yl]-cyclobutanol 29134 7-(4-aminophenethyl)-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine 29146 3-(4-{3-[4-(5-carbamoyl-1H-3-indolyl)-3-cyclohexenylamino]propylamino}-1-cyclohexenyl)-1H-5-indolecarboxamide 29147 3-(4-{7-[4-(5-carbamoyl-1H-3-indolyl)-3-cyclohexenylamino]heptylamino}-1-cyclohexenyl)-1H-5-indolecarboxamide 29148 3-(4-Heptylamino-cyclohex-1-enyl)-1H-indole-5-carboxylic acid amide 29155 4-(2-tert-Butyl-5-phenyl-1H-imidazol-4-yl)-pyridine 29156 4-(2-(5-amino-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)ethyl)benzenesulfonamide 29169 6-[3-(5-Amino-2-furan-2-yl-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)-propyl]-benzo[1,3]dioxole-5-sulfonic acid 29170 4-(3-(5-amino-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)propyl)benzenesulfonic acid 29171 4-(2-(5-amino-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)ethyl)-N,N-bis(2-chloroethyl)benzenesulfonamide 29311 1-(2,6-Difluoro-benzyl)-5-(3-methoxy-phenyl)-6-methyl-3-{2-[methyl-(2-pyridin-2-yl-ethyl)-amino]-ethyl}-1H-pyrimidine-2,4-dione 29373 (S)-3-bromo-N-((1-ethylpyrrolidin-2-yl)methyl)-2-hydroxy-6-methoxybenzamide 29461 (S)-2-Dimethylamino-3-(1H-indol-3-yl)-propionic acid 3,5-dimethyl-benzyl ester 29462 (S)-2-Acetylamino-3-(1H-indol-3-yl)-propionic acid 3,5-dimethyl-benzyl ester 29557 [1-(3,5-Dimethyl-benzyloxycarbonyl)-2-(1H-indol-3-yl)-ethyl]-trimethyl-ammonium 29586 5'-Deoxy-5'-(methylthio)-adenosine 29727 3-Methyl-5-phenyl-1,2,3,4,5,6-hexahydro-azepino[4,5-b]indole 29781 10-Ethyl-1-[2-(3-ethyl-3H-benzothiazol-2-ylidene)-ethylidene]-3-methyl-1,2,3,10-tetrahydro-10-aza-3a-azonia-pentaleno[1,2-b]naphthalene iodide 29782 (R)-1-(2,6-difluorobenzyl)-3-(1-(2-methoxybenzylamino)propan-2-yl)-5-(2-fluoro-3-methoxyphenyl)-6-methylpyrimidine-2,4(1H,3H)-dione 29783 1-(2,6-Difluoro-benzyl)-3-{(S)-2-[(5-ethyl-furan-2-ylmethyl)-amino]-propyl}-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 29793 Spantide 29813 3-Ethyl-1-(2-hydroxy-ethyl)-2-[3-(1,3,3-trimethyl-1,3-dihydro-indol-2-ylidene)-propenyl]-3H-naphtho[2,3-d]imidazol-1-ium chloride 29814 1,3-Diethyl-2-[3-(1-ethyl-3,3-dimethyl-1,3-dihydro-indol-2-ylidene)-propenyl]-3H-naphtho[2,3-d]imidazol-1-ium chloride 29824 (S)-1-(2,6-difluorobenzyl)-3-(2-(cyclopentylamino)propyl)-5-(2-fluoro-3-methoxyphenyl)-6-methylpyrimidine-2,4(1H,3H)-dione 29833 (R)-1-(2,6-difluorobenzyl)-5-(2-fluoro-3-methoxyphenyl)-6-methyl-3-(2-(pyridin-2-ylmethylamino)propyl)pyrimidine-2,4(1H,3H)-dione 29850 3-((S)-2-Benzylamino-propyl)-1-(2,6-difluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 29865 1-(2,6-Difluoro-benzyl)-3-[(S)-2-(1-ethyl-propylamino)-propyl]-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 29868 1-(2,6-Difluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-3-{(R)-2-[(thiazol-2-ylmethyl)-amino]-propyl}-1H-pyrimidine-2,4-dione 29899 5-Ethyl-4-[2-(3-ethyl-3H-benzothiazol-2-ylidene)-ethylidene]-2,3,4,5-tetrahydro-1H-naphtho[2',3':4,5]imidazo[1,2-a]pyridin-12-ylium iodide 29900 1,3-Diethyl-2-[3-(1,3,3-trimethyl-1,3-dihydro-indol-2-ylidene)-propenyl]-3H-imidazo[4,5-b]quinoxalin-1-ium chloride 29901 10-Ethyl-1-[2-(3-ethyl-3H-benzooxazol-2-ylidene)-ethylidene]-1,2,3,10-tetrahydro-10-aza-3a-azonia-pentaleno[1,2-b]naphthalene iodide 29932 9-Phenyl-2,3-dihydro-1H-indeno[2,1-c]pyridine 29968 1-(2,6-Difluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-3-{(S)-2-[(3-methyl-thiophen-2-ylmethyl)-amino]-propyl}-1H-pyrimidine-2,4-dione 30002 1,3-Diethyl-2-[3-(1,3,3-trimethyl-1,3-dihydro-indol-2-ylidene)-propenyl]-3H-naphtho[2,3-d]imidazol-1-ium chloride 30003 10-Ethyl-1-[2-(1,3,3-trimethyl-1,3-dihydro-indol-2-ylidene)-ethylidene]-1,2,3,10-tetrahydro-10-aza-3a-azonia-pentaleno[1,2-b]naphthalene iodide 30011 2-Amino-3-(1H-indol-3-yl)-propionic acid 3,5-dimethyl-benzyl ester 30093 2-Ethyl-9-phenyl-2,3,4,9-tetrahydro-1H-indeno[2,1-c]pyridine 30096 2-Methyl-9-phenyl-2,3,4,9-tetrahydro-1H-indeno[2,1-c]pyridinium 30138 2-Methyl-9-phenyl-2,3,4,4a-tetrahydro-1H-indeno[2,1-c]pyridine 30158 2-Benzyl-9-phenyl-2,3,4,4a-tetrahydro-1H-indeno[2,1-c]pyridine 30189 ((3R,4S)-1-Ethyl-4-hydroxy-4-phenyl-piperidin-3-yl)-phenyl-methanone 30190 ((3R,4S)-4-Hydroxy-1-methyl-4-phenyl-piperidin-3-yl)-phenyl-methanone 30192 2-Benzyl-9-phenyl-2,3,4,9-tetrahydro-1H-indeno[2,1-c]pyridine 30203 1-(2-Acetoxy-ethyl)-3-ethyl-2-[3-(1,3,3-trimethyl-1,3-dihydro-indol-2-ylidene)-propenyl]-3H-naphtho[2,3-d]imidazol-1-ium chloride 30209 2-Methyl-9-phenyl-2,3-dihydro-1H-indeno[2,1-c]pyridine 30239 1,3-Diethyl-2-[3-(1-methyl-1H-benzo[cd]indol-2-ylidene)-propenyl]-3H-naphtho[2,3-d]imidazol-1-ium chloride 30273 1,3-Diethyl-2-[3-(3-ethyl-3H-benzooxazol-2-ylidene)-propenyl]-3H-naphtho[2,3-d]imidazol-1-ium iodide 30274 1,3-Diethyl-2-[3-(3-ethyl-3H-benzothiazol-2-ylidene)-propenyl]-3H-naphtho[2,3-d]imidazol-1-ium iodide 30275 (2S,3S)-N-(2-methoxybenzyl)-2-phenylpiperidin-3-amine 30310 10-Ethyl-1-[2-(1,1,3-trimethyl-1,3-dihydro-benzo[e]indol-2-ylidene)-ethylidene]-1,2,3,10-tetrahydro-10-aza-3a-azonia-pentaleno[1,2-b]naphthalene iodide 30369 2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionic acid benzyl ester 30629 SID11114130 30818 SID11113746 30915 2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionic acid 3,5-dimethyl-benzyl ester 30936 2-Ethylamino-3-(1H-indol-3-yl)-propionic acid benzyl ester 30953 2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionic acid 2-methoxy-benzyl ester 31153 SID11114140 31519 2-Butyl-5-fluoro-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3H-quinazolin-4-one 31533 6-Methyl-2-propyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3H-quinazolin-4-one 31587 4'-(2-Butyl-8-methyl-4-oxo-4H-quinazolin-3-ylmethyl)-biphenyl-2-carboxylic acid 31589 4'-(2-Butyl-6-methyl-4-oxo-4H-quinazolin-3-ylmethyl)-biphenyl-2-carboxylic acid 31673 4'-(2-Butyl-5-methyl-4-oxo-4H-quinazolin-3-ylmethyl)-biphenyl-2-carboxylic acid 31718 Phosphoric acid mono-(4-{2-acetylamino-2-[2-oxo-1-(3-phenyl-propyl)-azepan-3-ylcarbamoyl]-ethyl}-phenyl) ester 31813 Paratoulene phosphate 31900 SID26756731 31917 4'-(2-Butyl-7-methyl-4-oxo-4H-quinazolin-3-ylmethyl)-biphenyl-2-carboxylic acid 31973 Octanoic acid 1-hydroxymethyl-2-octanoyloxy-ethyl ester 31985 4'-(2-Butyl-4-oxo-4H-quinazolin-3-ylmethyl)-biphenyl-2-carboxylic acid 32041 4'-(2-Butyl-4-oxo-4H-benzo[g]quinazolin-3-ylmethyl)-biphenyl-2-carboxylic acid 32105 2-Butyl-7-chloro-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3H-quinazolin-4-one 32118 6-Methyl-2-pentyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3H-quinazolin-4-one 32128 Phosphoric acid mono-(4-{2-acetylamino-2-[1-(4-naphthalen-1-yl-benzyl)-2-oxo-azepan-3-ylcarbamoyl]-ethyl}-phenyl) ester 32199 3-Isobutyl-1-methyl-7-propyl-3,7-dihydro-purine-2,6-dione 32200 1,3-Diallyl-7-methyl-3,7-dihydro-purine-2,6-dione 32210 Acetic acid 2-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydro-purin-7-yl)-ethyl ester 32212 1,3-Dipropyl-7-prop-2-ynyl-3,7-dihydro-purine-2,6-dione 32240 7-Allyl-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 32241 1,3,7-Tripropyl-3,7-dihydro-purine-2,6-dione 32261 3-Isobutyl-1-methyl-7-prop-2-ynyl-3,7-dihydro-purine-2,6-dione 32262 7-Allyl-3-isobutyl-1-methyl-3,7-dihydro-purine-2,6-dione 32294 SID14724940 32327 6-Amino-2-butyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3H-quinazolin-4-one 32328 1,3-Dibenzyl-3,7-dihydro-purine-2,6-dione 32329 1,3-Diisobutyl-3,7-dihydro-purine-2,6-dione 32401 2-Butyl-6-chloro-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3H-quinazolin-4-one 32408 SID11111404 32416 2-Butyl-6-fluoro-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3H-quinazolin-4-one 32428 1,3-Diethyl-3,7-dihydro-purine-2,6-dione 32448 1-(2-Hydroxy-ethyl)-3-methyl-3,7-dihydro-purine-2,6-dione 32453 1,3-Diallyl-3,7-dihydro-purine-2,6-dione 32454 3-(2-Hydroxy-ethyl)-1-methyl-3,7-dihydro-purine-2,6-dione 32480 1-Ethyl-3-methyl-3,7-dihydro-purine-2,6-dione 32502 3-Isopropyl-1-methyl-3,7-dihydro-purine-2,6-dione 32503 1,3-Dimethyl-7-prop-2-ynyl-3,7-dihydro-purine-2,6-dione 32507 2-Butyl-6-nitro-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3H-quinazolin-4-one 32508 7-Benzyl-3-isobutyl-1-methyl-3,7-dihydro-purine-2,6-dione 32530 (S)-3-(8-((dimethylamino)methyl)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)-4-(1-methyl-1H-indol-3-yl)-1H-pyrrole-2,5-dione 32532 7-Benzyl-1,3-dipropyl-3,7-dihydro-purine-2,6-dione (7-benzyl-1,3-dipropylxanthine) 32533 SID26746971 32559 4HOPh(CH2)2CO-DTyr(Me)-Phe-Gln-Asn-Lys(5C-Flu)-Pro-Arg-NH2 32564 2-Butyl-6-methyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3H-quinazolin-4-one 32568 1,7-Dimethyl-3-propyl-3,7-dihydro-purine-2,6-dione 32588 N-{2-Butyl-4-oxo-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3,4-dihydro-quinazolin-6-yl}-acetamide 32595 3,7-Dimethyl-1-propyl-3,7-dihydro-purine-2,6-dione 32620 2-Butyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3H-quinazolin-4-one 32648 {2-Butyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3,4-dihydro-quinazolin-6-yl}-methyl-carbamic acid isobutyl ester 32652 1,3-Dimethyl-7-propyl-3,7-dihydro-purine-2,6-dione 32687 {2-Butyl-4-oxo-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3,4-dihydro-quinazolin-6-yl}-carbamic acid isobutyl ester 32688 Pentanoic acid {2-butyl-4-oxo-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3,4-dihydro-quinazolin-6-yl}-amide 32695 dermorphin 32737 4HOPh(CH2)2CO-DTyr(Me)-Phe-Gln-Asn-Arg-Pro-Lys(6C-Flu)-NH2 32738 4HOPh(CH2)2CO-DTyr(Me)-Phe-Gln-Asn-Lys(6C-Rhm)-Pro-Arg-NH2 32747 3-{2-Butyl-4-oxo-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3,4-dihydro-quinazolin-6-yl}-1-isopropyl-1-methyl-urea 32763 7-Allyl-1,3-dimethyl-3,7-dihydro-purine-2,6-dione 32764 SID24824050 32807 (2-Fluoro-4-methyl-phenyl)-[6-methoxy-7-(piperidin-4-ylmethoxy)-quinazolin-4-yl]-amine 32832 (4-Chloro-2,6-difluoro-phenyl)-[6-methoxy-7-(piperidin-4-ylmethoxy)-quinazolin-4-yl]-amine 32833 (3aR,9bS)-3-propyl-2,3,3a,4,5,9b-hexahydro-1H-benzo[e]indol-9-ol 32837 SID11114171 32852 2-(4-((R)-2-((R)-2-(3-chlorophenyl)-2-hydroxyethylamino)propyl)phenoxy)acetic acid 32874 3-Isobutyl-1,7-dimethyl-3,7-dihydro-purine-2,6-dione 32931 (4-Chloro-2,6-difluoro-phenyl)-[6-methoxy-7-(1-methyl-piperidin-4-ylmethoxy)-quinazolin-4-yl]-amine 32991 SID26753559 32992 1-Allyl-3,7-dimethyl-3,7-dihydro-purine-2,6-dione 33079 2-Butyl-6-methoxy-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3H-quinazolin-4-one 33087 (R)-1-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine-7,8-diol 33258 (HO-LVA23)2-{2-[3-(4-Hydroxy-phenyl)-2-(methyl-4-Hydroxy-phenylacetyl-amino)-propionylamino]-3-phenyl-propionylamino}-pentanedioic acid 5-amide 1-[(2-carbamoyl-1-{1-[2-(1-carbamoyl-4-guanidino-butylcarbamoyl)-pyrrolidine-1-carbonyl]-4-guanidino-butylcarbamoyl}-ethyl)-amide] 33279 3-({[2-(4-Hydroxy-2-isopropyl-5-methyl-phenoxy)-ethyl]-methyl-amino}-methyl)-4-methoxy-2,5,6-trimethyl-phenol 33281 5-Chloro-8-methyl-1-vinyl-1,6,7,8,9,9a-hexahydro-2-thia-8-aza-benzo[cd]azulene 33306 3-(3-{3-[4-Fluoro-2-(2,2,2-trifluoro-ethoxy)-phenyl]-piperazin-1-yl}-propyl)-5-methyl-1H-pyrimidine-2,4-dione 33307 1-(3-Hydroxy-propyl)-5-((R)-2-{2-[2-(2,2,2-trifluoro-ethoxy)-phenoxy]-ethylamino}-propyl)-2,3-dihydro-1H-indole-7-carboxylic acid amide 33320 1-(1-{2-[4-(1-Cyclopropylmethyl-piperidin-4-yloxy)-2-(2,2,2-trifluoro-ethoxy)-phenyl]-acetyl}-piperidin-4-yl)-1,4-dihydro-benzo[d][1,3]oxazin-2-one 33321 4HOPh(CH2)2CO-DTyr(Me)-Phe-Gln-Asn-Lys(5C-Rhm)-Pro-Arg-NH2 33323 1-(1-{2-[2-(2,2,2-Trifluoro-ethoxy)-phenyl]-acetyl}-piperidin-4-yl)-1,4-dihydro-benzo[d][1,3]oxazin-2-one 33336 2-Butyl-6,7-dimethoxy-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3H-quinazolin-4-one 33370 (4-Chloro-2-fluoro-phenyl)-[6-methoxy-7-(3-morpholin-4-yl-propoxy)-quinazolin-4-yl]-amine 33373 doxazosin 33392 1-(1-{2-[4-(2-Morpholin-4-yl-ethoxy)-2-(2,2,2-trifluoro-ethoxy)-phenyl]-acetyl}-piperidin-4-yl)-1,4-dihydro-benzo[d][1,3]oxazin-2-one 33397 [2-(4-Methoxy-phenyl)-ethyl]-(1,2,3,4-tetrahydro-naphthalen-2-ylmethyl)-amine 33420 SID29215539 33439 1-(1-{2-[4-Morpholin-4-yl-2-(2,2,2-trifluoro-ethoxy)-phenyl]-acetyl}-piperidin-4-yl)-1,4-dihydro-benzo[d][1,3]oxazin-2-one 33466 N-{1-[2-(1H-Indol-3-yl)-ethyl]-piperidin-4-yl}-benzamide 33471 N-(4-chloro-2-fluorophenyl)-6-methoxy-7-(2-methoxyethoxy)quinazolin-4-amine 33472 (2-Fluoro-4-methyl-phenyl)-[6-methoxy-7-(1-methyl-piperidin-4-ylmethoxy)-quinazolin-4-yl]-amine 33473 (4-Bromo-2,6-difluoro-phenyl)-[6-methoxy-7-(1-methyl-piperidin-4-ylmethoxy)-quinazolin-4-yl]-amine 33496 3-Fluoro-4-[6-methoxy-7-(4-pyrrolidin-1-yl-but-2-enyloxy)-quinazolin-4-ylamino]-benzonitrile 33507 1-(1-{2-[4-(1-Acetyl-piperidin-4-yloxy)-phenyl]-acetyl}-piperidin-4-yl)-1,4-dihydro-benzo[d][1,3]oxazin-2-one 33508 1-(1-{2-[4-(1-Acetyl-piperidin-4-yloxy)-2-(2,2,2-trifluoro-ethoxy)-phenyl]-acetyl}-piperidin-4-yl)-1,4-dihydro-benzo[d][1,3]oxazin-2-one 33536 (4-Chloro-2-fluoro-phenyl)-{6-methoxy-7-[2-(1-methyl-piperidin-4-yl)-ethoxy]-quinazolin-4-yl}-amine 33537 (4-Bromo-2,6-difluoro-phenyl)-[6-methoxy-7-(piperidin-4-ylmethoxy)-quinazolin-4-yl]-amine 33573 1-(1-{2-[4-(1-Acetyl-piperidin-4-yloxy)-2-methoxy-phenyl]-acetyl}-piperidin-4-yl)-1,4-dihydro-benzo[d][1,3]oxazin-2-one 33576 Vandetanib 33597 1-{1-[3-(2,4-Dimethoxy-phenyl)-propionyl]-piperidin-4-yl}-1,4-dihydro-benzo[d][1,3]oxazin-2-one 33600 (4-Bromo-2-fluoro-phenyl)-[6-methoxy-7-(2-[1,2,3]triazol-1-yl-ethoxy)-quinazolin-4-yl]-amine 33613 3-Methyl-4-oxo-2-phenyl-4H-chromene-8-carboxylic acid {3-[4-(2-methoxy-phenyl)-piperazin-1-yl]-propyl}-amide 33635 2,6-Dimethyl-4-(4-nitro-phenyl)-pyridine-3,5-dicarboxylic acid 3-{[3-(4,4-diphenyl-piperidin-1-yl)-propyl]-amide} 5-methylamide 33664 SID26719835 33667 SID26749009 33675 SID26751986 33681 SID11113697 33695 cyclazosin 33734 2,6-Dimethyl-4-(4-nitro-phenyl)-1,4-dihydro-pyridine-3,5-dicarboxylic acid 3-amide 5-{[3-(4,4-diphenyl-piperidin-1-yl)-propyl]-amide} 33781 (R)-6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline 33859 (4-Chloro-2-fluoro-phenyl)-[6-methoxy-7-(2-morpholin-4-yl-ethoxy)-quinazolin-4-yl]-amine 33863 (4-Chloro-2-fluoro-phenyl)-{6-methoxy-7-[2-(4-methyl-piperazin-1-yl)-ethoxy]-quinazolin-4-yl}-amine 33870 SID11110868 33894 [2-Butyl-5-chloro-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-acetic acid 33912 (4-Bromo-2-fluoro-phenyl)-{6-methoxy-7-[2-(1-methyl-piperidin-4-yl)-ethoxy]-quinazolin-4-yl}-amine 33959 (4-Chloro-2-fluoro-phenyl)-{6-methoxy-7-[2-(methyl-pyridin-4-yl-amino)-ethoxy]-quinazolin-4-yl}-amine 33994 (LVA)2-{2-[3-(4-Hydroxy-phenyl)-2-(methyl-phenylacetyl-amino)-propionylamino]-3-phenyl-propionylamino}-pentanedioic acid 5-amide 1-[(2-carbamoyl-1-{1-[2-(1-carbamoyl-4-guanidino-butylcarbamoyl)-pyrrolidine-1-carbonyl]-4-guanidino-butylcarbamoyl}-ethyl)-amide] 34036 4HOPh(CH2)2CO-DTyr(Me)-Phe-Gln-Asn-Arg-Pro-Lys(6C-Rhm)-NH2 34050 4'-(3-Pyrrolidin-1-yl-propoxy)-biphenyl-4-carbonitrile 34139 4HOPh(CH2)2CO-DTyr(Me)-Phe-Gln-Asn-Arg-Pro-Lys(5C-Flu)-NH2 34140 4HOPh(CH2)2CO-DTyr(Me)-Phe-Gln-Asn-Arg-Pro-Lys(5C-Rhm)-NH2 34195 1-(2-hydroxy-4-nitrophenyl)-3-phenylurea 34197 SID29215187 34233 2-{3-[4-(5-Chloro-2-methoxy-phenyl)-piperazin-1-yl]-propylamino}-pyrimidine-4-carboxylic acid amide 34234 SID29215183 34237 1-(2-Hydroxy-5-nitro-phenyl)-3-phenyl-urea 34238 1-(2-Hydroxy-3-nitro-phenyl)-3-phenyl-urea 34239 1-(4-cyano-2-hydroxyphenyl)-3-phenylurea 34266 zotepine 34279 1-(1-{2-[4-(1-Acetyl-piperidin-4-yloxy)-2-trifluoromethoxy-phenyl]-acetyl}-piperidin-4-yl)-1,4-dihydro-benzo[d][1,3]oxazin-2-one 34309 1-{1-[2-(2,4-Dimethoxy-phenyl)-acetyl]-piperidin-4-yl}-1,4-dihydro-benzo[d][1,3]oxazin-2-one 34310 1-[1-(2,4-Dimethoxy-benzoyl)-piperidin-4-yl]-1,4-dihydro-benzo[d][1,3]oxazin-2-one 34325 3-Isopropoxy-5-methyl-6,7-dihydro-4H-thiopyrano[3,4-d]isoxazol-5-ium iodide 34326 2,5-Dimethyl-3-oxo-2,3,6,7-tetrahydro-4H-thiopyrano[3,4-d]isoxazol-5-ium iodide 34331 3-Methoxy-5-methyl-4,5,6,7-tetrahydro-isoxazolo[4,5-c]pyridine 34347 (4-Bromo-2-fluoro-phenyl)-[6-methoxy-7-(2-piperidin-4-yl-ethoxy)-quinazolin-4-yl]-amine 34373 3-Methoxy-5,5-dimethyl-4,5,6,7-tetrahydro-isoxazolo[4,5-c]pyridin-5-ium iodide 34374 3-Methoxy-5-methyl-6,7-dihydro-4H-thiopyrano[3,4-d]isoxazol-5-ium iodide 34398 4''-Oxazol-2-yl-biphenyl-2-sulfonic acid (3,4-dimethyl-isoxazol-5-yl)-amide 34432 SID26719799 34433 3-Ethoxy-5-methyl-6,7-dihydro-4H-thiopyrano[3,4-d]isoxazol-5-ium iodide 34434 5-Methyl-3-prop-2-ynyloxy-6,7-dihydro-4H-thiopyrano[3,4-d]isoxazol-5-ium iodide 34600 SID11113640 34620 1-(3-Bromo-4-cyano-2-hydroxy-phenyl)-3-(2-bromo-phenyl)-urea 34621 1-(2-Bromo-phenyl)-3-(4-chloro-3-cyano-2-hydroxy-phenyl)-urea 34622 1-(2-Bromo-phenyl)-3-(3-chloro-4-cyano-2-hydroxy-phenyl)-urea 34656 1-(2-bromophenyl)-3-(4-cyano-2-hydroxyphenyl)urea 34709 (4'-(3-((2R,5R)-2,5-dimethylpyrrolidin-1-yl)propoxy)biphenyl-4-yl)(morpholino)methanone 34912 13-Hydroxymethyl-10-isopropyl-9-methyl-5-octyl-3,9,12-triaza-tricyclo[6.6.1.0*4,15*]pentadeca-1,4,6,8(15)-tetraen-11-one (n-octyl-ILV) 34952 phorbol 12,13-dibutyrate 34997 (-)-indolactam V 35021 Trifluoro-methanesulfonic acid 7-propylamino-5,6,7,8-tetrahydro-naphthalen-1-yl ester 35022 Trifluoro-methanesulfonic acid 7-dipropylamino-5,6,7,8-tetrahydro-naphthalen-1-yl ester 35029 (1R,2R,3S,4R,5S)-4-(6-Amino-2-chloro-purin-9-yl)-1-hydroxymethyl-bicyclo[3.1.0]hexane-2,3-diol 35034 3-Methoxy-N-{2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-benzamide 35038 4-Amino-5-chloro-2-methoxy-N-{2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-benzamide 35063 4-(6-Cyclopentylamino-purin-9-yl)-1-hydroxymethyl-bicyclo[3.1.0]hexane-2,3-diol 35064 (1S,2R,3S,4R,5S)-4-(6-Amino-purin-9-yl)-2,3-dihydroxy-bicyclo[3.1.0]hexane-1-carboxylic acid ethylamide 35324 SID11113902 35352 K-252a analogue 35374 1-(2-Methoxy-phenyl)-4-[3-(5-methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl)-propyl]-piperazine 35417 7-nitro-1,2,3,4-tetrahydroisoquinoline 35420 1,2,3,4-tetrahydroisoquinoline-7-sulfonamide 35450 5-Fluoro-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole 35469 8-Acenaphthen-1-yl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 35499 5-Methoxy-1,2,3,4-tetrahydro-naphthalene-1-carboxylic acid {2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-amide 35529 1-(2-Methoxy-phenyl)-4-[4-(5-methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl)-butyl]-piperazine 35530 8-Methoxy-1,2,3,4-tetrahydro-naphthalene-1-carboxylic acid {3-[4-(2-methoxy-phenyl)-piperazin-1-yl]-propyl}-amide 35531 N-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(4-(2-methoxyphenyl)piperazin-1-yl)propanamide 35547 1-Biphenyl-3-ylmethyl-4-(2-methoxy-phenyl)-piperazine 35570 5-Nitro-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole 35583 1-(3-Methoxy-phenyl)-5-[4-(2-methoxy-phenyl)-piperazin-1-yl]-pentan-1-one 35603 1-(3-Methoxy-phenyl)-4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butan-1-one 35612 1-(2-Methoxy-phenyl)-4-(1-phenyl-1H-pyrrol-3-ylmethyl)-piperazine 35617 Dimethyl-[2-(3,7,8,9-tetrahydro-pyrano[3,2-e]indol-1-yl)-ethyl]-amine 35623 (R)-Trifluoro-methanesulfonic acid 2-(6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-yl)-3-trifluoromethanesulfonyloxy-phenyl ester 35639 [4-(1,3-Dimethyl-2,6-dioxo-2,3,6,9-tetrahydro-1H-purin-8-yl)-phenoxy]-acetic acid 35642 2-[4-(1,3-Dimethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-N-p-tolyl-acetamide 35672 (R)-11-(2,6-Dimethoxy-phenyl)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline 35696 1,3-Diethyl-7-methyl-8-[(E)-2-(3,4,5-trimethoxy-phenyl)-vinyl]-3,7-dihydro-purine-2,6-dione 35706 3-methyl-2-((R)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-yl)-benzonitrile 35756 5-Bromo-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole 35757 8-[(E)-2-(3,4-Dimethoxy-phenyl)-vinyl]-7-methyl-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 35790 1,3-Dipropyl-8-styryl-3,7-dihydro-purine-2,6-dione 35888 (5-Methoxy-chroman-3-yl)-dipropyl-amine 35897 N-(8-Amino-octyl)-2-[4-(2,6-dioxo-1,3-dipropyl-2,3,6,9-tetrahydro-1H-purin-8-yl)-phenoxy]-acetamide 35900 2-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,9-tetrahydro-1H-purin-8-yl)-phenoxy]-N,N-dimethyl-acetamide 35905 2-(3-Methyl-3,7,8,9-tetrahydro-pyrano[3,2-e]indol-1-yl)-ethylamine 35946 N-(4-cyanophenyl)-2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 35967 4-(6-Amino-purin-9-yl)-1-hydroxymethyl-bicyclo[3.1.0]hexane-2,3-diol 35994 4-Piperazin-1-yl-7-trifluoromethyl-pyrrolo[1,2-a]quinoxaline (desmethyl-CGS-12066B) 36005 (1S,2R,3S,4R,5S)-4-[2-Chloro-6-(3-iodo-benzylamino)-purin-9-yl]-2,3-dihydroxy-bicyclo[3.1.0]hexane-1-carboxylic acid methylamide 36015 4-[2-chloro-6-(3-iodobenzylamino)-9H-9-purinyl]-1-hydroxymethyl-(1R,2R,3S,4R,5S)-bicyclo[3.1.0]hexane-2,3-diol 36032 4-(2-Chloro-6-cyclopentylamino-purin-9-yl)-1-hydroxymethyl-bicyclo[3.1.0]hexane-2,3-diol 36065 1-Butyl-4-(2-methoxy-phenyl)-piperazine 36093 SID4244225 36099 N-[4-(4-Phenyl-piperazin-1-yl)-butyl]-benzamide 36107 N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)benzamide 36123 5-(2-Oxo-hexahydro-thieno[3,4-d]imidazol-6-yl)-pentanoic acid (2-{2-[4-(2,6-dioxo-1,3-dipropyl-2,3,6,9-tetrahydro-1H-purin-8-yl)-phenoxy]-acetylamino}-ethyl)-amide 36132 2-(3,7,8,9-Tetrahydro-pyrano[3,2-e]indol-1-yl)-ethylamine 36144 3-methyl-2-((R)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-yl)-phenol 36146 (1S,2R,3S,4R,5S)-4-(2-chloro-6-(methylamino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 36163 8-(4-Hydroxy-phenyl)-1,3-dimethyl-3,7-dihydro-purine-2,6-dione 36211 1-hydroxymethyl-4-[6-(3-iodobenzylamino)-9H-9-purinyl]-(1R,2R,3S,4R,5S)-bicyclo[3.1.0]hexane-2,3-diol 36217 [4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetic acid ethyl ester 36218 2-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,9-tetrahydro-1H-purin-8-yl)-phenoxy]-N-(4-hydroxy-phenyl)-acetamide 36240 2-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,9-tetrahydro-1H-purin-8-yl)-phenoxy]-N-{2-[ethyl-(4-hydroxy-benzyl)-amino]-ethyl}-acetamide; compound with acetic acid 36287 (R)-2-(6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-yl)-benzene-1,3-diol 36324 (R)-6-Methyl-11-phenyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline 36351 2-[(2S,3S)-3-(3,5-Bis-trifluoromethyl-benzyloxy)-2-phenyl-piperidin-1-yl]-acetamide 36357 (1S,5aR)-6-methyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylen-1-ylamine 36363 1,3-Dicyclohexyl-1-{2-[4-(2,6-dioxo-1,3-dipropyl-2,3,6,9-tetrahydro-1H-purin-8-yl)-phenoxy]-acetyl}-urea 36383 8-(4-Hydroxy-phenyl)-1,3-dipropyl-3,9-dihydro-purine-2,6-dione 36419 2-(4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)phenoxy)-N-p-tolylacetamide 36420 2-(4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)phenoxy)acetic acid 36479 5-Chloro-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole 36480 3-(1,2,3,6-Tetrahydro-pyridin-4-yl)-1H-indol-5-ol (desmethyl-RU-24696) 36481 3-(1,2,3,6-Tetrahydro-pyridin-4-yl)-1H-indole-5-carbonitrile 36525 SID26755675 36595 SID11111082 36611 [4-(2,6-Dioxo-1,3-dipropyl-2,3,6,9-tetrahydro-1H-purin-8-yl)-phenoxy]-acetic acid hydrazide 36626 SID11113615 36633 1-tert-Butylamino-3-(thiochroman-8-yloxy)-propan-2-ol 36725 [4-(2,6-Dioxo-1,3-dipropyl-2,3,6,9-tetrahydro-1H-purin-8-yl)-phenoxy]-acetic acid 2,5-dioxo-pyrrolidin-1-yl ester 36730 SID11114150 36732 (R)-2a-(4-(4-phenyl-5,6-dihydropyridin-1(2H)-yl)butyl)-2a,3,4,5-tetrahydrobenzo[cd]indol-2(1H)-one 36743 8-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-ylamine 36760 N-(2-Acetylamino-ethyl)-2-[4-(2,6-dioxo-1,3-dipropyl-2,3,6,9-tetrahydro-1H-purin-8-yl)-phenoxy]-acetamide 36763 1N-methyl-2,3-dihydroxy-4-[6-(3-iodobenzylamino)-9H-9-purinyl]-(1S,2R,3S,4R,5S)-bicyclo[3.1.0]hexane-1-carboxamide 36884 7-Methyl-1,3-dipropyl-8-[(E)-2-(2,3,4-trimethoxy-phenyl)-vinyl]-3,7-dihydro-purine-2,6-dione 36974 N-((1R,5aR)-6-methyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylen-1-yl)-acetamide 36988 (R)-6,11-Dimethyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline 36989 1-Ethoxy-1-ethyl-6-methyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylene 37006 (1S,5aR)-1,6-dimethyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylen-1-ol 37007 (1R,5aR)-1,6-dimethyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylen-1-ol 37069 (2S,3S)-3-(3,5-Bis-trifluoromethyl-benzyloxy)-1-methyl-2-phenyl-piperidine 37089 (1R,5aR)-6-methyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylen-1-ylamine 37090 N-((1S,5aR)-6-methyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylen-1-yl)-acetamide 37223 2-hydroxy-5-(2-(2-hydroxy-3-(4-(1-methyl-4-(trifluoromethyl)-1H-imidazol-2-yl)phenoxy)propylamino)ethoxy)benzamide 37245 SID11113947 37323 (R)-6-Methyl-1,4a,5,5a,6,7,8,10c-octahydro-6-aza-benzo[mno]aceanthrylene 37332 3-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-3-phenyl-propionylamino)-N-{1-[1-(carboxymethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-succinamic acid 37344 Naphthalene-1-sulfonic acid (3,4-dimethyl-isoxazol-5-yl)-amide 37353 (1R,5aR)-6-methyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylen-1-ol 37354 6-Methyl-5a,6,7,8-tetrahydro-5H-6-aza-benzo[mno]aceanthrylen-1-one 37476 (1R,5aR)-1,6-dimethyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylene 37553 (1S,5aR)-1,6-dimethyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylene 37555 2-(3,4,5-trimethoxyphenyl)ethanamine 37592 (1S,5aR)-6-methyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylen-1-ol 37828 (6S,10aR)-6-methoxy-1,6-dimethyl-1,2,3,6,10,10a-hexahydrofluoreno[3,4,5-defg]quinoline 37829 (1R,5aR)-1-methoxy-1,6-dimethyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylene 37860 1-Ethoxy-1-ethyl-6-methyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylene 37987 SID26754187 38032 2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-3-phenyl-propionylamino)-N*1*-{1-[1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-succinamide 38033 (S)-4-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-3-phenyl-propionylamino)-4-{(S)-1-[(S)-1-(carboxymethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propylcarbamoyl}-butyric acid 38645 N-(2-bromophenyl)imidazo[1,5-a]quinoxalin-4-amine 38764 SID26751608 38798 N-{3-[2'-(1-Methyl-1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-4-oxo-3,4-dihydro-quinazolin-6-yl}-N-pentyl-benzamide 38799 Pentanoic acid benzyl-{3-[2'-(1-methyl-1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-4-oxo-3,4-dihydro-quinazolin-6-yl}-amide 38852 N-[2'-(3,4-Dimethyl-isoxazol-5-ylsulfamoyl)-4-oxazol-2-yl-biphenyl-2-ylmethyl]-acetamide 38873 DiSodium salt; Phosphoric acid mono-[4-(butyl-{3-[2'-(1-methyl-1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-4-oxo-3,4-dihydro-quinazolin-6-yl}-carbamoyl)-phenyl] ester 39130 Furan-2-carboxylic acid {3-[2'-(1-methyl-1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-4-oxo-3,4-dihydro-quinazolin-6-yl}-pyridin-2-ylmethyl-amide 39159 N-{3-[2'-(1-Methyl-1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-4-oxo-3,4-dihydro-quinazolin-6-yl}-N-pyridin-2-ylmethyl-isonicotinamide 39170 N-{3-[2'-(1-Methyl-1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-4-oxo-3,4-dihydro-quinazolin-6-yl}-N-pyridin-3-ylmethyl-benzamide 39171 N-{3-[2'-(1-Methyl-1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-4-oxo-3,4-dihydro-quinazolin-6-yl}-N-pyridin-2-ylmethyl-benzamide 39222 4-[(Benzoyl-{3-[2'-(1-methyl-1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-4-oxo-3,4-dihydro-quinazolin-6-yl}-amino)-methyl]-benzoic acid methyl ester 39223 N-(4-Hydroxy-benzyl)-N-{3-[2'-(1-methyl-1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-4-oxo-3,4-dihydro-quinazolin-6-yl}-benzamide 39229 4-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-3-phenyl-propionylamino)-4-{1-[1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propylcarbamoyl}-butyric acid 39350 N-Butyl-4-hydroxy-N-{3-[2'-(1-methyl-1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-4-oxo-3,4-dihydro-quinazolin-6-yl}-benzamide 39383 Bu-His-DPhe-Arg-Trp-Gly-NH2 39672 SID11113872 39749 4-Hydroxy-N-{3-[2'-(1-methyl-1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-4-oxo-3,4-dihydro-quinazolin-6-yl}-N-pentyl-benzamide 39881 1-Ethyl-3-propyl-3,7-dihydro-purine-2,6-dione 39951 Tetradecanoic acid (2R,3S)-2-hydroxymethyl-5-oxo-tetrahydro-furan-3-ylmethyl ester 39952 [(2S,3R)-2-(2-Hydroxy-ethyl)-5-oxo-tetrahydro-furan-3-yl]-acetic acid tetradecyl ester 39959 Tetradecanoic acid 2-(2-hydroxy-ethyl)-5-oxo-tetrahydro-furan-3-yl ester 39965 ((2R,3R)-2-Hydroxymethyl-5-oxo-tetrahydro-furan-3-yl)-acetic acid tetradecyl ester 39979 N*1*-{(2R,3R,4S,5R,6R)-3,4,5-Tris-benzyloxy-6-[2-(1H-indol-3-yl)-ethoxy]-tetrahydro-pyran-2-ylmethyl}-pentane-1,5-diamine 39980 5-{(2S,3S,4R,5R,6S)-3,4-Bis-benzyloxy-5-(1H-imidazol-4-ylmethoxy)-6-[2-(1H-indol-3-yl)-ethoxy]-tetrahydro-pyran-2-ylmethoxy}-pentylamine 40060 3-[4-(2-Fluoro-phenyl)-piperazin-1-ylmethyl]-1H-pyrrolo[2,3-b]pyridine 40138 3-(4-Biphenyl-4-yl-piperazin-1-ylmethyl)-1H-pyrrolo[2,3-b]pyridine 40141 3-[4-(4-Propyl-phenyl)-piperazin-1-ylmethyl]-1H-pyrrolo[2,3-b]pyridine 40142 3-[4-(4-Ethyl-phenyl)-piperazin-1-ylmethyl]-1H-pyrrolo[2,3-b]pyridine 40143 3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-1H-pyrrolo[2,3-b]pyridine 40144 3-[4-(4-Vinyl-phenyl)-piperazin-1-ylmethyl]-1H-pyrrolo[2,3-b]pyridine 40145 3-[4-(4-Trifluoromethyl-phenyl)-piperazin-1-ylmethyl]-1H-pyrrolo[2,3-b]pyridine 40178 3-[4-(4-Methylsulfanyl-phenyl)-piperazin-1-ylmethyl]-1H-pyrrolo[2,3-b]pyridine 40352 5-{3,4,5-Tris-benzyloxy-6-[2-(1H-indol-3-yl)-ethoxy]-tetrahydro-pyran-2-ylmethoxy}-pentylamine 40636 2-Chloroadenosine 40648 5-{(2R,3S,5R,6R)-3-Benzyloxy-5-(1H-imidazol-4-ylmethoxy)-6-[2-(1H-indol-3-yl)-ethoxy]-tetrahydro-pyran-2-ylmethoxy}-pentylamine 40717 (5S,8R,11S,14R,17S,19aS)-5-Benzyl-11-(4-fluoro-benzyl)-8-((R)-1-hydroxy-ethyl)-14-(1H-indol-3-ylmethyl)-17-naphthalen-1-ylmethyl-tetradecahydro-3a,6,9,12,15,18-hexaaza-cyclopentacyclooctadecene-4,7,10,13,16,19-hexaone 40718 N-(5-{(2R,3R,4S,5R,6R)-3,4-Bis-benzyloxy-5-(4-fluoro-benzyloxy)-6-[2-(1H-indol-3-yl)-ethoxy]-tetrahydro-pyran-2-ylmethoxy}-pentyl)-acetamide 40823 5-{(2S,3S,4R,5R,6S)-3,4,5-Tris-benzyloxy-6-[2-(1H-indol-3-yl)-ethoxy]-tetrahydro-pyran-2-ylmethoxy}-pentylamine 40825 5-{(2S,3S,4R,5S,6S)-3,4,5-Tris-benzyloxy-6-[2-(1H-indol-3-yl)-ethoxy]-tetrahydro-pyran-2-ylmethoxy}-pentylamine 40889 5-{(2R,3S,5R,6R)-3,5-Bis-benzyloxy-6-[2-(1H-indol-3-yl)-ethoxy]-tetrahydro-pyran-2-ylmethoxy}-pentylamine 40961 3-[4-(4-Methoxy-phenyl)-piperazin-1-ylmethyl]-1H-pyrrolo[2,3-b]pyridine 40962 3-[4-(4-Fluoro-phenyl)-piperazin-1-ylmethyl]-1H-pyrrolo[2,3-b]pyridine 41054 N-(5-{4,5-Bis-benzyloxy-3-hydroxy-6-[2-(1H-indol-3-yl)-ethoxy]-tetrahydro-pyran-2-ylmethoxy}-pentyl)-acetamide 41125 (5S,8R,11S,14R,17S,19aS)-5-Benzyl-11-(4-fluoro-benzyl)-8-((R)-1-hydroxy-ethyl)-14-(1H-indol-3-ylmethyl)-17-naphthalen-2-ylmethyl-tetradecahydro-3a,6,9,12,15,18-hexaaza-cyclopentacyclooctadecene-4,7,10,13,16,19-hexaone 41126 5-((2R,3R,4S,5R,6R)-3,4,5-Tris-benzyloxy-6-methoxy-tetrahydro-pyran-2-ylmethoxy)-pentylamine 41198 11-hydroxy-N-propylnoraporphine 41457 1-Methyl-3,7-dipropyl-3,7-dihydro-purine-2,6-dione 41458 7-Ethyl-1-methyl-3-propyl-3,7-dihydro-purine-2,6-dione 41462 1-Methyl-3-propyl-3,7-dihydro-purine-2,6-dione 41608 N-[4-(3-Chloro-4-fluoro-phenylamino)-pyrido[3,2-d]pyrimidin-6-yl]-acrylamide 41664 N-(4-m-Tolylamino-quinazolin-6-yl)-acrylamide 41764 N-[4-(3-Chloro-4-fluoro-phenylamino)-7-(3-morpholin-4-yl-propoxy)-quinazolin-6-yl]-acrylamide 41766 N-[4-(3-Chloro-4-fluoro-phenylamino)-quinazolin-6-yl]-acrylamide 41969 4-(2-Amino-1-hydroxy-ethyl)-3-fluoro-benzene-1,2-diol (2-FNE) 42020 4-(2-Amino-1-hydroxy-ethyl)-5-fluoro-benzene-1,2-diol (6-FNE) 42238 N-(4-(3-bromophenylamino)quinazolin-6-yl)acrylamide 42358 N-[4-(3-Bromo-4-fluoro-phenylamino)-quinazolin-6-yl]-acrylamide 42381 SID26751946 42430 SID26755711 42509 (3-Benzyl-3H-benzoimidazol-5-yl)-quinazolin-4-yl-amine 42616 (1-Benzyl-1H-indol-5-yl)-quinazolin-4-yl-amine 42617 SID11111220 42743 N*4*-(2-Benzyl-1H-benzoimidazol-5-yl)-pyrido[3,4-d]pyrimidine-4,6-diamine 42744 N*4*-(1-Benzyl-1H-indazol-5-yl)-pyrido[3,4-d]pyrimidine-4,6-diamine 42746 N*4*-(1-Benzyl-1H-indol-5-yl)-pyrido[3,4-d]pyrimidine-4,6-diamine 42756 SID26753766 42762 (R,S) 7-[(3-Iodo-allyl)-propyl-amino]-5,6,7,8-tetrahydro-naphthalen-1-ol 42780 (2-Benzyl-1H-benzoimidazol-5-yl)-(6,7-dimethoxy-quinazolin-4-yl)-amine 42794 (2-Benzyl-1H-benzoimidazol-5-yl)-quinazolin-4-yl-amine 42853 (1-Benzyl-1H-benzoimidazol-5-yl)-quinazolin-4-yl-amine 42885 (1-Benzyl-1H-indazol-5-yl)-(6,7-dimethoxy-quinazolin-4-yl)-amine 42886 (1-Benzyl-1H-indazol-5-yl)-quinazolin-4-yl-amine 43103 N-[4-(3-Bromo-phenylamino)-3-cyano-quinolin-6-yl]-acrylamide 43104 But-2-ynoic acid [4-(3-chloro-4-fluoro-phenylamino)-3-cyano-quinolin-6-yl]-amide 43122 But-2-ynoic acid [4-(3-bromo-phenylamino)-3-cyano-quinolin-6-yl]-amide 43141 4-Dimethylamino-but-2-enoic acid [4-(3-bromo-phenylamino)-3-cyano-quinolin-6-yl]-amide 43162 But-2-ynoic acid [5-(3-bromo-phenylamino)-6-cyano-[1,8]naphthyridin-3-yl]-amide 43226 6,7-Dimethoxy-4-(4-phenoxy-phenylamino)-quinoline-3-carbonitrile 43264 (E)-4-Dimethylamino-but-2-enoic acid [4-(3-bromo-phenylamino)-3-cyano-[1,7]naphthyridin-6-yl]-amide 43265 But-2-ynoic acid [5-(3-chloro-4-fluoro-phenylamino)-6-cyano-[1,8]naphthyridin-3-yl]-amide 43268 (E)-4-Dimethylamino-but-2-enoic acid [5-(3-bromo-phenylamino)-6-cyano-[1,8]naphthyridin-3-yl]-amide 43290 (1-Benzyl-1H-indol-5-yl)-(6,7-dimethoxy-quinazolin-4-yl)-amine 43291 (2-Benzyl-2H-indazol-5-yl)-(6,7-dimethoxy-quinazolin-4-yl)-amine 43487 6-Methoxy-7-(3-morpholin-4-yl-propoxy)-4-(4-phenethyl-phenylamino)-quinoline-3-carbonitrile 43524 6-Methoxy-7-(3-morpholin-4-yl-propoxy)-4-(4-phenoxy-phenylamino)-quinoline-3-carbonitrile 43567 5-methoxy-alpha-methyltryptamine 43743 N-[5-(3-Bromo-phenylamino)-6-cyano-[1,8]naphthyridin-3-yl]-acrylamide 43964 Tyr-Pro-L-(NMe)Phe-D-Pro-NH2 44064 6,7-Dimethoxy-4-(3-phenoxy-phenylamino)-quinoline-3-carbonitrile 44185 (R)-2-{[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoyl]-methyl-amino}-3-(1H-indol-3-yl)-propionic acid 44191 (R)-5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoic acid 44234 1-(3,4-Dichloro-phenyl)-2-isopropylamino-ethanol 44622 1-Methyl-2-(3,4,5-trimethoxy-phenyl)-ethylamine 44700 2-(2,4-Dimethoxy-phenyl)-1-methyl-ethylamine 44885 4-(4,5-Dihydro-benzo[b]thiophen-7-yl)-1H-imidazole 44905 SID11114268 44906 4-(1,3-Dimethyl-4,5,6,7-tetrahydro-benzo[c]thiophen-4-yl)-1H-imidazole 44977 4-Benzo[b]thiophen-4-yl-1H-imidazole 44978 4-(6,7-Dihydro-benzo[b]thiophen-4-yl)-1H-imidazole 44979 4-(4,5,6,7-Tetrahydro-benzo[b]thiophen-4-yl)-1H-imidazole 45013 4-(4,5,6,7-Tetrahydro-benzo[b]thiophen-7-yl)-1H-imidazole 45028 (S)-4-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-4-(naphthalen-1-ylcarbamoyl)-butyric acid 45217 4-(1,3-Dimethyl-6,7-dihydro-benzo[c]thiophen-4-yl)-1H-imidazole 45294 2-[4-(3,4-Dihydro-benzo[c][1,2]dioxin-5-yl)-piperazin-1-ylmethyl]-tetrahydro-imidazo[1,5-a]pyridine-1,3-dione 45295 2-{4-[4-(9H-5,6-Dioxa-benzocyclohepten-1-yl)-piperazin-1-yl]-butyl}-hexahydro-pyrrolo[1,2-a]pyrazine-1,4-dione 45296 2-[4-(1H-Benzoimidazol-4-yl)-piperazin-1-ylmethyl]-tetrahydro-pyrrolo[1,2-c]imidazole-1,3-dione 45306 2-(4-Naphthalen-1-yl-piperazin-1-ylmethyl)-tetrahydro-imidazo[1,5-a]pyridine-1,3-dione 45319 (-)-8-Hydroxy-3,6,11-trimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-4-carbonitrile 45322 8-Hydroxy-3,6,11-trimethyl-3,4,5,6-tetrahydro-1H-2,6-methano-benzo[d]azocine-2-carboxylic acid amide 45334 (+)-8-Hydroxy-3,6,11-trimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-4-carboxylic acid amide 45342 2-(4-Naphthalen-1-yl-piperazin-1-ylmethyl)-tetrahydro-pyrrolo[1,2-c]imidazole-1,3-dione 45608 N-methyl-N-((E)-1-{[3-(5-methyl-1H-imidazol-4-yl)phenyl]amino}-2-nitrovinyl)amine 45733 2-[4-(4-Naphthalen-1-yl-piperazin-1-yl)-butyl]-tetrahydro-pyrrolo[1,2-c]imidazole-1,3-dione 45734 2-(4-Naphthalen-1-yl-piperazin-1-ylmethyl)-hexahydro-pyrrolo[1,2-a]pyrazine-1,4-dione 45841 SID26751858 45881 4-Amino-5-chloro-2-methoxy-benzoic acid 8-methyl-8-aza-bicyclo[3.2.1]oct-3-yl ester 45882 4-Amino-5-chloro-2-methoxy-benzoic acid 1-ethyl-piperidin-4-yl ester 45919 N-{4-[3-(4-Amino-1-oxo-1H-1lambda*4*-[1,2,5]thiadiazol-3-ylamino)-phenyl]-thiazol-2-yl}-guanidine 45922 N''-cyano-N-(3-{2-[(diaminomethylene)amino]-1,3-thiazol-4-yl}phenyl)-N'-methylguanidine 45947 N-(2-(5-methoxy-2-(3-methoxybenzyl)benzofuran-3-yl)ethyl)acetamide 45952 N-[3-(5-Methyl-1H-imidazol-4-yl)-phenyl]-1-oxo-1H-1lambda*4*-[1,2,5]thiadiazole-3,4-diamine 45979 SID26753194 46003 8-Cyclopentyl-1-methyl-3-propyl-3,7-dihydro-purine-2,6-dione 46065 1'-[4-methyl(phenyl)sulfonamido-3-phenylbutyl]spiro[2,3-dihydrobenzo[b]thiophene-1-oxide-3,4'-(hexahydropyridine)] 46164 8-Cyclopentyl-3-methyl-1-propyl-3,7-dihydro-purine-2,6-dione 46202 N-[2-(1-Benzyl-5-methoxy-1H-indol-3-yl)-ethyl]-acetamide 46204 N-(2-(5-methoxy-1-methyl-1H-indol-3-yl)ethyl)acetamide 46209 8-Phenethyl-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 46215 N-{4-[3-(1-Methylamino-2-nitro-vinylamino)-phenyl]-thiazol-2-yl}-guanidine 46216 N-{4-[4-(1-Methylamino-2-nitro-vinylamino)-phenyl]-thiazol-2-yl}-guanidine 46218 3-Methyl-1-propyl-8-thiophen-3-yl-3,7-dihydro-purine-2,6-dione 46233 SID26752040 46234 1,3-Dipropyl-8-thiophen-2-yl-3,7-dihydro-purine-2,6-dione 46266 1-Methyl-3-propyl-8-thiophen-3-yl-3,7-dihydro-purine-2,6-dione 46267 1,3-Dipropyl-8-pyridin-3-yl-3,7-dihydro-purine-2,6-dione 46303 1'-[4-phenyl-1-phenylsulfonyl-(3R,4S)-tetrahydro-1H-3-pyrrolylmethyl]spiro[2,3-dihydrobenzo[b]thiophene-3,4'-(hexahydropyridine)1-oxide] 46304 1-Methyl-3-propyl-8-pyridin-3-yl-3,7-dihydro-purine-2,6-dione 46312 1'-[4-phenyl-1-phenylsulfonyl-(3S,4S)-tetrahydro-1H-3-pyrrolylmethyl]spiro[2,3-dihydrobenzo[b]thiophene-3,4'-(hexahydropyridine)1,1-dioxide] 46336 3-Methyl-1-propyl-8-pyridin-3-yl-3,7-dihydro-purine-2,6-dione 46410 {(4S,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-10-benzyl-4-[(R)-1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-3,3,14,14-tetramethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradec-7-yl}-acetic acid 46497 {(4S,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-10-benzyl-4-[(R)-1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-3,3-dimethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradec-7-yl}-acetic acid 46498 3-(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-4-methylsulfanyl-butyrylamino}-3-phenyl-propionylamino)-3-(1H-imidazol-4-yl)-propionylamino]-4-methyl-pentanoylamino}-4-methylsulfanyl-butyrylamino)-succinamic acid 46517 3-Methyl-1-propyl-8-thiophen-2-yl-3,7-dihydro-purine-2,6-dione 46606 N-((1-(4-chlorobenzyl)-4-methoxy-1H-indol-2-yl)methyl)propionamide 46797 (2,3-Dichloro-4-{2-[2-hydroxy-2-(4-hydroxy-phenyl)-1-methyl-ethylamino]-ethyl}-phenylamino)-acetic acid 46804 N-{4-[3-(4-Methylamino-1-oxo-1H-1lambda*4*-[1,2,5]thiadiazol-3-ylamino)-phenyl]-thiazol-2-yl}-guanidine 46814 SID29215161 46820 SID11113752 46839 N''-cyano-N-methyl-N'-[3-(5-methyl-1H-imidazol-4-yl)phenyl]guanidine 46854 4-Amino-5-chloro-2-methoxy-benzoic acid 1-ethyl-piperidin-3-yl ester 46855 4-Amino-5-chloro-2-methoxy-benzoic acid 1-methyl-piperidin-4-yl ester 46873 (2,6-Dibromo-4-{2-[2-hydroxy-2-(4-hydroxy-phenyl)-1-methyl-ethylamino]-ethyl}-phenylamino)-acetic acid 46874 (2,5-Dichloro-4-{2-[2-hydroxy-2-(4-hydroxy-phenyl)-1-methyl-ethylamino]-ethyl}-phenylamino)-acetic acid 46884 SID17389844 47056 (4-{2-[2-Hydroxy-2-(4-hydroxy-phenyl)-1-methyl-ethylamino]-ethyl}-phenylamino)-acetic acid 47067 (3-Chloro-4-{2-[2-hydroxy-2-(4-hydroxy-phenyl)-1-methyl-ethylamino]-ethyl}-phenylamino)-acetic acid 47068 [Benzyl-(4-{2-[2-hydroxy-2-(4-hydroxy-phenyl)-1-methyl-ethylamino]-ethyl}-phenyl)-amino]-acetic acid 47109 SID26753172 47117 [Carboxymethyl-(4-{2-[2-hydroxy-2-(4-hydroxy-phenyl)-1-methyl-ethylamino]-ethyl}-phenyl)-amino]-acetic acid 47118 [(4-{2-[2-Hydroxy-2-(4-hydroxy-phenyl)-1-methyl-ethylamino]-ethyl}-phenyl)-methyl-amino]-acetic acid 47147 (2,6-Dichloro-4-{2-[2-hydroxy-2-(4-hydroxy-phenyl)-1-methyl-ethylamino]-ethyl}-phenylamino)-acetic acid 47179 SID26755680 47210 (2-Bromo-4-{2-[2-hydroxy-2-(4-hydroxy-phenyl)-1-methyl-ethylamino]-ethyl}-phenylamino)-acetic acid 47218 1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichloro-phenyl)-5-(4-hydroxy-4-phenyl-piperidin-1-yl)-pentan-2-one O-methyl-oxime 47233 2-(3-Chloro-4-{2-[2-hydroxy-2-(4-hydroxy-phenyl)-1-methyl-ethylamino]-ethyl}-phenylamino)-2-methyl-propionic acid 47240 {(4S,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-10-benzyl-4-[(R)-1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradec-7-yl}-acetic acid 47387 {(4R,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-10-benzyl-4-[(R)-1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-3,3,14,14-tetramethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradec-7-yl}-acetic acid 47447 Montelukast 47457 8-(4-Amino-phenyl)-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 47953 (2-Chloro-4-{2-[2-hydroxy-2-(4-hydroxy-phenyl)-1-methyl-ethylamino]-ethyl}-phenylamino)-acetic acid 47989 2-(4-{2-[2-Hydroxy-2-(4-hydroxy-phenyl)-1-methyl-ethylamino]-ethyl}-phenylamino)-2-methyl-propionic acid 48032 (4-{2-[2-Hydroxy-2-(4-hydroxy-phenyl)-1-methyl-ethylamino]-ethyl}-2-iodo-phenylamino)-acetic acid 48083 1-[1-[2-(3-Aza-bicyclo[3.2.2]non-3-yl)-2-oxo-ethyl]-5-(2-fluoro-phenyl)-9-methyl-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl]-3-[3-(1H-tetrazol-5-yl)-phenyl]-urea 48466 2-(4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzoylamino)-3-phenyl-propionic acid 48595 2-(4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzoylamino)-4-methyl-pentanoic acid 48596 2-(4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzoylamino)-3-methyl-butyric acid 48846 YGGFL-NH2 48898 SID11113941 49021 (4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzoylamino)-acetic acid 49783 SID11114029 50091 SID26751970 50094 SID11114170 50141 RS-(+/-)-6-Br-APD3-Allyl-6-bromo-1-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine-7,8-diol 50142 R-(+)-APD3-Allyl-1-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine-7,8-diol 50143 SID11110817 50185 SID26755662 50187 SID26755670 50214 N-Benzyl-N-{2-methyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3,4-dihydro-quinazolin-6-yl}-benzamide 50215 N-(2-Chloro-benzyl)-N-{2-ethyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3,4-dihydro-quinazolin-6-yl}-benzamide 50222 SID26752108 50224 N-Benzyl-N-{2-ethyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3,4-dihydro-quinazolin-6-yl}-isonicotinamide 50225 N-Benzyl-N-{2-ethyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3,4-dihydro-quinazolin-6-yl}-benzamide 50226 N-{2-Ethyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3,4-dihydro-quinazolin-6-yl}-N-(3-methyl-but-2-enyl)-benzamide 50232 (+/-)-APD3-Allyl-1-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine-7,8-diol 50269 SID11113791 50290 Gepirone 50327 Benzyl-{2-ethyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3,4-dihydro-quinazolin-6-yl}-carbamic acid isobutyl ester 50356 5-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-1,3-dihydro-indol-2-one 50504 N-{4-Oxo-2-propyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3,4-dihydro-quinazolin-6-yl}-N-phenyl-benzamide 50505 N-(2-Chloro-benzyl)-N-{2-methyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3,4-dihydro-quinazolin-6-yl}-benzamide 50798 5'-[2-(4-benzo[d]isothiazol-3-ylhexahydro-1-pyrazinyl)ethyl]spiro[cyclopentane-1,3'-(2',3'-dihydro-1'H-indole)]-2'-one 50799 6-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-3H-benzothiazol-2-one 50822 SID26751605 50846 N-Benzyl-N-{2-isopropyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3,4-dihydro-quinazolin-6-yl}-benzamide 50968 5-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-6-fluoro-1,3-dihydro-indol-2-one 50969 5-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-3,3-dimethyl-1,3-dihydro-indol-2-one 50970 5-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-1-ethyl-1,3-dihydro-indol-2-one 51162 SID29216385 51163 4-amino-5-chloro-N-[(1S-cis-hexahydro-1H-pyrrolizin-1-yl)-methyl]-2-methoxybenzenecarboxamide 51219 Benzyl-{2-butyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3,4-dihydro-quinazolin-6-yl}-carbamic acid isobutyl ester 51220 Thiophene-2-carboxylic acid benzyl-{2-isopropyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3,4-dihydro-quinazolin-6-yl}-amide 51221 Thiophene-2-carboxylic acid benzyl-{2-ethyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3,4-dihydro-quinazolin-6-yl}-amide 51291 4-amino-5-chloro-N-[(1R,7aR)-hexahydro-1H-pyrrolizin-1-ylmethyl]-2-methoxybenzamide 51451 3-{2-[4-(3,4-Dimethyl-phenyl)-piperazin-1-yl]-ethyl}-2,3-dihydro-isoindol-1-one (PD-18126) 51472 6-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-3H-benzooxazol-2-one 51473 8-[4-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-butyl]-8-aza-spiro[4.5]decane-7,9-dione 51902 teleocidin B-4 51909 3-{2-[4-(3,4-Dimethyl-phenyl)-piperidin-1-yl]-ethyl}-2,3-dihydro-isoindol-1-one 52238 (2S,5S)-9-Decyl-5-hydroxymethyl-2-isopropyl-1-methyl-1,4,5,6-tetrahydro-2H-benzo[e][1,4]diazocin-3-one 52276 5-{4-[2-(3,4,5-Trimethoxy-phenyl)-ethyl]-phenyl}-2,3-dihydro-imidazo[2,1-a]isoquinoline 52316 3-[2-(4-Phenyl-piperazin-1-yl)-ethyl]-2,3-dihydro-isoindol-1-one 52338 7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-2-ol 52359 3-{2-[4-(3,4-Dimethyl-phenyl)-piperazin-1-yl]-ethyl}-2,3-dihydro-isoindol-1-one 52364 (R)-3-{2-[4-(3,4-Dimethyl-phenyl)-piperazin-1-yl]-ethyl}-2,3-dihydro-isoindol-1-one 52464 (2S,3S,4R,5R)-5-[6-Amino-2-(3-cyclopentyl-propionylamino)-purin-9-yl]-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 52544 N-[6-Cyclopentylamino-9-((2R,3R,4S,5R)-3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-2-yl]-3-phenyl-propionamide 52580 N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-2-yl]-4-cyclohexyl-butyramide 52614 Cyclohexanecarboxylic acid [6-amino-9-((2R,3R,4S,5R)-3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-2-yl]-amide 52617 6-Phenyl-3-propyl-1,5-dihydro-pyrrolo[3,2-d]pyrimidine-2,4-dione 52683 N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-2-yl]-3-phenyl-propionamide 52857 8-{4-[2-(4-Benzyl-piperazin-1-yl)-2-oxo-ethoxy]-phenyl}-1-butyl-3,7-dihydro-purine-2,6-dione 52919 SID11113999 52938 2-chloro-N6-cyclopentyladenosine 52939 N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-2-yl]-2-cyclohexyl-acetamide 52962 8-(4-Bromo-phenyl)-1-butyl-3,7-dihydro-purine-2,6-dione 52983 3-Cyclopentyl-N-[6-cyclopentylamino-9-((2R,3R,4S,5R)-3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-2-yl]-propionamide 53010 N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-2-yl]-3-cyclopentyl-propionamide 53012 2-Cyclohexyl-N-[9-((2R,3R,4S,5R)-3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-6-ethylamino-9H-purin-2-yl]-acetamide 53156 (S)-3-{(S)-2-[(R)-2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-4-methyl-pentanoylamino}-N-((S)-1-{(S)-1-[(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 53161 2-[4-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-N-(2-hydroxy-ethyl)-acetamide 53201 N-(2-Amino-ethyl)-2-[4-(5,7-dioxo-6-propyl-4,5,6,7-tetrahydro-1H-imidazo[4,5-b]pyridin-2-yl)-phenoxy]-acetamide 53239 6-Butyl-2-{4-[2-(4-ethyl-piperazin-1-yl)-2-oxo-ethoxy]-phenyl}-1,4-dihydro-imidazo[4,5-b]pyridine-5,7-dione 53344 N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-2-yl]-3-((E)-phenyl)-acrylamide 53429 3-{(S)-2-[(S)-2-Acetylamino-3-(3H-imidazol-4-yl)-1-oxo-propylamino]-4-methyl-1-oxo-pentylamino}-N-(1-{(S)-1-[(S)-(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 53562 SID11113857 53671 endothelin-1 53754 8-Phenyl-3,7-dihydro-purine-2,6-dione 53865 4-(1-Butyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)-benzoic acid 54211 Eprosartan 54365 3-[2-Butyl-3-(4-hydroxy-3-methyl-benzyl)-3H-imidazol-4-yl]-2-thiophen-2-ylmethyl-acrylic acid 54435 2-Benzyl-3-[2-butyl-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-acrylic acid 54437 3-[2-Butyl-3-(4-nitro-benzyl)-3H-imidazol-4-yl]-2-thiophen-2-ylmethyl-acrylic acid 54465 [2-Butyl-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-acetic acid 54466 3-[2-Butyl-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-acrylic acid 54611 (2S)-2-{[(2S)-1-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-5-[(diaminomethylidene)amino]-2-[2-(methylamino)acetamido]pentanamido]-3-methylbutanamido]-3-(4-hydroxyphenyl)propanamido]-3-methylpentanamido]-3-(1H-imidazol-4-yl)propanoyl]pyrrolidin-2-yl]formamido}-3-phenylpropanoic acid 54825 Ac-Ser-Tyr-Ser-Nle-Glu-His-D-Phe-Arg-Trp-Gly-Lys-Pro-Val-NH2 54983 2-[2-Butyl-5-(2-carboxy-3-thiophen-2-yl-propenyl)-imidazol-1-ylmethyl]-benzoic acid 54998 (Z)-7-{(1R,2R,3R,5S)-3,5-Dihydroxy-2-[(E)-(S)-3-hydroxy-5-(3-trifluoromethyl-phenyl)-pent-1-enyl]-cyclopentyl}-hept-5-enoic acid 55020 3-[2-Butyl-3-(2-nitro-benzyl)-3H-imidazol-4-yl]-2-thiophen-2-ylmethyl-acrylic acid 55021 3-[2-Butyl-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-2-thiophen-2-ylmethyl-acrylic acid 55033 SID29216066 55034 SID29217531 55075 (3-Bromo-phenyl)-(8H-pyrrolo[3,2-g]quinazolin-4-yl)-amine 55077 7-[(1R,2R,3R,5S)-3,5-Dihydroxy-2-((R)-3-hydroxy-5-p-tolyl-pentyl)-cyclopentyl]-heptanoic acid 55078 7-[(1R,2R,3R,5S)-3,5-Dihydroxy-2-((R)-3-hydroxy-5-o-tolyl-pentyl)-cyclopentyl]-heptanoic acid 55115 7-{(1R,2R,3R,5S)-3,5-Dihydroxy-2-[(R)-3-hydroxy-5-(4-trifluoromethyl-phenyl)-pentyl]-cyclopentyl}-heptanoic acid 55139 Propionaldehyde O-(3-tert-butylamino-2-hydroxy-propyl)-oxime; compound with (E)-but-2-enedioic acid 55140 Propionaldehyde O-(2-hydroxy-3-isopropylamino-propyl)-oxime; compound with (E)-but-2-enedioic acid 55145 7-{(1R,2R,3R,5S)-3,5-Dihydroxy-2-[(R)-3-hydroxy-5-(3-trifluoromethyl-phenyl)-pentyl]-cyclopentyl}-heptanoic acid 55170 7-{(1R,2R,3R,5S)-2-[(R)-5-(2-Fluoro-phenyl)-3-hydroxy-pentyl]-3,5-dihydroxy-cyclopentyl}-heptanoic acid 55181 7-{(1R,2R,3R,5S)-3,5-Dihydroxy-2-[(R)-3-hydroxy-5-(2-trifluoromethyl-phenyl)-pentyl]-cyclopentyl}-heptanoic acid 55195 7-{(1R,2R,3R,5S)-2-[(R)-5-(3-Cyano-phenyl)-3-hydroxy-pentyl]-3,5-dihydroxy-cyclopentyl}-heptanoic acid 55196 7-{(1R,2R,3R,5S)-2-[(R)-5-(3-Ethyl-phenyl)-3-hydroxy-pentyl]-3,5-dihydroxy-cyclopentyl}-heptanoic acid 55265 3-tert-Butylamino-2-hydroxy-propionaldehyde O-ethyl-oxime; compound with (E)-but-2-enedioic acid 55266 2-Hydroxy-3-isopropylamino-propionaldehyde O-propyl-oxime; compound with (E)-but-2-enedioic acid 55295 2-Hydroxy-3-isopropylamino-propionaldehyde O-ethyl-oxime; compound with (E)-but-2-enedioic acid 55297 7-[3,5-Dihydroxy-2-(3-hydroxy-5-phenyl-pentyl)-cyclopentyl]-heptanoic acid 55298 7-{(1R,2R,3R,5S)-2-[(R)-5-(3-Fluoro-phenyl)-3-hydroxy-pentyl]-3,5-dihydroxy-cyclopentyl}-heptanoic acid 55337 7-{(1R,2R,3R,5S)-3,5-Dihydroxy-2-[(R)-3-hydroxy-5-(4-methoxy-phenyl)-pentyl]-cyclopentyl}-heptanoic acid 55338 7-{(1R,2R,3R,5S)-3,5-Dihydroxy-2-[(R)-3-hydroxy-5-(3-methoxy-phenyl)-pentyl]-cyclopentyl}-heptanoic acid 55373 Acetaldehyde O-(3-tert-butylamino-2-hydroxy-propyl)-oxime; compound with (E)-but-2-enedioic acid 55376 7-{(1R,2R,3R,5S)-3,5-Dihydroxy-2-[(R)-3-hydroxy-5-(2-methoxy-phenyl)-pentyl]-cyclopentyl}-heptanoic acid 55381 3-tert-Butylamino-2-hydroxy-propionaldehyde O-propyl-oxime; compound with (E)-but-2-enedioic acid 55384 SID26719716 55397 (3-Bromo-phenyl)-(8-methoxy-quinazolin-4-yl)-amine 55413 Acetaldehyde O-(2-hydroxy-3-isopropylamino-propyl)-oxime; compound with (E)-but-2-enedioic acid 55432 7-{2-[4-(3-Chloro-phenoxy)-3-hydroxy-butyl]-3,5-dihydroxy-cyclopentyl}-heptanoic acid 55467 7-[3,5-Dihydroxy-2-(3-hydroxy-octyl)-cyclopentyl]-heptanoic acid 55498 7-[(1R,2R,4S,5R)-3,5-Dihydroxy-2-((E)-(R)-3-hydroxy-4,4-dimethyl-oct-1-enyl)-cyclopentyl]-hept-5-enoic acid 55503 7-{(1R,2R,3R,5S)-2-[(R)-5-(4-Fluoro-phenyl)-3-hydroxy-pentyl]-3,5-dihydroxy-cyclopentyl}-heptanoic acid 55552 N-(3-bromophenyl)quinazolin-4-amine 55660 1-Propyl-3,7-dihydro-purine-2,6-dione 55852 5-(3-Hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]nonan-7-one 55962 (9S,10R,12R)-2,3,9,10,11,12-hexahydro-10-hydroxy-9-meth yl-1-oxo-9,12-epoxy-1H diindolo[1,2,3-fg:3',2',1'-kl]py rrolo[3,4-i][1,6]benzodiazocine-10-carboxylic acid methyl ester 56001 SID26751887 56052 N-(3-bromophenyl)-1H-pyrazolo[4,3-g]quinazolin-5-amine 56184 1,2,3,4,5,11-Hexahydro-6-(2-hydroxy)phenyl-3-methyl-2,6-methano-6H-azocino[4,5-b]indole 56422 10-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7-benzyl-3,3-dimethyl-6,9-dioxo-1,2-dithia-5,8-diaza-cycloundecane-4-carboxylic acid 56567 5-Chloro-N-(1-ethyl-4-methyl-[1,4]diazepan-6-yl)-2-methoxy-6-methylamino-nicotinamide 56848 5-Chloro-N-(1-ethyl-4-methyl-[1,4]diazepan-6-yl)-2-methoxy-4-methylamino-benzamide 56849 5-Bromo-N-(1-ethyl-4-methyl-[1,4]diazepan-6-yl)-2-methoxy-6-methylamino-nicotinamide 56862 6-Amino-5-chloro-N-(1-ethyl-4-methyl-[1,4]diazepan-6-yl)-2-methoxy-nicotinamide 56892 5-Chloro-6-ethylamino-N-(1-ethyl-4-methyl-[1,4]diazepan-6-yl)-2-methoxy-nicotinamide 56895 5-Bromo-6-ethylamino-N-(1-ethyl-4-methyl-[1,4]diazepan-6-yl)-2-methoxy-nicotinamide 56920 5-Bromo-N-(1-ethyl-4-methyl-[1,4]diazepan-6-yl)-2-methoxy-6-methylamino-nicotinamide 56972 5-Chloro-N-(1-ethyl-4-methyl-[1,4]diazepan-6-yl)-2-methoxy-6-methylamino-nicotinamide 57232 3-(4-Hydroxy-3-methoxy-phenyl)-2-pyridin-2-yl-acrylonitrile 57506 5-Chloro-N-(1-ethyl-4-methyl-[1,4]diazepan-6-yl)-2-methoxy-6-methylamino-nicotinamide 57537 5-Bromo-6-dimethylamino-N-(1-ethyl-4-methyl-[1,4]diazepan-6-yl)-2-methoxy-nicotinamide 57540 5-Bromo-N-(1-ethyl-4-methyl-[1,4]diazepan-6-yl)-2-methoxy-6-methylamino-nicotinamide 57620 3-[3-(Benzothiazol-2-ylsulfanyl)-4-hydroxy-5-methoxy-phenyl]-2-cyano-acrylamide 57632 (S)-7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-ol 57661 4-Amino-5-chloro-2-methoxy-benzoic acid (R)-(1-aza-bicyclo[2.2.2]oct-3-yl) ester 58020 3-(3-Iodo-4-phenoxy-phenyl)-2-pyridin-2-yl-acrylonitrile 58155 3-(4-Hydroxy-phenyl)-2-pyridin-2-yl-acrylonitrile 58182 4-Amino-5-chloro-2-methoxy-benzoic acid (S)-(1-aza-bicyclo[2.2.2]oct-3-yl) ester 58224 N,N-dimethyl-N-(4-(2-p-tolyl-6,7-dihydro-5H-benzo[7]annulene-8-carboxamido)benzyl)tetrahydro-2H-pyran-4-aminium chloride 58349 SID26751774 58465 (+)-N-(4-chlorophenyl)-3-(fluoromethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide 58482 (S)-N-((3R,6S,9S,15S,20aS)-6-((1H-indol-3-yl)methyl)-3-(cyclohexylmethyl)-9-(3-guanidinopropyl)-1,4,7,10,16-pentaoxoicosahydropyrrolo[1,2-a][1,4,7,10,13]pentaazacyclooctadecin-15-yl)-2-acetamido-3-phenylpropanamide 58653 6-(4-Methyl-piperazin-1-yl)-7,8-dihydro-benzo[k]phenanthridine 58836 (5S,11R,14S)-14-amino-5-benzyl-15-(4-hydroxyphenyl)-6,11-dimethyl-4,7,10,13-tetraoxo-3,6,9,12-tetraazapentadecan-1-oic acid 59082 (4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxymethyl)-phosphonic acid 59084 (R)-1-(3-Chloro-phenyl)-2-{(R)-2-[4-(2-hydroxy-ethoxy)-phenyl]-1-methyl-ethylamino}-ethanol 59114 (4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxymethyl)-methyl-phosphinic acid 59116 2-(4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxy)-acetamide 59323 (2S,6R,11S)-6,11-Dimethyl-3-(2-morpholin-4-yl-ethyl)-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocin-8-ol 59369 (2S,6R,11S)-6,11-Dimethyl-3-(2-piperidin-1-yl-ethyl)-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocin-8-ol 59370 (2S,6R,11S)-6,11-Dimethyl-3-(2-pyrrolidin-1-yl-ethyl)-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocin-8-ol 59499 (2S,6R,11S)-3-(2-Diethylamino-ethyl)-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocin-8-ol 59519 2-chloro-11-(4-methylpiperazin-1-yl)dibenzo[b,f][1,4]oxazepine 59532 (2S,6R,11S)-3-(2-Azepan-1-yl-ethyl)-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocin-8-ol 59539 8-Chloro-10-methoxy-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole 59545 [2-(5,6-Difluoro-indol-1-yl)-ethyl]-dimethyl-amine 59573 6-Chloro-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole 59706 (4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxymethyl)-phosphonic acid monoisopropyl ester 59734 (RS)-1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-m-tolyl-urea 59770 1-(4-Chloro-phenyl)-3-(1-methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-urea 59797 1-(4-Chloro-phenyl)-3-[2-oxo-1-(2-oxo-2-pyrrolidin-1-yl-ethyl)-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl]-urea 59816 2-(4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxy)-malonic acid 59826 (1S,2S)-2-(1H-Imidazol-4-yl)-cyclopentylamine 59834 {3-[3-(4-Chloro-phenyl)-ureido]-2-oxo-5-phenyl-2,3-dihydro-benzo[e][1,4]diazepin-1-yl}-acetic acid ethyl ester 59846 2-(4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxy)-N-hydroxy-acetamide 59847 (4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxy)-methanesulfonic acid 59848 SID29217493 59851 8-Chloro-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole 59852 6-Methoxy-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole 59878 8-Chloro-10-methyl-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole 60042 1-(2-chloro-2-phenylethyl)-6-(methylthio)-4-(piperidin-1-yl)-1H-pyrazolo[3,4-d]pyrimidine 60044 N-butyl-1-(2-chloro-2-phenylethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 60061 (2-Indol-1-ylethyl)dimethylamine 60062 [2-(6-Methoxy-indol-1-yl)-ethyl]-dimethyl-amine 60129 7,8-dichloro-1,2,3,4-tetrahydroisoquinoline 60171 7-Chloro-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole 60330 3-{[1-(3-Piperidin-4-yl-propionyl)-piperidine-3-carbonyl]-amino}-propionic acid 60418 [3-(4-Chloro-benzoylamino)-5-(2-fluoro-phenyl)-2-oxo-2,3-dihydro-benzo[e][1,4]diazepin-1-yl]-acetic acid ethyl ester 60419 (RS)-1-(4-Chloro-phenyl)-3-[5-(2-fluoro-phenyl)-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl]-urea 60462 {3-[3-(4-Chloro-phenyl)-ureido]-2-oxo-5-phenyl-2,3-dihydro-benzo[e][1,4]diazepin-1-yl}-acetic acid ethyl ester 60538 (threo)2-(1H-Imidazol-4-yl)-1-methyl-propylamine; compound with 2-(1H-imidazol-4-yl)-1-methyl-propylamine 60573 1-(2-chloro-2-phenylethyl)-6-(methylthio)-N-phenethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 60574 4-(1-(2-chloro-2-phenylethyl)-6-(ethylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-yl)morpholine 60592 2-[2-((3aR,9bR)-6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-4H-9-thia-2,4,6-triaza-fluorene-1,3-dione 60597 SID26756748 60632 4-(1-(2-chloro-2-phenylethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-yl)morpholine 61161 4-(2,4-Dichloro-phenylamino)-6-methoxy-7-(1-methyl-piperidin-4-ylmethoxy)-quinoline-3-carbonitrile 61163 4-(2,4-Dichloro-5-ethoxy-phenylamino)-6-methoxy-7-(1-methyl-piperidin-4-ylmethoxy)-quinoline-3-carbonitrile 61181 Tamsulosin 61187 6-Methoxy-7-(1-methyl-piperidin-4-ylmethoxy)-4-(3,4,5-trimethoxy-phenylamino)-quinoline-3-carbonitrile 61194 4-(2-Chloro-5-methoxy-phenylamino)-6-methoxy-7-(1-methyl-piperidin-4-ylmethoxy)-quinoline-3-carbonitrile 61196 6-Methoxy-4-(5-methoxy-2,4-dimethyl-phenylamino)-7-(1-methyl-piperidin-4-ylmethoxy)-quinoline-3-carbonitrile 61225 4-(2,4-Dichloro-5-methoxy-phenylamino)-6-methoxy-7-(1-methyl-piperidin-3-ylmethoxy)-quinoline-3-carbonitrile 61368 4-(2,4-Dichloro-5-methoxy-phenylamino)-6-methoxy-7-[2-(1-methyl-piperidin-4-yl)-ethoxy]-quinoline-3-carbonitrile 61484 2-phenylimidazoline 61508 N-butyl-1-(2-chloro-2-phenylethyl)-6-(ethylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 61510 1-(2-chloro-2-phenylethyl)-6-(ethylthio)-4-(piperidin-1-yl)-1H-pyrazolo[3,4-d]pyrimidine 61511 N-benzyl-1-(2-chloro-2-phenylethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 61525 4-(2,4-Dichloro-5-methoxy-phenylamino)-6-methoxy-7-(1-methyl-piperidin-4-ylmethoxy)-quinoline-3-carbonitrile 61539 4-(2,4-Dichloro-5-methoxy-phenylamino)-6-methoxy-7-(1-methyl-piperidin-4-yloxy)-quinoline-3-carbonitrile 61691 6-Chloro-5-methylsulfanyl-2,3-dihydro-indole-1-carboxylic acid pyridin-3-ylamide 61707 4-(2,4-Dichloro-5-methoxy-phenylamino)-6-methoxy-7-(1-methyl-piperidin-2-ylmethoxy)-quinoline-3-carbonitrile 61725 4-(2,4-Dimethyl-phenylamino)-6-methoxy-7-(1-methyl-piperidin-4-ylmethoxy)-quinoline-3-carbonitrile 61726 6-Methoxy-4-(5-methoxy-2-methyl-phenylamino)-7-(1-methyl-piperidin-4-ylmethoxy)-quinoline-3-carbonitrile 61773 4-Fluoro-5-(1-hydroxy-2-methylamino-ethyl)-benzene-1,2-diol (6-FEPI) 61800 2-phenyl-3-(piperidin-4-yl)-1H-indole 61811 3-(1-phenethylpiperidin-4-yl)-2-phenyl-1H-indole 62111 Bosutinib 62246 4-(2,4-Dichloro-5-methoxy-phenylamino)-6-methoxy-7-[3-(1-methyl-piperidin-4-yl)-propoxy]-quinoline-3-carbonitrile 62259 SID26751917 62284 1-[3-(2,2-Di-p-tolyl-acetylamino)-propyl]-4-phenyl-piperidine-4-carboxylic acid methyl ester 62518 4-Amino-N-(1-aza-tricyclo[3.3.1.1*3,7*]dec-4-yl)-5-chloro-2-methoxy-benzamide 62605 3-Fluoro-4-(1-hydroxy-2-methylamino-ethyl)-benzene-1,2-diol (2-FEPI) 62698 6-chloro-5-methyl-N-(pyridin-3-yl)indoline-1-carboxamide 62720 SID11114169 62740 4-Phenyl-1-[3-(2-p-tolyl-acetylamino)-propyl]-piperidine-4-carboxylic acid methyl ester 62798 (R)-4-(3,4-Difluoro-phenyl)-1,2-dimethyl-6-oxo-1,4,5,6-tetrahydro-pyridine-3-carboxylic acid {3-[4-cyano-4-(2,4-difluoro-phenyl)-piperidin-1-yl]-propyl}-amide 62817 SID26751556 62944 (R)-4-(3,4-Difluoro-phenyl)-2-methyl-6-oxo-1,4,5,6-tetrahydro-pyridine-3-carboxylic acid {3-[4-cyano-4-(2-cyano-4-fluoro-phenyl)-piperidin-1-yl]-propyl}-amide 63001 (R)-4-(3,4-Difluoro-phenyl)-2-methyl-6-oxo-1,4,5,6-tetrahydro-pyridine-3-carboxylic acid {3-[4-cyano-4-(2,4-difluoro-phenyl)-piperidin-1-yl]-propyl}-amide 63004 (R)-4-(3,4-Difluoro-phenyl)-1,2-dimethyl-6-oxo-1,4,5,6-tetrahydro-pyridine-3-carboxylic acid {3-[4-cyano-4-(2-cyano-4-fluoro-phenyl)-piperidin-1-yl]-propyl}-amide 63064 (R)-4-(3,4-Difluoro-phenyl)-2-methyl-6-oxo-1,4,5,6-tetrahydro-pyridine-3-carboxylic acid {3-[4-cyano-4-(4-fluoro-phenyl)-piperidin-1-yl]-propyl}-amide 63103 (R)-4-(3,4-Difluoro-phenyl)-2-methyl-6-oxo-1,4,5,6-tetrahydro-pyridine-3-carboxylic acid {3-[4-(2-cyano-4-fluoro-phenyl)-piperidin-1-yl]-propyl}-amide 63107 (R)-4-(3,4-Difluoro-phenyl)-2-methyl-6-oxo-1,4,5,6-tetrahydro-pyridine-3-carboxylic acid {3-[4-(4-fluoro-phenyl)-piperidin-1-yl]-propyl}-amide 63253 (R)-4-(3,4-Difluoro-phenyl)-1,2-dimethyl-6-oxo-1,4,5,6-tetrahydro-pyridine-3-carboxylic acid {3-[4-cyano-4-(4-fluoro-phenyl)-piperidin-1-yl]-propyl}-amide 63261 N-(1-Ethyl-pyrrolidin-2-ylmethyl)-2,3-dimethoxy-5-propyl-benzamide 63282 (R)-4-(3,4-Difluoro-phenyl)-1,2-dimethyl-6-oxo-1,4,5,6-tetrahydro-pyridine-3-carboxylic acid {3-[4-(2-cyano-4-fluoro-phenyl)-piperidin-1-yl]-propyl}-amide 63342 N-[3-(4-Cyano-4-phenyl-piperidin-1-yl)-propyl]-2,2-di-p-tolyl-acetamide 63367 N-(1-Ethyl-pyrrolidin-2-ylmethyl)-5-iodo-2,3-dimethoxy-benzamide (epidepride) 63636 N-(1-Ethyl-pyrrolidin-2-ylmethyl)-5-(2-fluoro-ethyl)-2,3-dimethoxy-benzamide 63637 N-(1-Ethyl-pyrrolidin-2-ylmethyl)-3-(3-fluoro-propyl)-2-hydroxy-5,6-dimethoxy-benzamide 63644 [2-(2,6-Dimethoxy-phenoxy)-ethyl]-(4-phenyl-thiochroman-2-ylmethyl)-amine 63658 N-(1-Ethyl-pyrrolidin-2-ylmethyl)-5-(3-fluoro-propyl)-2,3-dimethoxy-benzamide (FP-epidepride) 63677 [2-(2,6-Dimethoxy-phenoxy)-ethyl]-(4-phenyl-thiochroman-2-ylmethyl)-amine 63680 [2-(2,6-Dimethoxy-phenoxy)-ethyl]-(4-phenyl-chroman-2-ylmethyl)-amine 63692 N-(1-Ethyl-pyrrolidin-2-ylmethyl)-3-(2-fluoro-ethyl)-2-hydroxy-5,6-dimethoxy-benzamide 63697 N-(1-Ethyl-pyrrolidin-2-ylmethyl)-2,3-dimethoxy-benzamide 63702 [2-(2,6-Dimethoxy-phenoxy)-ethyl]-(4-phenyl-1,2,3,4-tetrahydro-naphthalen-2-ylmethyl)-amine 63729 N-(1-Ethyl-pyrrolidin-2-ylmethyl)-2-hydroxy-5,6-dimethoxy-3-propyl-benzamide 63741 5-bromo-N-((1-ethylpyrrolidin-2-yl)methyl)-2,3-dimethoxybenzamide 64002 5-(3-hydroxy-propyl)-7-methoxy-2-(3'-methoxy-4'-hydroxy-phenyl)-3-benzo[b]furanecarbaldehyde 64050 2-(4-Methyl-piperazin-1-yl)-4,6-di-thiophen-2-yl-pyrimidine 64051 4-Furan-3-yl-6-methyl-2-(4-methyl-piperazin-1-yl)-pyrimidine 64066 4-Furan-3-yl-2-(4-methyl-piperazin-1-yl)-pyrimidine 64070 4-Furan-2-yl-6-furan-3-yl-2-(4-methyl-piperazin-1-yl)-pyrimidine 64097 2-(4-Methyl-piperazin-1-yl)-4-phenyl-pyrimidine 64103 4,6-Di-furan-3-yl-2-(4-methyl-piperazin-1-yl)-pyrimidine 64104 2-{[2-(2,6-Dimethoxy-phenoxy)-ethylamino]-methyl}-4-phenyl-3,4-dihydro-2H-naphthalen-1-one 64134 2-(2-(benzyloxy)phenoxy)-N-(2-(2,6-dimethoxyphenoxy)ethyl)ethanamine 64144 1-(3-Acetyl-phenyl)-3-{3-[4-(4-fluoro-benzyl)-piperidin-1-yl]-propyl}-urea 64162 4-Furan-3-yl-2-(4-methyl-piperazin-1-yl)-6-thiophen-2-yl-pyrimidine 64202 4-Furan-2-yl-2-(4-methyl-piperazin-1-yl)-pyrimidine 64203 2-(4-Methyl-piperazin-1-yl)-4-thiophen-2-yl-pyrimidine 64233 4-Furan-3-yl-2-(4-methyl-piperazin-1-yl)-6-phenyl-pyrimidine 64264 2-(2-{2-[2-(dipropylamino)ethyl]piperidin-1-yl}acetyl)-2,9-diazatricyclo[9.4.0.0^{3,8}]pentadeca-1(11),3,5,7,12,14-hexaen-10-one 64265 2-(2-{4-[2-(dipropylamino)ethyl]piperidin-1-yl}acetyl)-2,9-diazatricyclo[9.4.0.0^{3,8}]pentadeca-1(11),3,5,7,12,14-hexaen-10-one 64271 [2-(2-Benzyl-phenoxy)-ethyl]-[2-(2,6-dimethoxy-phenoxy)-ethyl]-amine 64323 [2-(2,6-Dimethoxy-phenoxy)-ethyl]-(3-p-tolyl-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-amine 64390 2-(2-{4-[2-(diethylamino)ethyl]piperidin-1-yl}acetyl)-2,9-diazatricyclo[9.4.0.0^{3,8}]pentadeca-1(11),3,5,7,12,14-hexaen-10-one 64391 2-(2-{2-[2-(dibutylamino)ethyl]piperidin-1-yl}acetyl)-2,9-diazatricyclo[9.4.0.0^{3,8}]pentadeca-1(11),3,5,7,12,14-hexaen-10-one 64393 2-(2-{4-[2-(dimethylamino)ethyl]piperidin-1-yl}acetyl)-2,9-diazatricyclo[9.4.0.0^{3,8}]pentadeca-1(11),3,5,7,12,14-hexaen-10-one 64433 2-(2-{4-[2-(dibutylamino)ethyl]piperidin-1-yl}acetyl)-2,9-diazatricyclo[9.4.0.0^{3,8}]pentadeca-1(11),3,5,7,12,14-hexaen-10-one 64690 2-(2-{4-[4-(dimethylamino)butyl]piperidin-1-yl}acetyl)-2,9-diazatricyclo[9.4.0.0^{3,8}]pentadeca-1(11),3,5,7,12,14-hexaen-10-one 64769 SID26753266 64803 2-[2-(2-{2-[bis(2-methylpropyl)amino]ethyl}piperidin-1-yl)acetyl]-2,9-diazatricyclo[9.4.0.0^{3,8}]pentadeca-1(11),3,5,7,12,14-hexaen-10-one 64840 2-(2-{4-[4-(diethylamino)butyl]piperidin-1-yl}acetyl)-2,9-diazatricyclo[9.4.0.0^{3,8}]pentadeca-1(11),3,5,7,12,14-hexaen-10-one 64935 7-((S)-2-((R)-3-hydroxy-4-(3-(trifluoromethyl)phenyl)butyl)-5-oxopyrrolidin-1-yl)heptanoic acid 65241 8-aza-11-deoxyprostaglandin E1 65583 (S)-1-(3-(3-(4-fluorobenzyl)piperidin-1-yl)propyl)-3-(3-acetylphenyl)urea 65721 1-Phenethyl-4-(phenyl-propionyl-amino)-piperidine-4-carboxylic acid methyl ester 65834 2-(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-4-methylsulfanyl-butyrylamino}-3-phenyl-propionylamino)-3-(3H-imidazol-4-yl)-propionylamino]-4-methyl-pentanoylamino}-4-methylsulfanyl-butyrylamino)-succinamic acid 65835 2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-4-methylsulfanyl-butyrylamino}-3-phenyl-propionylamino)-3-(3H-imidazol-4-yl)-propionylamino]-4-methyl-pentanoic acid [1-(1-carbamoyl-propylcarbamoyl)-3-methylsulfanyl-propyl]-amide 65837 3-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-3-phenyl-propionylamino)-N-[1-(1-carbamoyl-2-methyl-propylcarbamoyl)-2-methyl-propyl]-succinamic acid 65972 3-(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-4-methylsulfanyl-butyrylamino}-3-phenyl-propionylamino)-3-phenyl-propionylamino]-4-methyl-pentanoylamino}-4-methylsulfanyl-butyrylamino)-succinamic acid 66050 Neurokinin B 66082 4-[1-Ethoxymethyl-5-(4-fluoro-phenyl)-1H-[1,2,3]triazol-4-yl]-pyridine 66373 H-Glu-Thr-Pro-Asp-c[Cys-Phe-Trp-Lys-Tyr-Cys]-Val-OH 66547 Befiradol 66586 2-(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-4-methylsulfanyl-butyrylamino}-3-phenyl-propionylamino)-3-(3H-imidazol-4-yl)-propionylamino]-4-methyl-pentanoylamino}-4-methylsulfanyl-butyrylamino)-succinic acid 66587 3-(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-4-methylsulfanyl-butyrylamino}-3-phenyl-propionylamino)-3-(4-hydroxy-phenyl)-propionylamino]-4-methyl-pentanoylamino}-4-methylsulfanyl-butyrylamino)-succinamic acid 66588 2-(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-4-methylsulfanyl-butyrylamino}-3-phenyl-propionylamino)-3-(3H-imidazol-4-yl)-propionylamino]-4-methyl-pentanoylamino}-4-methylsulfanyl-butyrylamino)-succinamide 66778 3-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-3-phenyl-propionylamino)-N-(1-carbamoyl-2-methyl-propyl)-succinamic acid 66779 3-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-3-phenyl-propionylamino)-succinamic acid 66780 (S)-5-((S)-1-((S)-1-(2-amino-2-oxoethylamino)-3-methyl-1-oxobutan-2-ylamino)-3-methyl-1-oxobutan-2-ylamino)-4-((S)-2-((R)-2-((S)-2-amino-3-(4-hydroxyphenyl)propanamido)propanamido)-3-phenylpropanamido)-5-oxopentanoic acid 66954 (1S,4S)-2-((S)-2-{(S)-2-[2-Amino-3-(4-phosphonooxy-phenyl)-propionylamino]-4-carboxy-butyrylamino}-4-carboxy-butyrylamino)-3-methyl-pentanoic acid 67094 C-(10,11-Dihydro-5H-dibenzo[a,d]cyclohepten-5-yl)-methylamine 67095 C-(9H-Fluoren-9-yl)-methylamine 67132 C-(5H-Dibenzo[a,d]cyclohepten-5-yl)-methylamine 67177 1-[5-(1H-Imidazol-4-yl)-pentyl]-3-methyl-thiourea 67179 4-(4-Phenyl-butyl)-1H-imidazole 67202 9-(Aminomethyl)-9,10-dihydroanthracene 67756 [(R)-1-Methyl-2-phenyl-1-((S)-1-phenyl-ethylcarbamoyl)-ethyl]-carbamic acid (R)-2-methyl-1-phenyl-propyl ester 67874 {(S)-1-[(R)-1-Methyl-2-phenyl-1-(7-ureido-heptylcarbamoyl)-ethylcarbamoyl]-2-phenyl-ethyl}-carbamic acid tert-butyl ester 67932 2-[4-Amino-5-(4-phenoxy-phenyl)-pyrrolo[2,3-d]pyrimidin-7-yl]-ethanol 67933 7-(2-Amino-ethyl)-5-(4-phenoxy-phenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine 67935 7-Isoxazolidin-4-yl-5-(4-phenoxy-phenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine 67948 [(R)-2-(2,3-Difluoro-phenyl)-1-methyl-1-(7-ureido-heptylcarbamoyl)-ethyl]-carbamic acid (S)-2-methyl-1-phenyl-propyl ester 67969 5-(4-Phenoxy-phenyl)-7-(tetrahydro-pyran-4-yl)-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine 68099 [(R)-1-Methyl-2-phenyl-1-(7-ureido-heptylcarbamoyl)-ethyl]-carbamic acid (S)-2-methyl-1-phenyl-propyl ester 68100 [(R)-1-(8-Hydroxy-octylcarbamoyl)-1-methyl-2-phenyl-ethyl]-carbamic acid (S)-2-methyl-1-phenyl-propyl ester 68117 5-(2,5-Dihydroxy-benzylamino)-N-[2-(4-fluoro-phenyl)-ethyl]-2-hydroxy-benzamide 68130 [(R)-2-(2-Fluoro-phenyl)-1-methyl-1-(7-ureido-heptylcarbamoyl)-ethyl]-carbamic acid (S)-2-methyl-1-phenyl-propyl ester 68135 [(R)-1-(8-Hydroxy-octylcarbamoyl)-1-methyl-2-phenyl-ethyl]-carbamic acid (R)-2-methyl-1-phenyl-propyl ester 68138 Ethanesulfonic acid (3-{4-[4-(1,3-dioxo-tetrahydro-pyrrolo[1,2-c]imidazol-2-yl)-butyl]-piperazin-1-yl}-phenyl)-amide 68222 5-(4-Phenoxy-phenyl)-7-piperidin-4-yl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine 68223 (R)-7-[4-(4-Methyl-piperazin-1-yl)-cyclohexyl]-5-(4-phenoxy-phenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine 68256 7-[4-(4-Methyl-piperazin-1-yl)-cyclohexyl]-5-(4-phenoxy-phenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine 68365 4-(4-Hydroxy-phenylazo)-benzene-1,3-diol 68398 2-(4-Hydroxy-phenyl)-benzothiazol-6-ol 68578 SID26752054 68624 (S)-N-(1-Carbamoyl-2-phenyl-ethyl)-2-[2-(4-hydroxy-phenyl)-acetylamino]-2-methyl-3-phenyl-propionamide 68740 [(S)-1-(1-Carbamoyl-2-phenyl-ethylcarbamoyl)-1-methyl-2-phenyl-ethyl]-carbamic acid tert-butyl ester 68741 [(R)-1-(1-Carbamoyl-2-phenyl-ethylcarbamoyl)-1-methyl-2-phenyl-ethyl]-carbamic acid tert-butyl ester 68799 2-(4-hydroxyphenyl)benzo[d]thiazole-4,6-diol 68838 {(S)-1-[(R)-1-(8-Carbamoyl-octylcarbamoyl)-2-phenyl-ethylcarbamoyl]-1-methyl-2-phenyl-ethyl}-carbamic acid tert-butyl ester 68854 1-(4-{(S)-4-Amino-1-[4-(4-methyl-piperazin-1-yl)-cyclohexyl]-1H-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxy-phenyl)-3-phenyl-urea 68862 5-(4-Phenoxy-phenyl)-7-(4-piperidin-1-yl-cyclohexyl)-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine 68863 5-(4-Phenoxy-phenyl)-7-pyrrolidin-3-yl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine 68864 5-(4-Phenoxy-phenyl)-7-(tetrahydro-furan-3-yl)-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine 68870 2-(3,4-Dihydroxy-phenyl)-benzothiazole-4,6-diol 68878 N-(4-{4-Amino-1-[4-(4-methyl-piperazin-1-yl)-cyclohexyl]-1H-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxy-phenyl)-2,2-dimethyl-3-phenyl-propionamide 68879 N-(4-{4-Amino-1-[4-(4-methyl-piperazin-1-yl)-cyclohexyl]-1H-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxy-phenyl)-3-methyl-3-phenyl-butyramide 68880 (1R,2R)-2-Phenyl-cyclopropanecarboxylic acid (4-{4-amino-1-[4-(4-methyl-piperazin-1-yl)-cyclohexyl]-1H-pyrazolo[3,4-d]pyrimidin-3-ylmethyl}-2-methoxy-phenyl)-amide 68901 {(S)-1-[1-(8-Methoxy-octylcarbamoyl)-2-phenyl-ethylcarbamoyl]-1-methyl-2-phenyl-ethyl}-carbamic acid tert-butyl ester 68902 {(S)-1-[(S)-1-(8-Hydroxy-octylcarbamoyl)-2-phenyl-ethylcarbamoyl]-1-methyl-2-phenyl-ethyl}-carbamic acid tert-butyl ester 68903 {(S)-1-[1-(4-Hydroxy-benzylcarbamoyl)-2-phenyl-ethylcarbamoyl]-1-methyl-2-phenyl-ethyl}-carbamic acid tert-butyl ester 68911 5-(4-Phenoxy-phenyl)-7-(4-piperidin-1-yl-cyclohexyl)-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine 68945 (4-{4-Amino-1-[4-(4-methyl-piperazin-1-yl)-cyclohexyl]-1H-pyrazolo[3,4-d]pyrimidin-3-yl}-phenyl)-phenyl-methanone 68947 3-(4-Benzylamino-3-methoxy-phenyl)-1-[4-(4-methyl-piperazin-1-yl)-cyclohexyl]-1H-pyrazolo[3,4-d]pyrimidin-4-ylamine 68975 N-(4-{4-Amino-1-[4-(4-methyl-piperazin-1-yl)-cyclohexyl]-1H-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxy-phenyl)-benzenesulfonamide 68976 (4-{4-Amino-1-[4-(4-methyl-piperazin-1-yl)-cyclohexyl]-1H-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxy-phenyl)-carbamic acid benzyl ester 69048 7-Methyl-2-propyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3H-imidazo[4,5-b]pyridine 69049 1-[4-(4-Methyl-piperazin-1-yl)-cyclohexyl]-3-(4-phenoxy-phenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-ylamine 69108 8-[2-((S)-2-tert-Butoxycarbonylamino-2-methyl-3-phenyl-propionylamino)-3-phenyl-propionylamino]-octanoic acid 69234 Benzofuran-2-carboxylic acid (4-{4-amino-1-[4-(4-methyl-piperazin-1-yl)-cyclohexyl]-1H-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxy-phenyl)-amide 69266 SID11111001 69333 {(S)-1-[1-(8-Hydroxy-octylcarbamoyl)-2-phenyl-ethylcarbamoyl]-1-methyl-2-phenyl-ethyl}-carbamic acid tert-butyl ester 69334 {(S)-1-[(R)-1-(8-Hydroxy-octylcarbamoyl)-2-phenyl-ethylcarbamoyl]-1-methyl-2-phenyl-ethyl}-carbamic acid tert-butyl ester 69346 (S)-2-[2-((S)-2-{(S)-2-[2-(4-Hydroxy-phenyl)-acetylamino]-3-phenyl-propionylamino}-3-phenyl-propionylamino)-acetylamino]-4-methyl-pentanoic acid ((S)-1-carbamoyl-3-methylsulfanyl-propyl)-amide 69368 SID26751740 69397 N-(4-{4-Amino-1-[4-(4-methyl-piperazin-1-yl)-cyclohexyl]-1H-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxy-phenyl)-3-phenyl-propionamide 69438 (2R,5R)-2-cyclohexyl-2-phenyl-5-((dimethylamino)methyl)-1,3-oxathiolane methiodide 69517 (E)-(1R,2R,3R,5R,12S,13R,16S)-16-Hydroxymethyl-5,9,12,13-tetramethyl-4-oxa-tricyclo[10.3.1.0*3,5*]hexadec-8-en-2-ol 70074 (4,5-Dihydro-oxazol-2-yl)-(2-propyl-cyclohexyl)-amine 70140 Vancomycin 70254 (4,5-Dihydro-oxazol-2-yl)-[3-(3-phenyl-propyl)-bicyclo[2.2.1]hept-2-yl]-amine 70255 (4,5-Dihydro-oxazol-2-yl)-(3-propyl-bicyclo[2.2.1]hept-2-yl)-amine 70256 (4,5-Dihydro-oxazol-2-yl)-(2-phenethyl-cyclohexyl)-amine 70345 N-(4-{(S)-4-Amino-1-[4-(4-methyl-piperazin-1-yl)-cyclohexyl]-1H-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxy-phenyl)-benzamide 70462 Thymeleatoxin 70556 1-[4-(4-Methyl-piperazin-1-yl)-cyclohexyl]-3-(4-phenylamino-phenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-ylamine 70557 3-{4-[(1H-Indol-2-ylmethyl)-amino]-phenyl}-1-[4-(4-methyl-piperazin-1-yl)-cyclohexyl]-1H-pyrazolo[3,4-d]pyrimidin-4-ylamine 70558 N-(4-{4-Amino-1-[4-(4-methyl-piperazin-1-yl)-cyclohexyl]-1H-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxy-phenyl)-phenylaminosulfonamide 70578 2-(5-tert-Butyl-1-methyl-1H-indol-3-yl)-ethylamine 70579 5-tert-Butyl-3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indole 70581 5-Methyl-3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indole 70607 5-Isopropyl-3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indole 70614 (4,5-Dihydro-oxazol-2-yl)-(2-phenyl-cyclohexyl)-amine 70622 (3-Benzyl-bicyclo[2.2.1]hept-2-yl)-(4,5-dihydro-oxazol-2-yl)-amine 70623 (4,5-Dihydro-oxazol-2-yl)-[3-(3-phenyl-allyl)-bicyclo[2.2.1]hept-2-yl]-amine 70656 (2-Benzyl-cyclohexyl)-(4,5-dihydro-oxazol-2-yl)-amine 70657 (4,5-Dihydro-oxazol-2-yl)-[2-(3-phenyl-propyl)-cyclohexyl]-amine 70662 5,6-dihydroxy-7-hydroxymethyl-3,11,11,14-tetramethyl-15-oxo-4-phenylcarbonyloxy-(14R)-tetracyclo[7.5.1.01,5.010,12]pentadeca-2,7-diene 70784 (2R,3R,4S,5R)-2-(6-(cyclohexylamino)-9H-purin-9-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol 70901 (S)-(4-Fluoromethyl-phenyl)-hydroxy-phenyl-acetic acid 1-aza-bicyclo[2.2.2]oct-3-yl ester 70974 5-tert-Butyl-3-(2-pyrrolidin-1-yl-ethyl)-1H-indole 70975 5-Ethyl-3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indole 71067 (R)-Hydroxy-(4-iodo-phenyl)-phenyl-acetic acid 1-aza-bicyclo[2.2.2]oct-3-yl ester 71068 (R)-(4-Fluoromethyl-phenyl)-hydroxy-phenyl-acetic acid 1-aza-bicyclo[2.2.2]oct-3-yl ester 71087 [2-(5-Ethyl-1H-indol-3-yl)-ethyl]-dimethyl-amine 71088 5-Ethyl-3-(2-pyrrolidin-1-yl-ethyl)-1H-indole 71089 [2-(5-Isopropyl-1H-indol-3-yl)-ethyl]-dimethyl-amine 71103 (R)-[4-(2-Fluoro-ethyl)-phenyl]-hydroxy-phenyl-acetic acid 1-aza-bicyclo[2.2.2]oct-3-yl ester 71123 5-Isopropyl-3-(2-pyrrolidin-1-yl-ethyl)-1H-indole 71442 5-(2-Amino-4-chloro-phenyl)-1,3-dimethyl-1,6-dihydro-pyrazolo[4,3-d]pyrimidin-7-one 71794 N-{4-[4-(2-{2-(3,5-Dimethyl-phenyl)-5-[2-(2,5-dimethyl-pyrrolidin-1-yl)-2-oxo-ethyl]-1H-indol-3-yl}-ethylamino)-butyl]-phenyl}-methanesulfonamide 71795 2-(2-(3,5-Dimethyl-phenyl)-3-{2-[4-(4-methanesulfonylamino-phenyl)-butylamino]-ethyl}-1H-indol-5-yl)-N,N-diethyl-acetamide 71803 7-Chloro-3-(3,5-dimethyl-phenyl)-6-nitro-4-((S)-2-piperidin-2-yl-ethoxy)-1H-quinolin-2-one 71812 (S)-Hydroxy-(4-iodo-phenyl)-phenyl-acetic acid 1-aza-bicyclo[2.2.2]oct-3-yl ester 71814 (S)-[4-(2-Fluoro-ethyl)-phenyl]-hydroxy-phenyl-acetic acid 1-aza-bicyclo[2.2.2]oct-3-yl ester 71820 2-(2-(3,5-Dimethyl-phenyl)-3-{2-[4-(4-methanesulfonylamino-phenyl)-butylamino]-ethyl}-1H-indol-5-yl)-N,N-dimethyl-acetamide 71853 (S)-[4-(3-Fluoro-propyl)-phenyl]-hydroxy-phenyl-acetic acid 1-aza-bicyclo[2.2.2]oct-3-yl ester 71870 7-Chloro-3-(3,5-dichloro-phenyl)-2-oxo-4-((S)-2-piperidin-2-yl-ethoxy)-1,2-dihydro-quinoline-6-carboxylic acid pyrimidin-4-ylamide 71871 Pyrazine-2-carboxylic acid [7-chloro-3-(3,5-dimethyl-phenyl)-2-oxo-4-((S)-2-piperidin-2-yl-ethoxy)-1,2-dihydro-quinolin-6-yl]-amide 71880 2-(3,5-Dimethyl-phenyl)-3-{2-[4-(4-methanesulfonylamino-phenyl)-butylamino]-ethyl}-1H-indole-5-carboxylic acid tert-butyl-ethyl-amide 71912 (2-(3,5-Dimethyl-phenyl)-3-{2-[4-(4-methanesulfonylamino-phenyl)-butylamino]-ethyl}-1H-indol-5-yl)-acetic acid ethyl ester 71913 N-{4-[4-(2-{2-(3,5-Dimethyl-phenyl)-5-[2-(2,5-dimethyl-pyrrolidin-1-yl)-1,1-dimethyl-2-oxo-ethyl]-1H-indol-3-yl}-ethylamino)-butyl]-phenyl}-methanesulfonamide 71914 N-[4-(4-{2-[5-(1,1-Dimethyl-2-oxo-2-pyrrolidin-1-yl-ethyl)-2-(3,5-dimethyl-phenyl)-1H-indol-3-yl]-ethylamino}-butyl)-phenyl]-methanesulfonamide 71915 2-(3,5-Dimethyl-phenyl)-3-{2-[4-(4-hydroxy-phenyl)-butylamino]-ethyl}-1H-indole-5-carboxylic acid diisobutylamide 71993 1-[7-Chloro-3-(3,5-dimethyl-phenyl)-2-oxo-4-((S)-2-piperidin-2-yl-ethoxy)-1,2-dihydro-quinolin-6-yl]-3-cyclopropyl-urea 71996 1-[7-Chloro-3-(3,5-dimethyl-phenyl)-2-oxo-4-(2-piperidin-2-yl-ethoxy)-1,2-dihydro-quinolin-6-yl]-3-cyclopropyl-urea 72021 1-[7-Chloro-3-(3,5-dimethyl-phenyl)-2-oxo-4-((S)-2-piperidin-2-yl-ethoxy)-1,2-dihydro-quinolin-6-yl]-3-pyrazin-2-yl-urea 72079 1-[7-Chloro-3-(3,5-dimethyl-phenyl)-2-oxo-4-(2-piperidin-2-yl-ethoxy)-1,2-dihydro-quinolin-6-yl]-3-pyridin-2-yl-urea 72080 1-[7-Chloro-3-(3,5-dimethyl-phenyl)-2-oxo-4-(2-piperidin-2-yl-ethoxy)-1,2-dihydro-quinolin-6-yl]-3-phenyl-urea 72084 2-(3,5-Dimethyl-phenyl)-3-{2-[4-(4-methanesulfonylamino-phenyl)-butylamino]-ethyl}-1H-indole-5-carboxylic acid diisopropylamide 72091 2-(3,5-Dimethyl-phenyl)-3-{2-[4-(4-hydroxy-phenyl)-butylamino]-ethyl}-1H-indole-5-carboxylic acid dimethylamide 72110 N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-5-(pyrrolidine-1-carbonyl)-1H-indol-3-yl]-ethylamino}-butyl)-phenyl]-methanesulfonamide 72113 2-(3,5-Dimethyl-phenyl)-3-{2-[4-(4-methanesulfonylamino-phenyl)-butylamino]-ethyl}-1H-indole-5-carboxylic acid dipropylamide 72181 2-(3,5-Dimethyl-phenyl)-3-{2-[4-(4-methanesulfonylamino-phenyl)-butylamino]-ethyl}-1H-indole-5-carboxylic acid diisobutylamide 72187 (H2C=CCH2)2-Tyr-Aib-Aib-Phe-Leu 72219 7-Chloro-3-indan-5-yl-2-oxo-4-((S)-2-piperidin-2-yl-ethoxy)-1,2-dihydro-quinoline-6-carboxylic acid pyrimidin-4-ylamide 72230 2-(2-(3,5-Dimethyl-phenyl)-3-{2-[4-(4-methanesulfonylamino-phenyl)-butylamino]-ethyl}-1H-indol-5-yl)-N,N-diethyl-isobutyramide 72231 2-(2-(3,5-Dimethyl-phenyl)-3-{2-[4-(4-methanesulfonylamino-phenyl)-butylamino]-ethyl}-1H-indol-5-yl)-N,N-dimethyl-isobutyramide 72232 2-(2-(3,5-Dimethyl-phenyl)-3-{2-[4-(4-methanesulfonylamino-phenyl)-butylamino]-ethyl}-1H-indol-5-yl)-2-methyl-propionic acid ethyl ester 72253 2-(2-(3,5-Dimethyl-phenyl)-3-{2-[4-(4-methanesulfonylamino-phenyl)-butylamino]-ethyl}-1H-indol-5-yl)-N,N-diethyl-propionamide 72254 2-(2-(3,5-Dimethyl-phenyl)-3-{2-[4-(4-methanesulfonylamino-phenyl)-butylamino]-ethyl}-1H-indol-5-yl)-propionic acid ethyl ester 72262 N-[4-(4-{2-[5-(7-Aza-bicyclo[2.2.1]heptane-7-carbonyl)-2-(3,5-dimethyl-phenyl)-1H-indol-3-yl]-ethylamino}-butyl)-phenyl]-methanesulfonamide 72263 N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-5-(2,5-dimethyl-pyrrolidine-1-carbonyl)-1H-indol-3-yl]-ethylamino}-butyl)-phenyl]-methanesulfonamide 72264 N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-5-(morpholine-4-carbonyl)-1H-indol-3-yl]-ethylamino}-butyl)-phenyl]-methanesulfonamide 72265 N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-5-(piperidine-1-carbonyl)-1H-indol-3-yl]-ethylamino}-butyl)-phenyl]-methanesulfonamide 72271 1-[7-Chloro-3-(3,5-dimethyl-phenyl)-2-oxo-4-((S)-2-piperidin-2-yl-ethoxy)-1,2-dihydro-quinolin-6-yl]-3-pyrimidin-4-yl-urea 72302 N-cyclopentyl-9-ethyl-9H-purin-6-amine 72303 SID11111511 72338 Pyrazine-2-carboxylic acid [7-chloro-3-(3,5-dimethyl-phenyl)-2-oxo-4-(2-piperidin-2-yl-ethoxy)-1,2-dihydro-quinolin-6-yl]-amide 72376 RES-701-1(1-10)/[A15]ET-3 72377 RES-701-1(1-10)/[A15]ET-1 72444 SRTX6b 72445 1-[7-Chloro-3-(3,5-dimethyl-phenyl)-2-oxo-4-(2-piperidin-2-yl-ethoxy)-1,2-dihydro-quinolin-6-yl]-3-pyrimidin-4-yl-urea 72464 N-[4-(4-{2-[5-(1,1-Dimethyl-2-morpholin-4-yl-2-oxo-ethyl)-2-(3,5-dimethyl-phenyl)-1H-indol-3-yl]-ethylamino}-butyl)-phenyl]-methanesulfonamide 72465 2-(2-(3,5-Dimethyl-phenyl)-3-{2-[4-(4-methanesulfonylamino-phenyl)-butylamino]-ethyl}-1H-indol-5-yl)-N,N-dipropyl-isobutyramide 72492 RES-701-1-C-terminal analogue 72493 ET-3 72494 RES-701-1(1-10)/[A15]SRTX6b 72497 2-(3,5-Dimethyl-phenyl)-3-{2-[4-(4-methanesulfonylamino-phenyl)-butylamino]-ethyl}-1H-indole-5-carboxylic acid ethyl-isopropyl-amide 72498 1-[7-Chloro-3-(3,5-dimethyl-phenyl)-2-oxo-4-(2-piperidin-2-yl-ethoxy)-1,2-dihydro-quinolin-6-yl]-3-pyridin-3-yl-urea 72520 7-Chloro-3-(4-iodo-3-methyl-phenyl)-2-oxo-4-((S)-2-piperidin-2-yl-ethoxy)-1,2-dihydro-quinoline-6-carboxylic acid pyrimidin-4-ylamide 72521 7-Chloro-3-(3,4-dimethyl-phenyl)-2-oxo-4-((S)-2-piperidin-2-yl-ethoxy)-1,2-dihydro-quinoline-6-carboxylic acid pyrimidin-4-ylamide 72529 2-(3,5-Dimethyl-phenyl)-3-{2-[4-(4-methanesulfonylamino-phenyl)-butylamino]-ethyl}-1H-indole-5-carboxylic acid butyl-ethyl-amide 72530 [S15]ET-1 72564 7-Chloro-3-(3,5-dimethyl-phenyl)-2-oxo-4-(2-piperidin-2-yl-ethoxy)-1,2-dihydro-quinoline-6-carboxylic acid pyrazin-2-ylamide 72565 2-[7-Chloro-3-(3,5-dimethyl-phenyl)-2-oxo-4-(2-piperidin-2-yl-ethoxy)-1,2-dihydro-quinolin-6-yl]-N-pyrimidin-4-yl-acetamide 72576 linear peptide of RES-701-1 72578 RES-701-1 72597 2-(3,5-Dimethyl-phenyl)-3-{2-[4-(4-methanesulfonylamino-phenyl)-butylamino]-ethyl}-1H-indole-5-carboxylic acid ethylamide 72647 7-Chloro-2-oxo-4-(2-piperidin-2-yl-ethoxy)-3-((S)-3,4,5-trimethyl-phenyl)-1,2-dihydro-quinoline-6-carboxylic acid pyrimidin-4-ylamide 72650 2-(3,5-Dimethyl-phenyl)-3-{2-[4-(4-methanesulfonylamino-phenyl)-butylamino]-ethyl}-1H-indole-5-carboxylic acid diethylamide 72651 2-(3,5-Dimethyl-phenyl)-3-{2-[4-(4-methanesulfonylamino-phenyl)-butylamino]-ethyl}-1H-indole-5-carboxylic acid dimethylamide 72653 (2-(3,5-Dimethyl-phenyl)-3-{2-[4-(4-hydroxy-phenyl)-butylamino]-ethyl}-1H-indol-5-yl)-morpholin-4-yl-methanone 72683 7-Chloro-3-(5-chloro-thiophen-2-yl)-2-oxo-4-((S)-2-piperidin-2-yl-ethoxy)-1,2-dihydro-quinoline-6-carboxylic acid pyrimidin-4-ylamide 72684 1-[7-Chloro-3-(3,5-dimethyl-phenyl)-2-oxo-4-((S)-2-piperidin-2-yl-ethoxy)-1,2-dihydro-quinolin-6-yl]-3-pyrimidin-5-yl-urea 72708 1-[7-Chloro-3-(3,5-dimethyl-phenyl)-2-oxo-4-(2-piperidin-2-yl-ethoxy)-1,2-dihydro-quinolin-6-yl]-3-pyrazin-2-yl-urea 72820 2-(3,5-Dimethyl-phenyl)-3-{2-[4-(4-hydroxy-phenyl)-butylamino]-ethyl}-1H-indole-5-carboxylic acid diethylamide 72860 7-Chloro-3-(3,4-dichloro-phenyl)-2-oxo-4-((S)-2-piperidin-2-yl-ethoxy)-1,2-dihydro-quinoline-6-carboxylic acid pyrimidin-4-ylamide 72878 3-aminocyclorphan 72932 5-(3-{[({[({[4-(1-{[2-(3,4-Dichloro-phenyl)-acetyl]-methyl-amino}-2-pyrrolidin-1-yl-ethyl)-phenylcarbamoyl]-methyl}-carbamoyl)-methyl]-carbamoyl}-methyl)-carbamoyl]-methyl}-thioureido)-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)-benzoic acid; compound with triethyl-amine 72957 5-{3-[({[4-(1-{[2-(3,4-Dichloro-phenyl)-acetyl]-methyl-amino}-2-pyrrolidin-1-yl-ethyl)-phenylcarbamoyl]-methyl}-carbamoyl)-methyl]-thioureido}-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)-benzoic acid; compound with triethyl-amine 72969 N-[(S)-1-(3-Amino-phenyl)-2-pyrrolidin-1-yl-ethyl]-2-(3,4-dichloro-phenyl)-N-methyl-acetamide 72970 N-[1-(4-Amino-phenyl)-2-pyrrolidin-1-yl-ethyl]-2-(3,4-dichloro-phenyl)-N-methyl-acetamide 72973 4-chloro-5-(4-(2-(2-ethoxyphenoxy)ethyl)piperazin-1-yl)-2-(7-(4-(2-isopropoxyphenyl)piperazin-1-yl)heptyl)pyridazin-3(2H)-one 72974 4-chloro-5-(4-(2-(2-ethoxyphenoxy)ethyl)piperazin-1-yl)-2-(7-(4-(2-ethoxyphenyl)piperazin-1-yl)heptyl)pyridazin-3(2H)-one 73008 N-[5-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-pyridin-2-yl]-2-bromo-benzamide 73066 butorphan 73067 Cyclorphan 73070 N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-3-chloro-phenyl]-5-fluoro-2-methyl-benzamide 73125 2-Amino-N-[5-(5H,11H-benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-pyridin-2-yl]-benzamide 73214 5-(3-{[4-(1-{[2-(3,4-Dichloro-phenyl)-acetyl]-methyl-amino}-2-pyrrolidin-1-yl-ethyl)-phenylcarbamoyl]-methyl}-thioureido)-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)-benzoic acid; compound with triethyl-amine 73215 5-{3-[4-(1-{[2-(3,4-Dichloro-phenyl)-acetyl]-methyl-amino}-2-pyrrolidin-1-yl-ethyl)-phenyl]-thioureido}-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)-benzoic acid; compound with triethyl-amine 73246 4-chloro-5-(4-(furan-2-carbonyl)piperazin-1-yl)-2-(7-(4-(2-isopropoxyphenyl)piperazin-1-yl)heptyl)pyridazin-3(2H)-one 73318 3-aminobutorphan 73423 4-chloro-5-(4-(2-(2-ethoxyphenoxy)ethyl)piperazin-1-yl)-2-(7-(4-(2-methoxyphenyl)piperazin-1-yl)heptyl)pyridazin-3(2H)-one 73608 2-Butyl-3-(2'-carboxy-biphenyl-4-ylmethyl)-5-chloro-3H-imidazole-4-carboxylic acid 73637 Ac-DPhe-Arg-Trp-NH2 73638 (S)-2-{(S)-2-[(S)-2-acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-3-phenyl-propionylamino}-5-guanidino-pentanoic acid [(S)-1-carbamoyl-2-(1H-indol-3-yl)-ethyl]-amide 73670 N-[5-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-pyridin-2-yl]-5-fluoro-2-methyl-benzamide 73695 N-[5-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-pyridin-2-yl]-N-(3-dimethylamino-propyl)-5-fluoro-2-methyl-benzamide 73743 N-[5-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-pyridin-2-yl]-2-chloro-6-fluoro-benzamide 73744 N-[5-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-pyridin-2-yl]-2,5-dichloro-benzamide 73764 Biphenyl-2-carboxylic acid [5-(5H,11H-benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-pyridin-2-yl]-amide 73779 N-[5-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-pyridin-2-yl]-2,5-difluoro-benzamide 73827 1-[1-[2-(3-Aza-bicyclo[3.2.2]non-3-yl)-2-oxo-ethyl]-5-(2-fluoro-phenyl)-9-methyl-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl]-3-m-tolyl-urea 73828 1-[1-[2-(3-Aza-bicyclo[3.2.2]non-3-yl)-2-oxo-ethyl]-5-(2-fluoro-phenyl)-9-methyl-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl]-3-(3-chloro-phenyl)-urea 73829 1-[1-[2-(3-Aza-bicyclo[3.2.2]non-3-yl)-2-oxo-ethyl]-5-(2-fluoro-phenyl)-9-methyl-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl]-3-(3-bromo-phenyl)-urea 73948 1H-Indole-2-carboxylic acid [(S)-1-(2-fluoro-phenyl)-4-oxo-3,4,6,7-tetrahydro-[1,4]diazepino[6,7,1-hi]indol-3-yl]-amide 73986 1-[1-[2-(3-Aza-bicyclo[3.2.2]non-3-yl)-2-oxo-ethyl]-5-(2-fluoro-phenyl)-9-methyl-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl]-3-(3-methylsulfanyl-phenyl)-urea 74113 N-[5-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-pyridin-2-yl]-2-chloro-4-fluoro-benzamide 74125 3-{3-[1-[2-(3-Aza-bicyclo[3.2.2]non-3-yl)-2-oxo-ethyl]-5-(2-fluoro-phenyl)-9-methyl-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl]-ureido}-benzoic acid 74129 N-[5-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-pyridin-2-yl]-2-chloro-benzamide 74161 N-[5-(3-Dimethylaminomethyl-5H,11H-benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-pyridin-2-yl]-5-fluoro-2-methyl-benzamide 74192 1-(3-Acetyl-phenyl)-3-[1-[2-(3-aza-bicyclo[3.2.2]non-3-yl)-2-oxo-ethyl]-5-(2-fluoro-phenyl)-9-methyl-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl]-urea 74193 1-[1-[2-(3-Aza-bicyclo[3.2.2]non-3-yl)-2-oxo-ethyl]-5-(2-fluoro-phenyl)-9-methyl-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl]-3-(3-methoxy-phenyl)-urea 74197 N-[5-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-pyridin-2-yl]-3-fluoro-2-methyl-benzamide 74324 SID26753615 74466 1-[1-[2-(3-Aza-bicyclo[3.2.2]non-3-yl)-2-oxo-ethyl]-5-(2-fluoro-phenyl)-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl]-3-m-tolyl-urea 74560 N-[5-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-pyridin-2-yl]-2-nitro-benzamide 74561 N-[5-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-pyridin-2-yl]-5-bromo-2-chloro-benzamide 74566 Imidazolidin-2-ylidene-(5-methyl-quinoxalin-6-yl)-amine 74594 N-[5-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-pyridin-2-yl]-2-chloro-5-pyridin-2-yl-benzamide 74792 3,5-Dihydroxy-4-(2-hydroxy-6-methoxycarbonyl-benzoyl)-benzoic acid 2-(4-hydroxy-benzyl)-cyclopentyl ester 74866 2-amino-6-(2,6-dichlorophenyl)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one 74871 Imidazolidin-2-ylidene-quinoxalin-6-yl-amine 74901 6-(2,6-Dichloro-phenyl)-8-methyl-2-[3-(4-methyl-piperazin-1-yl)-propylamino]-8H-pyrido[2,3-d]pyrimidin-7-one 74908 (4-Amino-5-chloro-2-methoxy-phenyl)-carbamic acid 2-diethylamino-ethyl ester 74909 (4-Amino-5-chloro-2-methoxy-phenyl)-carbamic acid 2-(4-methyl-piperidin-1-yl)-ethyl ester 74941 6-(2,6-dichlorophenyl)-8-methyl-2-(phenylamino)pyrido[2,3-d]pyrimidin-7(8H)-one 75006 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid 2-(4-hydroxy-benzoylamino)-cyclopentyl ester 75007 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid 4-(4-hydroxy-benzoylamino)-pyrrolidin-3-yl ester 75045 SID11111794 75046 6-Benzylamino-5,6,7,8-tetrahydro-naphthalene-2,3-diol 75193 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid 2-(4-hydroxy-benzyl)-cyclopentyl ester 75229 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid 3-(4-hydroxy-benzoylamino)-azepan-4-yl ester 75231 Ac-His-DPhe-Arg-Trp-NH2 75253 1-tert-butyl-3-(6-(2,6-dichlorophenyl)-2-(4-(diethylamino)butylamino)pyrido[2,3-d]pyrimidin-7-yl)urea 75258 TCMDC-140940 75277 1,2,3,4,4a,5,6,10b-Octahydro-benzo[f]quinoline-8,9-diol 75293 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid 2-(4-hydroxy-phenoxy)-cyclopentyl ester 75328 3-Chloro-N-[4-(2-chloro-phenyl)-piperazin-1-ylmethyl]-benzamide 75330 N-[4-(2-Cyano-phenyl)-piperazin-1-ylmethyl]-4-methyl-benzamide 75331 N-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-4-methyl-benzamide 75356 3-Chloro-N-[4-(2-methoxy-phenyl)-piperazin-1-ylmethyl]-benzamide 75435 (4-Amino-5-chloro-2-methoxy-phenyl)-carbamic acid 2-(3,5-dimethyl-piperidin-1-yl)-ethyl ester 75439 (4-Amino-5-chloro-2-methoxy-phenyl)-carbamic acid 2-(3-methyl-piperidin-1-yl)-ethyl ester 75477 1-benzyl-3-(6-(2,6-dichlorophenyl)-2-(3-(4-methylpiperazin-1-yl)propylamino)pyrido[2,3-d]pyrimidin-7-yl)urea 75502 1-cyclohexyl-3-(6-(2,6-dichlorophenyl)-2-(3-(4-methylpiperazin-1-yl)propylamino)pyrido[2,3-d]pyrimidin-7-yl)urea 75517 1-(6-(2,6-dichlorophenyl)-2-(3-(4-methylpiperazin-1-yl)propylamino)pyrido[2,3-d]pyrimidin-7-yl)-3-(4-methoxyphenyl)urea 75548 1-(2-amino-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl)-3-tert-butylurea 75565 (4-Amino-5-chloro-2-methoxy-phenyl)-carbamic acid 2-piperidin-1-yl-ethyl ester 75629 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid 4-(4-hydroxy-benzyl)-pyrrolidin-3-yl ester 75641 (2S,3R)-2-(3,5-Bis-trifluoromethyl-benzyloxy)-3-phenyl-morpholine 75661 1-tert-butyl-3-(6-(2,6-dichlorophenyl)-2-(4-(2-(diethylamino)ethoxy)phenylamino)pyrido[2,3-d]pyrimidin-7-yl)urea 75670 2-[(2S,3S)-2-(3,5-Bis-trifluoromethyl-benzyloxy)-3-phenyl-morpholin-4-yl]-acetamide 75673 6-(2,6-dichlorophenyl)-2-(3-(diethylamino)propylamino)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one 75699 (4-Amino-5-chloro-2-methoxy-phenyl)-carbamic acid 2-pyrrolidin-1-yl-ethyl ester 75703 3,5-Dihydroxy-4-(2-hydroxy-6-methoxycarbonyl-benzoyl)-benzoic acid 4-(4-hydroxy-benzyl)-pyrrolidin-3-yl ester 75712 [(2S,3S)-2-(3,5-Bis-trifluoromethyl-benzyloxy)-3-phenyl-morpholin-4-yl]-acetic acid methyl ester 75719 6-(2,6-dichlorophenyl)-8-methyl-2-(3-morpholinopropylamino)pyrido[2,3-d]pyrimidin-7(8H)-one 75727 6-Methyl-5,6,6a,7,8,12b-hexahydro-benzo[a]phenanthridine-10,11-diol 75740 (4-Amino-5-chloro-2-methoxy-phenyl)-carbamic acid 2-azepan-1-yl-ethyl ester 75748 4-Methyl-7-[3-(4-phenyl-piperazin-1-yl)-propoxy]-chromen-2-one 75749 4-Methyl-7-[3-(4-pyridin-2-yl-piperazin-1-yl)-propoxy]-chromen-2-one 75754 4-Methyl-7-[3-(4-pyrimidin-2-yl-piperazin-1-yl)-propoxy]-chromen-2-one 75758 (6aR,12bS)-6-Propyl-5,6,6a,7,8,12b-hexahydro-benzo[a]phenanthridine-10,11-diol 75775 6-(2,6-dichlorophenyl)-8-methyl-2-(4-(4-methylpiperazin-1-yl)phenylamino)pyrido[2,3-d]pyrimidin-7(8H)-one 75784 6-(2,6-dichlorophenyl)-2-(3-(2-(diethylamino)ethoxy)phenylamino)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one 75803 N-[4-(2-Chloro-phenyl)-piperazin-1-ylmethyl]-3-methyl-benzamide 75806 N-[4-(2-Chloro-phenyl)-piperazin-1-ylmethyl]-benzamide 75809 N-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-3-methyl-benzamide 75814 [(2S,3S)-2-(3,5-Bis-trifluoromethyl-benzyloxy)-3-phenyl-morpholin-4-yl]-acetic acid 75846 N-[4-(2-Cyano-phenyl)-piperazin-1-ylmethyl]-benzamide 75857 Tetradecanoic acid 2-hydroxymethyl-5-oxo-tetrahydro-furan-2-ylmethyl ester 75859 5-(((2S,3S)-2-(3,5-bis(trifluoromethyl)benzyloxy)-3-phenylmorpholino)methyl)-2H-1,2,4-triazol-3(4H)-one 75892 N-[4-(3-Naphthalen-1-yl-ureido)-butyl]-2-nitro-benzenesulfonamide 75893 N-[6-(3-Naphthalen-1-yl-ureido)-hexyl]-2-nitro-benzenesulfonamide 75895 8-(3-Oxa-tricyclo[3.2.1.0*2,4*]oct-6-yl)-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 75922 5-[(2S,3S)-2-(3,5-Bis-trifluoromethyl-benzyloxy)-3-phenyl-morpholin-4-ylmethyl]-2,4-dihydro-[1,2,4]triazol-3-one 75923 7-Methyl-2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-imidazo[1,2-a]pyridine 75936 N-{4-[(3-Naphthalen-1-yl-ureido)-methyl]-cyclohexylmethyl}-2-nitro-benzenesulfonamide 75981 1,2,3,4-Tetrahydro-naphthalene-2-carboxylic acid [6-(naphthalene-1-sulfonylamino)-hexyl]-amide 76120 Naphthalene-2-sulfonic acid (4-{[(1,2,3,4-tetrahydro-naphthalen-2-ylmethyl)-amino]-methyl}-cyclohexylmethyl)-amide 76131 4-Chloro-N-[4-(2-chloro-phenyl)-piperazin-1-ylmethyl]-benzamide 76169 4-Chloro-N-[4-(2-methoxy-phenyl)-piperazin-1-ylmethyl]-benzamide 76172 3-Chloro-N-[4-(2-cyano-phenyl)-piperazin-1-ylmethyl]-benzamide 76186 1,2,3,4-Tetrahydro-naphthalene-2-carboxylic acid {4-[(naphthalene-1-sulfonylamino)-methyl]-cyclohexylmethyl}-amide 76193 (2S,3S)-2-(3,5-Bis-trifluoromethyl-benzyloxy)-3-phenyl-morpholine 76199 2-(4-(6-(2,6-dichlorophenyl)-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-ylamino)phenyl)acetic acid 76236 Acetic acid 2-hydroxymethyl-5-oxo-4-tetradec-(E)-ylidene-tetrahydro-furan-2-ylmethyl ester 76255 4-Chloro-N-[4-(2-cyano-phenyl)-piperazin-1-ylmethyl]-benzamide 76290 N-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-benzamide 76310 4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-tetrahydro-4H-furo[3,4-d]pyrimidine-3-carboxylic acid {3-[4-(2-nitro-phenyl)-piperazin-1-yl]-propyl}-amide 76311 4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-tetrahydro-4H-furo[3,4-d]pyrimidine-3-carboxylic acid {3-[4-(2-carbamoyl-phenyl)-piperazin-1-yl]-propyl}-amide 76321 (2R,3R,4S,5R)-2-(2-Chloro-6-methoxyamino-purin-9-yl)-5-isoxazol-3-yl-tetrahydro-furan-3,4-diol 76322 (2R,3R,4S,5R)-2-[2-Chloro-6-(3-iodo-benzylamino)-purin-9-yl]-5-isoxazol-3-yl-tetrahydro-furan-3,4-diol 76325 (2R,3R,4S,5R)-2-(2-Chloro-6-methoxyamino-purin-9-yl)-5-vinyl-tetrahydro-furan-3,4-diol 76355 4-Methoxy-7-[3-(4-pyridin-2-yl-piperazin-1-yl)-propoxy]-chromen-2-one 76357 4-Methoxy-7-[3-(4-phenyl-piperazin-1-yl)-propoxy]-chromen-2-one 76359 (2R,3R,4S,5S)-2-(2-Chloro-6-methoxyamino-purin-9-yl)-5-chloromethyl-tetrahydro-furan-3,4-diol 76361 SID26752072 76365 N-[4-(2-Chloro-phenyl)-piperazin-1-ylmethyl]-4-methyl-benzamide 76385 Naphthalene-2-carboxylic acid [6-(2-nitro-benzenesulfonylamino)-hexyl]-amide 76397 4-Methoxy-7-[3-(4-pyrimidin-2-yl-piperazin-1-yl)-propoxy]-chromen-2-one 76400 4-Methoxy-7-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]-propoxy}-chromen-2-one 76404 5-(6-Benzylamino-purin-9-yl)-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid methylamide 76418 5-[(2S,3S)-2-(3,5-Bis-trifluoromethyl-benzyloxy)-3-phenyl-morpholin-4-ylmethyl]-2,4-dihydro-[1,2,4]triazol-3-one 76420 (2S,3S)-2-(3,5-Bis-trifluoromethyl-benzyloxy)-3-phenyl-4-(2H-[1,2,4]triazol-1-ylmethyl)-morpholine 76429 N-{4-[(Naphthalene-2-sulfonylamino)-methyl]-cyclohexylmethyl}-3-phenyl-2-(toluene-4-sulfonylamino)-propionamide 76440 7-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propoxy}-4-methyl-chromen-2-one 76447 5-Bromo-2,3-dihydro-benzofuran-7-carboxylic acid (1-ethyl-pyrrolidin-2-ylmethyl)-amide 76450 1-(3-{[4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-tetrahydro-4H-furo[3,4-d]pyrimidine-3-carbonyl]-amino}-propyl)-4-phenyl-piperidine-4-carboxylic acid methyl ester 76451 N-(1-Ethyl-pyrrolidin-2-ylmethyl)-5-iodo-2-methoxy-benzamide (iodopride) 76459 5-Iodo-2,3-dihydro-benzofuran-7-carboxylic acid (1-ethyl-pyrrolidin-2-ylmethyl)-amide ((S)-(-)IBF) 76493 1-[6-Amino-8-(3-chloro-phenyl)-9-methyl-9H-purin-2-ylethynyl]-cyclohexanol 76494 1-[6-Amino-8-(2-fluoro-phenyl)-9-methyl-9H-purin-2-ylethynyl]-cyclohexanol 76511 4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-tetrahydro-4H-furo[3,4-d]pyrimidine-3-carboxylic acid [3-(4-cyano-4-phenyl-piperidin-1-yl)-propyl]-amide 76519 1-(3-{[4-(4-Nitro-phenyl)-2,5-dioxo-1,2,5,7-tetrahydro-4H-furo[3,4-d]pyrimidine-3-carbonyl]-amino}-propyl)-4-phenyl-piperidine-4-carboxylic acid methyl ester 76525 (4R,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-5a-methyl-decahydro-benzo[d]azepin-2-one 76528 (1S,4S,5aS,9aS)-1,7,7-Tributyl-4-hydroxymethyl-5a-methyl-decahydro-benzo[d]azepin-2-one 76533 1-[6-Amino-8-(4-fluoro-phenyl)-9-methyl-9H-purin-2-ylethynyl]-cyclohexanol 76534 1-[6-Amino-8-(3-fluoro-phenyl)-9-methyl-9H-purin-2-ylethynyl]-cyclohexanol 76561 (1S,4S,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-5a-methyl-1-octyl-decahydro-benzo[d]azepin-2-one 76570 Naphthalene-1-sulfonic acid (4-{[(2,3-dihydro-benzo[1,4]dioxin-6-ylmethyl)-amino]-methyl}-cyclohexylmethyl)-amide 76647 3-Benzo[1,3]dioxol-5-yl-4-benzyl-5-hydroxy-5-(4-methoxy-phenyl)-5H-furan-2-one 76650 N-[6-(Naphthalene-1-sulfonylamino)-hexyl]-3-phenyl-2-(toluene-4-sulfonylamino)-propionamide 76666 8-(Hexahydro-2,5-methano-pentalen-3a-yl)-3-methyl-1-propyl-3,7-dihydro-purine-2,6-dione 76667 Naphthalene-1-sulfonic acid {4-[3-(3,4-dichloro-phenyl)-ureidomethyl]-cyclohexylmethyl}-amide 76672 1,2,3,4-Tetrahydro-naphthalene-2-carboxylic acid [6-(2-nitro-benzenesulfonylamino)-hexyl]-amide 76695 Naphthalene-1-sulfonic acid [6-(3-naphthalen-1-yl-ureido)-hexyl]-amide 76730 4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-tetrahydro-4H-furo[3,4-d]pyrimidine-3-carboxylic acid [3-(4,4-diphenyl-piperidin-1-yl)-propyl]-amide 76744 1,2,3,4-Tetrahydro-naphthalene-2-carboxylic acid {4-[(8-nitro-naphthalene-2-sulfonylamino)-methyl]-cyclohexylmethyl}-amide 76775 (4S,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-5a-methyl-decahydro-benzo[d]azepin-2-one 76810 (1S,4S,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-1,5a-dimethyl-decahydro-benzo[d]azepin-2-one 76819 1-(2-{[4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-tetrahydro-4H-furo[3,4-d]pyrimidine-3-carbonyl]-amino}-ethyl)-4-phenyl-piperidine-4-carboxylic acid methyl ester 76858 1-{3-[(4-Benzo[1,2,5]oxadiazol-5-yl-2,5-dioxo-1,2,5,7-tetrahydro-4H-furo[3,4-d]pyrimidine-3-carbonyl)-amino]-propyl}-4-phenyl-piperidine-4-carboxylic acid methyl ester 76859 1-{3-[(4-Benzo[1,3]dioxol-5-yl-2,5-dioxo-1,2,5,7-tetrahydro-4H-furo[3,4-d]pyrimidine-3-carbonyl)-amino]-propyl}-4-phenyl-piperidine-4-carboxylic acid methyl ester 76901 1-(4-{[4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-tetrahydro-4H-furo[3,4-d]pyrimidine-3-carbonyl]-amino}-butyl)-4-phenyl-piperidine-4-carboxylic acid methyl ester 77012 1-[6-Amino-8-(3-fluoro-phenyl)-9-methyl-9H-purin-2-ylethynyl]-cyclopentanol 77021 3-((3R,4R)-1-((S)-3-cyclohexyl-3-hydroxypropyl)-3,4-dimethylpiperidin-4-yl)phenol 77033 3-[6-Amino-2-(1-hydroxy-cyclohexylethynyl)-9-methyl-9H-purin-8-yl]-benzonitrile 77039 1-(6-Amino-8-furan-2-yl-9-methyl-9H-purin-2-ylethynyl)-cyclohexanol 77043 1-[6-Amino-8-(3-methoxy-phenyl)-9-methyl-9H-purin-2-ylethynyl]-cyclohexanol 77053 Aristeromycin 77068 1-(6-Amino-9-methyl-8-m-tolyl-9H-purin-2-ylethynyl)-cyclohexanol 77069 1-[6-Amino-8-(4-chloro-phenyl)-9-methyl-9H-purin-2-ylethynyl]-cyclohexanol 77207 Nalbuphine 77475 8-(3-Fluoro-phenyl)-9-methyl-9H-purin-6-ylamine 77476 1-(6-Amino-9-methyl-8-thiophen-2-yl-9H-purin-2-ylethynyl)-cyclohexanol 77498 1-[6-Amino-8-(3-fluoro-phenyl)-9-methyl-9H-purin-2-ylethynyl]-cycloheptanol 77499 1-(6-Amino-9-methyl-9H-purin-2-ylethynyl)-cyclohexanol 77509 3-[(3R,4R)-3,4-Dimethyl-1-((E)-3-phenyl-allyl)-piperidin-4-yl]-phenol 77536 3-[(3R,4R)-3,4-Dimethyl-1-(3-o-tolyl-allyl)-piperidin-4-yl]-phenol 77642 7-Chloro-3-(3,5-dimethyl-phenyl)-4-[2-((S)-6-ethyl-piperidin-2-yl)-ethoxy]-2-oxo-1,2-dihydro-quinoline-6-carboxylic acid pyrimidin-4-ylamide 77686 1-(6-Amino-9-methyl-8-pyridin-2-yl-9H-purin-2-ylethynyl)-cyclohexanol 77701 1-(6-Amino-9-methyl-8-phenyl-9H-purin-2-ylethynyl)-cyclohexanol 77702 (R)-1-(2-(2-hydroxyethyl)piperidin-1-yl)-3-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)prop-2-en-1-one 77726 9-Methyl-2-phenyl-5,9-dihydro-[1,2,4]triazolo[5,1-a][2,7]naphthyridine-6-carboxylic acid methyl ester 77756 1-[6-Amino-8-(3-fluoro-phenyl)-9-methyl-9H-purin-2-yl]-3-ethyl-pent-1-yn-3-ol 77762 SID26752182 77772 7-Chloro-3-(3,5-dimethyl-phenyl)-4-[2-((S)-(R)-6-methyl-piperidin-2-yl)-ethoxy]-2-oxo-1,2-dihydro-quinoline-6-carboxylic acid pyrimidin-4-ylamide 77773 7-Chloro-3-(3,5-dimethyl-phenyl)-4-[2-((S)-(S)-6-methyl-piperidin-2-yl)-ethoxy]-2-oxo-1,2-dihydro-quinoline-6-carboxylic acid pyrimidin-4-ylamide 77785 2-Cyclopentylethynyl-8-(3-fluoro-phenyl)-9-methyl-9H-purin-6-ylamine 77788 4-[6-Amino-8-(3-fluoro-phenyl)-9-methyl-9H-purin-2-yl]-2-methyl-but-3-yn-2-ol 77859 7-Chloro-3-((S)-3,5-dimethyl-4-methyl-phenyl)-4-[2-((S)-6-methyl-piperidin-2-yl)-ethoxy]-2-oxo-1,2-dihydro-quinoline-6-carboxylic acid pyrimidin-4-ylamide 77862 7-Chloro-3-(3,5-dimethyl-phenyl)-2-oxo-4-((S)-2-piperidin-2-yl-ethoxy)-1,2-dihydro-quinoline-6-carboxylic acid pyrimidin-4-ylamide 77959 7-Chloro-3-(3,5-dimethyl-phenyl)-4-[2-(3-methyl-piperidin-2-yl)-ethoxy]-6-nitro-1H-quinolin-2-one 77974 7-Chloro-3-(3,5-dimethyl-phenyl)-6-nitro-4-[2-(1,2,3,4-tetrahydro-isoquinolin-1-yl)-ethoxy]-1H-quinolin-2-one 78007 3-{(3R,4R)-1-[(E)-3-(2-Chloro-phenyl)-allyl]-3,4-dimethyl-piperidin-4-yl}-phenol 78132 (2-Amino-3-methyl-phenyl)-(4-{1-[4-(propane-2-sulfinyl)-phenyl]-ethylidene}-[1,4']bipiperidinyl-1'-yl)-methanone 78221 3-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-1H-quinazoline-2,4-dione 78278 6-(2-Fluoro-phenyl)-4-(1H-indol-3-ylmethyl)-4H-2,3,5,10b-tetraaza-benzo[e]azulene (0.5CHCl3) 78292 Phe-Gly-Gly-Phe-Thr-Gly-Ala-Arg-Lys-Ser-Ala-Arg-Lys-NH2 78300 (4-Fluoro-naphthalen-1-yl)-{4-[4-(propane-2-sulfonyl)-benzyl]-[1,4']bipiperidinyl-1'-yl}-methanone 78315 TCMDC-139245 78316 7-Chloro-3-(3,5-dimethyl-phenyl)-6-nitro-4-[(S)-2-(1,2,3,4-tetrahydro-isoquinolin-3-yl)-ethoxy]-1H-quinolin-2-one 78520 SID26731888 78560 Alsterpaullone 78639 7-Chloro-3-(3,5-dimethyl-phenyl)-4-[2-(5-methyl-piperidin-2-yl)-ethoxy]-6-nitro-1H-quinolin-2-one 78648 N-[4-(3-Bromo-phenylamino)-pyrido[3,2-d]pyrimidin-6-yl]-acrylamide 78758 (R)-2-Methoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol 78914 7-Chloro-2-oxo-4-[2-((S)-6-trifluoromethyl-piperidin-2-yl)-ethoxy]-3-(3,4,5-trimethyl-phenyl)-1,2-dihydro-quinoline-6-carboxylic acid pyrimidin-4-ylamide 79047 Rizatriptan 79259 4-Chloro-N-[6-(2-fluoro-phenyl)-4H-2,3,5,10b-tetraaza-benzo[e]azulen-4-yl]-benzamide 79260 1H-Indole-2-carboxylic acid [6-(2-fluoro-phenyl)-4H-2,3,5,10b-tetraaza-benzo[e]azulen-4-yl]-amide (0.1EtOAc) 79286 [6-(2-Fluoro-phenyl)-4H-2,3,5,10b-tetraaza-benzo[e]azulen-4-yl]-carbamic acid benzyl ester 79324 1-(4-Chloro-phenyl)-3-(1-methyl-6-phenyl-4H-2,3,5,10b-tetraaza-benzo[e]azulen-4-yl)-urea 79370 (+)6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-2,10,11-triol 79371 2-Chloro-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol 79380 (R)-(-)-2-methoxy-N-npropylnorapomorphine 79407 2-Methoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol 79409 SID26754246 79460 N-[4-(3-Bromo-phenylamino)-pyrido[4,3-d]pyrimidin-7-yl]-acrylamide 79472 3-(2'-Carboxy-biphenyl-4-ylmethyl)-5-hydroxymethyl-2-propyl-3H-imidazole-4-carboxylic acid ethyl ester 79484 1-(2'-Carboxy-biphenyl-4-ylmethyl)-2-propyl-1H-imidazole-4,5-dicarboxylic acid 79500 2-Butyl-3-(2'-carboxy-biphenyl-4-ylmethyl)-5-hydroxymethyl-3H-imidazole-4-carboxylic acid 79510 2-Butyl-5-chloro-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3H-imidazole-4-carboxylic acid 79517 1-(2'-Carboxy-biphenyl-4-ylmethyl)-2-hydroxymethyl-5-propyl-1H-pyrrole-3-carboxylic acid 79533 3-(2'-Carboxy-biphenyl-4-ylmethyl)-5-hydroxymethyl-2-propyl-3H-imidazole-4-carboxylic acid 79534 3-(2'-Carboxy-biphenyl-4-ylmethyl)-2-ethyl-5-hydroxymethyl-3H-imidazole-4-carboxylic acid 79542 1-(2'-Carboxy-biphenyl-4-ylmethyl)-3-methoxymethyl-5-propyl-1H-pyrrole-2-carboxylic acid 79572 N-[4-(3-Bromo-phenylamino)-pyrido[3,4-d]pyrimidin-6-yl]-acrylamide 79573 N-(4-m-Tolylamino-pyrido[3,4-d]pyrimidin-6-yl)-acrylamide 79660 [3-(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl)-propyl]-[2-(1,2,3,4-tetrahydro-naphthalen-1-yl)-ethyl]-amine 79688 N-[4-(3-Bromo-4-fluoro-phenylamino)-pyrido[3,4-d]pyrimidin-6-yl]-acrylamide 79705 6-(2-Fluoro-phenyl)-4-(1H-indol-3-ylmethyl)-1-trichloromethyl-4H-2,3,5,10b-tetraaza-benzo[e]azulene (0.5CHCl3) 79727 [3-(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl)-propyl]-phenethyl-amine 79728 [3-(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl)-propyl]-(3-phenyl-propyl)-amine 79736 6-(2-Fluoro-phenyl)-4-(1H-indol-3-ylmethyl)-1-methyl-4H-2,3,5,10b-tetraaza-benzo[e]azulene (0.5H2O.0.4Et2O) 79737 [6-(2-Fluoro-phenyl)-4-(1H-indol-3-ylmethyl)-4H-2,3,5,10b-tetraaza-benzo[e]azulen-1-ylmethyl]-dimethyl-amine (0.22CHCl3) 79757 1H-Indole-2-carboxylic acid [6-(2-fluoro-phenyl)-1-methyl-4H-2,3,5,10b-tetraaza-benzo[e]azulen-4-yl]-amide (0.2EtOAc) 79759 (6-Phenyl-4H-2,3,5,10b-tetraaza-benzo[e]azulen-4-yl)-carbamic acid benzyl ester (0.25EtOAc) 79760 1-(4-Chloro-phenyl)-3-(6-phenyl-4H-2,3,5,10b-tetraaza-benzo[e]azulen-4-yl)-urea 79773 6-(2-Fluoro-phenyl)-4-(1H-indol-3-ylmethyl)-1-phenyl-4H-2,3,5,10b-tetraaza-benzo[e]azulene (0.55CHCl3) 79799 N-[4-(6-Bromo-2,3-dihydro-indol-1-yl)-quinazolin-6-yl]-acrylamide 79800 N-[4-(3-Bromo-4-fluoro-phenylamino)-pyrido[3,2-d]pyrimidin-6-yl]-acrylamide 79801 N-[4-(3-Chloro-4-fluoro-phenylamino)-pyrido[3,4-d]pyrimidin-6-yl]-acrylamide 79958 1-Benzyl-4-[3-(3,4-dihydro-naphthalen-1-yl)-propyl]-piperazine 79990 N-[3-(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl)-propyl]-N'-phenyl-ethane-1,2-diamine 80024 1-[4-(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl)-butyl]-4-(3,4,5,6-tetrahydro-pyridin-2-yl)-piperazine 80048 1-[3-(7-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl)-propyl]-4-(3,4,5,6-tetrahydro-pyridin-2-yl)-piperazine 80081 1-cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine 80090 4'-(4,5-Bis-hydroxymethyl-2-propyl-imidazol-1-ylmethyl)-biphenyl-2-carboxylic acid 80091 1-(2'-Carboxy-biphenyl-4-ylmethyl)-5-hydroxymethyl-2-propyl-1H-imidazole-4-carboxylic acid 80114 1-[3-(1,2,3,4-Tetrahydro-naphthalen-1-yl)-propyl]-4-(3,4,5,6-tetrahydro-pyridin-2-yl)-piperazine 80121 N-(4-(3-bromophenylamino) quinazolin-7-yl)acrylamide 80149 1-Benzyl-4-[3-(5-methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl)-propyl]-piperazine 80156 N-[4-(3-Trifluoromethyl-phenylamino)-quinazolin-6-yl]-acrylamide 80234 N-[4-(4-Benzyloxy-phenylamino)-quinazolin-6-yl]-acrylamide 80235 N-[4-(4-Phenoxy-phenylamino)-quinazolin-6-yl]-acrylamide 80326 N-(4-m-Tolylamino-quinazolin-7-yl)-acrylamide 80327 N-[4-(3-Chloro-phenylamino)-quinazolin-7-yl]-acrylamide 80354 N-[4-(3-Chloro-phenylamino)-quinazolin-6-yl]-acrylamide 80528 N4-(3-bromophenyl)quinazoline-4,6-diamine 80931 N4-(3-bromophenyl)pyrido[3,2-d]pyrimidine-4,6-diamine 80973 N4-(3-bromophenyl)-N6-methylpyrido[3,4-d]pyrimidine-4,6-diamine 81022 N*4*-(3-Bromo-phenyl)-N*6*,N*6*-dimethyl-pyrido[3,4-d]pyrimidine-4,6-diamine 81028 N4-(3-bromophenyl)-N6-methylquinazoline-4,6-diamine 81146 N-(3-bromophenyl)-6-methoxypyrido[3,4-d]pyrimidin-4-amine 81204 N4-(3-bromophenyl)-N6-methylpyrido[3,2-d]pyrimidine-4,6-diamine 81230 N4-(3-bromophenyl)-N6,N6-dimethylpyrido[3,2-d]pyrimidine-4,6-diamine 81260 N*4*-(3-Bromo-phenyl)-pyrido[3,4-d]pyrimidine-4,6-diamine 81327 Dimethyl-[2-(5-[1,2,4]triazol-4-yl-1H-indol-3-yl)-ethyl]-amine 81385 N4-(3-bromophenyl)-N7-methylpyrido[2,3-d]pyrimidine-4,7-diamine 81388 3-(6-Amino-1-methyl-1H-indol-3-yl)-4-(1-methyl-1H-indol-3-yl)-pyrrole-2,5-dione 81403 3-(5-Chloro-1-methyl-1H-indol-3-yl)-4-(1-methyl-1H-indol-3-yl)-pyrrole-2,5-dione 81405 3,4-Bis-(1-methyl-1H-indol-3-yl)-pyrrole-2,5-dione 81407 SID11113656 81458 N4-(3-bromophenyl)-N7,N7-dimethylpyrido[2,3-d]pyrimidine-4,7-diamine 81508 N4-(3-bromophenyl)pyrido[4,3-d]pyrimidine-4,7-diamine 81539 N*4*-Benzyl-pyrido[4,3-d]pyrimidine-4,7-diamine 81694 4-{2-[2-(2,2-Dimethyl-propionyloxymethyl)-2H-tetrazol-5-yl]-6-hydroxy-benzoyl}-3,5-dihydroxy-benzoic acid (R)-2-((S)-4-hydroxy-benzoylamino)-cyclopentyl ester 81720 1-(4-Fluoro-phenyl)-4-(4-hydroxy-4-phenyl-piperidin-1-yl)-butan-1-one 81739 N4-(3-bromophenyl)-N7,N7-dimethylpyrido[4,3-d]pyrimidine-4,7-diamine 81979 3-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-Tyr-NH2 81999 4-(2-Acetylamino-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (R)-2-((S)-4-hydroxy-benzoylamino)-cyclopentyl ester 82000 3,5-Dihydroxy-4-[2-hydroxy-6-(2-methyl-2H-tetrazol-5-yl)-benzoyl]-benzoic acid (R)-2-((S)-4-hydroxy-benzoylamino)-cyclopentyl ester 82013 N-[(R)-5-(6-Cyclopentylamino-purin-9-yl)-4-hydroxy-2-hydroxymethyl-tetrahydro-furan-3-yl]-3,4-dimethyl-benzamide 82075 Biphenyl-4-carboxylic acid {4-[(5-chloro-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amino]-butyl}-amide 82098 4-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-Tyr-NH2 82099 4-N3-C6H4CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-Tyr-NH2 82115 4-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-Tyr-NH2 82116 4-N3-C6H4CH2CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-Tyr-NH2 82117 3,5-Dihydroxy-4-(2-hydroxy-6-methanesulfonylamino-benzoyl)-benzoic acid (R)-2-((S)-4-hydroxy-benzoylamino)-cyclopentyl ester 82133 N4-(3-bromophenyl)-N7-methylpyrido[4,3-d]pyrimidine-4,7-diamine 82139 3-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-Tyr-NH2 82197 24-benzyl-16-(1H-3-indolylmethyl)-25-methyl-13-[1-methyl-(1S)-propyl]perhydrodipyrido[1,2-a:1,2-d]pyrrolo[1,2-j][1,4,7,10,13,16]hexaazacyclooctadecine-6,12,15,18,23,26-hexaone 82248 24-(1H-5-imidazolylmethyl)-16-(1H-3-indolylmethyl)-13-[1-methyl-(1S)-propyl]perhydropyrido[1,2-d]pyrimido[1,6-a]pyrrolo[1,2-j][1,4,7,10,13,16]hexaazacyclooctadecine-6,12,15,18,23,26-hexaone 82253 18-(3-Amino-propyl)-6,15-dibenzyl-3-sec-butyl-16-methyl-1,4,7,13,16,19,24-heptaaza-tricyclo[19.4.0.0*9,13*]pentacosane-2,5,8,14,17,20-hexaone 82286 4-{2-[1-(2,2-Dimethyl-propionyloxymethyl)-1H-tetrazol-5-yl]-6-hydroxy-benzoyl}-3,5-dihydroxy-benzoic acid (R)-2-((S)-4-hydroxy-benzoylamino)-cyclopentyl ester 82301 2-benzylamino-3-(3,4-dichlorobenzyloxy)-1-[1-methylsulfonylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]-(2S)-propan-1-one 82314 N-[2-(5-Methoxy-6-nitro-1H-indol-3-yl)-ethyl]-acetamide 82315 N-(2-(2-iodo-5-methoxy-4-nitro-1H-indol-3-yl)ethyl)acetamide 82316 N-(2-(5-methoxy-4-nitro-1H-indol-3-yl)ethyl)acetamide 82353 N-[5-(6-Cyclopentylamino-purin-9-yl)-4-hydroxy-2-methyl-tetrahydro-furan-3-yl]-4-thiophen-2-yl-butyramide 82358 22-benzyl-13-(1H-3-indolylmethyl)-23-methyl-10-[1-methyl-(1R)-propyl]-1,8,11,14,20,23,25-heptaazatetracyclo[23.2.2.03,8.016,20]nonacosane-2,9,12,15,21,24-hexaone 82379 3-N3-C6H4CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-Tyr-NH2 82401 3,5-Dihydroxy-4-[2-hydroxy-6-(1-methyl-1H-tetrazol-5-yl)-benzoyl]-benzoic acid (R)-2-((S)-4-hydroxy-benzoylamino)-cyclopentyl ester 82402 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (1R,2R)-2-(4-hydroxy-benzoylamino)-cyclopentyl ester 82403 3,5-Dihydroxy-4-(2-hydroxy-6-trifluoromethanesulfonylamino-benzoyl)-benzoic acid (R)-2-((S)-4-hydroxy-benzoylamino)-cyclopentyl ester 82417 N-[5-(6-Cyclopentylamino-purin-9-yl)-4-hydroxy-2-hydroxymethyl-tetrahydro-furan-3-yl]-4-isopropyl-benzamide 82418 N-[5-(6-Cyclopentylamino-purin-9-yl)-4-hydroxy-2-hydroxymethyl-tetrahydro-furan-3-yl]-3-fluoro-4-methyl-benzamide 82433 N-[5-(6-Cyclopentylamino-purin-9-yl)-4-hydroxy-2-hydroxymethyl-tetrahydro-furan-3-yl]-4-thiophen-2-yl-butyramide 82441 3,5-Dihydroxy-4-[2-hydroxy-6-(2,2,2-trifluoro-acetylamino)-benzoyl]-benzoic acid (R)-2-((S)-4-hydroxy-benzoylamino)-cyclopentyl ester 82467 2-(Thiophene-2-carbonyl)-cyclohexanecarboxylic acid [5-(6-cyclopentylamino-purin-9-yl)-4-hydroxy-2-methyl-tetrahydro-furan-3-yl]-amide 82502 Trifluoro-methanesulfonic acid 6-({4-[(biphenyl-4-carbonyl)-amino]-butyl}-propyl-amino)-5,6,7,8-tetrahydro-naphthalen-1-yl ester 82504 1-Phenyl-cyclopentanecarboxylic acid [5-(6-cyclopentylamino-purin-9-yl)-4-hydroxy-2-methyl-tetrahydro-furan-3-yl]-amide 82508 2-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimethoxy-phenyl)-tetrahydro-furan-2-yl]-benzenesulfonyl}-ethanol 82632 N-(2-{4-[(S)-2-Benzylamino-3-(3,4-dichloro-benzyloxy)-propionyl]-piperazin-1-yl}-phenyl)-methanesulfonamide 82634 (S)-2-Benzylamino-3-(3,4-dichloro-benzyloxy)-1-[4-(2-methoxy-phenyl)-piperidin-1-yl]-propan-1-one 82738 SID26752009 82742 N-(2-(5-methoxy-1-methyl-4-nitro-1H-indol-3-yl)ethyl)acetamide 82783 N-(2-(2-iodo-5-methoxy-1-methyl-4-nitro-1H-indol-3-yl)ethyl)acetamide 82784 N-[2-(2-Iodo-5-methoxy-6-nitro-1H-indol-3-yl)-ethyl]-acetamide 82785 N-[2-(5-Methoxy-7-nitro-1H-indol-3-yl)-ethyl]-acetamide 82828 5-(6-Cyclopentylamino-purin-9-yl)-2-hydroxymethyl-tetrahydro-furan-3-ol 82830 N-{1-[(S)-2-Benzylamino-3-(3,4-dichloro-benzyloxy)-propionyl]-4-phenyl-piperidin-4-ylmethyl}-methanesulfonamide 82851 Benzo[1,3]dioxole-5-carboxylic acid [5-(6-cyclopentylamino-purin-9-yl)-4-hydroxy-2-hydroxymethyl-tetrahydro-furan-3-yl]-amide 82869 2-(6-Cyclopentylamino-purin-9-yl)-5-methyl-tetrahydro-furan-3,4-diol 82872 1-Phenyl-cyclohexanecarboxylic acid [5-(6-cyclopentylamino-purin-9-yl)-4-hydroxy-2-methyl-tetrahydro-furan-3-yl]-amide 82879 N-{1-[(S)-2-Benzylamino-3-(3,4-dichloro-benzyloxy)-propionyl]-piperidin-4-ylmethyl}-N-phenyl-methanesulfonamide 82920 N-(2-{1-[(S)-2-Benzylamino-3-(3,4-dichloro-benzyloxy)-propionyl]-piperidin-4-yl}-phenyl)-methanesulfonamide 82921 N-(2-{1-[(S)-2-Benzylamino-3-(3,4-dichloro-benzyloxy)-propionyl]-piperidin-4-yl}-phenyl)-N-methyl-methanesulfonamide 82934 1-(3,4,5-trimethoxybenzyl)-1,2,3,4-tetrahydroisoquinoline-6,7-diol 82942 16,24-dibenzyl-25-methyl-13-[1-methyl-(1S)-propyl]perhydropyrido[1,2-d]pyrimido[1,6-a]pyrrolo[1,2-j][1,4,7,10,13,16]hexaazacyclooctadecine-6,12,15,18,23,26-hexaone 82949 3-Chloro-N-[5-(6-cyclopentylamino-purin-9-yl)-4-hydroxy-2-hydroxymethyl-tetrahydro-furan-3-yl]-4-fluoro-benzamide 83018 SID26751781 83028 24-(1H-5-imidazolylmethyl)-16-(1H-3-indolylmethyl)-13-[1-methyl-(1S)-propyl]perhydrodipyrido[1,2-a:1,2-d]pyrrolo[1,2-j][1,4,7,10,13,16]hexaazacyclooctadecine-6,12,15,18,23,26-hexaone 83051 N-(2-(2-iodo-5-methoxy-1-methyl-1H-indol-3-yl)ethyl)acetamide 83064 (R)-6,10-dimethyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-ol 83076 (S)-2-Benzylamino-3-(3,4-dichloro-benzyloxy)-1-[4-(2-methoxy-phenyl)-piperazin-1-yl]-propan-1-one 83082 N-(S)-1-Aza-bicyclo[2.2.2]oct-3-yl-2-(1-methyl-1H-indol-3-yl)-2-oxo-acetamide 83092 2-[2-(4-Phenyl-piperazin-1-yl)-ethyl]-4,9-dihydro-2,4,9-triaza-fluorene-1,3-dione 83100 3,5-Dihydroxy-4-[2-hydroxy-6-(1H-tetrazol-5-yl)-benzoyl]-benzoic acid (1R,2R)-2-(4-hydroxy-benzoylamino)-cyclopentyl ester 83106 14,22-dibenzyl-23-methyl-11-[1-methyl-(1S)-propyl]-(5aR,11S,14R,16aS,22R,24aS)-perhydrotripyrrolo[1,2-a:1,2-d:1,2-j][1,4,7,10,13,16]hexaazacyclooctadecine-5,10,13,16,21,24-hexaone 83107 16,24-dibenzyl-13-[1-methyl-(1S)-propyl]perhydrodipyrido[1,2-a:1,2-d]pyrrolo[1,2-j][1,4,7,10,13,16]hexaazacyclooctadecine-6,12,15,18,23,26-hexaone 83117 2-benzylamino-3-(3,4-dichlorobenzyloxy)-1-spiro[2,3-dihydro-1H-indene-1,4'-(hexahydropyridine)]-1-yl-(2S)-propan-1-one 83118 (S)-2-Benzylamino-3-(3,4-dichloro-benzyloxy)-1-(4-o-tolyl-piperazin-1-yl)-propan-1-one 83150 (S)-2-Benzylamino-3-(3,4-dichloro-benzyloxy)-1-(4-o-tolyl-piperidin-1-yl)-propan-1-one 83161 N-[2-(2-Iodo-5-methoxy-1-methyl-6-nitro-1H-indol-3-yl)-ethyl]-acetamide 83168 3-(1-(1-benzylpiperidin-4-yl)-1H-indol-3-yl)-4-(1-methyl-1H-indol-3-yl)-1H-pyrrole-2,5-dione 83189 3-(1-Methyl-1H-indol-3-yl)-4-[1-(1-methyl-piperidin-4-yl)-1H-indol-3-yl]-pyrrole-2,5-dione 83217 3-(1-Methyl-1H-indol-3-yl)-4-[1-(1-pyridin-2-ylmethyl-piperidin-4-yl)-1H-indol-3-yl]-pyrrole-2,5-dione 83299 3-(1H-Indol-3-yl)-4-[1-(1-methyl-piperidin-4-yl)-1H-indol-3-yl]-pyrrole-2,5-dione 83315 3-[1-(1-Isopropyl-piperidin-4-yl)-1H-indol-3-yl]-4-(1-methyl-1H-indol-3-yl)-pyrrole-2,5-dione 83342 3-{2-[4-(2-Chloro-phenyl)-piperazin-1-yl]-ethyl}-1,5-dihydro-pyrimido[5,4-b]indole-2,4-dione 83354 3-[1-(1-Ethyl-piperidin-4-yl)-1H-indol-3-yl]-4-(1-methyl-1H-indol-3-yl)-pyrrole-2,5-dione 83355 4-{3-[4-(1-Methyl-1H-indol-3-yl)-2,5-dioxo-2,5-dihydro-1H-pyrrol-3-yl]-indol-1-yl}-piperidine-1-carboxylic acid tert-butyl ester 83387 18-dimethylaminomethyl-(18S)-17-oxa-4,14,21-triazahexacyclo[19.6.1.17,14.02,6.08,13.022,27]nonacosa-1(28),2(6),7(29),8(13),9,11,22(27),23,25-nonaene-3,5-dione; methane sulphonic acid salt 83427 3-[1-(1-Benzyl-pyrrolidin-3-yl)-1H-indol-3-yl]-4-(1-methyl-1H-indol-3-yl)-pyrrole-2,5-dione 83473 2-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyl}-4,9-dihydro-2,4,9-triaza-fluorene-1,3-dione 83492 SID26756513 83500 3-[1-(1-Cyclopropylmethyl-piperidin-4-yl)-1H-indol-3-yl]-4-(1-methyl-1H-indol-3-yl)-pyrrole-2,5-dione 83640 (S)-2-Benzylamino-3-(3,4-dichloro-benzyloxy)-1-(2-methanesulfonyl-2,8-diaza-spiro[4.5]dec-8-yl)-propan-1-one 83665 3-(1-methyl-1H-indol-3-yl)-4-(1-(piperidin-4-yl)-1H-indol-3-yl)-1H-pyrrole-2,5-dione 83784 5-Methyl-6-trifluoromethyl-2,3-dihydro-indole-1-carboxylic acid [6-(pyridin-2-ylmethoxy)-pyridin-3-yl]-amide 83874 3-Cyclopropylmethyl-6-ethyl-8-hydroxy-11-methyl-3,4,5,6-tetrahydro-2H-2,6-methano-benzo[d]azocin-1-one 84019 4-{4-[2-(4-Naphthalen-1-yl-piperazin-1-yl)-ethyl]-phenyl}-thiazol-2-ol 84046 1-{2-[4-(2-Methyl-thiazol-4-yl)-phenyl]-ethyl}-4-naphthalen-1-yl-piperazine 84048 5-Methyl-4-{4-[2-(4-naphthalen-1-yl-piperazin-1-yl)-ethyl]-phenyl}-thiazol-2-ylamine 84109 3,3-Dimethyl-5-[2-(4-naphthalen-1-yl-piperazin-1-yl)-ethyl]-1,3-dihydro-indol-2-one 84126 Methyl-(4-{4-[2-(4-naphthalen-1-yl-piperazin-1-yl)-ethyl]-phenyl}-thiazol-2-yl)-amine 84143 1-Naphthalen-1-yl-4-[2-(4-[1,2,3]thiadiazol-4-yl-phenyl)-ethyl]-piperazine 84144 6-[2-(4-Naphthalen-1-yl-piperazin-1-yl)-ethyl]-3H-benzooxazol-2-one 84146 5-[2-(4-Naphthalen-1-yl-piperazin-1-yl)-ethyl]-1,3-dihydro-indol-2-one 84148 4-{4-[2-(4-Naphthalen-1-yl-piperazin-1-yl)-ethyl]-phenyl}-thiazol-2-ylamine 84170 (+)-Cyclazocine 84172 1-Ethyl-5-[2-(4-naphthalen-1-yl-piperazin-1-yl)-ethyl]-1,3-dihydro-indol-2-one 84176 6-[2-(4-Naphthalen-1-yl-piperazin-1-yl)-ethyl]-3H-benzothiazol-2-one 84337 N-(2-{2-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetylamino}-ethyl)-2-(5-iodo-thiophen-2-yl)-acetamide 84390 dynorphin A 84497 Octanedioic acid (2-{2-[4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetylamino}-ethyl)-amide (thiophen-2-ylmethyl)-amide 84634 HTyr-Gly-Gly-Phe-Leu-Arg-Arg-lle-Arg-Pro-LysNH2 84649 [1-(2-{2-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetylamino}-ethylcarbamoyl)-2-thiophen-2-yl-ethyl]-carbamic acid tert-butyl ester 84683 8-Cyclopentyl-1,3-dimethyl-2-thioxo-1,2,3,7-tetrahydro-purin-6-one 84727 8-Cyclopentyl-1,3-dipropyl-3,7-dihydro-purine-2,6-dithione 84728 8-Cyclopentyl-1,3-dimethyl-6-thioxo-1,3,6,7-tetrahydro-purin-2-one 84729 8-Cyclopentyl-1,3-dimethyl-3,7-dihydro-purine-2,6-dithione 84950 2-Isobutoxy-7-methyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-pyrido[1,2-a]pyrimidin-4-one 84951 2-Isopropoxy-4-oxo-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-4H-pyrido[1,2-a]pyrimidine-7-carboxylic acid ethyl ester 84962 [5-tert-Butoxycarbonylamino-5-(2-{2-[4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetylamino}-ethylcarbamoyl)-pentyl]-carbamic acid benzyl ester 84966 1-(4-(piperidin-1-ylmethyl)benzyl)piperidine 84999 9-Methyl-2-propoxy-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-pyrido[1,2-a]pyrimidin-4-one 85143 [5-Amino-5-(2-{2-[4-(6-oxo-1,3-dipropyl-2-thioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetylamino}-ethylcarbamoyl)-pentyl]-carbamic acid benzyl ester TFA 85166 8-Furan-2-yl-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 85182 [5-Amino-5-(2-{2-[4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetylamino}-ethylcarbamoyl)-pentyl]-carbamic acid benzyl ester TFA 85372 7-Methyl-2-propoxy-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-pyrido[1,2-a]pyrimidin-4-one 85373 2-Propoxy-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-pyrido[1,2-a]pyrimidin-4-one 85407 2-Butoxy-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-pyrido[1,2-a]pyrimidin-4-one 85415 2-Methoxy-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-pyrido[1,2-a]pyrimidin-4-one 85450 SID11114032 85460 2-Ethoxy-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-pyrido[1,2-a]pyrimidin-4-one 85461 2-Isopropoxy-7-methyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-pyrido[1,2-a]pyrimidin-4-one 85498 7-(1-Hydroxy-ethyl)-2-isobutoxy-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-pyrido[1,2-a]pyrimidin-4-one 85500 2-Isopropoxy-4-oxo-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-4H-pyrido[1,2-a]pyrimidine-7-carboxylic acid 85577 8-Methyl-2-propoxy-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-pyrido[1,2-a]pyrimidin-4-one 85826 4-Benzo[1,3]dioxol-5-yl-6-ethoxy-1-(2-methoxy-benzyl)-2-oxo-1,2-dihydro-quinoline-3-carboxylic acid 85857 4-Benzo[1,3]dioxol-5-yl-1-(2-methoxy-benzyl)-2-oxo-1,2-dihydro-quinoline-3-carboxylic acid 85859 4-(2,4-Dimethoxy-phenyl)-6-ethoxy-1-(2-methoxy-benzyl)-2-oxo-1,2-dihydro-quinoline-3-carboxylic acid 85897 1-(2,5-Dimethoxy-benzyl)-6-ethoxy-4-(4-methoxy-phenyl)-2-oxo-1,2-dihydro-quinoline-3-carboxylic acid 85939 3-Benzo[1,3]dioxol-5-yl-5-ethoxy-1-(4-methoxy-benzyl)-1H-indole-2-carboxylic acid 85950 6-Ethoxy-1-(2-methoxy-benzyl)-4-(4-methoxy-phenyl)-2-oxo-1,2-dihydro-quinoline-3-carboxylic acid 85986 4-Benzo[1,3]dioxol-5-yl-5,6-dimethoxy-1-(2-methoxy-benzyl)-2-oxo-1,2-dihydro-quinoline-3-carboxylic acid 86018 4-Benzo[1,3]dioxol-5-yl-6-ethyl-1-(2-methoxy-benzyl)-2-oxo-1,2-dihydro-quinoline-3-carboxylic acid 86099 4-Benzo[1,3]dioxol-5-yl-1-benzo[1,3]dioxol-5-ylmethyl-2-oxo-1,2-dihydro-quinoline-3-carboxylic acid 86101 4-Benzo[1,3]dioxol-5-yl-1-(4-methoxy-benzyl)-2-oxo-1,2-dihydro-quinoline-3-carboxylic acid 86192 2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-3-benzyloxy-propionylamino}-acetylamino)-3-phenyl-propionylamino]-4-methyl-pentanoylamino}-3-hydroxy-butyric acid 86289 3-[1-[3-(3-Dimethylamino-propyl)-4,5,6,7-tetrahydro-1H-indol-2-yl]-meth-(Z)-ylidene]-5-ethanesulfonyl-1,3-dihydro-indol-2-one 86347 3-{2-[5-Methylsulfamoyl-2-oxo-1,2-dihydro-indol-(3Z)-ylidenemethyl]-4,5,6,7-tetrahydro-1H-indol-3-yl}-propionamide 86358 GNF-Pf-1389 86372 3-[1-[3-(3-Dimethylamino-propyl)-4,5,6,7-tetrahydro-1H-indol-2-yl]-meth-(Z)-ylidene]-2-oxo-2,3-dihydro-1H-indole-5-sulfonic acid methylamide 86388 2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-3-hydroxy-butyrylamino}-acetylamino)-3-phenyl-propionylamino]-4-methyl-pentanoylamino}-3-hydroxy-butyric acid 86426 3-[1-(3-Morpholin-4-ylmethyl-4,5,6,7-tetrahydro-1H-indol-2-yl)-meth-(Z)-ylidene]-2-oxo-2,3-dihydro-1H-indole-5-sulfonic acid methylamide 86446 [4-(3-{2-[5-Methylsulfamoyl-2-oxo-1,2-dihydro-indol-(3Z)-ylidenemethyl]-4,5,6,7-tetrahydro-1H-indol-3-yl}-propyl)-piperazin-1-yl]-acetic acid 86516 5-Ethanesulfonyl-3-[1-(3-morpholin-4-ylmethyl-4,5,6,7-tetrahydro-1H-indol-2-yl)-meth-(Z)-ylidene]-1,3-dihydro-indol-2-one 86531 [4-(3-{2-[5-Methylsulfamoyl-2-oxo-1,2-dihydro-indol-(3Z)-ylidenemethyl]-4,5,6,7-tetrahydro-1H-indol-3-yl}-propyl)-piperazin-1-yl]-acetic acid ethyl ester 86536 Propionic acid 1-[4-(4-fluoro-phenyl)-4-oxo-butyl]-3-methyl-4-phenyl-piperidin-4-yl ester 86593 [4-(3-{2-[5-Ethanesulfonyl-2-oxo-1,2-dihydro-indol-(3Z)-ylidenemethyl]-4,5,6,7-tetrahydro-1H-indol-3-yl}-propyl)-piperazin-1-yl]-acetic acid 86705 2-benzoyl-3-(3,4-dihydroxyphenyl)acrylonitrile 86707 2-[(S)-1-(3,5-Bis-trifluoromethyl-benzyloxymethyl)-2,2-diphenyl-ethylamino]-acetamide 86733 1-(1-methyl-1H-indol-5-yl)-3-(quinolin-4-yl)urea 86734 3-(3,4-dihydroxyphenyl)-2-(4-methylbenzoyl)acrylonitrile 86776 (E)-2-Cyano-3-(3,4-dihydroxy-phenyl)-N-(2,4-dimethoxy-phenyl)-acrylamide 86778 1-(1-methylindolin-5-yl)-3-(quinolin-4-yl)urea 86796 5-Ethanesulfonyl-3-[1-{3-[3-(4-hydroxy-piperidin-1-yl)-propyl]-4,5,6,7-tetrahydro-1H-indol-2-yl}-meth-(Z)-ylidene]-1,3-dihydro-indol-2-one 86805 2-Cyano-3-(3,4-dihydroxy-phenyl)-N-[2-(3,4-dimethoxy-phenyl)-ethyl]-acrylamide 86808 (E)-2-Cyano-N-cyclohexyl-3-(3,4-dihydroxy-phenyl)-acrylamide 86830 3-[1-{3-[3-(4-Hydroxy-piperidin-1-yl)-propyl]-4,5,6,7-tetrahydro-1H-indol-2-yl}-meth-(Z)-ylidene]-2-oxo-2,3-dihydro-1H-indole-5-sulfonic acid methylamide 86844 2-[(E)-2-Cyano-3-(3,4-dihydroxy-phenyl)-acryloylamino]-3-phenyl-propionic acid ethyl ester 86853 3-[1-{3-[3-(4-Methyl-piperazin-1-yl)-propyl]-4,5,6,7-tetrahydro-1H-indol-2-yl}-meth-(Z)-ylidene]-2-oxo-2,3-dihydro-1H-indole-5-sulfonic acid methylamide 86887 5-Ethanesulfonyl-3-[1-(3-{3-[4-(2-hydroxy-ethyl)-piperazin-1-yl]-propyl}-4,5,6,7-tetrahydro-1H-indol-2-yl)-meth-(Z)-ylidene]-1,3-dihydro-indol-2-one 86890 3-{2-[5-Ethanesulfonyl-2-oxo-1,2-dihydro-indol-(3Z)-ylidenemethyl]-4,5,6,7-tetrahydro-1H-indol-3-yl}-propionamide 86923 3-[1-(3-{3-[4-(2-Hydroxy-ethyl)-piperazin-1-yl]-propyl}-4,5,6,7-tetrahydro-1H-indol-2-yl)-meth-(Z)-ylidene]-2-oxo-2,3-dihydro-1H-indole-5-sulfonic acid methylamide 86941 3-[1-[3-(3-Morpholin-4-yl-propyl)-4,5,6,7-tetrahydro-1H-indol-2-yl]-meth-(Z)-ylidene]-2-oxo-2,3-dihydro-1H-indole-5-sulfonic acid methylamide 87051 (4S,7S,13S)-13-((S)-2-amino-3-(4-hydroxyphenyl)propanamido)-7-benzyl-3,3,14,14-tetramethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triazacyclotetradecane-4-carboxylic acid 87052 2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-3-tert-butoxy-propionylamino}-acetylamino)-3-phenyl-propionylamino]-4-methyl-pentanoylamino}-3-tert-butoxy-butyric acid 87053 2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-3-hydroxy-propionylamino}-acetylamino)-3-phenyl-propionylamino]-4-methyl-pentanoylamino}-3-tert-butoxy-butyric acid 87054 2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-3-tert-butoxy-butyrylamino}-acetylamino)-3-phenyl-propionylamino]-4-methyl-pentanoylamino}-3-hydroxy-butyric acid 87068 5-Ethanesulfonyl-3-[1-{3-[3-(4-methyl-piperazin-1-yl)-propyl]-4,5,6,7-tetrahydro-1H-indol-2-yl}-meth-(Z)-ylidene]-1,3-dihydro-indol-2-one 87077 9-Aminomethyl-9H-fluorene-3,4-diol 87110 6-Chloro-9-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine-7,8-diol 87111 6-(2-Dipropylamino-ethyl)-biphenyl-2,3,4'-triol 87124 6-(2-Amino-ethyl)-biphenyl-2,3-diol 87152 9-Aminomethyl-9H-fluorene-2,5,6-triol 87162 6-Chloro-9-(4-hydroxy-phenyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepine-7,8-diol 87172 2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-3-tert-butoxy-propionylamino}-acetylamino)-3-phenyl-propionylamino]-4-methyl-pentanoylamino}-3-hydroxy-butyric acid 87173 2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-3-tert-butoxy-butyrylamino}-acetylamino)-3-phenyl-propionylamino]-4-methyl-pentanoylamino}-3-hydroxy-butyric acid 87174 2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-3-hydroxy-butyrylamino}-acetylamino)-3-phenyl-propionylamino]-4-methyl-pentanoylamino}-3-tert-butoxy-butyric acid 87175 13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7-benzyl-3,3,14,14-tetramethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradecane-4-carboxylic acid 87188 (E)-2-Cyano-3-(3,4-dihydroxy-phenyl)-N-(2,6-dimethyl-phenyl)-acrylamide 87189 3-(3,4-Dihydroxy-phenyl)-2-(4-phenyl-piperazine-1-carbonyl)-acrylonitrile 87199 1-(4-Fluoro-phenyl)-4-(4-hydroxy-3-methyl-4-phenyl-piperidin-1-yl)-butan-1-one 87220 Tyrphostin AG-528 87221 SID26751708 87271 (S)-1-(4-(4-methoxybenzo[b]thiophen-2-yl)piperidin-1-yl)-3-(2-methyl-1H-indol-4-yloxy)propan-2-ol 87285 (S)-1-(1H-indol-4-yloxy)-3-(4-(6-fluorobenzo[b]thiophen-2-yl)piperidin-1-yl)propan-2-ol 87292 2-Ethyl-3-[2'-(5-oxo-4,5-dihydro-[1,2,4]oxadiazol-3-yl)-biphenyl-4-ylmethyl]-3H-benzoimidazole-4-carboxylic acid 87296 8-Cyclopropyl-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 87322 1-(4-Fluoro-phenyl)-4-(4-phenyl-piperidin-1-yl)-butan-1-one 87323 1-(1,2-dimethyl-1H-indol-5-yl)-3-(quinolin-4-yl)urea 87324 SID11111922 87326 2-[2-(2-{2-[(S)-2-Acetylamino-3-(4-phosphonooxy-phenyl)-propionylamino]-4-carboxy-butyrylamino}-4-carboxy-butyrylamino)-3-methyl-pentanoylamino]-pentanedioic acid 87330 3-[2'-(5-Oxo-4,5-dihydro-[1,2,4]oxadiazol-3-yl)-biphenyl-4-ylmethyl]-2-propyl-3H-benzoimidazole-4-carboxylic acid 87355 (E)-N-(2-Chloro-phenyl)-2-cyano-3-(3,4-dihydroxy-phenyl)-acrylamide 87359 2-Methoxy-3-[2'-(5-oxo-4,5-dihydro-[1,2,4]oxadiazol-3-yl)-biphenyl-4-ylmethyl]-3H-benzoimidazole-4-carboxylic acid 87383 SID11113600 87384 SID11111894 87386 (3S,3aR,4S,4aR,8aR,9aS)-4-[(Z)-2-((4R,5S)-1,6-Dimethyl-piperidin-2-yl)-vinyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 87387 2-Methylsulfanyl-3-[2'-(5-oxo-4,5-dihydro-[1,2,4]oxadiazol-3-yl)-biphenyl-4-ylmethyl]-3H-benzoimidazole-4-carboxylic acid 87390 Propionic acid 1-[4-(4-fluoro-phenyl)-4-oxo-butyl]-3-methyl-4-phenyl-piperidin-4-yl ester 87391 2-(5-Nitro-2-oxo-1,2-dihydro-indol-3-ylidene)-malononitrile 87417 1-(4-Fluoro-phenyl)-4-(4-hydroxy-3-methyl-4-phenyl-piperidin-1-yl)-butan-1-one 87420 2-(5-Hydroxy-3,4-dihydro-2H-naphthalen-1-ylidene)-malononitrile 87422 1-(2-methylbenzo[d]oxazol-6-yl)-3-(quinolin-4-yl)urea 87436 4-Chloro-2-(4-methyl-piperazin-1-yl)-6-p-tolyl-pyrimidine 87442 2-(5,6-dihydroxy-2,3-dihydro-1H-inden-1-ylidene)malononitrile 87444 Propionic acid 1-[4-(4-fluoro-phenyl)-4-oxo-butyl]-4-phenyl-piperidin-4-yl ester 87448 2-(2-oxoindolin-3-ylidene)malononitrile 87449 2-(6-hydroxy-5-methoxy-2-oxoindolin-3-ylidene)malononitrile 87452 4-[2-[1,6-dimethyl-(2R,6S)-hexahydro-2-pyridinyl]-(E)-1-ethenyl]-3-methyl-(3S,3aS,4R,4aS,8aS,9aR)-perhydrobenzo[f]isobenzofuran-1-one 87453 4-[2-[1,6-dimethyl-(2R,6S)-hexahydro-2-pyridinyl]-(E)-1-ethenyl]-3-methyl-(3S,3aR,4S,4aR,8aR,9aS)-perhydrobenzo[f]isobenzofuran-1-one 87454 (3S,3aS,4R,4aS,8aS,9aR)-4-[(Z)-2-((3R,5S)-1,6-Dimethyl-piperidin-2-yl)-vinyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 87455 3-[2'-(5-Oxo-4,5-dihydro-[1,2,4]oxadiazol-3-yl)-biphenyl-4-ylmethyl]-2-propoxy-3H-benzoimidazole-4-carboxylic acid 87458 2-(1H-Imidazol-2-ylmethylene)-malononitrile 87459 2-(3-Fluoro-4-methoxy-benzylidene)-malononitrile 87467 2-Ethylamino-3-[2'-(5-oxo-4,5-dihydro-[1,2,4]oxadiazol-3-yl)-biphenyl-4-ylmethyl]-3H-benzoimidazole-4-carboxylic acid 87469 2-Methylamino-3-[2'-(5-oxo-4,5-dihydro-[1,2,4]oxadiazol-3-yl)-biphenyl-4-ylmethyl]-3H-benzoimidazole-4-carboxylic acid 87470 4-Imidazol-1-yl-2-(4-methyl-piperazin-1-yl)-pyrimidine 87478 1-(3-chloro-4-methoxyphenyl)-3-(quinolin-4-yl)urea 87479 2-(1H-Indol-5-ylmethylene)-malononitrile 87480 2-(4-Methanesulfinyl-benzylidene)-malononitrile 87493 2-Ethoxy-3-[2'-(5-oxo-4,5-dihydro-[1,2,4]oxadiazol-3-yl)-biphenyl-4-ylmethyl]-3H-benzoimidazole-4-carboxylic acid 87504 (3S,3aS,4R,4aS,8aS,9aR)-4-((2R,6S)-1,6-Dimethyl-piperidin-2-ylethynyl)-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 87511 3-[2'-(5-Oxo-4,5-dihydro-[1,2,4]oxadiazol-3-yl)-biphenyl-4-ylmethyl]-2-propylsulfanyl-3H-benzoimidazole-4-carboxylic acid 87512 1-(4-(methylthio)phenyl)-3-(quinolin-4-yl)urea 87524 2-Butyl-3-[2'-(5-oxo-4,5-dihydro-[1,2,4]oxadiazol-3-yl)-biphenyl-4-ylmethyl]-3H-benzoimidazole-4-carboxylic acid 87527 4-Chloro-6-furan-3-yl-2-(4-methyl-piperazin-1-yl)-pyrimidine 87533 2-(5-hydroxy-2-oxoindolin-3-ylidene)malononitrile 87535 (3S,3aR,4R,4aS,8aR,9aS)-4-[(Z)-2-((3R,5S)-1,6-Dimethyl-piperidin-2-yl)-vinyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 87566 (3S,3aR,4S,4aR,8aR,9aS)-4-((2R,6S)-1,6-Dimethyl-piperidin-2-ylethynyl)-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 87568 2-Ethylsulfanyl-3-[2'-(5-oxo-4,5-dihydro-[1,2,4]oxadiazol-3-yl)-biphenyl-4-ylmethyl]-3H-benzoimidazole-4-carboxylic acid 87576 2-(4,5-dihydroxy-2,3-dihydro-1H-inden-1-ylidene)malononitrile 87577 2-(5,6-dihydroxy-2-oxoindolin-3-ylidene)malononitrile 87627 1-(4-(dimethylamino)phenyl)-3-(quinolin-4-yl)urea 87629 (3S,3aR,4R,4aS,8aR,9aS)-4-((2R,6S)-1,6-Dimethyl-piperidin-2-ylethynyl)-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 87654 2-(5-Hydroxy-1-methyl-2-oxo-1,2-dihydro-indol-3-ylidene)-malononitrile 87681 2-(2H-Pyrazol-3-ylmethylene)-malononitrile 87682 2-(4-Cyano-benzylidene)-malononitrile 87683 4-(2,2-Dicyano-vinyl)-1-hydroxy-pyridinium 87686 2-Chloro-4-(4-methyl-piperazin-1-yl)-6-p-tolyl-pyrimidine 87687 2-Chloro-4-furan-2-yl-6-(4-methyl-piperazin-1-yl)-pyrimidine 87689 2-Chloro-4-(4-methyl-piperazin-1-yl)-6-thiophen-2-yl-pyrimidine 87728 SID26756737 87732 SID24816508 87735 1-(4-(diethylamino)phenyl)-3-(quinolin-4-yl)urea 87754 4-Imidazol-1-yl-6-(4-methyl-piperazin-1-yl)-pyrimidine 87762 (S)-1-(1H-indol-4-yloxy)-3-(4-(benzo[b]thiophen-2-yl)piperidin-1-yl)propan-2-ol 87769 (S)-1-(1H-indol-4-yloxy)-3-(4-(4-methoxybenzo[b]thiophen-2-yl)piperidin-1-yl)propan-2-ol 87780 4-Chloro-2-(4-methyl-piperazin-1-yl)-6-thiophen-2-yl-pyrimidine 87804 3-(3,4-dihydroxyphenyl)-2-(4-fluorobenzoyl)acrylonitrile 87805 (E)-2-Cyano-3-(3,4-dihydroxy-phenyl)-N-(1-phenyl-ethyl)-acrylamide 87828 8-{2-[4-(2-Fluoro-phenyl)-piperazin-1-yl]-ethyl}-8-aza-spiro[4.5]decane-7,9-dione 87847 8-{2-[4-(2,5-Difluoro-phenyl)-piperazin-1-yl]-ethyl}-8-aza-spiro[4.5]decane-7,9-dione 87973 8-{2-[4-(2,5-Dichloro-phenyl)-piperazin-1-yl]-ethyl}-8-aza-spiro[4.5]decane-7,9-dione 88027 3-cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid phenylamide 88046 6-(2-Amino-ethyl)-biphenyl-2,3,4'-triol 88063 6-(2-Dipropylamino-ethyl)-biphenyl-2,3-diol 88079 6-Phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine-7,8-diol 88088 SID11113323 88123 SID11113601 88138 2-(2-chlorobenzoyl)-3-(3,4-dihydroxyphenyl)acrylonitrile 88173 (E)-3-(3,4-Dihydroxy-phenyl)-2-(2,4,6-trimethyl-benzoyl)-acrylonitrile 88174 3-(3,4-dihydroxyphenyl)-2-(thiophene-2-carbonyl)acrylonitrile 88177 (1S,11S)-4-methoxy-10-methyl-10-azatetracyclo[9.8.0.0^{2,7}.0^{14,19}]nonadeca-2,4,6,14(19),15,17-hexaen-5-ol 88182 (6aS,13bS)11-Chloro-7-methyl-5,6a,7,8,9,13b-hexahydro-6H-7-aza-benzo[6,7]cyclohepta[1,2-a]naphthalen-12-ol 88210 3-(3,4-dihydroxyphenyl)-2-(4-nitrobenzoyl)acrylonitrile 88214 (6aR,13bR)11-Chloro-7-methyl-5,6a,7,8,9,13b-hexahydro-6H-7-aza-benzo[6,7]cyclohepta[1,2-a]naphthalen-12-ol 88227 11-Chloro-7-methyl-5,6a,7,8,9,13b-hexahydro-6H-7-aza-benzo[6,7]cyclohepta[1,2-a]naphthalen-12-ol 88228 (6aR,13bS)11-Chloro-7-methyl-5,6a,7,8,9,13b-hexahydro-6H-7-aza-benzo[6,7]cyclohepta[1,2-a]naphthalen-12-ol 88230 11-Methoxy-7-methyl-5,6a,7,8,9,13b-hexahydro-6H-7-aza-benzo[6,7]cyclohepta[1,2-a]naphthalen-12-ol 88232 SID29215403 88246 (6aS,13bR)-11-chloro-7-methyl-6,6a,7,8,9,13b-hexahydro-5H-benzo[d]naphtho[2,1-b]azepin-12-ol 88463 8-{2-[4-(4-Fluoro-phenyl)-piperazin-1-yl]-ethyl}-8-aza-spiro[4.5]decane-7,9-dione 88493 (1R,11S)-4-methoxy-10-methyl-10-azatetracyclo[9.8.0.0^{2,7}.0^{14,19}]nonadeca-2,4,6,14(19),15,17-hexaen-5-ol 88494 7,11-Dimethyl-5,6a,7,8,9,13b-hexahydro-6H-7-aza-benzo[6,7]cyclohepta[1,2-a]naphthalen-12-ol 88501 (S)-2-{(2S,3S)-2-[(S)-2-((S)-2-{(S)-2-Acetylamino-3-[4-(difluoro-phosphono-methyl)-phenyl]-propionylamino}-4-carboxy-butyrylamino)-4-carboxy-butyrylamino]-3-methyl-pentanoylamino}-pentanedioic acid 88534 (1R,11S)-5-methoxy-10-methyl-10-azatetracyclo[9.8.0.0^{2,7}.0^{14,19}]nonadeca-2,4,6,14(19),15,17-hexaen-4-ol 88536 7-Methyl-5,6a,7,8,9,13b-hexahydro-6H-7-aza-benzo[6,7]cyclohepta[1,2-a]naphthalen-12-ol 88591 8-carboxamidocyclazocine 88658 Glu-Pro-Gln-pTyr-Glu-Glu-Ile-Pro-Ile-Tyr-Leu 88659 (S)-4-[(S)-2-Acetylamino-3-(4-phosphonooxy-phenyl)-propionylamino]-4-((S)-1-carbamoyl-3-cyclohexyl-propylcarbamoyl)-butyric acid 88661 3-cyclopropylmethyl-6-ethyl-11-methyl-1-oxo-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid amide 88713 (S)-2-[(2S,3S)-2-((S)-2-{(S)-2-[(S)-2-Acetylamino-3-(4-phosphono-phenyl)-propionylamino]-4-carboxy-butyrylamino}-4-carboxy-butyrylamino)-3-methyl-pentanoylamino]-pentanedioic acid 88714 Glu-Pro-Gln-F2Pmp-Glu-Glu-Ile-Pro-Ile-Tyr-Leu 88772 (S)-4-{(S)-2-Acetylamino-3-[4-(difluoro-phosphono-methyl)-phenyl]-propionylamino}-4-((S)-1-carbamoyl-3-cyclohexyl-propylcarbamoyl)-butyric acid 88787 {[4-((S)-2-Acetylamino-2-{(S)-1-[(3-cyclohexyl-propyl)-methyl-carbamoyl]-propylcarbamoyl}-ethyl)-phenyl]-difluoro-methyl}-phosphonic acid 88788 Phosphoric acid mono-[4-((S)-2-acetylamino-2-{(S)-1-[(3-cyclohexyl-propyl)-methyl-carbamoyl]-propylcarbamoyl}-ethyl)-phenyl] ester 88792 3-desoxy-3-carboxamidonaltrexone 88797 SID29215405 88800 SID26755041 88806 8-{2-[4-(2,5-Dichloro-phenyl)-piperazin-1-yl]-ethyl}-8-aza-spiro[4.5]decan-7-one 88812 [4-((S)-2-Acetylamino-2-{(S)-1-[(3-cyclohexyl-propyl)-methyl-carbamoyl]-propylcarbamoyl}-ethyl)-phenyl]-phosphonic acid 88815 Pramipexole 88827 (S)-4-[(S)-2-Acetylamino-3-(4-phosphono-phenyl)-propionylamino]-4-[(3-cyclohexyl-propyl)-methyl-carbamoyl]-butyric acid 88828 (S)-4-{(S)-2-Acetylamino-3-[4-(difluoro-phosphono-methyl)-phenyl]-propionylamino}-4-[(3-cyclohexyl-propyl)-methyl-carbamoyl]-butyric acid 88923 (R)-2-(4-Amino-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-6-ylamino)-propionamide 88929 2-(4-Amino-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-6-ylamino)-propionamide 88930 (S)-2-(4-Amino-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-6-ylamino)-propionamide 88936 N-(3-chloro-4-fluorophenyl)-6,7-dimethoxyquinazolin-4-amine 89004 2-(4-Methylamino-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-6-ylsulfanyl)-hexanoic acid amide 89122 1-[6-(2,6-Dichloro-phenyl)-2-(4-diethylamino-butylamino)-pyrido[2,3-d]pyrimidin-7-yl]-3-phenyl-urea 89123 1-[6-(2,6-Dichloro-phenyl)-2-(4-diethylamino-butylamino)-pyrido[2,3-d]pyrimidin-7-yl]-3-ethyl-urea 89326 1-tert-Butyl-3-{6-(2,6-dichloro-phenyl)-2-[3-(4-methyl-piperazin-1-yl)-propylamino]-pyrido[2,3-d]pyrimidin-7-yl}-urea 89378 1-((R)-5-Cyclohexyl-1-methyl-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-m-tolyl-urea 89526 SID26751629 89534 3-[4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-phenyl]-5-propyl-thiophene-2-sulfonic acid benzoylamide 89561 (6aR,10aR)-6,6,9-trimethyl-3-(2-methyloctan-2-yl)-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol 89572 3-[4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-phenyl]-5-pentyl-thiophene-2-sulfonic acid benzoylamide 89669 2-(4-bromo-2,5-dimethoxyphenyl)ethylamine 89682 9-Ethyl-8-phenylethynyl-9H-purin-6-ylamine 89688 4'-(1,1-dimethyl-heptyl)-3,5-dimethyl-biphenyl 89689 4-(1,1-dimethyl-heptyl)-3',5'-dimethyl-biphenyl-2-ol 89784 3-[4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-phenyl]-5-isobutyl-thiophene-2-sulfonic acid benzoylamide 89785 3-[4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-phenyl]-5-morpholin-4-ylmethyl-thiophene-2-sulfonic acid benzoylamide 89901 4-Fluoro-N-{2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-benzamide 89932 5-Ethyl-3-[4-(2-ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-phenyl]-thiophene-2-sulfonic acid benzoylamide 89948 4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-biphenyl-2-sulfonic acid benzoylamide 89983 3-[4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-phenyl]-5-methyl-thiophene-2-sulfonic acid benzoylamide 89985 3-[4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-phenyl]-5-trimethylsilanyl-thiophene-2-sulfonic acid benzoylamide 89986 5-Benzyl-3-[4-(2-ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-phenyl]-thiophene-2-sulfonic acid benzoylamide 90014 3-[4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-phenyl]-thiophene-2-sulfonic acid benzoylamide 90093 1-phenyl-4-((4-phenyl-1H-pyrrol-2-yl)methyl)piperazine 90244 4-(4-Chloro-phenyl)-1-[5-(4-fluoro-phenyl)-1H-pyrrol-2-ylmethyl]-piperidin-4-ol 90268 1-[5-(5-Ethanesulfonyl-2-methoxy-phenyl)-1H-pyrrol-2-ylmethyl]-4-(2-methoxy-phenyl)-piperazine 90269 1-[5-(4-Fluoro-phenyl)-1H-pyrrol-2-ylmethyl]-4-(2-methoxy-phenyl)-piperazine 90386 1-(4-Fluoro-phenyl)-4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butan-1-one 90416 7-Chloro-2-methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-6-ol 90449 7-Chloro-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-6-ol 90450 6-Chloro-1-phenyl-2-propyl-1,2,3,4-tetrahydro-isoquinolin-7-ol 90517 1-Phenyl-6-chloro-7-hydroxy-1,2,3,4-tetrahydroisoquinoline 90660 SID26752022 90664 SID11113850 90665 1-(4-Chloro-benzyl)-4-[3-(4-chloro-phenyl)-isoxazol-5-yl]-piperidine 90758 1-(1-Benzyl-piperidin-4-yl)-3-(3-methoxy-naphthalen-2-yl)-propan-2-one 90847 3-(4-Methyl-piperidin-1-ylmethyl)-1H-indole 90862 (1-Benzyl-piperidin-4-yl)-acetic acid 3-methoxy-naphthalen-2-yl ester 90866 SID46500376 90867 SID26755694 90873 4-Chloro-benzoic acid 1-benzyl-piperidin-4-ylmethyl ester 90874 3-Methoxy-naphthalene-2-carboxylic acid (1-benzyl-pyrrolidin-3-yl)-amide 90890 3-Methoxy-naphthalene-2-carboxylic acid 1-benzyl-piperidin-4-ylmethyl ester 90892 1-Benzyl-4-[2-(3-methoxy-naphthalen-2-yloxy)-ethyl]-piperidine 90988 3-(1-Benzyl-piperidin-4-yl)-1-(3-methoxy-naphthalen-2-yl)-propan-1-one 90998 3-(4-Phenyl-piperidin-1-ylmethyl)-1H-indole 91029 1-Benzyl-4-(3-methoxy-naphthalen-2-ylmethoxymethyl)-piperidine 91030 3-Methoxy-naphthalene-2-carboxylic acid 1-benzyl-pyrrolidin-3-ylmethyl ester 91060 N-((1-benzylpiperidin-4-yl)methyl)-3-methoxy-2-naphthamide 91207 1-(4-Chloro-benzyl)-4-[5-(4-chloro-phenyl)-isoxazol-3-yl]-piperidine 91269 4-[5-(4-Chloro-phenyl)-4-methyl-1H-pyrazol-3-yl]-1-phenethyl-piperidine 91270 1-(4-Chloro-benzyl)-4-[5-(4-chloro-phenyl)-2H-pyrazol-3-yl]-piperidine 91308 8-Chloro-5-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ol 91332 1-Benzyl-6-chloro-7-hydroxy-N-methyl-1,2,3,4-tetrahydroisoquinoline 91349 1-Phenyl-6-chloro-7-hydroxy-N-methyl-1,2,3,4-tetrahydroisoquinoline 91421 2-(1-amino-1-methylethylcarboxamido)-3-[1-methylsulfonylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]-3-oxo-(2S)-propyl octanoate; trifluoroacetate 91422 2-[1-aminomethylcarboxamido-2-hydroxy-(1S)-ethylcarboxamido]-3-[1-methylsulfonylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]-3-oxo-(2R)-propyl octanoate; Trifluoroacatate 91455 3-(4-Phenyl-piperazin-1-ylmethyl)-1H-indole 91570 2-[1-aminomethylcarboxamido-2-hydroxy-(1S)-ethylcarboxamido]-3-[1-methylsulfonylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]-3-oxo-(2S)-propyl octanoate; trifluoroactate 91575 1N-[1-benzyloxymethyl-2-[1-methylsulfonylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]-2-oxo-(1R)-ethyl]-2-aminomethylcarboxamido-3-hydroxy-(2S)-propanamide; Trifluoroacetate 91677 2-[1-[1-aminomethylcarboxamido-2-heptylcarbonyloxy-(1S)-ethylcarboxamido]-2-hydroxy-(1S)-ethylcarboxamido]-3-phenyl-(2S)-propanoic acid 91682 2-(1-amino-1-methylethylcarboxamido)-3-[1-methylsulfonylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]-3-oxo-(2R)-propyl octanoate; Trifluoroacetate 91683 2-[1-amino-2-hydroxy-(1S)-ethylcarboxamido]-3-[1-methylsulfonylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]-3-oxo-(2R)-propyl octanoate; Trifluoroacetate 91699 [3-(4-Chloro-phenyl)-3-pyridin-2-yl-propyl]-[4-(1H-imidazol-4-yl)-butyl]-methyl-amine 91722 1N-[1-benzyloxymethyl-2-[1-methylsulfonylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]-2-oxo-(1R)-ethyl]-2-amino-3-hydroxy-(2S)-propanamide; Trifluoroacetate 91855 4-(2-Chloro-phenyl)-1-[3-(2-oxo-5-thioxo-3,3-di-p-tolyl-pyrrolidin-1-yl)-propyl]-piperidine-4-carbonitrile 91857 1-[3-(2,5-Dioxo-3,3-di-p-tolyl-pyrrolidin-1-yl)-2-hydroxy-propyl]-4-o-tolyl-piperidine-4-carbonitrile 91858 4-(2-Chloro-phenyl)-1-[3-(2,5-dioxo-3,3-di-p-tolyl-pyrrolidin-1-yl)-propyl]-piperidine-4-carbonitrile 92035 1-[3-(2,5-Dioxo-3,3-di-p-tolyl-pyrrolidin-1-yl)-propyl]-4-o-tolyl-piperidine-4-carbonitrile 92039 1-[3-(2,4-Dioxo-5,5-di-p-tolyl-oxazolidin-3-yl)-propyl]-4-o-tolyl-piperidine-4-carbonitrile 92040 N-[3-(4-Cyano-4-phenyl-piperidin-1-yl)-propyl]-2-hydroxy-2,2-di-p-tolyl-acetamide 92602 12,13-dimethyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrrolo[3,4-c]carbazol-5-one 92605 12,13-diethyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrrolo[3,4-c]carbazol-5-one 92612 N-[3-(4-Cyano-4-o-tolyl-piperidin-1-yl)-propyl]-2-hydroxy-2,2-di-p-tolyl-acetamide 92654 12-(2,3-dihydroxypropyl)-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrrolo[3,4-c]carbazol-5-one 92673 12-methyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrrolo[3,4-c]carbazol-5-one 92677 12-(2,2-difluoroethyl)-13-methyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrrolo[3,4-c]carbazol-5-one 92683 2-(5-oxo-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrrolo[3,4-c]carbazol-12-yl)ethyl cyanide 92709 2-(13-ethyl-5-oxo-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrrolo[3,4-c]carbazol-12-yl)ethyl cyanide 92710 3-(5-oxo-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrrolo[3,4-c]carbazol-12-yl)propanoic acid 92744 SID26756836 92804 13-methyl-12-propyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrrolo[3,4-c]carbazol-5-one 92944 1-Butyl-3-{3-methoxy-2-propoxy-5-[5-(3,4,5-trimethoxy-phenyl)-tetrahydro-furan-2-yl]-phenyl}-1-hydroxy-urea 93086 1-Phenyl-cyclopentanecarboxylic acid 2-diethylamino-ethyl ester 93523 {2-[6-Oxo-3-(2-phenyl-pyrazolo[1,5-a]pyridin-3-yl)-6H-pyridazin-1-yl]-cyclohex-1-enyl}-acetic acid 93525 4-(6-oxo-3-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)pyridazin-1(6H)-yl)butanoic acid 93581 2-Fluoro-3-(1-hydroxy-2-methylamino-ethyl)-phenol (2-FPE) 93648 3-methyl-7-nitro-1,2,3,4-tetrahydroisoquinoline 94047 {2-[6-Oxo-3-(2-phenyl-pyrazolo[1,5-a]pyridin-3-yl)-6H-pyridazin-1-yl]-cyclopent-1-enyl}-acetic acid 94050 {2-[6-Oxo-3-(2-phenyl-pyrazolo[1,5-a]pyridin-3-yl)-6H-pyridazin-1-yl]-cyclohept-1-enyl}-acetic acid 94096 3-[(3R,4R)-1-(3-Hydroxy-cyclohexyl)-3,4-dimethyl-piperidin-4-yl]-phenol 94135 3-((3R,4R)-1-Cyclopentyl-3,4-dimethyl-piperidin-4-yl)-phenol 94136 3-((3R,4R)-1-Cyclohexyl-3,4-dimethyl-piperidin-4-yl)-phenol 94194 SID26752074 94196 Biphenyl-4-carboxylic acid {4-[(5-hydroxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-methyl-amino]-butyl}-amide 94225 (1R,2S)-2-(1H-imidazol-4-yl)cyclopropan-1-amine 94232 Biphenyl-4-carboxylic acid {4-[(5-methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-methyl-amino]-butyl}-amide 94234 Biphenyl-4-carboxylic acid {4-[(5-hydroxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amino]-butyl}-amide 94285 (1S,2S)-2-(2-aminoethyl)-1-(1H-imidazol-4-yl)cyclopropane 94286 C-[2-(1H-Imidazol-4-yl)-cyclopropyl]-methylamine 94337 Biphenyl-4-carboxylic acid {4-[(5-cyclopropylmethoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amino]-butyl}-amide 94339 6-({4-[(Biphenyl-4-carbonyl)-amino]-butyl}-propyl-amino)-5,6,7,8-tetrahydro-naphthalene-1-carboxylic acid amide 94375 Biphenyl-4-carboxylic acid {4-[(5-bromo-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amino]-butyl}-amide 94377 Biphenyl-4-carboxylic acid {4-[propyl-(1,2,3,4-tetrahydro-naphthalen-2-yl)-amino]-butyl}-amide 94381 C-[2-(1H-Imidazol-4-yl)-cyclopropyl]-methylamine 94382 C-[2-(1H-Imidazol-4-yl)-cyclopropyl]-methylamine 94393 C-[2-(1H-Imidazol-4-yl)-cyclopropyl]-methylamine 94395 4-Fluoro-3-(1-hydroxy-2-methylamino-ethyl)-phenol (6-FPE) 94435 (+)-(7-nitro-1,2,3,4-tetrahydroisoquinolin-3-yl)methanol 94453 2-[2-(1H-Imidazol-4-yl)-cyclopropyl]-ethylamine 94460 2-(4-Bromo-2-methoxy-phenyl)-1-methyl-ethylamine 94484 10,17-dihydroxy-4-methyl-(13R,17S)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10-trien-14-one 94504 2-(4-Bromo-phenyl)-1-methyl-ethylamine 94539 (1S,2R)-2-(1H-imidazol-4-yl)cyclopropan-1-amine 94605 SID26756758 94668 2-Ethyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-yloxy]-quinoline-4-carboxylic acid 94674 7-[3-(2-Cyclopropylmethyl-3-methoxymethyl-4-thiazol-4-yl-phenoxy)-propoxy]-8-propyl-chroman-2-carboxylic acid 94675 7-[3-(4-Acetyl-3-hydroxymethyl-2-propyl-phenoxy)-propoxy]-8-propyl-chroman-2-carboxylic acid 94677 2-Cyclopropyl-6-fluoro-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-yloxy]-quinoline-4-carboxylic acid 94678 2-Cyclopropyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-yloxy]-quinoline-4,5-dicarboxylic acid 94680 3-((3R,4R)-1-Benzo[b]thiophen-2-ylmethyl-3,4-dimethyl-piperidin-4-yl)-phenol 94708 2-Cyclopropyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-yloxy]-[1,5]naphthyridine-4-carboxylic acid 94765 4'-[3-Butyl-5-oxo-1-(2-trifluoromet hyl-phenyl)-15-dihydro-[124]tria zol-4-ylmethyl]-biphenyl-2-sulfonic acid t-butyloxycarbonylamide (L-162234) 94766 4'-[3-Butyl-1-(3-nitro-phenyl)-5-oxo-1,5-dihydro-[1,2,4]triazol-4-ylmethyl]-biphenyl-2-sulfonic acid 2-chloro-benzoylamide 94768 5,7-Dihydro-dibenzo[c,e]oxepine-1,2,3,9,10,11-hexaol 94794 3-((3R,4R)-1-Benzofuran-2-ylmethyl-3,4-dimethyl-piperidin-4-yl)-phenol 94819 3-(3,4-Dichloro-phenyl)-5-hydroxy-4-(4-methoxy-benzyl)-5-(4-methoxy-phenyl)-dihydro-furan-2-one 94835 3-[(3R,4R)-1-(3-Hydroxy-3-phenyl-cyclohexyl)-3,4-dimethyl-piperidin-4-yl]-phenol 94837 3-[(3R,4R)-3,4-Dimethyl-1-((Z)-3-phenyl-allyl)-piperidin-4-yl]-phenol 94958 Biphenyl-4-carboxylic acid {4-[(5-cyano-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amino]-butyl}-amide 94996 Methanesulfonic acid 6-({4-[(biphenyl-4-carbonyl)-amino]-butyl}-propyl-amino)-5,6,7,8-tetrahydro-naphthalen-1-yl ester 95062 Biphenyl-4-carboxylic acid {4-[(5-methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amino]-butyl}-amide 95079 2-Propyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-yloxy]-quinoline-4-carboxylic acid 95080 2-Cyclopropyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-yloxy]-[1,8]naphthyridine-4-carboxylic acid 95107 3-Benzo[1,3]dioxol-5-yl-4-benzyl-5-(3,4-dichloro-phenyl)-5-hydroxy-dihydro-furan-2-one 95116 2-Cyclopropyl-8-methyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-yloxy]-quinoline-4-carboxylic acid 95118 7-Chloro-2-cyclopropyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-yloxy]-quinoline-4-carboxylic acid 95180 2-Cyclopropyl-5-methyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-yloxy]-quinoline-4-carboxylic acid 95183 2-Cyclopropyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethoxy]-quinoline-4-carboxylic acid 95214 2-Methyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-yloxy]-quinoline-4-carboxylic acid 95222 2-Cyclopropyl-6-methoxy-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-yloxy]-quinoline-4-carboxylic acid 95239 (R)-2-(Benzylamino-methyl)-chroman-7-ol 95247 4-[3-(Naphthalen-1-ylmethoxy)-propyl]-1H-imidazole; compound with (Z)-but-2-enedioic acid 95285 4-(2-Benzylamino-ethoxy)-1,3-dihydro-indol-2-one 95286 butyloxy 2-{2-[3-chloro-4-(4-ethyl-5-methyloxycarbonyl-2-propyl-1H-1-imidazolylmethyl)phenyl]phenylsulfonyl}carbonylamino 95318 4-{3-[(4-Bromo-phenyl)-phenyl-methoxy]-propyl}-1H-imidazole; compound with (Z)-but-2-enedioic acid 95351 4-{3-[Phenyl-(4-trifluoromethyl-phenyl)-methoxy]-propyl}-1H-imidazole; compound with (Z)-but-2-enedioic acid 95354 4-{3-[Bis-(4-fluoro-phenyl)-methoxy]-propyl}-1H-imidazole; compound with (Z)-but-2-enedioic acid 95379 2-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-benzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxy-phenyl)-acetamide 95390 4-Methoxy-N-(3-phenyl-isoquinolin-1-yl)-benzamide 95437 4-methoxy-N-(3-phenyl-1,2,4-thiadiazol-5-yl)benzamide 95438 N-(4-Phenyl-thiazol-2-yl)-benzamide 95440 4-Chloro-N-(4-phenyl-thiazol-2-yl)-benzamide 95472 4-Bromo-N-(4-phenyl-thiazol-2-yl)-benzamide 95546 3-Chloro-N-(4-phenyl-thiazol-2-yl)-benzamide 95548 4-methoxy-N-(4-phenylthiazol-2-yl)benzamide 95584 4-Nitro-N-(4-phenyl-thiazol-2-yl)-benzamide 95585 2,4-Dichloro-N-(4-phenyl-thiazol-2-yl)-benzamide 95625 3,4-Dichloro-N-(4-phenyl-thiazol-2-yl)-benzamide 95633 N-[5-(3,4-Dimethoxy-phenyl)-1H-pyrazol-3-yl]-2-naphthalen-2-yl-acetamide 95686 4-(-1-amino-1-oxo-3-phenylpropan-2-ylamino)-3-(2-(2-(tert-butoxycarbonyl)-3-(1H-indol-3-yl)propanamido)-4-(methylthio)butanamido)-4-oxobutanoic acid 95738 4-(3-Benzhydryloxy-propyl)-1H-imidazole; compound with (Z)-but-2-enedioic acid 95813 Balanol 95860 5-Bromo-N-{4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-2,3-dimethoxy-benzamide 95878 4'-(5-Acetyl-4-ethyl-2-propyl-imidazol-1-ylmethyl)-3'-fluoro-biphenyl-2-sulfonic acid butyloxycarbonylamide (EXP970) 95881 9-Oxo-9H-fluorene-4-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide 95893 Benzyl-[2-(1H-indol-4-yloxy)-ethyl]-amine 95914 4-(3-Benzyloxy-propyl)-1H-imidazole; compound with (Z)-but-2-enedioic acid 95915 4-{3-[(4-Fluoro-phenyl)-phenyl-methoxy]-propyl}-1H-imidazole; compound with (Z)-but-2-enedioic acid 95916 4-{3-[(4-Chloro-phenyl)-phenyl-methoxy]-propyl}-1H-imidazole; compound with (Z)-but-2-enedioic acid 95917 N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-9H-fluorene-2-carboxamide 96185 3-(2-Benzylamino-ethoxy)-phenol 96225 5-Ethyl-3-(3-fluoro-2'-isopentyloxycarbonylsulfamoyl-biphenyl-4-ylmethyl)-2-propyl-3H-imidazole-4-carboxylic acid methyl ester (EXP408) 96291 N-(4-Phenyl-thiazol-2-yl)-4-trifluoromethyl-benzamide 96294 4-Methyl-N-(4-phenyl-thiazol-2-yl)-benzamide 96324 4-tert-Butyl-N-(4-phenyl-thiazol-2-yl)-benzamide 96326 Biphenyl-4-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide 96465 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (3R,4R)-4-(4-hydroxy-benzoylamino)-pyrrolidin-3-yl ester 96693 N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)benzo[b]thiophene-2-carboxamide 96729 4-(2,4-dichloro-5-methoxyphenylamino)-7-(5-((4-methylpiperazin-1-yl)methyl)thiophen-3-yl)quinoline-3-carbonitrile 96934 3N-phenyl-1-methyl-2-(1-methyl-3-phenylcarbamoyl-1H-2-indolyldisulfanyl)-1H-3-indolecarboxamide 97130 6-[(S)-(R)-3-Hydroxy-2-((1S,2R)-3-hydroxy-oct-1-enyl)-5-oxo-cyclopentylsulfanyl]-hexanoic acid 97494 ({(2E)-2-[(3aS,4S,5R,6aS)-5-hydroxy-4-((E)-{[(phenylamino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]ethyl}oxy)acetic acid 97497 (4E)-4-[(3aS,4S,6aR)-4-((E)-{[((3-chlorophenyl)amino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]pentanoic acid 97535 (4Z)-4-[(3aS,4S,5R,6aS)-5-hydroxy-4-((E)-{[(phenylamino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]butanoic acid 97557 (4Z)-4-[(3aS,4S,5R,6aS)-5-hydroxy-4-((E)-{[((3,4-dichloro-phenyl)amino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]butanoic acid 97558 (5Z)-5-[(3aS,4S,5R,6aS)-5-hydroxy-4-((E)-{[((3,4-dichlorophenyl)amino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]pentanoic acid 97569 3,5-Dimethyl-1,7-dihydro-benzo[1,2-c;5,4-c']dipyrazole 97579 1,7-Diethyl-3,5,8-trimethyl-1,7-dihydro-benzo[1,2-c;5,4-c']dipyrazole 97580 3,5-Dimethyl-1,7-dipropyl-1,7-dihydro-benzo[1,2-c;5,4-c']dipyrazole 97583 ({(2Z)-2-[(3aS,4S,5R,6aS)-5-hydroxy-4-((E)-{[(phenylamino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]ethyl}oxy)acetic acid 97584 (5E)-5-[(3aS,4S,5R,6aS)-5-hydroxy-4-((E)-{[((4-nitro-phenyl)amino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]pentanoic acid 97585 ({(2E)-2-[(3aS,4S,5R,6aS)-5-hydroxy-4-((E)-{[((3,4-dichloro-phenyl)amino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]ethyl}oxy)acetic acid 97586 (4E)-4-[(3aS,4S,5R,6aS)-5-hydroxy-4-((E)-{[((3,4-dichloro-phenyl)amino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]butanoic acid 97597 ({(2Z)-2-[(3aS,4S,5R,6aS)-5-hydroxy-4-((E)-{[((3-chlorophenyl)amino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]ethyl}oxy)acetic acid 97603 1,3,5,7,8-Pentamethyl-1,7-dihydro-benzo[1,2-c;5,4-c']dipyrazole 97618 (5E)-5-[(3aS,4S,6aR)-4-((E)-{[((4-nitrophenyl)amino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]pentanoic acid 97628 (4Z)-4-[(3aS,4S,5R,6aS)-5-hydroxy-4-((E)-{[((3-chlorophenyl)amino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]butanoic acid 97631 (4Z)-4-[(3aS,4S,6aR)-4-((E)-{[((3-chlorophenyl)amino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]butanoic acid 97640 ({(2E)-2-[(3aS,4S,5R,6aS)-5-hydroxy-4-((E)-{[((4-nitro-phenylamino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]ethyl}oxy)acetic acid 97650 (4E)-4-[(3aS,4S,5R,6aS)-5-hydroxy-4-((E)-{[((3-chlorophenyl)amino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]butanoic acid 97651 (5Z)-5-[(3aS,4S,6aR)-4-((E)-{[((3,4-dichlorophenyl)amino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]pentanoic acid 97728 9-Methoxy-1,2,3,4-tetrahydro-anthracen-2-ylamine 97730 (10-Methoxy-1,2,3,4-tetrahydro-phenanthren-2-yl)-dipropyl-amine 97731 7-Dipropylamino-4-methyl-5,6,7,8-tetrahydro-naphthalen-1-ol 97744 5-[(S)-(R)-3-Hydroxy-2-((1R,2R)-3-hydroxy-oct-1-enyl)-5-oxo-cyclopentylmethylsulfanyl]-pentanoic acid 97745 (E)-7-{(1R,2R,3R,5R)-5-Chloro-3-hydroxy-2-[(E)-(S)-3-hydroxy-4-(4-hydroxy-3-methyl-phenyl)-but-1-enyl]-cyclopentyl}-hept-5-enoic acid 97748 (8-Methoxy-5-methyl-1,2,3,4-tetrahydro-naphthalen-2-yl)-dipropyl-amine 97749 2-Dipropylamino-1,2,3,4-tetrahydro-anthracen-9-ol 97791 (5E)-5-[(3aS,4S,6aR)-4-((E)-{[(phenylamino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]pentanoic acid 97793 (5Z)-5-[(3aS,4S,5R,6aS)-5-hydroxy-4-((E)-{[(phenylamino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]pentanoic acid 97795 N-Benzyl-3-{2-[3-(2-benzylcarbamoyl-ethyl)-1H-indol-2-yldisulfanyl]-1H-indol-3-yl}-propionamide 97838 ({(2Z)-2-[(3aS,4S,5R,6aS)-5-hydroxy-4-((E)-{[((4-nitro-phenylamino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]ethyl}oxy)acetic acid 97841 (4Z)-4-[(3aS,4S,5R,6aS)-5-hydroxy-4-((E)-{[((4-nitro-phenylamino))carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]butanoic acid 97860 (R)-2-[(R)-2-(2-{(S)-2-[(R)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-3-hydroxy-2-methyl-propionylamino}-acetylamino)-3-phenyl-propionylamino]-4-methyl-pentanoic acid 97870 4-(2-{(1R,2R,3R,5R)-5-Fluoro-3-hydroxy-2-[(E)-(S)-3-hydroxy-4-(3-methoxymethyl-phenyl)-but-1-enyl]-cyclopentyl}-ethylsulfanyl)-butyric acid 97877 (4Z)-4-[(3aS,4S,6aR)-4-((E)-{[((3-chlorophenyl)amino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]butanoic acid 97886 4-{(S)-2-[(R)-3-Hydroxy-2-((1R,2R)-3-hydroxy-oct-1-enyl)-5-oxo-cyclopentyl]-ethylsulfanyl}-butyric acid 97887 {(S)-4-[(R)-3-Hydroxy-2-((1R,2R)-3-hydroxy-oct-1-enyl)-5-oxo-cyclopentyl]-butylsulfanyl}-acetic acid 97920 (E)-7-{(1R,2R,3R,5R)-5-Fluoro-3-hydroxy-2-[(E)-(S)-3-hydroxy-4-(3-methoxymethyl-phenyl)-but-1-enyl]-cyclopentyl}-hept-5-enoic acid 97921 (E)-7-{(1R,2R,3R,5R)-5-Chloro-3-hydroxy-2-[(E)-(S)-3-hydroxy-4-(3-methoxymethyl-phenyl)-but-1-enyl]-cyclopentyl}-hept-5-enoic acid 97937 7-{(1R,2R,3R,5R)-5-Chloro-3-hydroxy-2-[(E)-(S)-3-hydroxy-4-(3-methoxymethyl-phenyl)-but-1-enyl]-cyclopentyl}-heptanoic acid 97941 (R)-2-[(R)-2-(2-{(R)-2-[(R)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-3-hydroxy-2-methyl-propionylamino}-acetylamino)-3-phenyl-propionylamino]-4-methyl-pentanoic acid 98084 (5Z)-5-[(3aS,4S,6aR)-4-((E)-{[(phenylamino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]pentanoic acid 98086 3-{(S)-3-[(R)-3-Hydroxy-2-((1R,2R)-3-hydroxy-oct-1-enyl)-5-oxo-cyclopentyl]-propylsulfanyl}-propionic acid 98116 3-{2-[2-Acetylamino-2-(10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5-yl)-acetylamino]-4-methyl-pentanoylamino}-N-(1-{1-[1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 98121 4-(2-((1R,2R,3R)-3-hydroxy-2-((S,E)-3-hydroxy-4-(3-(methoxymethyl)phenyl)but-1-enyl)-5-oxocyclopentyl)ethylthio)butanoic acid 98157 4-(2-{(1R,2R,3R)-3-Hydroxy-2-[(E)-(S)-3-hydroxy-4-(4-hydroxy-3-methyl-phenyl)-but-1-enyl]-5-oxo-cyclopentyl}-ethylsulfanyl)-butyric acid 98202 (4E)-4-[(3aS,4S,5R,6aS)-5-hydroxy-4-((E)-{[((4-nitro-phenylamino))carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]butanoic acid 98204 (5Z)-5-[(3aS,4S,5R,6aS)-5-hydroxy-4-((E)-{[((4-nitro-phenyl)amino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]pentanoic acid 98246 (5Z)-5-[(3aS,4S,6aR)-4-((E)-{[((4-nitrophenyl)amino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]pentanoic acid 98248 ({(2Z)-2-[(3aS,4S,5R,6aS)-5-hydroxy-4-((E)-{[((3,4-dichloro-phenyl)amino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]ethyl}oxy)acetic acid 98410 1,7-Diethyl-3,5-dimethyl-1,7-dihydro-benzo[1,2-c;5,4-c']dipyrazole 98412 3,5-Dimethyl-8-nitro-1,7-dihydro-benzo[1,2-c;5,4-c']dipyrazole 98414 (5E)-5-[(3aS,4S,6aR)-4-((E)-{[((3,4-dichlorophenyl)amino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]pentanoic acid 98417 (5E)-5-[(3aS,4S,5R,6aS)-5-hydroxy-4-((E)-{[((3,4-dichlorophenyl)amino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]pentanoic acid 98418 ({(2E)-2-[(3aS,4S,5R,6aS)-5-hydroxy-4-((E)-{[((3-chlorophenyl)amino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]ethyl}oxy)acetic acid 98461 3,5,8-Trimethyl-1,7-dihydro-benzo[1,2-c;5,4-c']dipyrazole 98513 (4E)-4-[(3aS,4S,5R,6aS)-5-hydroxy-4-((E)-{[(phenylamino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]butanoic acid 98554 (R)-2-Amino-1-{4-[3-(4-cyclopropanecarbonyl-phenoxy)-propyl]-piperazin-1-yl}-propan-1-one 98651 10-Methoxy-1,2,3,4-tetrahydro-phenanthren-2-ylamine 98652 8-Methoxy-5-methyl-1,2,3,4-tetrahydro-naphthalen-2-ylamine 98821 8-Aza-bicyclo[3.2.1]octane-6-carboxylic acid methyl ester 98839 (R)-6-Chloro-2-methyl-1-phenyl-1,2,3,4-tetrahydro-isoquinolin-7-ol 98992 6-Chloro-1-phenyl-2-propyl-1,2,3,4-tetrahydro-isoquinolin-7-ol 98993 6-Chloro-1-phenyl-1,2,3,4-tetrahydro-isoquinolin-7-ol 98994 (S)-6-Chloro-2-methyl-1-phenyl-1,2,3,4-tetrahydro-isoquinolin-7-ol 99028 6-acetoxy-8-azonia-bicyclo[3.2.1]octane 99081 6-acetoxy-8-methyl-8-azonia-bicyclo[3.2.1]octane 99320 (2-Acetoxy-propyl)-trimethyl-ammonium 99414 N-[2-(2,7-Dimethoxy-naphthalen-1-yl)-ethyl]-propionamide 99462 (R)-2-Benzo[1,3]dioxol-5-yl-6-isopropoxy-4-(4-methoxy-phenyl)-2H-chromene-3-carboxylic acid 99612 (E)-1-[(S)-2-(2-Hydroxy-ethyl)-piperidin-1-yl]-3-(2-phenyl-pyrazolo[1,5-a]pyridin-3-yl)-propenone 99805 8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]indole-1-carbaldehyde 99816 R-(+)-1-(8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]indol-1-yl)-ethanone 99817 Dipropyl-(5,6,7,8-tetrahydro-1H-benzo[f]indol-7-yl)-amine 99851 Dipropyl-(6,7,8,9-tetrahydro-3H-benzo[e]indol-8-yl)-amine 99852 S-(-)-1-(8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]indol-1-yl)-ethanone 99988 Dipropyl-(S)-6,7,8,9-tetrahydro-3H-benzo[e]indol-8-yl-amine 99989 Dipropyl-(R)-6,7,8,9-tetrahydro-3H-benzo[e]indol-8-yl-amine 100025 Dimethyl-(6,7,8,9-tetrahydro-3H-benzo[e]indol-8-yl)-amine 100051 3-[(Benzyl-methyl-amino)-methyl]-8-(2,6-difluoro-benzyl)-5-oxo-2-{4-[(thiophene-3-carbonyl)-amino]-phenyl}-5,8-dihydro-imidazo[1,2-a]pyrimidine-6-carboxylic acid ethyl ester 100052 ethyl 8-(2,6-difluorobenzyl)-3-((benzyl(methyl)amino)methyl)-2-(4-(3-ethylureido)phenyl)-5-oxo-5,8-dihydroimidazo[1,2-a]pyrimidine-6-carboxylate 100071 3-[(Benzyl-methyl-amino)-methyl]-8-(2,6-difluoro-benzyl)-2-[4-(3-methoxy-ureido)-phenyl]-5-oxo-5,8-dihydro-imidazo[1,2-a]pyrimidine-6-carboxylic acid ethyl ester 100072 2-(4-Acryloylamino-phenyl)-3-[(benzyl-methyl-amino)-methyl]-8-(2,6-difluoro-benzyl)-5-oxo-5,8-dihydro-imidazo[1,2-a]pyrimidine-6-carboxylic acid ethyl ester 100122 2-[2-(2-{2-[2-(2-{2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-6-amino-hexanoylamino}-3-carboxy-propionylamino)-4-methylsulfanyl-butyrylamino]-4-carbamoyl-butyrylamino}-4-methyl-pentanoylamino)-acetylamino]-5-guanidino-pentanoic acid (Ac-His-Lys-Asp-Met-Gln-Leu-Gly-Arg) 100135 2-(4-Benzoylamino-phenyl)-3-[(benzyl-methyl-amino)-methyl]-8-(2,6-difluoro-benzyl)-5-oxo-5,8-dihydro-imidazo[1,2-a]pyrimidine-6-carboxylic acid ethyl ester 100174 H-His-Lys-AspMet-GIn-Leu-Gly-Arg-OH 100175 Ile-Ser-His-Lys-Asp-Met-Gln-Leu-Gly-Arg 100216 3-[(Benzyl-methyl-amino)-methyl]-2-(4-butyrylamino-phenyl)-8-(2,6-difluoro-benzyl)-5-oxo-5,8-dihydro-imidazo[1,2-a]pyrimidine-6-carboxylic acid ethyl ester 100246 3-[(Benzyl-methyl-amino)-methyl]-8-(2,6-difluoro-benzyl)-2-[4-(3-methoxy-ureido)-phenyl]-5-oxo-5,8-dihydro-imidazo[1,2-a]pyrimidine-6-carboxylic acid propyl ester 100279 3-[(Benzyl-methyl-amino)-methyl]-8-(2,6-difluoro-benzyl)-2-[4-(3-ethyl-ureido)-phenyl]-5-oxo-5,8-dihydro-imidazo[1,2-a]pyrimidine-6-carboxylic acid propyl ester 100287 Dimethyl-(6,7,8,9-tetrahydro-3H-benzo[e]indol-8-yl)-amine 100299 SID11111620 100307 3-[(Benzyl-methyl-amino)-methyl]-8-(2,6-difluoro-benzyl)-2-{4-[(furan-3-carbonyl)-amino]-phenyl}-5-oxo-5,8-dihydro-imidazo[1,2-a]pyrimidine-6-carboxylic acid ethyl ester 100345 AcMet-Ile-Lys-Ala-Phe-Thr-Glu-Met-Met-Val-Val-Ala-Ser-Gln-Leu-Alr-Ala-Asn-Ile-Ser-His-Lys-Asp-Met-Gln-Leu-Gly-Arg 100381 2,3-dimethoxy-7-methyl-6,7,8,9,14,15-hexahydro-5H-benzo[7,8]azecino[5,4-b]indole 100385 9-(tetrahydrofuran-2-yl)-9H-purin-6-amine 100406 AcMet-Val-Val-Ala-Ser-Gln-Leu-Arg-Ala-Asn-Ile-Ser-His-Lys-Asp-Met-Gln-Leu-Gly-Arg 100407 Phe-Thr-Glu-Met-Met-Val-Val-Ala-Ser-Gln-Leu-Alr-Ala-Asn-Ile-Ser-His-Lys-Asp-Met-Gln-Leu-Gly-Arg 100502 Dimethyl-(6,7,8,9-tetrahydro-3H-benzo[e]indol-8-yl)-amine 100662 4'-Chloro-2-(3,4,5-trimethoxy-benzoylamino)-biphenyl-4-carboxylic acid cyclohexylamide 100700 SID26754792 100713 3(1,2,3,4,5,11-Hexahydro-3-methyl-2,6-methano-9-methoxy-6H-azocino[4,5-b]indol-6-yl)phenol methanesulfonate 100720 3-[(Benzyl-methyl-amino)-methyl]-2-[4-(cyclopropanecarbonyl-amino)-phenyl]-8-(2,6-difluoro-benzyl)-5-oxo-5,8-dihydro-imidazo[1,2-a]pyrimidine-6-carboxylic acid ethyl ester 100721 3-[(Benzyl-methyl-amino)-methyl]-8-(2,6-difluoro-benzyl)-5-oxo-2-(4-propionylamino-phenyl)-5,8-dihydro-imidazo[1,2-a]pyrimidine-6-carboxylic acid ethyl ester 100765 3(1,2,3,4,5,11-Hexahydro-3-methyl-2,6-methano-10-methoxy-6H-azocino[4,5-b]indol-6-yl)phenol methanesulfonate 100776 9-Phenyl-9H-purin-6-ylamine 100867 SID11114176 100989 1,2,3,4,5,11-Hexahydro-6-phenyl-3-methyl-2,6-methano-6H-azocino[4,5-b]indole 101007 3(1,2,3,4,5,11-Hexahydro-3-methyl-2,6-methano-8-methoxy-6H-aocino[4,5-b]indol-6-yl)phenol methanesulfonate 101045 7-methyl-5,6,7,8,9,14,15,16-octahydroindolo[2',3':7,8]azecino[5,4-b]indole 101107 1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichloro-phenyl)-5-(4-hydroxy-4-phenyl-piperidin-1-yl)-pentan-2-one oxime 101122 [11-(2-Dimethylamino-ethylidene)-6,11-dihydro-dibenzo[b,e]oxepin-2-yl]-acetic acid 101148 11-(3-Dimethylamino-propylidene)-6,11-dihydro-dibenzo[b,e]oxepine-2-carboxylic acid 101227 11-(3-Thiomorpholin-4-yl-propylidene)-6,11-dihydro-dibenzo[b,e]oxepine-2-carboxylic acid 101255 11-(3-Pyrrolidin-1-yl-propylidene)-6,11-dihydro-dibenzo[b,e]oxepine-2-carboxylic acid; compound with but-2-enedioic acid 101256 3-[11-(3-Dimethylamino-propylidene)-6,11-dihydro-dibenzo[b,e]oxepin-2-yl]-acrylic acid; compound with but-2-enedioic acid 101257 3-[11-(3-Dimethylamino-propylidene)-6,11-dihydro-dibenzo[b,e]oxepin-2-yl]-propionic acid 101343 Benzo[g]quinazolin-4-yl-(3-bromo-phenyl)-amine 101358 9-cyclopentyladenine 101370 N-(3-bromophenyl)-3H-imidazo[4,5-g]quinazolin-8-amine 101371 (6,7-Dimethoxy-quinazolin-4-yl)-(3-ethynyl-4-fluoro-phenyl)-amine 101555 11-(2-Dimethylamino-ethylidene)-6,11-dihydro-dibenzo[b,e]oxepine-2-carboxylic acid; compound with but-2-enedioic acid 101593 9-Methyl-9H-adenine 101707 2-[11-(3-Dimethylamino-propylidene)-6,11-dihydro-dibenzo[b,e]oxepin-2-yl]-ethanol 101708 [11-(4-Dimethylamino-butylidene)-6,11-dihydro-dibenzo[b,e]oxepin-2-yl]-acetic acid 101787 11-(4-Dimethylamino-butylidene)-6,11-dihydro-dibenzo[b,e]oxepine-2-carboxylic acid 101788 11-(3-Diethylamino-propylidene)-6,11-dihydro-dibenzo[b,e]oxepine-2-carboxylic acid; compound with but-2-enedioic acid 101827 SID26758045 101900 17-hydroxymethyl-18-oxa-4,14,22-triazahexacyclo[20.6.1.17,14.02,6.08,13.023,28]triaconta-1(29),2(6),7(30),8(13),9,11,23(28),24,26-nonaene-3,5-dione 101913 11-(3-Dimethylamino-propylidene)-6,11-dihydro-dibenzo[b,e]oxepine-3-carboxylic acid 101915 11-(3-Dimethylamino-propylidene)-6,11-dihydro-dibenzo[b,e]oxepine-2-carboxylic acid; compound with but-2-enedioic acid 101939 18-hydroxymethyl-(18S)-17-oxa-4,14,21-triazahexacyclo[19.6.1.17,14.02,6.08,13.022,27]nonacosa-1(28),2(6),7(29),8(13),9,11,22(27),23,25-nonaene-3,5-dione 101941 3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thiophene-2-carboxylic acid benzo[1,3]dioxol-5-yl ester 101990 12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-benzyl-3,7,13-trioxo-1,4,8triaza-cyclotridecane-5-carboxylic acid amide 102004 9-Ethyl-9H-adenine 102053 SID11113868 102064 12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-benzyl-3,7,13-trioxo-1,4,8triaza-cyclotridecane-5-carboxylic acid amide 102065 12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-cyclohexyl-3,7,13-trioxo-1,4,8triaza-cyclotridecane-5-carboxylic acid amide 102087 3-[3-[4-[2-(3-fluorophenyl)ethyl]-1-piperazinyl]propyl]-5-(4H-1,2,4-triazol-4-yl)-1H-indole 102088 Benzyl-methyl-{1-[3-(5-[1,2,4]triazol-4-yl-1H-indol-3-yl)-propyl]-piperidin-4-yl}-amine 102091 5-Ethanesulfonyl-N-(1-ethyl-pyrrolidin-2-ylmethyl)-2-methoxy-benzamide ((S)-sultopride) 102144 2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-3-(1H-indol-3-yl)-propionylamino]-propionylamino}-N-{[2-(3H-imidazol-4-yl)-1-(3-methyl-1-propyl-butylcarbamoyl)-ethylcarbamoyl]-methyl}-3-methyl-butyramide 102147 3-(2-Fluoro-3-{4-[2-(3-fluoro-phenyl)-ethyl]-piperazin-1-yl}-propyl)-5-[1,2,4]triazol-4-yl-1H-indole 102190 N-{2-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-ethyl}-4-fluoro-benzamide 102268 2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-3-(1H-indol-3-yl)-propionylamino]-propionylamino}-N-{[2-(3H-imidazol-4-yl)-1-(1-isobutyl-hexylcarbamoyl)-ethylcarbamoyl]-methyl}-3-methyl-butyramide 102287 (S)-2-((S)-3-(4-Cyano-phenyl)-2-{3-[1-(2-methyl-benzyl)-3-pyrrolidin-1-ylmethyl-1H-indol-6-yl]-ureido}-propionylamino)-5-guanidino-pentanoic acid benzylamide 102288 (S)-5-Guanidino-2-[(S)-2-{3-[1-(2-methyl-benzyl)-3-pyrrolidin-1-ylmethyl-1H-indol-6-yl]-ureido}-3-(4-nitro-phenyl)-propionylamino]-pentanoic acid benzylamide 102323 (S)-2-[(S)-2-{3-[1-(4-Fluoro-benzyl)-3-pyrrolidin-1-ylmethyl-1H-indol-6-yl]-ureido}-3-(4-nitro-phenyl)-propionylamino]-5-guanidino-pentanoic acid benzylamide 102344 2-{2-[2-[2-(2,2-Dimethyl-propionylamino)-3-(3H-imidazol-4-yl)-propionylamino]-3-(1H-indol-3-yl)-propionylamino]-propionylamino}-N-{[2-(3H-imidazol-4-yl)-1-(1-isobutyl-hexylcarbamoyl)-ethylcarbamoyl]-methyl}-3-methyl-butyramide 102345 12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-3,7,13-trioxo-2-phenethyl-1,4,8triaza-cyclotridecane-5-carboxylic acid amide 102346 12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-benzyl-3,7,13-trioxo-1,4,8triaza-cyclotridecane-5-carboxylic acid amide 102355 (S)-3-{2-[(S)-2-Acetylamino-3-(1H-indol-3-yl)-propionylamino]-3-[4-(3-o-tolyl-ureido)-phenyl]-propionylamino}-N-((R)-1-carbamoyl-2-p-tolyl-ethyl)-succinamic acid 102382 3-(2-(dimethylamino)ethyl)-1H-indol-4-ol 102470 (S)-5-Guanidino-2-((S)-3-(4-methoxy-phenyl)-2-{3-[1-(2-methyl-benzyl)-3-piperidin-1-ylmethyl-1H-indol-6-yl]-ureido}-propionylamino)-pentanoic acid (3-phenyl-propyl)-amide 102471 (S)-2-[(S)-2-{3-[3-Diethylaminomethyl-1-(2-methyl-benzyl)-1H-indol-6-yl]-ureido}-3-(4-methoxy-phenyl)-propionylamino]-5-guanidino-pentanoic acid (3-phenyl-propyl)-amide 102472 (S)-5-Guanidino-2-((S)-3-(4-methoxy-phenyl)-2-{3-[1-(2-methyl-benzyl)-3-pyrrolidin-1-ylmethyl-1H-indol-6-yl]-ureido}-propionylamino)-pentanoic acid (3-phenyl-propyl)-amide 102494 (CH3)CCO-His-Trp-Ala-Val-Gly-His-Leu-Met-NH2 102573 3-[3-(4-Benzyl-piperazin-1-yl)-propyl]-5-[1,2,4]triazol-4-yl-1H-indole 102593 2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-3-(1H-indol-3-yl)-propionylamino]-propionylamino}-N-{[2-(3H-imidazol-4-yl)-1-(3-methyl-1-propyl-butylcarbamoyl)-ethylcarbamoyl]-methyl}-3-methyl-butyramide 102609 3-[3-(4-Benzyl-4-fluoro-piperidin-1-yl)-propyl]-5-[1,2,4]triazol-4-yl-1H-indole 102614 3-[3-(4-Benzyl-piperidin-1-yl)-propyl]-5-[1,2,4]triazol-4-yl-1H-indole 102659 12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-benzyl-1-methyl-3,7,13-trioxo-1,4,8triaza-cyclotridecane-5-carboxylic acid amide 102691 (S)-2-[(S)-2-{3-[3-Diethylaminomethyl-1-(3-methyl-benzyl)-1H-indol-6-yl]-ureido}-3-(4-methoxy-phenyl)-propionylamino]-5-guanidino-pentanoic acid (3-phenyl-propyl)-amide 102692 (S)-2-[(S)-2-{3-[1-(2-Chloro-benzyl)-3-pyrrolidin-1-ylmethyl-1H-indol-6-yl]-ureido}-3-(4-methoxy-phenyl)-propionylamino]-5-guanidino-pentanoic acid (3-phenyl-propyl)-amide 102693 (S)-2-((S)-3-(4-Cyano-phenyl)-2-{3-[1-(2,6-dichloro-benzyl)-3-pyrrolidin-1-ylmethyl-1H-indol-6-yl]-ureido}-propionylamino)-5-guanidino-pentanoic acid benzylamide 102700 11-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-benzyl-3,9,12-trioxo-1,4,8triaza-cyclododecane-5-carboxylic acid amide 102701 10-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7-benzyl-6,9-dioxo-1,2-dithia-5,8-diaza-cycloundecane-4-carboxylic acid amide 102705 Ac-His-Trp-Ala-Val-Gly-His-Leu-Met-NH2 102729 4-(4-Chloro-phenyl)-1-[5-(5-ethanesulfonyl-2-methoxy-phenyl)-1H-pyrrol-2-ylmethyl]-piperidin-4-ol 102730 Ac-His-Trp-Ala-Val-Ala-His-Leu-Met-NH2 102735 2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-3-(1H-indol-3-yl)-propionylamino]-propionylamino}-N-{[2-(3H-imidazol-4-yl)-1-(1-isobutyl-pentylcarbamoyl)-ethylcarbamoyl]-methyl}-3-methyl-butyramide 102760 (S)-2-[(S)-2-{3-[1-(4-Fluoro-benzyl)-3-pyrrolidin-1-ylmethyl-1H-indol-6-yl]-ureido}-3-(4-methoxy-phenyl)-propionylamino]-5-guanidino-pentanoic acid cyclohexylmethyl-amide 102788 Benzyl-{1-[2-fluoro-3-(5-[1,2,4]triazol-4-yl-1H-indol-3-yl)-propyl]-piperidin-4-yl}-methyl-amine 102799 Ac-His-Trp-Ala-Val-D-Ala-His-Leu-Met-NH2 102860 (S)-5-Amino-2-[(S)-2-{3-[1-(2,6-dichloro-benzyl)-3-pyrrolidin-1-ylmethyl-1H-indol-6-yl]-ureido}-3-(3,4-difluoro-phenyl)-propionylamino]-pentanoic acid benzylamide 102871 (S)-2-[(S)-2-{3-[3-Azetidin-1-ylmethyl-1-(4-fluoro-benzyl)-1H-indol-6-yl]-ureido}-3-(4-methoxy-phenyl)-propionylamino]-5-guanidino-pentanoic acid benzylamide 102872 (S)-5-Guanidino-2-((S)-3-(4-methoxy-phenyl)-2-{3-[3-piperidin-1-ylmethyl-1-(4-trifluoromethoxy-benzyl)-1H-indol-6-yl]-ureido}-propionylamino)-pentanoic acid cyclohexylmethyl-amide 102918 1-(8-ethyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-methoxyphenyl)urea 102920 SID26753604 102928 7-Methoxy-1-(2-morpholin-4-yl-ethyl)-1H-indazole-3-carboxylic acid 2-methoxy-benzylamide 102929 7-Methoxy-1-(2-morpholin-4-yl-ethyl)-1H-indazole-3-carboxylic acid (1,3,3-trimethyl-bicyclo[2.2.1]hept-2-yl)-amide 102932 2-Ethyl-7-methoxy-1-(2-morpholin-4-yl-ethyl)-1H-indole-3-carboxylic acid (1,3,3-trimethyl-bicyclo[2.2.1]hept-2-yl)-amide 102944 (S)-5-Guanidino-2-((S)-3-(4-methoxy-phenyl)-2-{3-[3-pyrrolidin-1-ylmethyl-1-(4-trifluoromethoxy-benzyl)-1H-indol-6-yl]-ureido}-propionylamino)-pentanoic acid cyclohexylmethyl-amide 102945 4-(6-{3-[(S)-1-[(S)-1-(Cyclohexylmethyl-carbamoyl)-4-guanidino-butylcarbamoyl]-2-(4-methoxy-phenyl)-ethyl]-ureido}-3-pyrrolidin-1-ylmethyl-indol-1-ylmethyl)-benzoic acid methyl ester 102946 N-Benzyl-2-[(S)-2-{3-[1-(2,6-dichloro-benzyl)-3-pyrrolidin-1-ylmethyl-1H-indol-6-yl]-ureido}-3-(3,4-difluoro-phenyl)-propionylamino]-4-methylsulfanyl-butyramide 102948 (S)-2-[(S)-2-{3-[3-Diethylaminomethyl-1-(4-fluoro-benzyl)-1H-indol-6-yl]-ureido}-3-(4-methoxy-phenyl)-propionylamino]-5-guanidino-pentanoic acid cyclohexylmethyl-amide 102981 1-(2-(furan-2-yl)-8-propyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-methoxyphenyl)urea 102998 2-[(S)-2-{3-[1-(2,6-Dichloro-benzyl)-3-pyrrolidin-1-ylmethyl-1H-indol-6-yl]-ureido}-3-(3,4-difluoro-phenyl)-propionylamino]-pentanedioic acid 5-amide 1-benzylamide 102999 2-[(S)-2-{3-[1-(2,6-Dichloro-benzyl)-3-pyrrolidin-1-ylmethyl-1H-indol-6-yl]-ureido}-3-(3,4-difluoro-phenyl)-propionylamino]-5-ureido-pentanoic acid benzylamide 103000 (S)-N-[1-Benzylcarbamoyl-2-(3H-imidazol-4-yl)-ethyl]-2-{3-[1-(2,6-dichloro-benzyl)-3-pyrrolidin-1-ylmethyl-1H-indol-6-yl]-ureido}-3-(3,4-difluoro-phenyl)-propionamide 103014 (S)-2-[(S)-2-{3-[1-(4-Fluoro-benzyl)-3-pyrrolidin-1-ylmethyl-1H-indol-6-yl]-ureido}-3-(4-methoxy-phenyl)-propionylamino]-5-guanidino-pentanoic acid (3-phenyl-propyl)-amide 103038 12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-benzyl-3,10,13-trioxo-1,4,9triaza-cyclotridecane-5-carboxylic acid amide 103039 12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-(4-nitro-benzyl)-3,7,13-trioxo-1,4,8triaza-cyclotridecane-5-carboxylic acid amide 103046 (S)-N-(2-Amino-1-benzylcarbamoyl-ethyl)-2-{3-[1-(2,6-dichloro-benzyl)-3-pyrrolidin-1-ylmethyl-1H-indol-6-yl]-ureido}-3-(3,4-difluoro-phenyl)-propionamide 103061 (S)-3-[2-[(S)-2-Acetylamino-3-(1H-indol-3-yl)-propionylamino]-6-(3-o-tolyl-ureido)-hexanoylamino]-N-((R)-1-carbamoyl-2-p-tolyl-ethyl)-succinamic acid 103067 1-(8-Allyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-methoxy-phenyl)-urea 103087 4-Amino-N-benzyl-2-[(S)-2-{3-[1-(2,6-dichloro-benzyl)-3-pyrrolidin-1-ylmethyl-1H-indol-6-yl]-ureido}-3-(3,4-difluoro-phenyl)-propionylamino]-butyramide 103088 (S)-6-Amino-2-[(S)-2-{3-[1-(2,6-dichloro-benzyl)-3-pyrrolidin-1-ylmethyl-1H-indol-6-yl]-ureido}-3-(3,4-difluoro-phenyl)-propionylamino]-hexanoic acid benzylamide 103200 (S)-3-{2-[(S)-2-Acetylamino-3-(1H-indol-3-yl)-propionylamino]-6-[3-(2-chloro-phenyl)-ureido]-hexanoylamino}-N-((R)-1-carbamoyl-2-p-tolyl-ethyl)-succinamic acid 103260 (S)-3-(2-[(S)-2-Acetylamino-3-(1H-indol-3-yl)-propionylamino]-3-{4-[3-(2-chloro-phenyl)-ureido]-phenyl}-propionylamino)-N-((R)-1-carbamoyl-2-p-tolyl-ethyl)-succinamic acid 103269 3-(3-{4-Fluoro-4-[2-(3-fluoro-phenyl)-ethyl]-piperidin-1-yl}-propyl)-5-[1,2,4]triazol-4-yl-1H-indole 103301 (R)-3-{2-[(R)-2-Acetylamino-3-(1H-indol-3-yl)-propionylamino]-3-[3-(3-o-tolyl-ureido)-phenyl]-propionylamino}-N-((S)-1-carbamoyl-2-p-tolyl-ethyl)-succinamic acid 103302 (S)-3-{2-[(S)-2-Acetylamino-3-(1H-indol-3-yl)-propionylamino]-3-[3-(3-o-tolyl-ureido)-phenyl]-propionylamino}-N-((R)-1-carbamoyl-2-p-tolyl-ethyl)-succinamic acid 103312 (S)-5-Guanidino-2-((S)-3-(4-methoxy-phenyl)-2-{3-[1-(3-methyl-benzyl)-3-piperidin-1-ylmethyl-1H-indol-6-yl]-ureido}-propionylamino)-pentanoic acid cyclohexylmethyl-amide 103329 (S)-2-[(S)-2-{3-[1-(4-Fluoro-benzyl)-3-piperidin-1-ylmethyl-1H-indol-6-yl]-ureido}-3-(4-methoxy-phenyl)-propionylamino]-5-guanidino-pentanoic acid cyclohexylmethyl-amide 103470 3-[3-(4-Benzyl-piperidin-1-yl)-2-fluoro-propyl]-5-[1,2,4]triazol-4-yl-1H-indole 103512 (6aR,9R)-7-Methyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid ((R)-sec-butyl)-amide 103700 1-[(2S,3S)-3-(3,5-Bis-trifluoromethyl-benzyloxy)-2-phenyl-piperidin-1-yl]-ethanone 103701 [(2S,3S)-3-(3,5-Bis-trifluoromethyl-benzyloxy)-2-phenyl-piperidin-1-yl]-acetic acid 103723 6-Methoxy-2-(2-methoxy-benzyl)-5-(2-morpholin-4-yl-ethyl)-2,5-dihydro-pyrido[4,3-b]indol-1-one 103744 2-[(2S,3S)-3-(3,5-Bis-trifluoromethyl-benzyloxy)-2-phenyl-piperidin-1-yl]-2-oxo-acetamide 103769 8-chloro-11-(4-methylpiperazin-1-yl)dibenzo[b,f][1,4]thiazepine 103780 [(2S,3S)-3-(3,5-Bis-trifluoromethyl-benzyloxy)-2-phenyl-piperidin-1-yl]-oxo-acetic acid methyl ester 103824 (2S,3S)-1-Benzyl-3-(3,5-bis-trifluoromethyl-benzyloxy)-2-phenyl-piperidine 103854 3-[(2S,3S)-3-(3,5-Bis-trifluoromethyl-benzyloxy)-2-phenyl-piperidin-1-yl]-propionamide 103857 [(2S,3S)-3-(3,5-Bis-trifluoromethyl-benzyloxy)-2-phenyl-piperidin-1-yl]-acetic acid methyl ester 103868 2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-3-(1H-indol-3-yl)-propionylamino]-propionylamino}-N-{[1-(1-butyl-pentylcarbamoyl)-2-(3H-imidazol-4-yl)-ethylcarbamoyl]-methyl}-3-methyl-butyramide 103869 2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-3-(1H-indol-3-yl)-propionylamino]-propionylamino}-N-{[2-(3H-imidazol-4-yl)-1-(1-isobutyl-3-methyl-butylcarbamoyl)-ethylcarbamoyl]-methyl}-3-methyl-butyramide 103870 2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-3-(1H-indol-3-yl)-propionylamino]-propionylamino}-N-{[2-(3H-imidazol-4-yl)-1-(1-propyl-butylcarbamoyl)-ethylcarbamoyl]-methyl}-3-methyl-butyramide 103880 2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-3-(1H-indol-3-yl)-propionylamino]-propionylamino}-N-{[2-(3H-imidazol-4-yl)-1-(1-isobutyl-heptylcarbamoyl)-ethylcarbamoyl]-methyl}-3-methyl-butyramide 103886 7-Methoxy-1-(2-morpholin-4-yl-ethyl)-1H-indole-3-carboxylic acid (1,3,3-trimethyl-bicyclo[2.2.1]hept-2-yl)-amide 103887 7-Methoxy-2-methyl-1-(2-morpholin-4-yl-ethyl)-1H-indole-3-carboxylic acid (1,3,3-trimethyl-bicyclo[2.2.1]hept-2-yl)-amide 103917 2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-3-(1H-indol-3-yl)-propionylamino]-propionylamino}-N-{[2-(3H-imidazol-4-yl)-1-(1-isobutyl-hexylcarbamoyl)-ethylcarbamoyl]-methyl}-3-methyl-butyramide 103943 SID11111344 103973 (7R,9aS)-7-(4-Fluoro-phenoxymethyl)-2-(5-fluoro-pyrimidin-2-yl)-octahydro-pyrido[1,2-a]pyrazine 104140 1-{10-[3-(4-Nitro-phenyl)-allyl]-9,10-diaza-tricyclo[4.2.1.1*2,5*]dec-9-yl}-propan-1-one 104152 3-[4-(4-Chloro-benzyl)-piperazin-1-yl]-1-ethyl-1,3,4,5-tetrahydro-benzo[b]azepin-2-one 104173 1-{10-[3-(3-Chloro-phenyl)-allyl]-9,10-diaza-tricyclo[4.2.1.1*2,5*]dec-9-yl}-propan-1-one 104179 (6aR,10aR)-3-heptyl-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol 104334 1-{10-[3-(3-Nitro-phenyl)-allyl]-9,10-diaza-tricyclo[4.2.1.1*2,5*]dec-9-yl}-propan-1-one 104408 2-[(2S,3S)-3-(2-Methoxy-benzylamino)-2-phenyl-piperidin-1-yl]-acetamide 104431 1-[10-(3-Naphthalen-1-yl-allyl)-9,10-diaza-tricyclo[4.2.1.1*2,5*]dec-9-yl]-propan-1-one 104444 7-Methoxy-1-(2-morpholin-4-yl-ethyl)-1H-indazole-3-carboxylic acid (phenyl-pyridin-2-yl-methyl)-amide 104447 2-[(2S,3S)-3-(3,5-Bis-trifluoromethyl-benzyloxy)-2-phenyl-piperidin-1-yl]-N,N-dimethyl-acetamide 104448 2-[(2S,3S)-3-(3,5-Bis-trifluoromethyl-benzyloxy)-2-phenyl-piperidin-1-yl]-N-methyl-acetamide 104449 4-[(2S,3S)-3-(3,5-Bis-trifluoromethyl-benzyloxy)-2-phenyl-piperidin-1-yl]-butyramide 104479 7-Methoxy-1-(2-morpholin-4-yl-ethyl)-1H-indazole-3-carboxylic acid (2-chloro-6-fluoro-benzyl)-isopropyl-amide 104505 4-[4-(2-Isochroman-1-yl-ethyl)-piperazin-1-yl]-benzenesulfonamide (U-101387) 104678 SID11111796 104857 D-Phe-Cys-Tyr-D-Trp-Arg-Thr-Pen-Thr-NH2 and4-[(4-Allyl-2,5-dimethyl-piperazin-1-yl)-(3-methoxy-phenyl)-methyl]-N,N-diethyl-benzamide (SNC 80) 104888 1-[10-(3-Phenyl-allyl)-9,10-diaza-tricyclo[4.2.1.1*2,5*]dec-9-yl]-propan-1-one 104890 4-[(4-Allyl-2,5-dimethyl-piperazin-1-yl)-(3-hydroxy-phenyl)-methyl]-N,N-diethyl-benzamide 104919 1-[3-(3-Phenyl-allyl)-3,8-diaza-bicyclo[3.2.1]oct-8-yl]-propan-1-one 104990 1-[8-(3-Phenyl-allyl)-3,8-diaza-bicyclo[3.2.1]oct-3-yl]-propan-1-one 105099 4-[(S)-((2R,5S)-4-Allyl-2,5-dimethyl-piperazin-1-yl)-(3-hydroxy-phenyl)-methyl]-N,N-diethyl-benzamide 105123 3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-2-methoxyimino-5-(3-methylcarbamoylmethyl-2-oxo-[1,4']bipiperidinyl-1'-yl)-pentyl]-N-ethyl-benzamide 105179 7-(3-(benzo[d][1,3]dioxol-5-yl)propyl)-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine 105211 N-[5-(3-Carbamoylmethyl-2-oxo-[1,4']bipiperidinyl-1'-yl)-3-(3,4-dichloro-phenyl)-2-methoxyimino-pentyl]-3,5-dichloro-N-ethyl-benzamide 105212 3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-2-methoxyimino-5-(3-methylcarbamoylmethyl-2-oxo-[1,4']bipiperidinyl-1'-yl)-pentyl]-N-ethyl-benzamide 105213 3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-2-methoxyimino-5-(3-methylcarbamoylmethyl-2-oxo-[1,4']bipiperidinyl-1'-yl)-pentyl]-N-ethyl-benzamide 105238 3-[4-(4-Chloro-benzyl)-piperazin-1-yl]-1-ethyl-3,4-dihydro-1H-quinolin-2-one 105248 1-Benzyl-3-methyl-3,7-dihydro-purine-2,6-dione 105249 3-Methyl-1-prop-2-ynyl-3,7-dihydro-purine-2,6-dione 105256 7-[2-(4-Benzyloxy-phenyl)-ethyl]-2-furan-2-yl-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 105260 7-[3-(4-Benzyloxy-phenyl)-propyl]-2-furan-2-yl-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 105263 4-[3-(5-Amino-2-furan-2-yl-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)-propyl]-benzene-1,2-diol 105285 3,5-Dichloro-N-{3-(3,4-dichloro-phenyl)-2-methoxyimino-5-[3-(2-morpholin-4-yl-2-oxo-ethyl)-2-oxo-[1,4']bipiperidinyl-1'-yl]-pentyl}-N-ethyl-benzamide 105286 N-[5-(3-Carbamoylmethyl-2-oxo-[1,4']bipiperidinyl-1'-yl)-3-(3,4-dichloro-phenyl)-2-methoxyimino-pentyl]-3,5-dichloro-N-ethyl-benzamide 105287 7-(4-Benzyloxy-benzyl)-2-furan-2-yl-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 105364 3,5-Dichloro-N-(3-(3,4-dichloro-phenyl)-5-{3-[2-(2-hydroxy-azetidin-1-yl)-2-oxo-ethyl]-2-oxo-[1,4']bipiperidinyl-1'-yl}-2-methoxyimino-pentyl)-N-ethyl-benzamide 105414 2-[4-(4-Chloro-benzyl)-piperazin-1-yl]-1-(2,3-dihydro-indol-1-yl)-ethanone 105420 4-[(S)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-yl)-(3-hydroxy-phenyl)-methyl]-N,N-diethyl-benzamide 105436 3,5-Dichloro-N-(3-(3,4-dichloro-phenyl)-5-{3-[2-(2-hydroxy-azetidin-1-yl)-2-oxo-ethyl]-2-oxo-[1,4']bipiperidinyl-1'-yl}-2-methoxyimino-pentyl)-N-ethyl-benzamide 105437 N-[5-(3-Carbamoylmethyl-2-oxo-[1,4']bipiperidinyl-1'-yl)-3-(3,4-dichloro-phenyl)-2-methoxyimino-pentyl]-3,5-dichloro-N-ethyl-benzamide 105452 4-[(S)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-yl)-(3-hydroxy-phenyl)-methyl]-N,N-diethyl-benzamide 105485 1-(2-{1'-[5-[(3,5-Dichloro-benzoyl)-ethyl-amino]-3-(3,4-dichloro-phenyl)-4-methoxyimino-pentyl]-2-oxo-[1,4']bipiperidinyl-3-yl}-acetyl)-1-methyl-piperidinium 105544 7-(4-Chloro-butyl)-1,3-dimethyl-3,7-dihydro-purine-2,6-dione 105545 7-(3-Chloro-propyl)-1,3-dimethyl-3,7-dihydro-purine-2,6-dione 105548 4-[2-(5-Amino-2-furan-2-yl-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)-ethyl]-phenol 105595 1-Allyl-7-(2-chloro-ethyl)-3-methyl-8-phenyl-3,7-dihydro-purine-2,6-dione 105598 3-Methyl-1-(3-phenyl-propyl)-3,7-dihydro-purine-2,6-dione 105599 3-Methyl-1-phenethyl-3,7-dihydro-purine-2,6-dione 105600 3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-5-(3-dimethylcarbamoylmethyl-2-oxo-[1,4']bipiperidinyl-1'-yl)-2-methoxyimino-pentyl]-N-ethyl-benzamide 105601 3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-5-(3-dimethylcarbamoylmethyl-2-oxo-[1,4']bipiperidinyl-1'-yl)-2-methoxyimino-pentyl]-N-ethyl-benzamide 105602 3,5-Dichloro-N-{3-(3,4-dichloro-phenyl)-2-methoxyimino-5-[3-(2-morpholin-4-yl-2-oxo-ethyl)-2-oxo-[1,4']bipiperidinyl-1'-yl]-pentyl}-N-ethyl-benzamide 105712 4-[(S)-((2R,5S)-4-Allyl-2,5-dimethyl-piperazin-1-yl)-(3-methoxy-phenyl)-methyl]-N,N-diethyl-benzamide 105735 3,5-Dihydroxy-4-(2-hydroxy-6-isopropoxycarbonyl-benzoyl)-benzoic acid (1R,2R)-2-(4-hydroxy-benzoylamino)-cyclopentyl ester 105789 3,5-Dichloro-N-{3-(3,4-dichloro-phenyl)-2-methoxyimino-5-[3-(2-morpholin-4-yl-2-oxo-ethyl)-2-oxo-[1,4']bipiperidinyl-1'-yl]-pentyl}-N-ethyl-benzamide 105797 1-Butyl-3,7-dihydro-purine-2,6-dione 105798 4-(2-Butoxycarbonyl-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (3R,4R)-4-(4-hydroxy-benzoylamino)-pyrrolidin-3-yl ester 105799 4-(2-Cyclohexylmethoxycarbonyl-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (3R,4R)-4-(4-hydroxy-benzoylamino)-pyrrolidin-3-yl ester 105800 3,5-Dihydroxy-4-(2-hydroxy-6-isobutoxycarbonyl-benzoyl)-benzoic acid (3R,4R)-4-(4-hydroxy-benzoylamino)-pyrrolidin-3-yl ester 105825 3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-5-(3-dimethylcarbamoylmethyl-2-oxo-[1,4']bipiperidinyl-1'-yl)-2-methoxyimino-pentyl]-N-ethyl-benzamide 105826 3,5-Dichloro-N-(3-(3,4-dichloro-phenyl)-5-{3-[2-(2-hydroxy-azetidin-1-yl)-2-oxo-ethyl]-2-oxo-[1,4']bipiperidinyl-1'-yl}-2-methoxyimino-pentyl)-N-ethyl-benzamide 105836 8-Bromo-6-methoxy-2a,3,4,5-tetrahydro-2H-naphtho[1,8-bc]furan-4-ylamine 105903 1-Phenethyl-3,7-dihydro-purine-2,6-dione 105904 1-Cyclopentyl-3,7-dihydro-purine-2,6-dione 105934 5'-amino-5'-deoxyadenosine 105937 4-(2-Ethoxycarbonyl-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (3R,4R)-4-(4-hydroxy-benzoylamino)-pyrrolidin-3-yl ester 105938 3,5-Dihydroxy-4-(2-hydroxy-6-methoxycarbonyl-benzoyl)-benzoic acid (3R,4R)-4-(4-hydroxy-benzoylamino)-pyrrolidin-3-yl ester 105945 4-(2-Ethoxycarbonyl-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (1R,2R)-2-(4-hydroxy-benzoylamino)-cyclopentyl ester 105946 3,5-Dihydroxy-4-(2-hydroxy-6-methoxycarbonyl-benzoyl)-benzoic acid (1R,2R)-2-(4-hydroxy-benzoylamino)-cyclopentyl ester 105950 (R)-1-(4-bromo-2,5-dimethoxyphenyl)propan-2-amine 105961 3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-2-[(Z)-methoxyimino]-5-(2-oxo-[1,4']bipiperidinyl-1'-yl)-pentyl]-N-methyl-benzamide 105982 (2R,3R,4S,5R)-2-(6-(3-iodobenzylamino)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 105991 4-(3-(5-amino-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)propyl)phenol 106023 4-(5-Amino-2-furan-2-yl-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-ylmethyl)-phenol 106038 Ac-DPhe-Arg-DTrp-NH2 106041 7-(2-Chloro-ethyl)-8-phenyl-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 106065 7-(3-(3,4-dimethoxyphenyl)propyl)-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine 106100 3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-2-methoxyimino-5-(2-oxo-[1,4']bipiperidinyl-1'-yl)-pentyl]-N-ethyl-benzamide 106223 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (3R,5R)-4-amino-2-((S)-4-hydroxy-benzoylamino)-cyclopentyl ester 106301 4-(Indan-5-ylamino)-5-[1-[3-methyl-5-(morpholine-4-carbonyl)-1H-pyrrol-2-yl]-meth-(Z)-ylidene]-5,7-dihydro-pyrrolo[2,3-d]pyrimidin-6-one 106303 5-[4-(4-Chloro-2-fluoro-phenylamino)-6-oxo-6,7-dihydro-pyrrolo[2,3-d]pyrimidin-(5Z)-ylidenemethyl]-4-methyl-1H-pyrrole-2-carboxylic acid (2-diethylamino-ethyl)-amide 106337 4-(Benzenesulfonylamino-methyl)-cyclohexanecarboxylic acid (3a,4,5,9b-tetrahydro-1H-benzo[e]indol-2-yl)-amide 106409 5-[4-(3-Ethynyl-phenylamino)-6-oxo-6,7-dihydro-pyrrolo[2,3-d]pyrimidin-(5Z)-ylidenemethyl]-4-methyl-1H-pyrrole-2-carboxylic acid (2-morpholin-4-yl-ethyl)-amide 106456 1-Allyl-3,7-dihydro-purine-2,6-dione 106457 1-Prop-2-ynyl-3,7-dihydro-purine-2,6-dione 106458 4-(2-Acetoxymethoxycarbonyl-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (3R,4R)-4-(4-hydroxy-benzoylamino)-pyrrolidin-3-yl ester 106459 4-[2-(2,2-Dimethyl-propionyloxymethoxycarbonyl)-6-hydroxy-benzoyl]-3,5-dihydroxy-benzoic acid (3R,4R)-4-(4-hydroxy-benzoylamino)-pyrrolidin-3-yl ester 106498 (6aR,12bS)-10-Bromo-6-methyl-5,6,6a,7,8,12b-hexahydro-benzo[a]phenanthridin-11-ol 106695 [14-(1H-Indol-3-ylmethyl)-5-isopropyl-8-methyl-4,7,10,13,16-pentaoxo-hexadecahydro-3a,6,9,12,15-pentaaza-cyclopentacyclopentadecen-11-yl]-acetic acid 106696 [8-(1H-Indol-3-ylmethyl)-11-isobutyl-14-isopropyl-12-methyl-4,7,10,13,16-pentaoxo-hexadecahydro-3a,6,9,12,15-pentaaza-cyclopentacyclopentadecen-5-yl]-acetic acid 106708 2-[(1-Methyl-cyclopropanecarbonyl)-amino]-benzothiazole-6-carboxylic acid (2-chloro-6-methyl-phenyl)-amide 106716 N-{4-[(7-Chloro-3a,4,5,9b-tetrahydro-1H-benzo[e]indol-2-ylamino)-methyl]-cyclohexylmethyl}-benzenesulfonamide 106749 2-(2-Cyclopropyl-acetylamino)-benzothiazole-6-carboxylic acid (2-chloro-6-methyl-phenyl)-amide 106752 2-[(2-Phenyl-cyclopropanecarbonyl)-amino]-benzothiazole-6-carboxylic acid (2-chloro-6-methyl-phenyl)-amide 106754 2-amino-4-methyl-N-(2,4,6-trimethylphenyl)-1,3-thiazole-5-carboxamide 106882 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (3S,5R)-4-hydroxy-2-((S)-4-hydroxy-benzoylamino)-cyclopentyl ester 106907 4-(2,4-Dichloro-phenylamino)-7-((E)-2-pyridin-4-yl-vinyl)-quinoline-3-carbonitrile 106945 2-[[(tert-butyloxy)carbonyl]-amino]-4-methyl-N-(2,4,6-trimethylphenyl)-1,3-thiazole-5-carboxamide 106952 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (3S,4R)-3-(4-hydroxy-benzoylamino)-oxepan-4-yl ester 106959 [14-(1H-Indol-3-ylmethyl)-11-isobutyl-8-isopropyl-4,5-dimethyl-3,6,9,12,15-pentaoxo-1,4,7,10,13pentaaza-cyclopentadec-2-yl]-acetic acid 106960 [14-(1H-Indol-3-ylmethyl)-11-isobutyl-8-isopropyl-4-methyl-3,6,9,12,15-pentaoxo-1,4,7,10,13pentaaza-cyclopentadec-2-yl]-acetic acid 106961 [(R)-8-(1H-Indol-3-ylmethyl)-11-isobutyl-14-isopropyl-4,7,10,13,16-pentaoxo-hexadecahydro-3a,6,9,12,15-pentaaza-cyclopentacyclopentadecen-5-yl]-acetic acid 107003 3-[8-(1H-Indol-3-ylmethyl)-11-isobutyl-14-isopropyl-4,7,10,13,16-pentaoxo-hexadecahydro-3a,6,9,12,15-pentaaza-cyclopentacyclopentadecen-5-yl]-propionic acid 107056 4-(2,4-Dichloro-5-methoxy-phenylamino)-7-pyridin-3-ylethynyl-quinoline-3-carbonitrile 107062 1-{5-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-thiophen-2-ylmethyl}-piperidin-2-one 107063 1-{5-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-thiophen-2-ylmethyl}-azepan-2-one 107064 4-(2,4-Dichloro-5-methoxy-phenylamino)-7-((E)-2-pyridin-4-yl-vinyl)-quinoline-3-carbonitrile 107067 4-(3-Chloro-4-fluoro-phenylamino)-5-[1-(3,5-dimethyl-1H-pyrrol-2-yl)-meth-(Z)-ylidene]-5,7-dihydro-pyrrolo[2,3-d]pyrimidin-6-one 107104 5-[4-(3-Chloro-4-fluoro-phenylamino)-6-oxo-6,7-dihydro-pyrrolo[2,3-d]pyrimidin-(5Z)-ylidenemethyl]-4-methyl-1H-pyrrole-2-carboxylic acid (2-diethylamino-ethyl)-amide 107105 4-(3-Chloro-4-fluoro-phenylamino)-5-[1-[5-(4-ethyl-piperazine-1-carbonyl)-3-methyl-1H-pyrrol-2-yl]-meth-(Z)-ylidene]-5,7-dihydro-pyrrolo[2,3-d]pyrimidin-6-one 107129 (S)-1-{5-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-thiophen-2-ylmethyl}-pyrrolidine-2-carboxylic acid methyl ester 107131 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (3R,4R)-3-(4-hydroxy-benzoylamino)-thiepan-4-yl ester 107132 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (3R,4R)-3-(4-hydroxy-benzoylamino)-1,1-dioxo-1lambda*6*-thiepan-4-yl ester 107133 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (1R,2S)-2-(4-hydroxy-benzoylamino)-cycloheptyl ester 107148 4-(3-Chloro-4-fluoro-phenylamino)-5-[1-[3-methyl-5-(4-methyl-piperazine-1-carbonyl)-1H-pyrrol-2-yl]-meth-(Z)-ylidene]-5,7-dihydro-pyrrolo[2,3-d]pyrimidin-6-one 107160 {5-[4-(2-Propoxy-phenyl)-piperazin-1-ylmethyl]-thiophen-3-yl}-methanol 107172 2-Fluoro-N-{4-[(7-methoxy-3a,4,5,9b-tetrahydro-1H-benzo[e]indol-2-ylamino)-methyl]-cyclohexylmethyl}-benzenesulfonamide 107184 2-(3-Phenyl-ureido)-benzothiazole-6-carboxylic acid (2,4,6-trimethyl-phenyl)-amide 107193 1-(5-Bromo-thiophen-2-ylmethyl)-4-(2-methoxy-phenyl)-piperazine 107194 5-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-thiophene-2-carbaldehyde 107195 1-{5-[4-(2-Propoxy-phenyl)-piperazin-1-ylmethyl]-thiophen-2-ylmethyl}-piperidin-2-one 107203 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (3S,4R)-3-(4-hydroxy-benzoylamino)-azepan-4-yl ester 107214 [14-(1H-Indol-3-ylmethyl)-11-isobutyl-8-isopropyl-5-methyl-3,6,9,12,15-pentaoxo-1,4,7,10,13pentaaza-cyclopentadec-2-yl]-acetic acid 107217 2-Acetylamino-benzothiazole-6-carboxylic acid (2,4,6-trimethyl-phenyl)-amide 107225 N-{4-[(7-Methoxy-3a,4,5,9b-tetrahydro-1H-benzo[e]indol-2-ylamino)-methyl]-cyclohexylmethyl}-benzenesulfonamide 107241 4-[(2-Fluoro-benzenesulfonylamino)-methyl]-cyclohexanecarboxylic acid (7-methoxy-3a,4,5,9b-tetrahydro-1H-benzo[e]indol-2-yl)-amide 107252 2-[(2-Methyl-cyclopropanecarbonyl)-amino]-benzothiazole-6-carboxylic acid (2-chloro-6-methyl-phenyl)-amide 107258 4-(Benzenesulfonylamino-methyl)-cyclohexanecarboxylic acid (7-hydroxy-3a,4,5,9b-tetrahydro-1H-benzo[e]indol-2-yl)-amide 107259 N-{4-[(7-Hydroxy-3a,4,5,9b-tetrahydro-1H-benzo[e]indol-2-ylamino)-methyl]-cyclohexylmethyl}-benzenesulfonamide 107304 5-[4-(1-Benzyl-1H-indol-5-ylamino)-6-oxo-6,7-dihydro-pyrrolo[2,3-d]pyrimidin-(5Z)-ylidenemethyl]-4-methyl-1H-pyrrole-2-carboxylic acid (2-morpholin-4-yl-ethyl)-amide 107305 4-(1-Benzyl-1H-indazol-5-ylamino)-5-[1-[3-methyl-5-(morpholine-4-carbonyl)-1H-pyrrol-2-yl]-meth-(Z)-ylidene]-5,7-dihydro-pyrrolo[2,3-d]pyrimidin-6-one 107306 4-(1-Benzyl-1H-indol-5-ylamino)-5-[1-[3-methyl-5-(morpholine-4-carbonyl)-1H-pyrrol-2-yl]-meth-(Z)-ylidene]-5,7-dihydro-pyrrolo[2,3-d]pyrimidin-6-one 107365 5-[4-(3-Chloro-4-fluoro-phenylamino)-6-oxo-6,7-dihydro-pyrrolo[2,3-d]pyrimidin-(5Z)-ylidenemethyl]-4-methyl-1H-pyrrole-2-carboxylic acid (2-morpholin-4-yl-ethyl)-amide 107368 4-(3-Chloro-4-fluoro-phenylamino)-5-[1-[5-(3,5-dimethyl-piperazine-1-carbonyl)-3-methyl-1H-pyrrol-2-yl]-meth-(Z)-ylidene]-5,7-dihydro-pyrrolo[2,3-d]pyrimidin-6-one 107375 4-(3-Chloro-4-fluoro-phenylamino)-5-[1-[3-methyl-5-(morpholine-4-carbonyl)-1H-pyrrol-2-yl]-meth-(Z)-ylidene]-5,7-dihydro-pyrrolo[2,3-d]pyrimidin-6-one 107406 1-{5-[4-(2-Propoxy-phenyl)-piperazin-1-ylmethyl]-thiophen-3-ylmethyl}-piperidin-2-one 107424 4-(2,4-Dichloro-5-methoxy-phenylamino)-6-methoxy-7-((E)-2-pyridin-4-yl-vinyl)-quinoline-3-carbonitrile 107440 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (3R,4R)-3-(4-hydroxy-benzoylamino)-piperidin-4-yl ester 107444 5-[4-(3-Chloro-4-fluoro-phenylamino)-6-oxo-6,7-dihydro-pyrrolo[2,3-d]pyrimidin-(5Z)-ylidenemethyl]-4-methyl-1H-pyrrole-2-carboxylic acid 107445 4-(2,4-Dichloro-5-methoxy-phenylamino)-6-methoxy-7-pyridin-3-ylethynyl-quinoline-3-carbonitrile 107478 1-{5-[4-(2-Propoxy-phenyl)-piperazin-1-ylmethyl]-thiophen-3-ylmethyl}-pyrrolidin-2-one 107479 1-{5-[4-(2-Propoxy-phenyl)-piperazin-1-ylmethyl]-thiophen-3-ylmethyl}-azepan-2-one 107503 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (3S,5R)-2-((S)-4-hydroxy-benzoylamino)-4-hydroxymethyl-cyclopentyl ester 107504 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (3R,5R)-4-aminomethyl-2-((S)-4-hydroxy-benzoylamino)-cyclopentyl ester 107505 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (3S,5R)-4-aminomethyl-2-((S)-4-hydroxy-benzoylamino)-cyclopentyl ester 107506 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (3R,5R)-2-((S)-4-hydroxy-benzoylamino)-4-hydroxymethyl-cyclopentyl ester 107554 (S)-1-[4-(4-benzhydrylthiosemicarbazido)-3-nitrobenzenesulfonyl]pyrrolidine-2-carboxylic acid{2-[(2-dimethylaminoethyl)methylamino]ethyl}amide (bradyzide) 107585 SID26751810 107601 1-{5-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-thiophen-2-ylmethyl}-piperidin-2-ol 107683 4-[4-Amino-5-(4-phenoxy-phenyl)-pyrrolo[2,3-d]pyrimidin-7-yl]-cyclopentane-1,2-diol 107684 7-Cyclopentyl-5-(2-phenoxy-phenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine 107721 7-Cyclopentyl-5-(3-phenoxy-phenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine 107734 4-(Benzenesulfonylamino-methyl)-cyclohexanecarboxylic acid (7-chloro-3a,4,5,9b-tetrahydro-1H-benzo[e]indol-2-yl)-amide 107735 4-(Benzenesulfonylamino-methyl)-cyclohexanecarboxylic acid (7-methoxy-3a,4,5,9b-tetrahydro-1H-benzo[e]indol-2-yl)-amide 107739 2-[(2-Pyrrolidin-1-ylmethyl-cyclopropanecarbonyl)-amino]-benzothiazole-6-carboxylic acid (2-chloro-6-methyl-phenyl)-amide 107740 2-[(2-Dimethylaminomethyl-cyclopropanecarbonyl)-amino]-benzothiazole-6-carboxylic acid (2-chloro-6-methyl-phenyl)-amide 107748 2-[4-Amino-5-(4-phenoxy-phenyl)-pyrrolo[2,3-d]pyrimidin-7-yl]-cyclopentanol 107756 3-[4-Amino-5-(4-phenoxy-phenyl)-pyrrolo[2,3-d]pyrimidin-7-yl]-cyclopentanol 107769 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (1R,2R)-2-(4-hydroxy-benzoylamino)-cycloheptyl ester 107771 2-[(2-Hydroxymethyl-cyclopropanecarbonyl)-amino]-benzothiazole-6-carboxylic acid (2-chloro-6-methyl-phenyl)-amide 107786 7-tert-Butyl-5-(4-phenoxy-phenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine 107787 (4-Phenoxy-phenyl)-quinazolin-4-yl-amine 107830 2-(3-Methyl-ureido)-benzothiazole-6-carboxylic acid (2,4,6-trimethyl-phenyl)-amide 107867 1-[4-(4-benzhydrylthiosemicarbazido)-3-nitrobenzenesulfonyl]-1H-pyrrole-2-carboxylic acid{2-[(2-dimethylaminoethyl)methylamino]ethyl}amide 107908 1'N-[1-(6-aminohexylcarbamoyl)-2-(1H-3-indolyl)-(1S)-ethyl]spiro[1H-indene-1,4'-(hexahydropyridine)]-1'-carboxamide 107920 1'N-[1-(4-aminobutylcarbamoyl)-2-(1H-3-indolyl)-(1R)-ethyl]spiro[1H-indene-1,4'-(hexahydropyridine)]-1'-carboxamide 107922 4-(2-Butyl-benzoimidazol-1-ylmethyl)-2,6-diiodo-phenol 107923 4-(2-Butyl-benzoimidazol-1-ylmethyl)-2-iodo-6-methyl-phenol 107928 1-{5-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-thiophen-2-ylmethyl}-pyrrolidin-2-one 107953 3-(2-Butyl-benzoimidazol-1-ylmethyl)-2,6-diiodo-phenol 107975 SID17402282 107982 6-amino-2-[2-(1H-3-indolyl)-1-spiro[1H-indene-1,4'-(hexahydropyridine)]-1-ylcarboxamido-(1S)-ethylcarboxamido]hexanoic acid 108051 7-tert-Butyl-5-(4-chloro-phenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine 108057 1'N-[1-(3-aminopropylcarbamoyl)-2-(1H-3-indolyl)-(1S)-ethyl]spiro[1H-indene-1,4'-(hexahydropyridine)]-1'-carboxamide 108066 1'N-[1-(3-aminomethylcyclohexylmethylcarbamoyl)-2-(1H-3-indolyl)-(1S)-ethyl]spiro[1H-indene-1,4'-(hexahydropyridine)]-1'-carboxamide 108072 ((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-thiophen-2-ylmethyl-amine 108087 7-Isopropyl-5-(4-phenoxy-phenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine 108177 N-[3-(1-{1-Cyclohexylmethyl-2-[4-(2,4-dimethyl-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-2,5-dioxo-imidazolidin-4-yl)-propyl]-guanidine 108187 N-[3-(1-{1-Cyclohexylmethyl-2-[4-(2,6-dimethyl-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-2,5-dioxo-imidazolidin-4-yl)-propyl]-guanidine 108188 N-(3-{1-[1-Cyclohexylmethyl-2-oxo-2-(4-o-tolyl-piperazin-1-yl)-ethyl]-2,5-dioxo-imidazolidin-4-yl}-propyl)-guanidine 108210 ((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-dipropyl-amine 108283 (R)-1-[4-(4-benzhydrylthiosemicarbazido)-3-nitrobenzenesulfonyl]pyrrolidine-2-carboxylic acid{2-[(2-dimethylaminoethyl)methylamino]ethyl}amide (bradyzide) 108294 (S)-2-(3,5-Dimethyl-benzyloxy)-1-phenyl-ethylamine 108401 1'N-[1-[3-aminomethyl-(1S,3R)-cyclohexylmethylcarbamoyl]-2-(1H-3-indolyl)-(1S)-ethyl]spiro[1H-indene-1,4'-(hexahydropyridine)]-1'-carboxamide 108402 Ala-Gly-cyclo[Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-Ser-Cys] (SRIF14) 108407 1'N-[1-(4-aminobutylcarbamoyl)-2-(1H-3-indolyl)ethyl]spiro[1H-indene-1,4'-(hexahydropyridine)]-1'-carboxamide 108453 {5-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-thiophen-2-yl}-methanol 108500 4-(2-Butyl-benzoimidazol-1-ylmethyl)-2,6-dichloro-phenol 108517 N-(3-{1-[1-Cyclohexylmethyl-2-oxo-2-(4-phenyl-piperidin-1-yl)-ethyl]-2,5-dioxo-imidazolidin-4-yl}-propyl)-guanidine 108520 (4-Methoxy-benzyl)-((R)-5-methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amine 108550 Benzyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amine 108562 2,6-Dibromo-4-(2-butyl-benzoimidazol-1-ylmethyl)-phenol 108576 5-[3-amino(imino)methylaminopropyl]-3-[3-methyl-1-spiro[2,3-dihydro-1H-indene-1,4'-(hexahydropyridine)]-1-ylcarbonyl-(1R)-butyl]-(5R)-tetrahydro-1H-2,4-imidazoledione 108602 5-[3-amino(imino)methylaminopropyl]-3-[1-benzyl-2-oxo-2-spiro[2,3-dihydro-1H-indene-1,4'-(hexahydropyridine)]-1-yl-(1R)-ethyl]-(5R)-tetrahydro-1H-2,4-imidazoledione 108613 4-(2-Butyl-benzoimidazol-1-ylmethyl)-2,6-dinitro-phenol 108630 ((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-(4-nitro-benzyl)-propyl-amine 108652 1'N-[1-[3-aminomethyl-(1R,3S)-cyclohexylmethylcarbamoyl]-2-(1H-3-indolyl)-(1S)-ethyl]spiro[1H-indene-1,4'-(hexahydropyridine)]-1'-carboxamide 108663 ((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-dipropyl-amine 108672 Furan-2-ylmethyl-((R)-5-methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amine 108673 Benzyl-((R)-5-methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-amine 108689 5-[3-amino(imino)methylaminopropyl]-3-[1-cyclohexylmethyl-2-oxo-2-spiro[1H-indene-1,4'-(hexahydropyridine)]-1-yl-(1R)-ethyl]-(5R)-tetrahydro-1H-2,4-imidazoledione 108701 (4-Fluoro-benzyl)-((R)-5-methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amine 108740 1'N-[1-(4-aminobutylcarbamoyl)-2-(1H-3-indolyl)-(1S)-ethyl]spiro[1H-indene-1,4'-(hexahydropyridine)]-1'-carboxamide 108752 SID11110697 108981 SID29215167 109046 5-(3-amino(imino)methylaminopropyl)-3-(1-(2-naphthylmethyl)-2-oxo-2-spiro[2,3-dihydro-1H-indene-1,4'-(hexahydropyridine)]-1-yl-(1R)-ethyl)-(5R)-tetrahydro-1H-2,4-imidazoledione 109060 4-(2-Butyl-benzoimidazol-1-ylmethyl)-2-methyl-6-nitro-phenol 109078 1-(2-Isochroman-1-yl-ethyl)-4-(4-methoxy-phenyl)-piperazine 109131 4-(2-Butyl-benzoimidazol-1-ylmethyl)-2,6-dimethyl-phenol 109166 Benzyl-((R)-5-methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amine 109189 ((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amine 109200 5-[3-amino(imino)methylaminopropyl]-3-[1-cyclohexylmethyl-2-oxo-2-spiro[2,3-dihydro-1H-indene-1,4'-(hexahydropyridine)]-1-yl-(1R)-ethyl]-(5R)-tetrahydro-1H-2,4-imidazoledione 109201 5-[3-amino(imino)methylaminopropyl]-3-[3-phenyl-1-spiro[2,3-dihydro-1H-indene-1,4'-(hexahydropyridine)]-1-ylcarbonylpropyl]-(5R)-tetrahydro-1H-2,4-imidazoledione 109210 6-(3-Guanidino-propyl)-12-(3H-imidazol-4-ylmethyl)-3-(1H-indol-3-ylmethyl)-9-methyl-2,5,8,11,14,17-hexaoxo-1,4,7,10,13,18hexaaza-cyclotricosane-23-carboxylic acid amide 109397 4-(2-Butyl-benzoimidazol-1-ylmethyl)-phenol 109406 isopropyl 7-(2,6-difluorobenzyl)-3-((benzyl(methyl)amino)methyl)-2-(4-isobutyramidophenyl)-4-oxo-4,7-dihydrothieno[2,3-b]pyridine-5-carboxylate 109422 4-(2-phenyl-5-(pyridin-4-yl)-1H-imidazol-4-yl)phenol 109433 4-(2-Butyl-benzoimidazol-1-ylmethyl)-2-methyl-phenol 109453 4-(2-Phenyl-5-pyridin-4-yl-1H-imidazol-4-yl)-benzoic acid methyl ester 109480 SID26752132 109498 4-(1-methyl-2-(piperidin-4-yl)-4-(3-(trifluoromethyl)phenyl)-1H-imidazol-5-yl)-N-((R)-1-phenylethyl)pyridin-2-amine 109514 (4aR,10bR)-4-propyl-3,4,4a,5,6,10b-hexahydro-2H-naphtho[1,2-b][1,4]oxazin-9-ol 109524 4-[2-(2-Butyl-benzoimidazol-1-yl)-ethyl]-2,6-diiodo-phenol 109662 5-Dimethylamino-naphthalene-1-sulfonic acid benzo[1,3]dioxol-5-ylamide 109666 3-Benzo[1,2,5]thiadiazol-5-yl-5-hydroxy-5-(4-methoxy-phenyl)-4-(3,4,5-trimethoxy-benzyl)-5H-furan-2-one 109740 3-Benzo[1,3]dioxol-5-yl-1-benzo[1,2,5]thiadiazol-5-ylmethyl-5-propoxy-1H-indole-2-carboxylic acid 109771 3-Benzo[1,3]dioxol-5-yl-1-benzo[1,2,5]oxadiazol-5-ylmethyl-5-propoxy-1H-indole-2-carboxylic acid 109812 Quinoxaline-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide 109813 N-{4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-butyl}-4-iodo-benzamide 110008 4-(2-phenyl-4-(3-(trifluoromethyl)phenyl)-1H-imidazol-5-yl)pyridine 110009 ((S)-1-Phenyl-ethyl)-{4-[2-piperidin-4-yl-5-(3-trifluoromethyl-phenyl)-3H-imidazol-4-yl]-pyrimidin-2-yl}-amine 110071 4-(4-(4-chlorophenyl)-2-phenyl-1H-imidazol-5-yl)pyridine 110193 9H-Fluorene-4-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-amide 110209 Imidazo[4,5-b]pyridine derivative 110210 N-{7-Methyl-2-propyl-3-[2'-(4-propyl-benzoylsulfamoyl)-biphenyl-4-ylmethyl]-3H-imidazo[4,5-b]pyridin-6-yl}-butyramide 110211 N-[3-(2'-Benzoylsulfamoyl-biphenyl-4-ylmethyl)-7-methyl-2-propyl-3H-imidazo[4,5-b]pyridin-6-yl]-butyramide 110214 Imidazo[4,5-b]pyridine derivative 110215 3-{2-Butyl-5-methyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3H-imidazo[4,5-b]pyridin-6-yl}-1,1-diphenyl-urea 110216 Pentanoic acid benzyl-{2-butyl-5-methyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3H-imidazo[4,5-b]pyridin-6-yl}-amide 110243 4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-biphenyl-2-sulfonic acid (3-cyclopentyl-propionyl)-amide 110260 N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-4-(pyridin-2-yl)benzamide 110268 Pentanoic acid [2-butyl-3-(2'-pentanoylsulfamoyl-biphenyl-4-ylmethyl)-3H-imidazo[4,5-b]pyridin-6-yl]-amide 110321 N-{4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-benzamide 110323 N-{4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-benzamide 110333 Imidazo[4,5-b]pyridine derivative 110334 4'-[2-Butyl-6-(3-isopropyl-3-methyl-ureido)-4-oxo-4H-quinazolin-3-ylmethyl]-biphenyl-2-sulfonic acid benzyloxycarbonylamide (L-162620) 110335 Imidazo[4,5-b]pyridine derivative 110358 N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)but-2-enyl)-9H-fluorene-2-carboxamide 110382 Acetic acid 2-methyl-2-aza-bicyclo[2.2.1]hept-6-yl ester 110387 Acetic acid 2-benzyl-2-aza-bicyclo[2.2.1]hept-5-yl ester 110389 5-Dimethylamino-naphthalene-1-sulfonic acid benzo[1,2,5]thiadiazol-5-ylamide 110409 3-Hydroxymethyl-5-[6-(3-iodo-benzylamino)-purin-9-yl]-cyclopentane-1,2-diol 110434 3-(4-Methoxy-phenyl)-1-(6-methyl-benzo[1,2,5]thiadiazol-5-ylmethyl)-5-propoxy-1H-indole-2-carboxylic acid 110472 1-Benzo[1,2,5]thiadiazol-5-ylmethyl-3-(4-methoxy-phenyl)-5-propoxy-1H-indole-2-carboxylic acid 110480 N6-Cyclopentyladenosine 110485 N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-phenyl]-2-trifluoromethyl-benzamide 110524 N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-phenyl]-2-methyl-benzamide 110567 N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-phenyl]-3-fluoro-2-methyl-benzamide 110568 N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-phenyl]-2-chloro-4-fluoro-benzamide 110629 1-Benzo[1,3]dioxol-5-ylmethyl-4-(4-methoxy-phenyl)-2-oxo-1,2-dihydro-benzo[4,5]furo[3,2-b]pyridine-3-carboxylic acid 110640 N-Butyl-N-{2-butyl-7-methyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3H-imidazo[4,5-b]pyridin-6-yl}-benzamide 110641 3-{2-Butyl-7-methyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3H-imidazo[4,5-b]pyridin-6-yl}-1,1-diphenyl-urea 110693 Imidazo[4,5-b]pyridine derivative 110729 N-{3-[2'-(3-Cyclopentyl-propionylsulfamoyl)-biphenyl-4-ylmethyl]-5,7-dimethyl-2-propyl-3H-imidazo[4,5-b]pyridin-6-yl}-butyramide 110730 Pentanoic acid {2-butyl-3-[2'-(3-cyclopentyl-propionylsulfamoyl)-biphenyl-4-ylmethyl]-5-methyl-3H-imidazo[4,5-b]pyridin-6-yl}-amide 110739 N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-phenyl]-2,4-dichloro-benzamide 110741 [1-(1,4-Dimethyl-piperazin-2-ylmethyl)-1H-indol-3-yl]-naphthalen-1-yl-methanone 110742 [1-(4-Methyl-morpholin-3-ylmethyl)-1H-indol-3-yl]-naphthalen-1-yl-methanone 110774 N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-phenyl]-2,3-dimethyl-benzamide 110776 [1-(1-Methyl-piperidin-2-ylmethyl)-1H-indol-3-yl]-naphthalen-1-yl-methanone 110799 1-Benzo[1,2,5]thiadiazol-5-ylmethyl-4-(4-methoxy-phenyl)-2-oxo-1,2-dihydro-benzo[4,5]furo[3,2-b]pyridine-3-carboxylic acid 110803 SID26751528 110810 N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-phenyl]-5-fluoro-2-methyl-benzamide 110833 3-Benzo[1,3]dioxol-5-yl-1-benzo[1,2,5]thiadiazol-5-ylmethyl-5,6-dimethoxy-1H-indole-2-carboxylic acid 110846 N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-phenyl]-2-chloro-benzamide 110876 N-{4-Oxo-2-propyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3,4-dihydro-quinazolin-6-yl}-N-pentyl-benzamide 110935 Pentanoic acid {2-butyl-3-[2'-(3-cyclopentyl-propionylsulfamoyl)-biphenyl-4-ylmethyl]-3H-imidazo[4,5-b]pyridin-6-yl}-amide 110936 Pentanoic acid [2-butyl-3-(2'-hexanoylsulfamoyl-biphenyl-4-ylmethyl)-3H-imidazo[4,5-b]pyridin-6-yl]-amide 111049 N-[2-(3,4-Dichloro-phenyl)-4-(4-hydroxy-4-phenyl-piperidin-1-yl)-butyl]-N-methyl-benzamide 111064 (2R,3R,4S,5R)-2-[2-Chloro-6-(3-iodo-benzylamino)-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 111128 N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-phenyl]-2-methoxy-benzamide 111185 Cetirizine 111257 N-methyl-2-{2-[4-(2-oxo-1,2,4,5-tetrahydro-3H-benzo[cd]indol-2a-yl)-butyl]-1,2,3,4-tetrahydro-beta-carbolin-9-yl}-acetamide 111258 1-Cyclohexyl-4-{1-[4-(4-methoxy-benzenesulfonyl)-phenyl]-vinyl}-piperidine 111270 SID11114137 111375 1-methyl-5-(4-propoxy-1,2,5-thiadiazol-3-yl)-1,2,3,6-tetrahydropyridine 111426 2-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-2,6-dihydro-3H-imidazo[1,2-c]quinazolin-5-one 111439 2a-(4-(4-phenyl-5,6-dihydropyridin-1(2H)-yl)butyl)-2a,3,4,5-tetrahydrobenzo[cd]indol-2(1H)-one 111443 5-(4-Methoxy-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2,3,6-tetrahydro-pyridine 111586 (R)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]indole-2-carbonitrile 111616 2-(1-Benzyl-1,2,3,6-tetrahydro-pyridin-4-yl)-1H-benzoimidazole 111652 5-Chloro-2-[1-(4-chloro-benzyl)-1,2,3,6-tetrahydro-pyridin-4-yl]-benzooxazole 111653 2-(1-Benzyl-1,2,3,6-tetrahydro-pyridin-4-yl)-5-chloro-benzothiazole 111929 4-Bromo-N-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-benzamide 111968 2-[1-(4-Chloro-benzyl)-1,2,3,6-tetrahydro-pyridin-4-yl]-1H-benzoimidazole 112040 5-Chloro-2-[1-(4-chloro-benzyl)-1,2,3,6-tetrahydro-pyridin-4-yl]-1H-benzoimidazole 112053 2-(1-Benzyl-1,2,3,6-tetrahydro-pyridin-4-yl)-benzooxazole 112222 1-((S)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-m-tolyl-urea 112236 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (R)-3-(4-hydroxy-benzoylamino)-azepan-4-yl ester 112340 3-Cyclopropylmethyl-5-ethyl-8-hydroxy-11-methyl-3,4,5,6-tetrahydro-2H-2,6-methano-benzo[d]azocin-1-one 112442 2-[1-(3-Chloro-benzyl)-1,2,3,6-tetrahydro-pyridin-4-yl]-benzothiazole 112443 5-Chloro-2-[1-(4-chloro-benzyl)-1,2,3,6-tetrahydro-pyridin-4-yl]-benzothiazole 112491 2-(1-Benzyl-1,2,3,6-tetrahydro-pyridin-4-yl)-benzothiazole 112492 2-(1-Benzyl-1,2,3,6-tetrahydro-pyridin-4-yl)-5-chloro-benzooxazole 112509 2-[1-(2-Chloro-benzyl)-1,2,3,6-tetrahydro-pyridin-4-yl]-benzothiazole 112518 2-(1-Benzyl-1,2,3,6-tetrahydro-pyridin-4-yl)-5-chloro-1H-benzoimidazole 112539 2-[1-(4-Chloro-benzyl)-1,2,3,6-tetrahydro-pyridin-4-yl]-benzothiazole 112909 (4aS,9aR)-4a-Ethyl-2-propyl-1,2,3,4,4a,9a-hexahydro-benzo[4,5]furo[2,3-c]pyridin-6-ol 113105 1-(2-Methoxy-phenyl)-3-(2-phenyl-quinazolin-4-yl)-urea 113237 4aS,9aR-(-)-cis-4a-Ethyl-2-methyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol 113285 (6aR,10aR)-9-(hydroxymethyl)-6,6-dimethyl-3-(2-methyloctan-2-yl)-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol 113574 4aS,9aR-(-)-cis-4a-ethyl-2-(2-phenylethyl)-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol 113594 N-butyl-N-(3-(4-(5-methylH-imidazo[1,2-a]pyridin-2-yl)phenoxy)propyl)butan-1-amine 113604 (4aS,9aR)-4a-Ethyl-2,9a-dimethyl-1,2,3,4,4a,9a-hexahydro-benzo[4,5]furo[2,3-c]pyridin-6-ol 113662 (4aS,9aR)-2-Cyclopentylmethyl-4a-ethyl-1,2,3,4,4a,9a-hexahydro-benzo[4,5]furo[2,3-c]pyridin-6-ol 113684 1-phenyl-3-(3-(pyridin-2-yl)isoquinolin-1-yl)urea 113702 1-(2-Pyridin-3-yl-quinazolin-4-yl)-3-o-tolyl-urea 113712 1-(2-(diethylamino)quinazolin-4-yl)-3-phenylurea 113722 1-Phenyl-3-(2-pyridin-4-yl-quinazolin-4-yl)-urea 113730 1-(2-Methoxy-phenyl)-3-(2-pyridin-2-yl-quinazolin-4-yl)-urea 113743 1-phenyl-3-(2-(pyridin-3-yl)quinazolin-4-yl)urea 113756 (2-Amino-ethyl)-carbamic acid 4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxymethyl ester 113863 1-phenyl-3-(2-(pyrrolidin-1-yl)quinazolin-4-yl)urea 114064 N-(3-(pyridin-2-yl)isoquinolin-1-yl)benzamide 114103 1-phenyl-3-(2-(pyridin-2-yl)quinazolin-4-yl)urea 114250 SID11114230 114333 2-(2,6-Dimethyl-benzyl)-4,5-dihydro-1H-imidazole 114346 1-phenyl-3-(quinazolin-4-yl)urea 114348 1-Phenyl-2-(3-pyridin-2-yl-isoquinolin-1-yl)-ethanone 114450 Des-AA1,2,5-[IAmp9,Tyr11]-SRIF 114491 (S)-2-{(R)-2-[(3,5-Dimethyl-benzoyl)-methyl-amino]-3-phenyl-propionylamino}-3-(1H-indol-3-yl)-propionic acid 114542 Trifluoro-methanesulfonic acid 11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b,e][1,4]diazepin-2-yl ester 114558 1-(4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)piperidin-1-yl)-2-methylpropan-1-one 114585 1-(benzylsulfonyl)-4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)piperidine 114586 4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)-1-(phenylsulfonyl)piperidine 114588 1-(butylsulfonyl)-4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)piperidine 114590 1-(isopropylsulfonyl)-4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)piperidine 114592 Trifluoro-methanesulfonic acid 11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b,e][1,4]diazepin-8-yl ester 114672 3-{4-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-piperazin-1-ylmethyl}-3,4-dihydro-2H-naphthalen-1-one 114704 1-(4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)piperidin-1-yl)butan-1-one 114706 1-(4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)piperidin-1-yl)propan-1-one 114707 4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)-1-(piperidin-4-yl)piperidine 114739 4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)-1-(propylsulfonyl)piperidine 114751 11-(4-Methyl-piperazin-1-yl)-5H-dibenzo[b,e][1,4]diazepin-8-ol 114768 butyl 4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)piperidine-1-carboxylate 114769 propyl 4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)piperidine-1-carboxylate 114772 methyl 4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)piperidine-1-carboxylate 114780 (5-Bromo-quinoxalin-6-yl)-(3aR,7aS)-octahydro-benzoimidazol-(2Z)-ylidene-amine 114810 SID11111975 114822 (5-Bromo-2-methyl-quinoxalin-6-yl)-imidazolidin-2-ylidene-amine 114834 1-[5-(1H-Imidazol-4-yl)-pentyl]-3-propyl-thiourea 114835 1-Ethyl-3-[5-(1H-imidazol-4-yl)-pentyl]-thiourea 114837 benzyl 4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)piperidine-1-carboxylate 114869 1-(4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)piperidin-1-yl)-2-phenylethanone 114871 cyclopropyl(4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)piperidin-1-yl)methanone 114912 ethyl 4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)piperidine-1-carboxylate 114916 2-Methoxy-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b,e][1,4]diazepine 114954 11-(4-Methyl-piperazin-1-yl)-5H-dibenzo[b,e][1,4]diazepin-2-ol 114994 8-Methoxy-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b,e][1,4]diazepine 115046 1-[5-(1H-Imidazol-4-yl)-pentyl]-3-phenethyl-thiourea 115053 1-Benzyl-3-[5-(1H-imidazol-4-yl)-pentyl]-thiourea 115054 1-[5-(1H-Imidazol-4-yl)-pentyl]-3-isopropyl-thiourea 115093 1-[5-(1H-Imidazol-4-yl)-pentyl]-3-phenyl-thiourea 115094 1-Cyclohexyl-3-[5-(1H-imidazol-4-yl)-pentyl]-thiourea 115168 3-(4-Hydroxy-phenyl)-2-methoxy-acrylic acid (3S,5R)-2-(6-amino-purin-9-yl)-4-(3-1H-imidazol-4-yl-acryloyloxy)-5-((S)-(R)-methylsulfanylmethyl)-tetrahydro-furan-3-yl ester 115196 8-Chloro-1-(4-chloro-phenyl)-[1,2,4]triazolo[4,3-a]quinoxalin-4-ylamine 115245 3-(3-Dimethylamino-propyl)-N-(4'-formyl-2'-methyl-biphenyl-4-yl)-4-methoxy-benzamide 115263 1-(ethylsulfonyl)-4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)piperidine 115272 2-(4-tert-Butyl-2,6-dimethyl-benzyl)-1-methyl-4,5-dihydro-1H-imidazole 115298 isobutyl 4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)piperidine-1-carboxylate 115336 2-(4-Bromo-2,6-dimethyl-benzyl)-4,5-dihydro-1H-imidazole 115349 isopropyl 4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)piperidine-1-carboxylate 115364 (5-Bromo-1,2,3,4-tetrahydro-quinoxalin-6-yl)-imidazolidin-2-ylidene-amine 115365 (5-Bromo-quinoxalin-6-yl)-[4-methyl-imidazolidin-(2E)-ylidene]-amine 115369 N-[(R)-4-(4-Acetylamino-4-phenyl-piperidin-1-yl)-2-(3,4-dichloro-phenyl)-butyl]-N-methyl-benzamide 115370 (5-Bromo-quinoxalin-6-yl)-thiazolidin-(2Z)-ylidene-amine 115505 Imidazolidin-2-ylidene-(5-iodo-quinoxalin-6-yl)-amine 115545 SID26751967 115579 (5-Chloro-quinoxalin-6-yl)-imidazolidin-2-ylidene-amine 115596 [2-(2,6-Dimethoxy-phenoxy)-ethyl]-((2S,3S)-3-p-tolyl-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-amine 115674 (5-Bromo-quinoxalin-6-yl)-oxazolidin-(2Z)-ylidene-amine 115843 Y-c[D-Pen-(2R,3R)-2-Me-(2')Nal-GSFC]KR-NH2 115844 Y-c[D-Pen-D-(2')Nal-GSFC]KR-NH2 115845 Y-c[D-Pen-(2')Nal-GSFC]KR-NH2 115872 3-(3-Dimethylamino-propyl)-4-methoxy-N-(4-pyridin-4-yl-phenyl)-benzamide 115874 Y-c[D-Pen-(2S,3R)-2-Me-(2')Nal-GSFC]KR-NH2 115875 Y-c[D-Pen-(2S,3S)-2-Me-(2')Nal-GSFC]KR-NH2 115876 Y-c[D-Pen-(2R,3S)-2-Me-(2')Nal-GSFC]KR-NH2 115895 1-(4-Chloro-benzyl)-3-[5-(1H-imidazol-4-yl)-pentyl]-thiourea 115945 3-(3-Dimethylamino-propyl)-N-(4-ethoxy-phenyl)-4-methoxy-benzamide 115958 Y-c[D-Pen-(3-I)Tyr-GSFC]KR-NH2 115960 N-[4-Methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-4-pyridin-4-yl-benzamide 115998 4-Methoxy-N-[2'-methyl-4'-(5-methyl-[1,2,4]oxadiazol-3-yl)-biphenyl-4-yl]-3-(4-methyl-piperazin-1-yl)-benzamide 116026 2-Methyl-biphenyl-4,4'-dicarboxylic acid 4-dimethylamide 4'-{[4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide} 116045 (7,8-Bis-benzyloxy-6-benzyloxymethyl-1,1-dioxo-3-phenyl-6,7,8,8a-tetrahydro-1H,4aH-4,5-dioxa-1lambda*6*-thia-naphthalen-2-yl)-phenyl-methanone 116254 7,8-Bis-benzyloxy-6-hydroxymethyl-3-methyl-6,7,8,8a-tetrahydro-4aH-4,5-dioxa-1-thia-naphthalene-2-carboxylic acid ethyl ester 116375 3-(3,4-Dimethyl-phenyl)-1-propyl-piperidine 116423 7-Benzyloxy-6-benzyloxymethyl-8-hydroxy-3-methyl-6,7,8,8a-tetrahydro-4aH-4,5-dioxa-1-thia-naphthalene-2-carboxylic acid ethyl ester 116449 Y-c[D-Pen-(3,5-diI)Tyr-GSFC]KR-NH2 116502 1-(8-Chloro-5-methylene-5H-dibenzo[a,d]cyclohepten-10-yl)-4-methyl-piperazine 116671 1-[4-(5-{4-[(R)-(4-Chloro-phenyl)-phenyl-methyl]-piperazin-1-ylmethyl}-furan-2-yl)-but-3-ynyl]-N-hydroxy-urea 116701 (7,8-Bis-benzyloxy-6-benzyloxymethyl-1-oxo-3-phenyl-6,7,8,8a-tetrahydro-1H,4aH-4,5-dioxa-1lambda*4*-thia-naphthalen-2-yl)-phenyl-methanone 116730 7,8-Bis-benzyloxy-6-hydroxymethyl-3-methyl-1-oxo-6,7,8,8a-tetrahydro-1H,4aH-4,5-dioxa-1lambda*4*-thia-naphthalene-2-carboxylic acid ethyl ester 116758 N-(1-Ethyl-pyrrolidin-2-ylmethyl)-2-iodo-6-methoxy-3-sulfamoyl-benzamide (iodosulpride) 116803 7,8-Bis-benzyloxy-6-benzyloxymethyl-3-methyl-6,7,8,8a-tetrahydro-4aH-4,5-dioxa-1-thia-naphthalene-2-carboxylic acid ethyl ester 116840 5-Iodo-2,3-dihydro-benzofuran-7-carboxylic acid [1-(4-fluoro-benzyl)-pyrrolidin-2-ylmethyl]-amide (IBF) 116846 7-Benzyloxy-6-benzyloxymethyl-8-hydroxy-3-methyl-1-oxo-6,7,8,8a-tetrahydro-1H,4aH-4,5-dioxa-1lambda*4*-thia-naphthalene-2-carboxylic acid ethyl ester 116848 candesartan 116874 N-(1-Ethyl-pyrrolidin-2-ylmethyl)-2-hydroxy-3-iodo-5,6-dimethoxy-benzamide (NCQ 298) 116910 5-Bromo-N-[1-(4-fluoro-benzyl)-pyrrolidin-2-ylmethyl]-2,3-dimethoxy-benzamide (NCQ115) 116966 7,8-Bis-benzyloxy-6-benzyloxymethyl-3-methyl-1-oxo-6,7,8,8a-tetrahydro-1H,4aH-4,5-dioxa-1lambda*4*-thia-naphthalene-2-carboxylic acid phenyl ester 117022 N*6*-Propyl-4,5,6,7-tetrahydro-benzothiazole-2,6-diamine 117025 (S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propionylamino)-5-guanidino-pentanoylamino]-N-((1S,2S)-1-{(1S,2S)-1-[(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 117036 7,8-Bis-benzyloxy-6-benzyloxymethyl-3-methyl-1-oxo-6,7,8,8a-tetrahydro-1H,4aH-4,5-dioxa-1lambda*4*-thia-naphthalene-2-carboxylic acid ethyl ester 117050 1-(8-Chloro-5-isopropylidene-5H-dibenzo[a,d]cyclohepten-10-yl)-4-methyl-piperazine 117116 11-(4-Methyl-piperazin-1-yl)-5H-dibenzo[b,e][1,4]diazepine 117172 1-(3',4',5'-Trimethoxy-biphenyl-4-ylmethyl)-1,2,3,4-tetrahydro-isoquinoline-6,7-diol 117251 N-[6-(6,7-Dihydroxy-1,2,3,4-tetrahydro-isoquinolin-1-ylmethyl)-naphthalen-2-yl]-4-(3-hexyl-ureido)-benzenesulfonamide 117462 N-(1-Ethyl-pyrrolidin-2-ylmethyl)-2-(2-fluoro-ethoxy)-3-methoxy-benzamide (FEOB) 117547 4-(3,5-Diiodo-4-methoxy-benzyl)-4,5,6,7-tetrahydro-thiazolo[5,4-c]pyridin-2-ylamine 117587 N-[4-(6,7-Dihydroxy-1,2,3,4-tetrahydro-isoquinolin-1-ylmethoxy)-phenyl]-4-(3-hexyl-ureido)-benzenesulfonamide 117646 5-(4-Hexyloxy-furazan-3-yl)-1-methyl-1,2,3,6-tetrahydro-pyridine 117748 N-[3'-(6,7-Dihydroxy-1,2,3,4-tetrahydro-isoquinolin-1-ylmethyl)-biphenyl-4-yl]-4-(3-hexyl-ureido)-benzenesulfonamide 117757 N-[3'-(6,7-Dihydroxy-1,2,3,4-tetrahydro-isoquinolin-1-ylmethyl)-biphenyl-3-yl]-4-(3-hexyl-ureido)-benzenesulfonamide 117792 N-[4'-(6,7-Dihydroxy-1,2,3,4-tetrahydro-isoquinolin-1-ylmethoxy)-biphenyl-3-yl]-4-(3-hexyl-ureido)-benzenesulfonamide 117853 5-(4-Chloro-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2,3,6-tetrahydro-pyridine 117854 Hexyl-[4-(1-methyl-1,2,5,6-tetrahydro-pyridin-3-yl)-[1,2,5]thiadiazol-3-yl]-amine 117865 N-[4-(6,7-Dihydroxy-1,2,3,4-tetrahydro-isoquinolin-1-ylmethyl)-phenyl]-4-(3-hexyl-ureido)-benzenesulfonamide 117892 5-(4-Butoxy-furazan-3-yl)-1-methyl-1,2,3,6-tetrahydro-pyridine 117990 3-Phenyl-pyrrolidine 118069 4-(3-chlorophenylcarbamoyloxy)-N,N,N-trimethylbut-2-yn-1-aminium chloride 118306 (1H-Imidazol-2-yl)-(5-methyl-quinoxalin-6-yl)-amine 118307 (1H-Benzoimidazol-5-yl)-(1H-imidazol-2-yl)-amine 118317 SID24841421 118351 (1S,2R,3S,4R,5S)-4-(1,3-Dibutyl-2,6-dioxo-1,2,3,6-tetrahydro-purin-7-yl)-2,3-dihydroxy-bicyclo[3.1.0]hexane-1-carboxylic acid methylamide 118382 (5-Bromo-quinoxalin-6-yl)-(1H-imidazol-2-yl)-amine 118501 N-[(S)-1-(2,5-Dihydro-pyrrol-1-ylmethyl)-3-methylsulfanyl-propyl]-N-methyl-2-(4-nitro-phenyl)-acetamide 118707 3,5,7-Triethoxy-2-phenyl-chromen-4-one 118746 3,5,7-Trimethoxy-2-phenyl-chromen-4-one 118813 (R)-Phosphoric acid mono-[(S)-(1S,3R,6R)-2,3-dihydroxy-4-(6-hydroxy-purin-9-yl)-bicyclo[3.1.0]hex-1-ylmethyl] ester 118866 1-(3,5-Diiodo-4-methoxy-benzyl)-1,2,3,4-tetrahydro-isoquinoline-6,7-diol 118879 N-(4-chlorophenyl)-4,5-dimethyl-6-(pyridin-4-ylmethyl)pyridazin-3-amine 119090 2-(2,4-Dimethoxy-phenyl)-3,5,7-trimethoxy-chromen-4-one 119095 (2-Bromo-phenyl)-(1H-imidazol-2-yl)-amine 119196 3-Methylsulfanyl-4,5,6,7-tetrahydro-benzo[c]thiophene-1-carboxylic acid hydrazide 119206 (1S,2R,3R,6R)-1-((S)-Hydroxymethyl)-4-(6-hydroxy-purin-9-yl)-bicyclo[3.1.0]hexane-2,3-diol 119207 (1S,2R,6S)-2,3-Dihydroxy-4-(6-hydroxy-purin-9-yl)-bicyclo[3.1.0]hexane-1-carboxylic acid (S,R)-methylamide 119223 (2,6-Dichloro-phenyl)-(1H-imidazol-2-yl)-amine 119229 (2R,4S)-4-(2-Amino-6-hydroxy-purin-9-yl)-1-((R)-(R)-1-hydroxymethyl)-bicyclo[3.1.0]hexane-2,3-diol 119261 1,3-Dibutyl-7-((1S,2R,3S,4R,5R)-3,4-dihydroxy-5-hydroxymethyl-bicyclo[3.1.0]hex-2-yl)-3,7-dihydro-purine-2,6-dione 119323 dimer[Phosphoric acid mono-[(1R,2R,3S,4R,5S)-2,3-dihydroxy-4-(6-hydroxy-purin-9-yl)-bicyclo[3.1.0]hex-1-ylmethyl] ester] 119340 (1H-Imidazol-2-yl)-(5-methyl-3,4-dihydro-2H-benzo[1,4]oxazin-6-yl)-amine 119342 (5-tert-Butyl-4-methoxy-2-methyl-phenyl)-(1H-imidazol-2-yl)-amine 119343 (4-tert-Butyl-3-methoxy-2,6-dimethyl-phenyl)-(1H-imidazol-2-yl)-amine 119344 (1H-Imidazol-2-yl)-(5-methyl-2,3-dihydro-benzo[1,4]dioxin-6-yl)-amine 119345 2'-C-methyladenosine 119368 SID11114036 119384 2-(3,4-Dichloro-phenyl)-N-[(S)-1-(2,5-dihydro-pyrrol-1-ylmethyl)-2-methyl-propyl]-N-methyl-acetamide 119428 N-(4-chlorophenyl)-5-(pyridin-4-ylmethyl)pyrido[2,3-d]pyridazin-8-amine 119463 N1-(4-chlorophenyl)-4-(pyridin-4-ylmethyl)phthalazine-1,7-diamine 119507 1N-methyl-1N-{4-methyl-2-[4-(4-methylhexahydro-1-pyrazinylcarbonyl)benzyloxy]phenyl}-4-[2-(2-ethyl-1H-1-imidazolyl)phenylcarboxamido]benzamide 119522 SID26754241 119580 Biphenyl-2-carboxylic acid (4-{5-[2-(4-dimethylamino-piperidin-1-yl)-2-oxo-ethylidene]-4,4-difluoro-2,3,4,5-tetrahydro-benzo[b]azepine-1-carbonyl}-phenyl)-amide 119710 4-Ethoxy-7-((E)-styryl)-furo[3,2-g]chromen-5-one 119790 N-(4-chlorophenyl)-8-(pyridin-4-ylmethyl)pyrido[3,2-d]pyridazin-5-amine 119805 2-Methyl-furan-3-carboxylic acid [4-({2-[3-([1,4']bipiperidinyl-1'-carbonyl)-phenoxy]-phenyl}-methyl-carbamoyl)-phenyl]-amide 119851 (1H-Imidazol-2-yl)-(4-methoxy-2-methyl-phenyl)-amine 119856 N-(4-chloro-3-(trifluoromethyl)phenyl)-4-(pyridin-4-ylmethyl)phthalazin-1-amine 119882 (1H-Imidazol-2-yl)-quinoxalin-6-yl-amine 119917 (3,4-Dimethoxy-2-methyl-phenyl)-(1H-imidazol-2-yl)-amine 119927 2-Methyl-furan-3-carboxylic acid (4-{5-[2-(4-dimethylamino-piperidin-1-yl)-2-oxo-ethylidene]-4,4-difluoro-2,3,4,5-tetrahydro-benzo[b]azepine-1-carbonyl}-phenyl)-amide 120056 N-(4-chloro-3-methoxyphenyl)-4-(pyridin-4-ylmethyl)phthalazin-1-amine 120057 N-(4-chlorophenyl)-1-(pyridin-4-ylmethyl)pyrido[3,4-d]pyridazin-4-amine 120107 2-Methyl-furan-3-carboxylic acid [4-(methyl-{4-methyl-2-[6-(4-methyl-piperazin-1-yl)-6-oxo-hexyloxy]-phenyl}-carbamoyl)-phenyl]-amide 120324 N-(1-Ethyl-pyrrolidin-2-ylmethyl)-6-hydroxy-2,3-dimethoxy-benzamide 120335 2-Methyl-furan-3-carboxylic acid (4-{[4'-([1,4']bipiperidinyl-1'-carbonyl)-biphenyl-2-yl]-methyl-carbamoyl}-phenyl)-amide 120336 1N-methyl-1N-{4-methyl-2-[6-(4-methylhexahydro-1-pyrazinyl)-6-oxohexyloxy]phenyl}-4-[2-(2-ethyl-1H-1-imidazolyl)phenylcarboxamido]benzamide 120408 2-Methyl-furan-3-carboxylic acid [4-({2-[4-([1,4']bipiperidinyl-1'-carbonyl)-benzyloxy]-4-methyl-phenyl}-methyl-carbamoyl)-phenyl]-amide 120480 (S)-3-bromo-N-((1-ethylpyrrolidin-2-yl)methyl)-2-hydroxy-5,6-dimethoxybenzamide 120535 Suc-Glu-Ala-Val-Gly-Phe-Ala-His-Leu-Asp-lle-lle-Trp-COOH 120536 Suc-Glu-Ala-Val-Tyr-Gly-Ala-His-Leu-Asp-lle-lle-Trp-COOH 120589 (R)-1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichloro-phenyl)-5-(4-hydroxy-4-phenyl-piperidin-1-yl)-pentan-2-one O-methyl-oxime 120590 (S)-1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichloro-phenyl)-5-(4-hydroxy-4-phenyl-piperidin-1-yl)-pentan-2-one O-methyl-oxime 120594 2-[(1R,2S)-1-(3,5-Bis-trifluoromethyl-benzyloxymethyl)-2-(3,4-dichloro-phenyl)-4-(4-hydroxy-4-phenyl-piperidin-1-yl)-butylamino]-acetamide 120595 1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichloro-phenyl)-5-(4-hydroxy-4-phenyl-piperidin-1-yl)-pentan-2-one oxime 120596 1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichloro-phenyl)-5-(4-hydroxy-4-phenyl-piperidin-1-yl)-pentan-2-one O-methyl-oxime 120674 (R)-(2,3-dimethoxyphenyl)(1-(4-fluorophenethyl)piperidin-4-yl)methanol 120695 N-(4-chlorophenyl)-4-(pyridin-4-ylmethyl)phthalazin-1-amine succinate 120702 N-(1-Benzyl-piperidin-4-yl)-5-bromo-2,3-dimethoxy-benzamide 120726 2-Methyl-furan-3-carboxylic acid [4-({2-[2-([1,4']bipiperidinyl-1'-carbonyl)-phenoxy]-phenyl}-methyl-carbamoyl)-phenyl]-amide 120759 2-Methyl-furan-3-carboxylic acid (4-{[2-(6-[1,4']bipiperidinyl-1'-yl-6-oxo-hexyloxy)-4-methyl-phenyl]-methyl-carbamoyl}-phenyl)-amide 120804 4-(1-Naphthalen-1-yl-ethyl)-1H-imidazole 120845 (1H-Imidazol-4-yl)-naphthalen-1-yl-methanone oxalic acid 120884 Suc-Glu-Ala-Gly-Tyr-Phe-Ala-His-Leu-Asp-lle-lle-Trp-COOH 121167 (4-Fluoro-naphthalen-1-yl)-(4-{2-[4-(4-methoxy-benzenesulfonyl)-phenyl]-[1,3]dioxolan-2-yl}-[1,4']bipiperidinyl-1'-yl)-methanone 121191 8-Acenaphthen-1-yl-1-(3-chloro-phenyl)-1,3,8-triaza-spiro[4.5]decan-4-one 121208 3'-Fluoro-4'-[6-(3-isopropyl-ureido)-4-oxo-2-propyl-4H-quinazolin-3-ylmethyl]-biphenyl-2-sulfonic acid 4-ethyl-2-fluoro-benzoylamide 121228 8-[(E)-2-(4-Methoxy-phenyl)-vinyl]-7-methyl-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 121246 2-ethyl-3-(3-fluoro-2'-(2-cyclopropylethyloxycarbonylaminosulphonyl)-biphenyl-4-ylmethyl)-6-(isopropylaminocarbonylamino)-3H-quinazolin-4-one 121251 Suc-Glu-Ala-Val-Tyr-Phe-Ala-His-Leu-Asp-lle-lle-Trp-COOH 121261 8-Acenaphthen-1-yl-1-(4-chloro-phenyl)-1,3,8-triaza-spiro[4.5]decan-4-one 121267 8-[(E)-2-(4-Chloro-phenyl)-vinyl]-7-methyl-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 121299 8-Acenaphthen-1-yl-1-(3-trifluoromethyl-phenyl)-1,3,8-triaza-spiro[4.5]decan-4-one 121328 Suc-Glu-Ala-Val-Tyr-Phe-Ala-His-Leu-Asp-lIe-Gly-Trp-COOH 121329 Suc-Glu-Ala-Val-Tyr-Phe-Ala-His-Leu-Gly-lle-lle-Trp-COOH 121340 4-(2,2-diphenylacetoxy)-1,1-dimethylpiperidinium iodide 121343 2-Ethyl-3-(3-fluoro-2'-(2-cyclopropylethyloxycarbonylaminosulphonyl)-biphenyl-4-ylmethyl)-6-(ethylaminocarbonylamino)-3H-quinazolin-4-one 121344 2-Butyl-3-(3-fluoro-2'-(2-cyclopropylethyloxycarbonylaminosulphonyl)-biphenyl-4-ylmethyl)-6-(isopropyl-methyl-aminocarbonylamino)-3H-quinazolin-4-one 121345 2-Butyl-3-(3-fluoro-2'-(butyloxycarbonylaminosulphonyl)-biphenyl-4-ylmethyl)-6-(isopropyl-methyl-aminocarbonylamino)-3H-quinazolin-4-one 121346 2-{4-[4-(1H-Benzoimidazol-4-yl)-piperazin-1-yl]-butyl}-tetrahydro-pyrrolo[1,2-c]imidazole-1,3-dione 121362 8-Acenaphthen-1-yl-1-(3-bromo-phenyl)-1,3,8-triaza-spiro[4.5]decan-4-one 121363 8-Acenaphthen-1-yl-1-(3-fluoro-phenyl)-1,3,8-triaza-spiro[4.5]decan-4-one 121368 Suc-Glu-Ala-Val-Tyr-Phe-Ala-Gly-Leu-Asp-lle-lle-Trp-COOH 121376 (S)-3-(1H-Indol-3-yl)-2-[(2-phenyl-cyclopropanecarbonyl)-amino]-propionic acid 121437 2-[(1S,2S)-1-(3,5-Bis-trifluoromethyl-benzyloxymethyl)-2-(3,4-dichloro-phenyl)-4-(4-hydroxy-4-phenyl-piperidin-1-yl)-butylamino]-acetamide 121443 2-[1-(3,5-Bis-trifluoromethyl-benzyloxymethyl)-2-(3,4-dichloro-phenyl)-4-(4-hydroxy-4-phenyl-piperidin-1-yl)-butylamino]-acetamide 121444 2-[(1R,2R)-1-(3,5-Bis-trifluoromethyl-benzyloxymethyl)-2-(3,4-dichloro-phenyl)-4-(4-hydroxy-4-phenyl-piperidin-1-yl)-butylamino]-acetamide 121455 3-[(1H-Imidazol-2-yl)-hydrazonomethyl]-1H-indol-5-ol 121462 8-Acenaphthen-1-yl-1-(3-methoxy-phenyl)-1,3,8-triaza-spiro[4.5]decan-4-one 121465 Suc-Glu-Ala-Val-Tyr-Phe-Gly-His-Leu-Asp-lle-lle-Trp-COOH 121466 Suc-Glu-Ala-Val-Tyr-Phe-Ala-His-Gly-Asp-lle-lle-Trp-COOH 121467 Suc-Glu-Ala-Val-Tyr-Phe-Ala-His-Leu-Asp-Gly-lle-Trp-COOH 121477 4-[1-(2,3-Dimethyl-phenyl)-ethyl]-1H-imidazole 121750 (2E)-N-butyl-2-[(5-isopropoxy-1H-indol-3-yl)methylene]hydrazinecarboximidamide 121824 2-methyl-3-(3-fluoro-2'-(3-methyl-butyloxycarbonylaminosulphonyl)-biphenyl-4-ylmethyl)-6-(N-isopropyl-N-methyl-aminocarbonylamino)-3H-quinazolin-4-one 121825 2-methyl-3-(3-fluoro-2'-(3-methyl-butyloxycarbonylaminosulphonyl)-biphenyl-4-ylmethyl)-6-(isopropylaminocarbonylamino)-3H-quinazolin-4-one 121826 2-ethyl-3-(3-fluoro-2'-(3-methyl-butyloxycarbonylaminosulphonyl)-biphenyl-4-ylmethyl)-6-(2-pyridylcarbonylamino)-3H-quinazolin-4-one 121827 2-ethyl-3-(3-fluoro-2'-(butyloxycarbonylaminosulphonyl)-biphenyl-4-ylmethyl)-6-(morpholinylcarbonylamino)-3H-quinazolin-4-one 121849 8-Acenaphthen-1-yl-1-(2-fluoro-phenyl)-1,3,8-triaza-spiro[4.5]decan-4-one 121870 N-(4-Dimethylamino-but-2-ynyl)-N-methyl-acetamide 121873 2-Butyl-3-(3-fluoro-2'-(3-methylbutyloxycarbonylaminosulphonyl)-biphenyl-4-ylmethyl)-6-(isopropyl-methyl-aminocarbonylamino)-3H-quinazolin-4-one 121874 2-Propyl-3-(3-fluoro-2'-(3-methylbutyloxycarbonylaminosulphonyl)-biphenyl-4-ylmethyl)-6-(morpholinylcarbonylamino)-3H-quinazolin-4-one 121894 SID26756729 121902 4'-[2-Ethyl-6-(3-isopropyl-3-methyl-ureido)-4-oxo-4H-quinazolin-3-ylmethyl]-3'-fluoro-biphenyl-2-sulfonic acid cyclopropylethyloxycarbonylamide (L-163579) 121925 (2E)-2-({5-[(3-methylbut-2-enyl)oxy]-1H-indol-3-yl}methylene)-N-pentylhydrazinecarboximidamide 122006 (2E)-2-[(5-oxo-4,5-dihydro-1H-pyrrolo[3,2-b]pyridin-3-yl)methylene]-N-pentylhydrazinecarboximidamide 122022 3'-Fluoro-4'-[6-(3-isopropyl-ureido)-4-oxo-2-propyl-4H-quinazolin-3-ylmethyl]-biphenyl-2-sulfonic acid (2-isobutoxy-acetyl)-amide 122023 Quinazolinone Analog 122041 7-Methyl-1,3-dipropyl-8-[(E)-2-(3,4,5-trimethoxy-phenyl)-vinyl]-3,7-dihydro-purine-2,6-dione 122042 8-[(E)-2-(2,4-Dimethoxy-phenyl)-vinyl]-7-methyl-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 122082 8-[(E)-2-(2,4-Dimethoxy-phenyl)-vinyl]-1,3-diethyl-7-methyl-3,7-dihydro-purine-2,6-dione 122100 2-methyl-3-(3-fluoro-2'-(2-cyclopropylethyloxycarbonylaminosulphonyl)-biphenyl-4-ylmethyl)-6-(N,N-dimethylaminocarbonylamino)-3H-quinazolin-4-one 122102 8-Acenaphthen-1-yl-1-(4-methoxy-phenyl)-1,3,8-triaza-spiro[4.5]decan-4-one 122137 8-Acenaphthen-1-yl-1-p-tolyl-1,3,8-triaza-spiro[4.5]decan-4-one 122185 6-(4-Chloro-phenyl)-7-isopropyl-5H-pyrrolo[2,3-b]pyrazine 122225 8-[(E)-2-(4-Methoxy-2,3-dimethyl-phenyl)-vinyl]-7-methyl-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 122243 N-(2-Dimethylamino-ethyl)-4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-N-methyl-benzenesulfonamide 122252 istradefylline 122354 4'-[2-Ethyl-6-(3-isopropyl-3-methyl-ureido)-4-oxo-4H-quinazolin-3-ylmethyl]-3'-fluoro-biphenyl-2-sulfonic acid 4-ethyl-benzoylamide 122394 2-ethyl-3-(3-fluoro-2'-(3-methyl-but-2-enyloxycarbonylaminosulphonyl)-biphenyl-4-ylmethyl)-6-(N-isopropyl-N-methyl-aminocarbonylamino)-3H-quinazolin-4-one 122397 8-Acenaphthen-1-yl-1-(3,5-dimethyl-phenyl)-1,3,8-triaza-spiro[4.5]decan-4-one 122429 2-((4-(4-chlorophenyl)piperazin-1-yl)methyl)H-pyrazolo[1,5-a]pyridine 122439 N-(1-Carbamoyl-2-phenyl-ethyl)-3-({2-[3-(1H-indol-3-yl)-2-(2-{2-[2-(4-sulfooxy-phenyl)-acetylamino]-hexanoylamino}-acetylamino)-propionylamino]-hexanoyl}-methyl-amino)-succinamic acid 122440 8-Acenaphthen-1-yl-1-(4-fluoro-phenyl)-1,3,8-triaza-spiro[4.5]decan-4-one 122445 7-Methyl-1,3-dipropyl-8-((E)-styryl)-3,7-dihydro-purine-2,6-dione 122485 4'-[2-Ethyl-6-(3-isopropyl-3-methyl-ureido)-4-oxo-4H-quinazolin-3-ylmethyl]-3'-fluoro-biphenyl-2-sulfonic acid (2-isobutoxy-acetyl)-amide 122486 2-ethyl-3-(3-fluoro-2'-(3-methyl-butyloxycarbonylaminosulphonyl)-biphenyl-4-ylmethyl)-6-(N-isopropyl-N-methyl-aminocarbonylamino)-3H-quinazolin-4-one 122504 2-ethyl-3-(3-fluoro-2'-(3-methyl-butyloxycarbonylaminosulphonyl)-biphenyl-4-ylmethyl)-6-(morpholinylcarbonylamino)-3H-quinazolin-4-one 122505 4'-[2-Ethyl-6-(3-ethyl-ureido)-4-oxo-4H-quinazolin-3-ylmethyl]-3'-fluoro-biphenyl-2-sulfonic acid 2-fluoro-benzoylamide 122506 4'-[2-Ethyl-6-(3-isopropyl-ureido)-4-oxo-4H-quinazolin-3-ylmethyl]-3'-fluoro-biphenyl-2-sulfonic acid 4-ethyl-2-fluoro-benzoylamide 122529 8-Acenaphthen-1-yl-1-m-tolyl-1,3,8-triaza-spiro[4.5]decan-4-one 122539 (2E)-N-heptyl-2-[(5-hydroxy-1H-indol-3-yl)methylene]-N-methylhydrazinecarboximidamide 122713 SID26753667 122998 1,3-Diethyl-8-[(E)-2-(4-methoxy-2,3-dimethyl-phenyl)-vinyl]-7-methyl-3,7-dihydro-purine-2,6-dione 122999 1,3-Diethyl-7-methyl-8-[(E)-2-(2,3,4-trimethoxy-phenyl)-vinyl]-3,7-dihydro-purine-2,6-dione 123036 8-[(E)-2-(2,4-Dimethoxy-3-methyl-phenyl)-vinyl]-1,3-diethyl-7-methyl-3,7-dihydro-purine-2,6-dione 123310 (S)-2-(5-Fluoro-6-trifluoromethyl-2,3-dihydro-indol-1-yl)-1-methyl-ethylamine 123311 (S)-2-(6-Ethylsulfanyl-5-fluoro-2,3-dihydro-indol-1-yl)-1-methyl-ethylamine 123314 (S)-1-Methyl-2-(2,3,8,9-tetrahydro-7H-pyrano[2,3-g]indol-1-yl)-ethylamine 123335 (S)-1-(6-chloro-5-fluoro-1H-indol-1-yl)propan-2-amine 123351 (S)-1-Methyl-2-(2,3,7,8-tetrahydro-furo[2,3-g]indol-1-yl)-ethylamine 123516 3-{[1-(2-Piperidin-4-yl-ethanesulfonyl)-piperidine-3-carbonyl]-amino}-propionic acid 123548 3-(2-Carboxy-ethylcarbamoyl)-piperidine-1-carboxylic acid piperidin-4-ylmethyl ester 123549 3-({1-[(Piperidin-4-ylmethyl)-carbamoyl]-piperidine-3-carbonyl}-amino)-propionic acid 123847 Cyclopropyl-{4-[2-(1H-imidazol-4-yl)-ethoxy]-phenyl}-methanone 123850 4-[3-(4-Ethynyl-phenoxy)-propyl]-1H-imidazole 123983 4-[3-(4-Butyl-phenoxy)-propyl]-1H-imidazole 123984 Cyclopropyl-{4-[3-(1H-imidazol-4-yl)-propoxy]-phenyl}-methanol 124033 10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionylamino)-16-(4-hydroxy-benzyl)-13-(1H-indol-3-ylmethyl)-3,3-dimethyl-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentaaza-cycloicosane-4-carboxylic acid (1-carbamoyl-2-hydroxy-propyl)-amide (D-Phe-Cys-Tyr-D-Trp-Lys-Gly-Pen-Thr-NH2) 124056 (S)-2-(6-Chloro-2,3-dihydro-indol-1-yl)-1-methyl-ethylamine 124058 (S)-1-Methyl-2-(6-methylsulfanyl-2,3-dihydro-indol-1-yl)-ethylamine 124099 (S)-2-(6-Chloro-5-fluoro-2,3-dihydro-indol-1-yl)-1-methyl-ethylamine 124111 4-(1-{6-[2-(3,4-dihydroxybenzyl)tetrahydro-1H-1-pyrrolyl]hexyl}tetrahydro-1H-2-pyrrolylmethyl)-1,2-benzenediol 124113 4-(1-Butyl-pyrrolidin-2-ylmethyl)-benzene-1,2-diol 124125 (S)-2-(6-Ethylsulfanyl-2,3-dihydro-indol-1-yl)-1-methyl-ethylamine 124126 SID11111954 124158 (S)-2-(5-Fluoro-6-methylsulfanyl-2,3-dihydro-indol-1-yl)-1-methyl-ethylamine 124176 3-({1-[3-(1-Methyl-piperidin-4-yl)-propionyl]-piperidine-3-carbonyl}-amino)-propionic acid 124184 (S)-2-(5-Fluoro-6-iodo-2,3-dihydro-indol-1-yl)-1-methyl-ethylamine 124205 4-(1-{6-[2-(3,4-dihydroxybenzyl)tetrahydro-1H-1-pyrrolyl]hexyl}tetrahydro-1H-2-pyrrolylmethyl)-1,2-benzenediol 124206 3-{[1-(3-Piperidin-4-yl-propionyl)-pyrrolidine-3-carbonyl]-amino}-propionic acid 124305 2-{[10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl)-propionylamino]-16-(4-hydroxy-benzyl)-7-(1-hydroxy-ethyl)-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentaaza-cycloicosane-4-carbonyl]-amino}-3-hydroxy-butyric acidD-Tyr-Cys-Tyr-D-Trp-Lys-Thr-Cys-Thr-OH 124306 2-{[10-(4-Amino-butyl)-19-(2-amino-2-phenyl-acetylamino)-16-benzyl-7-(1-hydroxy-ethyl)-13-(1H-indol-3-ylmethyl)-20,20-dimethyl-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentaaza-cycloicosane-4-carbonyl]-amino}-3-hydroxy-butyric acid D-PhGly-Pen-Phe-D-Trp-Lys-Thr-Cys-Thr-NH2 124307 3-Phenyl-3-{[1-(3-piperidin-4-yl-propionyl)-piperidine-3-carbonyl]-amino}-propionic acid 124308 5-Methyl-3-{[1-(3-piperidin-4-yl-propionyl)-piperidine-3-carbonyl]-amino}-hexanoic acid 124309 3-{[1-(3-Piperidin-4-yl-propionyl)-piperidine-3-carbonyl]-amino}-butyric acid 124310 3-{Methyl-[1-(3-piperidin-4-yl-propionyl)-piperidine-3-carbonyl]-amino}-propionic acid 124447 2-Hydroxy-3-{[1-(3-piperidin-4-yl-propionyl)-piperidine-3-carbonyl]-amino}-propionic acid 124457 H-Lys-Arg-Pro-Hyp-Gly-Thi-Ser-D-BT-OH (JMV1669) 124462 (S)-5-Phenyl-3-{[(R)-1-(3-piperidin-4-yl-propionyl)-piperidine-3-carbonyl]-amino}-pent-4-ynoic acid 124479 2-Methyl-10-(4-methyl-piperazin-1-yl)-2,4-dihydro-1,2,3,4,9-pentaaza-benzo[f]azulene 124498 (S)-3-Benzo[1,3]dioxol-5-yl-3-{[(R)-1-(3-piperidin-4-yl-propionyl)-piperidine-3-carbonyl]-amino}-propionic acid 124499 1-(3-Piperidin-4-yl-propionyl)-piperidine-3-carboxylic acid [2-(1H-tetrazol-5-yl)-ethyl]-amide 124520 2-{[1-(3-Piperidin-4-yl-propionyl)-piperidine-3-carbonyl]-amino}-succinic acid 1-methyl ester 124529 (S)-6,6-Dimethyl-3-{[(R)-1-(3-piperidin-4-yl-propionyl)-piperidine-3-carbonyl]-amino}-hept-4-ynoic acid 124553 Cyclopropyl-{4-[3-(1H-imidazol-4-yl)-propoxy]-phenyl}-methanone oxime 124586 7-Chloro-2-ethyl-10-(4-methyl-piperazin-1-yl)-2,4-dihydro-1,2,3,4,9-pentaaza-benzo[f]azulene 124635 3-(2-{4-[3-(1H-Imidazol-4-yl)-propoxy]-phenyl}-[1,3]dioxolan-2-yl)-propan-1-ol 124636 2-Ethyl-7-fluoro-10-(4-methyl-piperazin-1-yl)-2,4-dihydro-1,2,3,4,9-pentaaza-benzo[f]azulene 124748 8-Methoxy-quinolin-2-ylamine 124787 4-Hydroxy-1-{4-[3-(1H-imidazol-4-yl)-propoxy]-phenyl}-butan-1-one 124810 4-(1-{6-[2-(3,4-dihydroxybenzyl)tetrahydro-1H-1-pyrrolyl]hexyl}tetrahydro-1H-2-pyrrolylmethyl)-1,2-benzenediol 124849 4-(1-{6-[3,4-dihydroxyphenethyl(propyl)amino]hexyl}tetrahydro-1H-2-pyrrolylmethyl)-1,2-benzenediol 124859 D-Phe-Cys-Tyr-D-Trp-Lys-Thr-Pen-Thr-NH2 (CTP) 124860 19-(2-Amino-3-phenyl-propionylamino)-10-butyl-16-(4-hydroxy-benzyl)-7-(1-hydroxy-ethyl)-13-(1H-indol-3-ylmethyl)-3,3-dimethyl-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentaaza-cycloicosane-4-carboxylic acid (1-carbamoyl-2-hydroxy-propyl)-amide (D-Phe-Cys-Tyr-D-Trp-Nle-Thr-Pen-Thr-NH2) 124866 Cyclopropyl-{4-[4-(1H-imidazol-4-yl)-butoxy]-phenyl}-methanone 124961 Ethyl-(4,5,6,7-tetrahydro-2H-indazol-5-yl)-amine 125068 D-Phe-Cys-Tyr-D-Trp-Arg-Thr-Pen-Thr-NH2 (CTAP) 125071 (3-Methylsulfanyl-propyl)-propyl-(4,5,6,7-tetrahydro-2H-indazol-5-yl)-amine 125134 (S)-3-{[(R)-1-(3-Piperidin-4-yl-propionyl)-piperidine-3-carbonyl]-amino}-3-quinolin-3-yl-propionic acid 125173 3-{[(R)-1-(3-Piperidin-4-yl-propionyl)-piperidine-3-carbonyl]-amino}-propionic acid 125195 (2H-Benzo[1,4]oxazin-3-yl)-[4-(4-phenyl-piperazin-1-yl)-butyl]-amine; compound with but-2-enedioic acid 125199 3-{[(S)-1-(3-Piperidin-4-yl-propionyl)-piperidine-3-carbonyl]-amino}-propionic acid 125202 (S)-3-{[(R)-1-(3-Piperidin-4-yl-propionyl)-piperidine-3-carbonyl]-amino}-3-thiophen-2-yl-propionic acid 125208 bradykinin 125242 3-{[1-(3-Piperidin-4-yl-propionyl)-azepane-3-carbonyl]-amino}-propionic acid 125271 2-{[1-(3-Piperidin-4-yl-propionyl)-piperidine-3-carbonyl]-amino}-ethanesulfonic acid 125312 4-Oxo-1-[1-(3-piperidin-4-yl-propionyl)-piperidine-3-carbonyl]-piperidine-3-carboxylic acid 125359 2-formyl-4-methylphenyl phosphate 125395 H-DArg-Arg-Pro-Hyp-Gly-Thi-Ser-D-BT-OH (JMV1431) 125396 H-DArg-Arg-Pro-Hyp-Gly-Igl-Ser-D-BT-OH (JMV1638) 125469 D-PhGly-Cys-Tyr-D-Trp-Lys-Thr-Pen-Thr-NH2 125470 D-Phe-Cys-Tyr-Trp-Lys-Thr-Pen-Thr-NH2 125474 2-Carboxymethyl-5-methyl-benzoic acid 125475 2-(2-Carboxy-4-methyl-phenyl)-malonic acid 125615 (S)-1-(1H-indol-4-yloxy)-3-((2R,4S)-4-(4-methoxybenzo[b]thiophen-2-yl)-2-methylpiperidin-1-yl)propan-2-ol 125650 (S)-1-(1H-indol-4-yloxy)-3-((2S,4S)-4-(4-methoxybenzo[b]thiophen-2-yl)-2-methylpiperidin-1-yl)propan-2-ol 125724 (S)-1-(1H-indol-4-yloxy)-3-((2R,4R)-4-(4-methoxybenzo[b]thiophen-2-yl)-2-methylpiperidin-1-yl)propan-2-ol 125725 (S)-1-(1H-indol-4-yloxy)-3-((2S,4R)-4-(4-methoxybenzo[b]thiophen-2-yl)-2-methylpiperidin-1-yl)propan-2-ol 125741 (3-Methylsulfanyl-propyl)-(4,5,6,7-tetrahydro-2H-indazol-5-yl)-amine 125769 Phenethyl-(4,5,6,7-tetrahydro-2H-indazol-5-yl)-amine 125770 N-(4-Bromo-3-methyl-isoxazol-5-yl)-2,4,6-trimethyl-benzenesulfonamide 125799 Propyl-(4,5,6,7-tetrahydro-2H-indazol-5-yl)-(2-thiophen-2-yl-ethyl)-amine 125802 Biphenyl-4-sulfonic acid (4-bromo-3-methyl-isoxazol-5-yl)-amide 125804 N-(4-Chloro-3-methyl-isoxazol-5-yl)-benzenesulfonamide 125805 Biphenyl-4-sulfonic acid (3,4-dimethyl-isoxazol-5-yl)-amide 125808 (4,5,6,7-Tetrahydro-2H-indazol-5-yl)-(2-thiophen-2-yl-ethyl)-amine 125809 Phenethyl-propyl-(4,5,6,7-tetrahydro-2H-indazol-5-yl)-amine 125905 (2H-Benzo[1,4]oxazin-3-yl)-[5-(4-pyrimidin-2-yl-piperazin-1-yl)-pentyl]-amine; compound with but-2-enedioic acid 125939 (2H-Benzo[1,4]oxazin-3-yl)-[5-(4-pyridin-2-yl-piperazin-1-yl)-pentyl]-amine; compound with but-2-enedioic acid 125941 (2H-Benzo[1,4]oxazin-3-yl)-[3-(4-pyridin-2-yl-piperazin-1-yl)-propyl]-amine; compound with but-2-enedioic acid 125979 (2H-Benzo[1,4]oxazin-3-yl)-[4-(4-pyrimidin-2-yl-piperazin-1-yl)-butyl]-amine; compound with but-2-enedioic acid 126008 Naphthalene-1-sulfonic acid (4-bromo-3-methyl-isoxazol-5-yl)-amide 126049 (S)-1-(1H-indol-4-yloxy)-3-((2S,4R)-2-methyl-4-(4-methylbenzo[b]thiophen-2-yl)piperidin-1-yl)propan-2-ol 126251 (S)-1-(1H-indol-4-yloxy)-3-((2S,4R)-4-(6-methoxybenzo[b]thiophen-2-yl)-2-methylpiperidin-1-yl)propan-2-ol 126314 (S)-1-(1H-indol-4-yloxy)-3-((2S,4R)-4-(5-chlorobenzo[b]thiophen-2-yl)-2-methylpiperidin-1-yl)propan-2-ol 126389 (S)-1-(1H-indol-4-yloxy)-3-((2S,4R)-4-(6-fluorobenzo[b]thiophen-2-yl)-2-methylpiperidin-1-yl)propan-2-ol 126442 (S)-1-(1H-indol-4-yloxy)-3-((2S,4R)-4-(benzo[b]thiophen-2-yl)-2-methylpiperidin-1-yl)propan-2-ol 126476 5-Dimethylamino-naphthalene-1-sulfonic acid (4-bromo-3-methyl-isoxazol-5-yl)-amide 126477 Biphenyl-2-sulfonic acid (3,4-dimethyl-isoxazol-5-yl)-amide 126485 (2H-Benzo[1,4]oxazin-3-yl)-[3-(4-pyrimidin-2-yl-piperazin-1-yl)-propyl]-amine; compound with but-2-enedioic acid 126549 Propyl-(4,5,6,7-tetrahydro-2H-indazol-5-yl)-amine 126558 (2H-Benzo[1,4]oxazin-3-yl)-[3-(4-phenyl-piperazin-1-yl)-propyl]-amine; compound with but-2-enedioic acid 126559 (2H-Benzo[1,4]oxazin-3-yl)-methyl-[4-(4-pyrimidin-2-yl-piperazin-1-yl)-butyl]-amine 126560 (2H-Benzo[1,4]oxazin-3-yl)-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]-propyl}-amine; compound with but-2-enedioic acid 126572 6-phenyl-thieno[3,2-d]pyrimidin-4-ylamine 126641 2-(4-Amino-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-6-ylsulfanyl)-acetamide 126856 3-benzyl-6-chloro-4-methyl-2-oxo-2H-chromen-7-yl dimethylcarbamate 126932 4-[3-(3H-Imidazol-4-yl)-propyl]-pyridine 126933 2-[3-(3H-Imidazol-4-yl)-propyl]-pyridine 127130 Acetic acid (2S,3R)-2-hydroxymethyl-6-oxo-5-tetradec-(E)-ylidene-tetrahydro-pyran-3-yl ester 127157 Tetradecanoic acid (2R,4S)-2-hydroxymethyl-6-oxo-tetrahydro-pyran-4-yl ester 127309 Acetic acid (2S,3R)-2-hydroxymethyl-6-oxo-5-tetradecyl-tetrahydro-pyran-3-yl ester 127342 Acetic acid (2S,3R)-2-hydroxymethyl-6-oxo-5-tetradecylidene-tetrahydro-pyran-3-yl ester 127351 2-[6-(1-Carbamoyl-ethylsulfanyl)-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-4-ylsulfanyl]-propionamide 127352 2-(4-Amino-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-6-ylsulfanyl)-N-ethyl-acetamide 127355 3-(4-Amino-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-6-ylsulfanyl)-N-ethyl-propionamide 127381 2-[2-(3H-Imidazol-4-yl)-ethyl]-pyridine 127391 3-(4-Amino-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-6-ylsulfanyl)-propionamide 127415 3-[2-(3H-Imidazol-4-yl)-ethyl]-pyridine 127416 immethridine 127461 4-Amino-5-butyl-1-(3-chloro-phenyl)-1,5-dihydro-pyrazolo[3,4-d]pyrimidin-6-one 127485 3-((1H-imidazol-4-yl)methyl)pyridine 127512 {2-[7-Methoxy-1-(2-propionylamino-ethyl)-naphthalen-2-yloxy]-ethyl}-trimethyl-ammonium iodide 127543 2-((1H-imidazol-4-yl)methyl)pyridine 127547 Benzofuran-7-yl-[1-(2-morpholin-4-yl-ethyl)-1H-indol-3-yl]-methanone 127575 4-[2-(3H-Imidazol-4-yl)-ethyl]-pyridine 127576 3-[3-(3H-Imidazol-4-yl)-propyl]-pyridine 127577 4-[3-(3H-Imidazol-4-yl)-propyl]-piperidine 127595 (S)-2-(5,6-Dimethyl-2-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)-4-methyl-pentan-1-ol 127630 N-[2-(5,6-Dimethyl-2-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)-ethyl]-acetamide 127631 (5,6-Dimethyl-2-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)-pyridin-4-ylmethyl-amine 127633 1-[2-(5,6-Dimethyl-2-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)-ethyl]-imidazolidin-2-one 127837 1-(4-fluorophenyl)-4-(2-(isochroman-1-yl)ethyl)piperazine 127842 1-((R)-2-Isochroman-1-yl-ethyl)-4-(4-methoxy-phenyl)-piperazine 127944 N-[2-(2-Butoxy-7-methoxy-naphthalen-1-yl)-ethyl]-propionamide 128017 SID29217631 128026 N-[2-(2-Hydroxy-7-methoxy-naphthalen-1-yl)-ethyl]-propionamide 128136 N-{2-[2-(2-Hydroxy-ethoxy)-7-methoxy-naphthalen-1-yl]-ethyl}-propionamide 128138 N-{2-[2-(2-Iodo-ethoxy)-7-methoxy-naphthalen-1-yl]-ethyl}-propionamide 128140 N-[2-(7-Methoxy-2-propoxy-naphthalen-1-yl)-ethyl]-propionamide 128148 4-(5,6-Dimethyl-2-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)-cyclohexanol 128178 N-{2-[2-(2-Dimethylamino-ethoxy)-7-methoxy-naphthalen-1-yl]-ethyl}-propionamide 128180 N-[2-(2-Ethoxy-7-methoxy-naphthalen-1-yl)-ethyl]-propionamide 128190 (5,6-Dimethyl-2-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)-(1-phenyl-ethyl)-amine (DPEAP) 128353 (R)-3-(5,6-Dimethyl-2-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)-azepan-2-one 128449 (1R,2R)-2-(5,6-Dimethyl-2-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)-indan-1-ol 128450 1-[3-(5,6-Dimethyl-2-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)-propyl]-pyrrolidin-2-one 128511 8-{2-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-oxazol-4-ylmethyl}-8-aza-spiro[4.5]decane-7,9-dione 128514 1-{2-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-thiazol-4-ylmethyl}-piperidin-2-one 128554 {5-[4-(2-Phenoxy-phenyl)-piperazin-1-ylmethyl]-isoxazol-3-yl}-methanol 128586 1-{5-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-isoxazol-3-ylmethyl}-piperidin-2-one 128674 1-{2-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-oxazol-4-ylmethyl}-piperidin-2-one 128679 N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-2-methoxy-phenyl]-2,4-dichloro-benzamide 128712 1-{5-[4-(2-Phenoxy-phenyl)-piperazin-1-ylmethyl]-isoxazol-3-ylmethyl}-azepan-2-one 128716 N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-3-chloro-phenyl]-2,4-dichloro-benzamide 128763 SID26755285 129003 4-[4-((R)-2-Isochroman-1-yl-ethyl)-piperazin-1-yl]-benzenesulfonamide 129159 1-{2-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-oxazol-4-ylmethyl}-pyrrolidin-2-one 129194 1-{5-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-isoxazol-3-ylmethyl}-pyrrolidin-2-one 129211 7-[2-(4-Methoxy-benzoylamino)-6,6-dimethyl-bicyclo[3.1.1]hept-3-yl]-hept-5-enoic acid 129215 1-{2-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-thiazol-4-ylmethyl}-pyrrolidin-2-one 129233 1-{5-[4-(2-Phenoxy-phenyl)-piperazin-1-ylmethyl]-isoxazol-3-ylmethyl}-piperidin-2-one 129271 N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-2-chloro-phenyl]-5-fluoro-2-methyl-benzamide 129272 N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-3-chloro-phenyl]-3-fluoro-2-methyl-benzamide 129280 1-{2-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-oxazol-4-ylmethyl}-azepan-2-one 129294 7-[2-(2-Methoxy-benzoylamino)-6,6-dimethyl-bicyclo[3.1.1]hept-3-yl]-hept-5-enoic acid 129300 2-[2-(6-Trifluoromethyl-indol-1-yl)-ethyl]-decahydro-pyrido[1,2-a][1,4]diazepine 129306 N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-3-methyl-phenyl]-5-fluoro-2-methyl-benzamide 129322 2-[2-(6-Bromo-indol-1-yl)-ethyl]-decahydro-pyrido[1,2-a][1,4]diazepine 129334 1-{5-[4-(2-Phenoxy-phenyl)-piperazin-1-ylmethyl]-isoxazol-3-ylmethyl}-pyrrolidin-2-one 129387 N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-3-chloro-phenyl]-2-chloro-4-fluoro-benzamide 129389 1-Propyl-3-(3-trifluoromethyl-phenyl)-pyrrolidine 129395 N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-3-chloro-phenyl]-2,3-dimethyl-benzamide 129399 N-[4-(5-Dimethylamino-2,3,4,5-tetrahydro-benzo[b]azepine-1-carbonyl)-phenyl]-2-methyl-benzamide 129427 2-{2-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-oxazol-4-ylmethyl}-isoindole-1,3-dione 129435 N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-3-chloro-phenyl]-2-fluoro-3-trifluoromethyl-benzamide 129442 N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-2-methyl-phenyl]-2,4-dichloro-benzamide 129503 N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-3-chloro-phenyl]-2,5-dimethyl-benzamide 129520 1-[2-(6,7-Dimethoxy-isochroman-1-yl)-ethyl]-4-(4-fluoro-phenyl)-piperazine 129521 1-((S)-2-Isochroman-1-yl-ethyl)-4-(4-methoxy-phenyl)-piperazine 129637 N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-3-chloro-phenyl]-2-methyl-benzamide 129717 N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-3-methoxy-phenyl]-5-fluoro-2-methyl-benzamide 129817 7-{6,6-Dimethyl-2-[(naphthalene-2-carbonyl)-amino]-bicyclo[3.1.1]hept-3-yl}-hept-5-enoic acid 129838 7-{2-[(Benzo[1,3]dioxole-5-carbonyl)-amino]-6,6-dimethyl-bicyclo[3.1.1]hept-3-yl}-hept-5-enoic acid 129840 7-{6,6-Dimethyl-2-[(thiophene-2-carbonyl)-amino]-bicyclo[3.1.1]hept-3-yl}-hept-5-enoic acid 129853 Thiophene-3-carboxylic acid [3-(7-methanesulfonylamino-7-oxo-hept-2-enyl)-6,6-dimethyl-bicyclo[3.1.1]hept-2-yl]-amide 129854 7-{6,6-Dimethyl-2-[(thiazole-5-carbonyl)-amino]-bicyclo[3.1.1]hept-3-yl}-hept-5-enoic acid 129864 2-[2-(6-Chloro-indol-1-yl)-ethyl]-decahydro-pyrido[1,2-a][1,4]diazepine 129898 7-{6,6-Dimethyl-2-[(1-methyl-1H-pyrrole-3-carbonyl)-amino]-bicyclo[3.1.1]hept-3-yl}-hept-5-enoic acid 129917 7-[2-(4-Hydroxy-benzoylamino)-6,6-dimethyl-bicyclo[3.1.1]hept-3-yl]-hept-5-enoic acid 129924 3-Naphthalen-1-yl-1-propyl-pyrrolidine 129925 3-Phenyl-1-propyl-pyrrolidine 129935 7-{6,6-Dimethyl-2-[(1H-pyrrole-2-carbonyl)-amino]-bicyclo[3.1.1]hept-3-yl}-hept-5-enoic acid 129947 3-(1-Propyl-pyrrolidin-3-yl)-phenol 129986 Trifluoro-methanesulfonic acid 3-(1-propyl-pyrrolidin-3-yl)-phenyl ester 130021 Cyclohexanecarboxylic acid ((R)-1-phenethyl-pyrrolidin-2-ylmethyl)-amide 130026 2-{4-[4-(7-Chloro-2,3-dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-butyl}-1,1-dioxo-1,2-dihydro-1lambda*6*-benzo[d]isothiazol-3-one 130041 3-Naphthalen-1-yl-pyrrolidine 130049 7-[6,6-Dimethyl-2-(4-nitro-benzoylamino)-bicyclo[3.1.1]hept-3-yl]-hept-5-enoic acid 130051 7-{6,6-Dimethyl-2-[(5-methyl-thiophene-3-carbonyl)-amino]-bicyclo[3.1.1]hept-3-yl}-hept-5-enoic acid 130054 2-{4-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-butyl}-1,1-dioxo-1,2-dihydro-1lambda*6*-benzo[d]isothiazol-3-one 130086 7-{6,6-Dimethyl-2-[(5-phenyl-thiophene-3-carbonyl)-amino]-bicyclo[3.1.1]hept-3-yl}-hept-5-enoic acid 130087 4-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-1-(4-fluoro-phenyl)-butan-1-one 130098 N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-phenyl]-4-chloro-2-methoxy-benzamide 130112 1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-4-(4-phenyl-butyl)-piperazine 130144 N-{2-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-ethyl}-4-fluoro-benzamide 130189 Cyclohexanecarboxylic acid ((S)-1-phenethyl-pyrrolidin-2-ylmethyl)-amide 130190 4-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-1-phenyl-butan-1-one 130200 3-Furan-2-ylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocin-8-ol 130263 7-[2-(Biphenyl-4-sulfonylamino)-6,6-dimethyl-bicyclo[3.1.1]hept-3-yl]-hept-5-enoic acid 130269 7-[2-(2-Furan-3-yl-acetylamino)-6,6-dimethyl-bicyclo[3.1.1]hept-3-yl]-hept-5-enoic acid 130292 7-{2-[(5-Methanesulfonylamino-benzo[b]thiophene-3-carbonyl)-amino]-6,6-dimethyl-bicyclo[3.1.1]hept-3-yl}-hept-5-enoic acid 130293 7-{2-[(6-Hydroxy-benzo[b]thiophene-3-carbonyl)-amino]-6,6-dimethyl-bicyclo[3.1.1]hept-3-yl}-hept-5-enoic acid 130294 7-{2-[(5-Hydroxy-benzo[b]thiophene-3-carbonyl)-amino]-6,6-dimethyl-bicyclo[3.1.1]hept-3-yl}-hept-5-enoic acid 130298 7-{6,6-Dimethyl-2-[(thiophene-3-carbonyl)-amino]-bicyclo[3.1.1]hept-3-yl}-hept-5-enoic acid 130303 Thiophene-3-carboxylic acid {6,6-dimethyl-3-[6-(1H-tetrazol-5-yl)-hex-2-enyl]-bicyclo[3.1.1]hept-2-yl}-amide 130304 (Z)-7-((1R,2R,3S,5S)-2-Benzoylamino-6,6-dimethyl-bicyclo[3.1.1]hept-3-yl)-hept-5-enoic acid 130335 7-{2-[(4-Methoxy-thiophene-3-carbonyl)-amino]-6,6-dimethyl-bicyclo[3.1.1]hept-3-yl}-hept-5-enoic acid 130342 7-{6,6-Dimethyl-2-[(2-methyl-thiophene-3-carbonyl)-amino]-bicyclo[3.1.1]hept-3-yl}-hept-5-enoic acid 130402 (Z)-(R)-7-[(3R,4S,7S)-6,6-Dimethyl-2-(4-phenylazo-benzoylamino)-bicyclo[3.1.1]hept-3-yl]-hept-5-enoic acid 130430 5,7-Dimethyl-3-{1-[4-(1,1,3-trioxo-1,3-dihydro-1lambda*6*-benzo[d]isothiazol-2-yl)-butyl]-piperidin-4-yl}-3H-benzooxazol-2-one 130432 1-(2-Diethylamino-ethyl)-2-(4-ethoxy-benzyl)-1H-benzoimidazole-5-diazonium 130440 7-{2-[(Biphenyl-4-carbonyl)-amino]-6,6-dimethyl-bicyclo[3.1.1]hept-3-yl}-hept-5-enoic acid 130467 3-{1-[4-(1,1,3-Trioxo-1,3-dihydro-1lambda*6*-benzo[d]isothiazol-2-yl)-butyl]-piperidin-4-yl}-5,6,7,8-tetrahydro-3H-naphtho[2,3-d]oxazol-2-one 130470 1-[2-(4-Azido-3-iodo-phenyl)-ethyl]-4-(phenyl-propionyl-amino)-piperidine-4-carboxylic acid methyl ester 130490 7-{2-[(1H-Indole-3-carbonyl)-amino]-6,6-dimethyl-bicyclo[3.1.1]hept-3-yl}-hept-5-enoic acid 130491 7-{2-[(Benzo[b]thiophene-7-carbonyl)-amino]-6,6-dimethyl-bicyclo[3.1.1]hept-3-yl}-hept-5-enoic acid 130531 7-{2-[(5-Fluoro-benzo[b]thiophene-3-carbonyl)-amino]-6,6-dimethyl-bicyclo[3.1.1]hept-3-yl}-hept-5-enoic acid 130532 7-{2-[(Benzofuran-2-carbonyl)-amino]-6,6-dimethyl-bicyclo[3.1.1]hept-3-yl}-hept-5-enoic acid 130541 7-{2-[(Benzo[b]thiophene-3-carbonyl)-amino]-6,6-dimethyl-bicyclo[3.1.1]hept-3-yl}-hept-5-enoic acid 130552 4-{8-[1-(4-Chloro-phenyl)-ethyl]-4-oxo-1,3,8-triaza-spiro[4.5]dec-1-yl}-benzenediazonium 130575 7-{2-[(Benzo[b]thiophene-2-carbonyl)-amino]-6,6-dimethyl-bicyclo[3.1.1]hept-3-yl}-hept-5-enoic acid 130649 6-Fluoro-3-{1-[4-(1,1,3-trioxo-1,3-dihydro-1lambda*6*-benzo[d]isothiazol-2-yl)-butyl]-piperidin-4-yl}-3H-benzooxazol-2-one 130685 6-Methoxy-3-{1-[4-(1,1,3-trioxo-1,3-dihydro-1lambda*6*-benzo[d]isothiazol-2-yl)-butyl]-piperidin-4-yl}-3H-benzooxazol-2-one 130756 3-(3-Methanesulfonyl-phenyl)-1-propyl-pyrrolidine 130780 2-{2-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-ethyl}-1,1-dioxo-1,2-dihydro-1lambda*6*-benzo[d]isothiazol-3-one 130781 2-{4-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-butyl}-isoindole-1,3-dione 130784 2-{2-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-ethyl}-isoindole-1,3-dione 130785 N-{4-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-butyl}-4-fluoro-benzamide 130843 7-{6,6-Dimethyl-2-[(4,5,6,7-tetrahydro-benzo[b]thiophene-3-carbonyl)-amino]-bicyclo[3.1.1]hept-3-yl}-hept-5-enoic acid 130844 7-{6,6-Dimethyl-2-[(5-methyl-4-phenyl-thiophene-3-carbonyl)-amino]-bicyclo[3.1.1]hept-3-yl}-hept-5-enoic acid 130880 7-{2-[(5-Methoxy-thiophene-3-carbonyl)-amino]-6,6-dimethyl-bicyclo[3.1.1]hept-3-yl}-hept-5-enoic acid 130935 5-Methyl-3-{1-[4-(1,1,3-trioxo-1,3-dihydro-1lambda*6*-benzo[d]isothiazol-2-yl)-butyl]-piperidin-4-yl}-3H-benzooxazol-2-one 130936 6-Methyl-3-{1-[4-(1,1,3-trioxo-1,3-dihydro-1lambda*6*-benzo[d]isothiazol-2-yl)-butyl]-piperidin-4-yl}-3H-benzooxazol-2-one 130970 3-{1-[4-(1,1,3-Trioxo-1,3-dihydro-1lambda*6*-benzo[d]isothiazol-2-yl)-butyl]-piperidin-4-yl}-3H-benzooxazol-2-one 130984 3-{1-[4-(5-Nitro-1,1,3-trioxo-1,3-dihydro-1lambda*6*-benzo[d]isothiazol-2-yl)-butyl]-piperidin-4-yl}-3H-benzooxazol-2-one 131000 2-{4-[4-(2-Oxo-2,3-dihydro-benzoimidazol-1-yl)-piperidin-1-yl]-butyl}-isoindole-1,3-dione 131014 2-Oxo-3-{1-[4-(1,1,3-trioxo-1,3-dihydro-1lambda*6*-benzo[d]isothiazol-2-yl)-butyl]-piperidin-4-yl}-2,3-dihydro-benzooxazole-6-carboxylic acid methyl ester 131081 6,7-Dimethoxy-4-(3,4,5-trimethoxy-phenylamino)-quinoline-3-carbonitrile 131162 {2-[5-Azido-2-(4-ethoxy-benzyl)-benzoimidazol-1-yl]-ethyl}-diethyl-amine 131189 etonitazene 131190 8-[1-(4-Chloro-phenyl)-ethyl]-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 131221 1-[2-(4-Azido-phenyl)-ethyl]-4-(phenyl-propionyl-amino)-piperidine-4-carboxylic acid methyl ester 131330 14-[4-azido(methyl)anilino]-4-cyclopropylmethyl-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10-triene-10,17-diol (azidonaltrexone) 131331 14-[4-diazo(methyl)anilino]-4-cyclopropylmethyl-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10-triene-10,17-diol salt (naltrexonediazonium) 131332 1-(4-Azido-phenyl)-8-[1-(4-chloro-phenyl)-ethyl]-1,3,8-triaza-spiro[4.5]decan-4-one 131337 4-Methyl-3-{1-[4-(1,1,3-trioxo-1,3-dihydro-1lambda*6*-benzo[d]isothiazol-2-yl)-butyl]-piperidin-4-yl}-3H-benzooxazol-2-one 131346 1-(2-(4-(6-fluoro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)-3,4-dihydro-1H-isochromene-6-carboxamide 131689 fananserin 131923 ethyl 8-chloro-4-oxo-4,5-dihydro-[1,2,4]triazolo[1,5-a]quinoxaline-2-carboxylate 131924 ethyl 7-chloro-4-oxo-4,5-dihydro-[1,2,4]triazolo[1,5-a]quinoxaline-2-carboxylate 132006 ethyl 7-amino-4-oxo-4,5-dihydro-[1,2,4]triazolo[1,5-a]quinoxaline-2-carboxylate 132104 ethyl 4-oxo-4,5-dihydro-[1,2,4]triazolo[1,5-a]quinoxaline-2-carboxylate 132241 3-Phenyl-6-[4-(2-piperidin-1-yl-ethoxy)-phenyl]-3H-imidazo[4,5-b]pyridine 132243 5-(1-Phenyl-1H-benzoimidazol-5-yl)-1-(3-piperidin-1-yl-propyl)-1H-pyridin-2-one 132273 5-(4-Methoxy-phenyl)-1-phenyl-1H-benzoimidazole 132274 (2-Morpholin-4-yl-ethyl)-[5-(1-phenyl-1H-benzoimidazol-5-yl)-pyridin-2-yl]-amine 132517 {1-[4-(Benzenesulfonyl-methyl-amino)-3-(3-chloro-phenyl)-butyl]-piperidin-4-yl}-ethyl-carbamic acid benzyl ester 132520 {1-[(S)-4-(Benzenesulfonyl-methyl-amino)-3-phenyl-butyl]-piperidin-4-yl}-ethyl-carbamic acid benzyl ester 132585 4-(1-Phenyl-1H-benzoimidazol-5-yl)-1-(3-piperidin-1-yl-propyl)-1H-pyridin-2-one 132615 4-(1-Phenyl-1H-benzoimidazol-5-yl)-1-(3-piperidin-1-yl-propyl)-1H-pyrimidin-2-one 132616 5-(1-Phenyl-1H-benzoimidazol-5-yl)-1-(2-piperidin-1-yl-ethyl)-1H-pyridin-2-one 132617 4-(1-Phenyl-1H-benzoimidazol-5-yl)-1-(2-piperidin-1-yl-ethyl)-1H-pyridin-2-one 132626 1-Phenyl-5-[4-(2-piperidin-1-yl-ethoxy)-phenyl]-1H-benzoimidazole 132630 2-Phenyl-9-(1-phenyl-ethyl)-9H-1,3,9-triaza-fluoren-4-ylamine 132658 1-Phenyl-5-[6-(2-piperidin-1-yl-ethoxy)-pyridin-3-yl]-1H-benzoimidazole 132876 5,6-Dimethyl-2-phenyl-7-(1-phenyl-ethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine (ADPEP) 133063 Benzyl-{(S)-1-[2-(5-[1,2,4]triazol-4-yl-1H-indol-3-yl)-ethyl]-pyrrolidin-3-ylmethyl}-amine 133483 6-(4-Methoxy-phenyl)-3-phenyl-pyrazolo[1,5-a]pyrimidine 133823 SID26756746 133972 1-(6-Benzylamino-9-isopropyl-9H-purin-2-ylamino)-propan-2-ol 134024 Benzyl-(9-isopropyl-9H-purin-6-yl)-amine 134055 3-(6-Amino-9-isopropyl-9H-purin-2-ylamino)-propan-1-ol 134084 1-[(R)-5-(3-Aza-bicyclo[3.2.2]non-3-yl)-1-methyl-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl]-3-m-tolyl-urea 134085 1-(5-Azepan-1-yl-1-methyl-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-m-tolyl-urea 134103 1-(1-Methyl-2-oxo-5-pyrrolidin-1-yl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-m-tolyl-urea 134211 3-Benzo[1,3]dioxol-5-ylmethyl-8-(3,5-bis-trifluoromethyl-benzoyl)-1,3,8-triaza-spiro[4.5]decane-2,4-dione 134213 3-(3,5-Bis-trifluoromethyl-phenyl)-8-(naphthalene-1-carbonyl)-1,3,8-triaza-spiro[4.5]decane-2,4-dione 134214 3-(3,5-Bis-trifluoromethyl-phenyl)-8-(2,4,6-trimethyl-benzoyl)-1,3,8-triaza-spiro[4.5]decane-2,4-dione 134347 1-(2-chloro-2-phenylethyl)-6-(ethylthio)-N-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 134364 1-(2-chloro-2-phenylethyl)-N,N-diethyl-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 134475 (8-(dicyclopropylmethyl)-1,3-dipropylxanthine)8-Dicyclopropylmethyl-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 134534 N-benzyl-1-(2-chloro-2-phenylethyl)-6-(ethylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 134585 3-[2-(4-Amino-phenyl)-ethyl]-8-cyclopentyl-1-propyl-3,7-dihydro-purine-2,6-dione 134618 N-{4-[2-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tetrahydro-purin-3-yl)-ethyl]-phenyl}-isobutyramide 134637 ethyl 1-(2-chloro-2-phenylethyl)-4-(propylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 134671 3-[3-(3,5-Bis-trifluoromethyl-benzyl)-2,4-dioxo-1,3,8-triaza-spiro[4.5]dec-8-ylmethyl]-benzonitrile 134677 3-(6-Cyclopentylamino-9-isopropyl-9H-purin-2-ylamino)-propan-1-ol 134701 ethyl 1-(2-chloro-2-phenylethyl)-4-(cyclopropylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 134779 3-(3,5-Bis-trifluoromethyl-benzyl)-8-(2-naphthalen-1-yl-ethanesulfonyl)-1,3,8-triaza-spiro[4.5]decane-2,4-dione 134800 1-(3,5-Bis-trifluoromethyl-benzyl)-3-methyl-8-(naphthalene-1-carbonyl)-1,3,8-triaza-spiro[4.5]decane-2,4-dione 134821 6-Methyl-1,6-dihydro-2H-pyrrolo[3,2-e]indole-3-carboxylic acid pyridin-3-ylamide 134853 3-{[2-(1-Hydroxymethyl-2-methyl-propylamino)-9-isopropyl-9H-purin-6-ylamino]-methyl}-phenol 134881 Benzoic acid 8-aza-bicyclo[3.2.1]oct-6-yl ester 134928 SID29217495 134938 3-(3,5-Bis-trifluoromethyl-benzyl)-2,4-dioxo-1,3,8-triaza-spiro[4.5]decane-8-carboxylic acid m-tolylamide 134939 1-(2-chloro-2-phenylethyl)-6-(methylthio)-N-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 134941 1-Methyl-1,6,7,8-tetrahydro-pyrrolo[2,3-g]quinoline-5-carboxylic acid pyridin-3-ylamide 134942 1-(2-Chloro-2-phenyl-ethyl)-4-(2-ethoxy-ethylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid ethyl ester 134943 ethyl 1-(2-chloro-2-phenylethyl)-4-morpholino-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 134944 ethyl 4-(benzylamino)-1-(2-chloro-2-phenylethyl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 134970 8-(3,5-Bis-trifluoromethyl-benzoyl)-3-octyl-1,3,8-triaza-spiro[4.5]decane-2,4-dione 135004 8-(3,5-Bis-trifluoromethyl-benzoyl)-3-[2-(1H-indol-3-yl)-ethyl]-1,3,8-triaza-spiro[4.5]decane-2,4-dione 135136 1-(2-Chloro-2-phenyl-ethyl)-4-phenylamino-1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid ethyl ester 135172 8-(3,5-Bis-trifluoromethyl-benzoyl)-3-(4-methylsulfanyl-phenyl)-1,3,8-triaza-spiro[4.5]decane-2,4-dione 135176 ethyl 1-(2-chloro-2-phenylethyl)-4-(phenethylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 135206 1-(3,5-Bis-trifluoromethyl-benzyl)-8-(2-fluoro-benzoyl)-3-methyl-1,3,8-triaza-spiro[4.5]decane-2,4-dione 135241 3-Biphenyl-3-ylmethyl-8-(3,5-bis-trifluoromethyl-benzoyl)-1,3,8-triaza-spiro[4.5]decane-2,4-dione 135342 4-Nitro-benzoic acid 8-aza-bicyclo[3.2.1]oct-6-yl ester 135426 Cyclohexanecarboxylic acid 8-aza-bicyclo[3.2.1]oct-6-yl ester 135547 Propionic acid 8-methyl-8-aza-bicyclo[3.2.1]oct-6-yl ester 135599 Propionic acid 8-aza-bicyclo[3.2.1]oct-6-yl ester 135617 1-(3,5-Bis-trifluoromethyl-benzyl)-8-{2-[3-(3,4-dimethoxy-phenyl)-4-oxo-imidazolidin-1-yl]-acetyl}-3-methyl-1,3,8-triaza-spiro[4.5]decane-2,4-dione 135629 4-tert-Butylamino-1-(2-chloro-2-phenyl-ethyl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid ethyl ester 135645 1-(3,5-Bis-trifluoromethyl-benzyl)-8-(2,6-dichloro-benzoyl)-3-methyl-1,3,8-triaza-spiro[4.5]decane-2,4-dione 135646 8-[2-(4-Benzyl-piperidin-1-yl)-acetyl]-1-(3,5-bis-trifluoromethyl-benzyl)-3-methyl-1,3,8-triaza-spiro[4.5]decane-2,4-dione 135658 ethyl 1-(2-chloro-2-phenylethyl)-4-(pyrrolidin-1-yl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 135660 4-Butylamino-1-(2-chloro-2-phenyl-ethyl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid ethyl ester 135743 Benzoic acid 8-methyl-8-aza-bicyclo[3.2.1]oct-6-yl ester 135812 Carbonic acid 8-methyl-8-aza-bicyclo[3.2.1]oct-6-yl ester 2,2,2-trichloro-ethyl ester 135813 Cyclohexanecarboxylic acid 8-methyl-8-aza-bicyclo[3.2.1]oct-6-yl ester 136142 4-[4-(4-Fluoro-benzoyl)-piperidin-1-yl]-1-(4-fluoro-phenyl)-butan-1-one 136188 1-Phenyl-4-((S)-2-phenyl-4,5-dihydro-oxazol-4-ylmethyl)-piperazine 136305 16-Chloro-17,19-dihydroxy-4-methyl-3,7-dioxa-tricyclo[13.4.0.0*6,8*]nonadeca-1(19),9,11,15,17-pentaene-2,13-dione 13-{O-[2-(4-methyl-piperazin-1-yl)-2-oxo-ethyl]-oxime} 136423 2-(4-{3-[4-(3-Chloro-phenyl)-piperazin-1-yl]-propoxy}-phenyl)-1H-benzoimidazole 136425 2-(4-{3-[4-(4-Methoxy-phenyl)-piperazin-1-yl]-propoxy}-phenyl)-1H-benzoimidazole 136454 2-(4-{3-[4-(2-Chloro-phenyl)-piperazin-1-yl]-propoxy}-phenyl)-1H-benzoimidazole 136493 2a-[4-(6,7-Dihydro-4H-thieno[3,2-c]pyridin-5-yl)-butyl]-1-ethyl-2a,3,4,5-tetrahydro-1H-benzo[cd]indol-2-one 136494 2a-[4-(1,4,6,7-Tetrahydro-pyrazolo[4,3-c]pyridin-5-yl)-butyl]-2a,3,4,5-tetrahydro-1H-benzo[cd]indol-2-one 136495 2a-[4-(6,7-Dihydro-4H-furo[3,2-c]pyridin-5-yl)-butyl]-2a,3,4,5-tetrahydro-1H-benzo[cd]indol-2-one 136496 2a-[5-(3,4-Dihydro-1H-isoquinolin-2-yl)-pentyl]-2a,3,4,5-tetrahydro-1H-benzo[cd]indol-2-one 136528 N-(2-chloro-6-methylphenyl)-7-methoxyimidazo[1,5-a]quinoxalin-4-amine 136586 N-(2-chloro-6-methylphenyl)-7,8-dimethoxyimidazo[1,5-a]quinoxalin-4-amine 136587 N-(2,6-dimethylphenyl)-7,8-dimethoxyimidazo[1,5-a]quinoxalin-4-amine 136746 1-Phenyl-4-((S)-2-phenyl-4,5-dihydro-thiazol-4-ylmethyl)-piperazine 136757 1-[(S)-2-(5-Bromo-2-methoxy-phenyl)-4,5-dihydro-oxazol-4-ylmethyl]-4-phenyl-piperazine 136759 1-((4S,5S)-5-Methyl-2-phenyl-4,5-dihydro-oxazol-4-ylmethyl)-4-phenyl-piperazine 136761 1-[(4S,5R)-2-(5-Bromo-2-methoxy-phenyl)-5-methyl-4,5-dihydro-oxazol-4-ylmethyl]-4-phenyl-piperazine 136808 N-(2-chloro-6-methylphenyl)-8-methoxyimidazo[1,5-a]quinoxalin-4-amine 136809 N-(2-chloro-6-methylphenyl)-7-morpholinoimidazo[1,5-a]quinoxalin-4-amine 136877 N4-(2-chloro-6-methylphenyl)-N7,N7-diethylimidazo[1,5-a]quinoxaline-4,7-diamine 136906 2-{4-[3-(4-Methyl-piperazin-1-yl)-propoxy]-phenyl}-1H-benzoimidazole 136911 2-(4-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propoxy}-phenyl)-1H-benzoimidazole 136952 2a-[3-(3,4-Dihydro-1H-isoquinolin-2-yl)-propyl]-2a,3,4,5-tetrahydro-1H-benzo[cd]indol-2-one 136953 2a-[4-(6,7-Dihydro-4H-thieno[3,2-c]pyridin-5-yl)-butyl]-2a,3,4,5-tetrahydro-1H-benzo[cd]indol-2-one 136955 2a-[4-(3,4,6,7-Tetrahydro-imidazo[4,5-c]pyridin-5-yl)-butyl]-2a,3,4,5-tetrahydro-1H-benzo[cd]indol-2-one 136960 7-bromo-N-(2-chloro-6-methylphenyl)imidazo[1,5-a]quinoxalin-4-amine 136966 4-(2-chloro-6-methylphenylamino)imidazo[1,5-a]quinoxaline-7-carboxamide 136984 2a-[4-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-butyl]-1-methyl-2a,3,4,5-tetrahydro-1H-benzo[cd]indol-2-one 137019 N-(4-(2-chloro-6-methylphenylamino)imidazo[1,5-a]quinoxalin-7-yl)acetamide 137020 N4-(2-chloro-6-methylphenyl)imidazo[1,5-a]quinoxaline-4,7-diamine 137065 N-(2-chloro-6-methylphenyl)-6-methoxyimidazo[1,5-a]quinoxalin-4-amine 137074 2-(4-{3-[4-(4-Chloro-phenyl)-piperazin-1-yl]-propoxy}-phenyl)-1H-benzoimidazole 137080 2-{4-[3-(4-Pyrimidin-2-yl-piperazin-1-yl)-propoxy]-phenyl}-1H-benzoimidazole 137110 2-{4-[3-(4-Pyridin-2-yl-piperazin-1-yl)-propoxy]-phenyl}-1H-benzoimidazole 137111 2-(4-{3-[4-(2-Propylsulfanyl-phenyl)-piperazin-1-yl]-propoxy}-phenyl)-1H-benzoimidazole 137213 2a-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-butyl]-2a,3,4,5-tetrahydro-1H-benzo[cd]indol-2-one 137398 trans-N-[4-[2-(6-cyano-1,2,3,4-tetrahydroisoquinolin-2yl)-ethyl]cyclo-hexyl]-4-quinolinecarboxamide 137403 2-{4-[3-(4-Phenyl-piperazin-1-yl)-propoxy]-phenyl}-1H-benzoimidazole 137534 2-(furan-2-yl)-8-isopentyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine 138030 (1S,3R)-1-(aminomethyl)-3-phenyl-3,4-dihydro-1H-2-benzopyran-5,6-diol 138558 7-Chloro-2-cyclopentyl-10-(4-methyl-piperazin-1-yl)-2,4-dihydro-2,3,4,9-tetraaza-benzo[f]azulene 138560 2-[2-(1H-Imidazol-4-yl)-ethylsulfanyl]-5-(3-propoxy-phenyl)-1H-imidazole 138592 2,5-Dibutyl-4-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-[1,2,4]triazolidin-3-one 138594 4-((1S,2R)-2-(4-hydroxyphenethylamino)-1-hydroxypropyl)phenol 138595 7-Chloro-2-isobutyl-10-(4-methyl-piperazin-1-yl)-2,4-dihydro-2,3,4,9-tetraaza-benzo[f]azulene 138631 7-Chloro-2-ethyl-10-(4-methyl-piperazin-1-yl)-2,4-dihydro-2,3,4,9-tetraaza-benzo[f]azulene 138633 3-[2-(N',N''-Dicyclohexyl-guanidino)-3-naphthalen-2-yl-propionylamino]-1-azonia-bicyclo[2.2.2]octane dihydrochloride (diastereomeric mixture) 138636 [8-(Naphthalen-1-ylmethoxy)-11-oxo-5-propyl-5,11-dihydro-dibenzo[b,e][1,4]diazepin-10-yl]-acetic acid 138638 SID11114127 138726 7-Chloro-2-methyl-10-(4-methyl-piperazin-1-yl)-2,4-dihydro-2,3,4,9-tetraaza-benzo[f]azulene 138806 2-((3R,6S,9R,12S,17aS)-9-((1H-indol-3-yl)methyl)-6-isobutyl-3-isopropyl-1,4,7,10,13-pentaoxohexadecahydro-1H-pyrrolo[1,2-a][1,4,7,10,13]pentaazacyclopentadecin-12-yl)acetic acid 139011 {8-[(1H-Indole-2-carbonyl)-amino]-11-oxo-5-propyl-5,11-dihydro-dibenzo[b,e][1,4]diazepin-10-yl}-acetic acid 139043 4-{2-[2-(1H-Imidazol-4-yl)-ethylsulfanyl]-3H-imidazol-4-yl}-benzamide 139079 3-{2-[2-(1H-Imidazol-4-yl)-ethylsulfanyl]-3H-imidazol-4-yl}-benzamide 139126 1-{2-[4-(4-Fluoro-benzoyl)-piperidin-1-yl]-ethyl}-6-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-1,4-dihydro-benzo[d][1,3]oxazin-2-one 139127 2-Benzyl-7-fluoro-10-(4-methyl-piperazin-1-yl)-2,4-dihydro-2,3,4,9-tetraaza-benzo[f]azulene 139128 7-Fluoro-2-methyl-10-(4-methyl-piperazin-1-yl)-1-phenyl-2,4-dihydro-2,3,4,9-tetraaza-benzo[f]azulene 139131 2-[2-(1H-Imidazol-4-yl)-ethylsulfanyl]-5-phenyl-1H-imidazole 139138 5-(4-Chloro-phenyl)-2-[2-(1H-imidazol-4-yl)-ethylsulfanyl]-1H-imidazole 139156 1-{2-[4-(4-Fluoro-benzoyl)-piperidin-1-yl]-ethyl}-6-(4-morpholin-4-yl-butyl)-1,4-dihydro-benzo[d][1,3]oxazin-2-one 139158 3-{2-[4-(4-Fluoro-benzoyl)-piperidin-1-yl]-ethyl}-6-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-3H-benzothiazol-2-one 139159 3-{2-[4-(4-Fluoro-benzoyl)-piperidin-1-yl]-ethyl}-6-{2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-3H-benzothiazol-2-one 139162 [8-(2-1H-Indol-3-yl-acetylamino)-11-oxo-5-propyl-5,11-dihydro-dibenzo[b,e][1,4]diazepin-10-yl]-acetic acid 139201 {8-[(1H-Indole-3-carbonyl)-amino]-11-oxo-5-propyl-5,11-dihydro-dibenzo[b,e][1,4]diazepin-10-yl}-acetic acid 139213 5-(4-Butoxy-phenyl)-2-[2-(1H-imidazol-4-yl)-ethylsulfanyl]-1H-imidazole 139236 6,7-Difluoro-2-methyl-10-(4-methyl-piperazin-1-yl)-2,4-dihydro-2,3,4,9-tetraaza-benzo[f]azulene 139239 (4-{2-[2-(1H-Imidazol-4-yl)-ethylsulfanyl]-3H-imidazol-4-yl}-phenyl)-dimethyl-amine 139246 2-Ethyl-7-fluoro-10-(4-methyl-piperazin-1-yl)-2,4-dihydro-2,3,4,9-tetraaza-benzo[f]azulene 139271 2-[2-(1H-Imidazol-4-yl)-ethylsulfanyl]-5-(3-nitro-phenyl)-1H-imidazole 139272 5-(3-Bromo-phenyl)-2-[2-(1H-imidazol-4-yl)-ethylsulfanyl]-1H-imidazole 139273 7-Fluoro-2-methyl-10-(4-methyl-piperazin-1-yl)-2,4-dihydro-2,3,4,9-tetraaza-benzo[f]azulene 139274 Benzenesulfonic acid 4-{2-[2-(1H-imidazol-4-yl)-ethylsulfanyl]-3H-imidazol-4-yl}-phenyl ester 139282 (8-Benzyloxy-11-oxo-5,11-dihydro-dibenzo[b,e][1,4]diazepin-10-yl)-acetic acid 139323 2-amino-4-(4-((5,7-dimethyl-2-propyl-3H-imidazo[4,5-b]pyridin-3-yl)methyl)phenyl)quinoline-3-carboxylic acid 139338 [8-(Naphthalen-1-ylmethoxy)-11-oxo-5,11-dihydro-dibenzo[b,e][1,4]diazepin-10-yl]-acetic acid 139345 1-{(5S,8S)-3-Butyl-5-[2'-(2H-tetrazol-5-yl)-biphenyl-4-yl]-5,6,7,8-tetrahydro-imidazo[1,5-a]pyridin-8-yl}-pyrrolidine-2,5-dione 139361 6-Fluoro-2-methyl-10-(4-methyl-piperazin-1-yl)-2,4-dihydro-2,3,4,9-tetraaza-benzo[f]azulene 139362 7-Fluoro-1,2-dimethyl-10-(4-methyl-piperazin-1-yl)-2,4-dihydro-2,3,4,9-tetraaza-benzo[f]azulene 139371 {8-[(Naphthalene-1-carbonyl)-amino]-11-oxo-5-propyl-5,11-dihydro-dibenzo[b,e][1,4]diazepin-10-yl}-acetic acid 139374 2-[2-(1H-Imidazol-4-yl)-ethylsulfanyl]-5-(4-propyl-phenyl)-1H-imidazole 139378 1,3-Dibutyl-5-[2'-(2H-tetrazol-5-yl)-biphenyl-4-yl]-5,6-dihydro-imidazo[1,5-a]pyridine 139400 {8-[(Naphthalen-1-ylmethyl)-amino]-11-oxo-5-propyl-5,11-dihydro-dibenzo[b,e][1,4]diazepin-10-yl}-acetic acid 139401 2-[2-(1H-Imidazol-4-yl)-ethylsulfanyl]-5-(4-nitro-phenyl)-1H-imidazole 139435 [8-(1H-Indol-3-ylmethyl)-11-oxo-5-propyl-5,11-dihydro-dibenzo[b,e][1,4]diazepin-10-yl]-acetic acid 139447 N-Methyl-N-((S)-1-phenyl-2-pyrrolidin-1-yl-ethyl)-2-(4-trifluoromethyl-phenyl)-acetamide 139449 SID26757055 139472 3-{2-[4-(4-Fluoro-benzoyl)-piperidin-1-yl]-ethyl}-6-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]-propyl}-3H-benzothiazol-2-one 139473 3-{2-[4-(4-Fluoro-benzoyl)-piperidin-1-yl]-ethyl}-6-{4-[4-(3-trifluoromethyl-phenyl)-piperazin-1-yl]-butyl}-3H-benzothiazol-2-one 139573 4-(4-((2-ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridin-3-yl)methyl)phenyl)-3-(2H-tetrazol-5-yl)quinoline 139598 3-(2-{4-[Bis-(4-fluoro-phenyl)-methylene]-piperidin-1-yl}-ethyl)-6-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-3H-benzooxazol-2-one 139655 (E)-N-(4-amino-2-methylquinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)acrylamide 139705 1-(2-{4-[Bis-(4-fluoro-phenyl)-methylene]-piperidin-1-yl}-ethyl)-6-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-1,4-dihydro-benzo[d][1,3]oxazin-2-one 139706 3-(2-{4-[Bis-(4-fluoro-phenyl)-methylene]-piperidin-1-yl}-ethyl)-6-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-3H-benzothiazol-2-one 139707 3-{2-[4-(4-Fluoro-benzoyl)-piperidin-1-yl]-ethyl}-6-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-3H-benzooxazol-2-one 139726 N-{(S)-2-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1H-indol-3-yl)-2-methyl-propionylamino]-1-phenyl-ethyl}-succinamic acid 139765 3-{2-[4-(4-Fluoro-benzoyl)-piperidin-1-yl]-ethyl}-6-(4-morpholin-4-yl-butyl)-3H-benzothiazol-2-one 139851 3-Butyl-5-[2'-(2H-tetrazol-5-yl)-biphenyl-4-yl]-5,6-dihydro-imidazo[1,5-a]pyridine 139891 4-(4-((5,7-dimethyl-2-propyl-3H-imidazo[4,5-b]pyridin-3-yl)methyl)phenyl)-2-methylquinoline-3-carboxylic acid 139914 1-[2-((S)-4-Phenyl-cyclohex-3-enyl)-ethyl]-4-pyridin-2-yl-piperazine 139928 3-Benzylsulfanyl-4-oxo-4,5,6,7-tetrahydro-benzo[c]thiophene-1-carboxylic acid ethyl ester 139993 5-[4'-(2,4-Dibutyl-imidazol-1-ylmethyl)-biphenyl-2-yl]-2H-tetrazole 139994 1-{(5S,8S)-3-Butyl-1-chloro-5-[2'-(2H-tetrazol-5-yl)-biphenyl-4-yl]-5,6,7,8-tetrahydro-imidazo[1,5-a]pyridin-8-yl}-pyrrolidine-2,5-dione 140374 3-[2-(2-Acetylamino-3-biphenyl-4-yl-propionylamino)-4-methyl-pentanoylamino]-N-(1-{1-[1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 140379 3-[2-(2-Acetylamino-3-naphthalen-2-yl-propionylamino)-4-methyl-pentanoylamino]-N-(1-{1-[1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 140400 (S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-4-methyl-pentanoylamino]-N-{(S)-1-[(S)-(S)-1-((S)-1-carboxy-2-(S)-1H-indol-3-yl-ethylcarbamoyl)-2-methyl-butylcarbamoyl]-2-methyl-butyl}-succinamic acid 140401 3-{2-[2-Acetylamino-3-(4-hydroxy-phenyl)-propionylamino]-4-methyl-pentanoylamino}-N-(1-{1-[1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 140404 3-((R)-2-Acetylamino-3-phenyl-propionylamino)-N-{(S)-1-[(S)-1-((S)-(S)-1-carboxy-2-(S)-1H-indol-3-yl-ethylcarbamoyl)-2-methyl-butylcarbamoyl]-2-methyl-butyl}-succinamic acid 140434 2-Butyl-5-propyl-4-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-2,4-dihydro-pyrazol-3-one 140470 (S)-2-[(S)-2-((2S,5S)-2-{(S)-2-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-4-methyl-pentanoylamino]-3-phenyl-propionylamino}-3-methyl-pentanoylamino)-3-methyl-pentanoylamino]-3-(S)-1H-indol-3-yl-propionic acid 140510 (S)-3-[(S)-2-((S)-2-Acetylamino-3-phenyl-propionylamino)-4-methyl-pentanoylamino]-N-{(S)-1-[(S)-(S)-1-((S)-1-carboxy-2-(S)-1H-indol-3-yl-ethylcarbamoyl)-2-methyl-butylcarbamoyl]-2-methyl-butyl}-succinamic acid 140555 2-Butyl-8-propyl-5-[2'-(2H-tetrazol-5-yl)-biphenyl-4-yl]-5,6,7,8-tetrahydro-2H-[1,2,4]triazolo[4,3-a]pyridin-3-one 140760 (S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-3-phenyl-propionylamino]-N-{(S)-1-[(S)-(S)-1-((S)-1-carboxy-2-(S)-1H-indol-3-yl-ethylcarbamoyl)-2-methyl-butylcarbamoyl]-2-methyl-butyl}-succinamic acid 140909 [2-(1H-Benzoimidazol-4-yloxy)-ethyl]-benzyl-amine 141006 Benzyl-[2-(1H-indazol-4-yloxy)-ethyl]-amine 141007 Benzyl-[2-(2-trifluoromethyl-1H-benzoimidazol-4-yloxy)-ethyl]-amine 141037 Benzyl-[2-(6-chloro-2-trifluoromethyl-1H-benzoimidazol-4-yloxy)-ethyl]-amine 141038 2-Butyl-5-propyl-4-[1-[2'-(2H-tetrazol-5-yl)-biphenyl-4-yl]-meth-(Z)-ylidene]-2,4-dihydro-pyrazol-3-one 141043 Benzyl-[2-(2-methyl-1H-benzoimidazol-4-yloxy)-ethyl]-amine 141118 3-(4-methyl-2-((2-oxoindolin-3-ylidene)methyl)-1H-pyrrol-3-yl)propanoic acid 141202 ((2R,3S)-2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2-methoxy-benzyl)-amine 141205 SID26753276 141398 4-[(E)-2-(4-Amino-phenyl)-vinyl]-2-methyl-6-phenyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid diethyl ester 141438 7-Dipropylamino-5,6,7,8-tetrahydro-naphthalene-1-carboxylic acid methyl ester 141464 ((S)-8-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-dipropyl-ammonium 141478 7-Dipropylamino-5,6,7,8-tetrahydro-naphthalene-1-carboxylic acid methyl ester 141479 (R)-1-(7-Dipropylamino-5,6,7,8-tetrahydro-naphthalen-1-yl)-ethanone 141567 2-Methyl-6-phenyl-4-phenylethynyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid 5-benzyl ester 3-ethyl ester 141620 ((R)-8-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-dipropyl-amine 141724 4-(2-Benzylamino-ethoxy)-1,3-dihydro-benzoimidazol-2-one 141749 2-Methyl-6-phenyl-4-phenylethynyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid 3-ethyl ester 5-(4-nitro-benzyl) ester 141812 1H-Indole-2-carboxylic acid (4-{4-amino-1-[4-(4-methyl-piperazin-1-yl)-cyclohexyl]-1H-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxy-phenyl)-amide 141813 1-Methyl-1H-indole-2-carboxylic acid (4-{4-amino-1-[4-(4-methyl-piperazin-1-yl)-cyclohexyl]-1H-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxy-phenyl)-amide 141848 2-Methyl-6-phenyl-4-phenylethynyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid 3-benzyl ester 5-ethyl ester 141853 4-(2-Benzylamino-ethoxy)-1,3-dihydro-benzoimidazole-2-thione 141854 4-(2-Benzylamino-ethoxy)-6-chloro-1,3-dihydro-benzoimidazol-2-one 141886 4-(2-Benzylamino-ethoxy)-6-chloro-1,3-dihydro-benzoimidazole-2-thione 141982 2-Methyl-6-phenyl-4-phenylethynyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid diethyl ester 142025 3-{4-[(Furan-2-ylmethyl)-amino]-3-methoxy-phenyl}-1-[4-(4-methyl-piperazin-1-yl)-cyclohexyl]-1H-pyrazolo[3,4-d]pyrimidin-4-ylamine 142047 2-Methyl-6-phenyl-4-((E)-styryl)-1,4-dihydro-pyridine-3,5-dicarboxylic acid diethyl ester 142088 Trifluoro-methanesulfonic acid 7-dipropylamino-5,6,7,8-tetrahydro-naphthalen-1-yl ester 142091 Dipropyl-(1,2,3,4-tetrahydro-naphthalen-2-yl)-amine 142092 (S)-(8-Methyl-1,2,3,4-tetrahydro-naphthalen-2-yl)-dipropyl-amine 142093 (S)-(8-Phenyl-1,2,3,4-tetrahydro-naphthalen-2-yl)-dipropyl-amine 142141 Trifluoro-methanesulfonic acid 7-dipropylamino-5,6,7,8-tetrahydro-naphthalen-1-yl ester 142176 (S)-1-(7-Dipropylamino-5,6,7,8-tetrahydro-naphthalen-1-yl)-ethanone 142177 (R)-(8-Phenyl-1,2,3,4-tetrahydro-naphthalen-2-yl)-dipropyl-amine 142178 (R)-(8-Methyl-1,2,3,4-tetrahydro-naphthalen-2-yl)-dipropyl-amine 142294 SID11113966 142298 3,6-Dichloro-2-(2-isopropoxy-4-methyl-phenyl)-chromen-4-one 142325 5-Amino-3-(4-methoxy-phenyl)-thiazolo[3,2-a]pyrimidin-7-one 142710 Dipropyl-(1,2,3,4-tetrahydro-naphthalen-2-yl)-amine 142732 3-Pyridin-4-yl-quinoline-6,7-diol 142879 7-Chloro-3-(3,5-dimethyl-phenyl)-4-[2-(1-methyl-piperidin-2-yl)-ethoxy]-6-nitro-1H-quinolin-2-one 143025 7-Chloro-3-(3,5-dimethyl-phenyl)-6-nitro-4-((R)-2-pyrrolidin-2-yl-ethoxy)-1H-quinolin-2-one 143052 7-Chloro-3-(3,5-dimethyl-phenyl)-4-[2-((R)-1-methyl-piperidin-2-yl)-ethoxy]-6-nitro-1H-quinolin-2-one 143053 7-Chloro-3-(3,5-dimethyl-phenyl)-6-nitro-4-((R)-2-piperidin-2-yl-ethoxy)-1H-quinolin-2-one 143059 1,3,8-Trimethyl-3,7-dihydro-purine-2,6-dione 143071 7-Chloro-3-(3,5-dimethyl-phenyl)-6-nitro-4-(3-piperidin-2-yl-propoxy)-1H-quinolin-2-one 143072 4-(2-Azepan-2-yl-ethoxy)-7-chloro-3-(3,5-dimethyl-phenyl)-6-nitro-1H-quinolin-2-one 143119 7-Chloro-3-(3,5-dimethyl-phenyl)-6-nitro-4-(piperidin-3-ylmethoxy)-1H-quinolin-2-one 143146 4-((S)-2-Azetidin-2-yl-ethoxy)-7-chloro-3-(3,5-dimethyl-phenyl)-6-nitro-1H-quinolin-2-one 143154 7-Chloro-3-(3,5-dimethyl-phenyl)-4-[2-((S)-1-methyl-piperidin-2-yl)-ethoxy]-6-nitro-1H-quinolin-2-one 143178 7-Chloro-3-(3,5-dimethyl-phenyl)-6-nitro-4-((S)-2-pyrrolidin-2-yl-ethoxy)-1H-quinolin-2-one 143411 5'-methyl-1-(1-methyl-1-perhydro-2-naphthalenylethyl)-2'-phenylspiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole] 143412 1-(1-cyclodecyl-1-methylethyl)-5'-methyl-2'-phenylspiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole] 143449 1-(1-cyclononyl-1-methylethyl)-5'-methyl-2'-phenylspiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole] 143544 (E)-3-[6-(2,6-Dichloro-phenylsulfanylmethyl)-3-phenethyloxy-pyridin-2-yl]-acrylic acid 143594 3-(3,5-Bis-trifluoromethyl-phenyl)-N-(4-fluoro-phenyl)-N-piperidin-4-yl-propionamide 143762 N-(3,4-Dichloro-phenyl)-2-(3,5-dimethyl-phenoxy)-N-piperidin-4-yl-acetamide 144016 2-[3-(1-Benzyl-1H-indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-benzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxy-phenyl)-acetamide 144018 9-Benzyl-6-(3-guanidino-propyl)-12-(3H-imidazol-4-ylmethyl)-3-(1H-indol-3-ylmethyl)-2,5,8,11,14,17-hexaoxo-1,4,7,10,13,18hexaaza-cyclotricosane-23-carboxylic acid amide 144188 8-(3-Guanidino-propyl)-2-(3H-imidazol-4-ylmethyl)-11-(1H-indol-3-ylmethyl)-5-naphthalen-2-ylmethyl-3,6,9,12,20,24-hexaoxo-1,4,7,10,13,19hexaaza-cyclotetracosane-14-carboxylic acid amide 144189 5-Benzyl-8-(3-guanidino-propyl)-2-(3H-imidazol-4-ylmethyl)-11-(1H-indol-3-ylmethyl)-3,6,9,12,20,24-hexaoxo-1,4,7,10,13,19hexaaza-cyclotetracosane-14-carboxylic acid amide 144423 3-{7-[3-(2-Cyclopropylmethyl-3-methoxy-4-methylcarbamoyl-phenoxy)-propoxy]-8-propyl-chroman-2-yl}-propionic acid 144473 (O)C-(C6H4)-C(O)-c[His-D-Nal(2')-Arg-Trp-Lys]-NH2) (MK-7) 144572 N-Isopropyl-N-(4-methoxy-phenyl)-2-[3-(1-methyl-1H-indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-benzo[b][1,4]diazepin-1-yl]-acetamide 144618 2-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-benzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-phenyl-acetamide 144619 2-[3-(1H-Indol-3-ylmethyl)-3-methyl-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-benzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-phenyl-acetamide 144620 2-[3-(1H-Indol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-benzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxy-phenyl)-acetamide 144621 2-[3-(1H-Indazol-3-ylmethyl)-3-methyl-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-benzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-phenyl-acetamide 144623 (2R,3R,4S,5R)-2-[2-Chloro-6-(4-phenylsulfanyl-piperidin-1-ylamino)-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 144624 2-[2-Chloro-6-(1-methyl-2-phenyl-ethylamino)-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 144632 2-[2-Chloro-6-(1-methyl-2-phenyl-ethylamino)-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 144657 2-[3-(1H-Indol-3-ylmethyl)-3-methyl-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-benzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxy-phenyl)-acetamide 144841 (2R,3R,4S,5R)-2-[2-Chloro-6-(piperidin-1-ylamino)-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 144848 18-benzylaminomethyl-(18S)-17-oxa-4,14,21-triazahexacyclo[19.6.1.17,14.02,6.08,13.022,27]nonacosa-1(28),2(6),7(29),8(13),9,11,22(27),23,25-nonaene-3,5-dione 144873 N-[1-(1-{1-[1-(5-Amino-1-carbamoyl-pentylcarbamoyl)-2-(1H-indol-3-yl)-ethylcarbamoyl]-4-guanidino-butylcarbamoyl}-2-phenyl-ethylcarbamoyl)-2-(3H-imidazol-4-yl)-ethyl]-succinamic acid 144921 18-(4-methylhexahydro-1-pyrazinylmethyl)-(18S)-17-oxa-4,14,21-triazahexacyclo[19.6.1.17,14.02,6.08,13.022,27]nonacosa-1(28),2(6),7(29),8(13),9,11,22(27),23,25-nonaene-3,5-dione 144925 9-Benzyl-12-(3H-imidazol-4-ylmethyl)-3-(1H-indol-3-ylmethyl)-6-methyl-2,5,8,11,14,17-hexaoxo-1,4,7,10,13,18hexaaza-cyclotricosane-23-carboxylic acid amide 144926 9-Benzyl-6-(3-guanidino-propyl)-3-(1H-indol-3-ylmethyl)-12-methyl-2,5,8,11,14,17-hexaoxo-1,4,7,10,13,18hexaaza-cyclotricosane-23-carboxylic acid amide 144940 2-amino-2-(4-octylphenethyl)propane-1,3-diol 144959 LY-333531 144981 (O)C-(C6H4)-C(O)-c[His-D-Phe-Arg-Trp-Lys]-NH2) (MK-6) 144982 6-(3-Guanidino-propyl)-12-(3H-imidazol-4-ylmethyl)-3-(1H-indol-3-ylmethyl)-9-naphthalen-2-ylmethyl-2,5,8,11,14,17-hexaoxo-1,4,7,10,13,18hexaaza-cyclotricosane-23-carboxylic acid amide 145186 18-tetrahydro-1H-1-pyrrolylmethyl-(18S)-17-oxa-4,14,21-triazahexacyclo[19.6.1.17,14.02,6.08,13.022,27]nonacosa-1(28),2(6),7(29),8(13),9,11,22(27),23,25-nonaene-3,5-dione 145209 (2R,3S)-methyl 3-(bis(4-fluorophenyl)methoxy)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate 145223 (R)-2-(4-Fluoro-phenyl)-2-{1-[2-fluoro-3-(5-[1,2,4]triazol-4-yl-1H-indol-3-yl)-propyl]-piperidin-4-ylamino}-ethanol 145287 2-[2-Chloro-6-(morpholin-4-ylamino)-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 145391 3,5-dioxo-17-phenylsulfonamidomethyl-(17S)-18-oxa-4,14,21-triazahexacyclo[19.6.1.17,14.02,6.08,13.022,27]nonacosa-1(28),2(6),7(29),8(13),9,11,22(27),23,25-nonaene 145394 18-aminomethyl-(18S)-17-oxa-4,14,21-triazahexacyclo[19.6.1.17,14.02,6.08,13.022,27]nonacosa-1(28),2(6),7(29),8(13),9,11,22(27),23,25-nonaene-3,5-dione 145429 18-(1,4-oxazinan-4-ylmethyl)-(18S)-17-oxa-4,14,21-triazahexacyclo[19.6.1.17,14.02,6.08,13.022,27]nonacosa-1(28),2(6),7(29),8(13),9,11,22(27),23,25-nonaene-3,5-dione 145502 (R)-2-(4-Fluoro-phenyl)-2-{1-[3-(5-[1,2,4]triazol-4-yl-1H-indol-3-yl)-propyl]-piperidin-4-ylamino}-ethanol 145532 Benzyl-{(3R,4S)-3-fluoro-1-[3-(5-[1,2,4]triazol-4-yl-1H-indol-3-yl)-propyl]-piperidin-4-yl}-methyl-amine 145610 18-methylaminomethyl-(18S)-17-oxa-4,14,21-triazahexacyclo[19.6.1.17,14.02,6.08,13.022,27]nonacosa-1(28),2(6),7(29),8(13),9,11,22(27),23,25-nonaene-3,5-dione 145660 Benzyl-{(3S,4R)-3-fluoro-1-[3-(5-[1,2,4]triazol-4-yl-1H-indol-3-yl)-propyl]-piperidin-4-yl}-methyl-amine 145976 SID26752006 146092 4-(4-Benzyl-piperazin-1-yl)-1H-benzoimidazole 146093 4-(4-Benzyl-piperazin-1-yl)-2-trifluoromethyl-1H-benzoimidazole 146114 SID11111937 146128 4-(4-Benzyl-piperazin-1-yl)-5-chloro-1,3-dihydro-indol-2-one 146366 1-Methyl-4-(5-methylene-5H-dibenzo[a,d]cyclohepten-10-yl)-piperazine 146404 1-(2-Chloro-5-isopropylidene-5H-dibenzo[a,d]cyclohepten-10-yl)-4-methyl-piperazine 146413 1-(5-Isopropylidene-5H-dibenzo[a,d]cyclohepten-10-yl)-4-methyl-piperazine 146597 4-(4-Benzyl-piperazin-1-yl)-1,3-dihydro-indol-2-one 146638 1-benzyl-4-(3-hydroxyphenyl)piperazine 146648 4-(4-Benzyl-piperazin-1-yl)-7-bromo-1H-indole 146649 4-(4-Benzyl-piperazin-1-yl)-1H-indole 146683 4-(4-Benzyl-piperazin-1-yl)-1,3-dihydro-benzoimidazol-2-one 146684 4-(4-Benzyl-piperazin-1-yl)-5-chloro-1H-indole 146922 2-Phenyl-3-(2-piperidin-1-yl-ethyl)-1H-indole 146971 4-[5-(4-Chloro-phenyl)-3-(4-fluoro-phenyl)-1H-pyrrol-2-yl]-pyridine 147078 7-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-pyrazolo[1,5-a]pyridine 147331 3-[1-(8-Phenethyl-8-aza-bicyclo[3.2.1]oct-3-yl)-piperidin-4-yl]-2-phenyl-1H-indole 147412 1-{2-[4-(2-Phenyl-1H-indol-3-yl)-piperidin-1-yl]-ethyl}-imidazolidin-2-one 147444 3-(1-Methyl-piperidin-4-yl)-2-phenyl-1H-indole 147525 3-(1-Benzyl-piperidin-4-yl)-2-phenyl-1H-indole 147620 (4,5-Dihydro-1H-imidazol-2-yl)-(4'-methoxy-2-methyl-biphenyl-3-yl)-amine 147687 3-{6-((E)-2-Carboxy-vinyl)-5-[8-(4-methoxy-phenyl)-octyloxy]-pyridin-2-ylmethylsulfanylmethyl}-benzoic acid 147709 (2-Chloro-9-methyl-9H-purin-6-yl)-cyclopentyl-amine 147769 Rupatadine 147828 (4,5-Dihydro-1H-imidazol-2-yl)-(2,3'-dimethyl-biphenyl-3-yl)-amine 147863 SID11111196 148088 (4,5-Dihydro-1H-imidazol-2-yl)-(3'-fluoro-2-methyl-biphenyl-3-yl)-amine 148187 (4,5-Dihydro-1H-imidazol-2-yl)-(2-methyl-3'-trifluoromethyl-biphenyl-3-yl)-amine 148188 (3'-Chloro-2-methyl-biphenyl-3-yl)-(4,5-dihydro-1H-imidazol-2-yl)-amine 148243 (4,5-Dihydro-1H-imidazol-2-yl)-(2-methyl-biphenyl-3-yl)-amine 148252 (4,5-Dihydro-1H-imidazol-2-yl)-(3'-isopropyl-2-methyl-biphenyl-3-yl)-amine 148253 (4,5-Dihydro-1H-imidazol-2-yl)-(2-methyl-3-pyridin-3-yl-phenyl)-amine 148303 (4,5-Dihydro-1H-imidazol-2-yl)-(2-methyl-3-thiophen-3-yl-phenyl)-amine 148305 (4,5-Dihydro-1H-imidazol-2-yl)-(2-methyl-3-thiophen-2-yl-phenyl)-amine 148333 (4,5-Dihydro-1H-imidazol-2-yl)-(3'-methoxy-2-methyl-biphenyl-3-yl)-amine 148343 (4,5-Dihydro-1H-imidazol-2-yl)-(2',4'-dimethoxy-2-methyl-biphenyl-3-yl)-amine 148371 (6,7-Dimethoxy-quinazolin-4-yl)-(3-methyl-benzyl)-amine 148375 N-(3-Chloro-4-fluoro-phenyl)-N'-(6,7-dimethoxy-quinazolin-4-yl)-hydrazine 148402 (3-Chloro-4-fluoro-phenyl)-(6,7-dimethoxy-quinazolin-4-yl)-diazene 148479 Acetic acid 7-methoxy-4-(2-phenyl-cyclopropylamino)-quinazolin-6-yl ester 148504 2-[1,4']Bipiperidinyl-1'-yl-1-[2-(4-chloro-phenoxymethyl)-1-((S)-3-piperidin-3-yl-propyl)-1H-indol-3-yl]-ethanone 148595 (3R,3aS)-7,8-Dimethoxy-3-[4-(3-naphthalen-2-yl-propyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-chromeno[4,3-c]isoxazole 148655 (3R,3aS)-7,8-Dimethoxy-3-[4-((E)-5-phenyl-pent-4-enyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-chromeno[4,3-c]isoxazole 148724 (3R,3aS)-7,8-Dimethoxy-3-[4-((E)-4-methyl-5-phenyl-pent-4-enyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-chromeno[4,3-c]isoxazole 148765 4-(1H-imidazol-4-yl)butan-1-amine 148812 2-(4-Chloro-phenoxymethyl)-1-methyl-3-piperidin-1-ylmethyl-1H-indole 148884 [7-Methoxy-6-(2-morpholin-4-yl-ethoxy)-quinazolin-4-yl]-(2-phenyl-cyclopropyl)-amine 148955 4-(5-Fluoro-indan-2-ylmethyl)-4,5-dihydro-1H-imidazole 148963 3-(2-Methoxy-5-trifluoromethoxy-phenyl)-6-phenyl-1-oxa-7-aza-spiro[4.5]dec-3-ene 148978 (6,7-Dimethoxy-quinazolin-4-yl)-indan-1-yl-amine 149025 (6,7-Dimethoxy-quinazolin-4-yl)-isoquinolin-3-yl-amine 149029 (6,7-Dimethoxy-quinazolin-4-yl)-(2-phenyl-cyclopropyl)-amine 149030 (6,7-Dimethoxy-quinazolin-4-yl)-isoquinolin-4-yl-amine 149046 (6,7-Dimethoxy-quinazolin-4-yl)-isoquinolin-1-yl-amine 149084 (3R,3aS)-7,8-Dimethoxy-3-[4-((E)-5-phenyl-hex-4-enyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-chromeno[4,3-c]isoxazole 149103 (R)-4-Propyl-3,4,4a,5,6,10b-hexahydro-2H-naphtho[1,2-b][1,4]oxazin-9-ol 149133 5-{3-[2-Methoxy-5-(5-trifluoromethyl-tetrazol-1-yl)-phenyl]-6-phenyl-1-oxa-7-aza-spiro[4.5]dec-7-ylmethyl}-2,4-dihydro-[1,2,4]triazol-3-one 149138 4-(2,3-Dihydro-indol-1-yl)-6,7-dimethoxy-quinazoline 149233 (E)-N-(4-(3-bromophenylamino)quinazolin-6-yl)-4-(dimethylamino)but-2-enamide 149244 3-(2-Methoxy-5-trifluoromethoxy-phenyl)-6-phenyl-7-(1H-[1,2,4]triazol-3-ylmethyl)-1-oxa-7-aza-spiro[4.5]decane 149291 3-(2-Methoxy-phenyl)-6-phenyl-1-oxa-7-aza-spiro[4.5]dec-3-ene 149303 7-(1H-Imidazol-4-ylmethyl)-3-[2-methoxy-5-(5-trifluoromethyl-tetrazol-1-yl)-phenyl]-6-phenyl-1-oxa-7-aza-spiro[4.5]decane 149340 [6-(3-Dimethylamino-propoxy)-7-methoxy-quinazolin-4-yl]-(2-phenyl-cyclopropyl)-amine 149385 3-[2-Methoxy-5-(5-trifluoromethyl-tetrazol-1-yl)-phenyl]-6-phenyl-1-oxa-7-aza-spiro[4.5]decane 149386 3-(2-Methoxy-phenyl)-6-phenyl-1-oxa-7-aza-spiro[4.5]decane 149820 N-(4-(3-bromophenylamino)quinazolin-6-yl)but-2-ynamide 149831 1-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-methoxyphenyl)urea 149856 1-(8-butyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-methoxyphenyl)urea 149920 2-(2-(methylsulfinyl)benzylthio)-5-(4-fluorophenyl)-4-(pyridin-4-yl)pyrimidine 150023 N-[3-Chloro-4-((S)-3,4,11,11a-tetrahydro-1H,5H-2-oxa-4a,10-diaza-dibenzo[a,d]cycloheptene-10-carbonyl)-phenyl]-5-fluoro-2-methyl-benzamide 150231 HTry-Gly-Gly-Phe-Leu-Arg-Arg-lle-Arg-Pro-LysOH 150440 2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid amide 150448 7-Propyl-4,5,6,7,8,9-hexahydro-thiazolo[4,5-f]isoquinolin-2-ylamine 150449 8-Propyl-4,5,6,7,8,9-hexahydro-thiazolo[5,4-h]isoquinolin-2-ylamine 150472 6-Propyl-4,5,5a,6,7,8-hexahydro-thiazolo[4,5-f]quinolin-2-ylamine 150528 4-(4-Methyl-piperazin-1-yl)-pyrrolo[1,2-a]quinoxaline 150571 Biphenyl-2-carboxylic acid [3-hydroxy-4-(3,4,11,11a-tetrahydro-1H,5H-2-thia-4a,10-diaza-dibenzo[a,d]cycloheptene-10-carbonyl)-phenyl]-amide 150603 (-)-Trifluoro-methanesulfonic acid 3-(1-propyl-piperidin-3-yl)-phenyl ester 150635 2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-1-(3-hydroxymethyl-3,4-dihydro-1H-isoquinolin-2-yl)-propan-1-one 150674 1-{4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-butyl}-1H-benzotriazole 150809 Phosphoric acid mono-{2-((Z)-(S)-octadec-9-enoylamino)-3-[4-(pyridin-2-ylmethoxy)-phenyl]-propyl} ester 150810 Phosphoric acid mono-{(R)-2-((Z)-octadec-9-enoylamino)-3-[4-(pyridin-2-ylmethoxy)-phenyl]-propyl} ester 150822 Biphenyl-2-carboxylic acid [3-chloro-4-(3,4,11,11a-tetrahydro-1H,5H-2-thia-4a,10-diaza-dibenzo[a,d]cycloheptene-10-carbonyl)-phenyl]-amide 150858 Allyl-{1-[(S)-4-(benzenesulfonyl-methyl-amino)-3-methyl-3-phenyl-butyl]-piperidin-4-yl}-carbamic acid 4-nitro-benzyl ester 150865 5-Hydroxy-biphenyl-2-carboxylic acid [3-chloro-4-((S)-3,4,11,11a-tetrahydro-1H,5H-2-oxa-4a,10-diaza-dibenzo[a,d]cycloheptene-10-carbonyl)-phenyl]-amide 150873 6-Propyl-4,5,5a,6,7,8,9,9a-octahydro-thiazolo[4,5-f]quinolin-2-ylamine 150888 N*4*-(3-Bromo-phenyl)-quinazoline-4,7-diamine 150919 4-(1-Propyl-1,2,5,6-tetrahydro-pyridin-3-yl)-thiazol-2-ylamine 150920 7-Propyl-4,5,5a,6,7,8-hexahydro-thiazolo[4,5-f]isoquinolin-2-ylamine 150993 4-[(3-Bromophenyl)amino]-6,7-diaminoquinazoline 151031 5-Fluoro-biphenyl-2-carboxylic acid [3-chloro-4-(3,4,11,11a-tetrahydro-1H,5H-2-thia-4a,10-diaza-dibenzo[a,d]cycloheptene-10-carbonyl)-phenyl]-amide 151055 2-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-1H-benzotriazole 151056 1-(2-Methoxyphenyl)-4-propylpiperazine 151057 Allyl-{1-[(3S,4S)-1-(2-chloro-benzoyl)-4-phenyl-pyrrolidin-3-ylmethyl]-piperidin-4-yl}-carbamic acid 4-nitro-benzyl ester 151090 2-{4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-butyl}-1H-benzotriazole 151104 1-Ethyl-4-(2-methoxy-phenyl)-piperazine 151134 Biphenyl-2-carboxylic acid [4-(8-methyl-3,4,11,11a-tetrahydro-1H,5H-2-thia-4a,10-diaza-dibenzo[a,d]cycloheptene-10-carbonyl)-phenyl]-amide 151136 1-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-1H-benzotriazole 151137 1-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyl}-1H-benzotriazole 151139 2-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyl}-1H-benzotriazole 151341 Biphenyl-2-carboxylic acid [4-(3,4,11,11a-tetrahydro-1H,5H-2-thia-4a,10-diaza-dibenzo[a,d]cycloheptene-10-carbonyl)-phenyl]-amide 151348 Biphenyl-2-carboxylic acid [4-((R)-3,4,11,11a-tetrahydro-1H,5H-2-thia-4a,10-diaza-dibenzo[a,d]cycloheptene-10-carbonyl)-phenyl]-amide 151383 Biphenyl-2-carboxylic acid [4-((S)-3,4,11,11a-tetrahydro-1H,5H-2-thia-4a,10-diaza-dibenzo[a,d]cycloheptene-10-carbonyl)-phenyl]-amide 151410 1'-[4-phenyl-1-phenylsulfonyl-(3S,4S)-tetrahydro-1H-3-pyrrolylmethyl]spiro[2,3-dihydrobenzo[b]thiophenium-3,4'-(hexahydropyridine)]-1-olate 151439 alpha-MSH; Ac-Ser-Tyr-Ser-Met-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pro-Val-NH2 151444 4-(3-bromophenylamino)quinazoline-6,7-diol 151519 (3-Bromo-phenyl)-(5,6-dimethoxy-quinazolin-4-yl)-amine 151828 (3-Bromo-phenyl)-[1,3]dioxolo[4,5-g]quinazolin-8-yl-amine 151949 6-(4-methoxyphenyl)-3-(thiophen-3-yl)pyrazolo[1,5-a]pyrimidine 152030 8-(4-Chloro-5-methoxy-2-methyl-phenylamino)-3-(2-morpholin-4-yl-ethyl)-3H-imidazo[4,5-g]quinoline-7-carbonitrile 152061 3,6-Di-pyridin-4-yl-pyrazolo[1,5-a]pyrimidine 152078 [2-(6-Fluoro-2-methyl-chroman-8-yloxy)-ethyl]-[4-(4-methoxy-phenyl)-butyl]-amine 152080 Dipropyl-(6,7,8,9-tetrahydro-naphtho[1,2-b]furan-7-yl)-amine 152090 8-(2-Bromo-4-chloro-phenylamino)-3H-imidazo[4,5-g]quinoline-7-carbonitrile 152105 6-Fluoro-8-{2-[4-(4-methoxy-phenyl)-butylamino]-ethoxy}-chroman-4-one 152106 8-(5-Methoxy-2-methyl-phenylamino)-3-(2-morpholin-4-yl-ethyl)-3H-imidazo[4,5-g]quinoline-7-carbonitrile 152128 8-(2-Bromo-4-chloro-5-methoxy-phenylamino)-3-(2-morpholin-4-yl-ethyl)-3H-imidazo[4,5-g]quinoline-7-carbonitrile 152134 ((6S,7R)-6-Methyl-6,7,8,9-tetrahydro-naphtho[1,2-b]furan-7-yl)-dipropyl-amine 152137 Dipropyl-(6,7,8,9-tetrahydro-naphtho[2,1-b]furan-8-yl)-amine 152183 Dimethyl-(11-methyl-3,3a,8,12b-tetrahydro-2H-1-oxa-dibenzo[e,h]azulen-2-ylmethyl)-amine 152196 (S)-2-(3-tert-Butyl-5-methyl-benzyloxy)-1-phenyl-ethylamine 152197 2-(3,5-Bis-trifluoromethyl-benzyloxy)-1-methyl-1-phenyl-ethylamine 152204 8-(2-Chloro-5-methoxy-phenylamino)-3-(2-morpholin-4-yl-ethyl)-3H-imidazo[4,5-g]quinoline-7-carbonitrile 152205 8-(2-Chloro-5-methoxy-phenylamino)-3H-imidazo[4,5-g]quinoline-7-carbonitrile 152225 (S)-2-(3-Methoxy-5-methyl-benzyloxy)-1-phenyl-ethylamine 152243 8-(2-Bromo-4-chloro-5-methoxy-phenylamino)-3H-imidazo[4,5-g]quinoline-7-carbonitrile 152260 Dipropyl-(6,7,8,9-tetrahydro-naphtho[1,2-b]furan-8-yl)-amine 152261 (S)-2-(3-Bromo-5-methyl-benzyloxy)-1-phenyl-ethylamine 152288 6-(4-methoxyphenyl)-3-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidine 152295 (7aR,10aS)-8-Propyl-7,7a,8,9,10,10a-hexahydro-6H-1-oxa-8-aza-dicyclopenta[a,h]naphthalene 152300 (S)-2-(3,5-Dichloro-benzyloxy)-1-phenyl-ethylamine 152337 2-(3,5-Bis-trifluoromethyl-benzyloxy)-1-phenyl-propylamine (Diastereomer A) 152356 2-[(S)-2-(3,5-Bis-trifluoromethyl-benzyloxy)-1-phenyl-ethylamino]-acetamide 152360 2-{[(S)-2-(3,5-Bis-trifluoromethyl-benzyloxy)-1-phenyl-ethyl]-methyl-amino}-acetamide 152361 2-[1-(3,5-Bis-trifluoromethyl-phenyl)-ethoxy]-1-phenyl-ethylamine 152382 (S)-2-(3,5-Bis-trifluoromethyl-benzyloxy)-1-phenyl-ethylamine 152589 5-Fluoro-6-methyl-1-naphthalen-1-ylmethyl-2,3,4,4a,9,9a-hexahydro-1H-beta-carboline 152743 6-Fluoro-8-{2-[4-(4-methoxy-phenyl)-butylamino]-ethoxy}-chroman-4-one oxime 152744 6-Fluoro-8-{2-[4-(4-methoxy-phenyl)-butylamino]-ethoxy}-chroman-4-ol 152782 [2-(6-Fluoro-2,2-dimethyl-chroman-8-yloxy)-ethyl]-[4-(4-methoxy-phenyl)-butyl]-amine 152829 1-(3,4-Dimethoxy-benzyl)-6-methyl-2,3,4,9-tetrahydro-1H-beta-carboline 152927 [2-(6-Fluoro-2H-chromen-8-yloxy)-ethyl]-[4-(4-methoxy-phenyl)-butyl]-amine 152972 N-(3-{3-Butyl-4-[3-fluoro-2'-(2-fluoro-benzoylsulfamoyl)-5'-propyl-biphenyl-4-ylmethyl]-5-oxo-4,5-dihydro-[1,2,4]triazol-1-yl}-4-chloro-phenyl)-acetamide 153007 N-(3-{3-Butyl-4-[2'-(2-chloro-benzoylsulfamoyl)-3-fluoro-5'-propyl-biphenyl-4-ylmethyl]-5-oxo-4,5-dihydro-[1,2,4]triazol-1-yl}-4-chloro-phenyl)-acetamide 153043 4-{4-[2-(6-Fluoro-4-oxo-chroman-8-yloxy)-ethylamino]-butyl}-benzonitrile 153068 8-{2-[4-(2,3-Dihydro-benzofuran-5-yl)-butylamino]-ethoxy}-6-fluoro-chroman-4-one 153070 [2-(6-Fluoro-4-methoxy-chroman-8-yloxy)-ethyl]-[4-(4-methoxy-phenyl)-butyl]-amine 153090 8-[2-(4-Benzo[1,3]dioxol-5-yl-butylamino)-ethoxy]-6-fluoro-chroman-4-one 153105 1-(3,4-Dimethoxy-benzyl)-2,3,4,9-tetrahydro-1H-beta-carboline 153205 N-(3-{3-Butyl-4-[2'-(2-chloro-benzoylsulfamoyl)-biphenyl-4-ylmethyl]-5-oxo-4,5-dihydro-[1,2,4]triazol-1-yl}-4-chloro-phenyl)-propionamide 153206 Pentanoic acid (3-{3-butyl-4-[2'-(2-chloro-benzoylsulfamoyl)-biphenyl-4-ylmethyl]-5-oxo-4,5-dihydro-[1,2,4]triazol-1-yl}-4-chloro-phenyl)-amide 153207 N-{3-[3-Butyl-4-(3-fluoro-2'-(ethyloxtycarbonyl)sulfamoyl-5'-propyl-biphenyl-4-ylmethyl)-5-oxo-4,5-dihydro-[1,2,4]triazol-1-yl]-4-chloro-phenyl}-acetamide 153208 N-{3-[3-Butyl-4-(3-fluoro-5'-propyl-2'-(N-t-butyloxycarbonyl)-Sulfanamido-biphenyl-4-ylmethyl)-5-oxo-4,5-dihydro-[1,2,4]triazol-1-yl]-4-chloro-phenyl}-acetamide 153216 [2-(6-Fluoro-2-methyl-chroman-8-yloxy)-ethyl]-[3-(4-methoxy-phenyl)-propyl]-amine 153248 [2-(6-Fluoro-2-methyl-chroman-8-yloxy)-ethyl]-[2-(4-methoxy-phenyl)-ethyl]-amine 153259 1-(3,4-Dimethoxy-benzyl)-6,7-dimethyl-2,3,4,9-tetrahydro-1H-beta-carboline 153289 1-(3,4-Dimethoxy-benzyl)-7,8-dimethyl-2,3,4,9-tetrahydro-1H-beta-carboline 153307 6-Fluoro-8-{2-[2-(4-methoxy-phenyl)-ethylamino]-ethoxy}-chroman-4-ol 153308 [2-(6-Fluoro-2-methyl-chroman-8-yloxy)-ethyl]-[6-(4-methoxy-phenyl)-hexyl]-amine 153313 [2-(6-Fluoro-2-methyl-chroman-8-yloxy)-ethyl]-[5-(4-methoxy-phenyl)-pentyl]-amine 153339 6-Fluoro-8-{2-[2-(4-methoxy-phenyl)-ethylamino]-ethoxy}-chroman-4-one 153341 4-(1-(cyclopropylmethyl)-4-(4-fluorophenyl)-1H-imidazol-5-yl)pyridine 153349 4'-[3-Butyl-5-oxo-1-(2-trifluoromethyl-phenyl)-1,5-dihydro-[1,2,4]triazol-4-ylmethyl]-5-propyl-biphenyl-2-sulfonic acid(tert-butoxycarbonyl) amide 153350 4'-[3-Butyl-5-oxo-1-(2-trifluoromethyl-phenyl)-1,5-dihydro-[1,2,4]triazol-4-ylmethyl]-3'-fluoro-biphenyl-2-sulfonic acid(tert-butoxycarbonyl) amide 153359 (Z)-(2-(hydroxymethyl)-4-(3-isobutyl-5-methylhexylidene)-5-oxo-tetrahydrofuran-2-yl)methyl pivalate 153362 N-(3-{3-Butyl-4-[2'-(2-chloro-benzoylsulfamoyl)-5'-ethyl-biphenyl-4-ylmethyl]-5-oxo-4,5-dihydro-[1,2,4]triazol-1-yl}-4-chloro-phenyl)-propionamide 153363 4'-[3-Butyl-5-oxo-1-(2-trifluoromethyl-phenyl)-1,5-dihydro-[1,2,4]triazol-4-ylmethyl]-3'-fluoro-5-propyl-biphenyl-2-sulfonic acid 2-chloro-benzoylamide 153375 6-Fluoro-8-{2-[4-(4-hydroxy-phenyl)-butylamino]-ethoxy}-chroman-4-one 153381 1-(2-Bromo-3,4-dimethoxy-benzyl)-6-methyl-2,3,4,9-tetrahydro-1H-beta-carboline 153382 1-(2-Chloro-3,4-dimethoxy-benzyl)-6-methyl-2,3,4,9-tetrahydro-1H-beta-carboline 153386 6-Fluoro-8-{2-[4-(3-methoxy-phenyl)-butylamino]-ethoxy}-chroman-4-one 153388 8-{2-[4-(4-Ethoxy-phenyl)-butylamino]-ethoxy}-6-fluoro-chroman-4-one 153391 Pentanoic acid (3-{3-butyl-4-[2'-(2-chloro-benzoylsulfamoyl)-5'-ethyl-biphenyl-4-ylmethyl]-5-oxo-4,5-dihydro-[1,2,4]triazol-1-yl}-4-chloro-phenyl)-amide 153392 N-(3-{3-Butyl-4-[2'-(2-chloro-benzoylsulfamoyl)-biphenyl-4-ylmethyl]-5-oxo-4,5-dihydro-[1,2,4]triazol-1-yl}-4-chloro-phenyl)-acetamide 153428 6-Fluoro-8-[2-(4-phenyl-butylamino)-ethoxy]-chroman-4-one 153454 4-[[2'-[N-(tert-Butoxycarbonyl)sulfamoyl]biphenyl-4-yl]methyl]-5-n-butyl-2,4-dihydro-2-[5-(propionylamino)-2-(trifluoromethyl)phenyl]-3H-1,2,4-trizol-3-one 153460 8-Bromo-1-(3,4-dimethoxy-benzyl)-7-methyl-2,3,4,9-tetrahydro-1H-beta-carboline 153477 8-{2-[4-(4-Chloro-phenyl)-butylamino]-ethoxy}-6-fluoro-chroman-4-one 153478 6-Fluoro-8-{2-[4-(4-methylsulfanyl-phenyl)-butylamino]-ethoxy}-chroman-4-one 153479 6-Fluoro-8-{2-[4-(2-methoxy-phenyl)-butylamino]-ethoxy}-chroman-4-one 153480 (4S,5S)-4-(3,4-difluorophenyl)-N-(3-(4-(4-fluorophenyl)piperidin-1-yl)propyl)-5-methyl-2-oxooxazolidine-3-carboxamide 153509 8-{2-[4-(4-Dimethylamino-phenyl)-butylamino]-ethoxy}-6-fluoro-chroman-4-one 153593 8-{2-[4-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-butylamino]-ethoxy}-6-fluoro-chroman-4-one 153627 6-Fluoro-8-{2-[4-(4-methoxy-naphthalen-1-yl)-butylamino]-ethoxy}-chroman-4-one 153628 2-(2-{4-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-piperazin-1-yl}-ethyl)-indan-1-one 153664 8-{2-[(4-Benzo[1,3]dioxol-5-yl-butyl)-propyl-amino]-ethoxy}-6-fluoro-chroman-4-one 153739 4'-[3-Butyl-5-oxo-1-(2-trifluoromethyl-phenyl)-1,5-dihydro-[1,2,4]triazol-4-ylmethyl]-3'-fluoro-biphenyl-2-sulfonic acid 2-chloro-benzoylamide 153926 4'-[3-Butyl-5-oxo-1-(2-trifluoromethyl-phenyl)-1,5-dihydro-[1,2,4]triazol-4-ylmethyl]-5-propyl-biphenyl-2-sulfonic acid 2-chloro-benzoylamide 153927 4'-[3-Butyl-5-oxo-1-(2-trifluoromethyl-phenyl)-1,5-dihydro-[1,2,4]triazol-4-ylmethyl]-biphenyl-2-sulfonic acid 2-chloro-benzoylamide 154225 1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-(piperidin-4-yl)-3,4-dihydroquinazolin-2(1H)-one 154250 Octadec-9-enoic acid 2-hydroxymethyl-5-oxo-tetrahydro-furan-2-ylmethyl ester 154255 5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)-7-methoxy-3,4-dihydroquinazolin-2(1H)-one 154331 1,3-Bis-[(Z)-4-methyl-benzylimino]-2,3-dihydro-1H-isoindole 154480 1-[(Z)-2-(4-Chloro-phenyl)-ethylimino]-3-[(Z)-isopropylimino]-2,3-dihydro-1H-isoindole 154520 1,3-Bis-[(Z)-2-(4-fluoro-phenyl)-ethylimino]-2,3-dihydro-1H-isoindole 154521 N-(1-{1-[1-Carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-3-(2-{2-[(10,11-dihydro-5H-dibenzo[a,d]cycloheptene-5-carbonyl)-amino]-3,3-diphenyl-propionylamino}-4-methyl-pentanoylamino)-succinamic acid 154522 (S)-N-((1S,2S)-1-{(1S,2S)-1-[(S)-1-Carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-3-[(S)-2-((S)-2-diphenylacetylamino-3,3-diphenyl-propionylamino)-4-methyl-pentanoylamino]-succinamic acid 154527 1,3-Bis-[(Z)-2-p-tolyl-ethylimino]-2,3-dihydro-1H-isoindole 154558 1,3-Bis-[(Z)-2-(4-chloro-phenyl)-ethylimino]-2,3-dihydro-1H-isoindole 154657 Acetic acid 2-hydroxymethyl-4-[(Z)-octadec-9-en-(E)-ylidene]-5-oxo-tetrahydro-furan-2-ylmethyl ester 154684 methyl 5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)-2-oxo-1,2,3,4-tetrahydroquinazoline-7-carboxylate 154771 1'-(4-Pyridin-4-yl-butyl)-1',2',3',6'-tetrahydro-[2,4']bipyridinyl 154779 Nociceptin/orphanin FQ analogue 154798 SID26751783 154827 (S)-N-((1S,2S)-1-{(1S,2S)-1-[(S)-1-Carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-3-{(S)-2-[(S)-2-(2,2-dimethyl-propionylamino)-3,3-diphenyl-propionylamino]-4-methyl-pentanoylamino}-succinamic acid 154847 4-[4-(4-Thiophen-2-yl-3,6-dihydro-2H-pyridin-1-yl)-butyl]-pyridine 154986 (S)-N-((1S,2S)-1-{(1S,2S)-1-[(S)-1-Carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-3-{(S)-2-[(S)-2-(3-cyclohexyl-ureido)-3,3-diphenyl-propionylamino]-4-methyl-pentanoylamino}-succinamic acid 155002 3-(2-Dimethylamino-ethyl)-1H-indole-5-sulfonic acid methylamide 155006 SID29215485 155013 (S)-N-((1S,2S)-1-{(1S,2S)-1-[(S)-1-Carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-3-{(S)-2-[(S)-2-(cyclohexanecarbonyl-amino)-3,3-diphenyl-propionylamino]-4-methyl-pentanoylamino}-succinamic acid 155030 Acetic acid 2-hydroxymethyl-5-oxo-4-[(Z)-tetradec-9-en-(E)-ylidene]-tetrahydro-furan-2-ylmethyl ester 155045 SID26751577 155072 1,3-Bis-[(Z)-2-(4-fluoro-phenyl)-ethylimino]-2,3-dihydro-1H-pyrrolo[3,4-c]pyridine 155078 N-{3-[(E)-4-Methyl-benzylimino]-1-[(Z)-4-methyl-benzylimino]-2,3-dihydro-1H-isoindol-5-yl}-acetamide 155082 Acetic acid 3-hydroxymethyl-5-oxo-4-tetradec-(Z)-ylidene-tetrahydro-furan-3-ylmethyl ester 155108 (S)-2-[(2S,3S)-2-((2S,3S)-2-{(S)-2-[(S)-2-((S)-2-Acetylamino-3-phenyl-propionylamino)-4-methyl-pentanoylamino]-3-phenyl-propionylamino}-3-methyl-pentanoylamino)-3-methyl-pentanoylamino]-3-(1H-indol-3-yl)-propionic acid 155116 [1-(4-Fluoro-benzyl)-1H-benzoimidazol-2-yl]-{1-[2-(4-methoxy-phenyl)-ethyl]-piperidin-4-yl}-methanone 155128 5,6-Dichloro-1,3-bis-[(Z)-2-p-tolyl-ethylimino]-2,3-dihydro-1H-isoindole 155130 Acetic acid 2-hydroxymethyl-5-oxo-4-tetradec-(Z)-ylidene-tetrahydro-furan-2-ylmethyl ester 155165 (S)-N-((1S,2S)-1-{(1S,2S)-1-[(S)-1-Carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-3-{(S)-2-[(S)-3,3-diphenyl-2-(2,2,2-trifluoro-acetylamino)-propionylamino]-4-methyl-pentanoylamino}-succinamic acid 155173 (S)-N-((1S,2S)-1-{(1S,2S)-1-[(S)-1-Carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-3-[(S)-2-((S)-3,3-diphenyl-2-propionylamino-propionylamino)-4-methyl-pentanoylamino]-succinamic acid 155174 (S)-3-[(S)-2-((S)-2-Amino-3,3-diphenyl-propionylamino)-4-methyl-pentanoylamino]-N-((1S,2S)-1-{(1S,2S)-1-[(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 155183 6-((R)-2-{2-[4-(4-Chloro-phenoxy)-piperidin-1-yl]-ethyl}-pyrrolidine-1-sulfonyl)-1H-indole 155221 4-[4-(4-p-Tolyl-3,6-dihydro-2H-pyridin-1-yl)-butyl]-pyridine 155228 6-{(R)-2-[2-(4-Methyl-piperidin-1-yl)-ethyl]-pyrrolidine-1-sulfonyl}-1H-indole 155229 4-Methyl-1-{2-[(S)-1-(naphthalene-1-sulfonyl)-pyrrolidin-2-yl]-ethyl}-piperidine 155230 4-Methyl-1-{2-[(R)-1-(naphthalene-1-sulfonyl)-pyrrolidin-2-yl]-ethyl}-piperidine 155258 4-{4-[4-(4-Methoxy-phenyl)-3,6-dihydro-2H-pyridin-1-yl]-butyl}-pyridine 155259 4-{4-[4-(4-Chloro-phenyl)-3,6-dihydro-2H-pyridin-1-yl]-butyl}-pyridine 155260 4-[4-(4-Naphthalen-2-yl-3,6-dihydro-2H-pyridin-1-yl)-butyl]-pyridine 155264 Acetic acid 3-hydroxy-5-oxo-4-tetradec-(E)-ylidene-tetrahydro-furan-3-ylmethyl ester 155280 4-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-butyl]-pyridine 155291 3-[1-(4-Pyridin-4-yl-butyl)-1,2,3,6-tetrahydro-pyridin-4-yl]-1H-indole 155297 Tetradecanoic acid 3-hydroxymethyl-5-oxo-tetrahydro-furan-3-ylmethyl ester 155311 4-{4-[4-(4-Fluoro-phenyl)-3,6-dihydro-2H-pyridin-1-yl]-butyl}-pyridine 155358 2-{2-[2-(2-{2-[2-Acetylamino-3-(1H-indol-3-yl)-propionylamino]-4-methyl-pentanoylamino}-5-guanidino-pentanoylamino)-3-methyl-pentanoylamino]-3-methyl-pentanoylamino}-3-(1H-indol-3-yl)-propionic acid 155387 N-{4-Methoxy-3-[((2S,3S)-2-phenyl-piperidin-3-ylamino)-methyl]-phenyl}-N-methyl-methanesulfonamide 155423 (2-Isopropoxy-5-trifluoromethoxy-benzyl)-((2S,3S)-2-phenyl-piperidin-3-yl)-amine 155426 (2-Ethoxy-5-trifluoromethoxy-benzyl)-((2S,3S)-2-phenyl-piperidin-3-yl)-amine 155427 2-[((2S,3S)-2-Phenyl-piperidin-3-ylamino)-methyl]-4-trifluoromethoxy-phenol 155482 Nociceptin/orphanin FQ analogue 155483 2-[3-(4-Fluoro-phenoxy)-propyl]-5-methyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole 155485 5-Methyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole 155488 (S)-N-((1S,2S)-1-{(1S,2S)-1-[(S)-1-Carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-3-{(S)-4-methyl-2-[(S)-2-(3-methyl-ureido)-3,3-diphenyl-propionylamino]-pentanoylamino}-succinamic acid 155489 3-{2-[2-Amino-3-(1H-indol-3-yl)-propionylamino]-4-methyl-pentanoylamino}-N-(1-{1-[1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 155588 N-(1-{1-[1-Carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-3-{2-[4-(1H-indol-3-ylmethyl)-2,5-dioxo-imidazolidin-1-yl]-4-methyl-pentanoylamino}-succinamic acid 155589 15,18-Di-sec-butyl-9,12-bis-(1H-indol-3-ylmethyl)-6-isobutyl-10-methyl-5,8,11,14,17,20-hexaoxo-1-thia-4,7,10,13,16,19-hexaaza-cyclohenicosane-3-carboxylic acid 155590 [5,8-Di-sec-butyl-11,14-bis-(1H-indol-3-ylmethyl)-17-isobutyl-3,6,9,12,15,18-hexaoxo-1,4,7,10,13,16hexaaza-cyclooctadec-2-yl]-acetic acid 155605 1,3-Bis-[(Z)-2-(3-chloro-phenyl)-ethylimino]-2,3-dihydro-1H-isoindole 155606 1,3-Bis-[(Z)-2-(4-chloro-phenyl)-propylimino]-2,3-dihydro-1H-isoindole 155638 3-(2-{2-[(Adamantane-1-carbonyl)-amino]-3,3-diphenyl-propionylamino}-4-methyl-pentanoylamino)-N-(1-{1-[1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 155643 1,3-Bis-[(Z)-2-(4-fluoro-phenyl)-ethylimino]-5-propoxy-2,3-dihydro-1H-isoindole 155652 (S)-3-[(S)-2-((S)-2-Benzoylamino-3,3-diphenyl-propionylamino)-4-methyl-pentanoylamino]-N-((1S,2S)-1-{(1S,2S)-1-[(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 155666 (S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propionylamino)-4-methyl-pentanoylamino]-N-((S)-1-{(1S,2S)-1-[(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-phenyl-ethyl)-succinamic acid 155704 [3-(3,4-Dimethoxy-phenyl)-3-(2-{4-[1-(4-fluoro-benzyl)-1H-benzoimidazole-2-carbonyl]-piperidin-1-yl}-ethyl)-pyrrolidin-1-yl]-(3,4,5-trimethoxy-phenyl)-methanone 155705 5-Methoxy-1,3-bis-[(Z)-2-p-tolyl-ethylimino]-2,3-dihydro-1H-isoindole 155706 5-(2-Dimethylamino-ethoxy)-1,3-bis-[(Z)-2-(4-fluoro-phenyl)-ethylimino]-2,3-dihydro-1H-isoindole 155761 7-Methyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid (2-hydroxymethyl-2-methyl-butyl)-amide 155897 71 155966 (S)-N-((1S,2S)-1-{(1S,2S)-1-[(S)-1-Carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-3-((S)-2-{(S)-3,3-diphenyl-2-[(pyridine-3-carbonyl)-amino]-propionylamino}-4-methyl-pentanoylamino)-succinamic acid 156008 N-cyclohexyl-7-methyl-2-phenyl-1,8-naphthyridin-4-amine 156019 (S)-4-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propionylamino)-4-methyl-pentanoylamino]-4-((1S,2S)-1-{(1S,2S)-1-[(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butylcarbamoyl)-butyric acid 156035 3-[2-(2-Acetylamino-3,3-diphenyl-propionylamino)-4-methyl-pentanoylamino]-N-(1-{1-[1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 156204 4-chloro-7-methyl-2-phenyl-1,8-naphthyridine 156270 6-Methoxy-4-(4-phenoxy-phenylamino)-quinoline-3-carbonitrile 156271 5-Methoxy-4-(4-phenoxy-phenylamino)-quinoline-3-carbonitrile 156308 K-252a analogue 156321 1-{2-[(R)-3-(3,4-Dichloro-phenyl)-1-(3,4,5-trimethoxy-benzoyl)-pyrrolidin-3-yl]-ethyl}-4-phenyl-piperidine-4-carboxylic acid amide 156372 SID11110961 156414 7-bromo-2-phenyl-1,8-naphthyridin-4-ol 156452 (6,7-Dimethoxy-quinazolin-4-yl)-(4-phenoxy-phenyl)-amine 156494 3-{2-[2-Acetylamino-3-(1H-indol-3-yl)-propionylamino]-4-methyl-pentanoylamino}-N-(1-{1-[1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 156529 6-Methoxy-7-(2-morpholin-4-yl-ethoxy)-4-(4-phenoxy-phenylamino)-quinoline-3-carbonitrile 156531 7-(3-Morpholin-4-yl-propoxy)-4-(4-phenoxy-phenylamino)-quinoline-3-carbonitrile 156534 5,7-Dimethoxy-4-(4-phenoxy-phenylamino)-quinoline-3-carbonitrile 156550 (5-Dimethylamino-2-methoxy-benzyl)-((2S,3S)-2-phenyl-piperidin-3-yl)-amine 156551 (2S,3S)-N-(2-methoxy-5-(trifluoromethoxy)benzyl)-2-phenylpiperidin-3-amine 156554 4-(4-Phenoxy-phenylamino)-quinoline-3-carbonitrile 156555 7-Methoxy-4-(4-phenoxy-phenylamino)-quinoline-3-carbonitrile 156584 8-{(R)-1-Methyl-2-[4-(2,4,5-trifluoro-phenyl)-piperazin-1-yl]-ethyl}-8-aza-spiro[4.5]decane-7,9-dione 156767 1-(3,4-Dimethoxy-phenyl)-4-[4-(1-ethyl-propyl)-piperazin-1-yl]-butane-1,4-dione 157077 Biphenyl-4-sulfonic acid (4-piperazin-1-yl-quinolin-6-yl)-amide 157085 1-(4-Chloro-phenyl)-4-[4-(1-ethyl-propyl)-piperazin-1-yl]-butane-1,4-dione 157086 (2,5-Dimethoxy-benzyl)-((2S,3S)-2-phenyl-piperidin-3-yl)-amine 157124 (5-Chloro-2-methoxy-benzyl)-((2S,3S)-2-phenyl-piperidin-3-yl)-amine 157152 SID26752091 157153 2-Hydrazonomethyl-6-oxo-1,6-dihydro-[3,4']bipyridinyl-5-carbonitrile 157238 3-(fluoromethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide 157413 4-Amino-N-(9-chloro-2-furan-2-yl-[1,2,4]triazolo[1,5-c]quinazolin-5-yl)-butyramide 157420 N-(9-Chloro-2-furan-2-yl-[1,2,4]triazolo[1,5-c]quinazolin-5-yl)-3-iodo-benzamide 157426 3-Fluoromethyl-7-nitro-1,2,3,4-tetrahydro-isoquinoline 157427 8-chloro-2-(thiophen-3-yl)-[1,2,4]triazolo[1,5-a]quinoxalin-4(5H)-one 157430 1-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-2-[3-(3,4-dichloro-benzyl)-2-imino-2,3-dihydro-benzoimidazol-1-yl]-ethanone 157431 1-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-2-(2-imino-3-methyl-2,3-dihydro-benzoimidazol-1-yl)-ethanone 157451 3-Amino-N-(9-chloro-2-furan-2-yl-[1,2,4]triazolo[1,5-c]quinazolin-5-yl)-propionamide 157459 5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic acid (2-methyl-4-piperazin-1-yl-quinolin-6-yl)-amide 157530 [3-(9-Chloro-2-furan-2-yl-[1,2,4]triazolo[1,5-c]quinazolin-5-ylcarbamoyl)-propyl]-carbamic acid tert-butyl ester 157558 8-chloro-2-(thiophen-2-yl)-[1,2,4]triazolo[1,5-a]quinoxalin-4(5H)-one 157559 2-(thiophen-2-yl)-[1,2,4]triazolo[1,5-a]quinoxalin-4(5H)-one 157561 8-chloro-2-(furan-3-yl)-[1,2,4]triazolo[1,5-a]quinoxalin-4(5H)-one 157564 1-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-2-[2-imino-3-(2-piperidin-1-yl-ethyl)-2,3-dihydro-benzoimidazol-1-yl]-ethanone 157565 2-[3-(4-tert-Butyl-benzyl)-2-imino-2,3-dihydro-benzoimidazol-1-yl]-1-(3,5-di-tert-butyl-4-hydroxy-phenyl)-ethanone 157596 2-Ethyl-4-(4-nitro-phenyl)-6-propyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid 5-{[3-(4,4-diphenyl-piperidin-1-yl)-propyl]-amide} 3-ethylamide 157631 Pentanoic acid (9-chloro-2-furan-2-yl-[1,2,4]triazolo[1,5-c]quinazolin-5-yl)-amide 157632 N-(9-Chloro-2-furan-2-yl-[1,2,4]triazolo[1,5-c]quinazolin-5-yl)-butyramide 157635 8-chloro-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a]quinoxalin-4(5H)-one 157636 2-(furan-2-yl)-[1,2,4]triazolo[1,5-a]quinoxalin-4(5H)-one 157650 (2-Isopropoxy-benzyl)-((2S,3S)-2-phenyl-piperidin-3-yl)-amine 157665 N-(9-chloro-2-(furan-2-yl)-[1,2,4]triazolo[1,5-c]quinazolin-5-yl)propionamide 157675 N-(9-chloro-2-(furan-2-yl)-[1,2,4]triazolo[1,5-c]quinazolin-5-yl)benzamide 157676 (9-Chloro-2-furan-2-yl-[1,2,4]triazolo[1,5-c]quinazolin-5-yl)-carbamic acid tert-butyl ester 157684 (2-Difluoromethoxy-benzyl)-((2S,3S)-2-phenyl-piperidin-3-yl)-amine 157685 ((2S,3S)-2-Phenyl-piperidin-3-yl)-(2-trifluoromethoxy-benzyl)-amine 157716 3-[(Z)-3-Methoxy-isoxazol-5-ylmethoxyimino]-1-azonia-bicyclo[2.2.2]octane chloride 157717 3-[(Z)-3-Cyano-isoxazol-5-ylmethoxyimino]-1-azonia-bicyclo[2.2.2]octane chloride 157718 3-[(Z)-3-Chloro-isoxazol-5-ylmethoxyimino]-1-azonia-bicyclo[2.2.1]heptane chloride 157725 N-phenethyltrans-3,4-dimethyl-4-(3-hydroxyphenyl)piperidine 157750 3-[(Z)-3-Chloro-isoxazol-5-ylmethoxyimino]-1-azonia-bicyclo[2.2.2]octane chloride 157753 1-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-2-[2-imino-3-(4-methyl-benzyl)-2,3-dihydro-benzoimidazol-1-yl]-ethanone 157757 7-(benzyloxy)-2-morpholino-4H-chromen-4-one 157763 3-[(3-Methoxy-isoxazol-5-ylmethoxyimino)-methyl]-1-azonia-bicyclo[2.2.1]heptane chloride 157777 8-chloro-2-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-a]quinoxalin-4(5H)-one 157790 1-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-2-(2-imino-2,3-dihydro-benzoimidazol-1-yl)-ethanone 157791 1-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-2-[2-imino-3-(2-morpholin-4-yl-ethyl)-2,3-dihydro-benzoimidazol-1-yl]-ethanone 157802 2-(4-Amino-phenyl)-N-(9-chloro-2-furan-2-yl-[1,2,4]triazolo[1,5-c]quinazolin-5-yl)-acetamide 157806 5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic acid [4-(4-methyl-piperazin-1-yl)-quinolin-6-yl]-amide 157807 3-[(Z)-3-Bromo-isoxazol-5-ylmethoxyimino]-1-azonia-bicyclo[2.2.1]heptane chloride 157831 5-Amino-pentanoic acid (9-chloro-2-furan-2-yl-[1,2,4]triazolo[1,5-c]quinazolin-5-yl)-amide 157834 5-Chloro-naphthalene-2-sulfonic acid (4-piperazin-1-yl-quinolin-6-yl)-amide 157839 3-[(Z)-3-Cyano-isoxazol-5-ylmethoxyimino]-1-azonia-bicyclo[2.2.1]heptane chloride 157908 4-tert-Butyl-N-(4-piperazin-1-yl-quinolin-6-yl)-benzenesulfonamide 157934 2-(3-Butyl-2-imino-2,3-dihydro-benzoimidazol-1-yl)-1-(3,5-di-tert-butyl-4-hydroxy-phenyl)-ethanone 157954 1-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-2-(3-heptyl-2-imino-2,3-dihydro-benzoimidazol-1-yl)-ethanone 157971 2-(3-Benzyl-2-imino-2,3-dihydro-benzoimidazol-1-yl)-1-(3,5-di-tert-butyl-4-hydroxy-phenyl)-ethanone 157986 5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic acid [4-((S)-3-methyl-piperazin-1-yl)-quinolin-6-yl]-amide 157989 2-(2-Amino-ethoxymethyl)-6-ethyl-4-(4-nitro-phenyl)-1,4-dihydro-pyridine-3,5-dicarboxylic acid 3-{[3-(4,4-diphenyl-piperidin-1-yl)-propyl]-amide} 5-ethylamide 157991 2-(2-Amino-ethoxymethyl)-6-ethyl-4-(4-nitro-phenyl)-1,4-dihydro-pyridine-3,5-dicarboxylic acid 5-amide 3-{[3-(4,4-diphenyl-piperidin-1-yl)-propyl]-amide} 157992 2-(3-Amino-propoxymethyl)-6-ethyl-4-(4-nitro-phenyl)-1,4-dihydro-pyridine-3,5-dicarboxylic acid 5-amide 3-{[3-(4,4-diphenyl-piperidin-1-yl)-propyl]-amide} 158011 9-Chloro-2-furan-2-yl-6-propyl-6H-[1,2,4]triazolo[1,5-c]quinazolin-5-one 158021 3-[(Z)-3-Bromo-isoxazol-5-ylmethoxyimino]-1-azonia-bicyclo[2.2.2]octane chloride 158022 3-[(3-Bromo-isoxazol-5-ylmethoxyimino)-methyl]-1-azonia-bicyclo[2.2.2]octane chloride 158024 3-[(3-Bromo-isoxazol-5-ylmethoxyimino)-methyl]-1-azonia-bicyclo[2.2.1]heptane chloride 158033 5-Chloro-2-methyl-benzo[b]thiophene-3-sulfonic acid (4-piperazin-1-yl-quinolin-6-yl)-amide 158035 3-[(3-Cyano-isoxazol-5-ylmethoxyimino)-methyl]-1-azonia-bicyclo[2.2.1]heptane chloride 158036 3-[(3-Methoxy-isoxazol-5-ylmethoxyimino)-methyl]-1-azonia-bicyclo[2.2.2]octane chloride 158049 3-[(Z)-3-Methoxy-isoxazol-5-ylmethoxyimino]-1-azonia-bicyclo[2.2.1]heptane chloride 158053 5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic acid (4-piperazin-1-yl-quinolin-6-yl)-amide 158064 3-[(3-Chloro-isoxazol-5-ylmethoxyimino)-methyl]-1-azonia-bicyclo[2.2.2]octane chloride 158073 3-[(3-Chloro-isoxazol-5-ylmethoxyimino)-methyl]-1-azonia-bicyclo[2.2.1]heptane chloride 158074 3-[(3-Cyano-isoxazol-5-ylmethoxyimino)-methyl]-1-azonia-bicyclo[2.2.2]octane chloride 158093 N-(9-Chloro-2-furan-2-yl-[1,2,4]triazolo[1,5-c]quinazolin-5-yl)-2,2-dimethyl-propionamide 158139 8-methoxy-2-morpholino-4H-chromen-4-one 158169 5-Chloro-3-ethyl-benzo[b]thiophene-2-sulfonic acid (4-piperazin-1-yl-quinolin-6-yl)-amide 158225 2-(3,4-Dichloro-phenyl)-N-[(S)-1-(4-isothiocyanato-phenyl)-2-pyrrolidin-1-yl-ethyl]-N-methyl-acetamide 158226 2-Ethyl-4-(4-nitro-phenyl)-6-(2,2,2-trifluoro-ethoxymethyl)-1,4-dihydro-pyridine-3,5-dicarboxylic acid 3-amide 5-{[3-(4,4-diphenyl-piperidin-1-yl)-propyl]-amide} 158266 2-(4-Isothiocyanato-phenyl)-N-methyl-N-((S)-1-phenyl-2-pyrrolidin-1-yl-ethyl)-acetamide 158317 2-(4,5-Dichloro-2-isothiocyanato-phenyl)-N-methyl-N-((S)-1-phenyl-2-pyrrolidin-1-yl-ethyl)-acetamide 158347 SID11113703 158348 2-(3-Isothiocyanato-phenyl)-N-methyl-N-((S)-1-phenyl-2-pyrrolidin-1-yl-ethyl)-acetamide 158383 2-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-a]quinoxalin-4(5H)-one 158403 N-(9-chloro-2-(furan-2-yl)-[1,2,4]triazolo[1,5-c]quinazolin-5-yl)acetamide 158439 4-(9-Chloro-2-furan-2-yl-[1,2,4]triazolo[1,5-c]quinazolin-5-ylcarbamoyl)-butyric acid 158481 2-Ethyl-6-(4-methoxy-butyl)-4-(4-nitro-phenyl)-1,4-dihydro-pyridine-3,5-dicarboxylic acid 3-amide 5-{[3-(4,4-diphenyl-piperidin-1-yl)-propyl]-amide} 158482 2-Ethyl-6-methoxymethyl-4-(4-nitro-phenyl)-1,4-dihydro-pyridine-3,5-dicarboxylic acid 3-amide 5-{[3-(4,4-diphenyl-piperidin-1-yl)-propyl]-amide} 158511 ((S)-2-Methyl-5,6,7,8-tetrahydro-indolizin-7-yl)-dipropyl-amine 158534 Biphenyl-4-carboxylic acid [(4aS,10bR)-4-(2,3,4a,5,6,10b-hexahydro-1H-benzo[f]quinolin-4-yl)-butyl]-amide 158550 ((S)-1-Methyl-5,6,7,8-tetrahydro-indolizin-7-yl)-dipropyl-amine 158565 (R)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizine-1-carbaldehyde 158566 (S)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizine-3-carbaldehyde 158605 (R)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizine-3-carbaldehyde 158608 ((R)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizin-1-yl)-methanol 158618 Naltrindole analogue 158619 ((R)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizin-2-yl)-methanol 158620 ((S)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizin-2-yl)-methanol 158621 ((R)-1-Methyl-5,6,7,8-tetrahydro-indolizin-7-yl)-dipropyl-amine 158725 N*2*-(3-Amino-propyl)-N*6*-(4-chloro-phenyl)-8-isopropyl-9H-purine-2,6-diamine 158726 N*2*-Benzyl-N*6*-(4-chloro-phenyl)-8-isopropyl-9H-purine-2,6-diamine 158752 Naltrindole analogue 158753 (4-Chloro-phenyl)-(8-methyl-2-morpholin-4-yl-9H-purin-6-yl)-amine 158791 (4-Chloro-phenyl)-(2-morpholin-4-yl-8-propyl-9H-purin-6-yl)-amine 158795 NQLPpYNELNLGRREEpYDVLD 158900 [3-(2-Oxo-1,2-dihydro-quinolin-3-yl)-phenoxy]-acetic acid 158935 2-Hydroxy-5H-11-oxa-5-aza-benzo[a]fluoren-6-one 159009 ((R)-3-Methyl-5,6,7,8-tetrahydro-indolizin-7-yl)-dipropyl-amine 159010 ((S)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizin-3-yl)-methanol 159011 (S)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizine-1-carbaldehyde 159033 ((R)-2-Methyl-5,6,7,8-tetrahydro-indolizin-7-yl)-dipropyl-amine 159047 ((R)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizin-3-yl)-methanol 159075 ((S)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizin-1-yl)-methanol 159076 Dipropyl-(R)-5,6,7,8-tetrahydro-indolizin-7-yl-amine 159088 ((S)-3-Methyl-5,6,7,8-tetrahydro-indolizin-7-yl)-dipropyl-amine 159150 7-Hydroxy-10H-11-oxa-10-aza-benzo[b]fluoren-5-one 159154 (8-Isopropyl-2-morpholin-4-yl-9H-purin-6-yl)-(4-trifluoromethyl-phenyl)-amine 159155 1-[6-(4-Chloro-phenylamino)-8-isopropyl-9H-purin-2-yl]-4-phenyl-piperidin-4-ol 159175 3-[3-(2-Hydroxy-ethoxy)-phenyl]-1H-quinolin-2-one 159180 (4-Chloro-phenyl)-(8-ethyl-2-morpholin-4-yl-9H-purin-6-yl)-amine 159218 (4-Chloro-phenyl)-[2-(4,4-dimethoxy-piperidin-1-yl)-8-isopropyl-9H-purin-6-yl]-amine 159219 (4-Chloro-phenyl)-(8-isopropyl-2-morpholin-4-yl-9H-purin-6-yl)-amine 159266 22-cyclopropylmethyl-8-phenoxy-14-oxa-11,22-diazaheptacyclo[13.9.1.01,13.02,21.04,12.05,10.019,25]pentacosa-4(12),5(10),6,8,15(25),16,18-heptaene-2,16-diol 159268 22-cyclopropylmethyl-6-phenyl-14-oxa-11,22-diazaheptacyclo[13.9.1.01,13.02,21.04,12.05,10.019,25]pentacosa-4(12),5(10),6,8,15(25),16,18-heptaene-2,16-diol 159305 22-cyclopropylmethyl-8-phenyl-14-oxa-11,22-diazaheptacyclo[13.9.1.01,13.02,21.04,12.05,10.019,25]pentacosa-4(12),5(10),6,8,15(25),16,18-heptaene-2,16-diol 159374 22-cyclopropylmethyl-7-[2-(2-pyridyl)-(E)-1-ethenyl]-14-oxa-11,22-diazaheptacyclo[13.9.1.01,13.02,21.04,12.05,10.019,25]pentacosa-4(12),5(10),6,8,15(25),16,18-heptaene-2,16-diol 159375 2-(6-Cyclopentylamino-purin-9-yl)-ethanol 159376 Cyclopentyl-(9-cyclopentyl-9H-purin-6-yl)-amine 159382 Cyclopentyl-[9-(tetrahydro-furan-2-yl)-9H-purin-6-yl]-amine 159388 22-cyclopropylmethyl-7-phenoxy-14-oxa-11,22-diazaheptacyclo[13.9.1.01,13.02,21.04,12.05,10.019,25]pentacosa-4(12),5(10),6,8,15(25),16,18-heptaene-2,16-diol 159393 6-benzyloxy-22-cyclopropylmethyl-14-oxa-11,22-diazaheptacyclo[13.9.1.01,13.02,21.04,12.05,10.019,25]pentacosa-4(12),5(10),6,8,15(25),16,18-heptaene-2,16-diol 159394 22-cyclopropylmethyl-6-phenoxy-14-oxa-11,22-diazaheptacyclo[13.9.1.01,13.02,21.04,12.05,10.019,25]pentacosa-4(12),5(10),6,8,15(25),16,18-heptaene-2,16-diol 159412 22-cyclopropylmethyl-9-phenyl-14-oxa-11,22-diazaheptacyclo[13.9.1.01,13.02,21.04,12.05,10.019,25]pentacosa-4(12),5(10),6,8,15(25),16,18-heptaene-2,16-diol 159418 (2-Chloro-9-methyl-9H-purin-6-yl)-(1-phenyl-propyl)-amine 159425 2-Chloro-9-methyl-9H-purin-6-ylamine 159427 22-cyclopropylmethyl-7-phenyl-14-oxa-11,22-diazaheptacyclo[13.9.1.01,13.02,21.04,12.05,10.019,25]pentacosa-4(12),5(10),6,8,15(25),16,18-heptaene-2,16-diol 159430 4-(3-Chloro-4-fluoro-phenylamino)-7-methoxy-6-(3-morpholin-4-yl-propoxy)-quinoline-3-carbonitrile 159441 (2-Chloro-9-methyl-9H-purin-6-yl)-(1-phenyl-propyl)-amine 159451 9-Oxo-1-propyl-2,3,4a,9,10,10a-hexahydro-1H-4-oxa-9lambda*4*-thia-1-aza-phenanthren-6-ol 159457 N*6*-(4-Chloro-phenyl)-8-isopropyl-N*2*-propyl-9H-purine-2,6-diamine 159489 1-[8-Isopropyl-6-(4-trifluoromethyl-phenylamino)-9H-purin-2-yl]-piperidin-4-ol 159509 Naltrindole analogue 159528 1-[6-(4-Chloro-phenylamino)-8-isopropyl-9H-purin-2-yl]-4-methyl-piperidin-4-ol 159529 4-(4-Chloro-phenylamino)-6-isopropyl-2-morpholin-4-yl-5,6-dihydro-pyrrolo[3,4-d]pyrimidin-7-one 159538 Naltrindole analogue 159539 Cyclohexyl-(9-methyl-9H-purin-6-yl)-amine 159547 8-benzyloxy-22-cyclopropylmethyl-14-oxa-11,22-diazaheptacyclo[13.9.1.01,13.02,21.04,12.05,10.019,25]pentacosa-4(12),5(10),6,8,15(25),16,18-heptaene-2,16-diol 159548 22-cyclopropylmethyl-9-phenoxy-14-oxa-11,22-diazaheptacyclo[13.9.1.01,13.02,21.04,12.05,10.019,25]pentacosa-4(12),5(10),6,8,15(25),16,18-heptaene-2,16-diol 159549 9-benzyloxy-22-cyclopropylmethyl-14-oxa-11,22-diazaheptacyclo[13.9.1.01,13.02,21.04,12.05,10.019,25]pentacosa-4(12),5(10),6,8,15(25),16,18-heptaene-2,16-diol 159554 (4-Chloro-phenyl)-[2-(1,4-dioxa-8-aza-spiro[4.5]dec-8-yl)-8-isopropyl-9H-purin-6-yl]-amine 159555 1-[6-(4-Chloro-phenylamino)-8-isopropyl-9H-purin-2-yl]-piperidin-4-one 159566 (2-Chloro-9-methyl-9H-purin-6-yl)-phenyl-amine 159592 7-benzyloxy-22-cyclopropylmethyl-14-oxa-11,22-diazaheptacyclo[13.9.1.01,13.02,21.04,12.05,10.019,25]pentacosa-4(12),5(10),6,8,15(25),16,18-heptaene-2,16-diol 159693 4-Amino-5-butyl-1-phenyl-1,5-dihydro-pyrazolo[3,4-d]pyrimidin-6-one 159722 4-Amino-1-phenyl-5-propyl-1,5-dihydro-pyrazolo[3,4-d]pyrimidin-6-one 159723 4-Amino-5-ethyl-1-phenyl-1,5-dihydro-pyrazolo[3,4-d]pyrimidin-6-one 159909 Naltrindole analogue 159937 N-[4-(3-Chloro-4-fluoro-phenylamino)-3-cyano-7-(3-morpholin-4-yl-propoxy)-quinolin-6-yl]-acrylamide 159945 (1-Phenyl-propyl)-(9-phenyl-9H-purin-6-yl)-amine 159946 Phenyl-(9-phenyl-9H-purin-6-yl)-amine 159947 (1-Phenyl-propyl)-(9-phenyl-9H-purin-6-yl)-amine 159948 (9-Methyl-9H-purin-6-yl)-phenyl-amine 159958 4-(3-Ethynyl-phenylamino)-6,7-bis-(2-methoxy-ethoxy)-quinoline-3-carbonitrile 159963 Cyclopentyl-(9-phenyl-9H-purin-6-yl)-amine 159973 Cyclohexyl-(9-ethyl-9H-purin-6-yl)-amine 159978 Naltrindole analogue 160006 (cis)1-Propyl-2,3,10,10a-tetrahydro-1H,4aH-4-oxa-9-thia-1-aza-phenanthren-6-ol 160007 (+)-1-Propyl-2,3,10,10a-tetrahydro-1H,4aH-4-oxa-9-thia-1-aza-phenanthren-6-ol 160008 (-)-1-Propyl-2,3,10,10a-tetrahydro-1H,4aH-4-oxa-9-thia-1-aza-phenanthren-6-ol 160016 (trans)1-Propyl-2,3,10,10a-tetrahydro-1H,4aH-4-oxa-9-thia-1-aza-phenanthren-6-ol 160233 3-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-2-methyl-3H-pyrimido[5,4-b]indol-4(5H)-one 160333 4-Amino-1-(3-chloro-phenyl)-5-methyl-1,5-dihydro-pyrazolo[3,4-d]pyrimidin-6-one 160530 (S)-2,9-Dimethoxy-5,8,13,13a-tetrahydro-6H-isoquino[3,2-a]isoquinoline-3,10-diol 161009 1-Oxo-3-phenyl-1H-indene-2-carboxylic acid methyl ester 161107 4-Amino-1-(3-chloro-phenyl)-5-propyl-1,5-dihydro-pyrazolo[3,4-d]pyrimidin-6-one 161108 4-Amino-1,5-diphenyl-1,5-dihydro-pyrazolo[3,4-d]pyrimidin-6-one4-Amino-1-(3-chloro-phenyl)-5-ethyl-1,5-dihydro-pyrazolo[3,4-d]pyrimidin-6-one 161229 SID26751968 161305 3-(3-(ethoxy)-1,2,5-thiadiazol-4-yl)-1,2,5,6-tetrahydro-1-methylpyridine 161348 3-(4-butoxy-1,2,5-thiadiazol-3-yl)-1-methyl-1,2,5,6-tetrahydropyridine 161354 1-methyl-5-(4-(pentyloxy)-1,2,5-thiadiazol-3-yl)-1,2,3,6-tetrahydropyridine 161382 5-(4-Heptyloxy-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2,3,6-tetrahydro-pyridine 161659 (2S,3S)-3-(3,5-Bis-trifluoromethyl-benzyloxy)-1-(1H-imidazol-4-ylmethyl)-2-phenyl-piperidine 161708 (2R,3S)-ethyl 3-(bis(4-fluorophenyl)methoxy)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate 161789 (2S,3S)-3-(3,5-Bis-trifluoromethyl-benzyloxy)-2-phenyl-1-(1H-tetrazol-5-ylmethyl)-piperidine 161805 (5-Methyl-2-phosphono-phenyl)-phosphonic acid 161823 5-[(2S,3S)-3-(3,5-Bis-trifluoromethyl-benzyloxy)-2-phenyl-piperidin-1-ylmethyl]-2,4-dihydro-[1,2,4]triazole-3-thione 161824 (2S,3S)-3-(3,5-Bis-trifluoromethyl-benzyloxy)-1-furan-2-ylmethyl-2-phenyl-piperidine 162216 cis-(-)-7,8-dimethoxy-3-[4-(2-methyl-3-(4-fluoro)phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole 162263 (2S,3S)-3-(3,5-Bis-trifluoromethyl-benzyloxy)-1-(1H-imidazol-2-ylmethyl)-2-phenyl-piperidine 162275 (2S,3S)-3-(3,5-Bis-trifluoromethyl-benzyloxy)-1-oxazol-4-ylmethyl-2-phenyl-piperidine 162293 2-[6-Amino-2-((E)-hex-1-enyl)-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 162302 (2S,3S)-3-(3,5-Bis-trifluoromethyl-benzyloxy)-1-[1,3,4]oxadiazol-2-ylmethyl-2-phenyl-piperidine 162482 2-{6-Amino-2-[4-(4-methoxy-phenyl)-pyrazol-1-yl]-purin-9-yl}-5-hydroxymethyl-tetrahydro-furan-3,4-diol 162497 2,6-Diamino-hexanoic acid (1-tridecanoyl-piperidin-2-ylmethyl)-amide 162546 1-[6-Amino-9-(3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-2-yl]-1H-pyrazole-4-carboxylic acid methylamide 162599 2-[6-Amino-2-(1-benzyl-1H-pyrazol-4-yl)-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 162714 5-[(2S,3S)-3-(3,5-Bis-trifluoromethyl-benzyloxy)-2-phenyl-piperidin-1-ylmethyl]-2,4-dihydro-[1,2,4]triazol-3-one 162730 (2R,3R,4S,5R)-2-(6-amino-2-(hex-1-ynyl)-9H-purin-9-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol 162765 2-{6-Amino-2-[2-(4-methoxy-phenyl)-ethylamino]-purin-9-yl}-5-hydroxymethyl-tetrahydro-furan-3,4-diol 162789 1'-[2-(2-pyridyl)ethyl]spiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)]-4-one 162790 1'-[2-(1-naphthyl)ethyl]spiro[3,4-dihydro-1H-isochromene-3,4'-(hexahydropyridine)]-1-one 162847 (2-Chloro-5-trifluoromethyl-phenyl)-imidazolidin-2-ylidene-amine (St-587) 162990 7'-methylspiro[4,5-dihydro-1H-imidazole-4,2'-(1',2',3',4'-tetrahydronaphthalene)] 163008 (3,4-Dimethoxy-phenyl)-(6,7-dimethoxy-quinolin-4-yl)-amine 163263 1'-[2-(1-naphthyl)ethyl]spiro[2H-chromene-2,4'-(hexahydropyridine)] 163269 4-(3-Bromo-phenoxy)-6,7-dimethoxy-quinoline 163291 (3,4-Dimethoxy-phenyl)-(6,7-dimethoxy-quinazolin-4-yl)-amine 163294 N-[1'-[2-(1-naphthyl)ethyl]-4-oxospiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)]-7-yl]methanesulfonamide 163372 N-[4-oxo-1'-[2-(2-pyridyl)ethyl]spiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)]-7-yl]methanesulfonamide 163382 4-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-yl)-(3-methoxy-phenyl)-methyl]-N-ethyl-benzamide 163433 6-(3,5-dimethyl-4-isoxazolylsulfonamido)-1'-[2-(1-naphthyl)ethyl]-4-oxospiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)] 163437 N-[1'-[2-(1-naphthyl)ethyl]-4-oxospiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)]-6-yl]phenylmethanesulfonamide 163465 6-(1-methyl-1H-4-imidazolylsulfonamido)-1'-[2-(1-naphthyl)ethyl]-4-oxospiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)] 163466 N-[4-oxo-1'-[2-(2-pyridyl)ethyl]spiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)]-6-yl]methanesulfonamide 163496 N-[1'-[2-(2-methyl-1H-3-indolyl)ethyl]-4-oxospiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)]-7-yl]methanesulfonamide 163498 N-[1'-(2-methoxyphenethyl)-4-oxospiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)]-7-yl]methanesulfonamide 163503 1'-[2-(1-naphthyl)ethyl]spiro[2,3-dihydro-1H-indene-2,4'-(hexahydropyridine)]-1-one 163553 1'-[2-(1-naphthyl)ethyl]spiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)] 163585 (3-Bromo-phenyl)-(6,7-dimethoxy-quinolin-4-yl)-amine 163608 1-Aminomethyl-isochroman-5,6-diol 163617 4-(3-bromophenoxy)-6,7-dimethoxyquinazoline 163626 N-(5-phenylthiazol-2-yl)-5-(pyrrolidin-1-ylmethyl)pyridin-2-amine 163716 Phenyl-(5-phenyl-oxazol-2-yl)-amine 163722 1'-[2-(1-naphthyl)ethyl]spiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)]-4-one 163804 Tyr-D-Ala-Phe-Glu-Val-Val-Gly-NH2 163825 Acetic acid (R)-4-decyloxy-1-hydroxymethyl-3-oxo-1,3-dihydro-isobenzofuran-1-ylmethyl ester 163855 Acetic acid (R)-4-dodecyloxy-1-hydroxymethyl-3-oxo-1,3-dihydro-isobenzofuran-1-ylmethyl ester 163857 Acetic acid (S)-4-dodecyloxy-1-hydroxymethyl-3-oxo-1,3-dihydro-isobenzofuran-1-ylmethyl ester 163885 Acetic acid (S)-4-decyloxy-1-hydroxymethyl-3-oxo-1,3-dihydro-isobenzofuran-1-ylmethyl ester 163971 But-3-enoic acid (R)-1-acetoxymethyl-1-hydroxymethyl-3-oxo-1,3-dihydro-isobenzofuran-4-yl ester 163978 3-{1-[1-aminobutyl oxycarbonylamino-2-(1H-3-indolyl)ethylcarboxamido]-5-formamido-ortho-methoxy phenylaminopentylcarboxamido}-3-(1-carbamoyl-2-phenylethylcarbamoyl)propanoic acid 163980 2,2-Dimethyl-propionic acid (S)-4-dodecyloxy-1-hydroxymethyl-3-oxo-1,3-dihydro-isobenzofuran-1-ylmethyl ester 163981 Acetic acid (R)-4-benzyloxy-1-hydroxymethyl-3-oxo-1,3-dihydro-isobenzofuran-1-ylmethyl ester 163998 1-Aminomethyl-3-cyclohexyl-isochroman-5,6-diol 164011 Octanoic acid (S)-2-acetoxy-3-hydroxy-propyl ester 164031 3-{(S)-2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-6-[3-(2-chloro-phenyl)-ureido]-hexanoylamino}-N-(1-carbamoyl-2-phenyl-ethyl)-succinamic acid 164043 (S)-3-[(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-6-(3-o-tolyl-ureido)-hexanoylamino]-N-((S)-1-carbamoyl-2-phenyl-ethyl)-succinamic acid 164063 3-{1-[1-aminobutyl oxycarbonylamino-2-(1H-3-indolyl)ethylcarboxamido]-5-formamido-para-methyl phenylaminopentylcarboxamido}-3-(1-carbamoyl-2-phenylethylcarbamoyl)propanoic acid 164064 sincalide 164065 3-[2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-6-(3-o-tolyl-ureido)-hexanoylamino]-N-(1-carbamoyl-2-phenyl-ethyl)-N-methyl-succinamic acid 164078 3-{1-[1-aminobutyl oxycarbonylamino-2-(1H-3-indolyl)ethylcarboxamido]-5-formamidometa-methyl phenylaminopentylcarboxamido}-3-(1-carbamoyl-2-phenylethylcarbamoyl)propanoic acid 164088 3-[1-(3,5-Dichloro-phenyl)-ethoxy]-2-phenyl-piperidine 164135 7-{3-[4-(4-Fluoro-benzoyl)-piperidin-1-yl]-propoxy}-3-methyl-chromen-4-one 164236 2-(8-Bromo-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']difuran-4-yl)-1-methyl-ethylamine 164246 7-{3-[4-(4-Fluoro-benzoyl)-piperidin-1-yl]-propoxy}-3-hydroxymethyl-chromen-4-one 164345 3-[1-(3,5-Bis-trifluoromethyl-phenyl)-ethoxy]-2-phenyl-piperidine 164379 (6aR,12bR)-6-Methyl-5,6,6a,7,8,12b-hexahydro-benzo[a]phenanthridine-9,10-diol 164404 SID26751954 164463 N-[4-Phenyl-2-(5-phenyl-pyridin-3-yl)-oxazol-5-yl]-acetamide 164491 N-[2-(3-Hydroxy-naphthalen-2-yl)-4-phenyl-oxazol-5-yl]-acetamide 164493 N-{2-[5-(3-Fluoro-phenyl)-pyridin-3-yl]-4-phenyl-oxazol-5-yl}-acetamide 164637 (2S,3S)-3-(3,5-Bis-trifluoromethyl-benzyloxy)-2-phenyl-1-(4H-[1,2,4]triazol-3-ylmethyl)-piperidine 164638 5-{3-[1-(3,5-Dichloro-phenyl)-ethoxy]-2-phenyl-piperidin-1-ylmethyl}-2,4-dihydro-[1,2,4]triazol-3-one 164658 5-{3-[1-(3,5-Dichloro-phenyl)-ethoxy]-2-phenyl-piperidin-1-ylmethyl}-2,4-dihydro-[1,2,4]triazol-3-one 164670 2-Phenyl-3-(1-phenyl-ethoxy)-piperidine 164674 5-{3-[1-(3,5-Dichloro-phenyl)-ethoxy]-2-phenyl-piperidin-1-ylmethyl}-2,4-dihydro-[1,2,4]triazol-3-one 164686 5-{3-[1-(3,5-Bis-trifluoromethyl-phenyl)-ethoxy]-2-phenyl-piperidin-1-ylmethyl}-2,4-dihydro-[1,2,4]triazol-3-one 164688 3-[1-(3,5-Bis-trifluoromethyl-phenyl)-ethoxy]-2-phenyl-1-(1H-[1,2,4]triazol-3-ylmethyl)-piperidine 164814 3-[1-(3,5-Dichloro-phenyl)-ethoxy]-2-phenyl-piperidine 164838 3-[1-(3,5-Bis-trifluoromethyl-phenyl)-ethoxy]-2-phenyl-piperidine 164841 3-Benzyloxy-2-phenyl-piperidine 164875 (4aR,8aR)-4a-(3-Hydroxy-phenyl)-3,7-dimethyl-4,4a,5,6,7,8,8a,9-octahydro-1H-pyrrolo[3,2-g]isoquinoline-2-carboxylic acid diethylamide 164877 (4aR,8aS)-6-Ethyl-8a-(3-hydroxy-phenyl)-3-methyl-4,4a,5,6,7,8,8a,9-octahydro-1H-pyrrolo[2,3-g]isoquinoline-2-carboxylic acid diisopropylamide 164915 (4aR,8aS)-6-Ethyl-8a-(3-hydroxy-phenyl)-3-methyl-4,4a,5,6,7,8,8a,9-octahydro-1H-pyrrolo[2,3-g]isoquinoline-2-carboxylic acid diethylamide 165012 Vatalanib 165158 (4aR,8aS)-6-Ethyl-8a-(3-hydroxy-phenyl)-3-methyl-4,4a,5,6,7,8,8a,9-octahydro-1H-pyrrolo[2,3-g]isoquinoline-2-carboxylic acid amide 165184 4-(2,4-Dichloro-phenylamino)-6,7-dimethoxy-quinoline-3-carbonitrile 165209 (4aR,8aR)-7-Ethyl-4a-(3-hydroxy-phenyl)-3-methyl-4,4a,5,6,7,8,8a,9-octahydro-1H-pyrrolo[3,2-g]isoquinoline-2-carboxylic acid ethyl ester 165210 (4aR,8aR)-7-Ethyl-4a-(3-hydroxy-phenyl)-3-methyl-4,4a,5,6,7,8,8a,9-octahydro-1H-pyrrolo[3,2-g]isoquinoline-2-carbothioic acid diethylamide 165211 3-((4aS,12aR)-2-methyl-1,2,3,4,4a,5,12,12a-octahydropyrido[3,4-b]acridin-4a-yl)phenol 165265 Dimethyl-{3-[3-(5-thiophen-3-yl-pyridin-3-yl)-indol-1-yl]-propyl}-amine 165286 Dimethyl-{2-[3-(5-thiophen-3-yl-pyridin-3-yl)-indol-1-yl]-ethyl}-amine 165302 Dimethyl-{2-methyl-3-[3-(5-thiophen-3-yl-pyridin-3-yl)-indol-1-yl]-propyl}-amine 165303 1-(3-(4-methylpiperazin-1-yl)propyl)-3-(5-(thiophen-3-yl)pyridin-3-yl)-1H-indole 165310 N-{2-[5-(3-Methoxy-phenyl)-pyridin-3-yl]-4-phenyl-oxazol-5-yl}-acetamide 165317 N-{2-[5-(4-Methoxy-phenyl)-pyridin-3-yl]-4-phenyl-oxazol-5-yl}-acetamide 165318 N-{2-[5-(3-Chloro-phenyl)-pyridin-3-yl]-4-phenyl-oxazol-5-yl}-acetamide 165319 N-[4-Phenyl-2-(5-thiophen-3-yl-pyridin-3-yl)-oxazol-5-yl]-acetamide 165340 3-(5-Thiophen-3-yl-pyridin-3-yl)-1H-indole 165344 1-(2-Piperidin-1-yl-ethyl)-3-(5-thiophen-3-yl-pyridin-3-yl)-1H-indole 165355 (4aR,8aS)-6-Ethyl-8a-(3-hydroxy-phenyl)-3-methyl-4,4a,5,6,7,8,8a,9-octahydro-1H-pyrrolo[2,3-g]isoquinoline-2-carboxylic acid dimethylamide 165372 1-(2-Morpholin-4-yl-ethyl)-3-(5-thiophen-3-yl-pyridin-3-yl)-1H-indole 165385 1-(3-Piperidin-1-yl-propyl)-3-(5-thiophen-3-yl-pyridin-3-yl)-1H-indole 165469 2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid 3-ethyl ester 5-methyl ester 165584 2,4-Dimethyl-6-phenyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid diethyl ester 165749 4-(2,4-dichloro-5-methoxyphenylamino)-7-(4-((4-methylpiperazin-1-yl)methyl)phenyl)quinoline-3-carbonitrile 165774 SID11112188 165870 1-(1-Cyclohexylmethyl-4-phenyl-pyrrolidin-3-ylmethyl)-4-{3-[4-(1-methyl-1H-tetrazol-5-yl)-phenyl]-propyl}-piperidin-4-ol 165965 2-(4-(3-(1-(((3S,4S)-1-(cyclohexylmethyl)-4-phenylpyrrolidin-3-yl)methyl)-4-hydroxypiperidin-4-yl)propyl)phenyl)acetic acid 165967 4-(3-(1-(((3S,4S)-1-(cyclohexylmethyl)-4-phenylpyrrolidin-3-yl)methyl)-4-hydroxypiperidin-4-yl)propyl)benzoic acid 166055 4-(3-(4-(1H-tetrazol-5-yl)phenyl)propyl)-1-(((3S,4S)-1-(cyclohexylmethyl)-4-phenylpyrrolidin-3-yl)methyl)piperidin-4-ol 166060 4-(5-{3-[3-(2-Fluoro-5-trifluoromethyl-phenyl)-ureido]-phenyl}-2H-pyrazol-3-ylamino)-benzenesulfonamide 166083 4-[5-(3-Benzenesulfonylamino-phenyl)-2H-pyrazol-3-ylamino]-benzenesulfonamide 166086 4-[5-(3-Methanesulfonylamino-phenyl)-2H-pyrazol-3-ylamino]-benzenesulfonamide 166116 4-[5-(3-Hydroxy-phenyl)-2H-pyrazol-3-ylamino]-benzenesulfonamide 166117 4-[5-(3-Methoxy-phenyl)-2H-pyrazol-3-ylamino]-benzenesulfonamide 166118 4-[5-(4-Amino-phenyl)-2H-pyrazol-3-ylamino]-benzenesulfonamide 166119 4-[5-(3-Fluoro-4-hydroxy-phenyl)-2H-pyrazol-3-ylamino]-benzenesulfonamide 166134 4-[5-(4-Bromo-phenyl)-2H-pyrazol-3-ylamino]-benzenesulfonamide 166184 4-Ethyl-2,6-dimethyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid 3-ethyl ester 5-methyl ester 166217 5-(4-{3-[1-((3S,4S)-1-Cyclohexylmethyl-4-phenyl-pyrrolidin-3-ylmethyl)-4-hydroxy-piperidin-4-yl]-propyl}-phenyl)-2-methyl-1H-tetrazol-2-ium 166349 2-[4-(5-Methyl-2-phenyl-3H-imidazol-4-ylmethyl)-piperazin-1-yl]-pyrimidine 166358 2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid 3-benzyl ester 5-methyl ester 166379 2-[4-(2-Phenyl-3H-imidazol-4-ylmethyl)-piperazin-1-yl]-pyrimidine (NGD-94-1) 166424 4-[4-(2-Phenyl-3H-imidazol-4-ylmethyl)-piperazin-1-yl]-pyrimidine 166464 4-(2-Phenyl-3H-imidazol-4-ylmethyl)-3,4,5,6-tetrahydro-2H-[1,2']bipyrazinyl 166497 1-(2-Phenyl-3H-imidazol-4-ylmethyl)-4-pyridin-3-yl-piperazine 166538 SID26726578 166687 Cyclohexyl-{3-phenyl-4-[4-(3-phenyl-propyl)-piperidin-1-ylmethyl]-pyrrolidin-1-yl}-acetic acid 166820 3-(3-(1-(((3S,4S)-1-(cyclohexylmethyl)-4-phenylpyrrolidin-3-yl)methyl)-4-hydroxypiperidin-4-yl)propyl)benzoic acid 166953 2-[4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-5-oxo-3-(3,4,5-trimethoxy-benzyl)-2,5-dihydro-furan-2-yloxycarbonylamino]-3-methyl-butyric acid ethyl ester 166954 3-[4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-5-oxo-3-(3,4,5-trimethoxy-benzyl)-2,5-dihydro-furan-2-yloxycarbonylamino]-propionic acid ethyl ester 166972 Allyl-carbamic acid 4-benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-5-oxo-3-(3,4,5-trimethoxy-benzyl)-2,5-dihydro-furan-2-yl ester 166973 ((S)-1-Phenyl-ethyl)-carbamic acid 4-benzo[1,3]dioxol-5-yl-3-benzyl-2-(4-methoxy-phenyl)-5-oxo-2,5-dihydro-furan-2-yl ester 167044 1-((3S,4S)-1-Cyclohexylmethyl-4-phenyl-pyrrolidin-3-ylmethyl)-4-(3-phenyl-propyl)-piperidin-4-ol 167067 1-(((3S,4S)-1-(cyclohexylmethyl)-4-phenylpyrrolidin-3-yl)methyl)-4-(3-(pyridin-3-yl)propyl)piperidin-4-ol 167144 1-phenyl-4-((2-phenyl-1H-imidazol-4-yl)methyl)piperazine 167149 2-(3-(3-(1-(((3S,4S)-1-(cyclohexylmethyl)-4-phenylpyrrolidin-3-yl)methyl)-4-hydroxypiperidin-4-yl)propyl)phenyl)acetic acid 167150 3-(4-{3-[1-(1-Cyclohexylmethyl-4-phenyl-pyrrolidin-3-ylmethyl)-4-hydroxy-piperidin-4-yl]-propyl}-phenyl)-propionic acid 167151 1-(1-Cyclohexylmethyl-4-phenyl-pyrrolidin-3-ylmethyl)-4-{3-[4-(1H-tetrazol-5-ylmethyl)-phenyl]-propyl}-piperidin-4-ol 167168 1-(((3S,4S)-1-(cyclohexylmethyl)-4-phenylpyrrolidin-3-yl)methyl)-4-(3-(pyridin-2-yl)propyl)piperidin-4-ol 167202 1-(1-Cyclohexylmethyl-4-phenyl-pyrrolidin-3-ylmethyl)-4-(3-pyridin-4-yl-propyl)-piperidin-4-ol 167221 2-[4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-5-oxo-3-(3,4,5-trimethoxy-benzyl)-2,5-dihydro-furan-2-yloxycarbonylamino]-4-methyl-pentanoic acid ethyl ester 167222 ((S)-1-Naphthalen-1-yl-ethyl)-carbamic acid 4-benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-5-oxo-3-(3,4,5-trimethoxy-benzyl)-2,5-dihydro-furan-2-yl ester 167262 2-(3-(1-(((3S,4S)-1-(cyclohexylmethyl)-4-phenylpyrrolidin-3-yl)methyl)-4-hydroxypiperidin-4-yl)propyl)benzoic acid 167340 Methyl-carbamic acid 4-benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-5-oxo-3-(3,4,5-trimethoxy-benzyl)-2,5-dihydro-furan-2-yl ester 167341 [4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-5-oxo-3-(3,4,5-trimethoxy-benzyl)-2,5-dihydro-furan-2-yloxycarbonylamino]-acetic acid ethyl ester 167537 5-[2-(2,5-Dihydroxy-phenyl)-vinyl]-2-hydroxy-benzoic acid 167574 5-[2-(3,4-Dihydroxy-phenyl)-vinyl]-2-hydroxy-benzoic acid 167575 5-[2-(2,5-Dihydroxy-phenyl)-ethyl]-2-hydroxy-benzoic acid 167576 SID26755753 167577 SID26756741 167581 5-[2-(3,4-Dihydroxy-phenyl)-ethyl]-2-hydroxy-benzoic acid 167582 5-{[1-(2,5-Dihydroxy-phenyl)-meth-(E)-ylidene]-amino}-2-hydroxy-benzoic acid 167687 5-(6,7-Dihydroxy-naphthalen-2-yl)-2-hydroxy-benzoic acid 167718 5-(5,8-Dihydroxy-naphthalen-2-yl)-2-hydroxy-benzoic acid 167735 N-[4-(4-Hydroxy-7-methyl-[1,8]naphthyridin-2-yl)-phenyl]-acetamide 167746 3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sulfo-phenyl)-propionylamino]-hexanoylamino}-acetylamino)-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-N-phenethyl-succinamic acid 167747 2-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sulfo-phenyl)-propionylamino]-hexanoylamino}-acetylamino)-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-succinic acid 1-phenethyl ester 167759 Opioid Peptide [d-Ala(8)]Dynorphin derivative 167878 5-(5,6-Dihydroxy-naphthalen-2-yl)-2-hydroxy-benzoic acid 167940 7-methyl-2-propyl-1,8-naphthyridin-4-ol 167995 Doramapimod 167999 3-[[3-((3-{(2-Amino-ethyl)-[3-(bis-{3-[bis-(2-cyano-ethyl)-amino]-propyl}-amino)-propyl]-amino}-propyl)-{3-[bis-(2-cyano-ethyl)-amino]-propyl}-amino)-propyl]-(2-cyano-ethyl)-amino]-propionitrile 168006 1-(2-{Bis-[3-(bis-{3-[bis-(3-amino-propyl)-amino]-propyl}-amino)-propyl]-amino}-ethyl)-3,4-diphenyl-pyrrole-2,5-dione 168007 3-[[3-((3-{[2-(5-Amino-1,3-dioxo-1H,3H-benzo[de]isoquinolin-2-yl)-ethyl]-[3-(bis-{3-[bis-(2-cyano-ethyl)-amino]-propyl}-amino)-propyl]-amino}-propyl)-{3-[bis-(2-cyano-ethyl)-amino]-propyl}-amino)-propyl]-(2-cyano-ethyl)-amino]-propionitrile 168136 7-(dimethylamino)-2-phenyl-1,8-naphthyridin-4-ol 168177 1-[5-(4-Methyl-piperazin-1-yl)-2-oxo-1-propyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl]-3-m-tolyl-urea 168205 1-[5-(4-Methyl-piperazin-1-yl)-2-oxo-1-propyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl]-3-(3-trifluoromethyl-phenyl)-urea 168213 1-[5-(4-Methyl-piperazin-1-yl)-2-oxo-1-propyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl]-3-(3-propyl-phenyl)-urea 168226 1-((2S,4R)-2-Methyl-6-phenyl-2,4-dihydro-1H-3,5,10b-triaza-benzo[e]azulen-4-yl)-3-m-tolyl-urea 168255 1-[(S)-5-(4-Methyl-piperazin-1-yl)-2-oxo-1-propyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl]-3-m-tolyl-urea 168269 1-[1-Methyl-5-(4-methyl-piperazin-1-yl)-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl]-3-m-tolyl-urea 168281 3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-{[(tert-butoxy)carbonyl]amino}-3-(4-sulfophenyl)propanamido]hexanamido]acetamido}-3-(1H-indol-3-yl)propanamido]hexanamido]-6-phenoxyhexanoic acid 168282 3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sulfo-phenyl)-propionylamino]-hexanoylamino}-acetylamino)-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-7-phenyl-heptanoic acid 168338 3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sulfo-phenyl)-propionylamino]-hexanoylamino}-acetylamino)-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-7-phenyl-heptanoic acid 168421 3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-{[(tert-butoxy)carbonyl]amino}-3-(4-sulfophenyl)propanamido]hexanamido]acetamido}-3-(1H-indol-3-yl)propanamido]hexanamido]-6-phenoxyhexanoic acid 168422 3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sulfo-phenyl)-propionylamino]-hexanoylamino}-acetylamino)-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-7-phenyl-heptanoic acid 168483 2-(2-{Bis-[3-(bis-{3-[bis-(3-amino-propyl)-amino]-propyl}-amino)-propyl]-amino}-ethyl)-benzo[de]isoquinoline-1,3-dione 168492 3-[[3-((3-{[3-(Bis-{3-[bis-(2-cyano-ethyl)-amino]-propyl}-amino)-propyl]-[2-(5-nitro-1,3-dioxo-1H,3H-benzo[de]isoquinolin-2-yl)-ethyl]-amino}-propyl)-{3-[bis-(2-cyano-ethyl)-amino]-propyl}-amino)-propyl]-(2-cyano-ethyl)-amino]-propionitrile 168508 3-[(2S)-2-[(2R)-2-{2-[(2S)-2-[(2S)-2-{[(tert-butoxy)carbonyl]amino}-3-(4-sulfophenyl)propanamido]hexanamido]acetamido}-3-(1H-indol-3-yl)propanamido]hexanamido]-6-phenoxyhexanoic acid 168509 3-[(2S)-2-[(2R)-2-{2-[(2S)-2-[(2S)-2-{[(tert-butoxy)carbonyl]amino}-3-(4-sulfophenyl)propanamido]hexanamido]acetamido}-3-(1H-indol-3-yl)propanamido]hexanamido]-6-phenoxyhexanoic acid 168510 3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sulfo-phenyl)-propionylamino]-hexanoylamino}-acetylamino)-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-7-phenyl-heptanoic acid 168538 3-((1-methyl-1H-pyrrol-2-yl)methylene)indolin-2-one 168571 (1-Phenyl-ethyl)-(9H-2,4,9-triaza-fluoren-1-yl)-amine 168596 11-{2-[(Octahydro-quinolizin-1-ylmethyl)-amino]-acetyl}-5,11-dihydro-benzo[e]pyrido[3,2-b][1,4]diazepin-6-one 168637 11-[2-(Octahydro-quinolizin-1-ylmethylsulfanyl)-acetyl]-5,11-dihydro-benzo[e]pyrido[3,2-b][1,4]diazepin-6-one 168691 4-(3-chloro-4-(1-methyl-1H-imidazol-2-ylthio)phenylamino)-6-methoxy-7-(3-morpholinopropoxy)quinoline-3-carbonitrile 168698 N-(4-Benzoyl-2-methyl-phenyl)-2-(R)-octahydro-quinolizin-1-yl-acetamide 168722 (1-Phenyl-ethyl)-(9H-2,4,9-triaza-fluoren-1-yl)-amine 168890 (1-Phenyl-ethyl)-(6-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)-amine 169038 11-((S)-2-Octahydro-quinolizin-1-yl-thioacetyl)-5,11-dihydro-benzo[e]pyrido[3,2-b][1,4]diazepin-6-one 169097 Benzo[4,5]thieno[3,2-d]pyrimidin-4-yl-(1-phenyl-ethyl)-amine 169151 20-methyl-17,23-dioxa-4,14,20,26-tetraazahexacyclo[24.6.1.17,14.02,6.08,13.027,32]tetratriaconta-1(33),2(6),7(34),8(13),9,11,27(32),28,30-nonaene-3,5-dione 169152 20-(2-hydroxyethyl)-17,23-dioxa-4,14,20,26-tetraazahexacyclo[24.6.1.17,14.02,6.08,13.027,32]tetratriaconta-1(33),2(6),7(34),8(13),9,11,27(32),28,30-nonaene-3,5-dione 169168 (-)2-(2,5-Dimethoxy-4-methyl-phenyl)-1-methyl-ethylamine 169223 17,20,23-trimethyl-4,14,17,20,23,26-hexaazahexacyclo[24.6.1.17,14.02,6.08,13.027,32]tetratriaconta-1(33),2(6),7(34),8(13),9,11,27(32),28,30-nonaene-3,5-dione 169235 (R)-2-Methyl-6-phenyl-4-phenylethynyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid 3-((R)-2,2-dimethyl-[1,3]dioxolan-4-ylmethyl) ester 5-ethyl ester 169237 (S)-2-Methyl-6-phenyl-4-phenylethynyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid 5-benzyl ester 3-ethyl ester 169258 SID26755016 169346 (R)-2-Methyl-6-phenyl-4-phenylethynyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid 5-benzyl ester 3-ethyl ester 169457 SID26755655 169526 Benzyl-quinazolin-4-yl-amine 169852 1-(1-(2-(isopropyl(phenyl)amino)-2-oxoethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-3-yl)-3-phenylurea 169857 17,26-dimethyl-20,23-dioxa-4,14,17,26,29-pentaazahexacyclo[27.6.1.17,14.02,6.08,13.030,35]heptatriaconta-1(36),2(6),7(37),8(13),9,11,30(35),31,33-nonaene-3,5-dione 169917 20,23-dimethyl-17-oxa-4,14,20,23,26-pentaazahexacyclo[24.6.1.17,14.02,6.08,13.027,32]tetratriaconta-1(33),2(6),7(34),8(13),9,11,27(32),28,30-nonaene-3,5-dione 169920 3-(1-{2-[2-(2-Dimethylamino-ethoxy)-ethoxy]-ethyl}-1H-indol-3-yl)-4-(1-propyl-1H-indol-3-yl)-pyrrole-2,5-dione 169947 (S)-2-Methyl-6-phenyl-4-phenylethynyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid 3-((R)-2,2-dimethyl-[1,3]dioxolan-4-ylmethyl) ester 5-ethyl ester 169961 17,20-dimethyl-4,14,17,20,23-pentaazahexacyclo[21.6.1.17,14.02,6.08,13.024,29]hentriaconta-1(30),2(6),7(31),8(13),9,11,24(29),25,27-nonaene-3,5-dione 169962 SID11114153 169981 20,26-diethyl-17,23-dioxa-4,14,20,26,29-pentaazahexacyclo[27.6.1.17,14.02,6.08,13.030,35]heptatriaconta-1(36),2(6),7(37),8(13),9,11,30(35),31,33-nonaene-3,5-dione 169993 20-ethyl-17,23-dioxa-4,14,20,26-tetraazahexacyclo[24.6.1.1^{7,14}.0^{2,6}.0^{8,13}.0^{27,32}]tetratriaconta-1(33),2(6),7(34),8(13),9,11,27(32),28,30-nonaene-3,5-dione 170112 17,23-dimethyl-20-oxa-4,14,17,23,26-pentaazahexacyclo[24.6.1.17,14.02,6.08,13.027,32]tetratriaconta-1(33),2(6),7(34),8(13),9,11,27(32),28,30-nonaene-3,5-dione 170144 23-ethyl-17,20-dioxa-4,14,23,26-tetraazahexacyclo[24.6.1.17,14.02,6.08,13.027,32]tetratriaconta-1(33),2(6),7(34),8(13),9,11,27(32),28,30-nonaene-3,5-dione 170204 1-[3,5-di(trifluoromethyl)benzoyl]-5'-methyl-2'-(2-thienylmethyl)spiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole]-4',6'-dione 170218 1-[3,5-di(trifluoromethyl)benzoyl]-2'-[2-(1,4-oxazinan-4-yl)acetyl]-5'-phenylspiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole]-4',6'-dione 170219 2'-(3,4-dimethoxybenzoyl)-5'-[3,5-di(trifluoromethyl)benzyl]spiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole]-4',6'-dione 170220 1-acetyl-2'-[3,5-di(trifluoromethyl)benzoyl]-5'-phenylspiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole]-4',6'-dione 170229 ({4-[6-(2,6-Dichloro-phenyl)-8-methyl-7-oxo-7,8-dihydro-pyrido[2,3-d]pyrimidin-2-ylamino]-phenyl}-hydroxy-phosphinoylmethyl)-phosphonic acid 170242 ({4-[6-(2,6-Dichloro-phenyl)-8-methyl-7-oxo-7,8-dihydro-pyrido[2,3-d]pyrimidin-2-ylamino]-benzyl}-hydroxy-phosphinoylmethyl)-phosphonic acid 170243 {5-[6-(2,6-Dichloro-phenyl)-8-methyl-7-oxo-7,8-dihydro-pyrido[2,3-d]pyrimidin-2-ylamino]-2-phosphono-phenyl}-phosphonic acid 170244 {4-[6-(2,6-Dichloro-phenyl)-8-methyl-7-oxo-7,8-dihydro-pyrido[2,3-d]pyrimidin-2-ylamino]-2-phosphono-phenoxy}-acetic acid 170275 8-(4-Oxo-1-phenyl-1,3,8-triaza-spiro[4.5]dec-8-ylmethyl)-7,8-dihydro-3H-6,9-dioxa-3-aza-cyclopenta[a]naphthalene-2-carboxylic acid butyl ester 170276 8-(4-Oxo-1-phenyl-1,3,8-triaza-spiro[4.5]dec-8-ylmethyl)-7,8-dihydro-3H-6,9-dioxa-3-aza-cyclopenta[a]naphthalene-2-carbonitrile 170284 ({4-[6-(2,6-Dichloro-phenyl)-8-(3-dimethylamino-propyl)-7-oxo-7,8-dihydro-pyrido[2,3-d]pyrimidin-2-ylamino]-phenyl}-hydroxy-phosphinoylmethyl)-phosphonic acid 170318 ({3-[6-(2,6-Dichloro-phenyl)-8-methyl-7-oxo-7,8-dihydro-pyrido[2,3-d]pyrimidin-2-ylamino]-phenyl}-hydroxy-phosphinoylmethyl)-phosphonic acid 170328 4-Fluoro-N-[3-(1-methyl-4-piperidinyl)-1H-indol-5-yl]benzamide 170343 2'-(3-chlorobenzo[b]thiophen-2-ylcarbonyl)-5'-[3,5-di(trifluoromethyl)benzyl]spiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole]-4',6'-dione 170344 1-[3,5-di(trifluoromethyl)benzoyl]-2'-(2-methoxybenzoyl)-5'-methylspiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole]-4',6'-dione 170358 5'-[3,5-di(trifluoromethyl)benzyl]-1-methylsulfonyl-2'-(2-naphthylcarbonyl)spiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole]-4',6'-dione 170359 8-[(3-Phenyl-propylamino)-methyl]-7,8-dihydro-3H-6,9-dioxa-3-aza-cyclopenta[a]naphthalene-2-carboxylic acid (3-phenyl-propyl)-amide 170360 8-[(3-Phenyl-propylamino)-methyl]-7,8-dihydro-3H-6,9-dioxa-3-aza-cyclopenta[a]naphthalene-2-carboxylic acid methyl ester 170362 8-(4-Ethoxycarbonyl-piperidin-1-ylmethyl)-7,8-dihydro-3H-6,9-dioxa-3-aza-cyclopenta[a]naphthalene-2-carboxylic acid methyl ester 170385 8-[4-(2-Oxo-2,3-dihydro-benzoimidazol-1-yl)-piperidin-1-ylmethyl]-7,8-dihydro-3H-6,9-dioxa-3-aza-cyclopenta[a]naphthalene-2-carboxylic acid methyl ester 170411 1-(3,5-dimethyl-4-isoxazolylsulfonyl)-2'-[3,5-di(trifluoromethyl)benzoyl]-5'-phenylspiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole]-4',6'-dione 170419 8-(2-Hydroxymethyl-7,8-dihydro-3H-6,9-dioxa-3-aza-cyclopenta[a]naphthalen-8-ylmethyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 170436 1-[3,5-di(trifluoromethyl)benzoyl]-5'-methyl-2'-(2-naphthylsulfonyl)spiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole]-4',6'-dione 170454 1-acetyl-2'-(2-benzyloxyacetyl)-5'-[3,5-di(trifluoromethyl)benzyl]spiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole]-4',6'-dione 170455 2'-(2-benzyloxyacetyl)-5'-[3,5-di(trifluoromethyl)benzyl]spiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole]-4',6'-dione 170456 2'-[3,5-di(trifluoromethyl)benzoyl]-1-(3-oxo-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-ylsulfonyl)-5'-phenylspiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole]-4',6'-dione 170477 8-(4-Oxo-1-phenyl-1,3,8-triaza-spiro[4.5]dec-8-ylmethyl)-7,8-dihydro-3H-6,9-dioxa-3-aza-cyclopenta[a]naphthalene-2-carboxylic acid amide 170478 8-(4-Oxo-1-phenyl-1,3,8-triaza-spiro[4.5]dec-8-ylmethyl)-7,8-dihydro-3H-6,9-dioxa-3-aza-cyclopenta[a]naphthalene-2-carboxylic acid 170485 8-(4-Oxo-1-phenyl-1,3,8-triaza-spiro[4.5]dec-8-ylmethyl)-7,8-dihydro-3H-6,9-dioxa-3-aza-cyclopenta[a]naphthalene-2-carboxylic acid benzyl ester 170507 1-(2,2-dimethylpropanoyl)-2'-[3,5-di(trifluoromethyl)benzoyl]-5'-phenylspiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole]-4',6'-dione 170586 1-[3,5-di(trifluoromethyl)benzoyl]-2'-methylsulfonyl-5'-phenylspiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole]-4',6'-dione 170668 1-(2,5-dimethoxyphenylsulfonyl)-2'-[3,5-di(trifluoromethyl)benzoyl]-5'-phenylspiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole]-4',6'-dione 170768 6-(4-t-butylphenyl)-2-(4-morpholin-4-yl)pyran-4-one 170769 2-(4-methoxyphenyl)-6-morpholino-4H-pyran-4-one 170799 6-(4-(4-methylnaphthalen-1-yl)phenyl)-2-morpholin-4-yl-4H-thiopyran-4-one 170833 2-morpholin-4-yl-6-phenyl-4H-thiopyran-4-one 170907 2-(2-methoxyphenyl)-6-morpholino-4H-pyran-4-one 170938 SID29217598 170939 6-(3-fluorophenyl)-2-(4-morpholin-4-yl)pyran-4-one 171158 2-morpholino-6-(4-(naphthalen-1-yl)phenyl)-4H-thiopyran-4-one 171228 4-(4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-ylamino)benzamide 171234 2-((4-(4-amino-5-(3-methoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)phenethyl)(methyl)amino)ethanol 171245 N-[(R,R)-(E)-(3,4-dichlorobenzyl)-3-(2-oxoazepan-3-yl)carbamoyl]allyl-N-methyl-3,5-bis(trifluoromethyl)benzamide 171270 (2R,3S,4R,5R)-2-Hydroxymethyl-5-[6-((S)-2-hydroxy-1-methyl-2-phenyl-ethylamino)-purin-9-yl]-tetrahydro-furan-3,4-diol 171274 3-chloro-4-[16-methyl-(12S)-2,10-diazatetracyclo[11.2.1.02,12.04,9]hexadeca-4(9),5,7-trien-10-ylcarbonyl]-1-(2-phenylphenylcarboxamido)benzene 171275 1N-{4-[16-ethyl-2,10-diazatetracyclo[11.2.1.02,12.04,9]hexadeca-4(9),5,7-trien-10-ylcarbonyl]phenyl}-2-phenylbenzamide 171314 1N-{4-[6-chloro-16-ethyl-(12S)-2,10-diazatetracyclo[11.2.1.02,12.04,9]hexadeca-4(9),5,7-trien-10-ylcarbonyl]phenyl}-2-(4-methylphenyl)benzamide 171320 (4-benzylpiperazin-1-yl)(1H-indol-4-yl)methanone 171361 6-(3-bromophenyl)-2-morpholin-4-yl-4H-thiopyran-4-one 171362 2-(4-(benzo[b]thiophen-3-yl)phenyl)-6-morpholino-4H-thiopyran-4-one 171366 (4-Benzyl-piperazin-1-yl)-(1H-indol-6-yl)-methanone 171371 3-chloro-4-[16-ethyl-2,10-diazatetracyclo[11.2.1.02,12.04,9]hexadeca-4(9),5,7-trien-10-ylcarbonyl]-1-(2-phenylphenylcarboxamido)benzene 171405 3-[3'-(6-morpholin-4-yl-4-oxo-4H-thiopyran-2-yl)-biphenyl-2-yl]-acrylic acid methyl ester 171409 (4-Benzyl-piperazin-1-yl)-(6-methoxy-1H-indol-5-yl)-methanone 171446 6-(4-t-butylphenyl)-2-morpholin-4-yl-4H-thiopyran-4-one 171477 (2R,3S,4R,5R)-2-Hydroxymethyl-5-[6-(pyrrolidin-1-ylamino)-purin-9-yl]-tetrahydro-furan-3,4-diol 171481 6-(4-methoxyphenyl)-2-morpholin-4-yl-4H-thiopyran-4-one 171482 6-(4-chlorophenyl)-2-morpholin-4-yl-4H-thiopyran-4-one 171507 N-Methyl-N-[(E)-(R)-1-(1-methyl-1H-indol-3-ylmethyl)-3-((R)-2-oxo-azepan-3-ylcarbamoyl)-allyl]-3,5-bis-trifluoromethyl-benzamide 171508 N-[(E)-(R)-3-(1-Carbamoyl-cyclohexylcarbamoyl)-1-(4-chloro-benzyl)-allyl]-N-methyl-3,5-bis-trifluoromethyl-benzamide 171509 3-[N'-(3,5-Bis-trifluoromethyl-benzoyl)-N-(3,4-dichloro-benzyl)-N'-methyl-hydrazino]-N-((R)-2-oxo-azepan-3-yl)-propionamide 171513 4'-[3-((R)-3-Hydroxy-pyrrolidin-1-yl)-propoxy]-biphenyl-4-carbonitrile 171522 1N-{4-[6-chloro-16-methyl-(12S)-2,10-diazatetracyclo[11.2.1.02,12.04,9]hexadeca-4(9),5,7-trien-10-ylcarbonyl]phenyl}-2-trifluoromethylbenzamide 171526 1N-{4-[6-chloro-16-methyl-(12S)-2,10-diazatetracyclo[11.2.1.02,12.04,9]hexadeca-4(9),5,7-trien-10-ylcarbonyl]phenyl}-2-(4-methylphenyl)benzamide 171527 N-[(E)-(R)-1-(4-Chloro-benzyl)-3-((R)-2-oxo-azepan-3-ylcarbamoyl)-allyl]-N-methyl-3,5-bis-trifluoromethyl-benzamide 171542 4'-[3-(4-Amino-piperidin-1-yl)-propoxy]-biphenyl-4-carbonitrile 171551 6-cyclohexylmethoxy-2-(4-sulfamoylanilino)purine 171554 1N-{4-[6-chloro-16-ethyl-(12S)-2,10-diazatetracyclo[11.2.1.02,12.04,9]hexadeca-4(9),5,7-trien-10-ylcarbonyl]phenyl}-2-chlorobenzamide 171557 1N-{4-[6-chloro-16-methyl-(12S)-2,10-diazatetracyclo[11.2.1.02,12.04,9]hexadeca-4(9),5,7-trien-10-ylcarbonyl]phenyl}-2-chlorobenzamide 171562 4-[3-(4'-Chloro-biphenyl-4-yloxy)-propyl]-piperazine-1-carboxylic acid ethyl ester 171573 N-[(E)-(R)-1-(4,5-Dichloro-thiophen-2-ylmethyl)-3-((R)-2-oxo-azepan-3-ylcarbamoyl)-allyl]-N-methyl-3,5-bis-trifluoromethyl-benzamide 171574 4'-[3-((S)-3-Hydroxy-pyrrolidin-1-yl)-propoxy]-biphenyl-4-carbonitrile 171581 2-Methyl-N-[4-(2,3,4,5-tetrahydro-benzo[b][1,4]diazepine-1-carbonyl)-phenyl]-benzamide 171583 3-chloro-4-[16-ethyl-(12S)-2,10-diazatetracyclo[11.2.1.02,12.04,9]hexadeca-4(9),5,7-trien-10-ylcarbonyl]-1-(3-fluoro-5-methylphenylcarboxamido)benzene 171584 3-chloro-4-[16-methyl-(12R)-2,10-diazatetracyclo[11.2.1.02,12.04,9]hexadeca-4(9),5,7-trien-10-ylcarbonyl]-1-(2-phenylphenylcarboxamido)benzene 171585 3-chloro-4-[6-chloro-16-methyl-(12S)-2,10-diazatetracyclo[11.2.1.02,12.04,9]hexadeca-4(9),5,7-trien-10-ylcarbonyl]-1-[2-(4-methylphenyl)phenylcarboxamido]benzene 171592 3-[N'-(3,5-Bis-trifluoromethyl-benzoyl)-N'-methyl-N-naphthalen-2-ylmethyl-hydrazino]-N-((R)-2-oxo-azepan-3-yl)-propionamide 171604 4'-[3-((R)-3-Amino-pyrrolidin-1-yl)-propoxy]-biphenyl-4-carbonitrile 171605 4-[3-(3'-Cyano-biphenyl-4-yloxy)-propyl]-piperazine-1-carboxylic acid ethyl ester 171613 N-Methyl-N-[(E)-(R)-1-naphthalen-2-ylmethyl-3-((R)-2-oxo-azepan-3-ylcarbamoyl)-allyl]-3,5-bis-trifluoromethyl-benzamide 171618 N-[(E)-(R)-1-(4,5-Dibromo-thiophen-2-ylmethyl)-3-((R)-2-oxo-azepan-3-ylcarbamoyl)-allyl]-N-methyl-3,5-bis-trifluoromethyl-benzamide 171634 1N-{4-[6-chloro-16-methyl-(12S)-2,10-diazatetracyclo[11.2.1.02,12.04,9]hexadeca-4(9),5,7-trien-10-ylcarbonyl]phenyl}-2-fluorobenzamide 171641 4-[3-(2'-Nitro-biphenyl-4-yloxy)-propyl]-piperazine-1-carboxylic acid ethyl ester 171654 ((2R,5S)-4-benzyl-2,5-dimethylpiperazin-1-yl)(6-methoxy-1H-indol-5-yl)methanone 171680 N-[(E)-(R)-1-(4-Chloro-benzyl)-3-cycloheptylcarbamoyl-allyl]-N-methyl-3,5-bis-trifluoromethyl-benzamide 171683 4-[3-(4'-Nitro-biphenyl-4-yloxy)-propyl]-piperazine-1-carboxylic acid ethyl ester 171693 2-(3'-hydroxy-biphenyl-3-yl)-6-morpholin-4-yl-thiopyran-4-one 171694 6-(4-bromophenyl)-2-morpholin-4-yl-4H-thiopyran-4-one 171697 ((1R,3S)-4-Benzyl-2,5-dimethyl-piperazin-1-yl)-(6-methoxy-1H-indol-5-yl)-methanone 171723 (4-Benzyl-piperazin-1-yl)-(1H-indol-5-yl)-methanone 171728 SID24819082 171761 3-[N'-(3,5-Bis-trifluoromethyl-benzoyl)-N-(4,5-dibromo-thiophen-2-ylmethyl)-N'-methyl-hydrazino]-N-((R)-2-oxo-azepan-3-yl)-propionamide 171771 ((1S,3R)-4-Benzyl-2,5-dimethyl-piperazin-1-yl)-(1H-indol-5-yl)-methanone 171779 2-(3-methoxyphenyl)-6-morpholino-4H-pyran-4-one 171781 2-(4-fluorophenyl)-6-morpholino-4H-pyran-4-one 171785 2-(4-chlorophenyl)-6-morpholino-4H-pyran-4-one 171786 2-morpholino-6-phenyl-4H-pyran-4-one 171803 3-{1-[2-(2,3-Dihydro-benzo[1,4]dioxin-5-yloxy)-ethyl]-1,2,3,6-tetrahydro-pyridin-4-yl}-5-fluoro-1H-indole 171869 5-{2-[4-(1H-Pyrrolo[2,3-b]pyridin-3-yl)-3,6-dihydro-2H-pyridin-1-yl]-ethoxy}-quinoline 171872 5-{2-[4-(1H-Indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]-ethoxy}-quinoline 171873 1H-4-indolyl 2-[4-(1H-3-indolyl)-1,2,3,6-tetrahydro-1-pyridinyl]ethyl ether 171951 4-Methyl-4-{2-[3-(naphthalene-1-carbonyl)-indol-1-yl]-ethyl}-morpholin-4-ium 172197 3-{1-[2-(2,3-Dihydro-benzo[1,4]dioxin-5-yloxy)-ethyl]-1,2,3,6-tetrahydro-pyridin-4-yl}-1H-indole 172234 3-{1-[2-(1H-Indol-4-yloxy)-ethyl]-1,2,3,6-tetrahydro-pyridin-4-yl}-1H-pyrrolo[2,3-b]pyridine 172306 3-{1-[2-(2,3-Dihydro-benzo[1,4]dioxin-5-yloxy)-ethyl]-piperidin-4-yl}-6-fluoro-1H-indole 172307 3-{1-[2-(2,3-Dihydro-benzo[1,4]dioxin-5-yloxy)-ethyl]-1,2,3,6-tetrahydro-pyridin-4-yl}-1H-pyrrolo[2,3-b]pyridine 172359 2,2-Dimethyl-5-{4-[2-(3,4,5-trimethoxy-phenyl)-ethyl]-phenyl}-2,3-dihydro-imidazo[2,1-a]isoquinoline 172360 3,3-Dimethyl-6-{4-[2-(3,4,5-trimethoxy-phenyl)-ethyl]-phenyl}-3,4-dihydro-2H-pyrimido[2,1-a]isoquinoline 172362 7-Methyl-4-{4-[2-(3,4,5-trimethoxy-phenyl)-ethyl]-phenyl}-2,3-dihydro-6-oxa-1,3a-diaza-as-indacene 172398 5-{4-[2-(3,4,5-Trimethoxy-phenyl)-ethyl]-phenyl}-2,3-dihydro-imidazo[1,2-c]quinazoline 172428 6-{4-[2-(3,4,5-Trimethoxy-phenyl)-ethyl]-phenyl}-3,4-dihydro-2H-pyrimido[2,1-a]isoquinoline 172456 2-Methyl-5-{4-[2-(3,4,5-trimethoxy-phenyl)-ethyl]-phenyl}-2,3-dihydro-imidazo[2,1-a]isoquinoline 172534 3-Methyl-5-{4-[2-(3,4,5-trimethoxy-phenyl)-ethyl]-phenyl}-[1,2,4]triazolo[3,4-a]isoquinoline 172535 2-Methyl-5-{4-[2-(3,4,5-trimethoxy-phenyl)-ethyl]-phenyl}-imidazo[2,1-a]isoquinoline 172536 5-{4-[2-(3,4,5-Trimethoxy-phenyl)-ethyl]-phenyl}-imidazo[2,1-a]isoquinoline 172537 4-{4-[2-(3,4,5-Trimethoxy-phenyl)-ethyl]-phenyl}-2,3-dihydro-8-thia-1,3a-diaza-as-indacene 172875 (R)-2-fluoro-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol 172876 (R)-2-bromo-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol 172877 7-propyl-(6aR)-6a,7,8,9-tetrahydro-6H-benzo[de][1,3]dioxolo[5',4':5,6]benzo[g]quinolin-11-amine 172897 1-(2-methyl-2,3-dihydro-1H-indol-1-yl)-2-{4-[(4-methylphenyl)methyl]piperazin-1-yl}ethan-1-one 172941 4'-Oxazol-4-yl-biphenyl-2-sulfonic acid (3,4-dimethyl-isoxazol-5-yl)-amide 172972 4'-(5-Methyl-oxazol-4-yl)-biphenyl-2-sulfonic acid (3,4-dimethyl-isoxazol-5-yl)-amide 172985 3-((1H-pyrrol-2-yl)methylene)-5-(pyridin-3-yl)indolin-2-one 173023 (S)-2-Amino-N-{(R)-1-[(S)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-ethylcarbamoyl]-ethyl}-3-(4-hydroxy-phenyl)-propionamide 173040 4'-Benzooxazol-2-yl-biphenyl-2-sulfonic acid (3,4-dimethyl-isoxazol-5-yl)-amide 173063 2'-Amino-4'-isobutyl-biphenyl-2-sulfonic acid (3,4-dimethyl-isoxazol-5-yl)-amide 173064 4'-Isobutyl-biphenyl-2-sulfonic acid (3,4-dimethyl-isoxazol-5-yl)-amide 173079 4'-Oxazol-5-yl-biphenyl-2-sulfonic acid (3,4-dimethyl-isoxazol-5-yl)-amide 173159 {2-Butyl-5-chloro-3-[7-(1H-tetrazol-5-yl)-naphthalen-2-ylmethyl]-3H-imidazol-4-yl}-methanol 173160 {2-Butyl-5-chloro-1-[6-(1H-tetrazol-5-yl)-naphthalen-2-ylmethyl]-1H-imidazol-4-yl}-methanol 173183 {2-Butyl-5-chloro-3-[5-(1H-tetrazol-5-yl)-naphthalen-1-ylmethyl]-3H-imidazol-4-yl}-methanol 173185 6-(2-Butyl-4-chloro-5-hydroxymethyl-imidazol-1-ylmethyl)-1,2,3,4-tetrahydro-naphthalene-2-carboxylic acid 173200 4'-(2-Methyl-oxazol-4-yl)-biphenyl-2-sulfonic acid (3,4-dimethyl-isoxazol-5-yl)-amide 173210 {2-Butyl-5-chloro-3-[8-(1H-tetrazol-5-yl)-naphthalen-2-ylmethyl]-3H-imidazol-4-yl}-methanol 173212 6-(2-Butyl-5-chloro-4-hydroxymethyl-imidazol-1-ylmethyl)-1,2,3,4-tetrahydro-naphthalene-2-carboxylic acid 173215 1-[(2R)-2-methyl-2,3-dihydro-1H-indol-1-yl]-2-{4-[(4-methylphenyl)methyl]piperazin-1-yl}ethan-1-one 173229 {2-Butyl-5-chloro-3-[6-(1H-tetrazol-5-yl)-naphthalen-2-ylmethyl]-3H-imidazol-4-yl}-methanol 173230 {2-Butyl-5-chloro-3-[6-(1H-tetrazol-5-yl)-naphthalen-1-ylmethyl]-3H-imidazol-4-yl}-methanol 173231 {2-Butyl-5-chloro-3-[6-(1H-tetrazol-5-yl)-5,6,7,8-tetrahydro-naphthalen-2-ylmethyl]-3H-imidazol-4-yl}-methanol 173238 4'-Oxazol-2-ylmethyl-biphenyl-2-sulfonic acid (3,4-dimethyl-isoxazol-5-yl)-amide 173239 4'-(4-Methyl-oxazol-2-yl)-biphenyl-2-sulfonic acid (3,4-dimethyl-isoxazol-5-yl)-amide 173292 6-(2-Butyl-5-chloro-4-hydroxymethyl-imidazol-1-ylmethyl)-2-methyl-1,2,3,4-tetrahydro-naphthalene-2-carboxylic acid 173315 6-(2-Butyl-4-chloro-5-hydroxymethyl-imidazol-1-ylmethyl)-2-methyl-1,2,3,4-tetrahydro-naphthalene-2-carboxylic acid 173327 13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-benzyl-3,8,14-trioxo-1,4,9triaza-cyclotetradecane-5-carboxylic acid amide 173329 13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-3,8,14-trioxo-2-phenethyl-1,4,9triaza-cyclotetradecane-5-carboxylic acid amide 173330 13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-naphthalen-2-ylmethyl-3,8,14-trioxo-1,4,9triaza-cyclotetradecane-5-carboxylic acid amide 173332 {2-Butyl-5-chloro-1-[6-(1H-tetrazol-5-yl)-5,6,7,8-tetrahydro-naphthalen-2-ylmethyl]-1H-imidazol-4-yl}-methanol 173587 (S)-6-Amino-2-{(R)-2-[(S)-2-{(S)-2-[(R)-2-[(S)-2-amino-3-(1H-imidazol-4-yl)-propionylamino]-3-(1H-indol-3-yl)-propionylamino]-propionylamino}-3-(1H-indol-3-yl)-propionylamino]-3-phenyl-propionylamino}-hexanoic acid amide 173611 N-(3,5-bis(trifluoromethyl)benzyl)-N,7-dimethyl-8-oxo-5-p-tolyl-7,8-dihydro-1,7-naphthyridine-6-carboxamide 173688 (R)-2-amino-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol 173693 4'-(5-Methyl-oxazol-2-yl)-biphenyl-2-sulfonic acid (3,4-dimethyl-isoxazol-5-yl)-amide 173717 4'-(4,5-Dimethyl-oxazol-2-yl)-biphenyl-2-sulfonic acid (3,4-dimethyl-isoxazol-5-yl)-amide 173746 11-fluoro-7-propyl-(6aR)-6a,7,8,9-tetrahydro-6H-benzo[de][1,3]dioxolo[5',4':5,6]benzo[g]quinoline 173806 2-m-tolyl-2H-pyrazolo[3,4-c]quinolin-4-amine 173879 2-p-tolyl-2H-pyrazolo[3,4-c]quinolin-4-amine 173982 SID26747498 173984 2-(4-methoxyphenyl)-2H-pyrazolo[3,4-c]quinolin-4-amine 174034 (-)-trans-3-Cyclopropylmethyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinolin-9-ol 174118 N-[2-(5-Dimethylaminomethyl-furan-2-ylmethylsulfanyl)-ethyl]-4,6-dinitro-benzene-1,3-diamine 174123 2-{3-[3-(3-Benzoyl-phenyl)-ureido]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-benzo[b][1,4]diazepin-1-yl}-N-methyl-N-phenyl-acetamide 174157 2-phenyl-2H-pyrazolo[3,4-c]quinolin-4-amine 174159 2-{5-[2-(5-Dimethylaminomethyl-furan-2-ylmethylsulfanyl)-ethylamino]-2,4-dinitro-phenylamino}-benzonitrile 174167 (4aR,7S,7aR,12bS)-3-Cyclopropylmethyl-9-methoxy-2,3,4,4a,5,6,7,7a-octahydro-1H-8-oxa-3-aza-benzo[d]fluoren-7-ol 174199 N-[2-(5-Dimethylaminomethyl-furan-2-ylmethylsulfanyl)-ethyl]-4,6-dinitro-N'-propyl-benzene-1,3-diamine 174202 (4aR,7aR,12bS)-3-Cyclopropylmethyl-9-methoxy-2,3,4,4a,5,6-hexahydro-1H-8-oxa-3-aza-benzo[d]fluoren-7-one 174203 (4aR,7aR,12bS)-3-Cyclopropylmethyl-9-hydroxy-2,3,4,4a,5,6-hexahydro-1H-8-oxa-3-aza-benzo[d]fluoren-7-one 174239 13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-benzyl-3,8,14-trioxo-1,4,9triaza-cyclotetradecane-5-carboxylic acid amide 174240 13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-benzyl-2-methyl-3,8,14-trioxo-1,4,9triaza-cyclotetradecane-5-carboxylic acid amide 174242 (4aS,7aR,12bS)-3-Cyclopropylmethyl-9-hydroxy-2,3,4,4a,5,6-hexahydro-1H-8-oxa-3-aza-benzo[d]fluoren-7-one 174258 (4aS,7R,7aR,12bS)-3-Cyclopropylmethyl-2,3,4,4a,5,6,7,7a-octahydro-1H-8-oxa-3-aza-benzo[d]fluorene-7,9-diol 174296 (4aR,7aR,12bS)-9-Hydroxy-3-methyl-2,3,4,4a,5,6-hexahydro-1H-8-oxa-3-aza-benzo[d]fluoren-7-one 174371 7-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-6,12,17-trioxo-6,7,8,9,10,11,12,13,14,15,16,17,17a,18-tetradecahydro-5H-5a,11,16-triaza-cyclotetradeca[b]naphthalene-15-carboxylic acid amide 174372 13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-benzyl-1-methyl-3,8,14-trioxo-1,4,9triaza-cyclotetradecane-5-carboxylic acid amide 174373 13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-3,8,14-trioxo-2-phenethyl-1,4,9triaza-cyclotetradecane-5-carboxylic acid amide 174379 2-(2,4-Dioxo-5-phenyl-3-{3-[3-(3-trifluoromethyl-3H-diazirin-3-yl)-phenyl]-ureido}-2,3,4,5-tetrahydro-benzo[b][1,4]diazepin-1-yl)-N-isopropyl-N-phenyl-acetamide 174380 2-(2,4-Dioxo-5-phenyl-3-{3-[3-(3-trifluoromethyl-3H-diazirin-3-yl)-phenyl]-ureido}-2,3,4,5-tetrahydro-benzo[b][1,4]diazepin-1-yl)-N-isopropyl-N-(4-methoxy-phenyl)-acetamide 174390 H-Tyr-c[D-Orn-Aic-Glu]-NH2 174391 13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-(2-methyl-benzyl)-3,8,14-trioxo-1,4,9triaza-cyclotetradecane-5-carboxylic acid amide 174415 2-{3-[3-(3-Benzoyl-phenyl)-ureido]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-benzo[b][1,4]diazepin-1-yl}-N-(4-methoxy-phenyl)-N-methyl-acetamide 174434 1-(1-Benzyl-piperidin-4-yl)-1H-pyrrole-3-carbaldehyde 174467 N-[2-(5-Dimethylaminomethyl-furan-2-ylmethylsulfanyl)-ethyl]-N'-methyl-4,6-dinitro-benzene-1,3-diamine 174469 2-{3-[3-(3-Benzoyl-phenyl)-ureido]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-benzo[b][1,4]diazepin-1-yl}-N-isopropyl-N-(4-methoxy-phenyl)-acetamide 174473 N-[2-(5-Dimethylaminomethyl-furan-2-ylmethylsulfanyl)-ethyl]-N'-(4-fluoro-phenyl)-4,6-dinitro-benzene-1,3-diamine 174478 N-[2-(5-Dimethylaminomethyl-furan-2-ylmethylsulfanyl)-ethyl]-4,6-dinitro-N'-pyridin-2-ylmethyl-benzene-1,3-diamine 174483 2-[2,4-Dioxo-5-phenyl-3-(3-phenyl-ureido)-2,3,4,5-tetrahydro-benzo[b][1,4]diazepin-1-yl]-N-(4-methoxy-phenyl)-N-methyl-acetamide 174487 1-Benzyl-4-(2-ethynyl-pyrrol-1-yl)-piperidine 174488 1-Benzyl-4-(2-trimethylsilanylethynyl-pyrrol-1-yl)-piperidine 174489 PD-0173952 174510 N-[2-(5-Dimethylaminomethyl-furan-2-ylmethylsulfanyl)-ethyl]-N'-(3-morpholin-4-yl-propyl)-4,6-dinitro-benzene-1,3-diamine 174513 2-[1-(1-Benzyl-piperidin-4-yl)-1H-pyrrol-2-ylmethylene]-malononitrile 174514 1-Benzyl-4-(2-iodo-pyrrol-1-yl)-piperidine 174523 N-Benzyl-N'-[2-(5-dimethylaminomethyl-furan-2-ylmethylsulfanyl)-ethyl]-4,6-dinitro-benzene-1,3-diamine 174531 1-Benzyl-4-(2-phenylethynyl-pyrrol-1-yl)-piperidine 174532 1-Benzyl-4-(2-oxazol-5-yl-pyrrol-1-yl)-piperidine 174536 N-[2-(5-Dimethylaminomethyl-furan-2-ylmethylsulfanyl)-ethyl]-4,6-dinitro-N'-pyridin-3-ylmethyl-benzene-1,3-diamine 174540 N-(2-Dimethylamino-ethyl)-N'-[2-(5-dimethylaminomethyl-furan-2-ylmethylsulfanyl)-ethyl]-4,6-dinitro-benzene-1,3-diamine 174546 2-[2,4-Dioxo-5-phenyl-3-(3-phenyl-ureido)-2,3,4,5-tetrahydro-benzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxy-phenyl)-acetamide 174549 N-[2-(5-Dimethylaminomethyl-furan-2-ylmethylsulfanyl)-ethyl]-4,6-dinitro-N'-phenyl-benzene-1,3-diamine 174551 2-(2,4-Dioxo-5-phenyl-3-{3-[3-(3-trifluoromethyl-3H-diazirin-3-yl)-phenyl]-ureido}-2,3,4,5-tetrahydro-benzo[b][1,4]diazepin-1-yl)-N-(4-methoxy-phenyl)-N-methyl-acetamide 174552 [2-(5-Dimethylaminomethyl-furan-2-ylmethylsulfanyl)-ethyl]-[5-(N'-isopropylidene-hydrazino)-2,4-dinitro-phenyl]-amine 174553 [2-(5-Dimethylaminomethyl-furan-2-ylmethylsulfanyl)-ethyl]-(5-hydrazino-2,4-dinitro-phenyl)-amine 174562 1-(1-Benzyl-piperidin-4-yl)-1H-pyrrole-2-carbaldehyde 174566 2-[1-(1-Benzyl-piperidin-4-yl)-1H-pyrrol-3-ylmethylene]-malononitrile 174577 3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-2,6-dihydro-3H-imidazo[1,2-c]quinazolin-5-one 174594 1-Benzyl-4-(3-oxazol-5-yl-pyrrol-1-yl)-piperidine 174604 2-{3-[3-(3-Benzoyl-phenyl)-ureido]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-benzo[b][1,4]diazepin-1-yl}-N-isopropyl-N-phenyl-acetamide 174608 2-(2,4-Dioxo-5-phenyl-3-{3-[3-(3-trifluoromethyl-3H-diazirin-3-yl)-phenyl]-ureido}-2,3,4,5-tetrahydro-benzo[b][1,4]diazepin-1-yl)-N-methyl-N-phenyl-acetamide 174616 1-Benzyl-4-pyrrol-1-yl-piperidine 174627 (4aR,7S,7aR,12bS)-3-Cyclopropylmethyl-2,3,4,4a,5,6,7,7a-octahydro-1H-8-oxa-3-aza-benzo[d]fluorene-7,9-diol 174683 15-Amino-1-methyl-10-thia-tricyclo[7.5.1.0*2,7*]pentadeca-2,4,6-trien-4-ol 174684 7-Amino-6-ethyl-8,8-dimethyl-5,6,7,8-tetrahydro-naphthalen-2-ol 174685 3-Amino-4,4-dimethyl-1,2,3,4-tetrahydro-naphthalene-2,6-diol 174779 7-Amino-6-ethyl-8,8-dimethyl-5,6,7,8-tetrahydro-naphthalen-2-ol 174819 7-Amino-8,8-dimethyl-6-methylsulfanyl-5,6,7,8-tetrahydro-naphthalen-2-ol 174820 7-Amino-8,8-dimethyl-6-methylsulfanyl-5,6,7,8-tetrahydro-naphthalen-2-ol 174828 [2-(5-Dimethylaminomethyl-furan-2-ylmethylsulfanyl)-ethyl]-(2,4-dinitro-phenyl)-amine 174830 [2-(5-Dimethylaminomethyl-furan-2-ylmethylsulfanyl)-ethyl]-(5-fluoro-2,4-dinitro-phenyl)-amine 174831 [2-(5-Dimethylaminomethyl-furan-2-ylmethylsulfanyl)-ethyl]-(4-fluoro-2-nitro-phenyl)-amine 174858 7-Amino-6-mercapto-8,8-dimethyl-5,6,7,8-tetrahydro-naphthalen-2-ol 174911 7-Hydroxy-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid {1-[4-(3-hydroxy-phenyl)-3,4-dimethyl-piperidin-1-ylmethyl]-2-methyl-propyl}-amide 175051 7-Amino-6-methoxy-8,8-dimethyl-5,6,7,8-tetrahydro-naphthalen-2-ol 175070 7-Amino-6-methanesulfinyl-8,8-dimethyl-5,6,7,8-tetrahydro-naphthalen-2-ol 175100 7-Amino-6-methanesulfonyl-8,8-dimethyl-5,6,7,8-tetrahydro-naphthalen-2-ol 175678 N-(4-(2-chloro-6-methylphenylamino)imidazo[1,5-a]quinoxalin-8-yl)acetamide 175722 GNF-Pf-3427 175981 N4-(2-chloro-6-methylphenyl)-N8-(2-(dimethylamino)ethyl)imidazo[1,5-a]quinoxaline-4,8-diamine 175984 N4-(2-chloro-6-methylphenyl)-N8,N8-diethylimidazo[1,5-a]quinoxaline-4,8-diamine 175990 N-(2-chloro-6-methylphenyl)-8-(4-methylpiperazin-1-yl)imidazo[1,5-a]quinoxalin-4-amine 175991 N-(2-chloro-6-methylphenyl)-8-(piperazin-1-yl)imidazo[1,5-a]quinoxalin-4-amine 176006 N4-(2-chloro-6-methylphenyl)-N8-ethylimidazo[1,5-a]quinoxaline-4,8-diamine 176058 N4-(2-chloro-6-methylphenyl)-N8,N8-dimethylimidazo[1,5-a]quinoxaline-4,8-diamine 176069 N4-(2-chloro-6-methylphenyl)-N8-(2-morpholinoethyl)imidazo[1,5-a]quinoxaline-4,8-diamine 176106 N-(2-chloro-6-methylphenyl)-8-(3,5-dimethylpiperazin-1-yl)imidazo[1,5-a]quinoxalin-4-amine 176174 N-(2-chloro-6-methylphenyl)-7-(piperazin-1-yl)imidazo[1,5-a]quinoxalin-4-amine 176175 N-(2-chloro-6-methylphenyl)-7-(3,5-dimethylpiperazin-1-yl)imidazo[1,5-a]quinoxalin-4-amine 176176 N-(2-chloro-6-methylphenyl)-8-(3,5-dimethylpiperazin-1-yl)-7-methoxyimidazo[1,5-a]quinoxalin-4-amine 176246 N-(2-chloro-6-methylphenyl)-8-morpholinoimidazo[1,5-a]quinoxalin-4-amine 176272 N4-(2-chloro-6-methylphenyl)-N8-(3-morpholinopropyl)imidazo[1,5-a]quinoxaline-4,8-diamine 176273 N-(2-chloro-6-methylphenyl)-8-(4-ethylpiperazin-1-yl)imidazo[1,5-a]quinoxalin-4-amine 176274 4-(4-(2-chloro-6-methylphenylamino)imidazo[1,5-a]quinoxalin-8-yl)piperazine-1-carbaldehyde 176290 methyl 4-(2-chloro-6-methylphenylamino)imidazo[1,5-a]quinoxaline-8-carboxylate 176292 N-(2-chloro-6-methylphenyl)-8-fluoroimidazo[1,5-a]quinoxalin-4-amine 176326 8-bromo-N-(2-chloro-6-methylphenyl)imidazo[1,5-a]quinoxalin-4-amine 176338 N4-(2-chloro-6-methylphenyl)imidazo[1,5-a]quinoxaline-4,8-diamine 176361 4-(2-chloro-6-methylphenylamino)imidazo[1,5-a]quinoxaline-8-carbonitrile 176407 N-(2-chloro-6-methylphenyl)-9-methoxyimidazo[1,5-a]quinoxalin-4-amine 176418 (2,6-dichloro-phenyl)-(8-nitro-imidazo[1,5-a]quinoxalin-4-yl)-amine 176433 4-(2-chloro-6-methylphenylamino)imidazo[1,5-a]quinoxaline-7,8-diol 176461 (2-chloro-6-methyl-phenyl)-(8,9-dihydro-7,10-dioxa-2,5,11b-triaza-cyclopenta[a]anthracen-4-yl)-amine 176462 (2-chloro-6-methyl-phenyl)-(7,9-dioxa-2,5,10b-triaza-dicyclopenta[a,g]naphthalen-4-yl)-amine 176477 SID26751851 176486 N-(2,6-dimethylphenyl)-9-nitroimidazo[1,5-a]quinoxalin-4-amine 176522 N4-(2,6-dimethylphenyl)imidazo[1,5-a]quinoxaline-4,9-diamine 176525 9-(benzyloxy)-N-(2-chloro-6-methylphenyl)imidazo[1,5-a]quinoxalin-4-amine 176543 N-(2-chloro-6-methylphenyl)-8-(4-methyl-1,4-diazepan-1-yl)imidazo[1,5-a]quinoxalin-4-amine 176544 N4-(2-chloro-6-methylphenyl)-N7-(3-(dimethylamino)propyl)imidazo[1,5-a]quinoxaline-4,7-diamine 176567 4-(1-Allyl-1,2,5,6-tetrahydro-pyridin-3-yl)-thiazol-2-ylamine 176642 4-(1-Ethyl-1,2,5,6-tetrahydro-pyridin-3-yl)-thiazol-2-ylamine 176778 N4-(2-chloro-6-methylphenyl)-N7-(2-(dimethylamino)ethyl)-8-methoxyimidazo[1,5-a]quinoxaline-4,7-diamine 176786 2-(3,4-Dichloro-phenyl)-N-methyl-N-(1-phenyl-2-pyrrolidin-1-yl-ethyl)-acetamide 176803 8-[1-(3,4-Dichloro-phenyl)-meth-(E)-ylidene]-5-(3-hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]nonan-7-one 176821 N4-(2-chloro-6-fluorophenyl)-N7-(2-(dimethylamino)ethyl)-8-methoxyimidazo[1,5-a]quinoxaline-4,7-diamine 176841 N4-(2-chloro-6-methylphenyl)-8-methoxy-N7-(2-morpholinoethyl)imidazo[1,5-a]quinoxaline-4,7-diamine 176842 N-(2-chloro-6-methylphenyl)-8-methoxy-7-(2-morpholinoethoxy)imidazo[1,5-a]quinoxalin-4-amine 176853 N*4*-(2-Chloro-6-methyl-phenyl)-N*7*-(2-dimethylamino-ethyl)-8-methoxy-1-methyl-imidazo[1,5-a]quinoxaline-4,7-diamine 176877 ethyl 8-amino-4-oxo-4,5-dihydro-[1,2,4]triazolo[1,5-a]quinoxaline-2-carboxylate 176883 N-(2-chloro-6-methylphenyl)-7-(4-methylpiperazin-1-yl)imidazo[1,5-a]quinoxalin-4-amine 176884 N4-(2-chloro-6-methylphenyl)-N7-(2-(dimethylamino)ethyl)imidazo[1,5-a]quinoxaline-4,7-diamine 176891 senktide 176924 N-(2-chloro-6-methylphenyl)-7-methoxy-8-(2-morpholinoethoxy)imidazo[1,5-a]quinoxalin-4-amine 177077 3-hydroxy-4-methoxy-17-methyl-18-[1-phenyl-(E)-methylidene]-17-azapentacyclo[7.5.3.210,14.01,10.02,7]nonadeca-2(7),3,5-trien-13-one 177109 5-(3-Hydroxy-phenyl)-2-methyl-8-[1-phenyl-meth-(E)-ylidene]-2-aza-bicyclo[3.3.1]nonan-7-one 177149 13,22-dimethyl-2-(3-methyl-2-butenyl)-14-oxa-11,22-diazaheptacyclo[13.9.1.01,13.02,21.04,12.05,10.019,25]pentacosa-4(12),5(10),6,8,15,17,19(25)-heptaen-16-ol 177155 19-methoxy-24-methyl-26-(1-methylethylidene)-4,24-diazaheptacyclo[12.7.3.22,13.01,13.03,11.05,10.016,21]hexacosa-3(11),5(10),6,8,16(21),17,19-heptaen-20-ol 177169 2-[4-(2-Propoxy-phenyl)-piperazin-1-ylmethyl]-1H-benzoimidazole-4-carboxylic acid (1-aza-bicyclo[2.2.2]oct-3-yl)-amide 177193 2-[4-(2-Butoxy-phenyl)-piperazin-1-ylmethyl]-1H-benzoimidazole-4-carboxylic acid (1-aza-bicyclo[2.2.2]oct-3-yl)-amide 177195 13,22-dimethyl-2-[3-phenyl-(E)-2-propenyl]-14-oxa-11,22-diazaheptacyclo[13.9.1.01,13.02,21.04,12.05,10.019,25]pentacosa-4(12),5(10),6,8,15,17,19(25)-heptaen-16-ol 177225 2-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-1-(4-o-tolyl-piperazin-1-yl)-ethanone; compound with but-2-enedioic acid 177233 3-hydroxy-4-methoxy-17-methyl-18-[1-phenyl-(E)-ethylidene]-17-azapentacyclo[7.5.3.210,14.01,10.02,7]nonadeca-2(7),3,5-trien-13-one 177267 4-o-Tolyl-piperazine-1-carboxylic acid 4-chloro-3-(4-methyl-piperazin-1-yl)-phenyl ester; compound with (E)-but-2-enedioic acid 177307 4-o-Tolyl-piperazine-1-carboxylic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide; compound with (E)-but-2-enedioic acid 177308 2-[4-(1H-Benzoimidazol-4-yl)-piperazin-1-ylmethyl]-1H-benzoimidazole-4-carboxylic acid (1-aza-bicyclo[2.2.2]oct-3-yl)-amide 177339 4-Phenyl-piperazine-1-carboxylic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide; compound with (E)-but-2-enedioic acid 177347 2-[4-Chloro-3-(4-methyl-piperazin-1-yl)-phenoxy]-1-(4-o-tolyl-piperazin-1-yl)-ethanone; compound with (E)-but-2-enedioic acid 177369 2-(4-Benzo[1,3]dioxol-5-yl-piperazin-1-ylmethyl)-1H-benzoimidazole-4-carboxylic acid (1-aza-bicyclo[2.2.2]oct-3-yl)-amide 177472 19-methoxy-24-methyl-26-[1-phenyl-(E)-methylidene]-4,24-diazaheptacyclo[12.7.3.22,13.01,13.03,11.05,10.016,21]hexacosa-3(11),5(10),6,8,16(21),17,19-heptaen-20-ol 177504 19-methoxy-24-methyl-26-[1-phenyl-(E)-ethylidene]-4,24-diazaheptacyclo[12.7.3.22,13.01,13.03,11.05,10.016,21]hexacosa-3(11),5(10),6,8,16(21),17,19-heptaen-20-ol 177530 2-[4-Methoxy-3-(4-methyl-piperazin-1-yl)-phenylamino]-1-(4-o-tolyl-piperazin-1-yl)-ethanone; compound with but-2-enedioic acid 177565 4-(2,4-Dimethyl-phenyl)-piperazine-1-carboxylic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide; compound with (E)-but-2-enedioic acid 177586 26-[(E)-ethylidene]-19-methoxy-24-methyl-4,24-diazaheptacyclo[12.7.3.22,13.01,13.03,11.05,10.016,21]hexacosa-3(11),5(10),6,8,16(21),17,19-heptaen-20-ol 177599 2-[4-(2-Ethoxy-phenyl)-piperazin-1-ylmethyl]-1H-benzoimidazole-4-carboxylic acid (1-aza-bicyclo[2.2.2]oct-3-yl)-amide 177641 2-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-1H-benzoimidazole-4-carboxylic acid (1-aza-bicyclo[2.2.2]oct-3-yl)-amide 177779 3-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-but-1-ynyl]-pyridine 177840 6-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-but-1-ynyl]-pyridin-3-ylamine 177879 4-Phenyl-1-(4-phenyl-but-3-ynyl)-1,2,3,6-tetrahydro-pyridine 177893 5-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-but-1-ynyl]-pyridin-2-ylamine 177959 4-[3-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tetrahydro-purin-3-yl)-propylcarbamoyl]-benzenesulfonyl fluoride 177972 3-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-but-1-ynyl]-quinoline 177974 1-(4-Benzofuran-5-yl-but-3-ynyl)-4-phenyl-1,2,3,6-tetrahydro-pyridine 177993 H-Ile-Ser-Phe-Lys-AspMet-GIn-Leu-Gly-Arg-OH 178033 1-[4-(4-Methoxy-phenyl)-but-3-ynyl]-4-phenyl-1,2,3,6-tetrahydro-pyridine 178036 4-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-but-1-ynyl]-phenol 178039 4-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-but-1-ynyl]-phenylamine 178040 3-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-but-1-ynyl]-phenylamine 178057 4-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-but-1-ynyl]-isoquinoline 178058 2-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-but-1-ynyl]-pyridine 178059 4-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-but-1-ynyl]-pyridine 178066 1-[4-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-but-3-ynyl]-4-phenyl-1,2,3,6-tetrahydro-pyridine 178068 4-(2-Methoxy-phenyl)-piperazine-1-carboxylic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide; compound with (E)-but-2-enedioic acid 178072 2-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-but-1-ynyl]-phenylamine 178086 4-(2,6-Dimethyl-phenyl)-piperazine-1-carboxylic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide; compound with (E)-but-2-enedioic acid 178087 4-(5,6,7,8-Tetrahydro-naphthalen-1-yl)-piperazine-1-carboxylic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide; compound with (E)-but-2-enedioic acid 178088 4-(4-Methoxy-phenyl)-piperazine-1-carboxylic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide; compound with (E)-but-2-enedioic acid 178089 4-(3-Methoxy-phenyl)-piperazine-1-carboxylic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide; compound with (E)-but-2-enedioic acid 178095 5-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-but-1-ynyl]-1H-indole 178160 2-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-1H-benzoimidazole-4-carboxylic acid (1-aza-bicyclo[2.2.2]oct-3-yl)-amide 178194 3-(1-Propyl-piperidin-3-yl)-benzonitrile 178202 (4aR,8aS)-8a-(3-Hydroxy-phenyl)-3,6-dimethyl-4,4a,5,6,7,8,8a,9-octahydro-1H-pyrrolo[2,3-g]isoquinoline-2-carboxylic acid diethylamide 178203 3-((4aS,11aR)-2-Ethyl-1,2,3,4,5,6,11,11a-octahydro-pyrido[4,3-b]carbazol-4a-yl)-phenol 178227 (+)-Trifluoro-methanesulfonic acid 3-(1-propyl-piperidin-3-yl)-phenyl ester 178254 2-Methyl-6-phenyl-4-((E)-styryl)-pyridine-3,5-dicarboxylic acid diethyl ester 178309 (S)-1-[3-Fluoro-2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-5-phenethyl-3-(3-piperidin-1-yl-propyl)-imidazolidine-2,4-dione 178331 2-Cyclopentyl-6-methyl-4-phenylethynyl-pyridine-3,5-dicarboxylic acid 3-benzyl ester 5-ethyl ester 178343 (4aR,8aS)-6-Cyclopropylmethyl-8a-(3-hydroxy-phenyl)-3-methyl-4,4a,5,6,7,8,8a,9-octahydro-1H-pyrrolo[2,3-g]isoquinoline-2-carboxylic acid diethylamide 178365 2-Cyclobutyl-6-methyl-4-phenylethynyl-pyridine-3,5-dicarboxylic acid 3-benzyl ester 5-ethyl ester 178366 2-Methyl-6-phenyl-4-phenylethynyl-pyridine-3,5-dicarboxylic acid 5-benzyl ester 3-ethyl ester 178389 ethyl 4-ethyl-5-(ethylthiocarbonyl)-2-phenyl-6-propylnicotinate 178392 2,4-Dimethyl-6-phenyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid 5-ethyl ester 3-propyl ester 178428 diethyl 4-ethyl-2-methyl-6-phenyl-1,4-dihydropyridine-3,5-dicarboxylate 178454 (S)-3-(3-Morpholin-4-yl-propyl)-5-phenethyl-1-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-2-thioxo-imidazolidin-4-one 178484 (S)-5-(1H-Indol-3-ylmethyl)-3-piperidin-4-yl-1-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-imidazolidine-2,4-dione 178497 (S)-3-(3-Dimethylamino-propyl)-5-phenyl-1-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-2-thioxo-imidazolidin-4-one 178498 (S)-5-Phenethyl-3-(3-piperidin-1-yl-propyl)-1-{4-[2-(2H-tetrazol-5-yl)-phenyl]-thiophen-2-ylmethyl}-imidazolidine-2,4-dione 178499 (S)-5-Phenethyl-3-(3-piperidin-1-yl-propyl)-1-{5-[2-(2H-tetrazol-5-yl)-phenyl]-thiophen-2-ylmethyl}-imidazolidine-2,4-dione 178508 (S)-5-Phenethyl-3-(3-piperidin-1-yl-propyl)-1-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-imidazolidine-2,4-dione 178509 (S)-5-Phenethyl-3-(3-pyrrolidin-1-yl-propyl)-1-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-imidazolidine-2,4-dione 178519 (S)-3-(3-Dimethylamino-propyl)-5-phenethyl-1-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-2-thioxo-imidazolidin-4-one 178540 (S)-3-(3-Dimethylamino-propyl)-5-phenethyl-1-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-imidazolidine-2,4-dione 178599 (S)-5-Benzyl-3-(3-dimethylamino-propyl)-1-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-2-thioxo-imidazolidin-4-one 178636 diethyl 4-ethyl-2-methyl-6-phenylpyridine-3,5-dicarboxylate 178638 3-ethyl 5-propyl 4,6-dimethyl-2-phenylpyridine-3,5-dicarboxylate 178639 diethyl 2,4-dimethyl-6-phenylpyridine-3,5-dicarboxylate 178683 2-Ethyl-4-methyl-6-phenyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid diethyl ester 178693 2-hydroxyethyl 4,6-diethyl-5-(ethylthiocarbonyl)-2-phenylnicotinate 178703 4-[(4-Cyclopropylmethyl-2,5-dimethyl-piperazin-1-yl)-(3-methoxy-phenyl)-methyl]-N,N-diethyl-benzamide 178731 4-[(4-Butyl-2,5-dimethyl-piperazin-1-yl)-(3-methoxy-phenyl)-methyl]-N,N-diethyl-benzamide 178732 N,N-Diethyl-4-[(3-methoxy-phenyl)-(2,4,5-trimethyl-piperazin-1-yl)-methyl]-benzamide 178740 SID11111434 178741 4,6-Diethyl-5-ethylsulfanylcarbonyl-2-phenyl-nicotinic acid propyl ester 178743 ethyl 4,6-diethyl-5-(ethylthiocarbonyl)-2-phenylnicotinate 178764 4-[(2,5-Dimethyl-piperazin-1-yl)-(3-methoxy-phenyl)-methyl]-N,N-diethyl-benzamide 178866 2-Amino-N-[4-(2-amino-3-phenyl-propionylamino)-butyl]-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionamide 178893 2-Amino-N-{2-[2-amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionylamino]-ethyl}-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionamide 178925 2-Amino-N-{2-[2-amino-3-(4-hydroxy-phenyl)-propionylamino]-ethyl}-3-(4-hydroxy-phenyl)-propionamide 178930 2-Amino-N-{4-[2-amino-3-(4-hydroxy-phenyl)-propionylamino]-butyl}-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionamide 178966 2-Amino-N-[4-(2-amino-3-phenyl-propionylamino)-butyl]-3-phenyl-propionamide 178967 2-Amino-N-{4-[2-amino-3-(4-hydroxy-phenyl)-propionylamino]-butyl}-3-(4-hydroxy-phenyl)-propionamide 178971 2-Amino-N-{6-[2-amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionylamino]-hexyl}-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionamide 178972 2-Amino-N-{8-[2-amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionylamino]-octyl}-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionamide 178983 2-Amino-N-{6-[2-amino-3-(4-hydroxy-phenyl)-propionylamino]-hexyl}-3-(4-hydroxy-phenyl)-propionamide 179010 2-Amino-N-{8-[2-amino-3-(4-hydroxy-phenyl)-propionylamino]-octyl}-3-(4-hydroxy-phenyl)-propionamide 179045 2-Amino-N-{4-[2-amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionylamino]-butyl}-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionamide 179145 4-[[2,5-Dimethyl-4-(2-methyl-allyl)-piperazin-1-yl]-(3-methoxy-phenyl)-methyl]-N,N-diethyl-benzamide 179203 N,N-Diethyl-4-[(4-ethyl-2,5-dimethyl-piperazin-1-yl)-(3-methoxy-phenyl)-methyl]-benzamide 179204 4-[[2,5-Dimethyl-4-(3-phenyl-propyl)-piperazin-1-yl]-(3-methoxy-phenyl)-methyl]-N,N-diethyl-benzamide 179248 4-[(2,5-Dimethyl-4-phenethyl-piperazin-1-yl)-(3-methoxy-phenyl)-methyl]-N,N-diethyl-benzamide 179258 4-[(4-Benzyl-2,5-dimethyl-piperazin-1-yl)-(3-methoxy-phenyl)-methyl]-N,N-diethyl-benzamide 179259 4-[(4-But-2-enyl-2,5-dimethyl-piperazin-1-yl)-(3-methoxy-phenyl)-methyl]-N,N-diethyl-benzamide 179292 Acetic acid 2-hydroxymethyl-4-[(Z)-octadec-9-en-(Z)-ylidene]-5-oxo-tetrahydro-furan-2-ylmethyl ester 179314 4-[(2,5-Dimethyl-4-pentyl-piperazin-1-yl)-(3-methoxy-phenyl)-methyl]-N,N-diethyl-benzamide 179325 Methyl-{4-oxo-2-propyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3,4-dihydro-quinazolin-6-yl}-carbamic acid isobutyl ester 179444 Benzyl-{4-oxo-2-propyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3,4-dihydro-quinazolin-6-yl}-carbamic acid propyl ester 179472 Pentanoic acid benzyl-{4-oxo-2-propyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3,4-dihydro-quinazolin-6-yl}-amide 179613 ethyl 5-(ethylthiocarbonyl)-6-methyl-2-phenyl-4-propylnicotinate 179658 (3-Azepan-1-yl-propyl)-benzo[1,3]dioxol-5-ylmethyl-[3-(3,4-difluoro-phenyl)-isoxazol-5-yl]-amine 179685 (3-Azepan-1-yl-propyl)-benzo[1,3]dioxol-5-ylmethyl-[3-(4-iodo-phenyl)-isoxazol-5-yl]-amine 179798 {4-Oxo-2-propyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3,4-dihydro-quinazolin-6-yl}-carbamic acid isobutyl ester 179799 Benzyl-{4-oxo-2-propyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3,4-dihydro-quinazolin-6-yl}-carbamic acid isobutyl ester 179808 N,N-Diethyl-4-[(4-hexyl-2,5-dimethyl-piperazin-1-yl)-(3-methoxy-phenyl)-methyl]-benzamide 179828 (6aR,10aR)-3-(2-hexyl-1,3-dithian-2-yl)-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol 179856 (6aR,10aR)-3-(2-hexylbenzo[d][1,3]dithiol-2-yl)-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol 179857 (6aR,10aR)-3-(2-hexyl-1,3-dioxolan-2-yl)-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol 180083 (3-Azepan-1-yl-propyl)-benzo[1,3]dioxol-5-ylmethyl-[3-(3,5-dimethoxy-phenyl)-isoxazol-5-yl]-amine 180084 (3-Azepan-1-yl-propyl)-benzo[1,3]dioxol-5-ylmethyl-[3-(3,5-difluoro-phenyl)-isoxazol-5-yl]-amine 180141 (3-Azepan-1-yl-propyl)-benzo[1,3]dioxol-5-ylmethyl-[3-(3,4-dimethoxy-phenyl)-isoxazol-5-yl]-amine 180171 (6aR,10aR)-3-(1-hexylcyclopentyl)-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol 180173 (6aR,10aR)-3-(1,3-dithiolan-2-yl)-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol 180174 (6aR,10aR)-3-(2-hexyl-4,5-dimethyl-1,3-dithiolan-2-yl)-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol 180182 3-{5-[(3-Azepan-1-yl-propyl)-benzo[1,3]dioxol-5-ylmethyl-amino]-isoxazol-3-yl}-benzonitrile 180277 (3-Azepan-1-yl-propyl)-benzo[1,3]dioxol-5-ylmethyl-[3-(3-methoxy-phenyl)-isoxazol-5-yl]-amine 180278 (3-Azepan-1-yl-propyl)-benzo[1,3]dioxol-5-ylmethyl-[3-(2-methoxy-phenyl)-isoxazol-5-yl]-amine 180279 (3-Azepan-1-yl-propyl)-benzo[1,3]dioxol-5-ylmethyl-(3-p-tolyl-isoxazol-5-yl)-amine 180360 (3-Azepan-1-yl-propyl)-benzo[1,3]dioxol-5-ylmethyl-(3-m-tolyl-isoxazol-5-yl)-amine 180390 (3-Azepan-1-yl-propyl)-benzo[1,3]dioxol-5-ylmethyl-[3-(3-nitro-phenyl)-isoxazol-5-yl]-amine 180578 (3-Azepan-1-yl-propyl)-benzo[1,3]dioxol-5-ylmethyl-[3-(3-chloro-phenyl)-isoxazol-5-yl]-amine 180708 (3-Azepan-1-yl-propyl)-benzo[1,3]dioxol-5-ylmethyl-[3-(3-fluoro-phenyl)-isoxazol-5-yl]-amine 180736 (3-Azepan-1-yl-propyl)-benzo[1,3]dioxol-5-ylmethyl-[3-(4-methoxy-phenyl)-isoxazol-5-yl]-amine 180740 (3-Azepan-1-yl-propyl)-benzo[1,3]dioxol-5-ylmethyl-[3-(4-chloro-phenyl)-isoxazol-5-yl]-amine 181230 4-(3-Chloro-4-fluoro-phenylamino)-6,7-dimethoxy-quinoline-3-carbonitrile 181304 4-(4-Chloro-3-trifluoromethyl-phenyl)-1-(3,3-diphenyl-propyl)-piperidin-4-ol 181310 10-hydroxy-17-methoxy-4,13-dimethyl-(13R,17S)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10-trien-14-one 181311 cyprodime 181327 17-cyclopropylmethyl-10-methoxy-13-oxo-(1R,9R,10S)-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-3-yl 3-phenyl-(E)-2-propenoate 181413 4-cyclopropylmethyl-17-(3-phenylpropoxy)-(1S,5R,17S)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10-trien-14-one 181475 1-(3,3-Diphenyl-propyl)-4-(3-trifluoromethyl-phenyl)-piperidin-4-ol 181534 1-benzyloxy-3-spiro[1,3-dihydrobenzo[e]isobenzofuran-3,4'-(hexahydropyridine)]-1-yl-2-propanol 181535 4-phenyl-1-spiro[1,3-dihydrobenzo[e]isobenzofuran-3,4'-(hexahydropyridine)]-1-yl-2-butanol 181536 1-(2-fluorophenoxy)-3-spiro[1,3-dihydrobenzo[e]isobenzofuran-3,4'-(hexahydropyridine)]-1-yl-(2R)-propan-2-ol 181563 1-(5-fluoro-3,4-dihydro-2H-8-chromenyloxy)-3-spiro[1,3-dihydrobenzo[e]isobenzofuran-3,4'-(hexahydropyridine)]-1-yl-2-propanol 181583 4-(4-Chloro-3-trifluoromethyl-phenyl)-1-naphthalen-2-ylmethyl-piperidin-4-ol 181587 4-fluoro-7-[2-hydroxy-3-spiro[1,3-dihydrobenzo[e]isobenzofuran-3,4'-(hexahydropyridine)]-1-ylpropoxy]-1-indanone 181591 3-benzyloxy-17-cyclopropylmethyl-10-methoxy-(1R,9R,10S)-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-13-one 181592 17-cyclopropylmethyl-10-methoxy-3-(3-phenylpropoxy)-(1R,9R,10S)-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-13-one 181596 3-butoxy-17-cyclopropylmethyl-10-methoxy-(1R,9R,10S)-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-13-one 181597 3-butoxy-17-cyclopropylmethyl-10-(3-phenylpropoxy)-(1R,9R,10S)-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-13-one 181599 17-cyclopropylmethyl-3-hydroxy-10-(3-phenylpropoxy)-(1R,9R,10S)-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-13-one 181623 1'-(4-phenylbutyl)spiro[1,3-dihydrobenzo[e]isobenzofuran-3,4'-(hexahydropyridine)] 181627 1-Dimethylamino-3-(1H-indol-4-yloxy)-propan-2-ol 181683 (Z)-[2-(hydroxymethyl)-4-nonylidene-5-oxo-2,3-dihydrofur-2-yl]methyl 2-phenylacetate 181684 Biphenyl-4-carboxylic acid 4-biphenyl-4-ylmethylene-2-hydroxymethyl-5-oxo-tetrahydro-furan-2-ylmethyl ester 181720 17-cyclopropylmethyl-3-hexyloxy-10-methoxy-(1R,9R,10S)-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-13-one 181721 17-cyclopropylmethyl-3-methoxy-10-(3-phenylpropoxy)-(1R,9R,10S)-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-13-one 181727 (Z)-[4-decylidene-2-(hydroxymethyl)-5-oxo-2,3-dihydrofur-2-yl]methyl benzoate 181728 Phenyl-acetic acid 4-decylidene-2-hydroxymethyl-5-oxo-tetrahydro-furan-2-ylmethyl ester 181734 4-(4-Chloro-3-trifluoromethyl-phenyl)-1-(4-trifluoromethyl-benzyl)-piperidin-4-ol 181760 Biphenyl-4-carboxylic acid 4-decylidene-2-hydroxymethyl-5-oxo-tetrahydro-furan-2-ylmethyl ester 181836 1-(2-fluorophenoxy)-3-spiro[1,3-dihydrobenzo[e]isobenzofuran-3,4'-(hexahydropyridine)]-1-yl-(2S)-propan-2-ol 181872 1-phenoxy-3-spiro[1,3-dihydrobenzo[e]isobenzofuran-3,4'-(hexahydropyridine)]-1-yl-(2S)-propan-2-ol 181896 3-(2-Hydroxy-phenyl)-4-[1-(3-hydroxy-propyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]-pyrrole-2,5-dione 181957 Phenyl-acetic acid 4-biphenyl-4-ylmethylene-2-hydroxymethyl-5-oxo-tetrahydro-furan-2-ylmethyl ester 181965 1-(6-fluoro-3,4-dihydro-2H-8-chromenyloxy)-3-spiro[1,3-dihydrobenzo[e]isobenzofuran-3,4'-(hexahydropyridine)]-1-yl-2-propanol 181997 1-(3-ethylphenoxy)-3-spiro[1,3-dihydrobenzo[e]isobenzofuran-3,4'-(hexahydropyridine)]-1-yl-(2S)-propan-2-ol 182056 3,10-Diphenyl-10H-benzo[4,5]imidazo[2,1-c][1,2,4]triazin-4-one 182059 (6aR,12bS)-5,6,6a,7,8,12b-Hexahydro-benzo[a]phenanthridin-11-ol 182155 (2S,3S)-2-Methyl-3,7-diphenyl-5-propoxy-2,7-dihydro-3H-imidazo[1,2-c]pyrazolo[4,3-e]pyrimidine 182156 3-Phenyl-2-(9-phenyl-2-propoxy-9H-purin-6-ylamino)-propan-1-ol 182224 1-Dibutylcarbamoylmethyl-2-(2,2-dimethyl-pentyl)-4-(7-methoxy-benzo[1,3]dioxol-5-yl)-pyrrolidine-3-carboxylic acid 182239 6-Methoxy-5-methyl-1-phenyl-1,5-dihydro-pyrazolo[3,4-d]pyrimidin-4-one 182308 (3-{3-[4-(2-Methoxy-phenyl)-2,5-dioxo-2,5-dihydro-1H-pyrrol-3-yl]-pyrrolo[2,3-b]pyridin-1-yl}-propyl)-carbamic acid tert-butyl ester 182337 Benzoic acid 2-hydroxymethyl-4-nonylidene-5-oxo-tetrahydro-furan-2-ylmethyl ester 182355 Benzoic acid 4-biphenyl-4-ylmethylene-2-hydroxymethyl-5-oxo-tetrahydro-furan-2-ylmethyl ester 182356 Biphenyl-4-carboxylic acid 2-hydroxymethyl-4-nonylidene-5-oxo-tetrahydro-furan-2-ylmethyl ester 182361 (6aR,12bR)-5,6,6a,7,8,12b-Hexahydro-benzo[a]phenanthridin-11-ol 182437 (6aR,12bS)-6-Methyl-5,6,6a,7,8,12b-hexahydro-benzo[a]phenanthridin-11-ol 182445 (6aR,12bS)-5,6,6a,7,8,12b-Hexahydro-benzo[a]phenanthridin-9-ol 182548 (2R,3R)-2-Methyl-3,7-diphenyl-5-propoxy-2,7-dihydro-3H-imidazo[1,2-c]pyrazolo[4,3-e]pyrimidine 182585 (S)-2-Benzyl-7-phenyl-5-propoxy-2,7-dihydro-3H-imidazo[1,2-c]pyrazolo[4,3-e]pyrimidine 182586 (R)-8-Benzyl-3-phenyl-5-propoxy-7,8-dihydro-3H-imidazo[2,1-i]purine 182589 (R)-2-Benzyl-7-phenyl-5-propoxy-2,7-dihydro-3H-imidazo[1,2-c]pyrazolo[4,3-e]pyrimidine 182602 4-(3-Phenoxy-propyl)-1H-imidazole 182793 10-Benzyl-3-phenyl-10H-benzo[4,5]imidazo[2,1-c][1,2,4]triazin-4-one 182814 SID11112867 182843 2-Amino-N-[(R)-2-((R)-3a-benzyl-2-methyl-3-oxo-2,3,3a,4,6,7-hexahydro-pyrazolo[4,3-c]pyridin-5-yl)-1-benzyloxymethyl-2-oxo-ethyl]-2-methyl-propionamide 182871 (6aR,12bR)-5,6,6a,7,8,12b-Hexahydro-benzo[a]phenanthridin-9-ol 182874 9-butyl-8-(3,4,5-trimethoxybenzyl)-9H-purin-6-amine 182915 3-Phenyl-2-(9-phenyl-2-propoxy-9H-purin-6-ylamino)-propan-1-ol 182940 (S)-8-Benzyl-3-phenyl-5-propoxy-7,8-dihydro-3H-imidazo[2,1-i]purine 182948 (6aR,12bS)-6-Propyl-5,6,6a,7,8,12b-hexahydro-benzo[a]phenanthridin-11-ol 183064 5,7-Dimethyl-1-phenyl-1,7-dihydro-pyrazolo[3,4-d]pyrimidine-4,6-dione 183066 5-Methyl-1-phenyl-7-propyl-1,7-dihydro-pyrazolo[3,4-d]pyrimidine-4,6-dione 183101 6-(2,6-dichlorophenyl)-2-(4-hydroxyphenylamino)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one 183102 6-(2,6-dichlorophenyl)-2-(3-hydroxyphenylamino)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one 183112 5-Methyl-1-phenyl-6-propoxy-1,5-dihydro-pyrazolo[3,4-d]pyrimidin-4-one 183125 9-Butyl-8-(2,5-dimethoxy-benzyl)-9H-purin-6-ylamine 183155 6-(2,6-dichlorophenyl)-2-(3-(hydroxymethyl)phenylamino)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one 183181 6-(2,6-dichlorophenyl)-8-methyl-2-(p-tolylamino)pyrido[2,3-d]pyrimidin-7(8H)-one 183220 6-(2,6-Dichloro-phenyl)-2-[4-(2-diethylamino-ethoxy)-phenylamino]-8-ethyl-8H-pyrido[2,3-d]pyrimidin-7-one 183261 (S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-bicyclo[3.2.1]octan-6-ol 183936 (R)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-bicyclo[3.2.1]octan-6-ol 183972 (S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-bicyclo[3.2.1]octane-6-carboxylic acid 184086 (5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenesulfonyl fluoride 184158 7-nitro-3-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinoline 184292 (R)-1-(2,6-difluorobenzyl)-5-(3-methoxyphenyl)-6-methyl-3-(2-(methyl(pyridin-2-ylmethyl)amino)propyl)pyrimidine-2,4(1H,3H)-dione 184364 (S)-1-(6-chloro-5-(2-(pyridin-4-yl)vinyl)pyridin-3-yloxy)propan-2-amine 184427 SID26752042 184544 5-Methoxy-3-piperazin-1-yl-benzo[d]isothiazole (1.1HCl 0.15H2O) 184677 (R)-1-(2,6-difluorobenzyl)-5-(3-methoxyphenyl)-6-methyl-3-(2-(methyl(2-(pyridin-2-yl)ethyl)amino)propyl)pyrimidine-2,4(1H,3H)-dione 184788 4-Methoxy-3-piperazin-1-yl-benzo[d]isothiazole (1.1HCl) 184810 7-bromo-3-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinoline 184827 (2S,3R,4R,5R)-2,5-Bis-(3,4-dimethoxy-phenyl)-3,4-dimethyl-tetrahydro-furan 185299 1-Benzyl-7-phenyl-1H-1,3,4b,9-tetraaza-fluorene-2,4-dione 185306 1,3-Dibenzyl-1H-1,3,4b,9-tetraaza-fluorene-2,4-dione 185337 1-Benzyl-7-methoxy-3-propyl-1H-1,3,4b,9-tetraaza-fluorene-2,4-dione 185339 1-Benzyl-7-phenyl-3-propyl-1H-1,3,4b,9-tetraaza-fluorene-2,4-dione 185340 1-Benzyl-3-(4-methoxy-benzyl)-1H-1,3,4b,9-tetraaza-fluorene-2,4-dione 185409 1-Benzyl-3-cyclopropylmethyl-1H-1,3,4b,9-tetraaza-fluorene-2,4-dione 185410 1-Benzyl-3-ethyl-1H-1,3,4b,9-tetraaza-fluorene-2,4-dione 185471 1-(3-Methyl-benzyl)-3-propyl-1H-1,3,4b,9-tetraaza-fluorene-2,4-dione 185479 1-Benzyl-3-prop-2-ynyl-1H-1,3,4b,9-tetraaza-fluorene-2,4-dione 185480 3-Allyl-1-benzyl-1H-1,3,4b,9-tetraaza-fluorene-2,4-dione 185503 1-Methyl-3-propyl-1H-1,3,4b,9-tetraaza-fluorene-2,4-dione 185504 4-(1-Benzyl-2,4-dioxo-1,4-dihydro-2H-1,3,4b,9-tetraaza-fluoren-3-yl)-but-2-enoic acid methyl ester 185508 1-(4-Methoxy-benzyl)-3-propyl-1H-1,3,4b,9-tetraaza-fluorene-2,4-dione 185657 2-(7-Amino-imidazo[4,5-b]pyridin-3-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 185728 1-{4-[3-(1H-Imidazol-4-yl)-propoxy]-phenyl}-ethanone 185824 1-Benzyl-1H-1,3,4b,9-tetraaza-fluorene-2,4-dione 185825 1-Benzyl-7-methoxy-1H-1,3,4b,9-tetraaza-fluorene-2,4-dione 185929 1-Benzyl-3-cyclohexylmethyl-1H-1,3,4b,9-tetraaza-fluorene-2,4-dione 185961 1-Benzyl-3-isobutyl-1H-1,3,4b,9-tetraaza-fluorene-2,4-dione 185980 [(1S,3R)-3-Amino-1-hydroxy-5-(4-octyl-phenyl)-pentyl]-phosphonic acid 186010 [(R)-3-Amino-1-(R)-hydroxy-5-(4-octyl-phenyl)-pentyl]-phosphonic acid 186011 [(1R,3S)-3-Amino-1-hydroxy-5-(4-octyl-phenyl)-pentyl]-phosphonic acid 186026 1-Benzyl-7-tert-butyl-1H-1,3,4b,9-tetraaza-fluorene-2,4-dione 186088 1-Benzyl-7-tert-butyl-3-propyl-1H-1,3,4b,9-tetraaza-fluorene-2,4-dione 186120 1-Benzyl-3-propyl-1H-1,3,4b,9-tetraaza-fluorene-2,4-dione 186153 3-{(S)-7-[3-(2-Cyclopropylmethyl-3-methoxy-4-methylcarbamoyl-phenoxy)-propoxy]-8-propyl-chroman-2-yl}-propionic acid 186156 (E)-3-{6-(3-Amino-benzenesulfinylmethyl)-3-[8-(4-methoxy-phenyl)-octyloxy]-pyridin-2-yl}-acrylic acid 186191 2-(4-Fluoro-phenyl)-4-methoxy-3-pyridin-4-yl-1H-pyrrolo[2,3-b]pyridin-6-ylamine 186249 [3-Amino-2-hydroxy-5-(4-octyl-phenyl)-pentyl]-phosphonic acid; compound with [(E)-3-amino-5-(4-octyl-phenyl)-pent-1-enyl]-phosphonic acid 186278 [3-Amino-2-hydroxy-5-(4-octyl-phenyl)-pentyl]-phosphonic acid 186313 [3-Amino-5-(4-octyl-phenyl)-pentyl]-phosphonic acid 186330 2-amino-2-(hydroxymethyl)-4-(4-octylphenyl)butyl dihydrogen phosphate 186362 [3-Amino-3-hydroxymethyl-5-(4-octyl-phenyl)-pentyl]-phosphonic acid 186363 Phosphoric acid mono-[2-amino-4-(4-octyl-phenyl)-butyl] ester 186392 4-tert-Butyl-N-{6-[2-(5-hydroxymethyl-pyrimidin-2-yloxy)-ethoxy]-5-p-tolyl-pyrimidin-4-yl}-benzenesulfonamide 186442 [(1S,3S)-3-Amino-1-hydroxy-5-(4-octyl-phenyl)-pentyl]-phosphonic acid 186462 [3-Amino-1-hydroxy-5-(4-octyl-phenyl)-pentyl]-phosphonic acid 186506 3-Amino-5-(4-octyl-phenyl)-pentane-1-sulfonic acid 186507 3-amino-5-(4-octylphenyl)pentanoic acid 186508 4-amino-6-(4-octylphenyl)hexanoic acid 186705 1-(3-Chloro-benzyl)-8-phenyl-3,7-dihydro-purine-2,6-dione 187049 11-{2-[6-({8-[(6-Amino-hexyl)-methyl-amino]-octyl}-methyl-amino)-hexylamino]-acetyl}-5,11-dihydro-benzo[e]pyrido[3,2-b][1,4]diazepin-6-one 187088 11-{2-[6-methyl(8-methyl{6-[2-oxo-2-(6-oxo-6,11-dihydro-5H-benzo[e]pyrido[3,2-b][1,4]diazepin-11-yl)ethylamino]hexyl}aminooctyl)aminohexylamino]acetyl}-6,11-dihydro-5H-benzo[e]pyrido[3,2-b][1,4]diazepin-6-one 187230 tripitramine 187244 N-{6-[2-(5-Bromo-pyrimidin-2-yloxy)-ethoxy]-5-p-tolyl-pyrimidin-4-yl}-4-(2-hydroxy-1,1-dimethyl-ethyl)-benzenesulfonamide 187259 2-(4-{6-[2-(5-Bromo-pyrimidin-2-yloxy)-ethoxy]-5-p-tolyl-pyrimidin-4-ylsulfamoyl}-phenyl)-2-methyl-propionic acid. CH2Cl2 187303 N-{6-[2-(5-Bromo-pyrimidin-2-yloxy)-ethoxy]-5-p-tolyl-pyrimidin-4-yl}-4-tert-butyl-benzenesulfonamide 187354 4-tert-Butyl-N-{5-(4-hydroxymethyl-phenyl)-6-[2-(5-methylsulfanyl-pyrimidin-2-yloxy)-ethoxy]-pyrimidin-4-yl}-benzenesulfonamide 187685 8-(3-Phenoxy-benzyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 187686 1-Phenyl-8-[1,3,4]thiadiazolo[3,4-a]pyridazin-6-ylmethyl-1,3,8-triaza-spiro[4.5]decan-4-one 187688 8-Benzo[1,3]dioxol-5-ylmethyl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 187706 4-Oxo-1-phenyl-1,3,8-triaza-spiro[4.5]decane-8-carboxylic acid indan-1-yl ester 187707 4-Oxo-1-phenyl-1,3,8-triaza-spiro[4.5]decane-8-carboxylic acid 3-phenoxy-benzyl ester 187728 2-[8-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-4-oxo-1-phenyl-1,3,8-triaza-spiro[4.5]dec-3-yl]-N-methyl-acetamide 187736 N-[6-[2-(5-Bromo-pyrimidin-2-yloxy)-ethoxy]-5-(4-hydroxymethyl-phenyl)-pyrimidin-4-yl]-4-tert-butyl-benzenesulfonamide 187956 1-[1-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-piperidin-4-yl]-6-methyl-1,3-dihydro-benzoimidazol-2-one 188001 11-(2-{6-[(8-{[6-(2-Methoxy-benzylamino)-hexyl]-methyl-amino}-octyl)-methyl-amino]-hexylamino}-acetyl)-5,11-dihydro-benzo[e]pyrido[3,2-b][1,4]diazepin-6-one 188079 dimethyl2,6-dimethyl-4-{3-nitrileimino[3-(4-phenylhexahydro-1-pyridinyl)propylamino]methylaminophenyl}-1,4-dihydro-3,5-pyridinedicarboxylate 188114 [1-(2-Benzyl-1,3-dioxo-4a(R)-octahydro-pyrido[1,2-c]pyrimidin-5(S)-ylcarbamoyl)-2-(1H-indol-3-yl)-ethyl]-carbamic acid tert-butyl ester 188115 [(S)-1-((4aR,5R)-2-Benzyl-1,3-dioxo-octahydro-pyrido[1,2-c]pyrimidin-5-ylcarbamoyl)-2-(1H-indol-3-yl)-ethyl]-carbamic acid tert-butyl ester 188116 [(S)-1-((4aS,5S)-2-Benzyl-1,3-dioxo-octahydro-pyrido[1,2-c]pyrimidin-5-ylcarbamoyl)-2-(1H-indol-3-yl)-ethyl]-carbamic acid tert-butyl ester 188138 4-Oxo-1-phenyl-1,3,8-triaza-spiro[4.5]decane-8-carboxylic acid benzo[1,3]dioxol-5-ylmethyl ester 188139 4-Oxo-1-phenyl-1,3,8-triaza-spiro[4.5]decane-8-carboxylic acid 6-chloro-benzo[1,3]dioxol-5-ylmethyl ester 188141 3-Methylcarbamoylmethyl-4-oxo-1-phenyl-1,3,8-triaza-spiro[4.5]decane-8-carboxylic acid 6-chloro-benzo[1,3]dioxol-5-ylmethyl ester 188150 1-[1-(6-Nitro-benzo[1,3]dioxol-5-ylmethyl)-1,2,3,6-tetrahydro-pyridin-4-yl]-1,3-dihydro-benzoimidazol-2-one 188187 1-{3-[(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-amino]-propyl}-1,3-dihydro-benzoimidazol-2-one 188226 1-[1-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-piperidin-4-yl]-1,3-dihydro-benzoimidazol-2-one 188252 [3-(2-Oxo-2,3-dihydro-benzoimidazol-1-yl)-propyl]-carbamic acid 6-chloro-benzo[1,3]dioxol-5-ylmethyl ester 188396 4-(3-{3-[3-(4-Cyclohexyl-piperazin-1-yl)-propyl]-thioureido}-phenyl)-2,6-dimethyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid dimethyl ester 188414 4-[3-(3-{3-[4-(3-Methoxy-phenyl)-piperidin-1-yl]-propyl}-thioureido)-phenyl]-2,6-dimethyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid dimethyl ester 188415 1-(3-{3-[3-(4-Cyclohexyl-piperazin-1-yl)-propyl]-ureido}-phenyl)-3,5-dimethyl-1,4-dihydro-pyrazine-2,6-dicarboxylic acid dimethyl ester 188436 4-(2-Oxo-2,3-dihydro-benzoimidazol-1-yl)-piperidine-1-carboxylic acid 6-chloro-benzo[1,3]dioxol-5-ylmethyl ester 188462 dimethyl1-{3-[3-[4-(tert-butyl)hexahydro-1-pyridinyl]propylamino(nitrileimino)methylamino]phenyl}-3,5-dimethyl-1,4-dihydro-2,6-pyrazinedicarboxylate 188463 1-[3-(3-{3-[4-(3-Methoxy-phenyl)-piperidin-1-yl]-propyl}-thioureido)-phenyl]-3,5-dimethyl-1,4-dihydro-pyrazine-2,6-dicarboxylic acid dimethyl ester 188469 4-(3-{3-[3-(4-Cyclohexyl-piperazin-1-yl)-propyl]-ureido}-phenyl)-2,6-dimethyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid dimethyl ester 188505 1-[1-(2-Chloro-4-methyl-benzyl)-piperidin-4-yl]-1,3-dihydro-benzoimidazol-2-one 188507 1-[1-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-piperidin-4-yl]-1,4-dihydro-quinoxaline-2,3-dione 188533 N-(3-chloro-2-methylphenyl)-2-(N-(4-methoxyphenyl)phenylsulfonamido)acetamide 188581 1-[3-(3-{3-[4-(3-Methoxy-phenyl)-piperidin-1-yl]-propyl}-ureido)-phenyl]-3,5-dimethyl-1,4-dihydro-pyrazine-2,6-dicarboxylic acid dimethyl ester 188588 dimethyl3,5-dimethyl-1-{3-nitrileimino[3-(4-phenylhexahydro-1-pyridinyl)propylamino]methylaminophenyl}-1,4-dihydro-2,6-pyrazinedicarboxylate 188590 6,7-Dimethoxy-3-[4-(4-methoxy-phenyl)-thiazol-2-ylamino]-3H-isobenzofuran-1-one 188714 4-[4,4-Bis-(4-fluoro-phenyl)-butyl]-piperazine-1-carboxylic acid 2-(4-cyano-phenyl)-ethyl ester 188730 1H-Indole-2-carboxylic acid ((R)-1-methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-amide 188756 [(R)-1-((4aS,5R)-2-Benzyl-1,3-dioxo-octahydro-pyrido[1,2-c]pyrimidin-5-ylcarbamoyl)-2-(1H-indol-3-yl)-ethyl]-carbamic acid tert-butyl ester 188836 [(R)-1-((4aR,5R)-2-Benzyl-1,3-dioxo-octahydro-pyrido[1,2-c]pyrimidin-5-ylcarbamoyl)-2-(1H-indol-3-yl)-ethyl]-carbamic acid tert-butyl ester 188837 [(R)-1-((4aS,5S)-2-Benzyl-1,3-dioxo-octahydro-pyrido[1,2-c]pyrimidin-5-ylcarbamoyl)-2-(1H-indol-3-yl)-ethyl]-carbamic acid tert-butyl ester 188863 pGlu-Leu-Tyr-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Tyr-Ile-Leu 188869 N'-(2-hydroxybenzylidene)-2-(N-p-tolylphenylsulfonamido)acetohydrazide 188871 8-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 188877 [(S)-1-((4aS,5R)-2-Benzyl-1,3-dioxo-octahydro-pyrido[1,2-c]pyrimidin-5-ylcarbamoyl)-2-(1H-indol-3-yl)-ethyl]-carbamic acid tert-butyl ester 188955 5-Ethoxymethyl-5-hydroxymethyl-3-tetradec-(E)-ylidene-dihydro-furan-2-one 188982 Acetic acid 2-hydroxymethyl-4-tetradec-(E)-ylidene-tetrahydro-furan-2-ylmethyl ester 188985 5-Ethoxymethyl-5-hydroxymethyl-3-tetradec-(Z)-ylidene-dihydro-furan-2-one 188997 4-(3-Phenyl-propyl)-piperazine-1-carboxylic acid 2-(4-cyano-phenyl)-ethyl ester 189005 diethyl 2-(2-phenylacetamido)-4,5-dihydrothieno[2,3-c]pyridine-3,6(7H)-dicarboxylate 189033 {[(2-Benzoylamino-5-bromo-phenyl)-phenyl-methyl]-amino}-acetic acid ethyl ester 189039 (2R,8S,8aR)-2-Benzyl-8-[(R)-2-tert-butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-3-oxo-octahydro-indolizine-2-carboxylic acid methyl ester 189040 (2S,8S,8aR)-2-Benzyl-8-[(S)-2-tert-butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-3-oxo-octahydro-indolizine-2-carboxylic acid methyl ester 189057 (R)-1-(1-(3,3-dimethyl-2-oxobutyl)-2-oxo-5-(pyridin-2-yl)-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-(3-(methylamino)phenyl)urea 189066 1-[4-(3-Benzyloxy-4-methoxy-benzyl)-piperazin-1-yl]-3-(3-methyl-indol-1-yl)-propan-1-one 189098 1-{4-[3-(4-Chloro-phenoxy)-benzyl]-piperazin-1-yl}-3-(4-methoxy-phenylsulfanyl)-propan-1-one 189133 1-{4-[4,4-Bis-(4-fluoro-phenyl)-butyl]-piperazin-1-yl}-4-phenyl-butan-1-one 189135 4-[4,4-Bis-(4-fluoro-phenyl)-butyl]-piperazine-1-carboxylic acid [2-(4-ethoxy-phenyl)-ethyl]-amide 189176 4-(3-Phenyl-propyl)-piperazine-1-carboxylic acid 2-(4-ethoxy-phenyl)-ethyl ester 189230 1-{4-[4,4-Bis-(4-fluoro-phenyl)-butyl]-piperazin-1-yl}-3-(4-fluoro-phenyl)-propan-1-one 189267 4-[4,4-Bis-(4-fluoro-phenyl)-butyl]-piperazine-1-carboxylic acid 2-(4-fluoro-phenyl)-ethyl ester 189337 Trifluoro-methanesulfonic acid 6-dipropylamino-5,6,7,8-tetrahydro-naphthalen-2-yl ester 189344 Trifluoro-methanesulfonic acid 6-dipropylamino-5,6,7,8-tetrahydro-naphthalen-1-yl ester 189383 Trifluoro-methanesulfonic acid 7-dipropylamino-5,6,7,8-tetrahydro-naphthalen-2-yl ester 189637 {1-[4,4-Bis-(4-fluoro-phenyl)-butyl]-piperidin-4-yl}-carbamic acid 2-(4-cyano-phenyl)-ethyl ester 189664 (2S,5S,8R,13S)-13-amino-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 189698 (2S,5S,8R,12S)-12-amino-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 189733 1-{6-[(3R,4S)-3-(Benzo[1,3]dioxol-5-yloxymethyl)-4-(4-fluoro-phenyl)-piperidin-1-yl]-hexylamino}-3-(1H-indol-4-yloxy)-propan-2-ol 189769 1-(1H-Indol-4-yloxy)-3-[3-phenyl-3-(4-trifluoromethyl-phenoxy)-propylamino]-propan-2-ol 189899 (S)-1-(Naphthalen-1-yloxy)-3-[(S)-3-phenyl-3-(4-trifluoromethyl-phenoxy)-propylamino]-propan-2-ol 189934 (R)-1-(1H-Indol-4-yloxy)-3-[(S)-3-phenyl-3-(4-trifluoromethyl-phenoxy)-propylamino]-propan-2-ol 189960 N-[5-(S),8-(R)-dibenzyl-2-(S)-(1H-indol-3-ylmethyl)-3,6,11,14-tetraoxo-1,4,7,10-tetraaza-cyclotetradec-12-(R)-yl]-2-morpholin-4-yl-acetamide 189963 (1S,2R)-2-{[2-Hydroxy-3-(1H-indol-4-yloxy)-propylamino]-methyl}-1-phenyl-cyclopropanecarboxylic acid diethylamide 189994 (S)-1-(1H-Indol-4-yloxy)-3-[(S)-3-phenyl-3-(4-trifluoromethyl-phenoxy)-propylamino]-propan-2-ol 190006 1-(2-Cyclopentyl-phenoxy)-3-[3-phenyl-3-(4-trifluoromethyl-phenoxy)-propylamino]-propan-2-ol 190074 SID11113889 190271 Acetic acid (1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-9-acetoxy-4a,7b-dihydroxy-3-hydroxymethyl-1,1,6,8-tetramethyl-5-oxo-1,1a,1b,4,4a,5,7a,7b,8,9-decahydro-cyclopropa[3,4]benzo[1,2-e]azulen-9a-yl ester 190286 (S)-1-[(3S,4R)-3-(Benzo[1,3]dioxol-5-yloxymethyl)-4-(4-fluoro-phenyl)-piperidin-1-yl]-3-(1H-indol-4-yloxy)-propan-2-ol 190306 (R)-1-(Naphthalen-1-yloxy)-3-[(S)-3-phenyl-3-(4-trifluoromethyl-phenoxy)-propylamino]-propan-2-ol 190315 (R)-1-[(3S,4R)-3-(Benzo[1,3]dioxol-5-yloxymethyl)-4-(4-fluoro-phenyl)-piperidin-1-yl]-3-(1H-indol-4-yloxy)-propan-2-ol 190414 (2E)-2-[(5-hydroxy-1H-indol-3-yl)methylene]-N-pentylhydrazinecarboximidamide 190581 2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-6,7-dimethoxy-quinolin-4-ylamine 190655 1-(Naphthalen-1-yloxy)-3-{6-[3-phenyl-3-(4-trifluoromethyl-phenoxy)-propylamino]-hexylamino}-propan-2-ol 190656 1-{6-[(3R,4S)-3-(Benzo[1,3]dioxol-5-yloxymethyl)-4-(4-fluoro-phenyl)-piperidin-1-yl]-hexylamino}-3-(naphthalen-1-yloxy)-propan-2-ol 190658 6-Chloro-3-methyl-9-(3-methyl-but-2-enyloxy)-2,3,4,5-tetrahydro-1H-benzo[d]azepine 191163 SID26725296 191342 SID29215232 191481 (2R,3R,4S,5R)-2-[2-Chloro-6-((R)-1-methyl-2-phenoxy-ethylamino)-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 191524 (2R,3R,4S,5R)-2-[2-Chloro-6-((S)-1-methyl-2-phenoxy-ethylamino)-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 191569 (2R,3R,4S,5R)-2-[2-Chloro-6-(1-methyl-2-phenoxy-ethylamino)-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 191633 1-Methyl-2-phenyl-1,4,6,7-tetrahydro-1,3,4,5a,8-pentaaza-as-indacen-5-one 191734 2-Hexyloxy-3-(1-methyl-1,2,5,6-tetrahydro-pyridin-3-yl)-pyrazine 191834 1-(2,6-Difluoro-benzyl)-3-((S)-2-dimethylamino-3-phenyl-propyl)-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 191841 (3-Bromo-phenyl)-(5-nitro-quinazolin-4-yl)-amine 191845 3-((S)-2-Amino-3-phenyl-propyl)-1-(2,6-difluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 191913 3-((R)-2-Amino-3-phenyl-propyl)-1-(2,6-difluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 191929 (S)-1-(2,6-difluorobenzyl)-5-(2-fluoro-3-methoxyphenyl)-6-methyl-3-(2-(methylamino)-3-phenylpropyl)pyrimidine-2,4(1H,3H)-dione 191996 (-)-trans 42s,5S)-2-[3-[(2-Oxopropyl)sulfony1]-4-n-propoxy-5-[3-(phosphonooxy)propoxy]phenyl]-5-(3,4,5-trimethoxypheny1) tetrahydrofuran Monopotassium Salt 192029 3-(4-(2-(6-amino-9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxytetrahydrofuran-2-yl)-9H-purin-2-ylamino)ethyl)phenyl)propanoic acid 192091 (2R,3R,4R,5R)-5-(6-Cyclohexylamino-purin-9-yl)-2-hydroxymethyl-4-methoxy-tetrahydro-furan-3-ol 192098 Metrifudil 192100 (2S,3S,4R,5R)-2-Chloromethyl-5-[2-chloro-6-(4-phenylsulfanyl-piperidin-1-ylamino)-purin-9-yl]-tetrahydro-furan-3,4-diol 192127 2-Hydroxy-4-(4-nonyl-benzylamino)-butyric acid 192163 (2R,3R,4S,5R)-2-[6-((1R,2R)-2-Hydroxy-cyclopentylamino)-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 192168 Methyl-[3-(4-nonyl-benzylamino)-propyl]-phosphinic acid 192202 3-Hydroxy-4-(4-nonyl-benzylamino)-butyric acid 192335 1-{3-(3-Hydroxy-propoxy)-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimethoxy-phenyl)-tetrahydro-furan-2-yl]-benzenesulfonyl}-propan-2-one 192343 Phosphoric acid mono-[1-amino-1-hydroxymethyl-3-(4-octyl-phenyl)-propyl] ester 192344 (3-Amino-pentadecyl)-phosphonic acid 192376 1-(2,6-Difluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-3-((R)-4-methyl-2-methylamino-pentyl)-1H-pyrimidine-2,4-dione 192444 3-((R)-2-Amino-3-methyl-butyl)-1-(2,6-difluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 192449 2-Hydroxymethyl-5-[6-(1-methyl-2-phenyl-ethylamino)-purin-9-yl]-tetrahydro-furan-3,4-diol 192618 3-((R)-2-Amino-4-methyl-pentyl)-1-(2,6-difluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 192655 3-((S)-2-Amino-4-methyl-pentyl)-1-(2,6-difluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 192663 3-((R)-2-Amino-2-cyclohexyl-ethyl)-1-(2,6-difluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 192690 (R)-5-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimethoxy-phenyl)-tetrahydro-furan-2-yl]-benzenesulfonyl}-4-methyl-pentan-1-ol 192724 1-{3-(3-Morpholin-4-yl-propoxy)-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimethoxy-phenyl)-tetrahydro-furan-2-yl]-benzenesulfonyl}-propan-2-one 192752 3-((R)-2-Amino-propyl)-1-(2,6-difluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 192827 3-(tetradecylamino)propylphosphonic acid 192828 (3-Tridecylamino-propyl)-phosphonic acid 192854 (3-Dodecylamino-propyl)-phosphonic acid 192933 1-{3-(3-Imidazol-1-yl-propoxy)-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimethoxy-phenyl)-tetrahydro-furan-2-yl]-benzenesulfonyl}-propan-2-one 192984 {3-[4-(5-Heptyl-[1,2,4]oxadiazol-3-yl)-benzylamino]-propyl}-phosphonic acid 193008 3-Fluoro-4-(4-nonyl-benzylamino)-butyric acid 193037 2,2-Difluoro-4-(4-nonyl-benzylamino)-butyric acid 193064 {3-[4-(2-Heptyl-2H-tetrazol-5-yl)-benzylamino]-propyl}-phosphonic acid 193065 [3-(4-Nonanoyl-benzylamino)-propyl]-phosphonic acid 193087 R-(-)-11-hydroxy-aporphine 193099 3-((S)-2-Amino-3-methyl-butyl)-1-(2,6-difluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 193114 2-phenyl-3-(pyrimidin-4-yl)imidazo[1,2-a]pyrimidin-7-amine 193119 Tetradecanoic acid (R)-2-hydroxymethyl-5-oxo-tetrahydro-furan-2-ylmethyl ester 193127 [3-(3-Bromo-4-hexyloxy-5-methoxy-benzylamino)-propyl]-phosphonic acid 193134 (S)-5-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimethoxy-phenyl)-tetrahydro-furan-2-yl]-benzenesulfonyl}-4-methyl-pentan-1-ol 193150 [3-(4-Nonyl-benzylamino)-propyl]-phosphonic acid 193180 3-(2-Pyrrolidin-1-yl-ethyl)-5-[1,2,4]triazol-4-yl-1H-indole 193181 3-[3-(4-Phenethyl-piperazin-1-yl)-propyl]-5-[1,2,4]triazol-4-yl-1H-indole 193184 {3-[4-(4-Heptyl-phenyl)-butylamino]-propyl}-phosphonic acid 193185 [3-(4-Octyloxy-benzylamino)-propyl]-phosphonic acid 193209 {3-[4-(1-Hydroxy-nonyl)-benzylamino]-propyl}-phosphonic acid 193210 {3-[(4'-Hexyl-biphenyl-4-ylmethyl)-amino]-propyl}-phosphonic acid 193215 3-[3-(4-Methyl-piperazin-1-yl)-propyl]-5-[1,2,4]triazol-4-yl-1H-indole 193225 3-(3-bromo-5-methoxy-4-(octyloxy)benzylamino)propylphosphonic acid 193241 [3-(4-Nonyloxy-benzylamino)-propyl]-phosphonic acid 193244 2-Phenyl-3-{2-[(S)-(1,2,3,4-tetrahydro-naphthalen-1-yl)amino]-pyridin-4-yl}-imidazo[1,2-a]pyrimidin-7-ylamine 193286 2-benzyl-7-(4-fluorophenyl)-8-(pyridin-4-yl)-3,6-dihydroimidazo[4,5-e]indole 193289 3-(2-(benzylamino)pyridin-4-yl)-2-(4-fluorophenyl)imidazo[1,2-a]pyrimidin-7-amine 193290 2-Phenyl-3-[2-((S)-1-phenyl-ethylamino)-pyridin-4-yl]-imidazo[1,2-a]pyrimidin-7-ylamine 193294 [3-(10-Phenyl-decylamino)-propyl]-phosphonic acid 193331 (3-Pentadecylamino-propyl)-phosphonic acid 193368 2-(4-Fluoro-phenyl)-3-pyridin-4-yl-imidazo[1,2-a]pyrimidin-7-ylamine 193371 {3-[3-(4-Heptyl-phenyl)-propylamino]-propyl}-phosphonic acid 193372 {3-[2-(4-Octyl-phenyl)-ethylamino]-propyl}-phosphonic acid 193373 (3-Hexadecylamino-propyl)-phosphonic acid 193377 (R)-6-Isopropyl-11-methoxy-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline 193382 3-(3-{4-[2-(2-Fluoro-phenyl)-ethyl]-piperazin-1-yl}-propyl)-5-[1,2,4]triazol-4-yl-1H-indole 193391 (3-Amino-hexadecyl)-phosphonic acid 193401 (3-Amino-heptadecyl)-phosphonic acid 193403 (R)-6-Methyl-11-vinyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline 193412 N-[3-(2-{4-[3-(5-[1,2,4]Triazol-4-yl-1H-indol-3-yl)-propyl]-piperazin-1-yl}-ethyl)-phenyl]-acetamide 193454 11-Methoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline 193455 Trifluoro-methanesulfonic acid (R)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-yl ester 193462 [3-(3-Fluoro-4-octyloxy-benzylamino)-propyl]-phosphonic acid 193473 (3-Amino-octadecyl)-phosphonic acid 193483 1-((R)-6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-yl)-ethanone 193490 (R)-11-Methoxy-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline 193500 (3-Amino-13-phenyl-tridecyl)-phosphonic acid 193730 Acetic acid (R)-2-hydroxymethyl-4-[(Z)-octadec-9-en-(Z)-ylidene]-5-oxo-tetrahydro-furan-2-ylmethyl ester 193755 2-Phenyl-3-[2-((S)-1-phenyl-ethylamino)-pyrimidin-4-yl]-imidazo[1,2-a]pyrimidin-7-ylamine 193790 2-Phenyl-3-[2-((R)-1-phenyl-ethylamino)-pyrimidin-4-yl]-imidazo[1,2-a]pyrimidin-7-ylamine 193791 3-(2-Methoxy-pyrimidin-4-yl)-2-phenyl-imidazo[1,2-a]pyrimidin-7-ylamine 193829 3-(2-Methylsulfanyl-pyrimidin-4-yl)-2-phenyl-imidazo[1,2-a]pyrimidin-7-ylamine 193840 (R)-6-Isopropyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-ol 193843 Acetic acid (R)-2-hydroxymethyl-4-[(Z)-octadec-9-en-(E)-ylidene]-5-oxo-tetrahydro-furan-2-ylmethyl ester 193857 (S)-3-(2-(1-methoxypropan-2-ylamino)pyridin-4-yl)-2-phenylimidazo[1,2-a]pyrimidin-7-amine 193927 (R)-11-(2-Methoxy-phenyl)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline 193941 (R)-6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-11-carbonitrile 193964 6-[2-(2-Chloro-4-fluoro-phenyl)-imidazo[1,2-a]pyridin-3-yl]-2-(2,6-dichloro-phenyl)-4,5-dihydro-2H-pyridazin-3-one 193983 (R)-11-ethyl-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline 194012 3-[2-(4-Methyl-piperazin-1-yl)-ethyl]-5-[1,2,4]triazol-4-yl-1H-indole 194136 2-(2-chlorophenyl)-6-(2-(3-(trifluoromethyl)phenyl)imidazo[1,2-a]pyridin-3-yl)-4,5-dihydropyridazin-3(2H)-one 194174 6-[2-(2-Chloro-4-fluoro-phenyl)-imidazo[1,2-a]pyridin-3-yl]-2-(2-chloro-phenyl)-2H-pyridazin-3-one 194238 2-(2,6-dichlorophenyl)-6-(2-(4-fluorophenyl)imidazo[1,2-a]pyridin-3-yl)pyridazin-3(2H)-one 194262 2-(2,6-Dichloro-phenyl)-6-[2-(2,3-dichloro-phenyl)-imidazo[1,2-a]pyridin-3-yl]-2H-pyridazin-3-one 194274 3-[5-(Piperazine-1-carbonyl)-1H-indol-2-yl]-1H-quinolin-2-one 194356 N-[4-(2-{4-[3-(5-[1,2,4]Triazol-4-yl-1H-indol-3-yl)-propyl]-piperazin-1-yl}-ethyl)-phenyl]-acetamide 194389 3-(3-{4-[2-(3,4-Difluoro-phenyl)-ethyl]-piperazin-1-yl}-propyl)-5-[1,2,4]triazol-4-yl-1H-indole 194392 3-(3-{4-[2-(3,5-Difluoro-phenyl)-ethyl]-piperazin-1-yl}-propyl)-5-[1,2,4]triazol-4-yl-1H-indole 194393 3-(3-{4-[2-(4-Fluoro-phenyl)-ethyl]-piperazin-1-yl}-propyl)-5-[1,2,4]triazol-4-yl-1H-indole 194524 C-(8-Bromo-6-methoxy-4,5-dihydro-3H-naphtho[1,8-bc]furan-5-yl)-methylamine 194549 3-[5-(4-Methyl-piperazine-1-sulfonyl)-1H-indol-2-yl]-1H-quinolin-2-one 194553 3-[5-(Piperazine-1-sulfonyl)-1H-indol-2-yl]-1H-quinolin-2-one 194554 3-[5-(3-Amino-pyrrolidine-1-sulfonyl)-1H-indol-2-yl]-1H-quinolin-2-one 194559 C-(8-Bromo-6-methoxy-2a,3,4,5-tetrahydro-2H-naphtho[1,8-bc]furan-5-yl)-methylamine 194560 C-(8-Bromo-6-methoxy-2a,3,4,5-tetrahydro-2H-naphtho[1,8-bc]furan-5-yl)-methylamine 194563 2-(2-Oxo-1,2-dihydro-quinolin-3-yl)-1H-indole-5-sulfonic acid pyrrolidin-3-ylamide 194616 6-[4-(2-Morpholin-4-yl-ethoxy)-phenyl]-3-thiophen-3-yl-pyrazolo[1,5-a]pyrimidine 194619 (2S,3S,4R,5R)-3,4-dihydroxy-5-(6-(3-iodobenzylamino)-9H-purin-9-yl)-N-methyltetrahydrofuran-2-carboxamide 194620 3-Amino-4-hydroxy-5-[6-(3-iodo-benzylamino)-purin-9-yl]-tetrahydro-furan-2-carboxylic acid methylamide 194629 2-(2,6-dichlorophenyl)-6-(2-(2,4-difluorophenyl)imidazo[1,2-a]pyridin-3-yl)-4,5-dihydropyridazin-3(2H)-one 194630 6-[2-(2-Chloro-4-fluoro-phenyl)-imidazo[1,2-a]pyridin-3-yl]-2-o-tolyl-4,5-dihydro-2H-pyridazin-3-one 194631 6-[2-(2,3-Dichloro-phenyl)-imidazo[1,2-a]pyridin-3-yl]-2-o-tolyl-2H-pyridazin-3-one 194654 Benzyl-(2-methoxy-ethyl)-{2-[4-(3-thiophen-3-yl-pyrazolo[1,5-a]pyrimidin-6-yl)-phenoxy]-ethyl}-amine 194663 6-[2-(2-Chloro-4-fluoro-phenyl)-imidazo[1,2-a]pyridin-3-yl]-2-o-tolyl-2H-pyridazin-3-one 194731 4-(2-(4-(3-phenylpyrazolo[1,5-a]pyrimidin-6-yl)phenoxy)ethyl)morpholine 194734 6-(2-(2,4-difluorophenyl)imidazo[1,2-a]pyridin-3-yl)-2-o-tolyl-4,5-dihydropyridazin-3(2H)-one 194773 6-[2-(2-Chloro-4-fluoro-phenyl)-imidazo[1,2-a]pyridin-3-yl]-2-(2-chloro-phenyl)-4,5-dihydro-2H-pyridazin-3-one 194775 2-(2,6-Dichloro-phenyl)-6-[2-(2,4-difluoro-phenyl)-imidazo[1,2-a]pyridin-3-yl]-2H-pyridazin-3-one 194776 6-[2-(2,4-Difluoro-phenyl)-imidazo[1,2-a]pyridin-3-yl]-2-o-tolyl-2H-pyridazin-3-one 194788 4-(2-(4-(3-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-6-yl)phenoxy)ethyl)morpholine 194789 4-(3-Phenyl-pyrazolo[1,5-a]pyrimidin-6-yl)-1-(3-piperidin-1-yl-propyl)-1H-pyridin-2-one 194823 6-[2-(2-Chloro-4-fluoro-phenyl)-imidazo[1,2-a]pyridin-3-yl]-2-(2,6-dichloro-phenyl)-2H-pyridazin-3-one 194835 1-[3-(4-Methyl-piperazin-1-yl)-propyl]-4-(3-thiophen-3-yl-pyrazolo[1,5-a]pyrimidin-6-yl)-1H-pyridin-2-one 194868 1-[3-(4-Methyl-piperazin-1-yl)-propyl]-4-(3-phenyl-pyrazolo[1,5-a]pyrimidin-6-yl)-1H-pyridin-2-one 194892 5-nitroindoline-2,3-dione 194925 C-(6-Methoxy-2a,3,4,5-tetrahydro-2H-naphtho[1,8-bc]furan-5-yl)-methylamine 194926 C-(6-Methoxy-2a,3,4,5-tetrahydro-2H-naphtho[1,8-bc]furan-5-yl)-methylamine 194950 C-(6-Methoxy-4,5-dihydro-3H-naphtho[1,8-bc]furan-5-yl)-methylamine 194976 3-Benzimidazol-2-ylhydroquinolin-2-one 194984 6-(1H-Benzoimidazol-2-yl)-benzocyclohepten-7-one 194989 2-(2-Oxo-1,2-dihydro-quinolin-3-yl)-1H-indole-5-carboxylic acid pyrrolidin-3-ylamide 195019 3-[5-(3-Amino-pyrrolidine-1-carbonyl)-1H-indol-2-yl]-1H-quinolin-2-one 195051 5-Chloro-4-[4-(2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-piperazin-1-yl]-2-{7-[4-(2-isopropoxy-phenyl)-piperazin-1-yl]-heptyl}-2H-pyridazin-3-one 195052 5-Chloro-4-[4-(2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-piperazin-1-yl]-2-{7-[4-(2-ethoxy-phenyl)-piperazin-1-yl]-heptyl}-2H-pyridazin-3-one 195134 3-(5-{2-[(2-Methoxy-ethyl)-methyl-amino]-ethoxy}-1H-indol-2-yl)-1H-quinolin-2-one 195166 3-{5-[2-(4-Acetyl-piperazin-1-yl)-ethoxy]-1H-indol-2-yl}-1H-quinolin-2-one 195200 (2S,3S,4R,5R)-3-amino-4-hydroxy-N-methyl-5-(6-(methylamino)-9H-purin-9-yl)-tetrahydrofuran-2-carboxamide 195208 3-Amino-5-{6-[5-chloro-2-(3-methyl-isoxazol-5-ylmethoxy)-benzylamino]-purin-9-yl}-4-hydroxy-tetrahydro-furan-2-carboxylic acid methylamide 195248 6-[3-(2-Morpholin-4-yl-ethoxy)-phenyl]-3-thiophen-3-yl-pyrazolo[1,5-a]pyrimidine 195256 (2S,3S,4R,5R)-3,4-dihydroxy-N-methyl-5-(6-(methylamino)-9H-purin-9-yl)-tetrahydrofuran-2-carboxamide 195284 6-(4-(2-(piperidin-1-yl)ethoxy)phenyl)-3-(thiophen-3-yl)pyrazolo[1,5-a]pyrimidine 195288 5-{6-[5-Chloro-2-(3-methyl-isoxazol-5-ylmethoxy)-benzylamino]-purin-9-yl}-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid methylamide 195317 5-Chloro-4-[4-(2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-piperazin-1-yl]-2-{7-[4-(2-methoxy-phenyl)-piperazin-1-yl]-heptyl}-2H-pyridazin-3-one 195342 4-chloro-5-(4-((2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)piperazin-1-yl)-2-(7-(4-(2-methoxyphenyl)piperazin-1-yl)heptyl)pyridazin-3(2H)-one 195343 5-Chloro-2-{7-[4-(2-ethoxy-phenyl)-piperazin-1-yl]-heptyl}-4-[4-(furan-2-carbonyl)-piperazin-1-yl]-2H-pyridazin-3-one 195355 Dimethyl-{3-[4-(3-thiophen-3-yl-pyrazolo[1,5-a]pyrimidin-6-yl)-phenoxy]-propyl}-amine 195366 6-(4-(2-(piperidin-1-yl)ethoxy)phenyl)-3-(pyridin-3-yl)pyrazolo[1,5-a]pyrimidine 195370 4-chloro-5-(4-((2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)piperazin-1-yl)-2-(7-(4-(2-ethoxyphenyl)piperazin-1-yl)heptyl)pyridazin-3(2H)-one 195653 1-{3-[2-(2-Oxo-1,2-dihydro-quinolin-3-yl)-1H-indol-5-yloxy]-propyl}-piperidine-4-carboxylic acid 195654 3-[5-(4-Methyl-piperazine-1-carbonyl)-1H-indol-2-yl]-1H-quinolin-2-one 195678 3-[5-(2-Piperidin-1-yl-ethoxy)-1H-indol-2-yl]-1H-quinolin-2-one 195779 4-chloro-5-(4-((2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)piperazin-1-yl)-2-(7-(4-(2-isopropoxyphenyl)piperazin-1-yl)heptyl)pyridazin-3(2H)-one 195801 5-Chloro-4-[4-(furan-2-carbonyl)-piperazin-1-yl]-2-{7-[4-(2-methoxy-phenyl)-piperazin-1-yl]-heptyl}-2H-pyridazin-3-one 196009 5-Chloro-4-[4-(furan-2-carbonyl)-piperazin-1-yl]-2-{7-[4-(2-isopropoxy-phenyl)-piperazin-1-yl]-heptyl}-2H-pyridazin-3-one 196215 Zolmitriptan 196625 3-[5-(2-Carbamoyl-2-cyano-vinyl)-2-hydroxy-3-methoxy-benzylsulfanyl]-propionic acid 196634 (10S,13S)-13-Hydroxymethyl-10-isopropyl-9-methyl-3,9,12-triaza-tricyclo[6.6.1.0*4,15*]pentadeca-4,6,8(15)-trien-11-one 196740 Thieno analogue of kenpaullone 196824 4-amino-6-nitro-2-phenyl-[1,2,4]triazolo[4,3-a]quinoxalin-1(2H)-one 196867 Cyclopentyl-{4-[2-(4-fluoro-phenyl)-5-(4-methyl-piperazin-1-yl)-imidazo[4,5-b]pyridin-1-yl]-pyrimidin-2-yl}-amine 196913 4-[1-(2-Cyclopentylamino-pyrimidin-4-yl)-2-(3-trifluoromethyl-phenyl)-5H-imidazol-4-yl]-1-methyl-piperidin-4-ol 196987 (+/-)7-Fluoro-9-(4-methyl-piperazin-1-yl)-9,10-dihydro-4-thia-10a-aza-benzo[f]azulene 197006 2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-ylmethyl]-1,2,3,9-tetrahydro-carbazol-4-one 197227 (+/-)2-[4-(7-Fluoro-9,10-dihydro-4-thia-10a-aza-benzo[f]azulen-9-yl)-piperazin-1-yl]-ethanol 197233 5-(2,2-Dichloro-1-hexyl-cyclopropyl)-2-(6-isopropenyl-3-methyl-cyclohex-2-enyl)-benzene-1,3-diol 197244 4,6-Diamino-2-(4-methoxy-phenyl)-2H-[1,2,4]triazolo[4,3-a]quinoxalin-1-one 197254 5-(1-Hexyl-cyclopropyl)-2-(6-isopropenyl-3-methyl-cyclohex-2-enyl)-benzene-1,3-diol 197311 5-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-1-[4-(4-nitro-phenyl)-piperazin-1-yl]-pentan-1-one 197361 Dmt-Pro-Phe-Phe-NH2 197388 1-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-phenylurea 197398 Tyr-Pro-Phe-Phe-NH2 197427 5-(2-Hexyl-[1,3]dithiolan-2-yl)-2-(6-isopropenyl-3-methyl-cyclohex-2-enyl)-benzene-1,3-diol 197428 (6aR,10aR)-3-(2,2-dibromo-1-hexylcyclopropyl)-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol 197434 4-(3-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)ureido)benzenesulfonic acid 197514 5-[[(4-pyridyl)-amino]carbonyl]amino-8-methyl-2-(2-furyl)-pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine hydrochloride 197583 (+/-)9-(4-Ethyl-piperazin-1-yl)-7-fluoro-9,10-dihydro-4-thia-10a-aza-benzo[f]azulene 197622 1-(2-furan-2-yl-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-pyridin-4-yl-urea 197647 4-[5-(2-Cyclohexylamino-pyridin-4-yl)-4-(4-fluoro-phenyl)-oxazol-2-yl]-piperidin-4-ol 197679 (6aR,10aR)-3-(2,2-dichloro-1-hexylcyclopropyl)-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol 197712 5-(2,2-Dibromo-1-hexyl-cyclopropyl)-2-(6-isopropenyl-3-methyl-cyclohex-2-enyl)-benzene-1,3-diol 197726 Acetic acid 4-(1,4-dioxo-4,5-dihydro-[1,2,4]triazolo[4,3-a]quinoxalin-2-yl)-phenyl ester 197758 2-(4-Hydroxy-phenyl)-2H,5H-[1,2,4]triazolo[4,3-a]quinoxaline-1,4-dione 197766 N-[2-(4-{2-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-acetyl}-piperazin-1-yl)-benzyl]-methanesulfonamide 197771 6-Benzylamino-1-(2,6-dichloro-phenyl)-3,4-dihydro-1H-quinazolin-2-one 197772 2-Chloro-N-[1-(2,6-dichloro-phenyl)-2-oxo-1,2,3,4-tetrahydro-quinazolin-6-yl]-benzenesulfonamide 197805 N-[1-(2,6-Dichloro-phenyl)-2-oxo-1,2,3,4-tetrahydro-quinazolin-6-yl]-benzenesulfonamide 197809 2,5-Dichloro-N-[1-(2,6-dichloro-phenyl)-2-oxo-1,2,3,4-tetrahydro-quinazolin-6-yl]-benzenesulfonamide 197835 2-(4-{2-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-acetyl}-piperazin-1-yl)-benzonitrile 197859 2-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-1-(4-o-tolyl-piperazin-1-yl)-ethanone 197869 2-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-1-[4-(4-nitro-phenyl)-piperazin-1-yl]-ethanone 197889 4-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-1-[4-(4-nitro-phenyl)-piperazin-1-yl]-butan-1-one 197890 2-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-1-[4-(2-nitro-phenyl)-piperazin-1-yl]-ethanone 197904 6-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-1-[4-(4-nitro-phenyl)-piperazin-1-yl]-hexan-1-one 197905 2-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-1-[4-(4-aminomethyl-phenyl)-piperazin-1-yl]-ethanone 198029 1,3-diphenyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 198050 N-[4-(4-{2-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-acetyl}-piperazin-1-yl)-phenyl]-benzamide 198109 C-(4'-aminomethyl-biphenyl-4-yl)-methylamine 198139 (2-Methoxy-benzyl)-[(2S,3R)-2-(3-methoxy-phenyl)-1-aza-bicyclo[2.2.2]oct-3-yl]-amine 198173 N-[4-(4-{2-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-acetyl}-piperazin-1-yl)-benzyl]-methanesulfonamide 198187 1-(2,6-Dichloro-phenyl)-3,4-dihydro-1H-quinazolin-2-one 198188 N-[1-(2,6-Dichloro-phenyl)-2-oxo-1,2,3,4-tetrahydro-quinazolin-6-yl]-benzamide 198203 2-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-1-[4-(2-aminomethyl-phenyl)-piperazin-1-yl]-ethanone 198262 1-Isopropyl-6-methoxy-7-morpholin-4-yl-4-phenyl-1H-quinazolin-2-one 198316 1-(2,6-Dichloro-phenyl)-6-(2,4-difluoro-phenylsulfanyl)-3,4-dihydro-1H-quinazolin-2-one 198317 1-(2,6-Dichloro-phenyl)-6-(2,4-difluoro-phenylamino)-3,4-dihydro-1H-quinazolin-2-one 198383 N*3*-(3-Chloro-phenyl)-N*4*-m-tolyl-1H-pyrazolo[3,4-d]pyrimidine-3,4-diamine 198387 2-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-1-(4-phenyl-piperazin-1-yl)-ethanone 198392 5-Chloro-N-[1-(2,6-dichloro-phenyl)-2-oxo-1,2,3,4-tetrahydro-quinazolin-6-yl]-2-hydroxy-benzenesulfonamide 198449 N-[1-(2,6-Dichloro-phenyl)-2-oxo-1,2,3,4-tetrahydro-quinazolin-6-yl]-4-methyl-benzenesulfonamide 198481 N-[4-(4-{6-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-hexanoyl}-piperazin-1-yl)-phenyl]-methanesulfonamide 198493 3-Chloro-N-[1-(2,6-dichloro-phenyl)-2-oxo-1,2,3,4-tetrahydro-quinazolin-6-yl]-4-fluoro-benzenesulfonamide 198494 2,5-Dichloro-N-[1-(2,6-dichloro-phenyl)-2-oxo-1,2,3,4-tetrahydro-quinazolin-6-yl]-N-methyl-benzenesulfonamide 198513 5-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-1-[4-(4-amino-phenyl)-piperazin-1-yl]-pentan-1-one 198516 N-[4-(4-{2-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-acetyl}-piperazin-1-yl)-phenyl]-methanesulfonamide 198536 6-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-1-[4-(4-amino-phenyl)-piperazin-1-yl]-hexan-1-one 198538 2-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-1-[4-(4-amino-phenyl)-piperazin-1-yl]-ethanone 198542 N-[4-(4-{2-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-acetyl}-piperazin-1-yl)-phenyl]-acetamide 198574 2-(1-Phenyl-4-propylsulfanyl-1H-pyrazolo[3,4-d]pyrimidin-6-ylsulfanyl)-butyramide 198593 (S)-4-(2-(azetidin-2-yl)ethoxy)-7-chloro-2-oxo-N-(pyrimidin-4-yl)-3-(3,4,5-trimethylphenyl)-1,2-dihydroquinoline-6-carboxamide 198595 1-(2,6-difluorobenzyl)-5-((methyl(2-(pyridin-2-yl)ethyl)amino)methyl)-6-(4-nitrophenyl)-3-phenylthieno[2,3-d]pyrimidine-2,4(1H,3H)-dione 198596 1-(2,6-difluorobenzyl)-5-((methyl(phenethyl)amino)methyl)-6-(4-nitrophenyl)-3-phenylthieno[2,3-d]pyrimidine-2,4(1H,3H)-dione 198656 (5-(3-amino-3-methylbut-1-ynyl)-2-methoxyphenyl)(4-(2,4-difluorophenylamino)phenyl)methanone 198864 SID26754853 198917 (2-Chloro-benzyl)-[(2S,3S)-2-(3-chloro-phenyl)-1-aza-bicyclo[2.2.2]oct-3-yl]-amine 198951 [(2S,3S)-2-(3-Chloro-phenyl)-1-aza-bicyclo[2.2.2]oct-3-yl]-(2,4-dimethoxy-benzyl)-amine 199000 1-(2,6-difluorobenzyl)-6-(4-aminophenyl)-5-((benzyl(methyl)amino)methyl)-3-phenylthieno[2,3-d]pyrimidine-2,4(1H,3H)-dione 199033 1-(2,6-difluorobenzyl)-5-((benzyl(methyl)amino)methyl)-6-(4-nitrophenyl)-3-phenylthieno[2,3-d]pyrimidine-2,4(1H,3H)-dione 199282 N-(4-(1-(2,6-difluorobenzyl)-5-((benzyl(methyl)amino)methyl)-2,4-dioxo-3-phenyl-1,2,3,4-tetrahydrothieno[2,3-d]pyrimidin-6-yl)phenyl)acetamide 200569 5-(4-Heptyl-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2,3,6-tetrahydro-pyridine 200827 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-N-methyl-benzamide 200828 5-(2,5-Dihydroxy-benzylamino)-N-hexyl-2-hydroxy-benzamide 200891 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzenesulfonic acid 201063 7-fluoro-4-(4-methylpiperazin-1-yl)pyrrolo[1,2-a]quinoxaline 201073 7-Fluoro-4-piperazin-1-yl-pyrrolo[1,2-a]quinoxaline 201090 1-(3,4,5-Triiodo-benzyl)-1,2,3,4-tetrahydro-isoquinoline-6,7-diol 201124 N-[4-(6,7-Dihydroxy-1,2,3,4-tetrahydro-isoquinolin-1-ylmethyl)-2-iodo-phenyl]-acetamide 201125 1-(4-Amino-3,5-diiodo-benzyl)-1,2,3,4-tetrahydro-isoquinoline-6,7-diol 201221 (6aR,9R)-4,7-Dimethyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid (1-ethyl-propyl)-amide 201356 Tributyl-(4-{[2-(4-phenyl-butyryl)-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl]-amino}-benzyl)-phosphonium chloride 201411 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-N-tetradecyl-benzamide 201412 2-[(4-Hydroxy-3-nitro-phenylamino)-methyl]-benzene-1,4-diol 201413 2-[(4-Hydroxy-phenylamino)-methyl]-benzene-1,4-diol 201428 2-Amino-4-(4-hydroxy-phenyl)-6-(1H-imidazol-2-ylmethylsulfanyl)-pyridine-3,5-dicarbonitrile 201458 2-Amino-6-(1H-imidazol-2-ylmethylsulfanyl)-4-(3-methoxy-phenyl)-pyridine-3,5-dicarbonitrile 201553 9-Fluoro-4-piperazin-1-yl-pyrrolo[1,2-a]quinoxaline 201586 [4-(5-Butyl-3H-[1,2,4]triazolo[5,1-i]purin-8-yl)-phenyl]-dimethyl-amine 201592 5-Butyl-8-(4-ethoxy-phenyl)-3H-[1,2,4]triazolo[5,1-i]purine 201593 5-Butyl-8-(4-methoxy-phenyl)-3H-[1,2,4]triazolo[5,1-i]purine 201618 5-Butyl-8-(4-propoxy-phenyl)-3H-[1,2,4]triazolo[5,1-i]purine 201619 2-((1H-imidazol-2-yl)methylthio)-6-amino-4-(4-methoxyphenyl)pyridine-3,5-dicarbonitrile 201620 2-Amino-4-(3-hydroxy-phenyl)-6-(1H-imidazol-2-ylmethylsulfanyl)-pyridine-3,5-dicarbonitrile 201784 N-[4-(6,7-Dihydroxy-1,2,3,4-tetrahydro-isoquinolin-1-ylmethyl)-2-iodo-phenyl]-benzamide 201785 1-(3,5-Bis-trifluoromethyl-benzyl)-1,2,3,4-tetrahydro-isoquinoline-6,7-diol 201787 5-Butyl-8-phenyl-3H-[1,2,4]triazolo[5,1-i]purine 201803 1-(4-Amino-3-iodo-benzyl)-1,2,3,4-tetrahydro-isoquinoline-6,7-diol 201804 N-[4-(6,7-Dihydroxy-1,2,3,4-tetrahydro-isoquinolin-1-ylmethyl)-2,6-diiodo-phenyl]-acetamide 201826 5-Butyl-8-(4-trifluoromethyl-phenyl)-3H-[1,2,4]triazolo[5,1-i]purine 201833 5-(2-amino-4-oxo-1H-imidazol-5(4H)-ylidene)-2,3,4,5-tetrahydroazepino[3,4-b]indol-1(10H)-one 201921 (4-{[2-(2-tert-Butoxycarbonylamino-4-phenyl-butyryl)-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl]-amino}-benzyl)-tributyl-phosphonium chloride 201978 2-(2,4-Dichloro-phenoxymethyl)-1-methyl-3-piperidin-1-ylmethyl-1H-indole 201979 2-[1,4']Bipiperidinyl-1'-yl-1-[2-(4-chloro-phenoxymethyl)-1-(2-piperidin-4-yl-ethyl)-1H-indol-3-yl]-ethanone 202012 1'-[2-(4-Chloro-phenoxymethyl)-1-methyl-1H-indol-3-ylmethyl]-[1,4']bipiperidinyl 202024 2-((1H-imidazol-2-yl)methylthio)-6-amino-4-phenylpyridine-3,5-dicarbonitrile 202033 2-[1,4']Bipiperidinyl-1'-yl-1-[2-(4-chloro-phenoxymethyl)-1-methyl-1H-indol-3-yl]-ethanone 202034 1'-{2-[2-(4-Chloro-phenoxymethyl)-1-methyl-1H-indol-3-yl]-ethyl}-[1,4']bipiperidinyl 202134 N-(1-Benzyl-piperidin-4-yl)-2,3-dimethoxy-benzamide 202163 Ac-c[Cys-Glu-His-D-Nal(2')-Arg-Trp-Cys]-Pro-Pro-Lys-Asp-NH2 202165 Ac-c[Cys-Glu-His-D-(2')Nal-Arg-Trp-Gly-Cys]-Pro-Pro-Lys-Asp-NH2 202302 1-(4-Hydroxy-3,5-diiodo-benzyl)-1,2,3,4-tetrahydro-isoquinoline-6,7-diol 202347 1-(3,5-Diiodo-benzyl)-1,2,3,4-tetrahydro-isoquinoline-6,7-diol 202353 5-Chloro-1-ethyl-8-methyl-6,7,8,9-tetrahydro-2-thia-8-aza-benzo[cd]azulene 202354 1-Bromo-5-chloro-8-methyl-6,7,8,9-tetrahydro-2-oxa-8-aza-benzo[cd]azulene 202416 Ac-c[Cys-Glu-Pro-D-Phe-Arg-Trp-Cys]-Pro-Pro-Lys-Asp-NH2 202539 2-(4-Chloro-phenoxymethyl)-1-methyl-3-(2-piperidin-1-yl-ethyl)-1H-indole 202584 1-[1,4']Bipiperidinyl-1'-yl-2-[2-(4-chloro-phenoxymethyl)-1-methyl-1H-indol-3-yl]-ethane-1,2-dione 202609 (9-Benzyl-3,9-diaza-bicyclo[3.3.1]non-3-yl)-(5-bromo-2,3-dimethoxy-phenyl)-methanone 202612 4-Amino-N-(9-benzyl-9-aza-bicyclo[3.3.1]non-3-yl)-5-chloro-2-methoxy-benzamide 202694 SID11111780 202735 (R)-2-(2,2-diphenylacetamido)-5-guanidino-N-(4-hydroxybenzyl)pentanamide 202768 1'-[2-(4-Chloro-phenoxymethyl)-1-(2-piperidin-1-yl-ethyl)-1H-indol-3-ylmethyl]-[1,4']bipiperidinyl 202888 [4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-2,6-dipropyl-phenoxy]-p-tolyl-acetic acid 202913 Ac-c[Cys-Glu-His-D-Nal(2')-Arg-Trp-D-Cys]-Pro-Pro-Lys-Asp-NH2 202936 [4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-2,6-dipropyl-phenoxy]-(3-phenoxy-phenyl)-acetic acid 202995 Ac-c[Cys-Glu-Pro-D-Nal(2')-Arg-Trp-Cys]-Pro-Pro-Lys-Asp-NH2 203027 Ac-c[Pen-Glu-His-D-Phe-Arg-Trp-Cys]-Pro-Pro-Lys-Asp-NH2 203045 N-[1-(4-Fluoro-benzyl)-piperidin-4-yl]-2,3-dimethoxy-benzamide 203046 5-Bromo-N-[1-(4-fluoro-benzyl)-piperidin-4-yl]-2,3-dimethoxy-benzamide 203072 4-Amino-5-chloro-N-[1-(4-fluoro-benzyl)-piperidin-4-yl]-2-methoxy-benzamide 203127 2-[1,4']Bipiperidinyl-1'-yl-1-[2-(4-chloro-phenoxymethyl)-1-((R)-3-piperidin-3-yl-propyl)-1H-indol-3-yl]-ethanone 203192 [4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-2,6-dipropyl-phenoxy]-m-tolyl-acetic acid 203199 Biphenyl-3-yl-[4-(2-ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-2,6-dipropyl-phenoxy]-acetic acid 203223 [4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-2,6-dipropyl-phenoxy]-o-tolyl-acetic acid 203225 (2-Chloro-phenyl)-[4-(2-ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-2,6-dipropyl-phenoxy]-acetic acid 203347 [4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-2,6-dipropyl-phenoxy]-(4-ethyl-phenyl)-acetic acid 203494 [4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-2,6-dipropyl-phenoxy]-(4-phenoxy-phenyl)-acetic acid 203620 (3-Chloro-phenyl)-[4-(2-ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-2,6-dipropyl-phenoxy]-acetic acid 203621 (4-Chloro-phenyl)-[4-(2-ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-2,6-dipropyl-phenoxy]-acetic acid 203650 [4-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-2,6-dipropyl-phenoxy]-phenyl-acetic acid 204030 H-Tyr-D-Ala-(R or S)CalphaMPhe-Asp-Val-Val-Gly-NH2 204237 5-Butyl-2-phenyl-[1,2,4]triazolo[1,5-c]quinazoline 204317 N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[2-{5-[2-carboxyamino-3-(4-sulfo-phenyl)-propionylamino]-pentanoylamino}-3-(1H-indol-3-yl)-propionylamino]-4-methylsulfanyl-butyrylamino}-succinamic acid 204318 N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[2-{2-[2-carboxyamino-3-(4-sulfo-phenyl)-propionylamino]-acetylamino}-3-(1H-indol-3-yl)-propionylamino]-4-methylsulfanyl-butyrylamino}-succinamic acid 204342 3-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-1,2,3,4-tetrahydro-naphthalene-2-carbonyl)-amino]-N-{1-[1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-succinamic acid 204357 N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[2-{3-[2-carboxyamino-3-(4-sulfo-phenyl)-propionylamino]-benzoylamino}-3-(1H-indol-3-yl)-propionylamino]-4-methylsulfanyl-butyrylamino}-succinamic acid 204358 N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[2-{4-[2-carboxyamino-3-(4-sulfo-phenyl)-propionylamino]-butyrylamino}-3-(1H-indol-3-yl)-propionylamino]-4-methylsulfanyl-butyrylamino}-succinamic acid 204406 3-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-indane-2-carbonyl)-amino]-N-{1-[1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-succinamic acid 204407 3-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionyl}-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl)-amino]-N-{1-[1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-succinamic acid 204687 5-Butyl-2-phenyl-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine 204689 5-Butyl-2-(4-methoxy-phenyl)-[1,2,4]triazolo[1,5-c]quinazoline 204691 N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[2-(2-{2-[2-carboxyamino-3-(4-sulfo-phenyl)-propionylamino]-4-methylsulfanyl-butyrylamino}-acetylamino)-3-(1H-indol-3-yl)-propionylamino]-4-methylsulfanyl-butyrylamino}-succinamic acid 204692 N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[2-{6-[2-carboxyamino-3-(4-sulfo-phenyl)-propionylamino]-hexanoylamino}-3-(1H-indol-3-yl)-propionylamino]-4-methylsulfanyl-butyrylamino}-succinamic acid 204807 5-Butyl-2-(4-trifluoromethyl-phenyl)-[1,2,4]triazolo[1,5-c]quinazoline 204860 N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[2-{3-[2-carboxyamino-3-(4-sulfo-phenyl)-propionylamino]-propionylamino}-3-(1H-indol-3-yl)-propionylamino]-4-methylsulfanyl-butyrylamino}-succinamic acid 204881 5-Butyl-2-(4-methoxy-phenyl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine 204890 N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[2-{4-[2-carboxyamino-3-(4-sulfo-phenyl)-propionylamino]-benzoylamino}-3-(1H-indol-3-yl)-propionylamino]-4-methylsulfanyl-butyrylamino}-succinamic acid 205019 N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[2-{3-[2-carboxyamino-3-(4-sulfo-phenyl)-propionylamino]-2-methyl-benzoylamino}-3-(1H-indol-3-yl)-propionylamino]-4-methylsulfanyl-butyrylamino}-succinamic acid 205020 N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[2-{5-[2-carboxyamino-3-(4-sulfo-phenyl)-propionylamino]-2-methyl-benzoylamino}-3-(1H-indol-3-yl)-propionylamino]-4-methylsulfanyl-butyrylamino}-succinamic acid 205023 5-Butyl-2-(4-trifluoromethyl-phenyl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine 205066 N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[2-(2-{2-[2-carboxyamino-3-(4-sulfo-phenyl)-propionylamino]-cyclopentyl}-acetylamino)-3-(1H-indol-3-yl)-propionylamino]-4-methylsulfanyl-butyrylamino}-succinamic acid 205165 N-(4-isopropoxyphenyl)-4-(6-methoxy-7-(3-(piperidin-1-yl)propoxy)quinazolin-4-yl)piperazine-1-carboxamide 205249 Cyclopropanecarboxylic acid [3-(2-ethyl-benzooxazol-7-yl)-propyl]-amide 205250 N-[3-(2-Ethyl-benzooxazol-7-yl)-propyl]-isobutyramide 205268 (R)-N-((R)-1-(4-((1H-1,2,4-triazol-1-yl)methyl)-4-cyclohexylpiperidin-1-yl)-3-(4-chlorophenyl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 205295 N-[3-(2-Phenyl-benzooxazol-7-yl)-propyl]-acetamide 205365 4-[6-Methoxy-7-(3-morpholin-4-yl-propoxy)-quinazolin-4-yl]-piperazine-1-carboxylic acid (4-isopropoxy-phenyl)-amide 205386 (R)-3-[((2S,5S,11bR)-2-Benzyloxycarbonylamino-3-oxo-2,3,5,6,11,11b-hexahydro-1H-indolizino[8,7-b]indole-5-carbonyl)-amino]-4-phenyl-butyric acid 205387 (S)-3-[((2S,5S,11bR)-2-Benzyloxycarbonylamino-3-oxo-2,3,5,6,11,11b-hexahydro-1H-indolizino[8,7-b]indole-5-carbonyl)-amino]-4-phenyl-butyric acid 205417 (R)-N-((R)-1-(4-(2-((1H-1,2,4-triazol-1-yl)methyl)phenyl)piperazin-1-yl)-3-(4-chlorophenyl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 205427 4-[6-Methoxy-7-(2-piperidin-1-yl-ethoxy)-quinazolin-4-yl]-piperazine-1-carboxylic acid (4-isopropoxy-phenyl)-amide 205545 Cyclopropanecarboxylic acid {3-[2-(4-phenyl-butyl)-benzooxazol-7-yl]-propyl}-amide 205563 N-(3-Benzooxazol-7-yl-propyl)-butyramide 205575 N-[3-(2-Methyl-benzooxazol-7-yl)-propyl]-propionamide 205578 N-{3-[2-(4-Phenyl-butyl)-benzooxazol-7-yl]-propyl}-isobutyramide 205621 N-[3-(2-Methyl-benzooxazol-7-yl)-propyl]-isobutyramide 205629 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {1-(4-chloro-benzyl)-2-[4-(2-methanesulfonylamino-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-amide 205630 N-{3-[2-(4-Phenyl-butyl)-benzooxazol-7-yl]-propyl}-butyramide 205667 N-{3-[2-(4-Phenyl-butyl)-benzooxazol-7-yl]-propyl}-propionamide 205668 N-{3-[2-(4-Phenyl-butyl)-benzooxazol-7-yl]-propyl}-acetamide 205681 N-[3-(2-Ethyl-benzooxazol-7-yl)-propyl]-butyramide 205682 N-[3-(2-Ethyl-benzooxazol-7-yl)-propyl]-propionamide 205749 N-[3-(2-Propyl-benzooxazol-7-yl)-propyl]-acetamide 205750 1-Ethyl-3-[3-(2-ethyl-benzooxazol-7-yl)-propyl]-urea 205952 N-[3-(2-Ethyl-benzooxazol-7-yl)-propyl]-acetamide 205962 3-[3-(3-Acetyl-phenyl)-ureido]-2-[4-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-N-methyl-benzamide 206003 1-Ethyl-3-[3-(2-methyl-benzooxazol-7-yl)-propyl]-urea 206031 1-Ethyl-3-[3-(2-isopropyl-benzooxazol-7-yl)-propyl]-urea 206032 Cyclopropanecarboxylic acid [3-(2-isopropyl-benzooxazol-7-yl)-propyl]-amide 206033 N-[3-(2-Isopropyl-benzooxazol-7-yl)-propyl]-isobutyramide 206042 Cyclopropanecarboxylic acid [3-(2-methyl-benzooxazol-7-yl)-propyl]-amide 206062 N-[3-(2-Phenyl-benzooxazol-7-yl)-propyl]-isobutyramide 206063 N-[3-(2-Phenyl-benzooxazol-7-yl)-propyl]-butyramide 206064 N-[3-(2-Phenyl-benzooxazol-7-yl)-propyl]-propionamide 206094 1-Ethyl-3-[3-(2-phenyl-benzooxazol-7-yl)-propyl]-urea 206118 Cyclopropanecarboxylic acid [3-(2-phenyl-benzooxazol-7-yl)-propyl]-amide 206178 1-Ethyl-3-[3-(2-propyl-benzooxazol-7-yl)-propyl]-urea 206214 N-[3-(2-Isopropyl-benzooxazol-7-yl)-propyl]-butyramide 206215 N-[3-(2-Isopropyl-benzooxazol-7-yl)-propyl]-propionamide 206216 N-[3-(2-Isopropyl-benzooxazol-7-yl)-propyl]-acetamide 206263 Cyclopropanecarboxylic acid [3-(2-propyl-benzooxazol-7-yl)-propyl]-amide 206264 N-[3-(2-Propyl-benzooxazol-7-yl)-propyl]-isobutyramide 206266 4-[6-Methoxy-7-(2-methoxy-ethoxy)-quinazolin-4-yl]-piperazine-1-carboxylic acid (4-isopropoxy-phenyl)-amide 206308 N-[3-(2-Propyl-benzooxazol-7-yl)-propyl]-butyramide 206310 N-[3-(2-Propyl-benzooxazol-7-yl)-propyl]-propionamide 206317 N-[3-(2-Methyl-benzooxazol-7-yl)-propyl]-butyramide 206319 N-[3-(2-Methyl-benzooxazol-7-yl)-propyl]-acetamide 206320 N-(3-Benzooxazol-7-yl-propyl)-acetamide 206357 N-(3-Benzooxazol-7-yl-propyl)-propionamide 206454 N-(4-(4-(2,4-dichlorophenyl)piperazin-1-yl)butyl)-1H-indole-2-carboxamide 206489 Benzofuran-2-carboxylic acid {4-[4-(2,4-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide 206491 Isoquinoline-3-carboxylic acid {4-[4-(2,4-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide 206670 1-{4-[2-(1H-Imidazol-4-yl)-ethoxy]-phenyl}-ethanone 206696 1-(3-Acetyl-phenyl)-3-{2-[4-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-phenyl}-urea 206713 N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)benzofuran-2-carboxamide 206790 (E)-3-{2-[(E)-3-(2-Benzyloxy-3-methyl-phenyl)-allyl]-phenyl}-acrylic acid 206928 4-[3-(3-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyl}-ureido)-phenyl]-2,6-dimethyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid dimethyl ester 207045 6H,14H-naphthyl[3,4-a]pyrrolo[3,4-c]carbazole-5,7(5H,7H)-dione 207094 Isoquinoline-3-carboxylic acid {4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-amide 207150 N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-1H-indole-2-carboxamide 207151 5-chloro-N-(4-(4-(2,4-dichlorophenyl)piperazin-1-yl)butyl)-1H-indole-2-carboxamide 207252 3-thia-13,23-diazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,22}]tricosa-1,4(9),5,7,10,15,17(22),18,20-nonaene-12,14-dione 207303 2-{4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-butyl}-3,4-dihydro-2H-pyrazino[1,2-a]indol-1-one 207564 H-Tyr-D-Ala-Gly-Phe-D-Leu 207679 Tyr-D-Ser-Gly-Phe-Leu-Thr 207787 (E)-3-[6-(2,6-Dichloro-phenylsulfanylmethyl)-3-(4-fluoro-benzyloxy)-pyridin-2-yl]-acrylic acid 207790 (E)-3-{6-(2,6-Dichloro-phenylsulfanylmethyl)-3-[2-(4-fluoro-phenyl)-ethoxy]-pyridin-2-yl}-acrylic acid 207793 (E)-3-{3-[4-(4-Methoxy-phenyl)-butoxy]-6-phenylsulfanylmethyl-pyridin-2-yl}-acrylic acid 207807 [2-(6-Fluoro-chroman-8-yloxy)-ethyl]-[3-(5-fluoro-1H-indol-3-yl)-propyl]-amine 207817 (E)-3-{6-(2,6-Dichloro-phenylsulfanylmethyl)-3-[4-(4-methoxy-phenyl)-butoxy]-pyridin-2-yl}-acrylic acid 208083 (E)-3-[6-(2,6-Dichloro-phenylsulfanylmethyl)-3-(3-phenyl-propoxy)-pyridin-2-yl]-acrylic acid 208084 (E)-3-{6-(2,6-Dichloro-phenylsulfanylmethyl)-3-[2-(4-methoxy-phenyl)-ethoxy]-pyridin-2-yl}-acrylic acid 208085 (E)-3-[3-[2-(4-Chloro-phenyl)-ethoxy]-6-(2,6-dichloro-phenylsulfanylmethyl)-pyridin-2-yl]-acrylic acid 208205 (R)-5-Methylamino-5,6-dihydro-1H,4H-imidazo[4,5,1-ij]quinolin-2-one 208341 3-[2-Butyl-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-2-(5-methoxy-thiophen-2-ylmethyl)-acrylic acid 208398 2-(4-Amino-benzyl)-3-[2-butyl-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-acrylic acid 208399 3-[2-Butyl-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-2-(3,4-dichloro-benzyl)-acrylic acid 208420 3-[2-Butyl-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-2-(phenyl-thiophen-2-yl-methyl)-acrylic acid 208422 3-[2-Butyl-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-2-(4-methoxy-thiophen-2-ylmethyl)-acrylic acid 208462 3-[2-Butyl-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-2-(5-methyl-thiophen-2-ylmethyl)-acrylic acid 208489 3-[2-Butyl-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-2-thiophen-3-ylmethyl-acrylic acid 208490 3-[2-Butyl-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-2-(4-nitro-benzyl)-acrylic acid 208491 3-[2-Butyl-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-2-(2-methyl-benzyl)-acrylic acid 208506 (6,7-Diethoxy-quinazolin-4-yl)-(3-furan-2-yl-phenyl)-amine 208519 3-[2-Butyl-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-2-(3-methyl-thiophen-2-ylmethyl)-acrylic acid 208623 (6,7-Diethoxy-quinazolin-4-yl)-[3-(2-methyl-thiazol-4-yl)-phenyl]-amine 208652 (6,7-Diethoxy-quinazolin-4-yl)-(3-pyrimidin-5-yl-phenyl)-amine 208654 (6,7-Diethoxy-quinazolin-4-yl)-[3-(1H-[1,2,4]triazol-3-yl)-phenyl]-amine 208922 (6,7-Diethoxy-quinazolin-4-yl)-[3-(1H-pyrazol-3-yl)-phenyl]-amine 208937 (6,7-Diethoxy-quinazolin-4-yl)-(3-oxazol-4-yl-phenyl)-amine 208967 (6,7-Diethoxy-quinazolin-4-yl)-(3-thiazol-5-yl-phenyl)-amine 209019 (6,7-Diethoxy-2-ethyl-quinazolin-4-yl)-[3-(2-methyl-thiazol-4-yl)-phenyl]-amine 209053 (6,7-Diethoxy-2-methyl-quinazolin-4-yl)-[3-(2-methyl-thiazol-4-yl)-phenyl]-amine 209068 (6,7-Diethoxy-quinazolin-4-yl)-(3-thiazol-2-yl-phenyl)-amine 209072 [3-(2-Amino-thiazol-4-yl)-phenyl]-(6,7-diethoxy-quinazolin-4-yl)-amine 209129 4-(2-{3-[1-(4-Methoxy-phenyl)-meth-(E)-ylidene]-3H-inden-1-yl}-ethyl)-morpholine 209132 (6,7-Diethoxy-quinazolin-4-yl)-(3-thiazol-4-yl-phenyl)-amine 209314 11-(4-methyl-piperazin-1-yl)-dibenzo[b,f][1,4]oxazepine 209351 3-(2,6-dichlorobenzylidene)indolin-2-one 209411 4-[4-(4-Chloro-3-trifluoromethyl-phenyl)-4-hydroxy-piperidin-1-yl]-N,N-dimethyl-2,2-diphenyl-butyramide 209434 5-Bromo-3-[2-(4-fluoro-phenyl)-2-oxo-ethylidene]-1,3-dihydro-indol-2-one 209436 5-Bromo-3-(2-oxo-2-p-tolyl-ethylidene)-1,3-dihydro-indol-2-one 209453 4-(3'-hydroxyphenyl)amino-6,7-dimethoxyquinazoline 209532 3-(2-Oxo-2-phenyl-ethylidene)-1,3-dihydro-indol-2-one 209533 ethyl 2-cyano-2-(2-oxoindolin-3-ylidene)acetate 209535 2-Cyano-2-(2-oxo-1,2-dihydro-indol-3-ylidene)-acetamide 209616 6-(4-methyl-piperazin-1-yl)-11H-dibenzo[b,e]azepine 209771 5-[1-(4-Hydroxy-benzyl)-4-(4-methoxy-benzyl)-1H-imidazol-2-ylamino]-3-methyl-imidazole-2,4-dione 209772 5-[1,4-Bis-(4-methoxy-benzyl)-1H-imidazol-2-ylamino]-3-methyl-imidazole-2,4-dione 209773 4-(5-(4-hydroxybenzyl)-4-(4-methoxybenzyl)-1-methyl-1H-imidazol-2-ylamino)-1-methyl-1H-imidazole-2,5-dione 209935 5-methoxy-3-(4-oxo-2-thioxothiazolidin-5-ylidene)indolin-2-one 209967 3-(4-(trifluoromethyl)benzylidene)indolin-2-one 209968 SID26752252 210259 (cyclo-[L-propyl-D-phenylalanyl-L-isoleucyl-D-dehydropiperazyl-L-dehydropiperazyl-D(N-methyl)phenylalanyl])(L-365,209) 210290 3-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-2,2-dimethyl-oxazolidine-4-carboxylic acid [1-benzyl-2-(2-carbamoyl-pyrrolidin-1-yl)-2-oxo-ethyl]-amide 210314 16,24-dibenzyl-25-methyl-13-[1-methyl-(1S)-propyl]-(6aR,13S,16R,18aS,24R,26aS)-perhydrodipyrido[1,2-a:1,2-d]pyrrolo[1,2-j][1,4,7,10,13,16]hexaazacyclooctadecine-6,12,15,18,23,26-hexaone 210441 3-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-2,2-dimethyl-oxazolidine-4-carboxylic acid [1-(1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-ethyl]-amide 210442 3-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-oxazolidine-4-carboxylic acid [1-(1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-ethyl]-amide 210466 16-benzyl-24,25-dimethyl-13-[1-methyl-(1S)-propyl]-(6aR,13S,16R,18aS,24S,26aS)-perhydrodipyrido[1,2-a:1,2-d]pyrrolo[1,2-j][1,4,7,10,13,16]hexaazacyclooctadecine-6,12,15,18,23,26-hexaone 210471 N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-2-oxo-2H-1-benzopyran-3-carboxamide 210474 3-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-thiazolidine-4-carboxylic acid [1-(1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-ethyl]-amide 210484 3-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-oxazolidine-4-carboxylic acid [1-benzyl-2-(2-carbamoyl-pyrrolidin-1-yl)-2-oxo-ethyl]-amide 210490 SID26749048 210528 3-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-thiazolidine-4-carboxylic acid [1-benzyl-2-(2-carbamoyl-pyrrolidin-1-yl)-2-oxo-ethyl]-amide 210529 3-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-2,2-dimethyl-thiazolidine-4-carboxylic acid [1-benzyl-2-(2-carbamoyl-pyrrolidin-1-yl)-2-oxo-ethyl]-amide 210553 (R)-4-(4-Chloro-phenyl)-1-[4-(4-fluoro-phenyl)-4-hydroxy-butyl]-piperidin-4-ol 210555 (S)-4-(4-Chloro-phenyl)-1-[4-(4-fluoro-phenyl)-4-hydroxy-butyl]-piperidin-4-ol 210573 (S)1-(4-Fluoro-phenyl)-4-[4-(5-fluoro-pyrimidin-2-yl)-piperazin-1-yl]-butan-1-ol 210612 (S)-1-(4-Fluoro-phenyl)-4-(4-pyridin-2-yl-piperazin-1-yl)-butan-1-ol 210689 N7-(3-(1H-imidazol-1-yl)propyl)-N4-(3-bromophenyl)pyrido[4,3-d]pyrimidine-4,7-diamine 210710 (R)-1-(4-Fluoro-phenyl)-4-(4-pyridin-2-yl-piperazin-1-yl)-butan-1-ol 210896 N4-(3-bromophenyl)-N7-(3-morpholinopropyl)pyrido[4,3-d]pyrimidine-4,7-diamine 210898 N4-(3-bromophenyl)-N7-(2-morpholinoethyl)pyrido[4,3-d]pyrimidine-4,7-diamine 210903 N7-(2-(1H-imidazol-4-yl)ethyl)-N4-m-tolylpyrido[4,3-d]pyrimidine-4,7-diamine 211077 N7-(3-(1H-imidazol-1-yl)propyl)-N4-m-tolylpyrido[4,3-d]pyrimidine-4,7-diamine 211113 3-(4-(3-bromophenylamino)pyrido[4,3-d]pyrimidin-7-ylamino)propanoic acid 211290 3-(4-(3-bromophenylamino)pyrido[4,3-d]pyrimidin-7-ylamino)propane-1,2-diol 211337 N7-(2-(1H-imidazol-4-yl)ethyl)-N4-(3-bromophenyl)pyrido[4,3-d]pyrimidine-4,7-diamine 211437 3-(3-Piperidin-1-yl-bicyclo[2.2.2]oct-5-en-2-yl)-1H-indole 211438 3-(3-Pyrrolidin-1-yl-bicyclo[2.2.2]oct-5-en-2-yl)-1H-indole 211593 (S)-1-((2S,4R)-4-(5-fluorobenzo[b]thiophen-2-yl)-2-methylpiperidin-1-yl)-3-(2-methyl-1H-indol-4-yloxy)propan-2-ol 211633 4-(2-Amino-1-hydroxy-ethyl)-3,6-difluoro-benzene-1,2-diol (2,5-DiFNE) 211646 3,6-Difluoro-4-(1-hydroxy-2-methylamino-ethyl)-benzene-1,2-diol (2,5-DiFEPI) 211664 2,4-Difluoro-3-(1-hydroxy-2-methylamino-ethyl)-phenol (2,6-DiFPE) 211666 5-(2-Amino-1-hydroxy-ethyl)-3-fluoro-benzene-1,2-diol (5-FNE) 211728 5-(3-Phenyl-propyl)-1H-pyrazole-3-carboxylic acid 211729 5-Phenethyl-1H-pyrazole-3-carboxylic acid 211737 (S)-1-((2S,4R)-4-(benzo[b]thiophen-2-yl)-2-methylpiperidin-1-yl)-3-(2-methyl-1H-indol-4-yloxy)propan-2-ol 211837 (2R,4R)-1-[(R)-2-(2-Aza-tricyclo[3.3.1.1*3,7*]dec-2-yloxycarbonylamino)-3-(1H-indol-3-yl)-2-methyl-propionyl]-4-(2,4-difluoro-phenoxy)-pyrrolidine-2-carboxylic acid 211838 (2R,4R)-1-[(R)-2-(2-Aza-tricyclo[3.3.1.1*3,7*]dec-2-yloxycarbonylamino)-3-(1H-indol-3-yl)-2-methyl-propionyl]-4-(2,4-dichloro-phenoxy)-pyrrolidine-2-carboxylic acid 211839 (2R,4R)-1-[(R)-2-(2-Aza-tricyclo[3.3.1.1*3,7*]dec-2-yloxycarbonylamino)-3-(1H-indol-3-yl)-2-methyl-propionyl]-4-(4-nitro-phenoxy)-pyrrolidine-2-carboxylic acid 211853 (2R,4R)-1-[(R)-2-(2-Aza-tricyclo[3.3.1.1*3,7*]dec-2-yloxycarbonylamino)-3-(1H-indol-3-yl)-2-methyl-propionyl]-4-(4-iodo-phenoxy)-pyrrolidine-2-carboxylic acid 211854 (2R,4R)-1-[(R)-2-(2-Aza-tricyclo[3.3.1.1*3,7*]dec-2-yloxycarbonylamino)-3-(1H-indol-3-yl)-2-methyl-propionyl]-4-(4-fluoro-phenoxy)-pyrrolidine-2-carboxylic acid 211886 5-(1H-Indol-3-yl)-6-pyrrolidin-1-yl-bicyclo[2.2.2]octan-2-one 211892 (R)-1-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1H-indol-3-yl)-2-methyl-propionyl]-4-(4-chloro-phenyl)-pyrrolidine-2-carboxylic acid 211895 (S)-1-((2S,4R)-4-(4-methoxybenzo[b]thiophen-2-yl)-2-methylpiperidin-1-yl)-3-(2-methyl-1H-indol-4-yloxy)propan-2-ol 211908 5-(4-Methoxy-benzyl)-1H-pyrazole-3-carboxylic acid 211909 5-(4-Methyl-benzyl)-1H-pyrazole-3-carboxylic acid 211937 5-(1H-Indol-3-yl)-6-piperidin-1-yl-bicyclo[2.2.2]octan-2-one 211987 5-(4-Chloro-benzyl)-1H-pyrazole-3-carboxylic acid 212032 (2R,4R)-1-[(R)-2-(2-Aza-tricyclo[3.3.1.1*3,7*]dec-2-yloxycarbonylamino)-3-(1H-indol-3-yl)-2-methyl-propionyl]-4-(4-chloro-phenoxy)-pyrrolidine-2-carboxylic acid 212073 5-Phenyl-6-piperidin-1-yl-bicyclo[2.2.2]octan-2-one 212201 FGGFTGARKSARK 212202 FGGFTGARKSARK 212203 FGGFTGARKSARK 212342 (5-fluoro-1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone 212343 (5-chloro-1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone 212352 4-(3-(piperidin-1-yl)propoxy)benzonitrile 212357 {23-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-benzyl-14-carbamoyl-8,11-diisopropyl-3,6,9,12,17,24-hexaoxo-1,4,7,10,13,18hexaaza-cyclotetracos-5-yl}-acetic acid 212377 (5,7-difluoro-1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone 212378 2'-Methyl-4'-(5-methyl-4,5-dihydro-[1,2,4]oxadiazol-3-yl)-biphenyl-4-carboxylic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide 212398 5-(3-Chloro-phenyl)-1H-pyrazole-3-carboxylic acid 212423 (1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone 212434 SID26513823 212435 SID26513923 212437 2,4,5,6-tetrahydrocyclopenta[c]pyrazole-3-carboxylate 212452 1-(7-Methoxy-naphthalen-2-yl)-piperazine 212463 (1H-indol-2-yl)(piperazin-1-yl)methanone 212531 1-(4-(3-(piperidin-1-yl)propoxy)benzyl)piperidine 212563 5-Undecyl-1H-pyrazole-3-carboxylic acid 212564 4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid 212565 1H-pyrazole-3-carboxylic acid 212570 FGGFTGARKSARK 212595 FGGFTGARKSARK 212596 FGGFTGARKSARK 212625 15-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-3-phenyl-propionylamino)-2,5-diisopropyl-3,6,13,16-tetraoxo-1,4,7,12tetraaza-cyclohexadecane-8-carboxylic acid amide 212626 14-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-benzyl-3,8,15-trioxo-1,4,9triaza-cyclopentadecane-5-carboxylic acid {1-[1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-amide 212649 3-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-3-phenyl-propionylamino)-N-{1-[1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-succinamic acid 212650 3-[2-({2-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl}-amino)-3-phenyl-propionylamino]-N-{1-[1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-succinamic acid 212656 17-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-acetylamino}-3-phenyl-propionylamino)-2,5-diisopropyl-3,6,14,18-tetraoxo-1,4,7,13tetraaza-cyclooctadecane-8-carboxylic acid amide 212657 3-(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-hexanoylamino}-3-phenyl-propionylamino)-3-(3H-imidazol-4-yl)-propionylamino]-4-methyl-pentanoylamino}-hexanoylamino)-succinamic acid 212670 (7-methyl-1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone 212671 (7-amino-1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone 212672 (7-chloro-1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone 212710 FGGFTGARKSARK 212720 FGGFTGARKSARK 212722 FGGFTGARKSARK 212724 (4,5-dichloro-1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone 212732 1-Phenyl-2-(3-pyridin-2-yl-isoquinolin-1-yl)-propan-1-one 212751 (5,7-dichloro-1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone 212752 (7-bromo-1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone 212753 (6-bromo-1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone 212756 FGGFTGARKSARKLADE 212760 1-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-2-[8-(4-methyl-piperazin-1-yl)-naphthalen-2-yloxy]-ethanone 212773 (5-amino-1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone 212774 (5-hydroxy-1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone 212794 1-[4-(2,3-Dimethoxy-phenyl)-piperazin-1-yl]-2-[8-(4-methyl-piperazin-1-yl)-naphthalen-2-yloxy]-ethanone 212800 (5-methoxy-1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone 212801 (5-methyl-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone 212806 2-[8-(4-Methyl-piperazin-1-yl)-naphthalen-2-yloxy]-1-(4-o-tolyl-piperazin-1-yl)-ethanone 212828 FGGFTGARKSARK 212829 FGGFTGARKSARK 212830 FGGFTGARKSARK 212856 3-[2-(2-{2-[2-({2-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl}-amino)-3-phenyl-propionylamino]-3-phenyl-propionylamino}-4-methyl-pentanoylamino)-hexanoylamino]-succinamic acid 212869 (4-bromo-1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone 212903 (5-bromo-1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone 212980 (5,7-dimethyl-1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone 213018 1-Phenyl-3-pyridin-2-yl-isoquinoline 213053 2-[8-(4-Methyl-piperazin-1-yl)-naphthalen-2-yloxy]-1-[4-(2,4,6-trimethyl-phenyl)-piperazin-1-yl]-ethanone 213060 1-Methylsulfanyl-3-pyridin-2-yl-isoquinoline 213096 (S)-2-({(4R,7S,13S)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7-benzyl-14,14-dimethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradecane-4-carbonyl}-amino)-3-phenyl-propionic acid 213186 N-Benzoyl-N-(3-pyridin-2-yl-isoquinolin-1-yl)-benzamide 213197 (S)-3-[2-({(S)-2-[(S)-2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-4-methylsulfanyl-butyrylamino}-3-phenyl-propionylamino)-3-(3H-imidazol-4-yl)-propionylamino]-4-methyl-pentanoyl}-butyl-amino)-acetylamino]-succinamic acid 213239 (S)-3-[2-({(S)-2-[(S)-2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-4-methylsulfanyl-butylamino}-3-phenyl-propionylamino)-3-(3H-imidazol-4-yl)-propionylamino]-4-methyl-pentanoyl}-butyl-amino)-acetylamino]-succinamic acid 213245 3-Propyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ol 213247 3-Ethyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-6-ol 213256 (S)-3-((S)-2-{(S)-2-[(S)-2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-4-methylsulfanyl-butyrylamino}-3-phenyl-propionylamino)-3-(3H-imidazol-4-yl)-propionylamino]-4-methyl-pentanoylamino}-3,3-dimethyl-butyrylamino)-succinamic acid 213310 (S)-3-[2-({(S)-2-[(S)-2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-4-methylsulfanyl-butylamino}-3-phenyl-propionylamino)-3-(3H-imidazol-4-yl)-propionylamino]-3,3-dimethyl-butyryl}-butyl-amino)-acetylamino]-succinamic acid 213324 3-Propyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-6-ol 213325 6-Methoxy-3-propyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine 213372 6-Bromo-9-methoxy-3-propyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine 213396 6-Methoxy-3-methyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine 213403 (S)-3-((S)-2-{(S)-2-[(S)-2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-4-methylsulfanyl-butyrylamino}-3-phenyl-propionylamino)-3-(3H-imidazol-4-yl)-propionylamino]-propionylamino}-4-methylsulfanyl-butyrylamino)-succinamic acid 213432 3-Methyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-6-ol 213433 3-Ethyl-6-methoxy-2,3,4,5-tetrahydro-1H-benzo[d]azepine 213434 3-Cyclopropylmethyl-6-methoxy-2,3,4,5-tetrahydro-1H-benzo[d]azepine 213464 (S)-3-[2-({(S)-2-[(S)-2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-4-methylsulfanyl-butyrylamino}-3-phenyl-propionylamino)-3-(3H-imidazol-4-yl)-propionylamino]-3,3-dimethyl-butyryl}-butyl-amino)-acetylamino]-succinamic acid 213498 1-Methoxy-3-pyridin-2-yl-isoquinoline 213561 1-Methanesulfonyl-3-pyridin-2-yl-isoquinoline 213641 (S)-3-[2-({(S)-2-[(S)-2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-4-methylsulfanyl-butyrylamino}-3-phenyl-propionylamino)-3-(3H-imidazol-4-yl)-propionylamino]-4-methyl-pentanoyl}-isobutyl-amino)-acetylamino]-succinamic acid 213674 3-(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-4-methylsulfanyl-butyrylamino}-3-phenyl-propionylamino)-3-(1H-imidazol-4-yl)-propionylamino]-3,3-dimethyl-butyrylamino}-4-methylsulfanyl-butyrylamino)-succinamic acid 213747 3-Butyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-6-ol 213769 2-[[(tert-butyloxy)carbonyl]-amino]-4-methyl-N-(2,6-dichlorophenyl)-1,3-thiazole-5-carboxamide 213770 2-[[(tert-butyloxy)carbonyl]-amino]-4-methyl-N-(2-chloro-6-methylphenyl)-1,3-thiazole-5-carboxamide 213780 3-methoxy-N-(3-(pyridin-2-yl)isoquinolin-1-yl)benzamide 213784 2-[[(butylamino)-carbonyl]amino]-4-methyl-N-(2,4,6-trimethylphenyl)-1,3-thiazole-5-carboxamide 213807 Opioid Peptide [d-Ala(8)]Dynorphin derivative 213808 Opioid Peptide [d-Ala(8)]Dynorphin derivative 213825 2-[[(methoxy)carbonyl]-amino]-4-methyl-N-(2,4,6-trimethylphenyl)-1,3-thiazole-5-carboxamide 213836 2-[[(methylamino)-carbonyl]amino]-4-methyl-N-(2,4,6-trimethylphenyl)-1,3-thiazole-5-carboxamide 213855 2-[[(tert-butyloxy)carbonyl]-amino]-4-methyl-N-(2,6-dimethylphenyl)-1,3-thiazole-5-carboxamide 213857 N-(3-Pyridin-2-yl-isoquinolin-1-yl)-isobutyramide 213859 2-[(benzoyl)amino]-4-methyl-N-(2,4,6-trimethylphenyl)-1,3-thiazole-5-carboxamide 213861 3,4-dimethoxy-N-(3-(pyridin-2-yl)isoquinolin-1-yl)benzamide 213870 biphenyl-2-yl-[1-(4,5-dihydro-1H-imidazol-2-yl)-ethyl]-amine 213886 2-[[(tert-butyloxy)carbonyl]-amino]-4-methyl-N-(4-bromo-2,6-dimethylphenyl)-1,3-thiazole-5-carboxamide 213978 3-methyl-N-(3-(pyridin-2-yl)isoquinolin-1-yl)benzamide 213979 TCMDC-123886 213982 2-[[(furanyl)carbonyl]-amino]-4-methyl-N-(2-chloro-6-methylphenyl)-1,3-thiazole-5-carboxamide 213988 rac-2-(1-(biphenyl-2-yloxy)ethyl)-4,5-dihydro-1H-imidazole 214007 2-[[(tert-butyloxy)carbonyl]-amino]-4-methyl-N-(2-methoxy-6-methylphenyl)-1,3-thiazole-5-carboxamide 214016 2,4-dimethyl-N-(3-(pyridin-2-yl)isoquinolin-1-yl)benzamide 214018 Opioid Peptide [d-Ala(8)]Dynorphin derivative 214019 Opioid Peptide [d-Ala(8)]Dynorphin derivative 214047 2-[[(furanyl)carbonyl]-amino]-4-methyl-N-(2,4,6-trimethylphenyl)-1,3-thiazole-5-carboxamide 214195 Biphenyl-2-carboxylic acid [4-(2-dimethylaminomethyl-3,4-dihydro-2H-benzo[b][1,4]thiazepine-5-carbonyl)-phenyl]-amide 214201 FGGFTGARKCARKC 214202 FGGFTGCRKSARKC 214203 FGGFTGCRKSARKC 214204 (5-{4-[(Biphenyl-2-carbonyl)-amino]-benzoyl}-2,3,4,5-tetrahydro-benzo[b][1,4]thiazepin-2-yl)-acetic acid 214205 2-Butoxy-3-(1-methyl-1,2,5,6-tetrahydro-pyridin-3-yl)-pyrazine 214213 Opioid Peptide [d-Ala(8)]Dynorphin derivative 214214 Opioid Peptide [d-Ala(8)]Dynorphin derivative 214223 2-[[(tert-butyloxy)carbonyl]-amino]-4-methyl-N-(2-methylphenyl)-1,3-thiazole-5-carboxamide 214272 N-(2-Pyridin-2-yl-quinazolin-4-yl)-formamidine 214274 2-Ethoxy-3-(1-methyl-1,2,5,6-tetrahydro-pyridin-3-yl)-pyrazine 214275 2-Methoxy-3-(1-methyl-1,2,5,6-tetrahydro-pyridin-3-yl)-pyrazine 214280 Opioid Peptide [d-Ala(8)]Dynorphin derivative 214281 Opioid Peptide [d-Ala(8)]Dynorphin derivative 214312 2-Hexylsulfanyl-3-(1-methyl-1,2,5,6-tetrahydro-pyridin-3-yl)-pyrazine 214395 Opioid Peptide [d-Ala(8)]Dynorphin derivative 214470 2-(1-Methyl-1,2,5,6-tetrahydro-pyridin-3-yl)-3-propoxy-pyrazine 214499 4-methyl-N-(3-(pyridin-2-yl)isoquinolin-1-yl)benzamide 214509 N-(2-chloro-6-methylphenyl)-2-[(phenylcarbonyl)amino]-1,3-thiazole-5-carboxamide 214527 4-chloro-N-(3-(pyridin-2-yl)isoquinolin-1-yl)benzamide 214528 4-methoxy-N-(3-(pyridin-2-yl)isoquinolin-1-yl)benzamide 214529 N-(2-chloro-6-methylphenyl)-2-[(cyclopropylcarbonyl)amino]-1,3-thiazole-5-carboxamide 214539 2-[[(tert-butyloxy)carbonyl]-amino]-4-methyl-N-(2-isopropyl-6-methylphenyl)-1,3-thiazole-5-carboxamide 214545 2-[[(n-butylamino)carbonyl]-amino]-4-methyl-N-(2-chloro-6-methylphenyl)-1,3-thiazole-5-carboxamide 214546 2-[(benzoyl)-amino]-4-methyl-N-(2-chloro-6-methylphenyl)-1,3-thiazole-5-carboxamide 214555 2-[[(cyclopropyl)carbonyl]-amino]-4-methyl-N-(2-chloro-6-methylphenyl)-1,3-thiazole-5-carboxamide 214604 3,4-dimethyl-N-(3-(pyridin-2-yl)isoquinolin-1-yl)benzamide 214625 FGGFTGCRKSCRK 214626 FGGFTGCRKSCRK 214713 (2-Phenoxy-ethyl)-(3-phenoxy-propyl)-amine 214715 [2-(2-Chloro-phenoxy)-ethyl]-(3-phenoxy-propyl)-amine 214747 [2-(3-Chloro-phenoxy)-ethyl]-(3-phenoxy-propyl)-amine 214751 17,20-dioxa-4,12,14,23-tetraazahexacyclo[21.6.1.17,14.02,6.08,13.024,29]hentriaconta-1(30),2(6),7(31),8,10,12,24,26,28-nonaene-3,5-dione 214752 8-(1-Methyl-2-phenyl-ethyl)-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 214753 17,20,23,26-tetraoxa-4,14,29-triazahexacyclo[27.6.1.17,14.02,6.08,13.030,35]heptatriaconta-1(36),2(6),7(37),8,10,12,30,32,34-nonaene-3,5-dione 214822 17,20,23-trioxa-4,12,14,26,28-pentaazahexacyclo[24.6.1.17,14.02,6.08,13.027,32]tetratriaconta-1(33),2(6),7(34),8,10,12,27,29,31-nonaene-3,5-dione 214861 SID26755653 214863 17,20,23,26,29-pentaoxa-4,14,32-triazahexacyclo[30.6.1.17,14.02,6.08,13.033,38]tetraconta-1(39),2(6),7(40),8,10,12,33,35,37-nonaene-3,5-dione 214880 8-(1-Methyl-2-phenyl-ethyl)-1,3-dipropyl-3,9-dihydro-purine-2,6-dione 214945 [2-(4-Methoxy-phenoxy)-ethyl]-(3-phenoxy-propyl)-amine 214952 Indolylylmaleimide 2 214965 17,20-dioxa-4,14,23-triazahexacyclo[21.6.1.17,14.02,6.08,13.024,29]hentriaconta-1(30),2(6),7(31),8,10,12,24,26,28-nonaene-3,5-dione 214970 (3-Phenoxy-propyl)-(2-p-tolyloxy-ethyl)-amine 214972 (3-Phenoxy-propyl)-(2-m-tolyloxy-ethyl)-amine 214973 (3-Phenoxy-propyl)-(2-o-tolyloxy-ethyl)-amine 214994 Indolylylmaleimide 1 215039 [2-(3-Chloro-4-methyl-phenoxy)-ethyl]-(3-phenoxy-propyl)-amine 215041 (2-p-Tolyloxy-ethyl)-(3-m-tolyloxy-propyl)-amine 215048 [2-(4-Chloro-phenoxy)-ethyl]-[3-(4-fluoro-phenoxy)-propyl]-amine 215069 (2-p-Tolyloxy-ethyl)-(3-o-tolyloxy-propyl)-amine 215072 [3-(4-Bromo-phenoxy)-propyl]-[2-(4-chloro-phenoxy)-ethyl]-amine 215073 [2-(4-Chloro-phenoxy)-ethyl]-(3-p-tolyloxy-propyl)-amine 215091 2-(1-Methyl-1,2,5,6-tetrahydro-pyridin-3-yl)-3-pentylsulfanyl-pyrazine 215092 2-(1-Methyl-1,2,5,6-tetrahydro-pyridin-3-yl)-3-pentyloxy-pyrazine 215104 (2-Phenoxy-ethyl)-(3-p-tolyloxy-propyl)-amine 215127 8-(1-Methyl-2-phenyl-ethyl)-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 215158 CFGGFTGARKCARK 215159 CFGGFTGARKCARK 215160 CFGGFTCARKSARK 215172 [2-(4-Nitro-phenoxy)-ethyl]-(3-phenoxy-propyl)-amine 215188 ((R)-5-{4-[(Biphenyl-2-carbonyl)-amino]-benzoyl}-2,3,4,5-tetrahydro-benzo[b][1,4]thiazepin-2-yl)-acetic acid 215209 5-methoxy-3-(4-(4-phenyl-5,6-dihydropyridin-1(2H)-yl)butyl)-1H-indole 215220 Biphenyl-2-carboxylic acid {4-[2-(2,2-difluoro-ethyl)-3,4-dihydro-2H-benzo[b][1,4]thiazepine-5-carbonyl]-phenyl}-amide 215222 3-((R)-5-{4-[(Biphenyl-2-carbonyl)-amino]-benzoyl}-2,3,4,5-tetrahydro-benzo[b][1,4]thiazepin-2-yl)-propionic acid 215224 2-Chloro-3-(1-methyl-1,2,5,6-tetrahydro-pyridin-3-yl)-pyrazine 215225 5-(4-Hexylsulfanyl-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2,3,6-tetrahydro-pyridine 215237 Biphenyl-2-carboxylic acid {4-[2-(2-tetrazol-1-yl-ethyl)-3,4-dihydro-2H-benzo[b][1,4]thiazepine-5-carbonyl]-phenyl}-amide 215238 2-(5-{4-[(Biphenyl-2-carbonyl)-amino]-benzoyl}-2,3,4,5-tetrahydro-benzo[b][1,4]thiazepin-2-yl)-ethanesulfonic acid 215246 1-Methyl-5-(4-pentylsulfanyl-[1,2,5]thiadiazol-3-yl)-1,2,3,6-tetrahydro-pyridine 215254 FGGFTCARKCARK 215263 Biphenyl-2-carboxylic acid {4-[2-(2-hydroxy-ethyl)-3,4-dihydro-2H-benzo[b][1,4]thiazepine-5-carbonyl]-phenyl}-amide 215267 [3-(4-Fluoro-phenoxy)-propyl]-(2-p-tolyloxy-ethyl)-amine 215268 [3-(4-Bromo-phenoxy)-propyl]-(2-p-tolyloxy-ethyl)-amine 215282 cyclo[Cys6,Cys10]N/OFQ(1-13)NH2 215283 FGGFTGARKCARKC 215289 2-Heptyloxy-3-(1-methyl-1,2,5,6-tetrahydro-pyridin-3-yl)-pyrazine 215311 (2-p-Tolyloxy-ethyl)-(3-p-tolyloxy-propyl)-amine 215319 Biphenyl-2-carboxylic acid {4-[2-(2-fluoro-ethyl)-3,4-dihydro-2H-benzo[b][1,4]thiazepine-5-carbonyl]-phenyl}-amide 215351 3-((S)-5-{4-[(Biphenyl-2-carbonyl)-amino]-benzoyl}-2,3,4,5-tetrahydro-benzo[b][1,4]thiazepin-2-yl)-propionic acid 215370 7-Butyl-1-methyl-3-propyl-3,7-dihydro-purine-2,6-dione 215399 3-Ethyl-1-methyl-3,7-dihydro-purine-2,6-dione 215421 1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-4-indan-1-ylmethyl-piperazine 215458 1-Ethyl-3,7-dihydro-purine-2,6-dione 215525 3-Butyl-1-methyl-3,7-dihydro-purine-2,6-dione 215621 FGGFTGARKSARKL 215622 CFGGFTCARKSARK 215624 ((S)-5-{4-[(Biphenyl-2-carbonyl)-amino]-benzoyl}-2,3,4,5-tetrahydro-benzo[b][1,4]thiazepin-2-yl)-acetic acid 215643 1-Butyl-3-propyl-3,7-dihydro-purine-2,6-dione 215743 [2-(3,4-Dimethyl-phenoxy)-ethyl]-(3-phenoxy-propyl)-amine 215788 [2-(4-Chloro-phenoxy)-ethyl]-(3-phenoxy-propyl)-amine 215840 1-(2-Bicyclo[4.2.0]octa-1,3,5-trien-7-yl-ethyl)-4-(2,3-dihydro-benzo[1,4]dioxin-5-yl)-piperazine 215884 H-Thi-Lys-AspMet-GIn-Leu-Gly-Arg-OH 215885 H-Phe-Lys-AspMet-GIn-Leu-Gly-Arg-OH 215893 H-Ala-Asn-Ile-Ser-Phe-Lys-AspMet-GIn-Leu-Gly-Arg-OH 215924 H-Leu-Arg-Ala-Asn-Ile-Ser-Phe-Lys-AspMet-GIn-Leu-Gly-Arg-OH 215940 Hca-Lys-AspMet-GIn-Leu-Gly-Arg-OH 215972 spiro[4,5-dihydro-1H-imidazole-4,2'-(1',2',3',4'-tetrahydronaphthalene)] 215973 3-Benzylsulfanyl-4-oxo-4,5,6,7-tetrahydro-benzo[c]thiophene-1-carboxylic acid 215975 H-hPhe-Lys-AspMet-GIn-Leu-Gly-Arg-OH 215976 H-Phg-Lys-AspMet-GIn-Leu-Gly-Arg-OH 215977 H-Cha-Lys-AspMet-GIn-Leu-Gly-Arg-OH 215992 8-chlorospiro[1,2,3,4-tetrahydronaphthalene-2,4'-(4',5'-dihydro[1,3]oxazole)]-2'-amine 216176 H-DPhe-Lys-AspMet-GIn-Leu-Gly-Arg-OH 216400 8'-fluorospiro[4,5-dihydro-1H-imidazole-4,2'-(1',2',3',4'-tetrahydronaphthalene)] 216418 {4-[({[{[{[Carbamoylmethyl-(3-phenyl-propyl)-carbamoyl]-methyl}-(3-phenyl-propyl)-carbamoyl]-methyl}-(3-phenyl-propyl)-carbamoyl]-methyl}-hexanoyl-amino)-methyl]-benzyl}-phosphonic acid 216459 8'-methoxyspiro[4,5-dihydro-1H-imidazole-4,2'-(1',2',3',4'-tetrahydronaphthalene)] 216499 H-Thia-Lys-AspMet-GIn-Leu-Gly-Arg-OH 216501 H-His(1Me)-Lys-AspMet-GIn-Leu-Gly-Arg-OH 216502 H-His(3Me)-Lys-AspMet-GIn-Leu-Gly-Arg-OH 216521 (2R,3R,4S,5R)-2-{2-Cyclohexylamino-6-[(naphthalen-1-ylmethyl)-amino]-purin-9-yl}-5-hydroxymethyl-tetrahydro-furan-3,4-diol 216769 [4-({[({[[(Carbamoylmethyl-ethyl-carbamoyl)-methyl]-(3-phenyl-propyl)-carbamoyl]-methyl}-ethyl-carbamoyl)-methyl]-hexanoyl-amino}-methyl)-benzyl]-phosphonic acid 216872 5',7'-dichlorospiro[4,5-dihydro-1H-imidazole-4,2'-(1',2',3',4'-tetrahydronaphthalene)] 216950 SID26727996 216954 5'-methoxyspiro[4,5-dihydro-1H-imidazole-4,2'-(1',2',3',4'-tetrahydronaphthalene)] 216994 4-Hydroxy-3-methylsulfanyl-4,5,6,7-tetrahydro-benzo[c]thiophene-1-carboxylic acid ethyl ester 217001 6'-methoxyspiro[4,5-dihydro-1H-imidazole-4,2'-(1',2',3',4'-tetrahydronaphthalene)] 217002 7'-methoxyspiro[4,5-dihydro-1H-imidazole-4,2'-(1',2',3',4'-tetrahydronaphthalene)] 217005 2-Hydroxymethyl-5-{6-[(naphthalen-1-ylmethyl)-amino]-purin-9-yl}-tetrahydro-furan-3,4-diol 217031 3-Ethoxycarbonylmethylsulfanyl-4-oxo-4,5,6,7-tetrahydro-benzo[c]thiophene-1-carboxylic acid ethyl ester 217302 2-(4-(4-(5-fluoro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)butyl)isoindoline-1,3-dione 217303 {4-[({[({[(Carbamoylmethyl-isobutyl-carbamoyl)-methyl]-ethyl-carbamoyl}-methyl)-isobutyl-carbamoyl]-methyl}-hexanoyl-amino)-methyl]-benzyl}-phosphonic acid 217387 {4-[({[({[(Carbamoylmethyl-isobutyl-carbamoyl)-methyl]-isobutyl-carbamoyl}-methyl)-ethyl-carbamoyl]-methyl}-hexanoyl-amino)-methyl]-benzyl}-phosphonic acid 217431 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzoic acid methyl ester 217595 Phosphoric acid mono-[(2R,3S,5R)-5-(2-chloro-6-methylamino-purin-9-yl)-2-phosphonooxymethyl-tetrahydro-furan-3-yl] ester 217872 {4-[({[({[(Carbamoylmethyl-ethyl-carbamoyl)-methyl]-ethyl-carbamoyl}-methyl)-isobutyl-carbamoyl]-methyl}-hexanoyl-amino)-methyl]-benzyl}-phosphonic acid 217939 [({[(2R,3S,4R,5R)-5-[6-amino-2-(methylsulfanyl)-9H-purin-9-yl]-3,4-dihydroxyoxolan-2-yl]methoxy}(hydroxy)phosphoryl)oxy]phosphonic acid 218157 4-Amino-N-(1-butyl-piperidin-4-ylmethyl)-5-chloro-2-methoxy-benzamide 218159 3,4-Dihydro-2H-benzo[b][1,4]dioxepine-6-carboxylic acid 1-butyl-piperidin-4-ylmethyl ester 218188 Benzo[1,3]dioxole-4-carboxylic acid 1-butyl-piperidin-4-ylmethyl ester 218324 2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid 1-butyl-piperidin-4-ylmethyl ester 218369 c(Cys-Ser-c(Cys-Ser-Ser-Leu-Met-Asp-Lys-Gln-Cys)-Val-Tyr-Phe-Cys)-His-Leu-Leu-Ile-Ile-Trp 218370 c(Cys-Ser-c(Cys-Ser-Ser-Leu-Met-Asp-Lys-Gln-Cys)-Val-Tyr-Phe-Cys)-His-Leu-Asp-Leu-Ile-Trp 218591 c(Cys-Ser-Cys)-Ser-Ser-Leu-Met-Asp-Lys-Gln-c(Cys-Val-Tyr-Phe-Cys)-His-Leu-Asp-Ile-Ile-Trp 218622 1-[5-(4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-ylamino}-phenyl)-benzofuran-2-yl]-ethanone 218671 (4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-ylamino}-phenyl)-urea 218693 {4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-yl}-(4-trifluoromethyl-phenyl)-amine 218694 (4-Butyl-phenyl)-{4-[4-(piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-yl}-amine 218716 4-Amino-5-chloro-2-methoxy-benzoic acid 1-butyl-piperidin-4-ylmethyl ester 218764 5-(4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-ylamino}-phenyl)-1H-indole-3-carboxylic acid amide 218849 4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-ylamino}-benzamide 218850 1-(4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-ylamino}-phenyl)-ethanone 218851 (4-Benzothiazol-6-yl-phenyl)-{4-[4-(piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-yl}-amine 218874 (4-Nitro-phenyl)-{4-[4-(piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-yl}-amine 218884 (4-Methoxy-phenyl)-{4-[4-(piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-yl}-amine 218885 {4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-yl}-p-tolyl-amine 218886 N-(4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-ylamino}-phenyl)-acetamide 218887 (4-Chloro-phenyl)-{4-[4-(piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-yl}-amine 218933 {4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-yl}-(3,4,5-trimethoxy-phenyl)-amine 218955 Asp-Tyr-D-Phe-Gly-Trp-NMeNle-Asp-Phe-NH2 218963 4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-ylamino}-benzenesulfonamide 218965 (4-Methanesulfonyl-phenyl)-{4-[4-(piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-yl}-amine 218974 3-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-ylamino}-benzonitrile 218975 Phenyl-{4-[4-(piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-yl}-amine 218976 (4-Methanesulfinyl-phenyl)-{4-[4-(piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-yl}-amine 219000 (3,4-Difluoro-phenyl)-{4-[4-(piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-yl}-amine 219055 3'-amino-3'-deoxyadenosine 219060 5-[6-(4-Amino-3-iodo-benzylamino)-purin-9-yl]-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid methylamide 219064 N-(4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-ylamino}-phenyl)-methanesulfonamide 219065 4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-ylamino}-benzonitrile 219106 1-Benzo[b]thiophen-3-yl-3-[4-(2,3-dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propan-1-ol 219233 4-Amino-5-[2-chloro-6-(3-iodo-benzylamino)-purin-9-yl]-tetrahydro-furan-2-carboxylic acid methylamide 219271 (2R,3R,4S,5S)-4-Amino-5-hydroxymethyl-2-[6-(3-iodo-benzylamino)-purin-9-yl]-tetrahydro-furan-3-ol 219308 1-Benzo[b]thiophen-3-yl-3-[4-(1H-indol-4-yl)-piperazin-1-yl]-propan-1-ol 219334 SID11111644 219337 1-Benzo[b]thiophen-3-yl-3-[4-(1,2-dihydro-quinolin-2-yl)-piperazin-1-yl]-propan-1-ol 219368 1-(benzo[b]thiophen-3-yl)-3-(4-(quinolin-8-yl)piperazin-1-yl)propan-1-ol 219370 3-(9-methyl-2-phenethyl-2-aza-bicyclo[3.3.1]nonan-5-yl)phenol 219453 7-Methyl-2-phenyl-4-((E)-styryl)-1,4-dihydro-quinoline-3,6-dicarboxylic acid diethyl ester 219686 2-(4-Methylsulfanyl-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-6-ylsulfanyl)-pentanoic acid amide 219711 2-(4-Mercapto-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-6-ylsulfanyl)-butyramide 219712 2-(4-Mercapto-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-6-ylsulfanyl)-3-methyl-butyramide 219713 2-(4-Mercapto-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-6-ylsulfanyl)-hexanoic acid amide 219714 3-Methyl-2-(4-methylsulfanyl-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-6-ylsulfanyl)-butyramide 219732 (2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-(2-aminoethyl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 219775 2-(4-Methylsulfanyl-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-6-ylsulfanyl)-hexanoic acid amide 219794 6-[2-Oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyrido[3,2-b][1,4]diazepin-11-yl)-ethylamino]-hexanoic acid {8-[(6-amino-hexanoyl)-methyl-amino]-octyl}-methyl-amide 219811 2-(4-Methylsulfanyl-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-6-ylsulfanyl)-butyramide 219813 2-(4-Amino-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-6-ylsulfanyl)-hexanoic acid amide 219831 3-(4-(2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)-1-(5-fluorobenzo[b]thiophen-3-yl)propan-1-ol 219834 1-(5-Fluoro-benzo[b]thiophen-3-yl)-3-[4-(1H-indol-4-yl)-piperazin-1-yl]-propan-1-ol 219847 2-(4-Mercapto-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-6-ylsulfanyl)-pentanoic acid amide 219926 3-(4-(3,4-dihydro-2H-benzo[b][1,4]dioxepin-6-yl)piperazin-1-yl)-1-(5-fluorobenzo[b]thiophen-3-yl)propan-1-ol 220141 (4aR,10bR)-4-((E)-3-Iodo-allyl)-1,2,3,4,4a,5,6,10b-octahydro-benzo[f]quinolin-7-ol 220184 Azakenpaullone 220185 9-Bromo-5,12-dihydro-7H-4,5,12-triaza-dibenzo[a,e]azulen-6-one 220363 6-[5-Oxo-5-(6-oxo-5,6-dihydro-benzo[e]pyrido[3,2-b][1,4]diazepin-11-yl)-pentylamino]-hexanoic acid {8-[(6-amino-hexanoyl)-methyl-amino]-octyl}-methyl-amide 220538 6-[2-Oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyrido[3,2-b][1,4]diazepin-11-yl)-ethylamino]-hexanoic acid {8-[(6-{bis-[2-oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyrido[3,2-b][1,4]diazepin-11-yl)-ethyl]-amino}-hexanoyl)-methyl-amino]-octyl}-methyl-amide 220540 2-(4-Amino-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-6-ylsulfanyl)-pentanoic acid amide 220542 2-(4-Amino-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-6-ylsulfanyl)-3-methyl-butyramide 220543 2-(4-Amino-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-6-ylsulfanyl)-butyramide 220610 1-((E)-3-Iodo-allyl)-6-methoxy-1,2,3,4,4a,5,10,10a-octahydro-benzo[g]quinoline 220617 1-((E)-3-Iodo-allyl)-1,2,3,4,4a,5,10,10a-octahydro-benzo[g]quinoline 220630 1-Prop-2-ynyl-1,2,3,4,4a,5,10,10a-octahydro-benzo[g]quinolin-6-ol 220631 1-((E)-3-Iodo-allyl)-1,2,3,4,4a,5,10,10a-octahydro-benzo[g]quinolin-6-ol 220702 (4aR,10bR)-4-((E)-3-Iodo-allyl)-7-methoxy-1,2,3,4,4a,5,6,10b-octahydro-benzo[f]quinoline 220703 (4aR,10bR)-4-((E)-3-Iodo-allyl)-1,2,3,4,4a,5,6,10b-octahydro-benzo[f]quinoline 220748 ethyl 7-(2-methoxybenzyl)-3-((benzyl(methyl)amino)methyl)-2-(4-methoxyphenyl)-4-oxo-4,7-dihydrothieno[2,3-b]pyridine-5-carboxylate 220767 1-Methyl-2-(3,7,8,9-tetrahydro-pyrano[3,2-e]indol-1-yl)-ethylamine 220768 (S)-1-Methyl-2-(3,7,8,9-tetrahydro-pyrano[3,2-e]indol-1-yl)-ethylamine 220775 (R)-1-Methyl-2-(3,7,8,9-tetrahydro-pyrano[3,2-e]indol-1-yl)-ethylamine 220854 ethyl 3-(N-benzyl-N-methylaminomethyl)-7-(2,6-difluorobenzyl)-4,7-dihydro-2-(4-methoxyphenyl)-4-oxothieno[2,3b]pyridine-5-carboxylate 220874 1-Methyl-2-(3-methyl-3,7,8,9-tetrahydro-pyrano[3,2-e]indol-1-yl)-ethylamine 220875 ethyl 7-(2-methoxybenzyl)-2-(4-methoxyphenyl)-3-((methylamino)methyl)-4-oxo-4,7-dihydrothieno[2,3-b]pyridine-5-carboxylate 220898 5'-Iodo-1H,1'H-[2,3']biindolylidene-3,2'-dione 3-oxime 220945 11-{4-[6-({8-[(6-Amino-hexyl)-methyl-amino]-octyl}-methyl-amino)-hexylamino]-butyryl}-5,11-dihydro-benzo[e]pyrido[3,2-b][1,4]diazepin-6-one 221361 (6aS,10aS)-9-(hydroxymethyl)-6,6-dimethyl-3-(2-methyloctan-2-yl)-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol 221429 3-(4-Amino-3-iodo-phenyl)-N-(2-{2-[4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-acetylamino}-ethyl)-propionamide 221482 Tetradecanedioic acid ((S)-5-hydroxymethyl-2-isopropyl-1-methyl-3-(S)-oxo-1,2,3,4,5,6-hexahydro-benzo[e][1,4]diazocin-8-yl)-amide ((S)-5-hydroxymethyl-2-isopropyl-1-(S)-methyl-3-oxo-1,2,3,4,5,6-hexahydro-benzo[e][1,4]diazocin-9-yl)-amide 221517 (R)-1-(4-iodo-2,5-dimethoxyphenyl)propan-2-amine 221828 4-(2-Acetylsulfanyl-ethyl)-2-ethyl-3-ethylsulfanylcarbonyl-1-methyl-6-phenyl-5-propoxycarbonyl-pyridinium iodide 221830 2-Ethyl-3-(3-fluoro-propylsulfanylcarbonyl)-1-methyl-6-phenyl-5-propoxycarbonyl-4-propyl-pyridinium iodide 221831 2-Ethyl-3-ethylsulfanylcarbonyl-1-methyl-6-phenyl-5-propoxycarbonyl-4-propyl-pyridinium iodide 221832 2,4-Diethyl-3-ethylsulfanylcarbonyl-1-methyl-6-phenyl-5-propoxycarbonyl-pyridinium iodide 221852 3-Ethoxycarbonyl-4,6-diethyl-5-ethylsulfanylcarbonyl-2-phenyl-1-propyl-pyridinium iodide 221853 2-(2-Benzyloxy-ethyl)-3-ethylsulfanylcarbonyl-1-methyl-6-phenyl-5-propoxycarbonyl-4-propyl-pyridinium iodide 221855 3-Ethoxycarbonyl-4,6-diethyl-5-ethylsulfanylcarbonyl-1-methyl-2-phenyl-pyridinium iodide 221873 (1R,2R,5R)-2-{[(R)-1-(2,3-Dihydro-benzo[1,4]dioxin-2-yl)methyl]-amino}-5-phenoxy-cyclopentanol 221905 (1S,2S,5S)-2-{[(R)-1-(2,3-Dihydro-benzo[1,4]dioxin-2-yl)methyl]-amino}-5-phenoxy-cyclopentanol 221959 Bicyclo[2.2.1]hept-2-yl-(9-methyl-9H-purin-6-yl)-amine 221993 1-tert-Butyl-3-[3-(3,5-dimethoxy-phenyl)-7-(3-morpholin-4-yl-propylamino)-[1,6]naphthyridin-2-yl]-urea 222022 (1R,2R,5R)-2-{[(S)-1-(2,3-Dihydro-benzo[1,4]dioxin-2-yl)methyl]-amino}-5-phenoxy-cyclopentanol 222023 (1S,2S,5S)-2-{[(S)-1-(2,3-Dihydro-benzo[1,4]dioxin-2-yl)methyl]-amino}-5-phenoxy-cyclopentanol 222043 2,4-Diethyl-3-ethylsulfanylcarbonyl-5-(2-fluoro-ethoxycarbonyl)-1-methyl-6-phenyl-pyridinium iodide 222096 N-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-cyclohexylmethyl]-acetamide 222109 4-(3-Chloro-phenoxy)-6,7-dimethoxy-quinazoline 222110 4-(3-Chloro-phenylsulfanyl)-6,7-dimethoxy-quinazoline 222200 2-Cyclobutyl-5-ethoxycarbonyl-4-ethyl-3-ethylsulfanylcarbonyl-1-methyl-6-phenyl-pyridinium iodide 222631 Tyr-Gly-Gly-Trp-NMeNle-Asp-Phe-NH2 222692 7-Methyl-8-oxo-5-p-tolyl-7,8-dihydro-[1,7]naphthyridine-6-carboxylic acid (R)-[(S)-1-(3,5-bis-trifluoromethyl-phenyl)-ethyl]-methyl-amide 222694 7-Methyl-8-oxo-5-p-tolyl-7,8-dihydro-[1,7]naphthyridine-6-carboxylic acid (R)-[(R)-1-(3,5-bis-trifluoromethyl-phenyl)-ethyl]-methyl-amide 222745 1-(2-Isopropoxy-phenyl)-4-(4-pyrrolidin-1-ylmethyl-benzyl)-piperazine 222773 7-Methyl-8-oxo-5-p-tolyl-7,8-dihydro-[1,7]naphthyridine-6-carboxylic acid (S)-methyl-((S)-1-phenyl-ethyl)-amide 222860 4-[2-(1,3-Dioxo-1,3-dihydro-isoindol-2-yl)-ethyl]-3-ethoxycarbonyl-6-ethyl-5-ethylsulfanylcarbonyl-1-methyl-2-phenyl-pyridinium iodide 222909 [R-(R*,R*)]-2,2'-Diselenobis [alpha-amino-N-(phenylmethyl)-1H-indole-3-propanamide] 222910 [R-(R*,R*)]-2,2'-Diselenobis [N-(phenyl-methyl)-alpha-[(trifluoroacetyl)amino]-1H-indole-3-propanamide] 222953 1-(2-Isopropoxy-phenyl)-4-(3-piperidin-1-ylmethyl-benzyl)-piperazine 222954 (4-Fluoro-phenyl)-{3-[4-(2-isopropoxy-phenyl)-piperazin-1-ylmethyl]-benzyl}-amine 223003 5-{3-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-benzyl}-imidazolidine-2,4-dione 223051 4-(3-Chloro-4-fluoro-phenylamino)-7,8-dimethoxy-benzo[g]quinoline-3-carbonitrile 223165 2,2'-Diselenobis[N-[2-(diethylamino)ethyl]-1-methyl-1H-indole-3-carboxamide] 223166 2,2'-Diselenobis[N-[2-(diethylamino)ethyl]-1H-indole-3-carboxamide] 223187 4-(4-Chloro-5-methoxy-2-methyl-phenylamino)-7,8-dimethoxy-benzo[g]quinoline-3-carbonitrile 223205 2-Cyclopentyl-3-ethoxycarbonyl-4,6-diethyl-5-ethylsulfanylcarbonyl-1-methyl-pyridinium iodide 223206 3-Ethoxycarbonyl-4-ethyl-5-ethylsulfanylcarbonyl-1,6-dimethyl-2-phenyl-pyridinium iodide 223209 (S)-(2-Methoxy-benzyl)-((S)-2-phenyl-piperidin-3-yl)-amine 223237 2-Butyl-5-ethoxycarbonyl-4-ethyl-3-ethylsulfanylcarbonyl-1-methyl-6-phenyl-pyridinium iodide 223238 3-Ethoxycarbonyl-1,4,6-triethyl-5-ethylsulfanylcarbonyl-2-phenyl-pyridinium iodide 223311 2,2'-Diselenobis[N-methyl-1H-indole-3-carboxamide] 223343 2,2'-Diselenobis[N,1-dimethyl-1H-indole-3-carboxamide] 223400 (1R,3S,4R)-1-Aza-bicyclo[2.2.1]hept-3-yl-[(Z)-methoxyimino]-acetonitrile 223423 1-methyl-5-(4-(2-(2-(2-(2-(4-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)-1,2,5-thiadiazol-3-yloxy)ethoxy)ethoxy)ethoxy)ethoxy)-1,2,5-thiadiazol-3-yl)-1,2,3,6-tetrahydropyridine 223450 (1-Aza-bicyclo[2.2.1]hept-4-yl)-[(Z)-methoxyimino]-acetonitrile 223517 3-(1H-imidazol-4-yl)propyl isopropylcarbamate compound with (2E)-2,3-dihydroxybut-2-enedial (1:1); 0.25hydrate 223617 2-Amino-3-{2-[3-(2-amino-2-benzylcarbamoyl-ethyl)-1H-indol-2-yldisulfanyl]-1H-indol-3-yl}-N-benzyl-propionamide 223649 2,2'-Diselenobis[1-[2-(diethylamino)ethyl]-N-methyl-1H-indole-3-carboxamide] 223772 sodium (S)-2-(3-((2-(4,5-diphenyloxazol-2-yl)cyclohex-2-enyl)methyl)phenoxy)acetate 223806 1,3N-dimethyl-2-(1-methyl-3-methylcarbamoyl-1H-2-indolyldisulfanyl)-1H-3-indolecarboxamide0.5 H2O 223807 2,2'-Diselenobis[1-methyl-1H-indole-3-carboxylic acid] 223815 sodium 2-(3-((2-(4,5-diphenyloxazol-2-yl)cyclohex-1-enyl)methyl)phenoxy)acetate 223862 [4-(3-Chloro-benzoyloxy)-but-2-ynyl]-trimethyl-ammonium 223863 5-{4-[12-(4-Methoxy-[1,2,5]thiadiazol-3-yloxy)-dodecyloxy]-[1,2,5]thiadiazol-3-yl}-1-methyl-1,2,3,6-tetrahydro-pyridine 223880 1'-propylspiro[3,4-dihydro-2H-chromene-3,2'-(tetrahydro-1'H-pyrrole)]-5-ol 224034 (1,1,3,3-Tetramethyl-butyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester oxalic acid 224076 (2,2-Dimethyl-propyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester oxalic acid; 0.5hydrate 224085 (R)-3-{cyano-[(E)-hydroxyimino]-methyl}-1-azonia-bicyclo[2.2.2]octane 224211 (1R,3R,4R)-1-Aza-bicyclo[2.2.1]heptane-3-carbaldehyde O-methyl-oxime 224212 (1-Aza-bicyclo[3.2.1]oct-5-yl)-[(Z)-methoxyimino]-acetonitrile 224305 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-3-(2-nitro-benzyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 224392 (1R,3R,4R)-1-Aza-bicyclo[2.2.1]hept-3-yl-[(Z)-methoxyimino]-acetonitrile 224412 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-3-(4-methyl-benzyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 224444 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-3-(2-methoxy-benzyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 224478 N-(2-(furan-2-yl)-8-(3-phenylpropyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-2-(naphthalen-1-yl)acetamide 224479 N-(2-Furan-2-yl-8-phenethyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-2-naphthalen-1-yl-acetamide 224566 8-{2-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-ethyl}-8-aza-spiro[4.5]decane-7,9-dione 224600 1-{2-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-ethyl}-4,4-dimethyl-piperidine-2,6-dione 224602 1-{2-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-ethyl}-piperidine-2,6-dione 224681 N-[2-Furan-2-yl-8-(3-phenyl-propyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl]-2-phenyl-acetamide 224727 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-1-phenyl-3-propyl-1,3,8-triaza-spiro[4.5]decan-4-one 224728 3-Benzyl-8-[4-(4-fluoro-phenyl)-4-oxo-butyl]-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 224751 N-[2-Furan-2-yl-8-(3-methyl-butyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl]-2-phenyl-acetamide 224752 N-(2-(furan-2-yl)-8-phenethyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-2-phenylacetamide 224852 N-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-2-phenylacetamide 224870 1-{2-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-ethyl}-3-methyl-pyrrolidine-2,5-dione 224901 1-{2-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-ethyl}-pyrrolidine-2,5-dione 224902 2-{2-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-ethyl}-3a,4,7,7a-tetrahydro-isoindole-1,3-dione 224930 N-[2-Furan-2-yl-8-(3-methyl-butyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl]-2-naphthalen-1-yl-acetamide 224967 N-(2-Furan-2-yl-8-phenethyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-2-phenoxy-acetamide 224970 N-[2-Furan-2-yl-8-(3-methyl-butyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl]-2-phenoxy-acetamide 224991 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-3-(4-methoxy-benzyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 224992 3-Ethyl-8-[4-(4-fluoro-phenyl)-4-oxo-butyl]-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 225022 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-3-(4-nitro-benzyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 225037 (R)-Cyclohexyl-{(3S,4S)-3-phenyl-4-[4-(propyl-pyridin-2-yl-amino)-piperidin-1-ylmethyl]-pyrrolidin-1-yl}-acetic acid 225048 ((3S,4S)-3-((4-(allyl(pyrimidin-2-yl)amino)piperidin-1-yl)methyl)-4-phenylpyrrolidin-1-yl)(cyclohexyl)methanone 225075 ((3S,4S)-3-{4-[Allyl-(5-trifluoromethyl-pyridin-2-yl)-amino]-piperidin-1-ylmethyl}-4-phenyl-pyrrolidin-1-yl)-cyclohexyl-methanone 225083 N-[2-Furan-2-yl-8-(3-phenyl-propyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl]-2-phenoxy-acetamide 225114 (R)-2-cyclohexyl-2-((3S,4S)-3-phenyl-4-((4-(propyl(pyrimidin-2-yl)amino)piperidin-1-yl)methyl)pyrrolidin-1-yl)acetic acid 225151 (R)-Cyclohexyl-{(3S,4S)-3-(3-fluoro-phenyl)-4-[4-(propyl-pyrimidin-2-yl-amino)-piperidin-1-ylmethyl]-pyrrolidin-1-yl}-acetic acid 225155 (R)-2-cyclohexyl-2-((3S,4S)-3-phenyl-4-((4-(propyl(pyridin-3-yl)amino)piperidin-1-yl)methyl)pyrrolidin-1-yl)acetic acid 225187 (R)-3-cyclobutyl-2-((3S,4S)-3-(3-fluorophenyl)-4-((4-(propyl(pyrimidin-2-yl)amino)piperidin-1-yl)methyl)pyrrolidin-1-yl)propanoic acid 225253 2-{2-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-ethyl}-4,5,6,7-tetrahydro-isoindole-1,3-dione 225260 (R)-3-Cyclobutyl-2-[(3S,4S)-3-[4-(ethyl-pyrimidin-2-yl-amino)-piperidin-1-ylmethyl]-4-(3-fluoro-phenyl)-pyrrolidin-1-yl]-propionic acid 225274 (R)-3-Cyclobutyl-2-((3S,4S)-3-(3-fluoro-phenyl)-4-{4-[propyl-(4-trifluoromethyl-pyrimidin-2-yl)-amino]-piperidin-1-ylmethyl}-pyrrolidin-1-yl)-propionic acid 225284 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-3-(4-iodo-benzyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 225301 1-{2-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-ethyl}-3-methyl-pyrrole-2,5-dione 225320 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-3-isobutyl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 225321 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-3-pentyl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 225325 3-(2-Fluoro-benzyl)-8-[4-(4-fluoro-phenyl)-4-oxo-butyl]-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 225331 1-{2-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-ethyl}-pyrrole-2,5-dione 225332 2-{2-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-ethyl}-hexahydro-isoindole-1,3-dione 225349 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-3-(2-iodo-benzyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 225362 2-{2-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-ethyl}-5-methyl-isoindole-1,3-dione 225387 5-methoxy-1'-propylspiro[3,4-dihydro-2H-chromene-3,2'-(tetrahydro-1'H-pyrrole)] 225422 6-[6-(2-Chloro-phenyl)-4-phenyl-pyridin-2-yloxy]-2-methyl-hexanoic acid 225425 N4-(3-chlorophenyl)quinazoline-4,6-diamine 225434 (R)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-({(S)-2-[(S)-3-(1H-indol-3-yl)-2-(2-{(S)-2-[2-(4-sulfooxy-phenyl)-acetylamino]-hexanoylamino}-acetylamino)-propionylamino]-hexanoyl}-methyl-amino)-succinamic acid 225439 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-3-phenethyl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 225461 N-(3-methylphenyl)-6-[(1E)-3-methyltriaz-1-enyl]quinazolin-4-amine 225471 (R)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-{(S)-2-[(S)-3-(1H-indol-3-yl)-2-(2-{(S)-4-methylsulfanyl-2-[2-(4-sulfooxy-phenyl)-acetylamino]-butyrylamino}-acetylamino)-propionylamino]-4-methylsulfanyl-butyrylamino}-succinamic acid 225472 (R)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-{(S)-2-[(S)-3-(1H-indol-3-yl)-2-(2-{(S)-2-[2-(4-sulfooxy-phenyl)-acetylamino]-hexanoylamino}-acetylamino)-propionylamino]-hexanoylamino}-N-methyl-succinamic acid 225477 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-3-(3-methyl-butyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 225478 3-Butyl-8-[4-(4-fluoro-phenyl)-4-oxo-butyl]-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 225488 (R)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-{(S)-2-[(S)-3-(1H-indol-3-yl)-2-(2-{(S)-4-methylsulfanyl-2-[2-(4-sulfooxy-phenyl)-acetylamino]-butyrylamino}-acetylamino)-propionylamino]-4-methylsulfanyl-butyrylamino}-N-methyl-succinamic acid 225489 (S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-{(S)-2-[(S)-3-(1H-indol-3-yl)-2-(2-{(S)-4-methylsulfanyl-2-[2-(4-sulfooxy-phenyl)-acetylamino]-butyrylamino}-acetylamino)-propionylamino]-4-methylsulfanyl-butyrylamino}-N-methyl-succinamic acid 225504 N4-(3-methylphenyl)-4,6-quinazolinediamine 225529 (R)-3-Cyclobutyl-2-{(3S,4S)-3-(3-fluoro-phenyl)-4-[4-(propyl-pyrimidin-4-yl-amino)-piperidin-1-ylmethyl]-pyrrolidin-1-yl}-propionic acid 225547 SID26751844 225553 (R)-3-Cyclobutyl-2-((3S,4S)-3-(3-fluoro-phenyl)-4-{4-[(4-methoxy-pyrimidin-2-yl)-propyl-amino]-piperidin-1-ylmethyl}-pyrrolidin-1-yl)-propionic acid 225562 (R)-3-Cyclobutyl-2-((3S,4S)-3-(3-fluoro-phenyl)-4-{4-[propyl-(5-trifluoromethyl-pyrimidin-2-yl)-amino]-piperidin-1-ylmethyl}-pyrrolidin-1-yl)-propionic acid 225564 (R)-3-Cyclobutyl-2-((3S,4S)-3-(3-fluoro-phenyl)-4-{4-[(5-fluoro-pyrimidin-2-yl)-propyl-amino]-piperidin-1-ylmethyl}-pyrrolidin-1-yl)-propionic acid 225742 3-(4-Fluoro-benzyl)-8-[4-(4-fluoro-phenyl)-4-oxo-butyl]-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 225772 (S)-6-Bromo-2-methyl-1-phenyl-1,2,3,4-tetrahydro-isoquinolin-7-ol 225773 2-Methyl-1-phenyl-1,2,3,4-tetrahydro-isoquinoline-6,7-diol 225775 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-3-(2-methyl-benzyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 225789 Cyclohexyl-{(3S,4S)-3-[4-(cyclopropylmethyl-pyridin-2-yl-amino)-piperidin-1-ylmethyl]-4-phenyl-pyrrolidin-1-yl}-methanone 225811 1'-[4-(4-fluorophenylcarboxamido)butyl]-5-methoxyspiro[3,4-dihydro-2H-chromene-3,2'-(hexahydropyridine)] 225816 (2-Chloro-phenyl)-{(3S,4S)-3-phenyl-4-[4-(propyl-pyridin-2-yl-amino)-piperidin-1-ylmethyl]-pyrrolidin-1-yl}-methanone 225817 cyclohexyl((3S,4S)-3-phenyl-4-((4-(propyl(pyridin-2-yl)amino)piperidin-1-yl)methyl)pyrrolidin-1-yl)methanone 225825 ((3S,4S)-3-phenyl-4-((4-(propyl(pyridin-2-yl)amino)piperidin-1-yl)methyl)pyrrolidin-1-yl)(pyrrolidin-1-yl)methanone 225846 5-methoxy-1'-propylspiro[3,4-dihydro-2H-chromene-3,2'-(hexahydropyridine)] 225848 cyclobutyl((3S,4S)-3-phenyl-4-((4-(propyl(pyridin-2-yl)amino)piperidin-1-yl)methyl)pyrrolidin-1-yl)methanone 225857 5-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]-5-(3-isopropyl-4-methyl-pentanoyloxymethyl)tetrahydro-2-furanone 225876 5-methoxy-1'-[4-(4-methylphenylsulfonamido)butyl]spiro[3,4-dihydro-2H-chromene-3,2'-(hexahydropyridine)] 225896 5-hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]-5-(3-isopropyl-4-methyl-pentanoyloxymethyl)tetrahydro-2-furanone 225916 8-{4-[5-methoxyspiro[3,4-dihydro-2H-chromene-3,2'-(hexahydropyridine)]-1-yl]butyl}-8-azaspiro[4.5]decane-7,9-dione 226015 N-(3-bromophenyl)-6-[(1E)-3-methyltriaz-1-enyl]quinazolin-4-amine 226152 (R)-3-Cyclobutyl-2-{(3S,4S)-3-(3-fluoro-phenyl)-4-[4-(propyl-pyrimidin-5-yl-amino)-piperidin-1-ylmethyl]-pyrrolidin-1-yl}-propionic acid 226157 (R)-3-Cyclobutyl-2-[(3S,4S)-3-[4-(cyclopropylmethyl-pyrimidin-2-yl-amino)-piperidin-1-ylmethyl]-4-(3-fluoro-phenyl)-pyrrolidin-1-yl]-propionic acid 226221 {(3S,4S)-3-[4-(Allyl-pyridin-2-yl-amino)-piperidin-1-ylmethyl]-4-phenyl-pyrrolidin-1-yl}-cyclohexyl-methanone 226253 ((3S,4S)-3-((4-(allyl(pyridin-3-yl)amino)piperidin-1-yl)methyl)-4-phenylpyrrolidin-1-yl)(cyclohexyl)methanone 226418 (E)-2-(2-(hydroxymethyl)-4-(3-isobutyl-5-methylhexylidene)-5-oxo-tetrahydrofuran-2-yl)ethyl pivalate 227326 1-(4-Fluoro-phenyl)-4-(1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-butan-1-one 227480 SID29215552 227535 (S)-3-Fluoromethyl-1,2,3,4-tetrahydro-isoquinoline-7-sulfonic acid (4-chloro-phenyl)-amide 227536 (R)-3-Fluoromethyl-1,2,3,4-tetrahydro-isoquinoline-7-sulfonic acid (4-chloro-phenyl)-amide 227679 1-(4-Fluoro-phenyl)-3-(1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-propan-1-one 227789 (4R,7S,10R)-7-Benzyl-10-[(R)-3-(4-hydroxy-phenyl)-2-methylamino-propionylamino]-3,3-dimethyl-6,9-dioxo-1,2-dithia-5,8-diaza-cycloundecane-4-carboxylic acid 227889 (4R,7S,10R)-7-Benzyl-10-{[(2S,3R)-3-(4-hydroxy-phenyl)-pyrrolidine-2-carbonyl]-amino}-3,3-dimethyl-6,9-dioxo-1,2-dithia-5,8-diaza-cycloundecane-4-carboxylic acid 227910 (4R,7S,10R)-10-[((S)-2-Amino-6-hydroxy-1,2,3,4-tetrahydro-naphthalene-2-carbonyl)-amino]-7-benzyl-3,3-dimethyl-6,9-dioxo-1,2-dithia-5,8-diaza-cycloundecane-4-carboxylic acid 227992 (4R,7S,10R)-7-Benzyl-10-{[(2S,3S)-3-(4-hydroxy-phenyl)-pyrrolidine-2-carbonyl]-amino}-3,3-dimethyl-6,9-dioxo-1,2-dithia-5,8-diaza-cycloundecane-4-carboxylic acid 228038 Dimethyl-[2-(6-pyridin-3-yl-indol-1-yl)-ethyl]-amine 228056 (4R,7S,10R)-10-[(S)-2-Amino-3-(4-hydroxy-phenyl)-2-methyl-propionylamino]-7-benzyl-3,3-dimethyl-6,9-dioxo-1,2-dithia-5,8-diaza-cycloundecane-4-carboxylic acid 228057 (4R,7S,10R)-10-[(R)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7-benzyl-3,3-dimethyl-6,9-dioxo-1,2-dithia-5,8-diaza-cycloundecane-4-carboxylic acid 228082 (4R,7S,10R)-10-[((R)-2-Amino-5-hydroxy-indane-2-carbonyl)-amino]-7-benzyl-3,3-dimethyl-6,9-dioxo-1,2-dithia-5,8-diaza-cycloundecane-4-carboxylic acid 228083 (4R,7S,10R)-7-Benzyl-10-[((S)-7-hydroxy-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl)-amino]-3,3-dimethyl-6,9-dioxo-1,2-dithia-5,8-diaza-cycloundecane-4-carboxylic acid 228436 But-2-enedioic acid [4-(3-bromo-phenylamino)-pyrido[3,4-d]pyrimidin-6-yl]-amide (3-imidazol-1-yl-propyl)-amide 228463 N1-(4-(3-chloro-4-fluorophenylamino)pyrido[3,4-d]pyrimidin-6-yl)-N4-(3-morpholinopropyl)fumaramide 228506 (2,3,5,6,7,8-Hexahydro-naphtho[2,3-b]furan-7-yl)-dipropyl-amine 228523 But-2-enedioic acid [4-(3-bromo-phenylamino)-pyrido[3,4-d]pyrimidin-6-yl]-amide (3-diethylamino-propyl)-amide 228550 But-2-enedioic acid [4-(3-bromo-phenylamino)-pyrido[3,4-d]pyrimidin-6-yl]-amide (3-morpholin-4-yl-propyl)-amide 228551 But-2-enedioic acid [4-(3-bromo-phenylamino)-pyrido[3,4-d]pyrimidin-6-yl]-amide (3-dimethylamino-propyl)-amide 228575 Dimethyl-[2-(6-thiophen-3-yl-indol-1-yl)-ethyl]-amine 228576 Dimethyl-[2-(6-naphthalen-2-yl-indol-1-yl)-ethyl]-amine 228585 {2-[6-(3,6-Dihydro-2H-pyran-4-yl)-indol-1-yl]-ethyl}-dimethyl-amine 228587 (S)-1-{2-[4-(4-Carbamoyl-phenyl)-piperazin-1-yl]-ethyl}-isochroman-6-carboxylic acid methylamide 228593 8-[2-(3-Bromo-phenyl)-vinyl]-3,7-dimethyl-1-prop-2-ynyl-3,7-dihydro-purine-2,6-dione (BS-DMPX) 228603 4-[1-(2-Dimethylamino-ethyl)-1H-indol-6-yl]-tetrahydro-pyran-4-ol 228628 Dimethyl-{2-[6-(tetrahydro-pyran-4-yl)-indol-1-yl]-ethyl}-amine 228666 But-2-enedioic acid [4-(3-bromo-phenylamino)-quinazolin-6-yl]-amide (3-dimethylamino-propyl)-amide 228698 3-[4-(3-Bromo-phenylamino)-quinazolin-6-ylcarbamoyl]-acrylic acid 3-dimethylamino-propyl ester 228730 N-[4-(3-Bromo-phenylamino)-pyrido[3,4-d]pyrimidin-6-yl]-N-methyl-acrylamide 228759 4-[1-(2-Dimethylamino-ethyl)-1H-indol-6-yl]-tetrahydro-thiopyran-4-ol 228760 Dimethyl-{2-[6-(tetrahydro-thiopyran-4-yl)-indol-1-yl]-ethyl}-amine 228888 SID26753669 229058 4-(diethylamino)but-2-ynyl 2-cyclohexyl-2-hydroxy-2-phenylacetate 229082 Butyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amine 229083 Butyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-amine 229084 Benzyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-amine 229224 ((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amine 229225 ((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-isopropyl-amine 229226 (R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-ylamine 229255 {2-[6-(3,6-Dihydro-2H-thiopyran-4-yl)-indol-1-yl]-ethyl}-dimethyl-amine 229438 ((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-isopropyl-propyl-amine 229525 8-{4-[((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amino]-butyl}-8-aza-spiro[4.5]decane-7,9-dione 229580 N-[3-((3R,4R)-3,4-Dimethyl-1-phenethyl-piperidin-4-yl)-phenyl]-acetamide 229611 3-((3R,4R)-3,4-Dimethyl-1-phenethyl-piperidin-4-yl)-N-methyl-benzamide 229878 3-[(3R,4R)-3,4-Dimethyl-1-(3-phenyl-butyl)-piperidin-4-yl]-benzamide 229887 3-[(3R,4R)-3,4-Dimethyl-1-(3,5,5-trimethyl-hexyl)-piperidin-4-yl]-benzamide 229895 (4R,5S)-4-Phenyl-pyrrolidine-3-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 229911 3-[(3R,4R)-3,4-Dimethyl-1-(3-phenyl-propyl)-piperidin-4-yl]-benzamide 229913 3-[(3R,4R)-3,4-Dimethyl-1-(4-methylsulfanyl-benzyl)-piperidin-4-yl]-benzamide 229929 8-[4-((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-ylamino)-butyl]-8-aza-spiro[4.5]decane-7,9-dione 230003 3-((3R,4R)-3,4-Dimethyl-1-quinolin-2-ylmethyl-piperidin-4-yl)-benzamide 230110 [3-((3R,4R)-3,4-Dimethyl-1-phenethyl-piperidin-4-yl)-phenyl]-methanol 230213 3-((3R,4R)-3,4-Dimethyl-1-phenethyl-piperidin-4-yl)-benzamide 230564 8-[2-(3-Hydroxy-phenyl)-vinyl]-3,7-dimethyl-1-prop-2-ynyl-3,7-dihydro-purine-2,6-dione 230600 3-(3-Hydroxy-propyl)-8-[2-(3-methoxy-phenyl)-vinyl]-7-methyl-1-prop-2-ynyl-3,7-dihydro-purine-2,6-dione (MSX-2) 230679 (2R,3R,4S,5S)-3,4-dihydroxy-2-[6-(3-iodo-benzylamino)-purin-9-yl]-1-oxa-7-aza-spiro[4.4]nonan-6-one 230749 1-(3-chlorophenyl)-3-(8-ethyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 230755 2-(furan-2-yl)-8-(3-phenylpropyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine 230757 1-(3-chlorophenyl)-3-(2-(furan-2-yl)-8-propyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 230758 3-(2-Hydroxy-ethyl)-8-[2-(3-methoxy-phenyl)-vinyl]-7-methyl-1-prop-2-ynyl-3,7-dihydro-purine-2,6-dione 230786 8-[2-(3-Methoxy-phenyl)-vinyl]-3,7-dimethyl-1-prop-2-ynyl-3,7-dihydro-purine-2,6-dione (MS-DMPX) 230851 R(-)-N6-(2-Phenylisopropyl)adenosine 230877 1-(3-chlorophenyl)-3-(2-(furan-2-yl)-8-phenethyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 230878 2-(furan-2-yl)-8-propyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine 230889 4-[2-Chloro-6-(3-iodo-benzylamino)-purin-9-yl]-3,6-dioxa-bicyclo[3.1.0]hexane-2-carboxylic acid methylamide 231055 (E)-3-{(S)-2-Hydroxymethyl-4-[(Z)-nonadec-10-en-(Z)-ylidene]-5-oxo-tetrahydro-furan-2-yl}-acrylic acid methyl ester 231116 8-[2-(3-Bromo-phenyl)-vinyl]-3-(2-hydroxy-ethyl)-7-methyl-1-prop-2-ynyl-3,7-dihydro-purine-2,6-dione 231117 8-[2-(3-Amino-phenyl)-vinyl]-3,7-dimethyl-1-prop-2-ynyl-3,7-dihydro-purine-2,6-dione 231125 4-[2-Chloro-6-(3-iodo-benzylamino)-purin-9-yl]-1-hydroxymethyl-bicyclo[3.1.0]hexane-2,3-diol 231153 Phosphoric acid mono-(3-{8-[2-(3-methoxy-phenyl)-vinyl]-7-methyl-2,6-dioxo-1-prop-2-ynyl-1,2,6,7-tetrahydro-purin-3-yl}-propyl) esterdi sodium 231154 8-[2-(3-Bromo-phenyl)-vinyl]-3-(3-hydroxy-propyl)-7-methyl-1-prop-2-ynyl-3,7-dihydro-purine-2,6-dione 231184 1-(2-(furan-2-yl)-8-phenethyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-methoxyphenyl)urea 231245 8-ethyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine 231248 1-(3-chlorophenyl)-3-(2-(furan-2-yl)-8-(3-phenylpropyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 231250 1-(2-(furan-2-yl)-8-(3-phenylpropyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-methoxyphenyl)urea 231252 3-((S)-2-Hydroxymethyl-5-oxo-tetrahydro-furan-2-yl)-propionic acid tetradecyl ester 231299 (S)-5-Hydroxymethyl-3-[(Z)-octadec-9-en-(E)-ylidene]-5-[2-oxo-dihydro-furan-(3Z)-ylidenemethyl]-dihydro-furan-2-one 231321 (S)-3-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1H-indol-3-yl)-2-methyl-propionylamino]-4-phenyl-butyric acid 231382 (S)-5-Hydroxymethyl-3-[(Z)-octadec-9-en-(Z)-ylidene]-5-[2-oxo-dihydro-furan-(3E)-ylidenemethyl]-dihydro-furan-2-one 231388 7-Ethyl-9-(3-nitro-phenyl)-6,7,8,9-tetrahydro-5H-10-thia-7-aza-benzo[a]azulene 231394 3-(2-Hydroxymethyl-5-oxo-tetrahydro-furan-2-yl)-propionic acid tetradecyl ester 231404 Acetic acid (R)-2-hydroxymethyl-4-[(Z)-nonadec-10-en-(E)-ylidene]-5-oxo-tetrahydro-furan-2-ylmethyl ester 231405 (S)-5-Hydroxymethyl-3-[(Z)-octadec-9-en-(E)-ylidene]-5-[2-oxo-dihydro-furan-(3E)-ylidenemethyl]-dihydro-furan-2-one 231510 Acetic acid (R)-2-hydroxymethyl-4-[(Z)-nonadec-10-en-(Z)-ylidene]-5-oxo-tetrahydro-furan-2-ylmethyl ester 231543 (E)-3-((R)-2-Hydroxymethyl-5-oxo-tetrahydro-furan-2-yl)-acrylic acid tetradecyl ester 231633 (R)-3-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1H-indol-3-yl)-2-methyl-propionylamino]-4-phenyl-butyric acid 231653 (S)-5-Hydroxymethyl-3-[(Z)-octadec-9-en-(Z)-ylidene]-5-[2-oxo-dihydro-furan-(3Z)-ylidenemethyl]-dihydro-furan-2-one 231654 3-((R)-2-Hydroxymethyl-5-oxo-tetrahydro-furan-2-yl)-propionic acid tetradecyl ester 231655 4-(2,5-Dihydroxy-benzylamino)-N-(3-phenyl-propyl)-benzamide 231656 4-(2,5-dihydroxybenzylamino)-N-phenethylbenzamide 231729 9-(3-Bromo-phenyl)-7-ethyl-6,7,8,9-tetrahydro-5H-10-thia-7-aza-benzo[a]azulene 231898 N-Benzyl-5-(2,5-dihydroxy-benzylamino)-2-hydroxy-benzamide 231899 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-N-[2-(4-methoxy-phenyl)-ethyl]-benzamide 231942 7-Ethyl-9-phenyl-6,7,8,9-tetrahydro-5H-10-thia-7-aza-benzo[a]azulene 231943 7,8-Dimethoxy-3-methyl-1-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine 231966 (E)-3-((S)-2-Hydroxymethyl-5-oxo-tetrahydro-furan-2-yl)-acrylic acid tetradecyl ester 231967 (E)-3-{(S)-2-Hydroxymethyl-4-[(Z)-nonadec-10-en-(E)-ylidene]-5-oxo-tetrahydro-furan-2-yl}-acrylic acid methyl ester 231971 9-(3,4-Dichloro-phenyl)-7-ethyl-6,7,8,9-tetrahydro-5H-10-thia-7-aza-benzo[a]azulene 232013 (4-Methoxy-phenyl)-((R)-5-methyl-3-morpholin-4-ylmethyl-2,3-dihydro-[1,4]oxazino[2,3,4-hi]indol-6-yl)-methanone 232063 5-(2,5-dihydroxybenzylamino)-2-hydroxy-N-(2-morpholinoethyl)benzamide 232239 (5Z,8Z,11Z,14Z)-1-(3-Hydroxy-piperidin-1-yl)-icosa-5,8,11,14-tetraen-1-one 232240 (5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenethioic acid ((R)-2-hydroxy-1-methyl-ethyl)-amide 232279 (5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid (2-hydroxy-ethyl)-methyl-amide 232280 (5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid (2-hydroxy-butyl)-amide 232304 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-N-[2-(4-hydroxy-phenyl)-ethyl]-benzamide 232319 (5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid (2-hydroxy-1-hydroxymethyl-ethyl)-amide 232330 N-Benzyl-4-(2,5-dihydroxy-benzylamino)-benzamide 232332 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-N-(1,2,3,4-tetrahydro-naphthalen-2-yl)-benzamide 232382 5-(2,5-Dihydroxy-benzylamino)-N-dodecyl-2-hydroxy-benzamide 232393 (2-Fluoro-phenyl)-[2-methyl-1-((S)-1-methyl-2-morpholin-4-yl-ethyl)-1H-indol-3-yl]-methanone 232408 5-(2,5-dihydroxybenzylamino)-2-hydroxy-N-(3-phenylpropyl)benzamide 232600 (5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid (3-hydroxy-phenyl)-amide 232651 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-N-phenethyl-benzamide 232652 N-[2-(4-Bromo-phenyl)-ethyl]-5-(2,5-dihydroxy-benzylamino)-2-hydroxy-benzamide 232653 N-[2-(4-Chloro-phenyl)-ethyl]-5-(2,5-dihydroxy-benzylamino)-2-hydroxy-benzamide 232743 N-(4-hydroxybenzyl)icosa-5,8,11,14-tetraenamide 232788 (5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid (2-hydroxy-phenyl)-amide 232931 (5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenethioic acid (2-hydroxy-ethyl)-amide 233129 N-hydroxy-1-(4-methoxyphenylsulfonyl)piperidine-2-carboxamide 233922 (R)-N-((R)-1-(4-((1H-tetrazol-5-yl)methyl)-4-cyclohexylpiperidin-1-yl)-3-(4-chlorophenyl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 234033 2-(1-(((1R)-3-(2-(2-hydroxypropan-2-yl)phenyl)-1-(3-((E)-2-(8-methyl-5,6,7,8-tetrahydroquinolin-2-yl)vinyl)phenyl)propylthio)methyl)cyclopropyl)acetic acid 234098 2-[4-(2-Chloro-phenyl)-piperazin-1-ylmethyl]-1H-indole-6-carbonitrile 234111 (R)-2-(1-((3-(2-(2-hydroxypropan-2-yl)phenyl)-1-(3-(2-(5,6,7,8-tetrahydroquinolin-2-yl)vinyl)phenyl)propylthio)methyl)cyclopropyl)acetic acid 234112 [1-((R)-3-[2-(1-Hydroxy-1-methyl-ethyl)-phenyl]-1-{3-[(E)-2-(6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridin-2-yl)-vinyl]-phenyl}-propylsulfanylmethyl)-cyclopropyl]-acetic acid 234131 3-(4-Phenyl-piperazin-1-ylmethyl)-1H-indole-5-carbonitrile 234135 2-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-1H-indole-5-carbonitrile 234157 N-(5-(4-(2-methoxyphenyl)piperazin-1-yl)pentyl)H-pyrazolo[1,5-a]pyridine-3-carboxamide 234162 3-[4-(3,4-Dichloro-phenyl)-piperazin-1-ylmethyl]-1H-indole-5-carbonitrile 234165 2-[4-(3,4-Dichloro-phenyl)-piperazin-1-ylmethyl]-1H-indole-5-carbonitrile 234167 2-[4-(3,4-Dichloro-phenyl)-piperazin-1-ylmethyl]-1H-indole-6-carbonitrile 234168 2-[4-(2-Chloro-phenyl)-piperazin-1-ylmethyl]-1H-indole-5-carbonitrile 234169 2-((4-phenylpiperazin-1-yl)methyl)-1H-indole-5-carbonitrile 234175 (1-{(R)-1-{3-[(E)-2-(7,7-Dimethyl-6,7-dihydro-5H-[1]pyrindin-2-yl)-vinyl]-phenyl}-3-[2-(1-hydroxy-1-methyl-ethyl)-phenyl]-propylsulfanylmethyl}-cyclopropyl)-acetic acid 234180 (R)-2-(1-((1-(3-(2-(5,7-dihydrothieno[3,4-b]pyridin-2-yl)vinyl)phenyl)-3-(2-(2-hydroxypropan-2-yl)phenyl)propylthio)methyl)cyclopropyl)acetic acid 234181 (1-{(R)-1-{3-[(E)-2-(2,3-Dihydro-thieno[3,2-b]pyridin-5-yl)-vinyl]-phenyl}-3-[2-(1-hydroxy-1-methyl-ethyl)-phenyl]-propylsulfanylmethyl}-cyclopropyl)-acetic acid 234194 2-(4-Phenyl-piperazin-1-ylmethyl)-1H-indole-6-carbonitrile 234195 2-((4-(4-fluorophenyl)piperazin-1-yl)methyl)-1H-indole-5-carbonitrile 234216 (R)-2-(1-((1-(3-(2-(6,7-dihydro-5H-cyclopenta[b]pyridin-2-yl)vinyl)phenyl)-3-(2-(2-hydroxypropan-2-yl)phenyl)propylthio)methyl)cyclopropyl)acetic acid 234235 3-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-1H-indole-5-carbonitrile 234236 3-[4-(4-Fluoro-phenyl)-piperazin-1-ylmethyl]-1H-indole-5-carbonitrile 234244 (R)-2-(1-((1-(3-(2-(6,6-dimethyl-6,7-dihydro-5H-cyclopenta[b]pyridin-2-yl)vinyl)phenyl)-3-(2-(2-hydroxypropan-2-yl)phenyl)propylthio)methyl)cyclopropyl)acetic acid 234245 [1-((R)-3-[2-(1-Hydroxy-1-methyl-ethyl)-phenyl]-1-{3-[(E)-2-(7-methyl-6,7-dihydro-5H-[1]pyrindin-2-yl)-vinyl]-phenyl}-propylsulfanylmethyl)-cyclopropyl]-acetic acid 234274 3-[4-(2-Chloro-phenyl)-piperazin-1-ylmethyl]-1H-indole-5-carbonitrile 234375 N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)H-pyrazolo[1,5-a]pyridine-2-carboxamide 234449 N-(5-(4-(2-methoxyphenyl)piperazin-1-yl)pentyl)H-pyrazolo[1,5-a]pyridine-2-carboxamide 234531 (R)-N-((R)-3-(4-chlorophenyl)-1-(4-cyclohexyl-4-((2-methyl-2H-tetrazol-5-yl)methyl)piperidin-1-yl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 234538 N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)H-pyrazolo[1,5-a]pyridine-2-carboxamide 234539 N-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)H-pyrazolo[1,5-a]pyridine-2-carboxamide 234543 N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)H-pyrazolo[1,5-a]pyridine-3-carboxamide 234557 (1-{(R)-1-{3-[(E)-2-(8,8-Dimethyl-5,6,7,8-tetrahydro-quinolin-2-yl)-vinyl]-phenyl}-3-[2-(1-hydroxy-1-methyl-ethyl)-phenyl]-propylsulfanylmethyl}-cyclopropyl)-acetic acid 234591 (1-{(R)-1-{3-[(E)-2-(7,7-Dimethyl-5,6,7,8-tetrahydro-quinolin-2-yl)-vinyl]-phenyl}-3-[2-(1-hydroxy-1-methyl-ethyl)-phenyl]-propylsulfanylmethyl}-cyclopropyl)-acetic acid 234743 5-(((2S,3S)-2-(3,5-bis(trifluoromethyl)benzyloxy)-3-(4-fluorophenyl)morpholino)methyl)-2H-1,2,4-triazol-3(4H)-one 234848 N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)H-pyrazolo[1,5-a]pyridine-4-carboxamide 234862 etorphine 234867 N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)benzofuran-2-carboxamide 234869 N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)H-pyrazolo[1,5-a]pyridine-7-carboxamide 234931 N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)H-pyrazolo[1,5-a]pyridine-5-carboxamide 234947 (3R)-N-[(2R)-3-(4-chlorophenyl)-1-{4-cyclohexyl-4-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)methyl]piperidin-1-yl}-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 234948 (2S)-2-amino-3-(1H-imidazol-4-yl)-N-[(2R)-1-{1-methanesulfonyl-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}-3-(naphthalen-2-yl)-1-oxopropan-2-yl]propanamide 235232 4-[2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-3-(4-nitro-phenyl)-propionylamino]-4-{1-[1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propylcarbamoyl}-butyric acid 235233 3-[2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-3-(4-nitro-phenyl)-propionylamino]-N-{1-[1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-succinamic acid 235381 5-{(2R,3S)-3-Phenyl-2-[(R)-1-(3-trifluoromethyl-phenyl)-ethoxy]-morpholin-4-ylmethyl}-2,4-dihydro-[1,2,4]triazol-3-one 235396 N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]benzo[b]thiophene-2-carboxamide 235397 5-{(2R,3S)-2-[(S)-1-(3,5-Bis-trifluoromethyl-phenyl)-ethoxy]-3-phenyl-morpholin-4-ylmethyl}-2,4-dihydro-[1,2,4]triazol-3-one 235412 2-(7-Cyclopentyl-5,6-dimethyl-2-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)-butan-1-ol 235449 3-[2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-3-(4-iodo-phenyl)-propionylamino]-N-{1-[1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-succinamic acid 235491 (R)-1-(5-oxo-2,3,5,9b-tetrahydro-1H-pyrrolo[2,1-a]isoindol-9-yl)-3-(pyridin-2-yl)urea 235758 1-(5-(((S)-5-chloro-2,3-dihydro-1H-inden-2-ylamino)methyl)-1H-pyrazol-3-yl)-3-((S)-5-oxo-2,3,5,9b-tetrahydro-1H-pyrrolo[2,1-a]isoindol-9-yl)urea 235796 3-[2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-3-(4-chloro-phenyl)-propionylamino]-N-{1-[1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-succinamic acid 235896 (4R)-2-(3-heptylphenyl)thiazolidine-4-carboxylic acid 235917 5-(((2R,3S)-2-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-3-phenylmorpholino)methyl)-2H-1,2,4-triazol-3(4H)-one 235945 5-{(2R,3S)-2-[(R)-1-(3-Fluoro-5-trifluoromethyl-phenyl)-ethoxy]-3-phenyl-morpholin-4-ylmethyl}-2,4-dihydro-[1,2,4]triazol-3-one 235949 2,4-Dimethyl-6-phenyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid 5-benzyl ester 3-ethyl ester 235952 2-Methyl-6-phenyl-4-((E)-styryl)-1,4-dihydro-pyridine-3,5-dicarboxylic acid 3-benzyl ester 5-ethyl ester 236019 SID26752883 236071 2-[2-(4-Chloro-phenyl)-5,6-dimethyl-7-(1-phenyl-ethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino]-butan-1-ol 236084 3-[2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-3-(4-fluoro-phenyl)-propionylamino]-N-{1-[1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-succinamic acid 236085 3-[2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-3-(4-bromo-phenyl)-propionylamino]-N-{1-[1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-succinamic acid 236126 2-Furan-2-yl-5,6-dimethyl-7-(1-phenyl-ethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine 236157 5,6-Dimethyl-7-(1-phenyl-ethyl)-2-pyridin-4-yl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine 236168 3-[2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-3-(4-amino-phenyl)-propionylamino]-N-{1-[1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-succinamic acid 236169 4-[2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-3-(4-amino-phenyl)-propionylamino]-4-{1-[1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propylcarbamoyl}-butyric acid 236244 1,2,4-triazolo[1,5-a]pyrimidine 236286 5,6-Dimethyl-2-(1-oxy-pyridin-4-yl)-7-(1-phenyl-ethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine 236287 5,6-Dimethyl-7-(1-phenyl-ethyl)-2-pyrazin-2-yl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine 236314 5,6-Dimethyl-7-(1-phenyl-ethyl)-2-thiophen-2-yl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine 236372 4-(2,2-Diphenyl-vinyl)-2-methyl-6-phenyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid diethyl ester 236388 (4R)-2-(4-heptylphenyl)thiazolidine-4-carboxylic acid 236576 2-Methyl-6-(4-nitro-phenyl)-4-((E)-styryl)-1,4-dihydro-pyridine-3,5-dicarboxylic acid diethyl ester 236761 SID17412281 236789 2-Methyl-4-((E)-styryl)-6-p-tolyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid diethyl ester 236961 3-Amino-benzo[b]thiophene-2-carboxylic acid [4-(4-benzo[d]isothiazol-3-yl-piperazin-1-yl)-butyl]-amide 236962 1H-Indazole-3-carboxylic acid [4-(4-benzo[d]isothiazol-3-yl-piperazin-1-yl)-butyl]-amide 236964 2,3-Dihydro-1H-indole-7-carboxylic acid [4-(4-benzo[d]isothiazol-3-yl-piperazin-1-yl)-butyl]-amide 236988 3-Amino-thiophene-2-carboxylic acid [4-(4-benzo[d]isothiazol-3-yl-piperazin-1-yl)-butyl]-amide 237007 SID26751791 237035 2-Methyl-6-phenyl-4-((E)-styryl)-1,4-dihydro-pyridine-3,5-dicarboxylic acid 5-benzyl ester 3-ethyl ester 237139 degarelix 237192 6-(4-Pyrimidin-2-yl-piperazin-1-ylmethyl)-6,7-dihydro-5H-benzofuran-4-one 237194 6-{4-[5-(4-Fluoro-phenyl)-5-oxo-pentyl]-piperazin-1-ylmethyl}-6,7-dihydro-5H-benzofuran-4-one 237284 6-(4-Pyridin-2-yl-piperazin-1-ylmethyl)-6,7-dihydro-5H-benzofuran-4-one 237296 2-Amino-N-[4-(4-benzo[d]isothiazol-3-yl-piperazin-1-yl)-butyl]-nicotinamide 237297 1H-Indole-7-carboxylic acid [4-(4-benzo[d]isothiazol-3-yl-piperazin-1-yl)-butyl]-amide 237299 acyline 237300 4-Amino-thiophene-3-carboxylic acid [4-(4-benzo[d]isothiazol-3-yl-piperazin-1-yl)-butyl]-amide 237335 1,2,3,4-Tetrahydro-quinoline-8-carboxylic acid [4-(4-benzo[d]isothiazol-3-yl-piperazin-1-yl)-butyl]-amide 237463 N-[4-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-butyl]-nicotinamide 237472 3H-Benzoimidazole-4-carboxylic acid [4-(4-benzo[d]isothiazol-3-yl-piperazin-1-yl)-butyl]-amide 237550 Pyridine-2-carboxylic acid [4-(4-benzo[d]isothiazol-3-yl-piperazin-1-yl)-butyl]-amide 237594 6-{4-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-piperazin-1-ylmethyl}-6,7-dihydro-5H-benzofuran-4-one 237605 2-Amino-thiophene-3-carboxylic acid [4-(4-benzo[d]isothiazol-3-yl-piperazin-1-yl)-butyl]-amide 237633 4-Amino-N-[4-(4-benzo[d]isothiazol-3-yl-piperazin-1-yl)-butyl]-nicotinamide 237659 N-[4-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-butyl]-isonicotinamide 237719 3-Amino-N-[4-(4-benzo[d]isothiazol-3-yl-piperazin-1-yl)-butyl]-isonicotinamide 237741 (S)-1-{4-[3-(4-Fluoro-phenyl)-1H-pyrrolo[3,2-b]pyridin-2-yl]-pyridin-2-ylamino}-propan-2-ol 237750 Quinoline-8-carboxylic acid [4-(4-benzo[d]isothiazol-3-yl-piperazin-1-yl)-butyl]-amide 237751 1H-Indole-3-carboxylic acid [4-(4-benzo[d]isothiazol-3-yl-piperazin-1-yl)-butyl]-amide 237774 6-((4-(4-fluorobenzoyl)piperidin-1-yl)methyl)-6,7-dihydrobenzofuran-4(5H)-one 237775 QF-1004B 237776 6-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-6,7-dihydro-5H-benzofuran-4-one 238115 3-Amino-pyridine-2-carboxylic acid [4-(4-benzo[d]isothiazol-3-yl-piperazin-1-yl)-butyl]-amide 238160 1-(3-chlorophenyl)-3-(2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 238192 (4S,7S,13S)-13-[(S)-2-amino-3-(4-hydroxy-phenyl)-propionylamino]-7-(4-chloro-benzyl)-3,3,14,14-tetramethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradecane-4-carboxylic acid 238193 3-[(4-Benzyl-piperazin-1-yl)-(4-tert-butyl-phenyl)-methyl]-phenol 238225 Sodium salt 4'-(2-butyl-4-chloro-5-ethoxycarbonyl-6-phenyl-6H-pyrimidin-1-ylmethyl)-biphenyl-2-carboxylate 238233 1-{2-Furan-2-yl-8-[2-(2,4,5-tribromo-phenyl)-ethyl]-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl}-3-(4-methoxy-phenyl)-urea 238361 1-(3-chlorophenyl)-3-(2-(furan-2-yl)-8-(3-methylbut-2-enyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 238388 1-(2-(furan-2-yl)-8-(3-methylbut-2-enyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-methoxyphenyl)urea 238512 1-(3-chlorophenyl)-3-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 238513 2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine 238574 2-Butyl-4-chloro-6-methyl-1-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-1,6-dihydro-pyrimidine-5-carboxylic acid 238607 Sodium salt 4'-(2-butyl-5-ethoxycarbonyl-4-methyl-6-oxo-6H-pyrimidin-1-ylmethyl)-biphenyl-2-carboxylate 238608 Sodium salt 4'-(2-butyl-5-ethoxycarbonyl-6-oxo-6H-pyrimidin-1-ylmethyl)-biphenyl-2-carboxylate 238609 2-Butyl-6-chloro-4,4-dimethyl-1-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-1,4-dihydro-pyrimidine-5-carboxylic acid ethyl ester 238644 2-Butyl-4-chloro-6-methyl-1-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-1,6-dihydro-pyrimidine-5-carboxylic acid ethyl ester; potassium 238646 Sodium salt 4'-(2-butyl-5-ethoxycarbonyl-6-oxo-4-phenyl-6H-pyrimidin-1-ylmethyl)-biphenyl-2-carboxylate 238667 Sodium salt 4'-(2-butyl-6-chloro-5-ethoxycarbonyl-4,4-dimethyl-4H-pyrimidin-1-ylmethyl)-biphenyl-2-carboxylate 238673 2-Butyl-1-(2'-carboxy-biphenyl-4-ylmethyl)-4-(4-chloro-phenyl)-6-methyl-1,6-dihydro-pyrimidine-5-carboxylic acid ethyl ester 238684 1-(9-Chloro-2-furan-2-yl-[1,2,4]triazolo[1,5-c]quinazolin-5-yl)-3-(3-chloro-phenyl)-urea 238713 1-(9-Chloro-2-furan-2-yl-[1,2,4]triazolo[1,5-c]quinazolin-5-yl)-3-(4-methoxy-phenyl)-urea 238731 N-[(1-butyl-4-piperidinyl)methyl]-3,4-dihydro-2H-[1,3]-oxazino[3,2-a]-indole-10-carboxamide 238844 2-Furan-2-yl-8-[2-(2,4,5-tribromo-phenyl)-ethyl]-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 238878 1-(8-tert-butyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(3-chlorophenyl)urea 238903 1-(8-tert-butyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-methoxyphenyl)urea 238910 1-(3-{[5-Carbamoyl-6-(3,4-difluoro-phenyl)-4-ethyl-2-oxo-3,6-dihydro-2H-pyrimidine-1-carbonyl]-amino}-propyl)-4-phenyl-piperidine-4-carboxylic acid methyl ester 239022 2-Butyl-1-(2'-carboxy-biphenyl-4-ylmethyl)-4-chloro-6-methyl-1,6-dihydro-pyrimidine-5-carboxylic acid ethyl ester 239023 2-Butyl-1-(2'-carboxy-biphenyl-4-ylmethyl)-4,6-dimethyl-1,6-dihydro-pyrimidine-5-carboxylic acid ethyl ester 239059 2-Butyl-1-(2'-carboxy-biphenyl-4-ylmethyl)-6-methyl-4-phenyl-1,6-dihydro-pyrimidine-5-carboxylic acid ethyl ester 239090 1-(2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-methoxyphenyl)urea 239107 1-(3-Chloro-phenyl)-3-[2-furan-2-yl-8-(2-naphthalen-1-yl-ethyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl]-urea 239157 1-[2-Furan-2-yl-8-(2-naphthalen-1-yl-ethyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl]-3-(4-methoxy-phenyl)-urea 239174 8-tert-butyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine 239176 1-(8-butyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(3-chlorophenyl)urea 239341 2-Furan-2-yl-8-(2-naphthalen-1-yl-ethyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 239376 1-(3-Chloro-phenyl)-3-{2-furan-2-yl-8-[2-(2,4,5-tribromo-phenyl)-ethyl]-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl}-urea 239379 (S)-3-[((2S,5S,11bS)-2-Benzyloxycarbonylamino-3-oxo-2,3,5,6,11,11b-hexahydro-1H-indolizino[8,7-b]indole-5-carbonyl)-amino]-4-phenyl-butyric acid 2-trimethylsilanyl-ethyl ester 239413 (R)-3-[((2S,5S,11bS)-2-Benzyloxycarbonylamino-3-oxo-2,3,5,6,11,11b-hexahydro-1H-indolizino[8,7-b]indole-5-carbonyl)-amino]-4-phenyl-butyric acid 239504 (R)-3-[((2S,5S,11bR)-2-tert-Butoxycarbonylamino-3-oxo-2,3,5,6,11,11b-hexahydro-1H-indolizino[8,7-b]indole-5-carbonyl)-amino]-4-phenyl-butyric acid 239505 (R)-3-[((2S,5S,11bS)-2-Benzyloxycarbonylamino-3-oxo-2,3,5,6,11,11b-hexahydro-1H-indolizino[8,7-b]indole-5-carbonyl)-amino]-4-phenyl-butyric acid 2-trimethylsilanyl-ethyl ester 239506 (R)-3-[((2S,5S,11bR)-2-Benzyloxycarbonylamino-3-oxo-2,3,5,6,11,11b-hexahydro-1H-indolizino[8,7-b]indole-5-carbonyl)-amino]-4-phenyl-butyric acid 2-trimethylsilanyl-ethyl ester 239583 2-(furan-2-yl)-8-(3-methylbut-2-enyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine 239616 1-(3-chlorophenyl)-3-(2-(furan-2-yl)-8-isopentyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 239617 1-(2-(furan-2-yl)-8-isopentyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-methoxyphenyl)urea 239642 3,6-Dihydroxy-naphthalene-2-carboxylic acid (3-hydroxy-phenyl)-amide 239786 (S)-3-[((2S,5S,11bS)-2-Benzyloxycarbonylamino-3-oxo-2,3,5,6,11,11b-hexahydro-1H-indolizino[8,7-b]indole-5-carbonyl)-amino]-4-phenyl-butyric acid 239802 N-(1,3-Bis-cyclopropylmethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)-4-methoxy-benzenesulfonamide 239846 (R)-3-[(S)-2-(Adamantan-2-yloxycarbonylamino)-3-(1H-indol-3-yl)-2-methyl-propionylamino]-4-phenyl-butyric acid 239983 (S)-3-[(S)-2-(Adamantan-2-yloxycarbonylamino)-3-(1H-indol-3-yl)-2-methyl-propionylamino]-4-phenyl-butyric acid 239984 (S)-3-[((2S,5S,11bR)-2-Benzyloxycarbonylamino-3-oxo-2,3,5,6,11,11b-hexahydro-1H-indolizino[8,7-b]indole-5-carbonyl)-amino]-4-phenyl-butyric acid 2-trimethylsilanyl-ethyl ester 240163 3,5-Dihydroxy-naphthalene-2-carboxylic acid (3-hydroxy-phenyl)-amide 240294 N-[1,3-Bis-cyclopropylmethyl-7-(4-methoxy-benzyl)-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl]-4-methoxy-benzenesulfonamide 240306 8-Amino-7-(4-chloro-benzenesulfonyl)-1,3-bis-cyclopropylmethyl-3,7-dihydro-purine-2,6-dione 240310 8-Amino-1,3-bis-cyclopropylmethyl-7-propyl-3,7-dihydro-purine-2,6-dione 240311 8-Amino-1,3-bis-cyclopropylmethyl-3,7-dihydro-purine-2,6-dione 240312 8-Amino-1,3-bis-cyclopropylmethyl-7-isobutyl-3,7-dihydro-purine-2,6-dione 240315 8-Amino-1,3-bis-cyclopropylmethyl-7-(toluene-4-sulfonyl)-3,7-dihydro-purine-2,6-dione 240380 8-Amino-7-benzyl-1,3-bis-cyclopropylmethyl-3,7-dihydro-purine-2,6-dione 240416 1,3-Bis-cyclopropylmethyl-7-(4-methoxy-benzyl)-8-[1-methyl-pyrrolidin-(2Z)-ylideneamino]-3,7-dihydro-purine-2,6-dione 240884 5-Hydroxy-1H-indole-2-carboxylic acid 3-hydroxy-benzylamide 241031 8-Amino-1,3-bis-cyclopropylmethyl-7-methanesulfonyl-3,7-dihydro-purine-2,6-dione 241034 1,3-Bis(cyclopropylmethyl)-8-bis[(4-nitrophenylsulfonyl)amino]xanthine 241058 8-Amino-1,3-bis-cyclopropylmethyl-7-(propane-2-sulfonyl)-3,7-dihydro-purine-2,6-dione 241151 3-{[2-(2,6-Dimethoxy-phenoxy)-ethylamino]-methyl}-6,7-dimethoxy-1,2,3,4-tetrahydro-acridin-9-ol 241210 3-{[2-(2,6-Dimethoxy-phenoxy)-ethylamino]-methyl}-6,7-dimethoxy-1,2,3,4-tetrahydro-acridin-9-ylamine 241451 Furan-2-carboxylic acid (9-hydroxy-6,7-dimethoxy-1,2,3,4-tetrahydro-acridin-3-ylmethyl)-amide 241454 (2R,3R,4S,5R)-2-(6-Amino-purin-9-yl)-5-(1-methyl-1-phenyl-ethoxymethyl)-tetrahydro-furan-3,4-diol 241510 (2R,3R,4S,5S)-2-(6-(3-iodobenzylamino)-9H-purin-9-yl)-4-(aminomethyl)-5-(hydroxymethyl)-tetrahydrofuran-3-ol 241556 N-(9-Amino-6,7-dimethoxy-1,2,3,4-tetrahydro-acridin-3-ylmethyl)-4-trifluoromethyl-benzamide 241588 N-(9-Amino-6,7-dimethoxy-1,2,3,4-tetrahydro-acridin-3-ylmethyl)-2-trifluoromethyl-benzamide 241595 Furan-2-carboxylic acid (9-amino-6,7-dimethoxy-1,2,3,4-tetrahydro-acridin-3-ylmethyl)-amide 241630 Furan-2-carboxylic acid (9-amino-6,7-dimethoxy-2,3-dihydro-1H-cyclopenta[b]quinolin-2-ylmethyl)-amide 241981 (4-fluorophenyl)(piperidin-4-yl)methanone 242057 (1-Ethyl-piperidin-4-yl)-(4-fluoro-phenyl)-methanone 242058 (4-Fluoro-phenyl)-(1-methyl-piperidin-4-yl)-methanone 242292 1-Phenyl-4-(1-phenyl-1H-pyrrol-3-ylmethyl)-piperazine 242326 N-(2-Guanidino-ethyl)-N-(1-phenethyl-piperidin-4-yl)-propionamide 242526 1-Methyl-7,8-dihydro-1H-pyrrolo[2,3-e]indole-6-carboxylic acid pyridin-3-ylamide 242605 1-Phenyl-8-(1-phenyl-1H-pyrrol-3-ylmethyl)-1,3,8-triaza-spiro[4.5]decan-4-one 242609 3,5-Dihydro-2H-pyrrolo[2,3-f]indole-1-carboxylic acid pyridin-3-ylamide 242610 5-Ethyl-3,5-dihydro-2H-pyrrolo[2,3-f]indole-1-carboxylic acid pyridin-3-ylamide 242624 3-Methyl-5,6-dihydro-furo[3,2-f]indole-7-carboxylic acid pyridin-3-ylamide 242625 6,7-Dihydro-thieno[2,3-f]indole-5-carboxylic acid pyridin-3-ylamide 242626 5,7-Dimethyl-3,5-dihydro-2H-pyrrolo[2,3-f]indole-1-carboxylic acid phenylamide 242638 3-(2,3-Dimethyl-phenyl)-1-propyl-piperidine 242649 5-Benzyl-3,5-dihydro-2H-pyrrolo[2,3-f]indole-1-carboxylic acid pyridin-3-ylamide 242660 5-Methyl-3,5,6,7-tetrahydro-2H-pyrrolo[2,3-f]indole-1-carboxylic acid pyridin-3-ylamide 242675 3-(2,5-Dimethyl-phenyl)-1-propyl-piperidine 242694 4-(4-Chloro-phenyl)-1-(1-phenyl-1H-pyrrol-3-ylmethyl)-piperidin-4-ol 242709 3-(3,5-Dimethyl-phenyl)-piperidine 242710 3-(2,6-Dimethyl-phenyl)-1-propyl-piperidine 242716 SID26719802 242743 3-(3,5-Dimethyl-phenyl)-1-propyl-piperidine 242744 3-(2,3-Dimethyl-phenyl)-piperidine 242745 3-(3,4-Dimethyl-phenyl)-piperidine 242746 3-(2,4-Dimethyl-phenyl)-1-propyl-piperidine 242797 1-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-cyclohexyl}-1H-benzotriazole 242835 (3aS,7aR)-2-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-butyl]-hexahydro-isoindole-1,3-dione 242837 N-(3-Guanidino-propyl)-N-(1-phenethyl-piperidin-4-yl)-propionamide 242877 N-(6-Guanidino-hexyl)-N-(1-phenethyl-piperidin-4-yl)-propionamide 242880 N-(8-Guanidino-octyl)-N-(1-phenethyl-piperidin-4-yl)-propionamide 242898 H-Arg8-Arg9-Pro10-Tyr11-Ile12-Leu13 242918 N-(12-Guanidino-dodecyl)-N-(1-phenethyl-piperidin-4-yl)-propionamide 243070 6-Methyl-3,6-dihydro-2H-pyrrolo[2,3-e]indole-1-carboxylic acid pyridin-3-ylamide 243071 7-Methyl-3,7-dihydro-2H-pyrrolo[3,2-f]indole-1-carboxylic acid pyridin-3-ylamide 243095 4-Phenyl-1-(1-phenyl-1H-pyrrol-3-ylmethyl)-piperidine 243099 1-(1-Phenyl-1H-pyrrol-3-ylmethyl)-4-(3-trifluoromethyl-phenyl)-piperidin-4-ol 243129 4-Phenyl-1-(1-phenyl-1H-pyrrol-3-ylmethyl)-1,2,3,6-tetrahydro-pyridine 243130 1-(1-Phenyl-1H-pyrrol-3-ylmethyl)-4-pyridin-2-yl-piperazine 243171 H-Tyr-Val-Met-Gly-His-Phe-Arg-Trp-DAsp-Arg-Phe-Gly-OH 243190 (3aS,7aR)-2-{4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-cyclohexyl}-hexahydro-isoindole-1,3-dione 243253 (3aS,7aR)-2-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-cyclohexyl]-hexahydro-isoindole-1,3-dione 243279 (3aS,7aR)-2-{4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-butyl}-hexahydro-isoindole-1,3-dione 243313 2-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-cyclohexyl]-isoindole-1,3-dione 243344 2-{4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-cyclohexyl}-isoindole-1,3-dione 243485 SID26755703 243589 1-[1-(1-Phenyl-1H-pyrrol-3-ylmethyl)-piperidin-4-yl]-1,3-dihydro-benzoimidazol-2-one 243618 5,6-Dimethyl-3,5-dihydro-2H-pyrrolo[2,3-f]indole-1-carboxylic acid pyridin-3-ylamide 243619 5-Isopropyl-3,5-dihydro-2H-pyrrolo[2,3-f]indole-1-carboxylic acid pyridin-3-ylamide 243654 H-Tyr-Val-Met-Gly-His-Phe-Arg-Trp-Asp-Arg-Phe-Gly-NH2 243802 Phosphoric acid mono-[(1R,5S)-4-(2-bromo-6-methylamino-purin-9-yl)-1-phosphonooxymethyl-bicyclo[3.1.0]hex-2-yl] ester 243850 4-[3-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetrahydro-purin-3-yl)-propylcarbamoyl]-benzenesulfonyl fluoride 244014 4-[5-(4-Chloro-phenyl)-2H-pyrazol-3-yl]-1-phenethyl-piperidine 244026 Phosphoric acid mono-[(1R,5S)-4-(6-amino-2-iodo-purin-9-yl)-1-phosphonooxymethyl-bicyclo[3.1.0]hex-2-yl] ester 244114 Phosphoric acid mono-[(1R,5S)-4-(6-methylamino-2-methylselanyl-purin-9-yl)-1-phosphonooxymethyl-bicyclo[3.1.0]hex-2-yl] ester 244233 1-(2,4-difluorophenethyl)-4-(4-fluorophenylsulfonyl)piperidine 244505 (S)-3-[(R)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-3-phenyl-propionylamino]-N-{(S)-1-[(S)-(S)-1-((S)-1-carboxy-2-(S)-1H-indol-3-yl-ethylcarbamoyl)-2-methyl-butylcarbamoyl]-2-methyl-butyl}-succinamic acid 244612 (S)-4-((R)-2-Acetylamino-3-phenyl-propionylamino)-4-((S)-2-carboxy-1-{(S)-1-[(S)-(S)-1-((S)-1-carboxy-2-(S)-1H-indol-3-yl-ethylcarbamoyl)-2-methyl-butylcarbamoyl]-2-methyl-butylcarbamoyl}-ethylcarbamoyl)-butyric acid 244895 1-(2,4-difluorophenethyl)-4-(phenylsulfonyl)piperidine 245433 4-(3-(4-chlorophenyl)-3-hydroxypyrrolidin-1-yl)-1-(4-fluorophenyl)butan-1-one 245652 1-[(3R,4R)-1-cyclooctylmethyl-3-hydroxymethyl-4-piperidyl]-3-ethyl-1,3-dihydro-2H-benzimidazol-2-one 246543 N-((S)-1-Phenethyl-pyrrolidin-2-ylmethyl)-benzamide 246658 (Z)-3-(5-((6-(3-methoxyphenyl)-2-oxoindolin-3-ylidene)methyl)-2,4-dimethyl-1H-pyrrol-3-yl)propanoic acid 246664 2-Methoxy-5-methylsulfanyl-N-((S)-1-phenethyl-pyrrolidin-2-ylmethyl)-benzamide 246681 5-Methylsulfanyl-2,3-dihydro-benzofuran-7-carboxylic acid ((R)-1-phenethyl-pyrrolidin-2-ylmethyl)-amide 246695 5-Methoxy-2,3-dihydro-benzofuran-7-carboxylic acid ((S)-1-phenethyl-pyrrolidin-2-ylmethyl)-amide 247028 3-Methylsulfanyl-N-((R)-1-phenethyl-pyrrolidin-2-ylmethyl)-benzamide 247029 3-Methylsulfanyl-N-((S)-1-phenethyl-pyrrolidin-2-ylmethyl)-benzamide 247128 MCL-144 247227 (1R,3R,5S)-8-((S)-8-Ethoxy-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-3-phenyl-8-aza-bicyclo[3.2.1]octan-3-ol 247257 (1R,3R,5S)-8-((S)-8-Methoxy-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-3-(2-methoxy-phenyl)-8-aza-bicyclo[3.2.1]octan-3-ol 247286 (1R,3R,5S)-8-((S)-8-Methoxy-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-3-(3-trifluoromethyl-phenyl)-8-aza-bicyclo[3.2.1]octan-3-ol 247347 (1R,3R,5S)-3-Benzo[b]thiophen-3-yl-8-((S)-8-ethoxy-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-8-aza-bicyclo[3.2.1]octan-3-ol 247598 5-Hydroxy-2-(4-methoxy-phenyl)-7-methyl-chromen-4-one 247700 2-(3,4-Dihydroxy-phenyl)-3-hydroxy-7-methoxy-chromen-4-one 247782 8-Cyclopentyl-3-(3-fluoro-propyl)-1-propyl-3,7-dihydro-purine-2,6-dione 247785 (1R,3R,5S)-8-((S)-8-Ethoxy-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-3-naphthalen-2-yl-8-aza-bicyclo[3.2.1]octan-3-ol 247802 3,5,7-Trimethoxy-2-(4-methoxy-phenyl)-chromen-4-one 247803 Acetic acid 5,7-diacetoxy-4-oxo-2-phenyl-4H-chromen-3-yl ester 247805 SID26725076 247814 (1R,3R,5S)-8-((S)-8-Methoxy-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-3-naphthalen-2-yl-8-aza-bicyclo[3.2.1]octan-3-ol 247815 (1R,3R,5S)-8-((S)-8-Methoxy-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-3-phenyl-8-aza-bicyclo[3.2.1]octan-3-ol 247822 (1R,3R,5S)-3-Benzo[b]thiophen-3-yl-8-((S)-8-methoxy-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-8-aza-bicyclo[3.2.1]octan-3-ol 247826 5-Fluoro-1-[8-((S)-8-methoxy-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-8-aza-bicyclo[3.2.1]oct-2-en-3-yl]-1H-indole 247872 (1R,3R,5S)-8-((S)-8-Ethoxy-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-3-(3-trifluoromethyl-phenyl)-8-aza-bicyclo[3.2.1]octan-3-ol 247873 (1R,3R,5S)-8-((S)-8-Ethoxy-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-3-pyridin-2-yl-8-aza-bicyclo[3.2.1]octan-3-ol 247895 8-[8-((S)-8-Methoxy-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-8-aza-bicyclo[3.2.1]oct-2-en-3-yl]-quinoline 247909 (1R,3R,5S)-8-((S)-8-Methoxy-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-3-pyridin-2-yl-8-aza-bicyclo[3.2.1]octan-3-ol 247910 MCL-145 248112 8-((S)-8-Methoxy-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-3-naphthalen-1-yl-8-aza-bicyclo[3.2.1]oct-2-ene 248120 (S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-propionylamino]-N-((1S,2R)-1-{(1S,2R)-1-[(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 248363 (S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-3-carbamoyl-propionylamino]-N-((1S,2R)-1-{(1S,2R)-1-[(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 248364 (S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-3-(1H-indol-3-yl)-propionylamino]-N-((1S,2R)-1-{(1S,2R)-1-[(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 248575 3,5,7-Trimethoxy-2-(3,4,5-trimethoxy-phenyl)-chromen-4-one 248580 (S)-3-{2-[((R)-2-Acetylamino-3-phenyl-propionyl)-benzyl-amino]-acetylamino}-N-((1S,2R)-1-{(1S,2R)-1-[(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 248596 (S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-3-phenyl-propionylamino]-N-((1S,2R)-1-{(1S,2R)-1-[(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 248626 F-G-G-F-T-G-A-R-K-S-A-R-K-L-MeA-N-Q-CONH2 248627 F-G-G-F-T-G-Aib-R-K-S-Aib-R-K-L-A-N-Q-CONH2 248679 F-G-G-F-T-G-A-R-K-S-MeA-R-K-L-A-N-Q-CONH2 248749 (S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-4-phenyl-butyrylamino]-N-((1S,2R)-1-{(1S,2R)-1-[(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 248750 (R)-3-{[(R)-1-((R)-2-Acetylamino-3-phenyl-propionyl)-pyrrolidine-2-carbonyl]-amino}-N-((1R,2S)-1-{(1R,2S)-1-[(R)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 248767 (S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-5-amino-pentanoylamino]-N-((S)-1-{(1S,2R)-1-[(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-3-phenyl-propyl)-succinamic acid 248768 (S)-3-[(R)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-3-phenyl-propionylamino]-N-((1S,2R)-1-{(1S,2R)-1-[(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 248769 (S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-3-(4-hydroxy-phenyl)-propionylamino]-N-((1S,2R)-1-{(1S,2R)-1-[(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 248813 2'-Methyl-4'-(5-methyl-[1,3,4]oxadiazol-2-yl)-biphenyl-4-sulfonic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide 248847 (S)-3-{(S)-2-[(R)-2-Acetylamino-3-(1H-indol-3-yl)-propionylamino]-5-amino-pentanoylamino}-N-((1S,2R)-1-{(1S,2R)-1-[(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 248851 2'-Methyl-4'-(5-methyl-[1,2,4]oxadiazol-3-yl)-biphenyl-4-carboxylic acid [4-(2-fluoro-ethoxy)-3-(4-methyl-piperazin-1-yl)-phenyl]-amide 248873 2-Methyl-biphenyl-4,4'-dicarboxylic acid 4-amide 4'-{[4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide} 248903 4'-Carbamimidoyl-2'-methyl-biphenyl-4-carboxylic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide 248915 Methanesulfonic acid 4-{[2'-methyl-4'-(5-methyl-[1,3,4]oxadiazol-2-yl)-biphenyl-4-carbonyl]-amino}-2-(4-methyl-piperazin-1-yl)-phenyl ester 248971 (S)-3-{(S)-2-[(R)-2-Acetylamino-3-(4-hydroxy-phenyl)-propionylamino]-5-amino-pentanoylamino}-N-((1S,2R)-1-{(1S,2R)-1-[(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 249094 N-Cyclopropylmethyl-3-(3-hydroxy-phenyl)-2,2-dimethyl-3-methylamino-propionamide 249095 3-(3-Hydroxy-phenyl)-2,2-dimethyl-3-methylamino-N-naphthalen-1-ylmethyl-propionamide 249150 F-G-G-F-T-G-MeA-R-K-S-A-R-K-L-A-N-Q-COOH 249189 F-G-G-F-T-G-Aib-R-K-S-A-R-K-L-A-N-Q-COOH 249190 F-G-G-F-T-G-A-R-K-S-Aib-R-K-L-A-N-Q-COOH 249191 F-G-G-F-T-G-A-R-K-S-A-R-K-L-Aib-N-Q-COOH 249210 3-Cyano-2-ethyl-naphthalene-1-carboxylic acid ((S)-2-(3,4-dichloro-phenyl)-4-{4-[2-((S)-methanesulfinyl)-phenyl]-piperidin-1-yl}-butyl)-methyl-amide 249252 F-G-G-F-T-G-A-R-K-S-A-R-K-L-Aib-N-Q-CONH2 249253 6-(3-Guanidino-propyl)-3-(1H-indol-3-ylmethyl)-9-naphthalen-1-ylmethyl-2,5,8,11,14-pentaoxo-1,4,7,10,15pentaaza-cycloicosane-20-carboxylic acid amide 249459 F-G-G-F-T-G-A-R-K-S-MeA-R-K-L-A-N-Q-COOH 249460 F-G-G-F-T-G-Aib-R-K-S-A-R-K-L-A-N-Q-CONH2 249530 3-(Cyclopropylmethyl-methyl-amino)-3-(3-hydroxy-phenyl)-2,2-dimethyl-N-phenethyl-propionamide 249569 3-(Butyl-methyl-amino)-3-(3-hydroxy-phenyl)-2,2-dimethyl-N-phenethyl-propionamide 249637 F-G-G-F-T-G-A-R-K-S-Aib-R-K-L-A-N-Q-CONH2 249638 F-G-G-F-T-G-A-R-K-S-A-R-K-L-MeA-N-Q-COOH 249744 19-cyclopropylmethyl-6-nitro-11-oxa-8,19-diazahexacyclo[10.9.1.01,10.02,18.04,9.016,22]docosa-4(9),5,7,12,14,16(22)-hexaene-2,13-diol 249776 19-cyclopropylmethyl-6-benzylamino-11-oxa-8,19-diazahexacyclo[10.9.1.01,10.02,18.04,9.016,22]docosa-4(9),5,7,12,14,16(22)-hexaene-2,13-diol 249849 N-Benzyl-3-(3-hydroxy-phenyl)-2,2-dimethyl-3-methylamino-propionamide 249850 3-(3-Hydroxy-phenyl)-2,2-dimethyl-3-methylamino-N-phenethyl-propionamide 249919 2,2-Dimethyl-3-methylamino-N-phenethyl-3-phenyl-propionamide 249962 N-Cyclohexylmethyl-2,2-dimethyl-3-methylamino-3-phenyl-propionamide 249963 N-Benzyl-2,2-dimethyl-3-methylamino-3-phenyl-propionamide 250009 F-G-G-F-T-G-MeA-R-K-S-A-R-K-L-A-N-Q-CONH2 250045 19-cyclopropylmethyl-6-amino-11-oxa-8,19-diazahexacyclo[10.9.1.01,10.02,18.04,9.016,22]docosa-4(9),5,7,12,14,16(22)-hexaene-2,13-diol 250071 3-(3-Hydroxy-phenyl)-2,2-dimethyl-3-methylamino-N-(3-phenyl-propyl)-propionamide 250073 N-Cyclohexylmethyl-3-(3-hydroxy-phenyl)-2,2-dimethyl-3-methylamino-propionamide 250128 19-cyclopropylmethyl-6-phenyleaminomethyl-11-oxa-8,19-diazahexacyclo[10.9.1.01,10.02,18.04,9.016,22]docosa-4(9),5,7,12,14,16(22)-hexaene-2,13-diol 250135 ethyl 19-cyclopropylmethyl-2,13-dihydroxy-(10R)-11-oxa-8,19-diazahexacyclo[10.9.1.01,10.02,18.04,9.016,22]docosa-4(9),5,7,12,14,16(22)-hexaene-6-carboxylate 250151 19-cyclopropylmethyl-6-(1H-1-pyrrolyl)-11-oxa-8,19-diazahexacyclo[10.9.1.01,10.02,18.04,9.016,22]docosa-4(9),5,7,12,14,16(22)-hexaene-2,13-diol 250204 3,13-diazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,22}]tricosa-1(16),2(10),4(9),5,7,11(15),17,19,21-nonaen-12-one 250317 aldisin 250338 3-[((S)-4-Benzyl-2-methyl-piperazin-1-yl)-(4-tert-butyl-phenyl)-methyl]-phenol 250345 2-bromoaldisin 250364 4-(2-Amino-5-oxo-3,5-dihydro-imidazol-4-ylidene)-2-bromo-4,5,6,7-tetrahydro-1H-pyrrolo[2,3-c]azepin-8-one 250369 3-[(4-tert-Butyl-phenyl)-((S)-2,4-dibenzyl-piperazin-1-yl)-methyl]-phenol 250396 4-(2-Amino-3H-imidazol-4-yl)-2,3-dibromo-4,5,6,7-tetrahydro-1H-pyrrolo[2,3-c]azepin-8-one 250397 4,5-dibromopyrrole-2-carboxamide 250497 6-amino(imino)methylamino-19-cyclopropylmethyl-11-oxa-8,19-diazahexacyclo[10.9.1.01,10.02,18.04,9.016,22]docosa-4(9),5,7,12,14,16(22)-hexaene-2,13-diol; ditrifluoracetic acid 250516 19-cyclopropylmethyl-11-oxa-8,19-diazahexacyclo[10.9.1.01,10.02,18.04,9.016,22]docosa-4(9),5,7,12,14,16(22)-hexaene-2,13-diol 250528 19-cyclopropylmethyl-6-bromo-11-oxa-8,19-diazahexacyclo[10.9.1.01,10.02,18.04,9.016,22]docosa-4(9),5,7,12,14,16(22)-hexaene-2,13-diol 250529 19-cyclopropylmethyl-6-cyano-11-oxa-8,19-diazahexacyclo[10.9.1.01,10.02,18.04,9.016,22]docosa-4(9),5,7,12,14,16(22)-hexaene-2,13-diol 250597 3-[((R)-4-Benzyl-2-hydroxymethyl-piperazin-1-yl)-(4-tert-butyl-phenyl)-methyl]-phenol 250604 12-(3-hydroxypropyl)-9-isopropoxymethyl-6,7,12,13-tetrahydro-5H-indeno[2,1-a]pyrrolo[4,3-c]carbazol-5-one 250642 6,7,12,13-tetrahydro-5H-indeno[2,1-a]pyrrolo[4,3-c]carbazol-5-one 250749 SID29216291 250837 N-(4-chloro-2-fluorophenyl)-6,7-dimethoxyquinazolin-4-amine 250854 N-(4-chloro-2-fluorophenyl)-6-methoxy-7-(2-methoxyethoxy)cinnolin-4-amine 250855 2-chloro-4-fluoro-5-(6-methoxy-7-(2-methoxyethoxy)cinnolin-4-ylamino)phenol 250864 N-(2-fluorophenyl)-6,7-dimethoxyquinazolin-4-amine 250929 (3R,4S,5R)-2-(6-Cyclopentylamino-purin-9-yl)-5-methyl-tetrahydro-furan-3,4-diol 250967 (4S,7S,13S)-13-[(2S,3R)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-butyrylamino]-7-benzyl-3,3,14,14-tetramethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradecane-4-carboxylic acid 251013 3-[((R)-4-Benzyl-2-benzyloxymethyl-piperazin-1-yl)-(4-tert-butyl-phenyl)-methyl]-phenol 251020 3-[(4-Benzyl-piperidin-1-yl)-(4-tert-butyl-phenyl)-methyl]-phenol 251035 SID26755750 251040 3-[(1-Benzyl-piperidin-4-yl)-(4-tert-butyl-phenyl)-methyl]-phenol 251054 5-Benzyl-6-thioxo-[1,3,5]thiadiazinane-3-carboxylic acid 4-hydroxy-benzyl ester 251182 7-{3-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-propoxy}-chromen-4-one 251270 7-{3-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-propoxy}-3-methoxymethyl-chromen-4-one 251486 7-benzyl-18-cyclopropylmethyl-5-phenyl-10-oxa-7,18-diazahexacyclo[9.9.1.01,9.02,17.04,8.015,21]henicosa-4(8),5,11,13,15(21)-pentaene-2,12-diol 251497 7-{3-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-propoxy}-3-methyl-chromen-4-one 251499 7-{3-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-propoxy}-3-hydroxymethyl-chromen-4-one 251506 7-{3-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-propoxy}-2-hydroxymethyl-chromen-4-one 251507 7-{3-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-propoxy}-4-oxo-4H-chromene-3-carboxylic acid 251608 (2-Amino-3-methyl-phenyl)-(4-{1-[4-(propane-2-sulfonyl)-phenyl]-ethylidene}-[1,4']bipiperidinyl-1'-yl)-methanone 251632 7-{3-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-propoxy}-4-oxo-4H-chromene-3-carbaldehyde 251637 (4-Fluoro-naphthalen-1-yl)-(4-{1-[4-(propane-2-sulfinyl)-phenyl]-ethylidene}-[1,4']bipiperidinyl-1'-yl)-methanone 251728 4-[2-(3H-Imidazol-4-yl)-ethyl]-1-methyl-piperidine 252037 (S)-6-Propyl-4,5,5a,6,7,8-hexahydro-thiazolo[4,5-f]quinolin-2-ylamine 252070 (4-Fluoro-naphthalen-1-yl)-(4-{1-[4-(propane-2-sulfonyl)-phenyl]-ethylidene}-[1,4']bipiperidinyl-1'-yl)-methanone 252269 1-[1-(4-Fluoro-phenyl)-piperidin-4-yl]-4-(4-methoxy-phenoxy)-4-phenyl-butan-1-one 252286 Tetradecanoic acid (2S,3R)-2-hydroxymethyl-7-oxo-oxepan-3-yl ester 252618 3-{4-[3-Phenyl-3-(2-trifluoromethyl-phenoxy)-propyl]-piperazin-1-yl}-benzo[d]isothiazole 252672 4-(3H-Imidazol-4-ylmethylene)-piperidine 252730 3-{4-[3-(4-Nitro-phenoxy)-3-phenyl-propyl]-piperazin-1-yl}-benzo[d]isoxazole 252755 (3-Bromo-phenyl)-(1H-imidazo[4,5-h]quinazolin-6-yl)-amine 252756 (3-Bromo-phenyl)-(1H-1,6,8-triaza-cyclopenta[a]naphthalen-9-yl)-amine 252758 (3-Bromo-phenyl)-(1H-imidazo[4,5-f]quinazolin-9-yl)-amine 252918 3-{4-[3-Phenyl-3-(4-trifluoromethyl-phenoxy)-propyl]-piperazin-1-yl}-benzo[d]isothiazole 252919 4-(4-Amino-phenoxy)-1-[1-(4-fluoro-phenyl)-piperidin-4-yl]-4-phenyl-butan-1-one 252936 3-{4-[3-(2-Fluoro-phenoxy)-3-phenyl-propyl]-piperazin-1-yl}-benzo[d]isothiazole 252969 3-{4-[3-(2-Fluoro-phenoxy)-3-phenyl-propyl]-piperazin-1-yl}-benzo[d]isoxazole 253010 3-{4-[3-(4-Methoxy-phenoxy)-3-phenyl-propyl]-piperazin-1-yl}-benzo[d]isoxazole 253123 4-(2-Fluoro-phenoxy)-1-[1-(4-fluoro-phenyl)-piperidin-4-yl]-4-phenyl-butan-1-one 253400 {(4S,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-10-benzyl-4-[(S)-1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradec-7-yl}-acetic acid 253828 1-{5-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-1-methyl-1H-pyrrol-2-ylmethyl}-azocan-2-one 253940 6-[(1E)-3-acetyl-3-methyltriaz-1-enyl]-N-(3-methylphenyl)quinazolin-4-amine 254007 1-{5-[4-(2-Ethyl-phenyl)-piperazin-1-ylmethyl]-1-methyl-1H-pyrrol-2-ylmethyl}-piperidin-2-one 254037 ((2E)-3-{4-[(3-bromophenyl)amino]quinazolin-6-yl}-1-methyltriaz-2-enyl)methyl acetate 254051 1-{5-[4-(2-sec-Butoxy-phenyl)-piperazin-1-ylmethyl]-1-methyl-1H-pyrrol-2-ylmethyl}-piperidin-2-one 254067 1-{5-[4-(3-Chloro-phenyl)-piperazin-1-ylmethyl]-1-methyl-1H-pyrrol-2-ylmethyl}-piperidin-2-one 254084 1-{5-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-1H-pyrrol-2-ylmethyl}-piperidin-2-one 254086 Osanetant 254205 ((2E)-3-{4-[(3-bromophenyl)amino]quinazolin-6-yl}-1-methyltriaz-2-enyl)methanol 254264 8-Cyclopentyl-7-methyl-1-propyl-3,7-dihydro-purine-2,6-dione 254274 SID26755743 254276 C-(9H-Xanthen-9-yl)-methylamine 254311 8-Cyclopentyl-3-((E)-3-iodo-propenyl)-1-propyl-3,7-dihydro-purine-2,6-dione 254321 4-(10H-Anthracen-9-ylidene)-1-methyl-piperidine 254327 8-Cyclopentyl-1-(2-fluoro-propyl)-3-propyl-3,7-dihydro-purine-2,6-dione 254414 8-Cyclopentyl-3-(2-fluoro-propyl)-1-propyl-3,7-dihydro-purine-2,6-dione 254425 8-Cyclopentyl-1-(3-fluoro-propyl)-3,7-dihydro-purine-2,6-dione 254426 8-Cyclopentyl-1-ethoxymethyl-3-propyl-3,7-dihydro-purine-2,6-dione 254443 8-Cyclopentyl-3-ethoxymethyl-1-propyl-3,7-dihydro-purine-2,6-dione 254522 C-(9H-Thioxanthen-9-yl)-methylamine 254616 3-{4-[3-(4-Methoxy-phenoxy)-3-phenyl-propyl]-piperazin-1-yl}-benzo[d]isothiazole 254706 1-{5-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-1-methyl-1H-pyrrol-2-ylmethyl}-pyrrolidin-2-one 254976 (2-chloro-4-(phenylamino)phenyl)(o-tolyl)methanone 255369 [3-(2-chloro-6-methylamino-purin-9-yl)-2-phosphonomethyl-propyl]-phosphonic acid 255408 2-(pyridin-4-ylmethylamino)-N-(3-(trifluoromethyl)phenyl)benzamide 255480 Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Ser-Leu-Met-Asp-Lys-Glu-Cys) 255485 N-(3-Isoquinolin-4-yl-phenyl)-2-[(pyridin-4-ylmethyl)-amino]-benzamide 255493 Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Aoa-Val-Tyr-Phe-Cys) 255504 Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Apa-Val-Tyr-Phe-Cys) 255762 Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Val-Tyr-Phe-Cys) 255763 Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Val-Tyr-Phe-Cys) 255764 Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Aha-Val-Tyr-Phe-Cys) 255765 Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Ser-Ser-Val-Tyr-Phe-Cys) 255846 Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Asp-Lys-Glu-Val-Tyr-Phe-Cys) 256176 Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Ser-Val-Tyr-Phe-Cys) 256399 N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-1-methoxy-2-naphthamide 256556 N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-1H-indole-2-carboxamide 256582 N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-2-naphthamide 256812 H-(2S,3R)beta-MeTrp-c[Cys-Tyr-D-Trp-Arg-Thr-Pen]-Thr-NH2 256813 H-(2R,3S)beta-MeTrp-c[Cys-Tyr-D-Trp-Arg-Thr-Pen]-Thr-NH2 256814 H-(2S,3R)beta-MePhe-c[Cys-Tyr-D-Trp-Arg-Thr-Pen]-Thr-NH2 256909 H-D-Tca-c[Cys-Tyr-D-Trp-Arg-Thr-Pen]-Thr-NH2 256910 H-(2S,3S)beta-MeTrp-c[Cys-Tyr-D-Trp-Arg-Thr-Pen]-Thr-NH2 257028 H-D-Trp-c[Cys-Tyr-D-Trp-Arg-Thr-Pen]-Thr-NH2 257083 H-D-Tic-c[Cys-Tyr-D-Trp-Arg-Thr-Pen]-Thr-NH2 257084 H-(2R,3R)beta-MeTrp-c[Cys-Tyr-D-Trp-Arg-Thr-Pen]-Thr-NH2 257153 H-(2S,3S)beta-MePhe-c[Cys-Tyr-D-Trp-Arg-Thr-Pen]-Thr-NH2 257336 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzoic acid 3-hydroxy-phenyl ester 258036 2-(1H-Pyrrolo[2,3-b]pyridin-3-ylmethyl)-1,2,3,4-tetrahydro-isoquinoline 258050 3-(4-Phenethyl-piperidin-1-ylmethyl)-1H-pyrrolo[2,3-b]pyridine 258089 2-(4-Phenethyl-piperidin-1-ylmethyl)-1H-pyrrolo[2,3-b]pyridine 258123 2-(1H-Pyrrolo[2,3-b]pyridin-2-ylmethyl)-1,2,3,4-tetrahydro-isoquinoline 258171 2-[2-(4-Styryl-3,6-dihydro-2H-pyridin-1-yl)-ethyl]-1H-pyrrolo[2,3-b]pyridine 258205 2-{2-[4-(4-Chloro-phenyl)-piperazin-1-yl]-ethyl}-1H-pyrrolo[2,3-b]pyridine 258217 3-{2-[4-(4-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-1H-pyrrolo[2,3-b]pyridine 258520 Thiophene-2-sulfonic acid {4-[N'-(benzo[b]thiophene-2-carbonyl)-hydrazinocarbonyl]-cyclohexylmethyl}-amide 258521 N-{4-[N'-(Benzo[b]thiophene-2-carbonyl)-hydrazinocarbonyl]-cyclohexylmethyl}-4-methyl-benzenesulfonamide 258522 N-{4-[N'-(Benzo[b]thiophene-2-carbonyl)-hydrazinocarbonyl]-cyclohexylmethyl}-4-chloro-benzenesulfonamide 258532 N-{4-[N'-(Thiophene-2-carbonyl)-hydrazinocarbonyl]-cyclohexylmethyl}-benzenesulfonamide 258533 N-{4-[N'-(Benzo[b]thiophene-2-carbonyl)-hydrazinocarbonyl]-cyclohexylmethyl}-benzenesulfonamide 258581 Quinoline-8-sulfonic acid {4-[N'-(benzo[b]thiophene-2-carbonyl)-hydrazinocarbonyl]-cyclohexylmethyl}-amide 258603 2,4,6-Triisopropyl-N-{4-[N'-(thiophene-2-carbonyl)-hydrazinocarbonyl]-cyclohexylmethyl}-benzenesulfonamide 258604 Thiophene-2-sulfonic acid {4-[N'-(thiophene-2-carbonyl)-hydrazinocarbonyl]-cyclohexylmethyl}-amide 258605 4-Chloro-N-{4-[N'-(thiophene-2-carbonyl)-hydrazinocarbonyl]-cyclohexylmethyl}-benzenesulfonamide 258660 4-Methyl-N-{4-[N'-(thiophene-2-carbonyl)-hydrazinocarbonyl]-cyclohexylmethyl}-benzenesulfonamide 258688 Quinoline-8-sulfonic acid {4-[N'-(thiophene-2-carbonyl)-hydrazinocarbonyl]-cyclohexylmethyl}-amide 258714 3-Chloro-4-[4-(4-pyridin-2-yl-piperazin-1-yl)-butyl]-4H-benzo[f][1,4]oxazepin-5-one 258715 3-Chloro-4-[4-(4-pyrimidin-2-yl-piperazin-1-yl)-butyl]-4H-benzo[f][1,4]oxazepin-5-one 258720 N-{4-[N'-(Benzo[b]thiophene-2-carbonyl)-hydrazinocarbonyl]-cyclohexylmethyl}-4-bromo-benzenesulfonamide 258721 4-Bromo-N-{4-[N'-(thiophene-2-carbonyl)-hydrazinocarbonyl]-cyclohexylmethyl}-benzenesulfonamide 258735 N-{4-[N'-(Benzo[b]thiophene-2-carbonyl)-hydrazinocarbonyl]-cyclohexylmethyl}-2,4,6-triisopropyl-benzenesulfonamide 258905 Pentyl-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid 258941 (3-Methyl-butyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid 259005 3-(9-methoxy-13-methyl-5,7-dioxo-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrrolo[3,4-c]carbazol-12-yl)propyl cyanide 259025 (S)-5-{(S)-2-[Bis-((R)-sec-butyl)-amino]-1-hydroxy-ethyl}-1-(2-chloro-benzyl)-pyrrolidin-2-one 259026 (S)-5-{(R)-2-[Bis-((R)-sec-butyl)-amino]-1-hydroxy-ethyl}-1-(2-chloro-benzyl)-pyrrolidin-2-one 259069 (S)-5-{(S)-2-[Bis-((S)-sec-butyl)-amino]-1-hydroxy-ethyl}-1-(2-chloro-benzyl)-pyrrolidin-2-one 259078 2-(13-methyl-5,7-dioxo-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrrolo[3,4-c]carbazol-12-yl)ethyl cyanide 259079 12-(3-dimethylamino-2-hydroxypropyl)-9-methoxy-13-methyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrrolo[3,4-c]carbazol-5-one 259094 (R)-5-{(S)-2-[Bis-((R)-sec-butyl)-amino]-1-hydroxy-ethyl}-1-(2-chloro-benzyl)-pyrrolidin-2-one with sulphate 259095 (R)-5-{(R)-2-[Bis-((R)-sec-butyl)-amino]-1-hydroxy-ethyl}-1-(2-chloro-benzyl)-pyrrolidin-2-one 259096 (S)-5-{(S)-2-[((R)-sec-Butyl)-((S)-sec-butyl)-amino]-1-hydroxy-ethyl}-1-(2-chloro-benzyl)-pyrrolidin-2-one 259101 13-(3-dimethylamino-2-hydroxypropyl)-3-methoxy-12-methyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrrolo[3,4-c]carbazole-5,7-dione 259102 12-(3-dimethylamino-2-hydroxypropyl)-13-methyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrrolo[3,4-c]carbazole-5,7-dione 259106 12-(3-dimethylamino-2-hydroxypropyl)-13-methyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrrolo[3,4-c]carbazol-5-one 259114 (R)-5-{(R)-2-[((R)-sec-Butyl)-((S)-sec-butyl)-amino]-1-hydroxy-ethyl}-1-(2-chloro-benzyl)-pyrrolidin-2-one 259116 (R)-5-{(S)-2-[((R)-sec-Butyl)-((S)-sec-butyl)-amino]-1-hydroxy-ethyl}-1-(2-chloro-benzyl)-pyrrolidin-2-one 259148 12-(3-dimethylaminopropyl)-13-methyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrrolo[3,4-c]carbazol-5-one 259156 (R)-5-{(S)-2-[Bis-((S)-sec-butyl)-amino]-1-hydroxy-ethyl}-1-(2-chloro-benzyl)-pyrrolidin-2-one 259182 (S)-5-{(R)-2-[((R)-sec-Butyl)-((S)-sec-butyl)-amino]-1-hydroxy-ethyl}-1-(2-chloro-benzyl)-pyrrolidin-2-one 259202 12-(3-dimethylaminopropyl)-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrrolo[3,4-c]carbazol-5-one 259203 2-(3,9-dimethoxy-13-methyl-5-oxo-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrrolo[3,4-c]carbazol-12-yl)ethyl cyanide 259216 (S)-5-{(R)-2-[Bis-((S)-sec-butyl)-amino]-1-hydroxy-ethyl}-1-(2-chloro-benzyl)-pyrrolidin-2-one 259228 12-(3-aminopropyl)-13-methyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrrolo[3,4-c]carbazol-5-one 259240 benzyl (6R,9R,12R,16S,17R)-8-tert-butyl-6,12,17-trihydroxy-16-methyl-5,15,18-trioxo-2,4,14,19-tetraoxahexacyclo[8.7.2.0^{1,11}.0^{3,7}.0^{7,11}.0^{13,17}]nonadecan-9-yl carbonate 259267 9-azido-8-(tert-butyl)-6,12,17-trihydroxy-16-methyl-(6R,8R,9R,12R,16S,17R)-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,15,18-trione 259342 (2-Methyl-butyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid 259343 8-(tert-butyl)-6,12,17-trihydroxy-16-methyl-5,15,18-trioxo-(6R,8R,9R,12R,16S,17R)-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadec-9-yl acetate 259363 (1-Methyl-butyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid 259367 6-benzyloxy-8-(tert-butyl)-9,12,17-trihydroxy-16-methyl-(6R,8R,9R,12R,16S,17R)-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,15,18-trione 259462 (1-Methyl-heptyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid 259463 Heptyl-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid 259466 (1-Methyl-hexyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid 259475 Butyl-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid 259480 Octyl-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid 259508 Isobutyl-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid 259517 Isopropyl-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid 259554 Propyl-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid 259578 Hexyl-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid 259724 SID11111703 259871 6-benzyloxy-8-(tert-butyl)-9-fluoro-12,17-dihydroxy-16-methyl-(6R,8R,9R,12R,16S,17R)-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,15,18-trione 259872 6-benzyloxy-8-(tert-butyl)-9,12,17-trihydroxy-16-methyl-(6R,8R,9S,12R,16S,17R)-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,15,18-trione 259982 8-(tert-butyl)-9-chloro-6,12,17-trihydroxy-16-methyl-(6R,8R,9R,12R,16S,17R)-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,15,18-trione 259983 8-(tert-butyl)-9-fluoro-6,12,17-trihydroxy-16-methyl-(6R,8R,9R,12R,16S,17R)-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,15,18-trione 260017 8-(tert-butyl)-6,12,17-trihydroxy-16-methyl-9-methylamino-(6R,8R,9R,12R,16S,17R)-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,15,18-trione 260295 6-benzyloxy-8-(tert-butyl)-12,17-dihydroxy-16-methyl-(6R,8R,12R,16S,17R)-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,15,18-trione 260299 8-(tert-butyl)-6,12,17-trihydroxy-16-methyl-9-amino-(6R,8R,9R,12R,16S,17R)-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,15,18-trione 260331 8-(tert-butyl)-6,12,17-trihydroxy-16-methyl-9-ethylamino-(6R,8R,9R,12R,16S,17R)-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,15,18-trione 260495 4-{(7-Hydroxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-[3-(4-phenyl-piperazin-1-yl)-propyl]-amino}-butyronitrile 261036 7-({2-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-ethyl}-propyl-amino)-5,6,7,8-tetrahydro-naphthalen-2-ol 261075 (+)-7-[(4-(4-phenylpiperazin-1-yl)butyl)(propyl)amino]-5,6,7,8-tetrahydronaphthalen-2-ol 261076 7-({4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-butyl}-prop-2-ynyl-amino)-5,6,7,8-tetrahydro-naphthalen-2-ol 261078 7-({4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-butyl}-propyl-amino)-5,6,7,8-tetrahydro-naphthalen-2-ol 261089 7-{[2-(4-Phenyl-piperazin-1-yl)ethyl]propylamino}-5,6,7,8-tetrahydronaphthalen-2-ol 261095 7-{[2-(4-Phenyl-piperazin-1-yl)-ethyl]-prop-2-ynyl-amino}-5,6,7,8-tetrahydro-naphthalen-2-ol 261133 N-(2-{(7-Hydroxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-[3-(4-phenyl-piperazin-1-yl)-propyl]-amino}-ethyl)-benzamide 261137 (+)-7-{[4-(4-phenylpiperazin-1-yl)butyl]prop-2-ynylamino}-5,6,7,8-tetrahydronaphthalen-2-ol 261347 (1,3-dipropylxanthine)1,3-Dipropyl-3,7-dihydro-purine-2,6-dione 261373 SID11113528 261391 4-(2,6-Dioxo-1,3-dipropyl-2,3,6,9-tetrahydro-1H-purin-8-yl)-benzoic acid 261496 N-(4-{(7-Hydroxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-[3-(4-phenyl-piperazin-1-yl)-propyl]-amino}-butyl)-benzamide 261618 Ac-W-F-F-N-Y-Y-W 261619 bhg-F-N-Y-Y-W 261625 Cyclic (Gly1-Asp9) (Gly-Asn-Trp-His-Gly-Thr-Ala-Pro-Asp-Trp-Phe-Phe-Asn-Tyr-Tyr-Trp) 261765 Ac-bhg-F-N-Y-Y-W 261766 Ac-w-F-F-N-Y-Y-W 261767 W-F-F-N-Y-Y-W 262084 (6S,11R)-3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid 262085 (6S,11R)-3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid methyl ester 262217 (6S,11R)-3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid dimethylamide 262218 (6S,11R)-3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid methylamide 262251 (6S,11R)-3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carbonitrile 262285 (1R,9S,13S)-10-(cyclopropylmethyl)-1,13-dimethyl-10-azatricyclo[7.3.1.0^{2,7}]trideca-2(7),3,5-triene-4-carboxamide 262304 3-((4-(4-chlorophenyl)piperazin-1-yl)methyl)-7-methylH-pyrazolo[1,5-a]pyridine 262420 3-(indolin-1-yl)-4-(2-methoxyphenyl)-1H-pyrrole-2,5-dione 262421 2-chloro-5-(4-(2-nitrophenyl)-2,5-dioxo-2,5-dihydro-1H-pyrrol-3-ylamino)benzoic acid 262422 2-chloro-5-(4-(3-nitrophenyl)-2,5-dioxo-2,5-dihydro-1H-pyrrol-3-ylamino)benzoic acid 262468 3-(3-chlorophenylamino)-4-(4-methoxyphenyl)-1H-pyrrole-2,5-dione 262520 [3-Chloro-4-(3-fluoro-benzyloxy)-phenyl]-{6-[2-(2-methanesulfonyl-ethylamino)-thiazol-4-yl]-quinazolin-4-yl}-amine 262522 (1-Benzyl-1H-indazol-5-yl)-{6-[2-(2-methanesulfonyl-ethylamino)-thiazol-4-yl]-quinazolin-4-yl}-amine 262547 (4-Benzyloxy-3-chloro-phenyl)-{6-[2-(2-methanesulfonyl-ethylamino)-thiazol-4-yl]-quinazolin-4-yl}-amine 262779 (3-Chloro-4-fluoro-phenyl)-{6-[2-(2-methanesulfonyl-ethylamino)-thiazol-4-yl]-quinazolin-4-yl}-amine 262807 (4-Benzyloxy-phenyl)-{6-[2-(2-methanesulfonyl-ethylamino)-thiazol-4-yl]-quinazolin-4-yl}-amine 262893 3-((4-(4-chlorophenyl)piperazin-1-yl)methyl)-7-ethynyl-pyrazolo[1,5-a]pyridine 262959 {6-[2-(2-Methanesulfonyl-ethylamino)-thiazol-4-yl]-quinazolin-4-yl}-[4-(3-trifluoromethyl-benzyloxy)-phenyl]-amine 262985 (3-((4-(4-chlorophenyl)piperazin-1-yl)methyl)H-pyrazolo[1,5-a]pyridin-6-yl)methanol 263143 4-[4-(4-Fluoro-phenyl)-5-pyridin-4-yl-1H-pyrrol-2-yl]-benzoic acid 263458 1-[2-(4-Phenyl-cyclohex-3-enyl)-ethyl]-4-pyridin-2-yl-piperazine 263483 6-Methyl-4,5,5a,6,7,8-hexahydro-thiazolo[4,5-f]quinolin-2-ylamine 263517 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 263537 1-(4-Phenyl-cyclohex-3-enyl)-4-pyridin-2-yl-piperazine 263539 1-Pyridin-2-yl-4-[2-(4-thiophen-2-yl-cyclohex-3-enyl)-ethyl]-piperazine 263553 1-Pyridin-2-yl-4-(4-thiophen-2-yl-cyclohex-3-enylmethyl)-piperazine 263554 1-Pyridin-2-yl-4-(4-pyridin-2-yl-cyclohex-3-enyl)-piperazine 263558 S-(-)-Lisuride 263562 (R)-5,6-Dihydro-4H-imidazo[4,5,1-ij]quinolin-5-yl-methyl-amine 263572 1-[2-((R)-4-Phenyl-cyclohex-3-enyl)-ethyl]-4-pyridin-2-yl-piperazine 263583 1-Pyridin-2-yl-4-(4-thiophen-2-yl-cyclohex-3-enyl)-piperazine 263586 (R)-5-Propylamino-5,6-dihydro-1H,4H-imidazo[4,5,1-ij]quinolin-2-one 263587 (R)-5-Dimethylamino-5,6-dihydro-1H,4H-imidazo[4,5,1-ij]quinolin-2-one 263590 (R)-5,6-Dihydro-4H-imidazo[4,5,1-ij]quinolin-5-yl-dimethyl-amine 263669 1-Pyridin-2-yl-4-[2-(4-pyridin-2-yl-cyclohex-3-enyl)-ethyl]-piperazine 264427 (2S,5S)-2-Decyl-5-hydroxymethyl-1-methyl-1,4,5,6-tetrahydro-2H-benzo[e][1,4]diazocin-3-one 264428 (2S,5S)-5-Hydroxymethyl-1-methyl-2-tetradecyl-1,4,5,6-tetrahydro-2H-benzo[e][1,4]diazocin-3-one 264454 (2S,5S)-2-Dodecyl-5-hydroxymethyl-1-methyl-1,4,5,6-tetrahydro-2H-benzo[e][1,4]diazocin-3-one 264618 2,3-Dihydro-1H-cyclopenta[a]naphthalene-2-carboxylic acid [5-(2-ethyl-pyridin-4-yl)-1H-pyrazol-3-yl]-amide 264620 N-[5-(4-Chloro-phenyl)-2H-pyrazol-3-yl]-2-naphthalen-1-yl-acetamide 264841 Indan-2-carboxylic acid (5-phenyl-1H-pyrazol-3-yl)-amide 264859 Indan-2-carboxylic acid [5-(4-isopropoxy-phenyl)-1H-pyrazol-3-yl]-amide 264860 N-[5-(4-Chloro-phenyl)-2H-pyrazol-3-yl]-2-phenyl-acetamide 264867 N-(3-(4-chlorophenyl)-1H-pyrazol-5-yl)-2,3-dihydro-1H-indene-2-carboxamide 264939 Indan-2-carboxylic acid [5-(3-chloro-phenyl)-1H-pyrazol-3-yl]-amide 264957 N-[5-(4-Chloro-phenyl)-2H-pyrazol-3-yl]-2-naphthalen-2-yl-acetamide 264960 2,3-Dihydro-1H-cyclopenta[a]naphthalene-2-carboxylic acid (5-pyridin-4-yl-1H-pyrazol-3-yl)-amide 265000 2,3-Dihydro-1H-cyclopenta[a]naphthalene-2-carboxylic acid [5-(3,4-dimethoxy-phenyl)-1H-pyrazol-3-yl]-amide 265059 Indan-2-carboxylic acid (5-p-tolyl-1H-pyrazol-3-yl)-amide 265300 N-[5-(4-Chloro-phenyl)-2H-pyrazol-3-yl]-4-phenyl-butyramide 265458 Indan-2-carboxylic acid [5-(4-methoxy-phenyl)-1H-pyrazol-3-yl]-amide 265487 Indan-2-carboxylic acid [5-(3,4-dimethoxy-phenyl)-1H-pyrazol-3-yl]-amide 265524 Indan-2-carboxylic acid [5-(2-chloro-phenyl)-1H-pyrazol-3-yl]-amide 266639 1H-Indole-2-carboxylic acid {4-[2-(5-cyano-1,3-dihydro-isoindol-2-yl)-ethyl]-cyclohexyl}-amide 266930 (E)-N-{4-[2-(5-Cyano-1,3-dihydro-isoindol-2-yl)-ethyl]-cyclohexyl}-3-(4-fluoro-phenyl)-acrylamide 267144 Quinoline-4-carboxylic acid {4-[2-(5-cyano-1,3-dihydro-isoindol-2-yl)-ethyl]-cyclohexyl}-amide 267145 (E)-3-(4-Fluoro-phenyl)-N-{4-[2-(5-trifluoromethyl-1,3-dihydro-isoindol-2-yl)-ethyl]-cyclohexyl}-acrylamide 267147 (E)-3-(4-Fluoro-phenyl)-N-{4-[2-(5-methoxy-1,3-dihydro-isoindol-2-yl)-ethyl]-cyclohexyl}-acrylamide 267153 Methanesulfonic acid 2-(2-{4-[(E)-3-(4-fluoro-phenyl)-acryloylamino]-cyclohexyl}-ethyl)-2,3-dihydro-1H-isoindol-5-yl ester 267154 (E)-N-{4-[2-(5-Bromo-1,3-dihydro-isoindol-2-yl)-ethyl]-cyclohexyl}-3-(4-fluoro-phenyl)-acrylamide 267155 (E)-N-{4-[2-(5-Cyano-1,3-dihydro-isoindol-2-yl)-ethyl]-cyclohexyl}-3-(3-methoxy-phenyl)-acrylamide 267177 (5S,14R)-5,8-Dibenzyl-12-{4-[2-(2-hydroxy-ethoxy)-ethyl]-piperazine-1-carbonyl}-2-(1H-indol-3-ylmethyl)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 267366 (R)-4-(2-(2-(2-methylpyrrolidin-1-yl)ethyl)benzofuran-5-yl)benzonitrile 267392 N-(3-Acetylamino-4,5-dihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-2-[(2S,5R,8R,12S)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-3,6,11,14-tetraoxo-1,4,7,10tetraaza-cyclotetradec-12-yl]-acetamide 267511 (2S,5R,8R,12R)-5,8-Dibenzyl-12-(2-[1,4']bipiperidinyl-1'-yl-2-oxo-ethyl)-2-(1H-indol-3-ylmethyl)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 267537 (2S,5R,8R,12S)-5,8-Dibenzyl-12-(2-[1,4']bipiperidinyl-1'-yl-2-oxo-ethyl)-2-(1H-indol-3-ylmethyl)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 267538 2-[(2S,5R,8R,12R)-5,8-Dibenzyl-2-(1H-indol-3-ylmethyl)-3,6,11,14-tetraoxo-1,4,7,10tetraaza-cyclotetradec-12-yl]-N-(2-dimethylamino-ethyl)-acetamide 267665 (2S,5R,8R)-5,8-Dibenzyl-2-(1H-indol-3-ylmethyl)-3,6,11,14-tetraoxo-1,4,7,10tetraaza-cyclotetradecane-12-carboxylic acid (3-acetylamino-4,5-dihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-amide 267725 N-(3-Acetylamino-4,5-dihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-2-[(2S,5R,8R,12R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-3,6,11,14-tetraoxo-1,4,7,10tetraaza-cyclotetradec-12-yl]-acetamide 268185 Biphenyl-2-carboxylic acid [4-(5H,11H-benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-phenyl]-amide 268216 Biphenyl-2-carboxylic acid [4-(2-chloro-5,6,7,8-tetrahydro-thieno[3,2-b]azepine-4-carbonyl)-phenyl]-amide 268254 Biphenyl-2-carboxylic acid [3-chloro-4-(5,6,7,8-tetrahydro-thieno[3,2-b]azepine-4-carbonyl)-phenyl]-amide 268255 2,4-Dichloro-N-[4-(2-chloro-5,6,7,8-tetrahydro-thieno[3,2-b]azepine-4-carbonyl)-phenyl]-benzamide 268258 N-[3-Chloro-4-(5,6,7,8-tetrahydro-thieno[3,2-b]azepine-4-carbonyl)-phenyl]-5-fluoro-2-methyl-benzamide 268270 5-[4-(5-Chloro-2-methoxy-benzyl)-piperazin-1-yl]-2,2-dimethyl-1,2,6,7-tetrahydro-5H-azepino[3,2,1-hi]indol-4-one 268271 5-[4-(2-Methoxy-5-methyl-benzyl)-piperazin-1-yl]-2,2-dimethyl-1,2,6,7-tetrahydro-5H-azepino[3,2,1-hi]indol-4-one 268284 N-[3-Chloro-4-(4,5-dihydro-2H-9-thia-1,2,6-triaza-cyclopenta[e]azulene-6-carbonyl)-phenyl]-5-fluoro-2-methyl-benzamide 268300 2-Methyl-5-[4-(4-methyl-benzyl)-piperazin-1-yl]-1,2,6,7-tetrahydro-5H-azepino[3,2,1-hi]indol-4-one 268313 N-[3-Chloro-4-(4,5-dihydro-2H-9-thia-1,2,6-triaza-cyclopenta[e]azulene-6-carbonyl)-phenyl]-5-fluoro-2-methyl-benzamide 268316 Biphenyl-2-carboxylic acid [3-chloro-4-(4,5-dihydro-2H-9-thia-1,2,6-triaza-cyclopenta[e]azulene-6-carbonyl)-phenyl]-amide 268319 Cyclohexanecarboxylic acid [4-(2-methyl-4,5-dihydro-2H-9-thia-1,2,6-triaza-cyclopenta[e]azulene-6-carbonyl)-phenyl]-amide 268323 2-Methyl-N-[4-(2-methyl-4,5-dihydro-2H-9-thia-1,2,6-triaza-cyclopenta[e]azulene-6-carbonyl)-phenyl]-benzamide 268324 2-Chloro-N-[4-(4,5-dihydro-2H-9-thia-1,2,6-triaza-cyclopenta[e]azulene-6-carbonyl)-phenyl]-4-fluoro-benzamide 268339 5-[4-(4-Chloro-benzyl)-piperazin-1-yl]-2-methyl-1,2,6,7-tetrahydro-5H-azepino[3,2,1-hi]indol-4-one 268352 N-[4-(4,5-Dihydro-2H-9-thia-1,2,6-triaza-cyclopenta[e]azulene-6-carbonyl)-phenyl]-5-fluoro-2-methyl-benzamide 268371 2,2-Dimethyl-5-[4-(4-methyl-benzyl)-piperazin-1-yl]-1,2,6,7-tetrahydro-5H-azepino[3,2,1-hi]indol-4-one 268372 5-[4-(4-Chloro-benzyl)-piperazin-1-yl]-2,2-dimethyl-1,2,6,7-tetrahydro-5H-azepino[3,2,1-hi]indol-4-one 268433 5-[4-(4-Chloro-benzyl)-piperazin-1-yl]-1,2,6,7-tetrahydro-5H-azepino[3,2,1-hi]indol-4-one 268434 5-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1,2,6,7-tetrahydro-5H-azepino[3,2,1-hi]indol-4-one 268438 5-[4-(2-Methoxy-4-methyl-benzyl)-piperazin-1-yl]-2,2-dimethyl-1,2,6,7-tetrahydro-5H-azepino[3,2,1-hi]indol-4-one 268557 Biphenyl-2-carboxylic acid [4-(5H,11H-benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-3-chloro-phenyl]-amide 268602 N-[4-(4,5-Dihydro-2H-9-thia-1,2,6-triaza-cyclopenta[e]azulene-6-carbonyl)-phenyl]-2-methyl-benzamide 268666 2,4-Dichloro-N-[4-(2-methyl-4,5-dihydro-2H-9-thia-1,2,6-triaza-cyclopenta[e]azulene-6-carbonyl)-phenyl]-benzamide 269052 2-Phenyl-2-{4-[3-(5-[1,2,4]triazol-4-yl-1H-indol-3-yl)-propyl]-piperazin-1-yl}-acetamide 269496 8-Ethyl-1-oxo-6-phenyl-3,4-dihydro-1H-thiopyrano[3,4-c]pyridine-5-carboxylic acid propyl ester 269654 5-(2-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)ethyl)-6,7-dihydrobenzofuran-4(5H)-one 269725 6-Ethyl-5-(2-hydroxy-ethylsulfanylcarbonyl)-2-phenyl-4-propyl-nicotinic acid propyl ester 269751 1-[19-Benzyl-13-carbamoylmethyl-22-(4-ethoxy-benzyl)-16-isopropyl-12,15,18,21,24-pentaoxo-7,8-dithia-11,14,17,20,23-pentaaza-spiro[5.19]pentacosane-10-carbonyl]-pyrrolidine-2-carboxylic acid [1-(carbamoylmethyl-carbamoyl)-4-guanidino-butyl]-amide 269755 5-Ethylsulfanylcarbonyl-6-(2-fluoro-ethyl)-2-phenyl-4-propyl-nicotinic acid propyl ester 269769 4,6-Diethyl-5-ethylsulfanylcarbonyl-2-phenyl-nicotinic acid 2-fluoro-ethyl ester 269776 3-[3-(4-Furan-3-ylmethyl-piperazin-1-yl)-propyl]-5-[1,2,4]triazol-4-yl-1H-indole 269783 6-Ethyl-5-ethylsulfanylcarbonyl-2-phenyl-4-propyl-nicotinic acid 2,2,3,3,3-pentafluoro-propyl ester 269822 6-Ethyl-5-ethylsulfanylcarbonyl-2-phenyl-4-propyl-nicotinic acid 3-fluoro-propyl ester 269823 6-Ethyl-5-ethylsulfanylcarbonyl-4-(3-hydroxy-propyl)-2-phenyl-nicotinic acid propyl ester 269825 6-Ethyl-5-ethylsulfanylcarbonyl-4-(3-fluoro-propyl)-2-phenyl-nicotinic acid propyl ester 269837 4-Amino-N-(8-benzoyl-8-aza-bicyclo[3.2.1]oct-3-yl)-5-chloro-2-methoxy-benzamide 269864 6-(2-Benzyloxy-ethyl)-5-ethylsulfanylcarbonyl-2-phenyl-4-propyl-nicotinic acid propyl ester 269865 5-Ethylsulfanylcarbonyl-6-(2-hydroxy-ethyl)-2-phenyl-4-propyl-nicotinic acid propyl ester 269995 6-Ethyl-5-(2-fluoro-ethylsulfanylcarbonyl)-2-phenyl-4-propyl-nicotinic acid propyl ester 270021 5-Oxo-2-phenyl-4-propyl-7,8-dihydro-5H-thiopyrano[4,3-b]pyridine-3-carboxylic acid ethyl ester 270037 1-[5-(3-Aza-bicyclo[3.2.2]non-3-yl)-1-methyl-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl]-3-m-tolyl-urea 270050 1-(1-Methyl-2-oxo-5-piperidin-1-yl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-m-tolyl-urea 270097 6-Ethyl-5-ethylsulfanylcarbonyl-2-(3-fluoro-phenyl)-4-propyl-nicotinic acid propyl ester 270105 6-Ethyl-5-ethylsulfanylcarbonyl-2-(2-fluoro-phenyl)-4-propyl-nicotinic acid propyl ester 270106 4-[2-(1,3-Dioxo-1,3-dihydro-isoindol-2-yl)-ethyl]-6-ethyl-5-ethylsulfanylcarbonyl-2-phenyl-nicotinic acid ethyl ester 270139 5-[1,2,4]Triazol-4-yl-3-{3-[4-(4-trifluoromethyl-benzyl)-piperazin-1-yl]-propyl}-1H-indole 270510 6-Ethyl-5-ethylsulfanylcarbonyl-4-(2-hydroxy-ethyl)-2-phenyl-nicotinic acid propyl ester 270511 6-Ethyl-5-(3-fluoro-propylsulfanylcarbonyl)-2-phenyl-4-propyl-nicotinic acid propyl ester 271599 [2-(4-Bromo-2,5-dimethoxy-phenyl)-1-methyl-ethyl]-methyl-amine 271992 2-(4-Bromo-2-methoxy-phenyl)-ethylamine 271998 Bremazocine 272019 2-(4-Iodo-2-methoxy-phenyl)-1-methyl-ethylamine 272050 2-(2-Bromo-6-methoxy-phenyl)-1-methyl-ethylamine 272091 2-(2-Methoxy-4-methyl-phenyl)-ethylamine 272092 Methyl-[1-methyl-2-(4-propyl-phenyl)-ethyl]-amine 272121 (S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid [(1S,2S)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-propyl]-amide 272122 (S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid [(1S,2R)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-propyl]-amide 272123 (S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid [(S)-1-((1S,2S)-1-carbamoyl-2-phenyl-propylcarbamoyl)-2-phenyl-ethyl]-amide 272140 (S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid [(S)-1-((1R,2S)-1-carbamoyl-2-phenyl-propylcarbamoyl)-2-phenyl-ethyl]-amide 272225 (S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid [(1R,2R)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-propyl]-amide 272266 (S)-2-({(S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrrolidine-2-carbonyl}-amino)-3-phenyl-propionic acid 272398 (S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid [(S)-1-((1R,2R)-1-carbamoyl-2-phenyl-propylcarbamoyl)-2-(1H-indol-3-yl)-ethyl]-amide 272407 morphine-6-O-beta-glucuronide 272413 N*4*-(3-Bromo-phenyl)-N*6*-(3-morpholin-4-yl-propyl)-pyrido[3,4-d]pyrimidine-4,6-diamine 272537 N*4*-(3-Bromo-phenyl)-N*6*-(2-dimethylamino-ethyl)-N*6*-methyl-pyrido[3,4-d]pyrimidine-4,6-diamine 272567 2-[{3-[4-(3-Bromo-phenylamino)-pyrido[3,4-d]pyrimidin-6-ylamino]-propyl}-(2-hydroxy-ethyl)-amino]-ethanol 272568 N*4*-(3-Bromo-phenyl)-N*6*-(2-morpholin-4-yl-ethyl)-pyrido[3,4-d]pyrimidine-4,6-diamine 272706 (S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid [(S)-1-((1S,2S)-1-carbamoyl-2-phenyl-propylcarbamoyl)-2-(1H-indol-3-yl)-ethyl]-amide 272728 {4-[1-(4-Amino-benzyl)-2,6-dioxo-3-propyl-2,3,6,9-tetrahydro-1H-purin-8-yl]-phenoxy}-acetic acid 272733 (S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid [(S)-1-((1R,2S)-1-carbamoyl-2-phenyl-propylcarbamoyl)-2-(1H-indol-3-yl)-ethyl]-amide 272747 {4-[3-(4-Amino-3-iodo-benzyl)-2,6-dioxo-1-propyl-2,3,6,9-tetrahydro-1H-purin-8-yl]-phenoxy}-acetic acid 272753 {4-[3-(4-Amino-benzyl)-2,6-dioxo-1-propyl-2,3,6,9-tetrahydro-1H-purin-8-yl]-phenoxy}-acetic acid 272758 2-(2-Methoxy-4-methyl-phenyl)-1-methyl-ethylamine 272759 [2-(2-Methoxy-4-methyl-phenyl)-1-methyl-ethyl]-methyl-amine 272778 N*4*-(3-Bromo-phenyl)-N*6*-(4-dimethylamino-butyl)-pyrido[3,4-d]pyrimidine-4,6-diamine 272779 N*4*-(3-Bromo-phenyl)-N*6*-(2-dimethylamino-ethyl)-pyrido[3,4-d]pyrimidine-4,6-diamine 272781 (4-{3-[2-(4-Amino-phenyl)-ethyl]-2,6-dioxo-1-propyl-2,3,6,9-tetrahydro-1H-purin-8-yl}-phenoxy)-acetic acid 272814 N*4*-(3-Bromo-phenyl)-N*6*-(3-dimethylamino-propyl)-pyrido[3,4-d]pyrimidine-4,6-diamine 272840 (S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid [(S)-1-((1S,2R)-1-carbamoyl-2-phenyl-propylcarbamoyl)-2-phenyl-ethyl]-amide 272841 (S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid [(S)-1-((1R,2R)-1-carbamoyl-2-phenyl-propylcarbamoyl)-2-phenyl-ethyl]-amide 272842 (S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid [(1R,2S)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-propyl]-amide 272878 N*4*-(3-Bromo-phenyl)-N*6*-[3-(4-methyl-piperazin-1-ylamino)-propyl]-pyrido[3,4-d]pyrimidine-4,6-diamine 272879 2-[{2-[4-(3-Bromo-phenylamino)-pyrido[3,4-d]pyrimidin-6-ylamino]-ethyl}-(2-hydroxy-ethyl)-amino]-ethanol 272920 (S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid [(S)-1-((1S,2R)-1-carbamoyl-2-phenyl-propylcarbamoyl)-2-(1H-indol-3-yl)-ethyl]-amide 273000 N*4*-(3-Bromo-phenyl)-N*6*-pyridin-3-ylmethyl-pyrido[3,4-d]pyrimidine-4,6-diamine 273013 N*4*-(3-Bromo-phenyl)-N*6*-(3-imidazol-1-yl-propyl)-pyrido[3,4-d]pyrimidine-4,6-diamine 273047 N*4*-(3-Bromo-phenyl)-N*6*-[2-(3H-imidazol-4-yl)-ethyl]-pyrido[3,4-d]pyrimidine-4,6-diamine 273103 N*4*-(3-Bromo-phenyl)-N*6*-(2-pyridin-2-yl-ethyl)-pyrido[3,4-d]pyrimidine-4,6-diamine 273114 3-(2-(naphthalen-2-ylmethyl)phenyl)acrylic acid 273124 Tyr-Gly-Gly-Phe-Leu-Arg-Arg-c(Cys-Arg-Pro-Lys-Leu-Cys) 273217 1-[4-(3-Bromo-phenylamino)-pyrido[3,4-d]pyrimidin-6-ylamino]-3-diethylamino-propan-2-ol 273282 Tyr-Gly-Gly-Phe-leu-c(Cys-Arg-Ile-Arg-Cys)-lys 273283 Tyr-Gly-Gly-Phe-c(Cys-Arg-Arg-Ile-Cys)-Arg-lys 273354 Naphthalene-1-sulfonic acid [2-(4-{[(3-methoxy-6,7,8,9-tetrahydro-5H-benzocyclohepten-6-ylmethyl)-amino]-methyl}-piperidin-1-yl)-ethyl]-amide 273356 SID24826288 273387 N-(4-Pyridin-2-yl-thiazol-2-yl)-benzamide 273390 3-Chloro-N-(4-pyridin-2-yl-thiazol-2-yl)-benzamide 273467 Dipropyl-(4-trimethylsilanylethynyl-cyclohex-3-enyl)-amine 273468 4-ethynyl-N,N-dipropylcyclohex-3-enamine 273484 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-[4-(2-diethylaminomethyl-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-amide 273523 (3-Bromo-phenyl)-[6-(4-methyl-piperazin-1-yl)-pyrido[3,4-d]pyrimidin-4-yl]-amine 273539 (6-{4-[(4'-Methyl-biphenyl-2-carbonyl)-amino]-benzoyl}-3,4,5,6-tetrahydro-azepino[4,3,2-cd]indol-1-yl)-acetic acid ethyl ester 273554 2-({2-[4-(3-Bromo-phenylamino)-pyrido[3,4-d]pyrimidin-6-ylamino]-ethyl}-methyl-amino)-ethanol 273582 3-[4-(3-Bromo-phenylamino)-pyrido[3,4-d]pyrimidin-6-ylamino]-propionic acid 273596 2-[8-(3-Amino-propyl)-6-benzo[b]thiophen-3-yl-imidazo[1,2-a]pyrazin-2-yl]-N-cyclohexyl-isobutyramide 273597 3-(6-Benzo[b]thiophen-3-yl-2-phenyl-imidazo[1,2-a]pyrazin-8-yl)-propylamine 273659 2-[8-(3-Amino-propyl)-6-benzo[b]thiophen-3-yl-imidazo[1,2-a]pyrazin-2-yl]-N-[2-(1H-indol-3-yl)-ethyl]-isobutyramide 273677 1-Phenyl-3-(4-pyridin-2-yl-thiazol-2-yl)-urea 273704 N*6*-Methyl-N*4*-m-tolyl-pyrido[3,4-d]pyrimidine-4,6-diamine 273731 Biphenyl-2-carboxylic acid [4-(1,3,4,5-tetrahydro-azepino[4,3,2-cd]indole-6-carbonyl)-phenyl]-amide 273735 2-[8-(3-Amino-propyl)-6-benzo[b]thiophen-3-yl-imidazo[1,2-a]pyrazin-2-yl]-N-butyl-isobutyramide 273778 3-[6-(3-Nitro-phenyl)-2-phenyl-imidazo[1,2-a]pyrazin-8-yl]-propylamine 273779 N*6*-(2-Morpholin-4-yl-ethyl)-N*4*-m-tolyl-pyrido[3,4-d]pyrimidine-4,6-diamine 273785 Biphenyl-2-carboxylic acid [4-(2-oxo-1,2,2a,3,4,5-hexahydro-azepino[4,3,2-cd]indole-6-carbonyl)-phenyl]-amide 273816 N-(3-Phenyl-[1,2,4]thiadiazol-5-yl)-benzamide 273836 4'-Methyl-biphenyl-2-carboxylic acid [4-(1,3,4,5-tetrahydro-azepino[4,3,2-cd]indole-6-carbonyl)-phenyl]-amide 273862 4-Dipropylamino-cyclohex-1-enecarbonitrile 273894 (4-Dipropylamino-cyclohexylidene)-acetonitrile 273895 2-(4-Dipropylamino-cyclohexylidene)-malononitrile 273937 Tyr-Gly-Gly-Phe-c(Cys-Arg-Arg-Ile-Arg-(D-Pro)-Lys-Leu-Cys) 273938 Tyr-Gly-Gly-Phe-Leu-Arg-Arg-c((D-Cys)-Arg-Pro-Lys-(D-Cys))-Lys 274021 4-Hydroxy-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benzamide (LUF5437) 274159 4'-Methyl-biphenyl-2-carboxylic acid [4-(1-methyl-1,3,4,5-tetrahydro-azepino[4,3,2-cd]indole-6-carbonyl)-phenyl]-amide 274211 4'-Methyl-biphenyl-2-carboxylic acid [4-(1-acetyl-1,3,4,5-tetrahydro-azepino[4,3,2-cd]indole-6-carbonyl)-phenyl]-amide 274213 Biphenyl-2-carboxylic acid [3-chloro-4-(1,3,4,5-tetrahydro-azepino[4,3,2-cd]indole-6-carbonyl)-phenyl]-amide 274214 5-Fluoro-2-methyl-N-[4-(1,3,4,5-tetrahydro-azepino[4,3,2-cd]indole-6-carbonyl)-phenyl]-benzamide 274277 (Trans)-4-Methoxy-cyclohexanecarboxylic acid (3-phenyl-[1,2,4]thiadiazol-5-yl)-amide 274314 3-Fluoro-2-methyl-N-[4-(1,3,4,5-tetrahydro-azepino[4,3,2-cd]indole-6-carbonyl)-phenyl]-benzamide 274333 Biphenyl-2-carboxylic acid [2-chloro-4-(1,3,4,5-tetrahydro-azepino[4,3,2-cd]indole-6-carbonyl)-phenyl]-amide 274393 [4-(3-Phenyl-[1,2,4]thiadiazol-5-ylcarbamoyl)-phenoxy]-acetic acid 274428 [4-(3-Phenyl-1-phenylethynyl-prop-2-ynylidene)-cyclohexyl]-dipropyl-amine 274431 Dipropyl-[4-(3-trimethylsilanyl-1-trimethylsilanylethynyl-prop-2-ynylidene)-cyclohexyl]-amine 274457 [4-(1-Ethynyl-prop-2-ynylidene)-cyclohexyl]-dipropyl-amine 274460 (4-Phenylethynyl-cyclohex-3-enyl)-dipropyl-amine 274464 6-{4-[(Biphenyl-2-carbonyl)-amino]-3-chloro-benzoyl}-3,4,5,6-tetrahydro-1H-azepino[4,3,2-cd]indole-2-sulfonic acid 274465 6-{4-[(Biphenyl-2-carbonyl)-amino]-benzoyl}-3,4,5,6-tetrahydro-1H-azepino[4,3,2-cd]indole-2-sulfonic acid 274466 Biphenyl-2-carboxylic acid [4-(2-chloro-1,3,4,5-tetrahydro-azepino[4,3,2-cd]indole-6-carbonyl)-phenyl]-amide 274548 1-(2-chlorophenyl)-3-(2-(furan-2-yl)-8-propyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 274549 1-(2-(furan-2-yl)-8-propyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(3-methoxyphenyl)urea 274550 1-(2-(furan-2-yl)-8-propyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(2-methoxyphenyl)urea 274614 1-(2-(furan-2-yl)-8-propyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-p-tolylurea 274615 1-(benzo[d][1,3]dioxol-5-yl)-3-(2-(furan-2-yl)-8-propyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 274786 RES-701-1-C-terminal analogue 274787 RES-701-1-C-terminal analogue 274805 4-(3-(8-butyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)ureido)benzenesulfonic acid 274806 1-(4-chlorophenyl)-3-(2-(furan-2-yl)-8-propyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 274830 1-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(2-methoxyphenyl)urea 274831 1-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-(trifluoromethyl)phenyl)urea 274832 1-(8-butyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-phenylurea 274922 1-(4-fluorophenyl)-3-(2-(furan-2-yl)-8-propyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 274945 RES-701-1-C-terminal analogue 274946 RES-701-1-C-terminal analogue 274949 1-(benzo[d][1,3]dioxol-5-yl)-3-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 274950 1-(2-(furan-2-yl)-8-propyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-(trifluoromethyl)phenyl)urea 274951 1-(4-bromophenyl)-3-(2-(furan-2-yl)-8-propyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 274970 RES-701-1-C-terminal analogue 274974 1-(3,4-dichlorophenyl)-3-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 275048 RES-701-1-C-terminal analogue 275049 RES-701-1-C-terminal analogue 275114 1-(8-butyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-chlorophenyl)urea 275115 1-(8-butyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(2-chlorophenyl)urea 275199 RES-701-1-C-terminal analogue 275200 RES-701-1-C-terminal analogue 275241 N-(8-butyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-2-phenylacetamide 275242 N-(2-(furan-2-yl)-8-propyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-2-phenylacetamide 275312 1-(4-bromophenyl)-3-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 275343 1-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-p-tolylurea 275346 1-(8-butyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(2-methoxyphenyl)urea 275347 N-(8-ethyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-2-phenylacetamide 275354 1-(8-ethyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-nitrophenyl)urea 275377 1-(4-fluorophenyl)-3-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 275382 1-(8-butyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-(trifluoromethyl)phenyl)urea 275392 1-(8-butyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-fluorophenyl)urea 275395 1-(4-bromophenyl)-3-(8-butyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 275456 1-(4-bromophenyl)-3-(8-ethyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 275471 1-(3,4-dichlorophenyl)-3-(8-ethyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 275493 1-(8-ethyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-p-tolylurea 275511 4-(3-(8-ethyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)ureido)benzenesulfonic acid 275548 1-(benzo[d][1,3]dioxol-5-yl)-3-(8-ethyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 275721 1-(8-butyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(3-methoxyphenyl)urea 275848 1-(8-butyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-nitrophenyl)urea 275849 1-(2-(furan-2-yl)-8-propyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-nitrophenyl)urea 275917 (S)-3-{[1-({1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-cyclohexanecarbonyl}-amino)-cyclohexanecarbonyl]-amino}-N-{(S)-1-[(S)-1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-succinamic acid 275945 1-(benzo[d][1,3]dioxol-5-yl)-3-(8-butyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 275973 1-(8-butyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-p-tolylurea 275977 1-(8-butyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(3,4-dichlorophenyl)urea 276022 1-(8-ethyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-phenylurea 276027 1-(2-chlorophenyl)-3-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 276054 1-(4-chlorophenyl)-3-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 276066 (S)-3-[(1-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-cyclopropanecarbonyl)-amino]-N-{(S)-1-[(S)-1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-succinamic acid 276092 1-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(3-methoxyphenyl)urea 276093 1-(4-chlorophenyl)-3-(8-ethyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 276094 1-((S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-3-phenyl-propionylamino)-cyclopropanecarboxylic acid {(S)-1-[(S)-1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-amide 276096 1-(3,4-dichlorophenyl)-3-(2-(furan-2-yl)-8-propyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 276123 1-(2-(furan-2-yl)-8-propyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-phenylurea 276124 1-(2-chlorophenyl)-3-(8-ethyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)urea 276125 1-((S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-3-phenyl-propionylamino)-cyclopentanecarboxylic acid {(S)-1-[(S)-1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-amide 276126 (S)-3-({1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-cyclohexanecarbonyl}-amino)-N-{(S)-1-[(S)-1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-succinamic acid 276127 1-(8-ethyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(3-methoxyphenyl)urea 276128 4-(3-(2-(furan-2-yl)-8-propyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)ureido)benzenesulfonic acid 276129 (S)-3-[(1-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-cyclopentanecarbonyl)-amino]-N-{(S)-1-[(S)-1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-succinamic acid 276167 1-(8-ethyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(2-methoxyphenyl)urea 276175 1-(8-ethyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-(trifluoromethyl)phenyl)urea 276176 1-((S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-3-phenyl-propionylamino)-cyclohexanecarboxylic acid {(S)-1-[(S)-1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-amide 276177 (S)-3-[(S)-2-({1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-cyclohexanecarbonyl}-amino)-3-phenyl-propionylamino]-N-{(S)-1-[(S)-1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-succinamic acid 276221 (S)-3-[(1-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-cyclohexanecarbonyl)-amino]-N-{(S)-1-[(S)-1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-succinamic acid 276222 1-(8-ethyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-fluorophenyl)urea 276224 1-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-nitrophenyl)urea 276276 10-[2-Chloro-4-(5-fluoro-2-methyl-benzoylamino)-benzoyl]-10,11-dihydro-5H-benzo[e]pyrrolo[1,2-a][1,4]diazepine-3-carboxylic acid 276410 Biphenyl-2-carboxylic acid [3-chloro-4-(3-dimethylaminomethyl-5H,11H-benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-phenyl]-amide 276411 Biphenyl-2-carboxylic acid {3-chloro-4-[3-(4-dimethylamino-piperidine-1-carbonyl)-5H,11H-benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl]-phenyl}-amide 276412 Biphenyl-2-carboxylic acid {3-chloro-4-[3-(4-methyl-piperazine-1-carbonyl)-5H,11H-benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl]-phenyl}-amide; compound with 3-carboxy-3-hydroxy-pentanedioic acid 276426 10-{4-[(Biphenyl-2-carbonyl)-amino]-2-chloro-benzoyl}-10,11-dihydro-5H-benzo[e]pyrrolo[1,2-a][1,4]diazepine-3-carboxylic acid 276437 Biphenyl-2-carboxylic acid [4-(3-dimethylaminomethyl-5H,11H-benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-2-methoxy-phenyl]-amide 276448 Biphenyl-2-carboxylic acid [3-chloro-4-(3-{[(2-dimethylamino-ethyl)-methyl-amino]-methyl}-5H,11H-benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-phenyl]-amide 276470 Biphenyl-2-carboxylic acid {3-chloro-4-[3-(4-dimethylamino-piperidin-1-ylmethyl)-5H,11H-benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl]-phenyl}-amide 276471 Biphenyl-2-carboxylic acid [4-(3-[1,4']bipiperidinyl-1'-ylmethyl-5H,11H-benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-3-chloro-phenyl]-amide 276503 Biphenyl-2-carboxylic acid {3-chloro-4-[3-(4-methyl-piperazin-1-ylmethyl)-5H,11H-benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl]-phenyl}-amide 276624 5,6,7-Trimethyl-2-p-tolyl-chromen-4-one 276734 Sorafenib 276907 Biphenyl-2-carboxylic acid {3-methoxy-4-[3-(4-methyl-piperazin-1-ylmethyl)-5H,11H-benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl]-phenyl}-amide 276908 Biphenyl-2-carboxylic acid [4-(3-dimethylaminomethyl-5H,11H-benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-3-hydroxy-phenyl]-amide 277341 Naphthalene-1-sulfonic acid [2-(4-{[(1-hydroxy-7-methoxy-1,2,3,4-tetrahydro-naphthalen-1-ylmethyl)-amino]-methyl}-piperidin-1-yl)-ethyl]-amide 277367 Naphthalene-1-sulfonic acid (2-{4-[(3-methoxy-6,7,8,9-tetrahydro-5H-benzocyclohepten-6-ylamino)-methyl]-piperidin-1-yl}-2-oxo-ethyl)-amide 277368 4'-(6-Isopropyl-4-oxo-2-propyl-4H-quinazolin-3-ylmethyl)-biphenyl-2-sulfonic acid cyclopropanecarbonyl-amide 277382 N-[2-(4-{[(1-Hydroxy-7-methoxy-1,2,3,4-tetrahydro-naphthalen-1-ylmethyl)-amino]-methyl}-piperidin-1-yl)-ethyl]-3-methyl-benzenesulfonamide 277396 1-[2-(5-Chloro-2-oxo-benzothiazol-3-yl)-acetyl]-piperidine-4-carboxylic acid (3-methoxy-6,7,8,9-tetrahydro-5H-benzocyclohepten-6-ylmethyl)-amide 277439 1-[2-(5-Chloro-2-oxo-benzothiazol-3-yl)-acetyl]-piperidine-4-carboxylic acid (1-hydroxy-7-methoxy-1,2,3,4-tetrahydro-naphthalen-1-ylmethyl)-amide 277440 5-Chloro-3-[2-(4-{[(1-hydroxy-7-methoxy-1,2,3,4-tetrahydro-naphthalen-1-ylmethyl)-amino]-methyl}-piperidin-1-yl)-2-oxo-ethyl]-3H-benzothiazol-2-one 277586 4-(7-Fluoro-3,4-dihydro-naphthalen-2-ylmethyl)-4,5-dihydro-1H-imidazole 277592 4-(8-Fluoro-3,4-dihydro-naphthalen-2-ylmethyl)-4,5-dihydro-1H-imidazole 277611 4'-(2-Butyl-6-isopropyl-4-oxo-4H-quinazolin-3-ylmethyl)-biphenyl-2-sulfonic acid benzoylamide 277612 4'-(2-Butyl-6-isopropyl-4-oxo-4H-quinazolin-3-ylmethyl)-biphenyl-2-sulfonic acid (1-methyl-cyclopropanecarbonyl)-amide 277613 4'-(2-Butyl-6-isopropyl-4-oxo-4H-quinazolin-3-ylmethyl)-biphenyl-2-sulfonic acid (6-amino-hexanoyl)-amide 277614 6-[4'-(6-Isopropyl-4-oxo-2-propyl-4H-quinazolin-3-ylmethyl)-biphenyl-2-sulfonylamino]-6-oxo-hexanoic acid 277649 Spiro[(1,3-diazacyclopent-1-ene)-5:2''-(trans-1'',2'',3'',4''-4'a,9',9'a,10-octahydroantrhacene)] 277680 2-Methyl-6-pyrrolidin-1-yl-hex-4-ynal oxime 277699 Quinazolinone Biphenyl Acylsulfonamide derivative 277761 4(5)-{Spiro[cycloprpane-2':2''-(1'',2'',3'',4''-tetrahydronaphthalene)]-1'-yl}-4,5-dihydroimidazole 277796 [3-(2'-Benzoylsulfamoyl-biphenyl-4-ylmethyl)-4-oxo-2-propyl-3,4-dihydro-quinazolin-6-yl]-methyl-carbamic acid isobutyl ester 277797 {2-Butyl-3-[2'-(cyclopropanecarbonyl-sulfamoyl)-biphenyl-4-ylmethyl]-4-oxo-3,4-dihydro-quinazolin-6-yl}-methyl-carbamic acid isobutyl ester 277798 4'-(6-Dimethylamino-4-oxo-2-propyl-4H-quinazolin-3-ylmethyl)-biphenyl-2-sulfonic acid benzoylamide 277859 {6-[4'-(2-Butyl-6-isopropyl-4-oxo-4H-quinazolin-3-ylmethyl)-biphenyl-2-sulfonylamino]-6-oxo-hexyl}-carbamic acid tert-butyl ester 277860 4'-(2-Butyl-6-isopropyl-4-oxo-4H-quinazolin-3-ylmethyl)-biphenyl-2-sulfonic acid (3-cyclopentyl-propionyl)-amide 277861 4'-(2-Butyl-6-isopropyl-4-oxo-4H-quinazolin-3-ylmethyl)-biphenyl-2-sulfonic acid 4-fluoro-benzoylamide 277943 4'-(2-Butyl-6-isopropyl-4-oxo-4H-quinazolin-3-ylmethyl)-biphenyl-2-sulfonic acid (1H-tetrazole-5-carbonyl)-amide 277944 Quinazolinone Biphenyl Acylsulfonamide derivative 277972 4'-(6-Dimethylamino-4-oxo-2-propyl-4H-quinazolin-3-ylmethyl)-biphenyl-2-sulfonic acid cyclopropanecarbonyl-amide 277975 4'-(2-Butyl-6-dimethylamino-4-oxo-4H-quinazolin-3-ylmethyl)-biphenyl-2-sulfonic acid cyclopropanecarbonyl-amide 277977 4'-(2-Butyl-6-isopropyl-4-oxo-4H-quinazolin-3-ylmethyl)-biphenyl-2-sulfonic acid (thiophene-2-carbonyl)-amide 278009 5-Chloro-3-(2-{4-[(3-methoxy-6,7,8,9-tetrahydro-5H-benzocyclohepten-6-ylamino)-methyl]-piperidin-1-yl}-2-oxo-ethyl)-3H-benzothiazol-2-one 278010 Naphthalene-1-sulfonic acid [2-(4-{2-[(1-hydroxy-7-methoxy-1,2,3,4-tetrahydro-naphthalen-1-ylmethyl)-amino]-ethyl}-piperidin-1-yl)-ethyl]-amide 278011 Naphthalene-1-sulfonic acid [2-(4-{[(6-hydroxy-3-methoxy-6,7,8,9-tetrahydro-5H-benzocyclohepten-6-ylmethyl)-amino]-methyl}-piperidin-1-yl)-ethyl]-amide 278024 4-Benzofuran-2-ylmethyl-4,5-dihydro-1H-imidazole 278025 4-Indan-2-ylmethyl-4,5-dihydro-1H-imidazole 278049 4'-(2-Butyl-6-isopropyl-4-oxo-4H-quinazolin-3-ylmethyl)-biphenyl-2-sulfonic acid cyclopropanecarbonyl-amide 278118 3-Chloro-N-[2-(4-{[(1-hydroxy-7-methoxy-1,2,3,4-tetrahydro-naphthalen-1-ylmethyl)-amino]-methyl}-piperidin-1-yl)-ethyl]-2-methyl-benzenesulfonamide 278121 Naphthalene-1-sulfonic acid [2-(4-{[(1-hydroxy-6-methoxy-indan-1-ylmethyl)-amino]-methyl}-piperidin-1-yl)-ethyl]-amide 278166 4-(8-Chloro-naphthalen-2-ylmethyl)-4,5-dihydro-1H-imidazole 278169 3-{(R)-7-[3-(2-Cyclopropylmethyl-3-methoxy-4-methylcarbamoyl-phenoxy)-propoxy]-8-propyl-chroman-2-yl}-propionic acid 278221 7-[3-(4-Dimethylcarbamoyl-3-methoxy-2-propyl-phenoxy)-propoxy]-8-propyl-chroman-2-carboxylic acid 278226 [Cys-Trp-Arg-Nva-Arg-Tyr-NH2]2 278260 7-[3-(2-Cyclopropylmethyl-3-methoxy-4-methylcarbamoyl-phenoxy)-propoxy]-8-propyl-chroman-2-carboxylic acid 278393 4-(8-Chloro-3,4-dihydro-naphthalen-2-ylmethyl)-4,5-dihydro-1H-imidazole 278421 4-(3,4-Dihydro-naphthalen-2-ylmethyl)-4,5-dihydro-1H-imidazole 278422 Atipamezole 278453 4-(1,2,3,7b-Tetrahydro-cyclopropa[a]naphthalen-1a-ylmethyl)-4,5-dihydro-1H-imidazole 278484 1-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-piperidin-4-yl]-5-methyl-1,3-dihydro-benzoimidazol-2-one 278485 1-[1-(7-Fluoro-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-piperidin-4-yl]-5-methyl-1,3-dihydro-benzoimidazol-2-one 278566 6-Dimethylamino-2-methyl-hex-4-ynal oxime 278604 1-(4-Bromo-benzyl)-3-[3-(3-isopropoxy-phenyl)-4-oxo-3,4-dihydro-quinazolin-2-ylmethyl]-urea 278630 1-(4-Bromo-phenyl)-3-[3-(3-isopropoxy-phenyl)-4-oxo-3,4-dihydro-quinazolin-2-ylmethyl]-thiourea 278656 1-(2-Chloro-5-methylene-5H-dibenzo[a,d]cyclohepten-10-yl)-4-methyl-piperazine 278669 3-{3-[3-(3-Isopropoxy-phenyl)-4-oxo-3,4-dihydro-quinazolin-2-ylmethyl]-ureido}-benzoic acid ethyl ester 278687 3-Methyl-7-pyrrolidin-1-yl-hept-5-yn-2-one 278707 7-[3-(4-Carbamoyl-3-methoxy-2-propyl-phenoxy)-propoxy]-8-propyl-chroman-2-carboxylic acid 278715 5-(3-Butoxy-isothiazol-4-yl)-1-methyl-1,2,3,6-tetrahydro-pyridine 278733 7-[3-(4-Isopropylcarbamoyl-3-methoxy-2-propyl-phenoxy)-propoxy]-8-propyl-chroman-2-carboxylic acid 278734 7-[3-(3-Methoxy-4-methylcarbamoyl-2-propyl-phenoxy)-propoxy]-8-propyl-chroman-2-carboxylic acid 278739 7-Dimethylamino-hept-5-yn-2-one 278792 5-(3-Hexyloxy-isothiazol-4-yl)-1-methyl-1,2,3,6-tetrahydro-pyridine 278793 5-(4-Butoxy-thiophen-3-yl)-1-methyl-1,2,3,6-tetrahydro-pyridine 278887 5-Chloro-1-[1-(2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-piperidin-4-yl]-1,3-dihydro-benzoimidazol-2-one 278997 5-Fluoro-1-[1-(6-fluoro-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-piperidin-4-yl]-1,3-dihydro-benzoimidazol-2-one 279010 5-(3,4-Dichloro-benzyl)-3-(3-methoxy-phenyl)-1H-[1,2,4]triazole 279030 5-(4-Hexyloxy-thiophen-3-yl)-1-methyl-1,2,3,6-tetrahydro-pyridine 279084 3-(3-Bromo-benzyl)-5-(3-methoxy-phenyl)-1H-[1,2,4]triazole 279085 5-[2-(3,4-Dichloro-phenyl)-ethyl]-3-(3-methoxy-phenyl)-1H-[1,2,4]triazole 279217 1-[3-(3-Isopropoxy-phenyl)-4-oxo-3,4-dihydro-quinazolin-2-ylmethyl]-3-m-tolyl-urea 279228 5-Bromo-1-[1-(2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-piperidin-4-yl]-1,3-dihydro-benzoimidazol-2-one 279251 1-[3-(3-Isopropoxy-phenyl)-4-oxo-3,4-dihydro-quinazolin-2-ylmethyl]-3-(4-nitro-phenyl)-urea 279274 2-[2-chloro-6-(methylamino)-9H-purin-9-yl]-4-fluoro-5-(hydroxymethyl)tetrahydrofuran-3-ol 279275 5-{2-chloro-6-[(3-iodobenzyl)amino]-9H-purin-9-yl}-3-fluoro-4-hydroxy-N-methyltetrahydrofuran-2-carboxamide 279347 1-[3-(3-Isopropoxy-phenyl)-4-oxo-3,4-dihydro-quinazolin-2-ylmethyl]-3-(4-trifluoromethyl-phenyl)-urea 279372 5-(3-Methoxy-phenyl)-3-naphthalen-2-ylmethyl-1H-[1,2,4]triazole 279440 5-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(3-pyrrolidin-1-ylmethyl-phenyl)-1H-[1,2,4]triazole 279441 5-Fluoro-1-[1-(5-methyl-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-piperidin-4-yl]-1,3-dihydro-benzoimidazol-2-one 279473 5-Methyl-1-[1-(6-methyl-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-piperidin-4-yl]-1,3-dihydro-benzoimidazol-2-one 279477 3-(4-Azido-phenyl)-5-[3-(2,5-dihydro-pyrrol-1-ylmethyl)-phenyl]-1-methyl-1H-[1,2,4]triazole 279521 1-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-piperidin-4-yl]-5-methoxy-1,3-dihydro-benzoimidazol-2-one 279573 2-(11,15-dimethoxy-3-methyl-13-oxa-3-azahexacyclo[13.2.2.12,8.01,6.06,14.07,12]icosa-7,9,11-trien-16-yl)-3-methyl-2-butanol 279574 3-cyclopropylmethyl-18-methyl-(15S)-13,16-dioxa-3-azaheptacyclo[13.5.2.12,8.01,6.06,14.07,12.015,19]tricosa-7,9,11-trien-11-ol 279670 3-(3,4-dimethylbenzyl)-5-(3-methoxyphenyl)-1H-1,2,4-triazole 279704 3-(2,3-Difluoro-benzyl)-5-(3-methoxy-phenyl)-1H-[1,2,4]triazole 279736 5-(3,4-Dichloro-phenyl)-3-(3-methoxy-phenyl)-1H-[1,2,4]triazole 280027 1-[1-(6,7-Dimethyl-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-piperidin-4-yl]-5-fluoro-1,3-dihydro-benzoimidazol-2-one 280029 1-[1-(6,7-Dimethyl-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-piperidin-4-yl]-5-methyl-1,3-dihydro-benzoimidazol-2-one 280062 5-Chloro-1-[1-(6-methyl-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-piperidin-4-yl]-1,3-dihydro-benzoimidazol-2-one 280211 3-cyclopropylmethyl-18,18-dimethyl-(15S)-13,16-dioxa-3-azaheptacyclo[13.5.2.12,8.01,6.06,14.07,12.015,19]tricosa-7,9,11-trien-11-ol 280212 2-[11,15-dimethoxy-3-methyl-(14R,15S)-13-oxa-3-azahexacyclo[13.2.2.12,8.01,6.06,14.07,12]icosa-7,9,11-trien-16-yl]-3,3-dimethyl-2-butanol 280245 3-cyclopropylmethyl-18-methyl-(15S)-13,16-dioxa-3-azaheptacyclo[13.5.2.12,8.01,6.06,14.07,12.015,19]tricosa-7,9,11-trien-11-ol 280379 2-{2-chloro-6-[(3-iodobenzyl)amino]-9H-purin-9-yl}-4-fluoro-5-(hydroxymethyl)tetrahydrofuran-3-ol 280428 2-[1-Pyridin-2-yl-meth-(E)-ylidene]-3,4-dihydro-2H-naphthalen-1-one 280519 2-(3-cyclopropylmethyl-11-hydroxy-15-methoxy-13-oxa-3-azahexacyclo[13.2.2.12,8.01,6.06,14.07,12]icosa-7,9,11-trien-16-yl)-2-propanol 280606 8-(R)-Acenaphthen-1-yl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 280679 3,17,17,18-tetramethyl-13,16-dioxa-3-azaheptacyclo[13.5.2.12,8.01,6.06,14.07,12.015,19]tricosa-7,9,11-trien-11-ol 280896 (2-Methoxy-benzyl)-[(2S,3S)-2-(3-methoxy-phenyl)-1-aza-bicyclo[2.2.2]oct-3-yl]-amine 280897 [(2S,3S)-2-(3-Chloro-phenyl)-1-aza-bicyclo[2.2.2]oct-3-yl]-(2-methoxy-benzyl)-amine 280899 (2-Methoxy-benzyl)-((2S,3R)-2-phenyl-1-aza-bicyclo[2.2.2]oct-3-yl)-amine 280958 [(2R,3S)-2-(3-Chloro-phenyl)-1-aza-bicyclo[2.2.2]oct-3-yl]-(2,4-dimethoxy-benzyl)-amine 281487 (2-Methoxy-benzyl)-((2S,3S)-2-phenyl-1-aza-bicyclo[2.2.2]oct-3-yl)-amine 281491 [(2S,3R)-2-(3-Chloro-phenyl)-1-aza-bicyclo[2.2.2]oct-3-yl]-(2-methoxy-benzyl)-amine 281510 4-[2-(4-Amino-5-phenyl-pyrrolo[2,3-d]pyrimidin-7-yl)-3-hydroxy-propyl]-phenol 281542 2-[4-Amino-5-(3-methoxy-phenyl)-pyrrolo[2,3-d]pyrimidin-7-yl]-3-(4-methoxy-phenyl)-propan-1-ol 281700 1-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-{3-[(1H-tetrazol-5-ylamino)-methyl]-phenyl}-urea 281701 1-((R)-5-Cyclohexyl-1-methyl-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-[3-(1H-tetrazol-5-ylamino)-phenyl]-urea 281720 4-(4-amino-7-cyclobutyl-7H-pyrrolo[2,3-d]pyrimidin-5-yl)phenol 281721 7-cyclobutyl-5-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine 281732 5-{[1-(2,5-Dihydroxy-phenyl)-meth-(E)-ylidene]-amino}-2-hydroxy-benzoic acid ethyl ester 281739 2-{3-[4-Amino-5-(3-hydroxy-phenyl)-pyrrolo[2,3-d]pyrimidin-7-yl]-pyrrolidin-1-yl}-acetamide 281740 {3-[4-Amino-5-(3-hydroxy-phenyl)-pyrrolo[2,3-d]pyrimidin-7-yl]-pyrrolidin-1-yl}-acetic acid methyl ester 281760 N-tert-Butoxy-2-[5-(2,5-dihydroxy-benzylamino)-2-hydroxy-phenyl]-acetamide 281763 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzoic acid naphthalen-2-yl ester 281770 (S)-3-{(S)-2-[(R)-2-(2-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(4-sulfooxy-phenyl)-propionylamino]-hexanoylamino}-acetylamino)-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-N-methyl-N-phenethyl-succinamic acid 281771 (S)-N-(1-Benzyl-2-phenyl-ethyl)-3-{(S)-2-[(R)-2-(2-{(S)-2-[(S)-2-tert-butoxycarbonylamino-3-(4-sulfooxy-phenyl)-propionylamino]-hexanoylamino}-acetylamino)-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-succinamic acid 281793 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzoic acid naphthalen-1-yl ester 281827 7-cyclopentyl-5-(3-methoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine 281829 7-cyclopentyl-5-(4-methoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine 281860 3-(4-amino-7-cyclopentyl-7H-pyrrolo[2,3-d]pyrimidin-5-yl)phenol 281861 4-(4-amino-7-cyclopentyl-7H-pyrrolo[2,3-d]pyrimidin-5-yl)phenol 281899 3-{4-Amino-7-[1-hydroxymethyl-2-(4-methoxy-phenyl)-ethyl]-7H-pyrrolo[2,3-d]pyrimidin-5-yl}-phenol 281925 {3-[4-Amino-5-(3-methoxy-phenyl)-pyrrolo[2,3-d]pyrimidin-7-yl]-cyclobutyl}-methanol 281926 3-(4-Amino-5-phenyl-pyrrolo[2,3-d]pyrimidin-7-yl)-cyclobutanol 281927 3-(4-Amino-5-phenyl-pyrrolo[2,3-d]pyrimidin-7-yl)-cyclopentanol 281928 3-(4-amino-7-cyclobutyl-7H-pyrrolo[2,3-d]pyrimidin-5-yl)phenol 281945 1-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-[3-(1H-tetrazol-5-ylamino)-phenyl]-urea 281973 1-{4-Methyl-3-[methyl-(1H-tetrazol-5-yl)-amino]-phenyl}-3-((R)-1-methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-urea 282005 1-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-[1-(1H-tetrazol-5-yl)-2,3-dihydro-1H-indol-6-yl]-urea 282097 (5-{[1-(2,5-Dihydroxy-phenyl)-meth-(E)-ylidene]-amino}-2-hydroxy-phenyl)-acetic acid 282116 1-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-[4-methyl-3-(1H-tetrazol-5-ylamino)-phenyl]-urea 282139 methyl 2-(4-(4-amino-5-(3-hydroxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)piperidin-1-yl)acetate 282182 7-cyclobutyl-5-(3-methoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine 282184 7-cyclobutyl-5-(4-methoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine 282204 3-[4-Amino-5-(4-methoxy-phenyl)-pyrrolo[2,3-d]pyrimidin-7-yl]-pyrrolidine-1-carboxylic acid tert-butyl ester 282205 4-(4-Amino-7-pyrrolidin-3-yl-7H-pyrrolo[2,3-d]pyrimidin-5-yl)-phenol 282224 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzoic acid 3,5-dimethyl-benzyl ester 282228 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzoic acid 4-isopropyl-benzyl ester 282244 2-((2-(4-(4-amino-5-(3-methoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)piperidin-1-yl)ethyl)(methyl)amino)ethanol 282256 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzoic acid 3-phenyl-butyl ester 282299 [5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-phenyl]-acetic acid ethyl ester 282301 [5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-phenyl]-acetic acid methyl ester 282302 [5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-phenyl]-acetic acid 282315 2-({3-[4-Amino-5-(3-methoxy-phenyl)-pyrrolo[2,3-d]pyrimidin-7-yl]-cyclobutylmethyl}-amino)-ethanol 282344 7-cyclopentyl-5-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine 282345 5,7-diphenyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine 282346 3-[4-Amino-5-(3-methoxy-phenyl)-pyrrolo[2,3-d]pyrimidin-7-yl]-cyclobutanecarboxylic acid (2-hydroxy-ethyl)-amide 282375 7-(1-(2-((2-methoxyethyl)(methyl)amino)ethyl)piperidin-4-yl)-5-(3-methoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine 282405 (S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(4-sulfooxy-phenyl)-propionylamino]-hexanoylamino}-acetylamino)-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-N-(2,2-diphenyl-ethyl)-succinamic acid 282428 (S)-3-{(R)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionyl]-6-[(Z)-3-(4-hydroxy-phenyl)-acryloylamino]-hexanoylamino}-N-((S)-1-carbamoyl-2-phenyl-ethyl)-succinamic acid 282429 (S)-3-[(R)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionyl]-6-(3-o-tolyl-ureido)-hexanoylamino]-N-((S)-1-carbamoyl-2-phenyl-ethyl)-N-methyl-succinamic acid 282433 (S)-3-{N'-[2-((3aS,7S)-2-tert-Butoxycarbonylamino-3-1H-indol-3-yl-propionylamino)-6-(3-o-tolyl-ureido)-hexyl]-hydrazino}-N-((S)-1-carbamoyl-2-phenyl-ethyl)-N-methyl-succinamic acid 282434 3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-6-[(S)-3-((1S,2S)-o-tolyl)-ureido]-hexanoylamino}-4-[N'-((S)-1-carbamoyl-2-phenyl-ethyl)-hydrazino]-butyric acid 282435 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzoic acid 3-phenyl-propyl ester 282436 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzoic acid phenethyl ester 282445 (S)-3-{(S)-2-[(R)-2-(2-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(4-sulfooxy-phenyl)-propionylamino]-hexanoylamino}-acetylamino)-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-N-(2,2-diphenyl-ethyl)-succinamic acid 282446 (S)-3-{(S)-2-[(R)-2-(2-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(4-sulfooxy-phenyl)-propionylamino]-hexanoylamino}-acetylamino)-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-N-phenethyl-succinamic acid 282482 2-(4-Amino-5-phenyl-pyrrolo[2,3-d]pyrimidin-7-yl)-3-phenyl-propan-1-ol 282487 (S)-3-{(S)-2-[(R)-2-(2-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(4-sulfooxy-phenyl)-propionylamino]-hexanoylamino}-acetylamino)-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-N-phenethyl-succinamic acid 282488 (S)-N-(1-Benzyl-2-phenyl-ethyl)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-butoxycarbonylamino-3-(4-sulfooxy-phenyl)-propionylamino]-hexanoylamino}-acetylamino)-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-succinamic acid 282498 1-((R)-5-Cyclohexyl-1-methyl-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-{4-methyl-3-[methyl-(1H-tetrazol-5-yl)-amino]-phenyl}-urea 282499 [5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzyl]-phosphonic acid diethyl ester 282500 N-Benzyloxy-2-[5-(2,5-dihydroxy-benzylamino)-2-hydroxy-phenyl]-acetamide 282501 (5-{[1-(2,5-Dihydroxy-phenyl)-meth-(E)-ylidene]-amino}-2-hydroxy-phenyl)-acetic acid methyl ester 282511 5-(2,5-Dihydroxy-benzylamino)-2,N-dihydroxy-benzamide 282512 [5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzyl]-phosphonic acid 282517 2-(4-Amino-5-phenyl-pyrrolo[2,3-d]pyrimidin-7-yl)-4-phenyl-butan-1-ol 282539 (5-{[1-(2,5-Dihydroxy-phenyl)-meth-(E)-ylidene]-amino}-2-hydroxy-phenyl)-acetic acid ethyl ester 282575 (S)-3-{N'-[(S)-2-{N'-[2-((S)-tert-Butoxycarbonylamino)-3-(1H-indol-3-yl)-propionyl]-hydrazino}-6-(3-o-tolyl-ureido)-hexyl]-hydrazino}-N-((S)-1-carbamoyl-2-phenyl-ethyl)-succinamic acid 282582 7-{1-[2-(2-Methoxy-ethylamino)-ethyl]-piperidin-4-yl}-5-(3-methoxy-phenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine 282584 (R)-4-[(R)-4-Amino-5-(4-hydroxy-phenyl)-pyrrolo[2,3-d]pyrimidin-7-yl]-2-ethoxycarbonylmethyl-pyrrolidine-1-carboxylic acid tert-butyl ester 282595 2-(4-(4-amino-5-(3-hydroxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)piperidin-1-yl)-N,N-dimethylacetamide 282602 N-tert-Butoxy-2-(5-{[1-(2,5-dihydroxy-phenyl)-meth-(E)-ylidene]-amino}-2-hydroxy-phenyl)-acetamide 282603 N-tert-Butoxy-5-(2,5-dihydroxy-benzylamino)-2-hydroxy-benzamide 282604 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzoic acid 3,7-dimethyl-octyl ester 282606 (S)-3-[(S)-2-[N'-((S)-2-tert-Butoxycarbonylamino-3-1H-indol-3-yl-propyl)-hydrazino]-6-(3-o-tolyl-ureido)-hexanoylamino]-N-((S)-1-carbamoyl-2-phenyl-ethyl)-succinamic acid 282626 2-(4-(4-amino-5-(3-methoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)piperidin-1-yl)acetamide 282627 methyl 2-(4-(4-amino-5-(3-methoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)piperidin-1-yl)acetate 282629 3-(4-amino-7-(1-(2-hydroxyethyl)piperidin-4-yl)-7H-pyrrolo[2,3-d]pyrimidin-5-yl)phenol 282631 2-(4-(4-amino-5-(3-hydroxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)piperidin-1-yl)acetamide 282650 (S)-3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-6-[(S)-3-((S)-4-hydroxy-phenyl)-acryloylamino]-hexanoylamino}-4-[N'-((S)-1-carbamoyl-2-phenyl-ethyl)-hydrazino]-butyric acid 282651 3-(N'-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-6-[(Z)-3-(4-hydroxy-phenyl)-acryloylamino]-hexyl}-hydrazino)-N-((S)-1-carbamoyl-2-phenyl-ethyl)-succinamic acid 282662 2-(4-(4-amino-5-(3-methoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)piperidin-1-yl)ethanol 282674 {(R)-4-[(S)-4-Amino-5-(4-hydroxy-phenyl)-pyrrolo[2,3-d]pyrimidin-7-yl]-pyrrolidin-2-yl}-acetic acid ethyl ester 282689 3-(N'-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-6-[(Z)-3-(4-hydroxy-phenyl)-acryloylamino]-hexyl}-hydrazino)-N-((S)-1-carbamoyl-2-phenyl-ethyl)-N-methyl-succinamic acid 282739 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzoic acid benzyl ester 282752 3-[4-Amino-5-(3-methoxy-phenyl)-pyrrolo[2,3-d]pyrimidin-7-yl]-pyrrolidine-1-carboxylic acid tert-butyl ester 282759 3-[4-Amino-5-(4-hydroxy-phenyl)-pyrrolo[2,3-d]pyrimidin-7-yl]-pyrrolidine-1-carboxylic acid tert-butyl ester 282768 N-Benzyloxy-5-(2,5-dihydroxy-benzylamino)-2-hydroxy-benzamide 282772 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzoic acid biphenyl-4-yl ester 282784 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzoic acid phenyl ester 282791 N-Benzyloxy-2-(5-{[1-(2,5-dihydroxy-phenyl)-meth-(E)-ylidene]-amino}-2-hydroxy-phenyl)-acetamide 282792 5-{[1-(2,5-Dihydroxy-phenyl)-meth-(E)-ylidene]-amino}-2-hydroxy-N-methoxy-benzamide 282820 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzoic acid 3,3-dimethyl-butyl ester 282824 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzoic acid tert-butyl ester 282825 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzoic acid ethyl ester 282862 3-(4-Amino-7-pyrrolidin-3-yl-7H-pyrrolo[2,3-d]pyrimidin-5-yl)-phenol 282890 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzoic acid cyclohexylmethyl ester 282897 3-[4-Amino-5-(3-hydroxy-phenyl)-pyrrolo[2,3-d]pyrimidin-7-yl]-pyrrolidine-1-carboxylic acid tert-butyl ester 282957 (S)-3-[(R)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionyl]-6-(3-o-tolyl-ureido)-hexanoylamino]-N-((S)-1-carbamoyl-2-phenyl-ethyl)-succinamic acid 283010 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzoic acid (E)-3-phenyl-allyl ester 283041 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzoic acid 2-methyl-3-phenyl-propyl ester 283043 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzoic acid 4-phenyl-butyl ester 283047 N-[3-(2'-Benzoylsulfamoyl-biphenyl-4-ylmethyl)-4-oxo-2-propyl-3,4-dihydro-quinazolin-6-yl]-benzamide 283085 N-{1-(8-Aza-spiro[4.5]decane-8-carbonyl)-3-[(E)-2-(4-methyl-piperazin-1-yl)-vinylcarbamoyl]-propyl}-3,5-dichloro-benzamide; compound with (Z)-but-2-enedioic acid 283175 (R)-4-[(R)-4-Amino-5-(4-hydroxy-phenyl)-pyrrolo[2,3-d]pyrimidin-7-yl]-2-hydroxymethyl-pyrrolidine-1-carboxylic acid tert-butyl ester 283179 5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-N-methoxy-benzamide 283212 (S)-3-{(R)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionyl]-6-[(Z)-3-(4-hydroxy-phenyl)-acryloylamino]-hexanoylamino}-N-((S)-1-carbamoyl-2-phenyl-ethyl)-N-methyl-succinamic acid 283246 3-{(S)-2-{N'-[(S)-2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propyl]-hydrazino}-6-[3-((S)-4-hydroxy-phenyl)-acryloylamino]-hexanoylamino}-N-(1-carbamoyl-2-phenyl-ethyl)-succinamic acid 283378 N-[1-(8-Aza-spiro[4.5]decane-8-carbonyl)-3-(2-dimethylamino-ethylcarbamoyl)-propyl]-3,5-dichloro-benzamide oxalic acid 283435 5-Dipentylcarbamoyl-5-[((R)-naphthalene-2-carbonyl)-amino]-pentanoic acid 283514 1-(4-Chloro-phenyl)-3-((R)-1-methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-urea 283516 N-[1-(8-Aza-spiro[4.5]decane-8-carbonyl)-3-(2-morpholin-4-yl-ethylcarbamoyl)-propyl]-3,5-dichloro-benzamide 283543 1-(4-Chloro-phenyl)-3-((S)-1-methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-urea 283868 (2-Chloro-5-methoxy-phenyl)-[6-methoxy-7-(4-methyl-piperazin-1-ylmethoxy)-quinazolin-4-yl]-amine 283888 (4aR,11bR)-4-Isobutyl-2,3,4a,5,6,8,9,11b-octahydro-4H-1,10-dioxa-4-aza-cyclopenta[b]phenanthrene 283889 (4aR,11bR)-4-Propyl-2,3,4a,5,6,8,9,11b-octahydro-4H-1,10-dioxa-4-aza-cyclopenta[b]phenanthrene 283995 (4aR,11bR)-2,3,4a,5,6,8,9,11b-Octahydro-4H-1,10-dioxa-4-aza-cyclopenta[b]phenanthrene 283996 (4aR,11bR)-4-Methyl-2,3,4a,5,6,8,9,11b-octahydro-4H-1,10-dioxa-4-aza-cyclopenta[b]phenanthrene 283997 (4aR,11bR)-4-Cyclopropylmethyl-2,3,4a,5,6,8,9,11b-octahydro-4H-1,10-dioxa-4-aza-cyclopenta[b]phenanthrene 284154 N-(5-chlorobenzo[d][1,3]dioxol-4-yl)-6-methoxy-7-((1-methylpiperidin-4-yl)methoxy)quinazolin-4-amine 284173 [2-Benzylcarbamoyl-1-(1H-indol-3-ylmethyl)-1-phenethylcarbamoyl-ethyl]-carbamic acid adamantan-2-yl ester 284174 [1-(1H-Indol-3-ylmethyl)-1-phenethylcarbamoyl-2-phenylcarbamoyl-ethyl]-carbamic acid adamantan-2-yl ester 284292 4-(4-{2-Amino-2-[(R)-1-(3-phenyl-propylcarbamoyl)-ethylcarbamoyl]-ethyl}-3,5-dimethyl-phenoxymethyl)-benzoic acid 284481 1-[19-Benzyl-13-carbamoylmethyl-22-(4-ethoxy-benzyl)-16-isopropyl-12,15,18,21,24-pentaoxo-7,8-dithia-11,14,17,20,23-pentaaza-spiro[5.19]pentacosane-10-carbonyl]-pyrrolidine-2-carboxylic acid (1-carbamoyl-4-guanidino-butyl)-amide 284522 2-Amino-3-[4-(4-cyano-benzyloxy)-2,6-dimethyl-phenyl]-N-[(R)-1-(3-phenyl-propylcarbamoyl)-ethyl]-propionamide 284604 N-Benzyl-2-phenoxy-nicotinamide 284741 N-{(S)-2-[(S)-2-(Adamantan-2-yloxycarbonylamino)-3-(1H-indol-3-yl)-2-methyl-propionylamino]-1-phenyl-ethyl}-succinamic acid 284742 N-{(S)-2-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1H-indol-3-yl)-2-methyl-propionylamino]-3-phenyl-propyl}-succinamic acid 284851 N-{(R)-2-[(S)-2-(Adamantan-2-yloxycarbonylamino)-3-(1H-indol-3-yl)-2-methyl-propionylamino]-3-phenyl-propyl}-succinamic acid 284883 2-Amino-3-[4-(4-fluoro-benzyloxy)-2,6-dimethyl-phenyl]-N-[(R)-1-(3-phenyl-propylcarbamoyl)-ethyl]-propionamide 285017 [1-(1H-Indol-3-ylmethyl)-1-phenethylcarbamoyl-2-(3-phenyl-propylcarbamoyl)-ethyl]-carbamic acid adamantan-2-yl ester 285018 [2-[2-(4-Hydroxy-phenyl)-ethylcarbamoyl]-1-(1H-indol-3-ylmethyl)-1-phenethylcarbamoyl-ethyl]-carbamic acid adamantan-2-yl ester 285019 [1-[2-(4-Hydroxy-phenyl)-ethylcarbamoyl]-1-(1H-indol-3-ylmethyl)-2-phenethylcarbamoyl-ethyl]-carbamic acid adamantan-2-yl ester 285021 {1-(1H-Indol-3-ylmethyl)-1-phenethylcarbamoyl-2-[2-(4-sulfooxy-phenyl)-ethylcarbamoyl]-ethyl}-carbamic acid adamantan-2-yl ester 285083 N-{(R)-2-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1H-indol-3-yl)-2-methyl-propionylamino]-3-phenyl-propyl}-succinamic acid 285325 2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-2-methyl-N-[(R)-1-(3-phenyl-propylcarbamoyl)-ethyl]-propionamide 285327 2-Amino-3-[2,6-dimethyl-4-(4-nitro-benzyloxy)-phenyl]-N-[(R)-1-(3-phenyl-propylcarbamoyl)-ethyl]-propionamide 285350 {1-(1H-Indol-3-ylmethyl)-2-phenethylcarbamoyl-1-[2-(4-sulfooxy-phenyl)-ethylcarbamoyl]-ethyl}-carbamic acid adamantan-2-yl ester 285372 2-(2-{4-[4-(4-tert-Butyl-phenylamino)-phenoxy]-6-methoxy-quinolin-7-yloxy}-ethylamino)-ethanol 285459 [1-(1H-Indol-3-ylmethyl)-1,2-bis-phenethylcarbamoyl-ethyl]-carbamic acid adamantan-2-yl ester 285535 N-{(S)-2-[(S)-2-(Adamantan-2-yloxycarbonylamino)-3-(1H-indol-3-yl)-2-methyl-propionylamino]-3-phenyl-propyl}-succinamic acid 285679 (4aR,11bR)-4-Propyl-1,2,3,4,4a,5,6,8,9,11b-decahydro-10-oxa-4-aza-cyclopenta[b]phenanthrene 285680 (4aR,11bR)-4-Propyl-3,4,4a,8,9,11b-hexahydro-2H,5H-1,6,10-trioxa-4-aza-cyclopenta[b]phenanthrene 286002 2-(5-Thiophen-2-yl-1H-indol-3-yl)-ethylamine 286003 Dimethyl-[2-(5-thiophen-2-yl-1H-indol-3-yl)-ethyl]-amine 286009 Dimethyl-[2-(5-thiophen-3-yl-1H-indol-3-yl)-ethyl]-amine 286049 3-(6-Methoxy-pyridin-3-yl)-7-phenyl-imidazo[1,2-a]pyridine 286117 {2-[5-(5-Chloro-thiophen-2-yl)-1H-indol-3-yl]-ethyl}-dimethyl-amine 286161 3-(Adamantan-2-yloxycarbonylamino)-3-(1H-indol-3-ylmethyl)-N-phenethyl-succinamic acid benzyl ester 286180 4-[2-(5,5-Dimethyl-hex-1-ynyl)-cyclopropyl]-1H-imidazole 286725 2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-N-[(R)-1-(3-phenyl-propylcarbamoyl)-ethyl]-propionamide 286755 1-[3-(3-Dimethylaminomethyl-piperidin-1-yl)-propyl]-4-(3-phenyl-imidazo[1,2-a]pyridin-7-yl)-1H-pyridin-2-one 286756 1-{3-[(2-Methoxy-ethyl)-methyl-amino]-propyl}-4-(3-phenyl-imidazo[1,2-a]pyridin-7-yl)-1H-pyridin-2-one 286831 3-(4-Allyloxy-2,6-dimethyl-phenyl)-2-amino-N-[(R)-1-(3-phenyl-propylcarbamoyl)-ethyl]-propionamide 286834 2-Amino-3-(4-methoxy-2,6-dimethyl-phenyl)-N-[(R)-1-(3-phenyl-propylcarbamoyl)-ethyl]-propionamide 286960 2-Amino-N-cyclopropylmethyl-3-(4-hydroxy-2,6-dimethyl-phenyl)-N-[(R)-1-(3-phenyl-propylcarbamoyl)-ethyl]-propionamide 286980 4-[4-(3-Phenyl-imidazo[1,2-a]pyridin-7-yl)-benzyl]-piperazine-1-carboxylic acid methylamide 287441 (3S,3aR,4R,4aS,8aR,9aS)-4-[2-((2R,6S)-1,6-Dimethyl-piperidin-2-yl)-ethyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 287505 3-[2-(2,5-Dimethyl-pyrrolidin-1-yl)-ethyl]-5-thiophen-2-yl-1H-indole 287513 3-(2-Pyrrolidin-1-yl-ethyl)-5-thiophen-2-yl-1H-indole 287530 Cyclohexyl-[3-[4-(2-ethyl-5-phenethyl-2H-pyrazol-3-yl)-piperidin-1-ylmethyl]-4-(3-fluoro-phenyl)-pyrrolidin-1-yl]-acetic acid 287531 (R)-2-((3S,4S)-3-((4-(3-benzyl-1-ethyl-1H-pyrazol-5-yl)piperidin-1-yl)methyl)-4-(3-fluorophenyl)pyrrolidin-1-yl)-3-cyclobutylpropanoic acid 287552 (3-Bromo-phenyl)-(1,3,5,8-tetraaza-anthracen-4-yl)-amine 287561 3-p-Tolyloxymethyl-thiophene-2-sulfonic acid (4-bromo-3-methyl-isoxazol-5-yl)-amide 287612 Dimethyl-{2-[5-(5-methyl-thiophen-2-yl)-1H-indol-3-yl]-ethyl}-amine 287618 5-(5-Chloro-thiophen-2-yl)-3-(2-pyrrolidin-1-yl-ethyl)-1H-indole 287619 3-[2-(2,5-Dihydro-pyrrol-1-yl)-ethyl]-5-thiophen-2-yl-1H-indole 287629 3-[2-((S)-2-Methoxymethyl-pyrrolidin-1-yl)-ethyl]-5-thiophen-2-yl-1H-indole 287630 {(S)-1-[2-(5-Thiophen-2-yl-1H-indol-3-yl)-ethyl]-pyrrolidin-2-yl}-methanol 287653 (R)-2-((3S,4S)-3-((4-(3-benzyl-1-ethyl-1H-pyrazol-5-yl)piperidin-1-yl)methyl)-4-(3-fluorophenyl)pyrrolidin-1-yl)-3-methylbutanoic acid 287685 2-(2,4,6-Trimethyl-phenoxymethyl)-thiophene-3-sulfonic acid (4-bromo-3-methyl-isoxazol-5-yl)-amide 287695 (R)-2-((3S,4S)-3-((4-(3-benzyl-1-ethyl-1H-pyrazol-5-yl)piperidin-1-yl)methyl)-4-(3-fluorophenyl)pyrrolidin-1-yl)-3-ethylpentanoic acid 287698 N-[4-[4-(Acetylamino-methyl)-4-phenyl-piperidin-1-yl]-2-(3,4-dichloro-phenyl)-butyl]-N-methyl-benzamide 287728 N-{3-[2-Amino-3-cyano-6-(2-hydroxy-phenyl)-pyridin-4-yl]-phenyl}-3-piperidin-1-yl-propionamide 287789 (3-{4-[5-(4-Cyano-phenyl)-2H-pyrazol-3-yl]-piperidin-1-ylmethyl}-4-phenyl-pyrrolidin-1-yl)-cyclohexyl-acetic acid 287801 2-(2,4-Dimethyl-phenoxymethyl)-thiophene-3-sulfonic acid (4-bromo-3-methyl-isoxazol-5-yl)-amide 287808 7-{3,5-Dihydroxy-2-[3-hydroxy-4-(thiazol-2-ylsulfanyl)-butyl]-cyclopentyl}-heptanoic acid 287809 7-{2-[4-(3-Chloro-phenylsulfanyl)-3-hydroxy-butyl]-3,5-dihydroxy-cyclopentyl}-heptanoic acid 287907 3-(2,4-Dimethyl-phenoxymethyl)-thiophene-2-sulfonic acid (4-bromo-3-methyl-isoxazol-5-yl)-amide 287916 Acetic acid 1-[4-(benzoyl-methyl-amino)-3-(3,4-dichloro-phenyl)-butyl]-4-phenyl-piperidin-4-yl ester 287918 (2R,3S)-2-[(2S,3S)-3-[4-(5-Benzyl-2-ethyl-2H-pyrazol-3-yl)-piperidin-1-ylmethyl]-4-(3-fluoro-phenyl)-pyrrolidin-1-yl]-3-methyl-pentanoic acid 287949 2-morpholino-4H-chromen-4-one 288020 Cyclohexyl-{3-[4-(4-phenethyl-2-propyl-2H-pyrazol-3-yl)-piperidin-1-ylmethyl]-4-phenyl-pyrrolidin-1-yl}-acetic acid 288021 Cyclohexyl-{3-[4-(2-methyl-4-phenethyl-2H-pyrazol-3-yl)-piperidin-1-ylmethyl]-4-phenyl-pyrrolidin-1-yl}-acetic acid 288029 3-(Benzo[1,3]dioxol-5-yloxymethyl)-thiophene-2-sulfonic acid (4-bromo-3-methyl-isoxazol-5-yl)-amide 288054 (R)-2-((3S,4S)-3-((4-(3-benzyl-1-ethyl-1H-pyrazol-5-yl)piperidin-1-yl)methyl)-4-phenylpyrrolidin-1-yl)-2-cyclobutylacetic acid 288080 4-(3-Phenyl-imidazo[1,2-a]pyridin-7-yl)-1-(3-piperidin-1-yl-propyl)-1H-pyridin-2-one 288147 (3-Bromo-phenyl)-(2-methyl-1H-imidazo[4,5-g]quinazolin-8-yl)-amine 288249 Cyclohexyl-[3-[4-(2-ethyl-5-naphthalen-1-yl-2H-pyrazol-3-yl)-piperidin-1-ylmethyl]-4-(3-fluoro-phenyl)-pyrrolidin-1-yl]-acetic acid 288250 Cyclohexyl-{3-[4-(5-naphthalen-1-yl-2H-pyrazol-3-yl)-piperidin-1-ylmethyl]-4-phenyl-pyrrolidin-1-yl}-acetic acid 288297 5-Oxo-tetrahydro-furan-2-carboxylic acid {3-[2-amino-3-cyano-6-(2-hydroxy-phenyl)-pyridin-4-yl]-phenyl}-amide 288503 7-{3,5-Dihydroxy-2-[3-hydroxy-4-(thiophen-2-ylsulfanyl)-butyl]-cyclopentyl}-heptanoic acid 288552 7-[4-(4-Methanesulfonyl-piperazin-1-ylmethyl)-phenyl]-3-phenyl-imidazo[1,2-a]pyridine 288571 N-[2-(3,4-Dichloro-phenyl)-4-(4-hydroxymethyl-4-phenyl-piperidin-1-yl)-butyl]-N-methyl-benzamide 288629 7-{2-[4-(3-Fluoro-phenylsulfanyl)-3-hydroxy-butyl]-3,5-dihydroxy-cyclopentyl}-heptanoic acid 288632 2-(Benzo[1,3]dioxol-5-yloxymethyl)-thiophene-3-sulfonic acid (4-bromo-3-methyl-isoxazol-5-yl)-amide 288635 Cyclohexyl-(3-(3-fluoro-phenyl)-4-{4-[5-(4-methoxy-phenyl)-2H-pyrazol-3-yl]-piperidin-1-ylmethyl}-pyrrolidin-1-yl)-acetic acid 288636 [3-{4-[5-(4-Chloro-phenyl)-2H-pyrazol-3-yl]-piperidin-1-ylmethyl}-4-(3-fluoro-phenyl)-pyrrolidin-1-yl]-cyclohexyl-acetic acid 288637 Cyclohexyl-[3-{4-[5-(2,4-dichloro-phenyl)-2H-pyrazol-3-yl]-piperidin-1-ylmethyl}-4-(3-fluoro-phenyl)-pyrrolidin-1-yl]-acetic acid 288643 2-(6-Chloro-benzo[1,3]dioxol-5-yloxymethyl)-thiophene-3-sulfonic acid (4-bromo-3-methyl-isoxazol-5-yl)-amide 288681 1-{4-[4-(3-Phenyl-imidazo[1,2-a]pyridin-7-yl)-benzyl]-piperazin-1-yl}-ethanone 288714 (3-Bromo-phenyl)-(1H-pyrazolo[3,4-g]quinazolin-8-yl)-amine 288833 (3-Bromo-phenyl)-(1H-1,2,3,5,7-pentaaza-cyclopenta[b]naphthalen-8-yl)-amine 288954 (3-Bromo-phenyl)-[9-chloro-3-(2-dimethylamino-ethyl)-3H-imidazo[4,5-g]quinazolin-8-yl]-amine 289042 Macrocyclic Quinazolinone analogue 289043 Macrocyclic Quinazolinone analogue 289044 Macrocyclic Quinazolinone analogue 289161 Macrocyclic Quinazolinone analogue 289207 7-[3,5-Dihydroxy-2-(3-hydroxy-4-phenoxy-butyl)-cyclopentyl]-heptanoic acid 289213 Thiophene-2-carboxylic acid [2-(3,4-dichloro-phenyl)-4-(4-hydroxy-4-phenyl-piperidin-1-yl)-butyl]-methyl-amide 289239 2-(6-Propyl-benzo[1,3]dioxol-5-yloxymethyl)-thiophene-3-sulfonic acid (4-bromo-3-methyl-isoxazol-5-yl)-amide 289306 ethyl 4-(4-amino-7-phenyl-7H-pyrrolo[2,3-d]pyrimidin-5-yl)benzoate 289323 7-[3,5-Dihydroxy-2-(3-hydroxy-4-phenylamino-butyl)-cyclopentyl]-heptanoic acid 289324 7-[3,5-Dihydroxy-2-(3-hydroxy-4-phenylsulfanyl-butyl)-cyclopentyl]-heptanoic acid 289336 N-[2-(3,4-Dichloro-phenyl)-4-(4-ethoxy-4-phenyl-piperidin-1-yl)-butyl]-N-methyl-benzamide 289384 2-p-Tolyloxymethyl-thiophene-3-sulfonic acid (4-bromo-3-methyl-isoxazol-5-yl)-amide 289405 (3-(4-amino-5-phenyl-7H-pyrrolo[2,3-d]pyrimidin-7-yl)phenyl)methanol 289406 (2-(4-amino-5-phenyl-7H-pyrrolo[2,3-d]pyrimidin-7-yl)phenyl)methanol 289481 Dodecanoic acid (3S,3aR,8R,8aS)-3-hydroxymethyl-8-isopropyl-8-methyl-1-oxo-1,2,3,3a,8,8a-hexahydro-indeno[1,2-c]pyrrol-6-yl ester 289654 (2R,3R)-2-[(2S,3S)-3-[4-(5-Benzyl-2-ethyl-2H-pyrazol-3-yl)-piperidin-1-ylmethyl]-4-(3-fluoro-phenyl)-pyrrolidin-1-yl]-3-methyl-pentanoic acid 289655 (R)-2-((3S,4S)-3-((4-(3-benzyl-1-ethyl-1H-pyrazol-5-yl)piperidin-1-yl)methyl)-4-(3-fluorophenyl)pyrrolidin-1-yl)-3,3-dimethylbutanoic acid 289658 (3-Bromo-phenyl)-(3-methyl-3H-imidazo[4,5-g]quinazolin-8-yl)-amine 289674 (4-(4-amino-5-phenyl-7H-pyrrolo[2,3-d]pyrimidin-7-yl)phenyl)methanol 289682 2-[3-[4-(5-Benzyl-2-ethyl-2H-pyrazol-3-yl)-piperidin-1-ylmethyl]-4-(3-fluoro-phenyl)-pyrrolidin-1-yl]-2,3-dimethyl-butyric acid 289683 (R)-[(2S,3S)-3-[4-(5-Benzyl-2-ethyl-2H-pyrazol-3-yl)-piperidin-1-ylmethyl]-4-(3-fluoro-phenyl)-pyrrolidin-1-yl]-cyclohexyl-acetic acid 289684 (R)-2-((3S,4S)-3-((4-(3-benzyl-1-ethyl-1H-pyrazol-5-yl)piperidin-1-yl)methyl)-4-phenylpyrrolidin-1-yl)-2-cyclohexylacetic acid 289721 1-(4-Fluoro-phenyl)-4-[4-(1,2,3,4-tetrahydro-naphthalen-1-yl)-piperazin-1-yl]-butan-1-one 289750 Dodecanoic acid (3S,3aR,8S,8aS)-3-hydroxymethyl-8-isopropyl-8-methyl-1-oxo-1,2,3,3a,8,8a-hexahydro-indeno[1,2-c]pyrrol-6-yl ester 289865 (7,8-Dihydroxy-4-propyl-1,2,3,4,4a,5,6,10b-octahydro-benzo[f]quinolin-2-yl)-acetonitrile 289872 2-Methyl-4-propyl-1,2,3,4,4a,5,6,10b-octahydro-benzo[f]quinolin-9-ol 289918 3-(6-Propyl-benzo[1,3]dioxol-5-yloxymethyl)-thiophene-2-sulfonic acid (4-bromo-3-methyl-isoxazol-5-yl)-amide 289919 3-(2,4,6-Trimethyl-phenoxymethyl)-thiophene-2-sulfonic acid (4-bromo-3-methyl-isoxazol-5-yl)-amide 289960 (3S,3aR,8R,8aS)-6-Dec-1-ynyl-3-hydroxymethyl-8-isopropyl-8-methyl-3,3a,8,8a-tetrahydro-2H-indeno[1,2-c]pyrrol-1-one 290009 (6aR,9R)-7-Methyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid (1-methyl-pentyl)-amide 290048 Cyclohexyl-{3-[4-(4-phenethyl-1-propyl-1H-pyrazol-3-yl)-piperidin-1-ylmethyl]-4-phenyl-pyrrolidin-1-yl}-acetic acid 290058 2-[3-[4-(5-Benzyl-2-ethyl-2H-pyrazol-3-yl)-piperidin-1-ylmethyl]-4-(3-fluoro-phenyl)-pyrrolidin-1-yl]-2,3-dimethyl-butyric acid 290089 4-Chloro-N-{2-[4-(1,2,3,4-tetrahydro-naphthalen-1-yl)-piperazin-1-yl]-ethyl}-benzamide 290165 (6aR,9R)-7-Methyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid (1-methyl-hexyl)-amide 290180 4-chloro-5,7-diphenyl-7H-pyrrolo[2,3-d]pyrimidine 290202 N-{4-Oxo-2-propyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-3,4-dihydro-quinazolin-6-yl}-benzamide 290203 N-[3-(2'-Benzoylsulfamoyl-biphenyl-4-ylmethyl)-4-oxo-2-propyl-3,4-dihydro-quinazolin-6-yl]-N-pentyl-benzamide 290204 4'-[6-(3-Isopropyl-ureido)-4-oxo-2-propyl-4H-quinazolin-3-ylmethyl]-biphenyl-2-sulfonic acid acetyl-amide 290212 8-Adamantan-1-yl-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 290345 Cyclohexyl-{3-[4-(1-methyl-4-phenethyl-1H-pyrazol-3-yl)-piperidin-1-ylmethyl]-4-phenyl-pyrrolidin-1-yl}-acetic acid 290349 7-{3,5-Dihydroxy-2-[3-hydroxy-4-(3-trifluoromethyl-phenylsulfanyl)-butyl]-cyclopentyl}-heptanoic acid 290462 2-(4-(4-amino-5-(3-methoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzylamino)ethanol 290463 2-(4-(4-amino-5-phenyl-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzylamino)ethanol 290466 (6aR,9R)-7-Methyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid (1-methyl-butyl)-amide 290471 5,7-diphenyl-3H-pyrrolo[2,3-d]pyrimidin-4(7H)-one 290482 (3-Bromo-phenyl)-(1-methyl-1H-imidazo[4,5-g]quinazolin-8-yl)-amine 290483 (3-Bromo-phenyl)-(1-thia-3,5,7-triaza-cyclopenta[b]naphthalen-8-yl)-amine 290489 7-[3,5-Dihydroxy-2-(3-hydroxy-4-m-tolylsulfanyl-butyl)-cyclopentyl]-heptanoic acid 290634 2-(2-(4-amino-5-phenyl-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzylamino)ethanol 290694 4-[6-(3-Chloro-phenylamino)-9-ethyl-9H-purin-2-ylamino]-cyclohexanol 290728 5-(3-chlorophenyl)-7-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine 290729 5-(3-methoxyphenyl)-7-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine 290769 1-{4-[2-(1H-Imidazol-4-yl)-ethylsulfanyl]-phenyl}-ethanone 290801 (3-(4-amino-5-(3-methoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)phenyl)methanol 290845 (6aR,9R)-7-Methyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid ((R)-1-methyl-pentyl)-amide 290857 3-(1-Methyl-1H-indol-3-ylmethylene)-1,3-dihydro-pyrrolo[2,3-b]pyridin-2-one 290923 1-{4-[3-(1H-Imidazol-4-yl)-propylsulfanyl]-phenyl}-ethanone 290951 (3-Bromo-phenyl)-[3-(2-dimethylamino-ethyl)-3H-imidazo[4,5-g]quinazolin-8-yl]-amine 290960 (3-Bromo-phenyl)-[1-(2-dimethylamino-ethyl)-1H-imidazo[4,5-g]quinazolin-8-yl]-amine 290987 Macrocyclic Quinazolinone analogue 290988 Macrocyclic Quinazolinone analogue 290989 4'-[6-(3-Isopropyl-ureido)-4-oxo-2-propyl-4H-quinazolin-3-ylmethyl]-biphenyl-2-sulfonic acid benzoylamide 291034 4-Fluoro-N-{2-[4-(1,2,3,4-tetrahydro-naphthalen-1-yl)-piperazin-1-yl]-ethyl}-benzamide 291139 Thiophene-3-carboxylic acid [2-(3,4-dichloro-phenyl)-4-(4-hydroxy-4-phenyl-piperidin-1-yl)-butyl]-methyl-amide 291140 (R)-2-((3S,4S)-3-((4-(3-benzyl-1-ethyl-1H-pyrazol-5-yl)piperidin-1-yl)methyl)-4-(3-fluorophenyl)pyrrolidin-1-yl)-3-cyclopropylpropanoic acid 291154 4-[3-(4-Methoxy-phenoxy)-propyl]-1H-imidazole 291250 2-(3-(4-amino-5-phenyl-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzylamino)ethanol 291268 Naphthalene-1-carboxylic acid [2-(3,4-dichloro-phenyl)-4-(4-hydroxy-4-phenyl-piperidin-1-yl)-butyl]-methyl-amide 291273 Acetic acid 1-{3-(3,4-dichloro-phenyl)-4-[ethyl-(thiophene-2-carbonyl)-amino]-butyl}-4-phenyl-piperidin-4-yl ester 291582 (R) 3-Bromo-N-[1-(4-fluoro-benzyl)-pyrrolidin-2-ylmethyl]-2-hydroxy-5,6-dimethoxy-benzamide 291621 7-[3-(Hexane-1-sulfinylmethyl)-7-oxa-bicyclo[2.2.1]hept-2-yl]-hept-5-enoic acid 291623 [1-(4-Fluoro-phenyl)-4-methyl-2,3-dihydro-1H-indol-3-ylmethyl]-dimethyl-amine 291645 (R) N-(1-Benzyl-pyrrolidin-2-ylmethyl)-5-bromo-2,3-dimethoxy-benzamide 291646 N-{2-[4-(1,2,3,4-Tetrahydro-naphthalen-1-yl)-piperazin-1-yl]-ethyl}-benzamide 291691 5-Methyl-2-{(R)-2-(1-methyl-1H-indol-3-yl)-1-[(S)-4-methyl-2-(3-pyridin-2-yl-ureido)-pentanoylamino]-ethyl}-oxazole-4-carboxylic acid 291723 N-[(R)-2-(1H-Indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-4-trifluoromethoxy-benzamidine 291729 1-tert-Butyl-3-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-urea 291736 2-(4-Diethylamino-but-2-ynyl)-isoindole-1,3-dione 291737 1-(4-diethylamino-2-butynyl)spiro[tetrahydro-1H-imidazole-4,1'-(2',3'-dihydro-1'H-indene)]-2,5-dione 291773 3,5-Dichloro-N-(1-ethyl-pyrrolidin-2-ylmethyl)-2,6-dimethoxy-benzamide 291817 [5-(4-{4-[(R)-2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzyl)-2,4-dioxo-thiazolidin-3-yl]-acetic acid 291847 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (S)-3-(4-hydroxy-benzoylamino)-azepan-4-yl ester 291899 5-Bromo-3-(5-bromo-6-hydroxy-2'-methoxy-biphenyl-3-ylmethylene)-1,3-dihydro-pyrrolo[2,3-b]pyridin-2-one 291954 N-[(R)-2-(1H-Indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-2-(3-trifluoromethyl-phenyl)-acetamide 291960 2-(1-(2-(2,3-dihydrobenzofuran-5-yl)ethyl)pyrrolidin-3-yl)-2,2-diphenylacetamide 291966 5-Methyl-2-{(R)-2-(1-methyl-1H-indol-3-yl)-1-[(S)-4-methyl-2-(3-phenyl-ureido)-pentanoylamino]-ethyl}-1H-imidazole-4-carboxylic acid 291967 5-Methyl-2-((R)-2-(1-methyl-1H-indol-3-yl)-1-{(S)-4-methyl-2-[(1-oxa-4-aza-spiro[4.5]decane-4-carbonyl)-amino]-pentanoylamino}-ethyl)-oxazole-4-carboxylic acid 291993 2-[(R)-1-[(S)-2-(3-Benzyl-ureido)-4-methyl-pentanoylamino]-2-(1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid 291994 Azepane-1-carboxylic acid {(S)-1-[(R)-2-(1H-indol-3-yl)-1-(5-methyl-4-methylcarbamoyl-oxazol-2-yl)-ethylcarbamoyl]-3-methyl-butyl}-amide 292032 5-Methyl-2-((R)-2-(1-methyl-1H-indol-3-yl)-1-{(S)-4-methyl-2-[3-(2-methyl-cyclohexyl)-ureido]-pentanoylamino}-ethyl)-1H-imidazole-4-carboxylic acid 292116 N-[(R)-2-(1H-Indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-benzamidine 292129 13-(2-Amino-ethyl)-19-benzyl-22-(4-ethoxy-benzyl)-16-isopropyl-12,15,18,21,24-pentaoxo-7,8-dithia-11,14,17,20,23-pentaaza-spiro[5.19]pentacosane-10-carboxylic acid (1-carbamoyl-4-guanidino-butyl)-amide 292130 (2-{[13-(2-Amino-ethyl)-19-benzyl-22-(4-ethoxy-benzyl)-16-isopropyl-12,15,18,21,24-pentaoxo-7,8-dithia-11,14,17,20,23-pentaaza-spiro[5.19]pentacosane-10-carbonyl]-amino}-5-guanidino-pentanoylamino)-acetic acid 292253 N-[(R)-2-(1H-Indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-acetamidine 292261 1-(4-Fluoro-phenyl)-4-methyl-3,4,5,6-tetrahydro-1H-azepino[3,4,5-cd]indole 292301 2-[(R)-1-[(S)-2-(3-Adamantan-1-yl-ureido)-4-methyl-pentanoylamino]-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid 292346 2-Methylsulfanylmethyl-4-propyl-1,2,3,4,4a,5,6,10b-octahydro-benzo[f]quinoline-7,8-diol 292347 7-Phenyl-5-o-tolyl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine 292353 2-Methylsulfanylmethyl-4-propyl-1,2,3,4,4a,5,6,10b-octahydro-benzo[f]quinoline-8,9-diol 292354 5-(4-methoxyphenyl)-7-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine 292372 (8,9-Dihydroxy-4-propyl-1,2,3,4,4a,5,6,10b-octahydro-benzo[f]quinolin-2-yl)-acetonitrile 292408 4-tert-Butyl-N-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-benzamidine 292411 (endo)-7-(3-Heptylsulfanyl-7-oxa-bicyclo[2.2.1]hept-2-yl)-hept-5-enoic acid 292542 N-(1-Cyclohexylmethyl-piperidin-3-ylmethyl)-4-[2-(3,3,3-triphenyl-propionylamino)-acetylamino]-butyramide 292571 7-[3-(3-Phenyl-propylsulfanylmethyl)-7-oxa-bicyclo[2.2.1]hept-2-yl]-hept-5-enoic acid 292572 (E)7-(3-Hex-3-enylsulfanylmethyl-7-oxa-bicyclo[2.2.1]hept-2-yl)-hept-5-enoic acid 292631 (6aR,9R)-7-Methyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid (R)-sec-butylamide 292718 5-Methyl-2-((R)-2-(1-methyl-1H-indol-3-yl)-1-{(S)-4-methyl-2-[3-(4-methyl-cyclohexyl)-ureido]-pentanoylamino}-ethyl)-1H-imidazole-4-carboxylic acid 292755 (6aR,9R)-7-Methyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid ((R)-1-methyl-hexyl)-amide 292763 (6aR,9R)-7-Methyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid ((R)-1-methyl-butyl)-amide 292764 (6aR,9R)-7-Methyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid (1-ethyl-propyl)-amide 292777 2-(4-(4-amino-5-(3-methoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)phenyl)-N-(2-hydroxyethyl)acetamide 292844 (E)-7-(3-Hex-2-enylsulfanylmethyl-7-oxa-bicyclo[2.2.1]hept-2-yl)-hept-5-enoic acid 292854 5-Methyl-2-((R)-2-(1-methyl-1H-indol-3-yl)-1-{(S)-4-methyl-2-[3-(1,2,3,4-tetrahydro-naphthalen-1-yl)-ureido]-pentanoylamino}-ethyl)-oxazole-4-carboxylic acid 292856 2-[(R)-1-[(S)-2-(3-Cyclopentyl-ureido)-4-methyl-pentanoylamino]-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid 292863 5-Methyl-2-((R)-2-(1-methyl-1H-indol-3-yl)-1-{(S)-4-methyl-2-[3-(3-methyl-cyclohexyl)-ureido]-pentanoylamino}-ethyl)-1H-imidazole-4-carboxylic acid 292963 9-(4-Methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f]azulene 292968 1-(4-Fluoro-phenyl)-4-methyl-2,2a,3,4,5,6-hexahydro-1H-azepino[3,4,5-cd]indole 292969 1-(4-Fluoro-phenyl)-2,2a,3,4,5,6-hexahydro-1H-azepino[3,4,5-cd]indole 292981 7-[3-(2-Hydroxy-hexylsulfanylmethyl)-7-oxa-bicyclo[2.2.1]hept-2-yl]-hept-5-enoic acid 293058 benzyl 2-[1-[1-[1-amino-2-carbamoyl-(1S)-ethylcarboxamido]-2-methyl-(1S)-propylcarboxamido]-2-phenyl-(1S)-ethylcarboxamido]-(2S)-propanoate 293061 benzyl 2-[1-[1-[1-[1-amino-2-hydroxy-(1S)-ethylcarboxamido]-2-carbamoyl-(1S)-ethylcarboxamido]-2-methyl-(1S)-propylcarboxamido]-2-phenyl-(1S)-ethylcarboxamido]-(2S)-propanoate 293062 benzyl 2-[1-[1-amino-2-methyl-(1S)-propylcarboxamido]-2-phenyl-(1S)-ethylcarboxamido]-(2S)-propanoate 293101 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (1R,2R)-1-(4-hydroxy-benzoylamino)-indan-2-yl ester 293107 7-Chloro-9-(4-methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f]azulene 293117 (S)-7-[3-(1-Methyl-hexylsulfanylmethyl)-7-oxa-bicyclo[2.2.1]hept-2-yl]-hept-5-enoic acid 293118 7-(3-Cyclohexylmethylsulfanylmethyl-7-oxa-bicyclo[2.2.1]hept-2-yl)-hept-5-enoic acid 293159 2-[(R)-1-[(S)-2-(3-Cycloheptyl-ureido)-4-methyl-pentanoylamino]-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid 293242 N-{2-[(1-Cyclohexylmethyl-piperidin-3-ylmethyl)-carbamoyl]-ethyl}-4-(3,3,3-triphenyl-propionylamino)-butyramide 293248 2-[(R)-1-[(S)-2-(3-Cyclopentyl-ureido)-4-methyl-pentanoylamino]-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-1H-imidazole-4-carboxylic acid 293266 7-(3-Ethylsulfanylmethyl-7-oxa-bicyclo[2.2.1]hept-2-yl)-hept-5-enoic acid 293267 7-(3-Butylsulfanylmethylsulfanylmethyl-7-oxa-bicyclo[2.2.1]hept-2-yl)-hept-5-enoic acid 293281 7-(3-Methylsulfanylmethyl-7-oxa-bicyclo[2.2.1]hept-2-yl)-hept-5-enoic acid 293285 1-(4-Diethylamino-but-2-ynyl)-3,3-diphenyl-pyrrolidine-2,5-dione 293299 5-Methyl-2-((R)-2-(1-methyl-1H-indol-3-yl)-1-{(S)-4-methyl-2-[3-(1-methyl-cyclohexyl)-ureido]-pentanoylamino}-ethyl)-oxazole-4-carboxylic acid 293300 2-[(R)-1-{(S)-2-[(3,4-Dihydro-2H-quinoline-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid 293301 2-[(R)-1-{(S)-2-[(Indole-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid 293346 (R) 3-Bromo-N-[1-(4-fluoro-benzyl)-pyrrolidin-2-ylmethyl]-2-hydroxy-6-methoxy-benzamide 293377 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (R)-2-(4-hydroxy-benzoylamino)-indan-1-yl ester 293378 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (R)-2-(4-hydroxy-benzoylamino)-cyclopentyl ester 293402 7-[3-(2-Phenoxy-ethylsulfanylmethyl)-7-oxa-bicyclo[2.2.1]hept-2-yl]-hept-5-enoic acid 293417 1-(4-Diisopropylamino-but-2-ynyl)-3,3-diphenyl-pyrrolidine-2,5-dione 293424 1-(4-Diethylamino-but-2-ynyl)-3-phenyl-pyrrolidine-2,5-dione 293462 1-{4-[4-(1H-Imidazol-4-yl)-butoxy]-phenyl}-ethanone 293501 [(R)-2-(1H-Indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-carbamic acid tert-butyl ester 293502 (R)-2-(1H-Indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethylamine 293515 2-[(R)-1-[(S)-2-(3-Cyclohexyl-ureido)-4-methyl-pentanoylamino]-2-(1-ethyl-1H-indol-3-yl)-ethyl]-5-methyl-1H-imidazole-4-carboxylic acid 293537 2,4-Difluoro-N-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-benzamidine 293542 (E)-7-[3-(3-Phenyl-allylsulfanylmethyl)-7-oxa-bicyclo[2.2.1]hept-2-yl]-hept-5-enoic acid 293588 N-[(R)-2-(1H-Indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-4-methoxy-benzamidine 293668 [(R)-2-(1H-Indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-carbamic acid benzyl ester 293706 (E)-7-[3-(2-Methyl-hex-2-enylsulfanylmethyl)-7-oxa-bicyclo[2.2.1]hept-2-yl]-hept-5-enoic acid 293713 7-(3-Phenethylsulfanylmethyl-7-oxa-bicyclo[2.2.1]hept-2-yl)-hept-5-enoic acid 293820 5-Methyl-2-{(R)-2-(1-methyl-1H-indol-3-yl)-1-[(S)-4-methyl-2-(3-phenyl-ureido)-pentanoylamino]-ethyl}-oxazole-4-carboxylic acid 293852 N-[(R)-2-(1H-Indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-4-trifluoromethyl-benzamidine 293900 1-(2,4-Difluoro-phenyl)-3-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-urea 293959 Dimethyl-[3-(2-methyl-6H-dibenzo[b,e]oxepin-11-ylidene)-propyl]-amine; compound with but-2-enedioic acid 293983 Biphenyl-2-carboxylic acid [4-(5,6,7,8-tetrahydro-thieno[3,2-b]azepine-4-carbonyl)-phenyl]-amide 294055 2-[(R)-1-[(S)-2-(3-Cyclohexyl-ureido)-4-methyl-pentanoylamino]-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-1H-imidazole-4-carboxylic acid 294061 1'-(4-diethylamino-2-butynyl)spiro[10,11-dihydro-5H-dibenzo[a,d]cycloheptene-5,3'-(tetrahydro-1'H-pyrrole)]-2',5'-dione 294062 1'-(4-diisopropylamino-2-butynyl)spiro[9H-fluorene-9,3'-(tetrahydro-1'H-pyrrole)]-2',5'-dione 294138 2-[(R)-1-{(S)-2-[(2,3-Dihydro-indole-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid 294144 7-(3-Octylsulfanylmethyl-7-oxa-bicyclo[2.2.1]hept-2-yl)-hept-5-enoic acid 294157 2-[(R)-1-{(S)-2-[3-(3-Fluoro-phenyl)-ureido]-4-methyl-pentanoylamino}-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid 294158 2-[(R)-1-{(S)-2-[3-(2-Fluoro-phenyl)-ureido]-4-methyl-pentanoylamino}-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid 294190 N-[4-(8-Dimethylamino-5,6,7,8-tetrahydro-thieno[3,2-b]azepine-4-carbonyl)-phenyl]-2-methyl-benzamide 294268 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (R)-4-(4-hydroxy-benzoylamino)-pyrrolidin-3-yl ester 294269 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (R)-1-(4-hydroxy-benzoylamino)-indan-2-yl ester 294270 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (1R,2S)-1-(4-hydroxy-benzoylamino)-indan-2-yl ester 294277 13-(2-Amino-ethyl)-19-benzyl-22-(4-ethoxy-benzyl)-16-isopropyl-12,15,18,21,24-pentaoxo-7,8-dithia-11,14,17,20,23-pentaaza-spiro[5.19]pentacosane-10-carboxylic acid [1-(carbamoylmethyl-carbamoyl)-4-guanidino-butyl]-amide 294278 13-(2-Amino-ethyl)-19-benzyl-22-(4-ethoxy-benzyl)-16-isopropyl-12,15,18,21,24-pentaoxo-7,8-dithia-11,14,17,20,23-pentaaza-spiro[5.19]pentacosane-10-carboxylic acid (1-carbamoyl-4-guanidino-butyl)-amide 294295 Biphenyl-2-carboxylic acid [3-methoxy-4-(5,6,7,8-tetrahydro-thieno[3,2-b]azepine-4-carbonyl)-phenyl]-amide 294320 Biphenyl-2-carboxylic acid [4-(5,6,7,8-tetrahydro-furo[3,2-b]azepine-4-carbonyl)-phenyl]-amide 294321 Biphenyl-2-carboxylic acid [4-(5,6,7,8-tetrahydro-1H-pyrrolo[3,2-b]azepine-4-carbonyl)-phenyl]-amide 294322 (S)-7-Chloro-9-(4-methyl-piperazin-1-yl)-9,10-dihydro-4-thia-10a-aza-benzo[f]azulene 294346 2-[(R)-1-[(S)-2-(3-Bicyclo[2.2.1]hept-2-yl-ureido)-4-methyl-pentanoylamino]-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid 294349 7-Chloro-1-(4-fluoro-phenyl)-8,9-dimethoxy-4-methyl-2,2a,3,4,5,6-hexahydro-1H-azepino[3,4,5-cd]indole 294368 N'-[5-(4-{4-[(S)-2-Hydroxy-3-(2-oxo-2,3-dihydro-1H-benzoimidazol-4-yloxy)-propylamino]-piperidin-1-yl}-benzylidene)-4-oxo-4,5-dihydro-thiazol-2-yl]-N,N-dimethyl-guanidine 294471 7-[3-(Hexane-1-sulfonylmethyl)-7-oxa-bicyclo[2.2.1]hept-2-yl]-hept-5-enoic acid 294486 2-{[13-(2-Amino-ethyl)-19-benzyl-22-(4-ethoxy-benzyl)-16-isopropyl-12,15,18,21,24-pentaoxo-7,8-dithia-11,14,17,20,23-pentaaza-spiro[5.19]pentacosane-10-carbonyl]-amino}-5-guanidino-pentanoic acid 294487 13-(2-Amino-ethyl)-19-benzyl-22-(4-ethoxy-benzyl)-16-isopropyl-12,15,18,21,24-pentaoxo-7,8-dithia-11,14,17,20,23-pentaaza-spiro[5.19]pentacosane-10-carboxylic acid (1-carbamoyl-5-guanidino-pentyl)-amide 294752 N-[5-(2-{1-[4-((R)-3,5-Dioxo-[1,2,4]oxadiazolidin-2-ylmethyl)-phenyl]-piperidin-4-ylamino}-1-hydroxy-ethyl)-2-hydroxy-phenyl]-methanesulfonamide 294835 1-(4-Fluoro-phenyl)-8,9-dimethoxy-4-methyl-3,4,5,6-tetrahydro-1H-azepino[3,4,5-cd]indole 294844 1-(4-Fluoro-phenyl)-8,9-dimethoxy-4-methyl-2,2a,3,4,5,6-hexahydro-1H-azepino[3,4,5-cd]indole 294935 5,5-Diphenyl-3-(4-pyrrolidin-1-yl-but-2-ynyl)-imidazolidine-2,4-dione 294950 1-(4-Fluoro-phenyl)-8,9-dimethoxy-2,2a,3,4,5,6-hexahydro-1H-azepino[3,4,5-cd]indole 295007 [6-(3,5-Dimethyl-biphenyl-4-ylcarbamoyl)-benzothiazol-2-yl]-carbamic acid tert-butyl ester 295068 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (S)-1-(4-hydroxy-benzoylamino)-indan-2-yl ester 295071 3-(4-Diethylamino-but-2-ynyl)-5,5-diphenyl-imidazolidine-2,4-dione 295184 1'-(4-diethylamino-2-butynyl)spiro[9H-fluorene-9,3'-(tetrahydro-1'H-pyrrole)]-2',5'-dione 295195 1'-(4-tetrahydro-1H-1-pyrrolyl-2-butynyl)spiro[2,3-dihydro-1H-indene-1,3'-(tetrahydro-1'H-pyrrole)]-2',5'-dione 295198 2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid ethyl ester 295235 Biphenyl-2-carboxylic acid (4-{8-[methyl-(2-pyridin-3-yl-ethyl)-amino]-5,6,7,8-tetrahydro-thieno[3,2-b]azepine-4-carbonyl}-phenyl)-amide 295257 Biphenyl-2-carboxylic acid [4-(1-methyl-5,6,7,8-tetrahydro-1H-pyrrolo[3,2-b]azepine-4-carbonyl)-phenyl]-amide 295258 2-Methyl-N-[4-(5,6,7,8-tetrahydro-thieno[3,2-b]azepine-4-carbonyl)-phenyl]-benzamide 295323 7-(3-Propylcarbamoylmethylsulfanylmethyl-7-oxa-bicyclo[2.2.1]hept-2-yl)-hept-5-enoic acid 295324 7-[3-(2-Pentylsulfanyl-ethyl)-7-oxa-bicyclo[2.2.1]hept-2-yl]-hept-5-enoic acid 295334 7-(3-Heptylsulfanylmethyl-7-oxa-bicyclo[2.2.1]hept-2-yl)-hept-5-enoic acid 295452 2-[(R)-1-[(S)-2-(3-Bicyclo[2.2.1]hept-2-yl-ureido)-4-methyl-pentanoylamino]-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-1H-imidazole-4-carboxylic acid 295453 2-[(R)-1-[(S)-2-(3-Adamantan-2-yl-ureido)-4-methyl-pentanoylamino]-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid 295465 7-(3-Phenylsulfanylmethyl-7-oxa-bicyclo[2.2.1]hept-2-yl)-hept-5-enoic acid 295467 7-(3-Methylsulfanylmethylsulfanylmethyl-7-oxa-bicyclo[2.2.1]hept-2-yl)-hept-5-enoic acid 295544 4-Chloro-N-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-benzamidine 295564 2-[(R)-1-[(S)-2-(3-Cycloheptyl-ureido)-4-methyl-pentanoylamino]-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-1H-imidazole-4-carboxylic acid 295576 1'-(4-diethylamino-2-butynyl)spiro[2,3-dihydro-1H-indene-1,3'-(tetrahydro-1'H-pyrrole)]-2',5'-dione 295616 2-Chloro-N-[4-(5,6,7,8-tetrahydro-thieno[3,2-b]azepine-4-carbonyl)-phenyl]-benzamide 295682 7-(3-Butylsulfanylmethyl-7-oxa-bicyclo[2.2.1]hept-2-yl)-hept-5-enoic acid 295716 Biphenyl-2-carboxylic acid [4-(8-dimethylamino-5,6,7,8-tetrahydro-thieno[3,2-b]azepine-4-carbonyl)-phenyl]-amide 296013 sodium salt of 4-tert-Butyl-N-[6-(2-hydroxy-ethoxy)-5-(2-methoxy-phenoxy)-[2,2']bipyrimidinyl-4-yl]-benzenesulfonamide 296221 (1S,2R,3S,4R,5S)-4-[2-Chloro-6-(3-chloro-benzylamino)-purin-9-yl]-2,3-dihydroxy-bicyclo[3.1.0]hexane-1-carboxylic acid methylamide 296229 3-{5-[6-(3-Chloro-phenylamino)-pyrimidin-4-yl]-pyridin-3-ylamino}-propan-1-ol 296230 (1S,2R,3S,4R,5S)-4-(6-(5-chloro-2-methoxybenzylamino)-2-chloro-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 296241 3-Benzyl-8-cyclopentyl-1-propyl-3,7-dihydro-purine-2,6-dione 296242 3-[6''-(3-Chloro-phenylamino)-[2,2'']bipyrazinyl-6-ylamino]-propan-1-ol 296244 3-{4-[6-(3-Chloro-phenylamino)-pyrazin-2-yl]-pyridin-2-ylamino}-propan-1-ol 296245 3-{4-[6-(3-Chloro-phenylamino)-pyrazin-2-yl]-pyridin-3-ylamino}-propan-1-ol 296246 3-{5-[6-(3-Chloro-phenylamino)-pyrazin-2-yl]-oxazol-2-ylamino}-propan-1-ol 296248 3-{5-[6-(3-Chloro-phenylamino)-pyrazin-2-yl]-pyridin-3-ylamino}-propan-1-ol 296261 3-{5-[6-(3-Chloro-phenylamino)-pyrazin-2-yl]-thiazol-2-ylamino}-propan-1-ol 296269 5-(4-Chloro-phenyl)-4-(2,4-dichloro-phenyl)-thiazole-2-carboxylic acid piperidin-1-ylamide 296273 4-(4-Chloro-phenyl)-5-(2,4-dichloro-phenyl)-thiazole-2-carboxylic acid piperidin-1-ylamide 296279 2-(2,4-Dichloro-phenyl)-1-(4-fluoro-phenyl)-5-methyl-1H-imidazole-4-carboxylic acid piperidin-1-ylamide 296280 2-(2,4-Dichloro-phenyl)-1-(4-methoxy-phenyl)-5-methyl-1H-imidazole-4-carboxylic acid piperidin-1-ylamide 296281 2-(2,4-Dichloro-phenyl)-5-methyl-1-(4-trifluoromethyl-phenyl)-1H-imidazole-4-carboxylic acid piperidin-1-ylamide 296282 1-(5-Chloro-pyridin-2-yl)-2-(2,4-dichloro-phenyl)-5-methyl-1H-imidazole-4-carboxylic acid piperidin-1-ylamide 296285 [1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-methyl-1H-imidazol-4-yl]-(4-hydroxy-piperidin-1-yl)-methanone 296286 [1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-methyl-1H-imidazol-4-yl]-(3,4-dihydro-1H-isoquinolin-2-yl)-methanone 296287 1-(4-Bromo-phenyl)-2-(2,4-dichloro-phenyl)-5-methyl-1H-imidazole-4-carboxylic acid piperidin-1-ylamide 296288 1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-ethyl-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 296289 1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-methyl-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 296291 1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-methyl-1H-imidazole-4-carboxylic acid pyrrolidin-1-ylamide 296292 1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-methyl-1H-imidazole-4-carboxylic acid azepan-1-ylamide 296293 1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-methyl-1H-imidazole-4-carboxylic acid morpholin-4-ylamide 296294 1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-methyl-1H-imidazole-4-carboxylic acid (4-hydroxy-cyclohexyl)-amide 296295 1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-methyl-1H-imidazole-4-carboxylic acid cyclopentylamide 296296 5-Chloro-1-(4-chloro-phenyl)-2-(2,4-dichloro-phenyl)-1H-imidazole-4-carboxylic acid piperidin-1-ylamide 296297 5-Bromo-1-(4-chloro-phenyl)-2-(2,4-dichloro-phenyl)-1H-imidazole-4-carboxylic acid piperidin-1-ylamide 296298 1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-fluoromethyl-1H-imidazole-4-carboxylic acid piperidin-1-ylamide 296300 H-Tyr-Val-Met-Gly-His-Phe-Arg-D-Trp-Asp-Arg-Phe-Gly-OH 296301 Ac-Tyr-Val-Nle-Gly-His-D-Phe-Arg-Trp-Asp-Arg-Phe-Gly-NH2 296305 1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-methyl-1H-imidazole-4-carboxylic acid bicyclo[2.2.1]hept-2-ylamide 296306 1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-methyl-1H-imidazole-4-carboxylic acid tert-butoxy-amide 296307 1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-methyl-1H-imidazole-4-carboxylic acid 4-trifluoromethyl-benzylamide 296308 1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-methyl-1H-imidazole-4-carboxylic acid diethylamide 296309 1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-methyl-1H-imidazole-4-carboxylic acid tert-butyl ester 296312 1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-methyl-1H-imidazole-4-carboxylic acid cyclohexylamide 296313 1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-methyl-1H-imidazole-4-carboxylic acid cycloheptylamide 296323 2-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-5-methyl-1H-imidazole-4-carboxylic acid piperidin-1-ylamide 296326 H-Tyr-Val-Nle-Gly-His-D-Phe-Arg-D-Nal(2'')-Asp-Arg-Phe-Gly-NH2 296327 H-Tyr-Val-Nle-Gly-His-Phe-Arg-Trp-Asp-Arg-Phe-Gly-NH 296329 H-Tyr-Val-Nle-Gly-His-D-Nal(2'')-Arg-D-Trp-Asp-Arg-Phe-Gly-NH2 296330 H-Tyr-Val-Nle-Gly-His-D-Nal(2'')-Arg-D-Phe-Asp-Arg-Phe-Gly-NH2 296331 H-Tyr-Val-Nle-Gly-D-Nal(2'')-Phe-Arg-Trp-Asp-Arg-Phe-Gly-NH2 296332 H-Tyr-Val-Nle-Gly-His-Phe-Arg-Trp-Asp-Arg-Phe-Gly-OH 296333 1-(4-chlorophenyl)-5-cyano-2-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 296368 (R)-3-Fluoromethyl-1,2,3,4-tetrahydro-isoquinoline-7-sulfonic acid ethylamide 296372 (R)-3-Fluoromethyl-1,2,3,4-tetrahydro-isoquinoline-7-sulfonic acid (3,3,3-trifluoro-propyl)-amide 296373 (R)-3-Fluoromethyl-1,2,3,4-tetrahydro-isoquinoline-7-sulfonic acid (3-methoxy-propyl)-amide 296378 (R)-3-Fluoromethyl-1,2,3,4-tetrahydro-isoquinoline-7-sulfonic acid propylamide 296379 (R)-3-Fluoromethyl-1,2,3,4-tetrahydro-isoquinoline-7-sulfonic acid (2,2,2-trifluoro-ethyl)-amide 296383 (R)-3-Fluoromethyl-1,2,3,4-tetrahydro-isoquinoline-7-sulfonic acid amide 296384 3-(fluoromethyl)-N-(2,2,2-trifluoroethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide 296385 4-(Benzothiazol-5-ylamino)-6-(benzyl-methyl-amino)-[1,3,5]triazin-2-ol 296389 N-Benzothiazol-6-yl-6-chloro-N''-(1-methyl-1-phenyl-ethyl)-[1,3,5]triazine-2,4-diamine 296393 (R)-3-Fluoromethyl-7-(thiomorpholine-4-sulfonyl)-1,2,3,4-tetrahydro-isoquinoline 296394 N-ethyl-3-(fluoromethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide 296399 N-[4-(Benzothiazol-6-ylamino)-6-(1-methyl-1-phenyl-ethylamino)-[1,3,5]triazin-2-yl]-hydroxylamine 296403 N-Benzothiazol-6-yl-6-methoxy-N''-(1-methyl-1-phenyl-ethyl)-[1,3,5]triazine-2,4-diamine 296405 4-(Benzothiazol-6-ylamino)-6-(1-methyl-1-phenyl-ethylamino)-[1,3,5]triazin-2-ol 296406 4-(Benzothiazol-6-ylamino)-6-benzylamino-[1,3,5]triazin-2-ol 296414 4-(Benzothiazol-6-ylamino)-6-(benzyl-ethyl-amino)-[1,3,5]triazin-2-ol 296415 4-(Benzothiazol-6-ylamino)-6-(benzyl-isopropyl-amino)-[1,3,5]triazin-2-ol 296419 4-(Benzothiazol-6-yl-methyl-amino)-6-(1-methyl-1-phenyl-ethylamino)-[1,3,5]triazin-2-ol 296420 4-(3H-Benzoimidazol-5-ylamino)-6-(1-methyl-1-phenyl-ethylamino)-[1,3,5]triazin-2-ol 296421 3-Fluoromethyl-1,2,3,4-tetrahydro-isoquinoline-7-sulfonic acid (3-methoxy-propyl)-amide 296425 3-(fluoromethyl)-N-propyl-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide 296429 (+)-3-(fluoromethyl)-N-(3,3,3-trifluoropropyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide 296442 (+)-3-(fluoromethyl)-7-(thiomorpholinosulfonyl)-1,2,3,4-tetrahydroisoquinoline 296493 2-Furan-2-yl-N*5*-[1-(5-methyl-isoxazol-3-ylmethyl)-piperidin-4-ylmethyl]-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296512 2-Furan-2-yl-N*5*-[1-(5-methyl-isoxazol-3-ylmethyl)-piperidin-3-ylmethyl]-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296513 2-Furan-2-yl-5-[4-(5-methyl-isoxazol-3-ylmethyl)-piperazin-1-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 296531 2-Furan-2-yl-5-[4-(5-methyl-isoxazol-3-ylmethyl)-[1,4]diazepan-1-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 296532 2-Furan-2-yl-N*5*-{2-[(5-methyl-isoxazol-3-ylmethyl)-amino]-ethyl}-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296552 2-Furan-2-yl-N*5*-[(R)-1-(5-methyl-isoxazol-3-ylmethyl)-pyrrolidin-2-ylmethyl]-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296554 2-Furan-2-yl-N*5*-methyl-N*5*-{2-[methyl-(5-methyl-isoxazol-3-ylmethyl)-amino]-ethyl}-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296560 2-Furan-2-yl-N*5*-{2-[methyl-(5-methyl-isoxazol-3-ylmethyl)-amino]-ethyl}-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296596 N5-(((R)-1-(2,6-difluorobenzyl)pyrrolidin-2-yl)methyl)-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296598 N*5*-[(R)-1-(4-Chloro-benzyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296602 N*5*-((R)-1-Benzofuran-2-ylmethyl-pyrrolidin-2-ylmethyl)-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296604 N*5*-[(R)-1-(2-Chloro-3,6-difluoro-benzyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296614 N*5*-[(R)-1-(3,5-Dichloro-benzyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296616 2-Furan-2-yl-7-phenyl-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 296619 2-Furan-2-yl-N*5*-[(R)-1-(2,4,5-trifluoro-benzyl)-pyrrolidin-2-ylmethyl]-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296620 2-Furan-2-yl-N*5*-((R)-1-quinolin-2-ylmethyl-pyrrolidin-2-ylmethyl)-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296621 N*5*-[(R)-1-(3-Chloro-2-fluoro-6-trifluoromethyl-benzyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296625 2-Furan-2-yl-N*5*-[1-(5-methyl-isoxazol-3-ylmethyl)-piperidin-4-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296630 1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(3-fluoro-benzenesulfonyl)-piperidine 296631 1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(2-fluoro-benzenesulfonyl)-piperidine 296634 2-Furan-2-yl-N*5*-methyl-N*5*-[(R)-1-(5-methyl-isoxazol-3-ylmethyl)-pyrrolidin-2-ylmethyl]-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296635 2-Furan-2-yl-N*5*-[(R)-1-(2,3,6-trifluoro-benzyl)-pyrrolidin-2-ylmethyl]-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296636 N*5*-[(R)-1-(2,4-Dichloro-benzyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296637 2-Furan-2-yl-N*5*-((R)-1-pyridin-2-ylmethyl-pyrrolidin-2-ylmethyl)-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296641 2-Furan-2-yl-N*5*-[1-(5-methyl-isoxazol-3-ylmethyl)-piperidin-3-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296642 5-[4-(2-Chloro-benzyl)-piperazin-1-yl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 296654 2-Furan-2-yl-N*5*-[(R)-1-(3-methyl-benzyl)-pyrrolidin-2-ylmethyl]-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296655 2-Furan-2-yl-N*5*-((R)-1-pyridin-3-ylmethyl-pyrrolidin-2-ylmethyl)-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296660 2-(4-Benzenesulfonyl-piperidin-1-yl)-1-(2,4-difluoro-phenyl)-ethanone 296661 2-Furan-2-yl-N*5*-methyl-N*5*-[(R)-1-(5-methyl-isoxazol-3-ylmethyl)-piperidin-2-ylmethyl]-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296662 2-Furan-2-yl-N*5*-[(R)-1-(2,4,6-trifluoro-benzyl)-pyrrolidin-2-ylmethyl]-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296670 N*5*-[(R)-1-(2,4-Difluoro-benzyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296671 2-Furan-2-yl-N*5*-((R)-1-furan-2-ylmethyl-pyrrolidin-2-ylmethyl)-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296672 5-[4-(3-Chloro-benzyl)-piperazin-1-yl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 296674 N*5*-[(R)-1-(3-Fluoro-benzyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296675 2-Furan-2-yl-N*5*-((R)-1-pyridin-4-ylmethyl-pyrrolidin-2-ylmethyl)-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296676 2-Furan-2-yl-7-m-tolyl-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 296678 N*5*-[(R)-1-(5-Chloro-furan-2-ylmethyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296681 N*5*-[(R)-1-(2-Chloro-benzyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296685 4-(4-Azetidin-1-yl-benzenesulfonyl)-1-[2-(2,4-difluoro-phenyl)-ethyl]-4-fluoro-piperidine 296689 N*5*-[(R)-1-(2-Fluoro-5-trifluoromethyl-benzyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296690 5-[4-(3,5-Dimethyl-isoxazol-4-ylmethyl)-piperazin-1-yl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 296691 N*5*-[(R)-1-(3,5-Difluoro-benzyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296692 N*5*-[(R)-1-(3,5-Dimethyl-isoxazol-4-ylmethyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296694 N*5*-[(R)-1-(2,3-Difluoro-benzyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296695 N*5*-[(R)-1-(3,5-Dichloro-pyridin-4-ylmethyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296707 N*5*-[(R)-1-(3-Chloro-benzyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296708 4-Benzenesulfonyl-1-[2-(2,4-difluoro-phenyl)-ethyl]-4-fluoro-piperidine 296709 N*5*-[(R)-1-(2,5-Difluoro-benzyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296710 N*5*-[(R)-1-(3-Chloro-1-methyl-1H-pyrazol-4-ylmethyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296713 N*5*-[(R)-1-(3-Chloro-2-fluoro-benzyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamin 296714 N*5*-[(R)-1-(2-Chloro-pyridin-4-ylmethyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296715 N*5*-[(R)-1-(2-Fluoro-4-trifluoromethyl-benzyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 296716 2-Furan-2-yl-5-[4-(2,4,6-trifluoro-benzyl)-piperazin-1-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 296729 2-Furan-2-yl-7-(3,4,5-trimethoxy-phenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 296745 2-Furan-2-yl-7-p-tolyl-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 296753 2-(furan-2-yl)-7-(2-methoxyphenyl)-[1,2,4]triazolo[1,5-f]pyrimidin-5-amine 296762 7-(3-Amino-phenyl)-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 296763 2-Furan-2-yl-7-o-tolyl-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 296766 2-Furan-2-yl-7-(3-methoxy-phenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 296768 2-Furan-2-yl-7-(2,3,4-trimethoxy-phenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 296773 2-Furan-2-yl-7-(4-methoxy-phenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 296798 1-(2,4-difluorophenethyl)-4-fluoro-4-(4-fluorophenylsulfonyl)piperidine 296817 1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(4-pyrazol-1-yl-benzenesulfonyl)-piperidine 296821 2-Furan-2-yl-7-thiophen-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 296824 7-(2,4-Dimethoxy-phenyl)-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 296825 7-(3,4-Dimethoxy-phenyl)-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 296837 1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(4-[1,2,3]triazol-1-yl-benzenesulfonyl)-piperidine 296852 7-(2,5-Dimethoxy-phenyl)-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 296856 4-(4-Chloro-benzenesulfonyl)-1-[2-(2,4-difluoro-phenyl)-ethyl]-4-fluoro-piperidine 296859 7-(2,6-Dimethoxy-phenyl)-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 296864 4-{1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-piperidine-4-sulfonyl}-benzonitrile 296866 7-(2,3-Dimethoxy-phenyl)-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 296871 7-Biphenyl-3-yl-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 296872 3-[1-(3-Dimethylamino-propyl)-1H-indazol-3-yl]-4-(1-vinyl-1H-indol-3-yl)-pyrrole-2,5-dione 296873 Dimethyl-(2-{(3R,3aS)-3-[4-((E)-2-methyl-3-phenyl-allyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-chromeno[4,3-c]isoxazol-7-yloxy}-ethyl)-amine 296874 3-[1-(1,2-Dihydro-pyridin-2-yl)-1H-indazol-3-yl]-4-[1-(1,4,4a,8a-tetrahydro-naphthalen-2-yl)-1H-indol-3-yl]-pyrrole-2,5-dione 296875 3-(1-Piperazin-1-yl-1H-indazol-3-yl)-4-[1-(1,4,4a,8a-tetrahydro-naphthalen-2-yl)-1H-indol-3-yl]-pyrrole-2,5-dione 296877 1-(2-Cyclohexyl-ethyl)-4-[2-(3H-imidazol-4-yl)-ethyl]-piperidine 296885 1-(2-Cyclohexyl-ethyl)-4-(3H-imidazol-4-ylmethylene)-piperidine 296890 Acetic acid (3R,3aS)-3-[4-((E)-2-methyl-3-phenyl-allyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-chromeno[4,3-c]isoxazol-7-ylester 296896 3-[1-(3-Dimethylamino-propyl)-1H-indazol-3-yl]-4-(1-phenyl-1H-indol-3-yl)-pyrrole-2,5-dione 296900 3-[1-(3-Dimethylamino-propyl)-1H-indazol-3-yl]-4-[1-(1,4,4a,8a-tetrahydro-naphthalen-2-yl)-1H-indol-3-yl]-pyrrole-2,5-dione 296902 1-(3-Cyclohexyl-propyl)-4-(3H-imidazol-4-ylmethyl)-piperidine 296903 [3-(5-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin-7-yl)-phenyl]-methanol 296906 (3R,3aS)-7-Methoxy-3-[4-((E)-2-methyl-3-phenyl-allyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-chromeno[4,3-c]isoxazole 296908 Methoxy-acetic acid (3R,3aS)-3-[4-((E)-2-methyl-3-phenyl-allyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-chromeno[4,3-c]isoxazol-7-yl ester 296909 2-Furan-2-yl-7-{3-[(methyl-phenethyl-amino)-methyl]-phenyl}-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 296913 3-[1-(3-Dimethylamino-propyl)-1H-indazol-3-yl]-4-(1-thiophen-2-yl-1H-indol-3-yl)-pyrrole-2,5-dione 296916 2-Furan-2-yl-7-pyridin-4-yl-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 296917 3-[1-(3-Dimethylamino-propyl)-1H-indazol-3-yl]-4-[1-(1,4,4a,8a-tetrahydro-naphthalen-1-yl)-1H-indol-3-yl]-pyrrole-2,5-dione 296922 (3R,3aS)-3-[4-((E)-2-Methyl-3-phenyl-allyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-chromeno[4,3-c]isoxazol-7-ol 296926 3-[1-(3-Dimethylamino-propyl)-1H-indazol-3-yl]-4-(1-pyridin-3-yl-1H-indol-3-yl)-pyrrole-2,5-dione 296928 Cyclopropanecarboxylic acid (3R,3aS)-3-[4-((E)-2-methyl-3-phenyl-allyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-chromeno[4,3-c]isoxazol-7-yl ester 296931 Acrylic acid (3R,3aS)-3-[4-((E)-2-methyl-3-phenyl-allyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-chromeno[4,3-c]isoxazol-7-ylester 296932 1-{(3R,3aR)-3-[4-((E)-5-Phenyl-pent-4-enyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-isoxazolo[4,3-c]quinolin-5-yl}-ethanone 296933 (3R,3aS)-7-(2-Methoxy-ethoxy)-3-[4-((E)-2-methyl-3-phenyl-allyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-chromeno[4,3-c]isoxazole 296937 3-(1H-Indazol-3-yl)-4-(1-pyridin-3-yl-1H-indol-3-yl)-pyrrole-2,5-dione 296943 2,2-Dimethyl-propionic acid (3R,3aS)-3-[4-((E)-2-methyl-3-phenyl-allyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-chromeno[4,3-c]isoxazol-7-yl ester 296944 2-Furan-2-yl-7-pyridin-3-yl-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 296945 2-Furan-2-yl-7-pyridin-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 296952 (3R,3aS)-7-[2-(2-Ethoxy-ethoxy)-ethoxy]-3-[4-((E)-2-methyl-3-phenyl-allyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-chromeno[4,3-c]isoxazole 296953 3-(5-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin-7-yl)-benzonitrile 296954 3-[1-(3-Dimethylamino-propyl)-1H-indazol-3-yl]-4-(1-isoquinolin-4-yl-1H-indol-3-yl)-pyrrole-2,5-dione 296955 3-[1-(3-Dimethylamino-propyl)-1H-indazol-3-yl]-4-(1-quinolin-3-yl-1H-indol-3-yl)-pyrrole-2,5-dione 296957 1-Cyclohexylmethyl-4-(3H-imidazol-4-ylmethyl)-piperidine 296962 1-Cyclohexylmethyl-4-[2-(3H-imidazol-4-yl)-ethyl]-piperidine 296966 Isonicotinic acid (3R,3aS)-3-[4-((E)-2-methyl-3-phenyl-allyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-chromeno[4,3-c]isoxazol-7-yl ester 296967 (3R,3aS)-7-Cyclopentyloxy-3-[4-((E)-2-methyl-3-phenyl-allyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-chromeno[4,3-c]isoxazole 296974 3-(1-Benzo[b]thiophen-2-yl-1H-indol-3-yl)-4-[1-(3-dimethylamino-propyl)-1H-indazol-3-yl]-pyrrole-2,5-dione 296975 3-(1-Morpholin-2-yl-1H-indazol-3-yl)-4-[1-(1,4,4a,8a-tetrahydro-naphthalen-2-yl)-1H-indol-3-yl]-pyrrole-2,5-dione 296976 1-Cyclohexylmethyl-4-(3H-imidazol-4-ylmethylene)-piperidine 296977 1-(2-Cyclohexyl-ethyl)-4-(3H-imidazol-4-ylmethyl)-piperidine 296981 2-Furan-2-yl-7-(4-isopropyl-phenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 296983 7-{3-[4-(4-Fluoro-phenyl)-piperidin-1-ylmethyl]-phenyl}-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 296986 2-(3-Phenoxy-phenyl)-1H-benzoimidazole-5-carboxylic acid amide 296994 2-p-Tolyl-1H-benzoimidazole-5-carboxylic acid amide 296996 1-Cyclohexyl-4-[2-(3H-imidazol-4-yl)-ethyl]-piperidine 297003 1-Cyclohexyl-4-(3H-imidazol-4-ylmethylene)-piperidine 297010 2-Naphthalen-2-yl-1H-benzoimidazole-5-carboxylic acid amide 297011 2-[3-(3,4-Dichloro-phenoxy)-phenyl]-1H-benzoimidazole-5-carboxylic acid amide 297046 7-(3-{4-[2-Fluoro-4-(2-methoxy-ethoxy)-phenyl]-piperazin-1-ylmethyl}-phenyl)-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 297047 7-(3-{4-[2-Chloro-4-(2-methoxy-ethoxy)-phenyl]-piperazin-1-ylmethyl}-phenyl)-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 297048 2-Furan-2-yl-7-(3-{4-[3-methoxy-4-(2-methoxy-ethoxy)-phenyl]-piperazin-1-ylmethyl}-phenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 297049 2-Furan-2-yl-7-(3-{4-[4-(2-methoxy-ethoxy)-2-methyl-phenyl]-piperazin-1-ylmethyl}-phenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 297057 2-Furan-2-yl-7-[3-(4-phenyl-piperazin-1-ylmethyl)-phenyl]-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 297058 2-Furan-2-yl-7-(3-{4-[4-(2-methoxy-ethoxy)-phenyl]-piperazin-1-ylmethyl}-phenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 297059 2-(4-Phenoxy-phenyl)-1H-benzoimidazole-4-carboxylic acid amide 297066 2-Phenyl-1H-benzoimidazole-5-carboxylic acid amide 297070 1-Ethyl-4-(3H-imidazol-4-ylmethylene)-piperidine 297081 2-(4-Ethoxy-phenyl)-1H-benzoimidazole-5-carboxylic acid amide 297082 2-(4-phenoxyphenyl)-1H-benzo[d]imidazole-5-carboxylic acid 297083 2-Furan-2-yl-7-[3-(4-phenyl-piperidin-1-ylmethyl)-phenyl]-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 297089 4-(3H-Imidazol-4-ylmethyl)-1-isopropyl-piperidine 297090 4-[2-(3H-Imidazol-4-yl)-ethyl]-1-isopropyl-piperidine 297095 2-(4-Phenoxy-phenyl)-1H-benzoimidazole-5-carbonitrile 297096 5-Nitro-2-(4-phenoxy-phenyl)-1H-benzoimidazole 297106 4-(3H-Imidazol-4-ylmethylene)-1-isopropyl-piperidine 297107 1-Cyclohexyl-4-(3H-imidazol-4-ylmethyl)-piperidine 297119 7-{3-[4-(3,4-Dichloro-phenyl)-piperazin-1-ylmethyl]-phenyl}-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 297127 2-[4-(4-Carbamoyl-phenoxy)-phenyl]-1H-benzoimidazole-5-carboxylic acid amide 297135 2-[4-(3-Hydroxy-phenoxy)-phenyl]-1H-benzoimidazole-5-carboxylic acid amide 297145 2-[4-(4-Chloro-3-hydroxy-phenoxy)-phenyl]-1H-benzoimidazole-5-carboxylic acid amide 297152 2-Furan-2-yl-7-(3-{4-[4-(2-methoxy-ethoxy)-phenyl]-piperidin-1-ylmethyl}-phenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 297153 2-[4-(Naphthalen-2-yloxy)-phenyl]-1H-benzoimidazole-5-carboxylic acid amide 297162 2-{4-[3-(5-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin-7-yl)-benzyl]-piperazin-1-yl}-5-(2-methoxy-ethoxy)-benzonitrile 297163 5-{4-[3-(5-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin-7-yl)-benzyl]-piperazin-1-yl}-2-(2-methoxy-ethoxy)-benzonitrile 297164 2-(4-Phenoxy-phenyl)-1H-benzoimidazol-5-ylamine 297166 7-(3-{4-[2,6-Difluoro-4-(2-methoxy-ethoxy)-phenyl]-piperazin-1-ylmethyl}-phenyl)-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 297167 7-(3-{4-[3,5-Difluoro-4-(2-methoxy-ethoxy)-phenyl]-piperazin-1-ylmethyl}-phenyl)-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 297169 2-Furan-2-yl-7-[3-(4-thiazol-2-yl-piperazin-1-ylmethyl)-phenyl]-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 297179 SID29217525 297180 2-[4-(3,4-Dichloro-phenoxy)-phenyl]-1H-benzoimidazole-5-carboxylic acid amide 297181 2-(4-Phenoxy-phenyl)-1H-benzoimidazole-5-sulfonic acid amide 297186 2-(4-phenoxyphenyl)-1H-benzo[d]imidazole-5-carboxamide 297187 2-[4-(3-Chloro-phenoxy)-phenyl]-1H-benzoimidazole-5-carboxylic acid amide 297191 2-[4-(4-Methoxy-phenoxy)-phenyl]-1H-benzoimidazole-5-carboxylic acid amide 297195 2-[4-(3-Chloro-4-methyl-phenoxy)-phenyl]-1H-benzoimidazole-5-carboxylic acid amide 297196 2-[4-(4-Chloro-3-trifluoromethyl-phenoxy)-phenyl]-1H-benzoimidazole-5-carboxylic acid amide 297197 2-(4-Phenoxy-phenyl)-1H-benzoimidazole-5-carboxylic acid methylamide 297201 2-Furan-2-yl-7-(3-{4-[3-(2-methoxy-ethoxy)-phenyl]-piperazin-1-ylmethyl}-phenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 297203 2-(4-p-Tolyloxy-phenyl)-1H-benzoimidazole-5-carboxylic acid amide 297207 2-[4-(2-Fluoro-5-trifluoromethyl-phenoxy)-phenyl]-1H-benzoimidazole-5-carboxylic acid amide 297208 2-[4-(3,4-Dimethyl-phenoxy)-phenyl]-1H-benzoimidazole-5-carboxylic acid amide 297209 2-[4-(3,4-Dimethoxy-phenoxy)-phenyl]-1H-benzoimidazole-5-carboxylic acid amide 297218 1-{(1R,2S)-2-[(S)-3-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-o-tolyl-urea 297220 1-(3-Cyano-phenyl)-3-{(1R,2S)-2-[4-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-urea 297224 4-(3H-Imidazol-4-ylmethylene)-1-methyl-piperidine 297227 2-Amino-4-(3-fluoro-phenyl)-6-(2-hydroxy-ethylsulfanyl)-pyridine-3,5-dicarbonitrile 297228 2-Amino-4-(4-fluoro-phenyl)-6-(2-hydroxy-ethylsulfanyl)-pyridine-3,5-dicarbonitrile 297229 N-(4-Benzoyl-phenyl)-2-[4-(2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide 297230 1-{2-[4-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-(3-methoxy-phenyl)-urea 297237 1-(3-Acetyl-phenyl)-3-{2-[4-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-urea 297239 1-(3-Acetyl-phenyl)-3-{(1R,2S)-2-[4-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-urea 297240 1-Ethyl-4-(3H-imidazol-4-ylmethyl)-piperidine 297243 1-{(1R,2S)-2-[(S)-3-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-(2-methoxy-phenyl)-urea 297252 2-Amino-6-(2-hydroxy-ethylsulfanyl)-4-(3-methoxy-phenyl)-pyridine-3,5-dicarbonitrile 297253 1-Ethyl-4-[2-(3H-imidazol-4-yl)-ethyl]-piperidine 297257 2-Amino-6-(2-hydroxy-ethylsulfanyl)-4-(4-methoxy-phenyl)-pyridine-3,5-dicarbonitrile 297258 1-(3-Acetyl-phenyl)-3-[2-(4-fluoro-benzyl)-piperidin-1-yl]-urea 297261 2-Amino-6-(2-hydroxy-ethylsulfanyl)-4-phenyl-pyridine-3,5-dicarbonitrile 297263 2-Amino-6-(2-hydroxy-ethylsulfanyl)-4-(3-trifluoromethyl-phenyl)-pyridine-3,5-dicarbonitrile 297269 2-Amino-6-(2-hydroxy-ethylsulfanyl)-4-(4-trifluoromethyl-phenyl)-pyridine-3,5-dicarbonitrile 297273 2-amino-4-(benzo[d][1,3]dioxol-5-yl)-6-(2-hydroxyethylthio)pyridine-3,5-dicarbonitrile 297275 1-{(1R,2S)-2-[(S)-3-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-phenyl-urea 297286 1-[2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-methoxy-phenyl)-ethyl]-3-(3,5-dichloro-phenyl)-urea 297290 2-Amino-6-(2-hydroxy-ethylsulfanyl)-4-m-tolyl-pyridine-3,5-dicarbonitrile 297291 2-Amino-6-(2-hydroxy-ethylsulfanyl)-4-p-tolyl-pyridine-3,5-dicarbonitrile 297299 2-Amino-4-(4-dimethylamino-phenyl)-6-(2-hydroxy-ethylsulfanyl)-pyridine-3,5-dicarbonitrile 297302 1-[(1R,2S)-2-(4-Benzyl-piperidin-1-ylmethyl)-cyclohexyl]-3-(3-cyano-phenyl)-urea 297307 2-Amino-6-(2-hydroxy-ethylsulfanyl)-4-(3-hydroxy-phenyl)-pyridine-3,5-dicarbonitrile 297308 2-Amino-6-(2-hydroxy-ethylsulfanyl)-4-(4-hydroxy-phenyl)-pyridine-3,5-dicarbonitrile 297312 [2-(4-tert-Butyl-phenyl)-ethyl]-[2-(4-cyclohexyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethyl]-amine 297319 1-(3-Acetyl-phenyl)-3-[(1R,2S)-2-(4-benzyl-piperidin-1-ylmethyl)-cyclohexyl]-urea 297320 4-[2-(3H-Imidazol-4-yl)-ethyl]-1-methyl-piperidine 297321 1-[2-(4-Benzyl-piperidin-1-ylmethyl)-cyclohexyl]-3-(3-methoxy-phenyl)-urea 297327 2-Amino-4-(3-difluoromethoxy-phenyl)-6-(2-hydroxy-ethylsulfanyl)-pyridine-3,5-dicarbonitrile 297328 2-Amino-4-(4-difluoromethoxy-phenyl)-6-(2-hydroxy-ethylsulfanyl)-pyridine-3,5-dicarbonitrile 297333 1-{(1R,2S)-2-[4-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-(3-methoxy-phenyl)-urea 297334 methimepip 297335 1-[2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethyl]-3-(3,5-dichloro-phenyl)-urea 297342 2-Amino-6-(2-hydroxy-ethylsulfanyl)-4-(3-trifluoromethoxy-phenyl)-pyridine-3,5-dicarbonitrile 297349 2-Amino-6-(2-hydroxy-ethylsulfanyl)-4-(4-trifluoromethoxy-phenyl)-pyridine-3,5-dicarbonitrile 297422 1-[2-Amino-2-(2-fluoro-phenyl)-ethyl]-3-(2,6-difluoro-benzyl)-5-(3-methoxy-phenyl)-[1,3,5]triazinane-2,4,6-trione 297437 (R)-1-(2,6-difluorobenzyl)-3-(2-amino-2-phenylethyl)-5-(3-methoxyphenyl)-1,3,5-triazinane-2,4,6-trione 297455 2-[4-(6-Fluoro-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-quinolin-6-yl-acetamide 297462 1-(2-Amino-4-methyl-pentyl)-3-(2,6-difluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-[1,3,5]triazinane-2,4,6-trione 297486 N-{4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-4-fluoro-benzamide 297490 1-((R)-3-Amino-5-methyl-hexyl)-3-(2,6-difluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-[1,3,5]triazinane-2,4,6-trione 297493 N-(2-(4-(2,3-dichlorophenyl)piperazin-1-yl)vinyl)benzofuran-2-carboxamide 297494 N-{4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-nicotinamide 297496 N-{4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-4-(1H-imidazol-2-yl)-benzamide 297499 2-Chloro-N-{4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-benzamide 297501 1-[3-Amino-3-(3-fluoro-phenyl)-propyl]-3-(2,6-difluoro-benzyl)-5-(3-methoxy-phenyl)-[1,3,5]triazinane-2,4,6-trione 297503 3-Chloro-N-{4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-benzamide 297507 N-{4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-isonicotinamide 297518 Quinoxaline-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-amide 297520 (R)-1-(2,6-difluorobenzyl)-3-(2-amino-2-phenylethyl)-5-(2-fluoro-3-methoxyphenyl)-1,3,5-triazinane-2,4,6-trione 297525 N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)but-2-enyl)-4-(pyridin-2-yl)benzamide 297527 1-(3-Amino-3-o-tolyl-propyl)-3-(2,6-difluoro-benzyl)-5-(3-methoxy-phenyl)-[1,3,5]triazinane-2,4,6-trione 297541 1-[2-Amino-2-(2-fluoro-phenyl)-ethyl]-3-(2,6-difluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-[1,3,5]triazinane-2,4,6-trione 297542 1-(3-Amino-3-thiophen-2-yl-propyl)-3-(2,6-difluoro-benzyl)-5-(3-methoxy-phenyl)-[1,3,5]triazinane-2,4,6-trione 297545 1-(3-Amino-3-pyridin-3-yl-propyl)-3-(2,6-difluoro-benzyl)-5-(3-methoxy-phenyl)-[1,3,5]triazinane-2,4,6-trione 297570 N-{4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-4-pyridin-3-yl-benzamide 297571 1-((R)-2-Amino-2-phenyl-ethyl)-3-(2-fluoro-3-methoxy-phenyl)-5-(2-methyl-benzyl)-[1,3,5]triazinane-2,4,6-trione 297574 1-[3-Amino-3-(2-fluoro-phenyl)-propyl]-3-(2,6-difluoro-benzyl)-5-(3-methoxy-phenyl)-[1,3,5]triazinane-2,4,6-trione 297577 1-[3-Amino-3-(4-fluoro-phenyl)-propyl]-3-(2,6-difluoro-benzyl)-5-(3-methoxy-phenyl)-[1,3,5]triazinane-2,4,6-trione 297579 1-((R)-2-Amino-2-phenyl-ethyl)-3-(2-fluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-[1,3,5]triazinane-2,4,6-trione 297589 1-[3-Amino-3-(2-chloro-phenyl)-propyl]-3-(2,6-difluoro-benzyl)-5-(3-methoxy-phenyl)-[1,3,5]triazinane-2,4,6-trione 297590 N-{4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-4-pyridin-4-yl-benzamide 297601 N-{4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-2-fluoro-benzamide 297606 1-(3-Amino-2-phenyl-propyl)-3-(2,6-difluoro-benzyl)-5-(3-methoxy-phenyl)-[1,3,5]triazinane-2,4,6-trione 297613 N-{4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-4-pyrimidin-2-yl-benzamide 297621 1-(3-Amino-3-phenyl-propyl)-3-(2,6-difluoro-benzyl)-5-(3-methoxy-phenyl)-[1,3,5]triazinane-2,4,6-trione 297625 N-{4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-3-fluoro-benzamide 297626 N-(2-(4-(2,3-dichlorophenyl)piperazin-1-yl)vinyl)benzo[b]thiophene-2-carboxamide 297647 1-((R)-2-Amino-2-phenyl-ethyl)-3-(2-bromo-6-fluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-[1,3,5]triazinane-2,4,6-trione 297650 1-((R)-2-Amino-2-phenyl-ethyl)-3-(2-fluoro-3-methoxy-phenyl)-5-(2-trifluoromethoxy-benzyl)-[1,3,5]triazinane-2,4,6-trione 297653 Pyridine-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-amide 297675 1-((R)-2-Amino-2-phenyl-ethyl)-3-(2-chloro-6-fluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-[1,3,5]triazinane-2,4,6-trione 297678 4-Chloro-N-{4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-benzamide 297679 N-{4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-2-iodo-benzamide 297685 1-((R)-2-Amino-2-phenyl-ethyl)-3-(2-fluoro-3-methoxy-phenyl)-5-(2-fluoro-6-trifluoromethyl-benzyl)-[1,3,5]triazinane-2,4,6-trione 297690 1-((R)-2-Amino-2-phenyl-ethyl)-3-(2-fluoro-3-methoxy-phenyl)-5-(2-methoxy-benzyl)-[1,3,5]triazinane-2,4,6-trione 297700 N-{4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-3-iodo-benzamide 297701 N-{4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-4-iodo-benzamide 297706 1-((R)-2-Amino-2-phenyl-ethyl)-3-(2,6-dichloro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-[1,3,5]triazinane-2,4,6-trione 297718 1-((R)-2-Amino-2-phenyl-ethyl)-3-(2-chloro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-[1,3,5]triazinane-2,4,6-trione 297738 N-{4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-butyl}-4-pyridin-3-yl-benzamide 297739 1-((S)-3-Amino-3-phenyl-propyl)-3-(2,6-difluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-[1,3,5]triazinane-2,4,6-trione 297742 N-{4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-2-methoxy-benzamide 297750 1-((R)-2-Amino-2-phenyl-ethyl)-3-[1-(2,6-difluoro-phenyl)-ethyl]-5-(2-fluoro-3-methoxy-phenyl)-[1,3,5]triazinane-2,4,6-trione 297762 N-{4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-3-methoxy-benzamide 297769 2-[3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-fluoro-3-methoxy-phenyl)-2,4,6-trioxo-[1,3,5]triazinan-1-ylmethyl]-benzonitrile 297776 Des-AA1,2,4,5-[D-Trp8]SRIF 297777 Des-AA1,2,4,5,13-[D-Trp8]-SRIF 297778 Des-AA1,4,5,13-[Tyr2,D-Trp8]-SRIF 297783 1-[4-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phenyl)-butyl]-3-(3-chloro-phenyl)-urea 297784 2-[3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-fluoro-3-methoxy-phenyl)-2,4,6-trioxo-[1,3,5]triazinan-1-ylmethyl]-3-chloro-benzonitrile 297785 cyclo(7-12) Des-AA1,2,5-[Glu7,D-Trp8,(NMe)IAmp9,m-I-Tyr11,Lys12]SRIF 297786 cyclo(7-12) Des-AA1,2,5-[Glu7,D-Trp8,IAmp9,m-I-Tyr11,hhLys12]SRIF 297787 cyclo(7-12) Des-AA1,2,5-[Glu7,D-Trp8,(NMe)IAmp9,m-I-Tyr11,hhLys12]SRIF 297804 1-((R)-2-Amino-2-phenyl-ethyl)-3-(2-chloro-pyridin-3-ylmethyl)-5-(2-fluoro-3-methoxy-phenyl)-[1,3,5]triazinane-2,4,6-trione 297805 Des-AA1,2,5-[(NalphaMe)Lys4,D-Nal8,IAmp9]SRIF 297807 cyclo(7-12) Des-AA1,2,5-[Glu7,D-Trp8,IAmp9,m-I-Tyr11,D-hhLys12]SRIF 297808 cyclo(7-12) Des-AA1,2,5-[Glu7,D-Trp8,(NMe)IAmp9,m-I-Tyr11,D-hhLys12]SRIF 297812 1-[2-(2'-Chloro-biphenyl-4-yl)-4-cyclopentylamino-butyl]-3-(3,5-dichloro-phenyl)-urea 297813 1-[4-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phenyl)-butyl]-3-(3-trifluoromethyl-phenyl)-urea 297819 1-[4-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phenyl)-butyl]-3-(3-chloro-4-fluoro-phenyl)-urea 297821 Des-AA1,2,5-[(NalphaMe)D-Nal8,IAmp9]SRIF 297822 Des-AA1,2,5-[D-Nal8,(NalphaMe)IAmp9]SRIF 297824 Des-AA1,2,5-[D-Nal8,IAmp9,(NalphaMe)Phe11]SRIF 297825 Des-AA1,2,5-[D-Nal8,IAmp9,(NalphaMe)Thr12]SRIF 297833 Des-AA1,2,4,12,13-[D-Trp8]SRIF 297834 Des-AA1,2,5,12,13-[D-Trp8]SRIF 297835 Des-AA1,2,5,12,13-[D-Trp8,IAmp9]SRIF 297836 Des-AA1,2,4,5,6,12,13-[D-Trp8]SRIF 297837 Des-AA1,2,4,5,11,12,13-[D-Trp8]SRIF 297838 Des-AA1,2,4,5,10,12,13-[D-Trp8]SRIF 297847 1-[4-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phenyl)-butyl]-3-(3,4-difluoro-phenyl)-urea 297850 Des-AA1,2,5-[D-Nal8,IAmp9,(NalphaMe)Ser13]SRIF 297851 Des-AA1,2,5-[D-Nal8,IAmp9,(NalphaMe)Cys14]SRIF 297856 1-[4-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phenyl)-butyl]-3-phenyl-urea 297857 Des-AA1,5-[Tyr2,D-Trp8,IAmp9]SRIF CH-288 297858 cyclo(6-11) Des-AA1,5-[Tyr2,Glu6,D-Trp8,IAmp9,Dab11]SRIF 297869 Des-AA1,2,5-[D-Trp8,IAmp9,(NalphaMe)Ser13]SRIF 297870 Des-AA1,2,5-[D-Trp8,IAmp9,(NalphaMe)Cys14]SRIF 297874 cyclo(6-12) Des-AA1,5-[Tyr2,Glu6,D-Trp8,IAmp9,Lys12]SRIF 297878 Des-AA1,2,5-[(NalphaMe)Cys3,D-Trp8,IAmp9]SRIF 297879 Des-AA1,2,5-[D-Trp8,(NalphaMe)IAmp9]SRIF 297880 Des-AA1,2,5-[D-Trp8,IAmp9,(NalphaMe)Thr12]SRIF 297881 Des-AA1,2,5-[D-Trp8,(NalphaMe)IAmp9,Tyr11]SRIF 297882 Des-AA1,2,5-[D-Trp8,(NalphaMe)IAmp9,m-I-Tyr11]SRIF 297885 1-[4-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phenyl)-butyl]-3-(2-trifluoromethyl-phenyl)-urea 297891 1-[4-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phenyl)-butyl]-3-(3,4-dichloro-phenyl)-urea 297893 1-[4-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phenyl)-butyl]-3-(3,5-dichloro-phenyl)-urea 297895 1-[4-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phenyl)-butyl]-3-(3,5-bis-trifluoromethyl-phenyl)-urea 297901 Des-AA1,2,5-[D-Trp8,IAmp9,(NalphaMe)Ser13]SRIF-(Lys)2 297902 Des-AA1,2,5-[D-Nal8,IAmp9,(NalphaMe)Cys14]SRIF-(Lys)3 297903 Des-AA1,2,5-[D-Nal8,IAmp9,(NalphaMe)Cys14]SRIF-Lys 297904 Des-AA1,2,5-[D-Trp8,IAmp9,(NalphaMe)Cys14]SRIF-(Lys)3 297905 Des-AA1,2,5-[D-Trp8,IAmp9,(NalphaMe)Cys14]SRIF-Lys 297912 Des-AA1,2,5-[D-Trp8,IAmp9,Tyr11]Cbm-SRIF 297913 Des-AA1,2,5-[D-Trp8,(NalphaMe)IAmp9,Tyr11]Cbm-SRIF 297914 Des-AA1,2,5-[D-Trp8,IAmp9,m-I-Tyr11]Cbm-SRIF 297915 Des-AA1,2,5-[D-Trp8,(NalphaMe)IAmp9,m-I-Tyr11]Cbm-SRIF 297916 1-[4-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phenyl)-butyl]-3-m-tolyl-urea 297928 1-(2-Biphenyl-4-yl-4-cyclopentylamino-butyl)-3-(3,5-dichloro-phenyl)-urea 297931 Des-AA1,5-[Tyr2,D-Trp8,(NalphaMe)IAmp9]SRIF 297932 Des-AA1,5-[Tyr2,D-Trp8,IAmp9]Cbm-SRIF 297933 cyclo(7-12) Des-AA1,5-[Tyr2,Glu7,D-Trp8,IAmp9,Dab12]SRIF 297934 cyclo(7-12) Des-AA1,5-[Tyr2,Glu7,D-Trp8,IAmp9,Orn12]SRIF 297935 cyclo(7-12) Des-AA1,5-[Tyr2,Glu7,D-Trp8,IAmp9,Lys12]SRIF 297936 cyclo(7-12) Des-AA1,5-[Tyr2,Glu7,D-Trp8,IAmp9,hLys12]SRIF 297937 cyclo(7-12) Des-AA1,5-[Tyr2,Glu7,D-Trp8,IAmp9,hhLys12]SRIF 297938 cyclo(7-12) Des-AA1,5-[Tyr2,Glu7,D-Trp8,IAmp9,D-hLys12]SRIF 297942 Des-AA1,2,5-[D-Nal8,(NalphaMe)IAmp9,Tyr11]SRIF 297943 Des-AA1,2,5-[D-Nal8,(NalphaMe)IAmp9,Tyr11]Cbm-SRIF 297952 Des-AA1,5-[Tyr2,D-Trp8,(NalphaMe)IAmp9]Cbm-SRIF 297953 Des-AA1,5-[m-I-Tyr2,D-Trp8,(NalphaMe)IAmp9]Cbm-SRIF 297954 Des-AA1,2,5-[D-Trp8,Tyr11]SRIF 297955 Des-AA1,2,5-[D-Trp8,IAmp9,Tyr11]SRIF [Tyr11]CH-275 297956 (4R,7S,10R,13S,16R,19S,22R,25S,28R,31S,34R,37S)-37-{2-[(2S)-2-[(2S)-6-amino-2-[(2S)-2-[(2S)-2-[(2S)-2-{[(2S)-1-[(2S)-2-[(2S)-2-[(2S)-2-{[(2S)-1-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-amino-3-hydroxypropanamido]propanamido]-3-carbamoylpropanamido]-3-hydroxypropanamido]-3-carbamoylpropanoyl]pyrrolidin-2-yl]formamido}propanamido]-4-(methylsulfanyl)butanamido]propanoyl]pyrrolidin-2-yl]formamido}-5-[(diaminomethylidene)amino]pentanamido]-4-carboxybutanamido]-5-[(diaminomethylidene)amino]pentanamido]hexanamido]propanamido]acetamido}-19,34-bis(4-aminobutyl)-13,25,28-tribenzyl-31-(carbamoylmethyl)-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecaazacyclooctatriacontane-4-carboxylic acid 297958 cyclo(7-12) Des-AA1,5-[Tyr2,Glu7,D-Trp8,IAmp9,Dab(betaAla)12]SRIF 297961 Des-AA1,2,5-[D-Agl8(NbetaMe,2-naphthoyl),IAmp9,Tyr11]SRIF 297962 Des-AA1,2,5-[L-Agl8(NbetaMe,2-naphthoyl),IAmp9, Tyr11]SRIF 297963 Des-AA1,2,5-[D-Agl8(NbetaMe,2-naphthoyl),IAmp9, m-I-Tyr11]SRIF 297964 Des-AA1,2,5-[D-Agl8(NbetaMe,2-naphthoyl),IAmp9, m-I-Tyr11]Cbm-SRIF 297965 Des-AA1,2,4,13-[D-Trp8]SRIF 297972 Des-AA5-[D-Trp8]SRIF 297973 Des-AA1,2,5-[D-Trp8,IAmp9]SRIF CH-275 297974 Des-AA1,2,5-[D-Nal8,IAmp9]SRIF 297975 Des-AA1,2,5-[(NalphaMe)Cys3,D-Nal8,IAmp9]SRIF 297976 cyclo(7-12) Des-AA1,5-[Tyr2,Glu7,D-Trp8,IAmp9,Orn(betaAla)12]SRIF 297977 cyclo(7-12) Des-AA1,5-[Tyr2,Glu7,D-Trp8,IAmp9,Orn(Gaba)12]SRIF 297978 cyclo(7-12) Des-AA1,5-[Tyr2,Glu7,D-Trp8,IAmp9,Lys(Gaba)12]SRIF 297979 cyclo(7-12) Des-AA1,5-[m-I-Tyr2,Glu7,D-Trp8,IAmp9,Lys12]SRIF 297981 cyclo(7-12) Des-AA1,2,5-[Glu7,D-Trp8,IAmp9,Tyr11,Lys12]SRIF 297982 cyclo(7-12) Des-AA1,2,5-[Glu7,D-Trp8,(NMe)IAmp9,Tyr11,Lys12]SRIF 297986 1-[4-Cyclopentylamino-2-(4-pyridin-4-yl-phenyl)-butyl]-3-(3,5-dichloro-phenyl)-urea 297987 1-[2-(3'-Cyano-biphenyl-4-yl)-4-ethylamino-butyl]-3-(3,5-dichloro-phenyl)-urea 297989 2-(3-Fluoro-phenyl)-benzo[h]chromen-4-one 297992 4-Thiomorpholin-4-yl-benzo[g]chromen-2-one 297993 4-Morpholino-2H-benzo[h]chromen-2-one 297996 2-Morpholin-4-yl-6-phenyl-chromen-4-one 297997 8-Phenyl-2-piperidin-1-yl-chromen-4-one 297998 8-Methoxy-4-morpholin-4-yl-chromen-2-one 298002 4-morpholino-2H-chromen-2-one 298006 6-Chloro-4-morpholin-4-yl-chromen-2-one 298009 1-[2-(4'-Chloro-biphenyl-4-yl)-4-cyclopentylamino-butyl]-3-(3,5-dichloro-phenyl)-urea 298011 2-Morpholin-4-yl-pyrido[1,2-a]pyrimidin-4-one 298018 2-(3-Hydroxy-pyrrolidin-1-yl)-benzo[h]chromen-4-one 298022 1-[4-Cyclopentylamino-2-(3'-fluoro-biphenyl-4-yl)-butyl]-3-(3,5-dichloro-phenyl)-urea 298023 1-[4-Cyclopentylamino-2-(3'-trifluoromethoxy-biphenyl-4-yl)-butyl]-3-(3,5-dichloro-phenyl)-urea 298026 8-Phenyl-2-thiomorpholin-4-yl-chromen-4-one 298027 4-(4-Oxo-8-phenyl-4H-chromen-2-yl)-1lambda*4*-thiomorpholin-1-ol anion 298030 SID24802694 298031 6-Methyl-4-morpholino-coumarin 298032 2-Thiomorpholin-4-yl-pyrido[1,2-a]pyrimidin-4-one 298038 2-Pyrrolidin-1-yl-pyrimido[2,1-a]isoquinolin-4-one 298041 1-[4-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phenyl)-butyl]-3-(3-methoxy-phenyl)-urea 298046 2-(4-Amino-phenyl)-benzo[h]chromen-4-one 298048 1-Morpholin-4-yl-benzo[f]chromen-3-one 298049 2-morpholino-4H-pyrimido[2,1-a]isoquinolin-4-one 298051 1-[4-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phenyl)-butyl]-3-(4-trifluoromethyl-phenyl)-urea 298053 1-[2-(3'-Cyano-biphenyl-4-yl)-4-cyclopentylamino-butyl]-3-(3,5-dichloro-phenyl)-urea 298057 2-Morpholin-4-yl-benzo[h]chromene-4-thione 298058 8-Methyl-4-morpholin-4-yl-chromen-2-one 298060 2-(2,5-Dihydro-pyrrol-1-yl)-pyrimido[2,1-a]isoquinolin-4-one 298067 2-thiomorpholino-4H-benzo[h]chromen-4-one 298069 2-((R)-3-Hydroxy-pyrrolidin-1-yl)-pyrimido[2,1-a]isoquinolin-4-one 298076 2-(piperidin-1-yl)-4H-benzo[h]chromen-4-one 298079 8-Methyl-2-morpholin-4-yl-chromen-4-one 298082 2-Pyrrolidin-1-yl-benzo[h]chromen-4-one 298084 2-(2-Fluoro-phenyl)-benzo[h]chromen-4-one 298085 1-[2-(3'-Cyano-biphenyl-4-yl)-4-methylamino-butyl]-3-(3,5-dichloro-phenyl)-urea 298086 2-Morpholin-4-yl-7,8,9,10-tetrahydro-benzo[h]chromen-4-one 298091 2-(2,3-Dihydroxy-propylamino)-pyrimido[2,1-a]isoquinolin-4-one 298094 2-morpholino-4H-benzo[g]chromen-4-one 298095 2-(2-Methyl-morpholin-4-yl)-benzo[h]chromen-4-one 298096 2-(2,6-Dimethyl-morpholin-4-yl)-benzo[h]chromen-4-one 298098 1-[2-(3'-Cyano-biphenyl-4-yl)-4-dimethylamino-butyl]-3-(3,5-dichloro-phenyl)-urea 298101 2-[1,4]Oxazepan-4-yl-benzo[h]chromen-4-one 298102 SID26665252 298105 7-Methoxy-2-morpholin-4-yl-chromen-4-one 298106 6-methoxy-4-morpholino-2H-chromen-2-one 298107 1-[2-(3'-Chloro-biphenyl-4-yl)-4-cyclopentylamino-butyl]-3-(3,5-dichloro-phenyl)-urea 298110 1-[2-(4'-Cyano-biphenyl-4-yl)-4-cyclopentylamino-butyl]-3-(3,5-dichloro-phenyl)-urea 298112 3-morpholino-1H-benzo[f]chromen-1-one 298113 4-Morpholin-4-yl-benzo[g]chromen-2-one 298114 7-methoxy-4-morpholino-2H-chromen-2-one 298115 2-((2S,6R)-2,6-Dimethyl-morpholin-4-yl)-pyrimido[2,1-a]isoquinolin-4-one 298116 2-(2,2-Dimethyl-morpholin-4-yl)-pyrimido[2,1-a]isoquinolin-4-one 298122 2-(2,2-Dimethyl-morpholin-4-yl)-benzo[h]chromen-4-one 298124 1-(3-Chloro-phenyl)-3-[2-(3'-cyano-biphenyl-4-yl)-4-dimethylamino-butyl]-urea 298127 (1R,4R)-2-(2-Oxa-5-aza-bicyclo[2.2.1]hept-5-yl)-benzo[h]chromen-4-one 298128 1-[4-Cyclopentylamino-2-(4-pyridin-3-yl-phenyl)-butyl]-3-(3,5-dichloro-phenyl)-urea 298132 N-(4'-{4-[3-(3,5-Dichloro-phenyl)-ureidomethyl]-1-methyl-piperidin-4-yl}-biphenyl-3-yl)-acetamide 298133 2-[(2-Hydroxy-2-phenyl-ethyl)-methyl-amino]-pyrimido[2,1-a]isoquinolin-4-one 298172 1-[2-(3'-Cyano-biphenyl-4-yl)-4-isopropylamino-butyl]-3-(3,5-dichloro-phenyl)-urea 298187 1-(3,5-Dichloro-phenyl)-3-[1-methyl-4-(4-pyridin-3-yl-phenyl)-piperidin-4-ylmethyl]-urea 298192 1-(4-Chloro-phenyl)-3-[2-(3'-cyano-biphenyl-4-yl)-4-dimethylamino-butyl]-urea 298198 1-[2-(3'-Cyano-biphenyl-4-yl)-4-dimethylamino-butyl]-3-(3,4-difluoro-phenyl)-urea 298204 1-[2-(3'-Cyano-biphenyl-4-yl)-4-dimethylamino-butyl]-3-(3,5-difluoro-phenyl)-urea 298214 1-[2-(3'-Cyano-biphenyl-4-yl)-4-dimethylamino-butyl]-3-(4-fluoro-phenyl)-urea 298216 Universal ligand 298228 [(N4-Bzdig)0]BB(7-14) 298229 [(N4-Bzdig)0,Nle14]BB(7-14) 298231 1-[4-(3'-Chloro-biphenyl-4-yl)-1-methyl-piperidin-4-ylmethyl]-3-(3,5-dichloro-phenyl)-urea 298235 1-[2-(3'-Cyano-biphenyl-4-yl)-4-dimethylamino-butyl]-3-(3-fluoro-phenyl)-urea 298240 1-(3,5-Dichloro-phenyl)-3-(1-methyl-4-p-tolyl-piperidin-4-ylmethyl)-urea 298259 1-[2-(3'-Cyano-biphenyl-4-yl)-4-dimethylamino-butyl]-3-phenyl-urea 298260 4-[3-(3,5-Dichloro-phenyl)-ureidomethyl]-4-(4-pyridin-3-yl-phenyl)-piperidine-1-sulfonic acid dimethylamide 298266 1-(3-chloro-4-fluorophenyl)-3-(2-(3'-cyanobiphenyl-4-yl)-4-(dimethylamino)butyl)urea 298267 1-[4-(3'-Cyano-biphenyl-4-yl)-1-cyclohexyl-piperidin-4-ylmethyl]-3-(3,5-dichloro-phenyl)-urea 298268 1-(2-Furan-2-yl-8-propyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-isopropyl-urea 298269 1-Cyclohexyl-3-[2-furan-2-yl-8-(3-methyl-butyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl]-urea 298271 (2-Furan-2-yl-8-phenethyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-ylcarbamoyl)-methyl-ammonium chloride 298272 1-(2-Furan-2-yl-8-octyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-p-tolyl-urea 298274 1-[4-(3'-Cyano-biphenyl-4-yl)-1-(2-methoxy-ethyl)-piperidin-4-ylmethyl]-3-(3,5-dichloro-phenyl)-urea 298275 1-tert-Butyl-3-(2-furan-2-yl-8-propyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-urea 298276 1-[4-(3'-Cyano-biphenyl-4-yl)-1-cyclopropylmethyl-piperidin-4-ylmethyl]-3-(3,5-dichloro-phenyl)-urea 298277 1-[4-(3'-Cyano-biphenyl-4-yl)-1-methyl-piperidin-4-ylmethyl]-3-(3,5-dichloro-phenyl)-urea 298278 1-[2-Furan-2-yl-8-(3-methyl-butyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl]-3-pentyl-urea 298280 1-Cyclohexyl-3-(8-cyclohexylmethyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-urea 298282 1-[2-Furan-2-yl-8-(3-phenyl-propyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl]-3-isopropyl-urea 298284 ethyl 2-[4-({[4-(furan-2-yl)-11-(3-methylbutyl)-3,5,6,8,10,11-hexaazatricyclo[7.3.0.0^{2,6}]dodeca-1(12),2,4,7,9-pentaen-7-yl]carbamoyl}amino)phenyl]acetate 298285 1-(3,5-Dichloro-phenyl)-3-[4-(4-pyridin-3-yl-phenyl)-piperidin-4-ylmethyl]-urea 298287 1-[4-(3'-Cyano-biphenyl-4-yl)-1-propyl-piperidin-4-ylmethyl]-3-(3,5-dichloro-phenyl)-urea 298288 1-[4-(3'-Cyano-biphenyl-4-yl)-1-isopropyl-piperidin-4-ylmethyl]-3-(3,5-dichloro-phenyl)-urea 298289 1-tert-Butyl-3-[2-furan-2-yl-8-(3-phenyl-propyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl]-urea 298292 1-[2-Furan-2-yl-8-(3-methyl-butyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl]-3-p-tolyl-urea 298295 3-(2-Furan-2-yl-8-phenethyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-ylcarbamoyl)-propyl-ammonium chloride 298296 1-(3,5-Dichloro-phenyl)-3-[1-methanesulfonyl-4-(4-pyridin-3-yl-phenyl)-piperidin-4-ylmethyl]-urea 298298 1-[4-(3'-Cyano-biphenyl-4-yl)-1-ethyl-piperidin-4-ylmethyl]-3-(3,5-dichloro-phenyl)-urea 298299 1-[4-(3'-Cyano-biphenyl-4-yl)-1-cyclobutyl-piperidin-4-ylmethyl]-3-(3,5-dichloro-phenyl)-urea 298301 tert-butyl 4-(2-(furan-2-yl)-8-phenethyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-ylamino)-4-oxobutylcarbamate 298302 1-(3,5-Dichloro-phenyl)-3-[4-(3'-formyl-biphenyl-4-yl)-1-methyl-piperidin-4-ylmethyl]-urea 298303 1-[4-(3'-cyano-biphenyl-4-yl)-1-cyclopentyl-piperidin-4-ylmethyl]-3-(3,5-dichloro-phenyl)-urea 298304 1-Cyclohexyl-3-(2-furan-2-yl-8-octyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-urea 298305 1-[1-Butyl-4-(3'-cyano-biphenyl-4-yl)-piperidin-4-ylmethyl]-3-(3,5-dichloro-phenyl)-urea 298306 1-[1-sec-Butyl-4-(3'-cyano-biphenyl-4-yl)-piperidin-4-ylmethyl]-3-(3,5-dichloro-phenyl)-urea 298307 1-(2-Furan-2-yl-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-pentyl-urea 298308 3-[2-Furan-2-yl-8-(3-methyl-butyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-ylcarbamoyl]-propyl-ammonium chloride 298309 1-(2-Furan-2-yl-8-octyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-pentyl-urea 298310 1-tert-Butyl-3-[2-furan-2-yl-8-(3-methyl-butyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl]-urea 298311 {4-[3-(2-Furan-2-yl-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-ureido]-phenyl}-acetic acid ethyl ester 298314 tert-butyl 4-(2-(furan-2-yl)-8-isopentyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-ylamino)-4-oxobutylcarbamate 298316 4'-(2-Butyl-4-oxo-1,3-diaza-spiro[4.4]non-1-en-3-ylmethyl)-2'-ethoxymethyl-biphenyl-2-sulfonic acid (4,5-dimethyl-isoxazol-3-yl)-amide 298317 {4-[3-(2-Furan-2-yl-8-octyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-ureido]-phenyl}-acetic acid ethyl ester 298323 Biphenyl-4-carboxylic acid [4-(3-dimethylamino-pyrrolidin-1-yl)-phenyl]-amide 298343 1-[4-(3'-Cyano-biphenyl-4-yl)-1-methyl-piperidin-4-ylmethyl]-3-phenyl-urea 298352 2-(2-Furan-2-yl-8-phenethyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-ylcarbamoyl)-ethyl-ammonium chloride 298354 1-[4-(3'-Cyano-biphenyl-4-yl)-1-methyl-piperidin-4-ylmethyl]-3-(3-cyano-phenyl)-urea 298355 1-(4-Chloro-3-trifluoromethyl-phenyl)-3-[4-(3'-cyano-biphenyl-4-yl)-1-methyl-piperidin-4-ylmethyl]-urea 298356 1-(8-Cyclohexylmethyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-pentyl-urea 298360 1-(2-Furan-2-yl-8-phenethyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-isopropyl-urea 298361 2-Furan-2-yl-8-octyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 298366 {4-[3-(8-Cyclohexylmethyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-ureido]-phenyl}-acetic acid ethyl ester 298371 1-tert-Butyl-3-(2-furan-2-yl-8-phenethyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-urea 298377 8-Cyclohexylmethyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 298378 1-(8-Cyclohexylmethyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-p-tolyl-urea 298383 1-[2-Furan-2-yl-8-(3-methyl-butyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl]-3-isopropyl-urea 298394 1-Cyclohexyl-3-(2-furan-2-yl-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-urea 298396 1-[4-(3'-Cyano-biphenyl-4-yl)-1-methyl-piperidin-4-ylmethyl]-3-(2,5-dichloro-phenyl)-urea 298399 5-Oxo-5-phenyl-pentanoic acid [4-(3-dimethylamino-pyrrolidin-1-yl)-phenyl]-amide 298402 3,5-Dichloro-N-[4-(3'-cyano-biphenyl-4-yl)-1-methyl-piperidin-4-ylmethyl]-benzenesulfonamide 298404 3,5-Dichloro-N-[4-(3'-cyano-biphenyl-4-yl)-1-methyl-piperidin-4-ylmethyl]-benzamide 298408 1-[4-(3'-Cyano-biphenyl-4-yl)-1-methyl-piperidin-4-ylmethyl]-3-(3,4-difluoro-phenyl)-urea 298416 N-[4-(3'-Cyano-biphenyl-4-yl)-1-methyl-piperidin-4-ylmethyl]-2-(3,5-dichloro-phenyl)-acetamide 298432 N-[4-(3-Dimethylamino-pyrrolidin-1-yl)-phenyl]-6-phenyl-nicotinamide 298474 5-(4-Chloro-phenyl)-5-oxo-pentanoic acid [4-(3-dimethylamino-pyrrolidin-1-yl)-phenyl]-amide 298483 4-(4-Chloro-phenyl)-cyclohexanecarboxylic acid [4-(3-dimethylamino-pyrrolidin-1-yl)-phenyl]-amide 298486 4-Phenyl-cyclohexanecarboxylic acid [4-(3-dimethylamino-pyrrolidin-1-yl)-phenyl]-amide 298504 N-[4-(3-Dimethylamino-pyrrolidin-1-yl)-phenyl]-6-(4-methoxy-phenyl)-nicotinamide 298514 {3-[((R)-4-Fluoro-benzenesulfonyl)-methyl-amino]-1,2,3,4-tetrahydro-carbazol-9-yl}-acetic acid 298521 2-Biphenyl-4-yl-N-[4-(3-dimethylamino-pyrrolidin-1-yl)-phenyl]-acetamide 298525 1-[4-(3-Dimethylamino-pyrrolidin-1-yl)-phenyl]-3-(3-phenyl-propyl)-urea 298538 1-[4-(3-Dimethylamino-pyrrolidin-1-yl)-phenyl]-3-[3-(4-methoxy-phenyl)-propyl]-urea 298626 3,4,5,6-Tetrahydro-2H-[1,2']bipyridinyl-5'-carboxylic acid [4-(3-dimethylamino-pyrrolidin-1-yl)-phenyl]-amide 298638 N-[4-(3-Dimethylamino-pyrrolidin-1-yl)-phenyl]-4-thiophen-2-yl-benzamide 298769 Biphenyl-4-carboxylic acid [4-(3-methylamino-pyrrolidin-1-yl)-phenyl]-amide 298786 Biphenyl-4-carboxylic acid {4-[3-(ethyl-methyl-amino)-pyrrolidin-1-yl]-phenyl}-amide 298809 (3,5-Dimethoxy-phenyl)-(5-phenyl-oxazol-2-yl)-amine 298816 (5-Phenyl-oxazol-2-yl)-(3,4,5-trimethoxy-phenyl)-amine 298832 N,N-Diethyl-4-methoxy-3-(5-phenyl-oxazol-2-ylamino)-benzenesulfonamide 298833 (5-Ethanesulfonyl-2-methoxy-phenyl)-(5-phenyl-oxazol-2-yl)-amine 298835 Naltrindole analogue 298842 Naltrindole analogue 298848 [5-(2-Chloro-phenyl)-oxazol-2-yl]-(5-ethanesulfonyl-2-methoxy-phenyl)-amine 298855 [5-(3-Chloro-phenyl)-oxazol-2-yl]-(5-ethanesulfonyl-2-methoxy-phenyl)-amine 298857 Naltrindole analogue 298865 Biphenyl-4-carboxylic acid {4-[3-(benzyl-methyl-amino)-pyrrolidin-1-yl]-phenyl}-amide 298871 3-[2-(5-Ethanesulfonyl-2-methoxy-phenylamino)-oxazol-5-yl]-benzonitrile 298872 (5-Ethanesulfonyl-2-methoxy-phenyl)-[5-(3-methoxy-phenyl)-oxazol-2-yl]-amine 298891 Biphenyl-4-carboxylic acid {4-[3-(methyl-pyridin-2-ylmethyl-amino)-pyrrolidin-1-yl]-phenyl}-amide 298893 (5-Ethanesulfonyl-2-methoxy-phenyl)-[5-(3-fluoro-phenyl)-oxazol-2-yl]-amine 298908 Biphenyl-4-carboxylic acid {4-[3-(cyclopropylmethyl-methyl-amino)-pyrrolidin-1-yl]-phenyl}-amide 298933 Biphenyl-4-carboxylic acid (4-{3-[methyl-(3-phenyl-propyl)-amino]-pyrrolidin-1-yl}-phenyl)-amide 298957 Biphenyl-4-carboxylic acid {4-[3-(acetyl-methyl-amino)-pyrrolidin-1-yl]-phenyl}-amide 298977 Nociceptin/orphanin FQ analogue 298978 Nociceptin/orphanin FQ analogue 298979 Nociceptin/orphanin FQ analogue 298986 Nociceptin/orphanin FQ analogue 298987 Nociceptin/orphanin FQ analogue 298988 Nociceptin/orphanin FQ analogue 298995 Nociceptin/orphanin FQ analogue 298996 Nociceptin/orphanin FQ analogue 298997 Nociceptin/orphanin FQ analogue 299009 biphenyl-4-carboxylic acid [6-(3-methylamino-pyrrolidin-1-yl)-pyridin-3-yl]-amide 299026 N-(4-(4-(3-chlorobenzyloxy)-3-chlorophenylamino)-3-cyano-7-ethoxyquinolin-6-yl)-4-(dimethylamino)but-2-enamide 299027 4-(4-Methyl-piperazin-1-yl)-but-2-enoic acid [4-(4-benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299028 1-{(E)-3-[4-(4-Benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-ylcarbamoyl]-allyl}-aziridine-2-carboxylic acid methyl ester 299031 4-Dimethylamino-but-2-enoic acid (4-{3-chloro-4-[(1,6-dihydro-pyridin-3-ylmethyl)-amino]-phenylamino}-3-cyano-7-methoxy-quinolin-6-yl)-amide 299033 4-Dimethylamino-but-2-enoic acid [4-(3-chloro-4-pentyloxy-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299035 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(furan-2-ylmethoxy)-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide 299039 2-{2-Chloro-4-[3-cyano-6-(4-dimethylamino-but-2-enoylamino)-7-ethoxy-quinolin-4-ylamino]-phenoxymethyl}-1-methyl-3H-imidazol-1-ium 299040 4-Dimethylamino-but-2-enoic acid {4-[4-(benzothiazol-2-ylmethoxy)-3-chloro-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide 299041 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(quinolin-4-ylmethoxy)-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide 299042 2-{[4-(4-Benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-ylamino]-methyl}-acrylic acid 299045 2-{2-Chloro-4-[3-cyano-6-(4-dimethylamino-but-2-enoylamino)-7-methoxy-quinolin-4-ylamino]-phenylsulfanyl}-1-methyl-3H-imidazol-1-ium 299046 4-Dimethylamino-but-2-enoic acid [4-(1-benzenesulfonyl-1H-indol-5-ylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299047 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(2,4-difluoro-benzyloxy)-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide 299050 4-Dimethylamino-but-2-enoic acid [4-(4-benzyloxy-3-cyano-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299053 4-Dimethylamino-but-2-enoic acid [4-(1-benzyl-2,3-dihydro-1H-indol-5-ylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299054 4-(2-Methoxymethyl-pyrrolidin-1-yl)-but-2-enoic acid [4-(4-benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299055 4-Piperidin-1-yl-but-2-enoic acid [4-(4-benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299056 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(thiophen-2-ylmethoxy)-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide 299057 4-(1,4,7-Trioxa-10-aza-cyclododec-10-yl)-but-2-enoic acid [4-(4-benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299058 4-Pyrrolidin-1-yl-but-2-enoic acid [4-(4-benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299062 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(phenylaminomethyl-amino)-phenylamino]-3-cyano-7-methoxy-quinolin-6-yl}-amide 299064 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(3-methyl-benzyloxy)-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide 299068 4-Dimethylamino-but-2-enoic acid [4-(3-chloro-4-phenoxy-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299069 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(naphthalen-1-ylmethoxy)-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide 299070 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(naphthalen-2-ylmethoxy)-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide 299071 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(2-chloro-benzyloxy)-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide 299077 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(2-fluoro-benzyloxy)-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide 299080 4-Dimethylamino-but-2-enoic acid [4-(3-chloro-4-morpholin-4-yl-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299081 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-((S)-indan-1-yloxy)-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide 299082 4-Azetidin-1-yl-but-2-enoic acid [4-(4-benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299083 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(3-fluoro-benzyloxy)-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide 299084 4-(4-Methoxy-piperidin-1-yl)-but-2-enoic acid [4-(4-benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299085 4-(4,4-Dihydroxy-piperidin-1-yl)-but-2-enoic acid [4-(4-benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299088 4-Dimethylamino-but-2-enoic acid [4-(4-benzyloxy-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299089 N-[4-(4-Benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-3-(1H-imidazol-4-yl)-acrylamide 299090 N-[4-(4-Benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-2-morpholin-4-ylmethyl-acrylamide 299091 4-Dimethylamino-but-2-enoic acid (4-{3-chloro-4-[(naphthalen-1-ylmethyl)-amino]-phenylamino}-3-cyano-7-ethoxy-quinolin-6-yl)-amide 299092 4-Dimethylamino-but-2-enoic acid [4-(3-chloro-4-cyclohexylmethoxy-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299097 4-Dimethylamino-but-2-enoic acid [4-(4-benzylamino-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299099 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(4-fluoro-benzyloxy)-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide 299108 Ethenesulfonic acid [4-(4-benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299110 4-Dimethylamino-but-2-enoic acid [4-(4-benzyloxy-3-chloro-phenylamino)-3-cyano-7-methoxy-quinolin-6-yl]-amide 299111 4-(2,6-Dimethyl-piperidin-1-yl)-but-2-enoic acid [4-(4-benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299115 4-Dimethylamino-but-2-enoic acid [4-(4-benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299116 4-Dimethylamino-but-2-enoic acid {3-cyano-4-[3,5-dichloro-4-(3-fluoro-benzyloxy)-phenylamino]-7-ethoxy-quinolin-6-yl}-amide 299117 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(3,5-difluoro-benzyloxy)-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide 299120 neratinib 299123 4-Dimethylamino-but-2-enoic acid [4-(3-chloro-4-phenethyloxy-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299124 4-Diisopropylamino-but-2-enoic acid [4-(4-benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299125 4-Dimethylamino-but-2-enoic acid [4-(1-benzyl-1H-indol-5-ylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299126 4-[(2-Methoxy-ethyl)-methyl-amino]-but-2-enoic acid [4-(4-benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299127 4-[(2-Hydroxy-ethyl)-methyl-amino]-but-2-enoic acid [4-(4-benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299132 4-Dimethylamino-but-2-enoic acid [4-(4-benzylamino-3-chloro-phenylamino)-3-cyano-7-methoxy-quinolin-6-yl]-amide 299134 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(4-chloro-benzyloxy)-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide 299136 4-Dimethylamino-but-2-enoic acid [4-(3-chloro-4-imidazol-1-yl-phenylamino)-3-cyano-7-methoxy-quinolin-6-yl]-amide 299137 N-(4-(3-chloro-4-(5-phenylthiazol-2-ylthio)phenylamino)-3-cyano-7-methoxyquinolin-6-yl)-4-(dimethylamino)but-2-enamide 299138 N-(4-(3-chloro-4-(4-phenylthiazol-2-ylthio)phenylamino)-3-cyano-7-ethoxyquinolin-6-yl)-4-(dimethylamino)but-2-enamide 299144 N-[4-(4-Benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-2-dimethylaminomethyl-acrylamide 299145 4-Dimethylamino-but-2-enoic acid [4-(4-benzyloxy-phenylamino)-3-cyano-7-methoxy-quinolin-6-yl]-amide 299146 4-Morpholin-4-yl-but-2-enoic acid [4-(4-benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299147 4-Thiomorpholin-4-yl-but-2-enoic acid [4-(4-benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299149 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(pyrimidin-2-ylsulfanyl)-phenylamino]-3-cyano-7-methoxy-quinolin-6-yl}-amide 299150 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(3-cyano-benzyloxy)-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide 299152 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(pyridin-3-ylmethoxy)-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide 299156 4-Dimethylamino-but-2-enoic acid [4-(4-benzyloxy-3,5-dichloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299158 4-Dimethylamino-but-2-enoic acid [4-(1-benzyl-1H-indazol-5-ylamino)-3-cyano-7-methoxy-quinolin-6-yl]-amide 299160 4-[Bis-(2-hydroxy-propyl)-amino]-but-2-enoic acid [4-(4-benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299162 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(pyridin-4-yloxy)-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide 299163 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(4-phenyl-thiazol-2-ylmethyl)-phenylamino]-3-cyano-7-methoxy-quinolin-6-yl}-amide 299164 3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-fluoro-phenyl)-6-methyl-1-(2-trifluoromethyl-benzyl)-1H-pyrimidine-2,4-dione 299166 1-(2,6-Difluoro-benzyl)-3-((R)-2-dimethylamino-3-methyl-butyl)-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 299171 1-(2,6-Difluoro-benzyl)-3-((S)-2-dimethylamino-2-phenyl-ethyl)-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 299174 1-(2,6-Difluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-3-[(S)-2-(methyl-pyridin-2-ylmethyl-amino)-propyl]-1H-pyrimidine-2,4-dione 299175 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-6-methyl-5-(4-methylsulfanyl-phenyl)-1H-pyrimidine-2,4-dione 299176 5-Benzo[1,3]dioxol-5-yl-1-(2,6-difluoro-benzyl)-6-methyl-3-((R)-2-methylamino-2-phenyl-ethyl)-1H-pyrimidine-2,4-dione 299178 3-((R)-2-Amino-2-phenyl-ethyl)-1-cyclopropylmethyl-5-(2-fluoro-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 299179 3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-fluoro-phenyl)-1-(5-fluoro-2-trifluoromethyl-benzyl)-6-methyl-1H-pyrimidine-2,4-dione 299187 3-[(2R)-amino-2-phenylethyl]-1-(2,6-difluorobenzyl)-5-(2-fluoro-3-methoxyphenyl)-6-methylpyrimidin-2,4-dione 299192 1-(2,6-Difluoro-benzyl)-3-((S)-2-dimethylamino-3-methyl-butyl)-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 299195 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2-bromo-benzyl)-5-(2-fluoro-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 299196 3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-fluoro-phenyl)-1-isobutyl-6-methyl-1H-pyrimidine-2,4-dione 299197 (R)-1-(2-chloro-6-fluorobenzyl)-3-(2-amino-2-phenylethyl)-5-(2-fluorophenyl)-6-methylpyrimidine-2,4(1H,3H)-dione 299198 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-6-methyl-5-(4-phenoxy-phenyl)-1H-pyrimidine-2,4-dione 299203 3-((S)-2-Cyclobutylamino-propyl)-1-(2,6-difluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 299210 1-(2,6-Difluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-3-((R)-2-methylamino-2-phenyl-ethyl)-1H-pyrimidine-2,4-dione 299211 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(thiazol-2-ylsulfanyl)-phenylamino]-3-cyano-7-methoxy-quinolin-6-yl}-amide 299212 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(2-methoxy-benzyloxy)-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide 299213 4-Dimethylamino-but-2-enoic acid {4-[4-(4-benzyloxy-benzyloxy)-3-chloro-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide 299214 3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-fluoro-phenyl)-1-(2-methoxy-ethyl)-6-methyl-1H-pyrimidine-2,4-dione 299215 3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-chloro-phenyl)-1-(2,6-difluoro-benzyl)-6-methyl-1H-pyrimidine-2,4-dione 299217 3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-fluoro-phenyl)-6-methyl-1-(2-methyl-benzyl)-1H-pyrimidine-2,4-dione 299218 4-Dimethylamino-but-2-enoic acid [4-(3-benzyloxy-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299219 4-(1H-Imidazol-4-yl)-but-2-enoic acid [4-(4-benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299220 N-[4-(4-Benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-3-quinolin-8-yl-acrylamide 299221 3-((S)-2-Amino-2-cyclohexyl-ethyl)-1-(2,6-difluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 299229 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-((R)-1-phenyl-ethoxy)-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide 299233 (R)-1-(2,6-difluorobenzyl)-3-(2-amino-2-phenylethyl)-5-(2-fluorophenyl)-6-methylpyrimidine-2,4(1H,3H)-dione 299237 4-Dimethylamino-but-2-enoic acid [4-(3-chloro-4-imidazol-1-ylmethyl-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 299238 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-((R)-indan-1-yloxy)-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide 299245 3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-fluoro-phenyl)-1-(2-methoxy-benzyl)-6-methyl-1H-pyrimidine-2,4-dione 299246 4-Dimethylamino-but-2-enoic acid {4-[4-(benzyl-methyl-amino)-3-chloro-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide 299247 N-[4-(4-Benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-3-(2-dimethylamino-phenyl)-acrylamide 299248 (R)-1-(2,6-difluorobenzyl)-3-(2-amino-2-phenylethyl)-5-(3-methoxyphenyl)-6-methylpyrimidine-2,4(1H,3H)-dione 299250 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-5-(2-fluoro-3-methyl-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 299254 4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-((S)-1-phenyl-ethoxy)-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide 299264 1-(2,6-Difluoro-benzyl)-5-(2,3-dihydro-benzo[1,4]dioxin-6-yl)-6-methyl-3-((R)-2-methylamino-2-phenyl-ethyl)-1H-pyrimidine-2,4-dione 299265 3-((R)-2-Amino-2-phenyl-ethyl)-5-benzo[1,3]dioxol-5-yl-1-(2,6-difluoro-benzyl)-6-methyl-1H-pyrimidine-2,4-dione 299266 1-(2,6-Difluoro-benzyl)-3-((R)-2-dimethylamino-2-phenyl-ethyl)-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 299267 3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-fluoro-phenyl)-6-methyl-1-(2-trifluoromethylsulfanyl-benzyl)-1H-pyrimidine-2,4-dione 299270 3-((S)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 299272 1-(2,6-Difluoro-benzyl)-5-(3-methoxy-phenyl)-6-methyl-3-((R)-2-methylamino-2-phenyl-ethyl)-1H-pyrimidine-2,4-dione 299275 1-(2,6-Difluoro-benzyl)-3-((S)-2-dimethylamino-4-methyl-pentyl)-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 299280 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-5-(2,3-dihydro-benzo[1,4]dioxin-6-yl)-6-methyl-1H-pyrimidine-2,4-dione 299284 {4''-[3-((2R,5R)-2,5-Dimethyl-pyrrolidin-1-yl)-propoxy]-biphenyl-4-yl}-morpholin-4-yl-methanone 299285 3-((R)-2-Amino-2-phenyl-ethyl)-1-benzyl-5-(2-fluoro-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 299290 2-(4-Benzyloxy-phenyl)-N-[1-(2-pyrrolidin-1-yl-ethyl)-1H-benzoimidazol-5-yl]-acetamide 299302 2-(4-Benzyl-piperidin-1-ylmethyl)-3,4-dihydro-2H-naphthalen-1-one 299311 3-((R)-2-Amino-2-phenyl-ethyl)-1-(4-fluoro-benzyl)-5-(2-fluoro-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 299315 2-(4-(benzyloxy)phenyl)-N-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-6-yl)acetamide 299327 3-((R)-2-Amino-2-phenyl-ethyl)-1-(3-fluoro-benzyl)-5-(2-fluoro-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 299330 2-(4-(benzyloxy)phenyl)-N-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)acetamide 299331 3-((R)-2-Amino-2-phenyl-ethyl)-1-cyclohexylmethyl-5-(2-fluoro-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 299332 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2-chloro-4-fluoro-benzyl)-5-(2-fluoro-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 299345 2-(4-Phenoxy-benzylamino)-N-[3-(2-pyrrolidin-1-yl-ethyl)-3H-benzoimidazol-5-yl]-acetamide 299350 3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-fluoro-phenyl)-6-methyl-1-phenethyl-1H-pyrimidine-2,4-dione 299352 (R)-1-(2-fluorobenzyl)-3-(2-amino-2-phenylethyl)-5-(2-fluorophenyl)-6-methylpyrimidine-2,4(1H,3H)-dione 299356 2-(4-(benzyloxy)phenyl)-N-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-4-yl)acetamide 299363 2-(4-Benzyloxy-phenyl)-N-[3-(2-pyrrolidin-1-yl-ethyl)-3H-benzoimidazol-5-yl]-acetamide 299367 3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-fluoro-phenyl)-6-methyl-1-pyridin-2-ylmethyl-1H-pyrimidine-2,4-dione 299372 2-(4-Benzyloxy-phenyl)-N-[2-(2-pyrrolidin-1-yl-ethyl)-2H-indazol-6-yl]-acetamide 299376 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2-chloro-benzyl)-5-(2-fluoro-phenyl)-6-methyl-1H-pyrimidine-2,4-dione 299388 2-(4-Benzyloxy-phenyl)-N-[1-(2-pyrrolidin-1-yl-ethyl)-2H-indazol-5-yl]-acetamide 299390 3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-fluoro-phenyl)-6-methyl-1-pyridin-3-ylmethyl-1H-pyrimidine-2,4-dione 299401 2-(4-Benzyloxy-phenyl)-N-[1-(2-pyrrolidin-1-yl-ethyl)-2H-indazol-4-yl]-acetamide 299416 (3-Chloro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-methanone 299419 4-Benzyl-1-chroman-3-ylmethyl-piperidine 299421 Cyclopropyl-[2-(4-cyclopropyl-piperazin-1-yl)-quinolin-6-yl]-methanone 299426 1-Benzyl-4-(1,2,3,4-tetrahydro-naphthalen-2-ylmethyl)-piperazine 299427 2-(4-Cyclopentyl-piperazin-1-yl)-quinoline 299428 (R)-2-Quinolin-2-yl-octahydro-pyrido[1,2-a]pyrazine 299434 (3,5-Difluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-methanone 299435 {2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-phenyl-methanone 299437 3-{2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-benzonitrile 299448 Cyclopropyl-(4-{2-[2-((R)-2-methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-phenyl)-methanone 299451 6-Chloro-2-(4-cyclopropyl-piperazin-1-yl)-quinoline 299455 1-(3-{2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-phenyl)-ethanone 299456 {2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-p-tolyl-methanone 299457 (4-Methoxy-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-methanone 299458 7-Chloro-2-(4-cyclopropyl-piperazin-1-yl)-quinoline 299462 3-(4-Benzyl-piperidin-1-ylmethyl)-chroman-4-one 299463 3-(4-Benzyl-piperidin-1-ylmethyl)-chromen-4-one 299464 1-(3-{2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-phenyl)-propan-1-ol 299467 1-benzyl-4-((3,4-dihydro-2H-chromen-2-yl)methyl)piperazine 299469 4-{2-[2-((S)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-benzonitrile 299470 (2-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-methanone 299473 5,7-Dichloro-2-(4-cyclopropyl-piperazin-1-yl)-quinoline 299474 2-(4-Cyclopropyl-piperazin-1-yl)-6-methoxy-quinoline 299479 1-(3-{2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-phenyl)-ethanol 299480 (3-{2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-phenyl)-methanol 299481 (4-Dimethylamino-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-methanone 299482 (4-Fluoro-3-methyl-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-methanone 299484 1-[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-piperazin-1-yl]-5-[1,2]dithiolan-3-yl-pentan-1-one 299490 1-Benzyl-4-(2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-piperazine 299491 2-(4-Cyclopropyl-piperazin-1-yl)-6-trifluoromethyl-quinoline 299492 (3-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-methanone 299503 4-Benzyl-1-chroman-2-ylmethyl-piperidine 299504 4-Benzyl-1-(2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-piperidine 299505 1-[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-piperazin-1-yl]-2-[1,2]dithiolan-3-yl-ethanone 299508 (4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-methanone 299509 4-Benzyl-1-indan-2-ylmethyl-piperidine 299510 4-Benzyl-1-(1,2,3,4-tetrahydro-naphthalen-2-ylmethyl)-piperidine 299513 2-(4-Cyclopropyl-piperazin-1-yl)-quinoline-6-carbonitrile 299514 6-Cyclohexyl-2-(4-cyclopropyl-piperazin-1-yl)-quinoline 299516 (4-Chloro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-methanone 299519 Furan-2-carboxylic acid ((R)-2-{4-[3-(4-cyclopropanecarbonyl-phenoxy)-propyl]-piperazin-1-yl}-1-methyl-2-oxo-ethyl)-amide 299526 1-(3-{2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-phenyl)-propan-1-one 299528 2-(4-Benzyl-piperidin-1-ylmethyl)-chroman-4-one 299529 2-(4-Benzyl-piperazin-1-ylmethyl)-3,4-dihydro-2H-naphthalen-1-one 299536 4-Benzyl-1-(7-methoxy-1,2,3,4-tetrahydro-naphthalen-2-ylmethyl)-piperidine 299542 2-(4-Cyclopropyl-piperazin-1-yl)-6-pyrazol-1-yl-quinoline 299543 [2-(4-Cyclopropyl-piperazin-1-yl)-quinolin-6-yl]-(4-fluoro-phenyl)-methanone 299544 4-Benzyl-1-(8-methoxy-1,2,3,4-tetrahydro-naphthalen-2-ylmethyl)-piperidine 299545 (4-Chloro-3-methyl-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-methanone 299546 Cyclopropyl-(3-{2-[2-((R)-2-methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-phenyl)-methanone 299547 (4-{2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-phenyl)-methanol 299568 [4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-piperazin-1-yl]-[1,2]dithiolan-3-yl-methanone 299576 2-(4-Propyl-piperazin-1-yl)-quinoline 299603 2-(4-Isopropyl-piperazin-1-yl)-quinoline 299604 2-[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-piperazin-1-yl]-[1,4]naphthoquinone 299636 2-[4-(1-Ethyl-propyl)-piperazin-1-yl]-quinoline 299647 2-(4-Cyclopropyl-piperazin-1-yl)-quinoline 299780 9-(4-Methyl-piperazin-1-yl)-3,4-dithia-7a-aza-cyclopenta[f]azulene 299800 11-(4-Methyl-piperazin-1-yl)-5H-benzo[e]pyrrolo[1,2-a]azepine 299805 8-Chloro-11-(4-methyl-piperazin-1-yl)-5H-benzo[e]pyrrolo[1,2-a]azepine 299819 3-Methyl-11-(4-methyl-piperazin-1-yl)-5H-benzo[e]pyrrolo[1,2-a]azepine 299877 1-(2-Methoxy-phenyl)-4-[1-(2-trifluoromethyl-phenyl)-1H-pyrrol-3-ylmethyl]-piperazine 299879 [4-(2-Methyl-1-propyl-1H-indole-3-carbonyl)-naphthalen-2-ylcarbamoyl]-methyl-ammonium chloride 299887 (3S,4aR,6S,8R,8aR,10aR)-6-Acetoxy-3-furan-3-yl-4a,8a-dimethyl-1,5-dioxo-dodecahydro-2-oxa-phenanthrene-8-carboxylic acid methyl ester 299896 (3S,4aR,6S,8R,8aR,10aR)-3-Furan-3-yl-6-methoxymethoxy-4a,8a-dimethyl-1,5-dioxo-dodecahydro-2-oxa-phenanthrene-8-carboxylic acid methyl ester 299949 1-(2-methoxyphenyl)-4-((1-o-tolyl-1H-pyrrol-3-yl)methyl)piperazine 299966 methyl 2-(3-((4-(2-methoxyphenyl)piperazin-1-yl)methyl)-1H-pyrrol-1-yl)-3-methylbenzoate 299997 (2-Methyl-1-propyl-1H-indol-3-yl)-(3-nitro-naphthalen-1-yl)-methanone 299998 (3S,4aR,6S,8R,8aR,10aR)-3-Furan-3-yl-6-hydroxy-4a,8a-dimethyl-1,5-dioxo-dodecahydro-2-oxa-phenanthrene-8-carboxylic acid methyl ester 300019 (3-Amino-naphthalen-1-yl)-(2-methyl-1-propyl-1H-indol-3-yl)-methanone 300042 2-(3-((4-(2-methoxyphenyl)piperazin-1-yl)methyl)-1H-pyrrol-1-yl)benzonitrile 300044 (4-Benzyloxy-3-chloro-phenyl)-(1,3,8a,9-tetraaza-fluoren-4-yl)-amine 300073 4-(6-Chloro-3-piperidin-4-yl-indole-1-sulfonyl)-phenylamine 300084 4-[5-Methoxy-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-indole-1-sulfonyl]-phenylamine 300103 (2-Benzyl-1H-benzoimidazol-5-yl)-(1,3,8a,9-tetraaza-fluoren-4-yl)-amine 300114 [3-Chloro-4-(3-fluoro-benzyloxy)-phenyl]-(1,3,8a,9-tetraaza-fluoren-4-yl)-amine 300135 1-(2-Chloro-benzenesulfonyl)-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole 300151 1-(2-Fluoro-benzenesulfonyl)-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole 300180 (3-Chloro-4-fluoro-phenyl)-(1,3,8a,9-tetraaza-fluoren-4-yl)-amine 300181 4-[3-(1,2,3,6-Tetrahydro-pyridin-4-yl)-indole-1-sulfonyl]-phenylamine 300198 5-Fluoro-3-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-cyclohexyl}-1H-indole 300222 3-{4-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-cyclohexyl}-5-fluoro-1H-indole 300316 5-Fluoro-3-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-cyclohexyl}-1H-indole 300326 6-[4-(4-Benzoimidazol-1-yl-piperidin-1-ylmethyl)-phenyl]-5-phenyl-nicotinonitrile 300327 3-(2,6-Dichloro-phenyl)-5-methyl-isoxazole-4-carboxylic acid (4-diethylamino-2-trifluoromethyl-phenyl)-amide 300332 (2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-[4-(5-fluoro-1H-indol-3-yl)-cyclohexyl]-amine 300333 5-Fluoro-3-[cis-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl]-1H-indole 300340 3-(2-Chloro-phenyl)-5-methyl-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 300341 6-{4-[4-(2-Methyl-benzoimidazol-1-yl)-piperidin-1-ylmethyl]-phenyl}-5-phenyl-nicotinonitrile 300342 3-(2,6-Dichloro-phenyl)-5-methyl-isoxazole-4-carboxylic acid (4-diethylamino-2-methyl-phenyl)-amide 300347 3-(2-Bromo-phenyl)-5-methyl-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 300348 3-(2,6-Dichloro-phenyl)-5-methyl-isoxazole-4-carboxylic acid [2-(2-methyl-1,2,3,4-tetrahydro-isoquinolin-1-ylmethyl)-phenyl]-amide 300349 5-Fluoro-3-[trans-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl]-1H-indole 300355 5-Phenyl-6-{4-[(4-[1,2,3]thiadiazol-4-yl-benzylamino)-methyl]-phenyl}-nicotinonitrile 300362 5-Methyl-3-(2-nitro-phenyl)-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 300363 3-(2,6-Dichloro-phenyl)-5-methyl-isoxazole-4-carboxylic acid (2-diethylcarbamoyl-phenyl)-amide 300375 6-{4-[4-(6-Fluoro-1H-benzoimidazol-2-yl)-piperidin-1-ylmethyl]-phenyl}-5-phenyl-nicotinonitrile 300382 3-Biphenyl-2-yl-5-methyl-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 300383 3-(2,6-Dichloro-phenyl)-5-methyl-isoxazole-4-carboxylic acid [2-(piperidine-1-carbonyl)-phenyl]-amide 300402 3-(2-Methoxy-phenyl)-5-methyl-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 300403 3-(3-Chloro-phenyl)-5-methyl-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 300410 3-(2,6-Dichloro-phenyl)-5-methyl-isoxazole-4-carboxylic acid [2-(azepane-1-carbonyl)-phenyl]-amide 300417 6-{4-[4-(6-Methyl-1H-benzoimidazol-2-yl)-piperidin-1-ylmethyl]-phenyl}-5-phenyl-nicotinonitrile 300432 6-{4-[4-(1H-Benzoimidazol-2-yl)-piperidin-1-ylmethyl]-phenyl}-5-phenyl-nicotinonitrile 300437 3-(2,6-dichloro-phenyl)-5-methyl-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 300438 5-Methyl-3-phenyl-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 300439 3-(4-Chloro-phenyl)-5-methyl-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 300440 3-(2,6-Dichloro-phenyl)-5-methyl-isoxazole-4-carboxylic acid (2-cyano-4-diethylamino-phenyl)-amide 300447 3-{4-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-cyclohexyl}-5-fluoro-1H-indole 300453 2-(1-{4-[3-Phenyl-5-(1H-tetrazol-5-yl)-pyridin-2-yl]-benzyl}-piperidin-4-yl)-1H-benzoimidazole 300458 3-(2,6-Dichloro-phenyl)-5-(2-[1,3]dioxan-2-yl-ethyl)-isoxazole-4-carboxylic acid (4-diethylamino-2-methyl-phenyl)-amide 300462 [4-(5-Fluoro-1H-indol-3-yl)-cyclohexyl]-[2-(1H-indol-4-yloxy)-ethyl]-amine 300463 1-{1-[4-(6-Hydroxy-5-isobutyl-3-phenyl-1,6-dihydro-pyrazin-2-yl)-benzyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 300471 1-(1-{4-[3-Phenyl-5-(1H-tetrazol-5-yl)-pyridin-2-yl]-benzyl}-piperidin-4-yl)-1H-benzoimidazole 300472 3-(2,6-Dichloro-phenyl)-5-methyl-isoxazole-4-carboxylic acid [4-(ethyl-propyl-amino)-phenyl]-amide 300479 [4-(5-Fluoro-1H-indol-3-yl)-cyclohexyl]-[2-(1H-indol-4-yloxy)-ethyl]-amine 300482 3-(2,6-Dichloro-phenyl)-5-(2-[1,3]dioxan-2-yl-ethyl)-isoxazole-4-carboxylic acid [2-(piperidine-1-carbonyl)-phenyl]-amide 300486 1-{1-[4-(3-Phenyl-quinolin-2-yl)-benzyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 300491 3-(2,6-Dichloro-phenyl)-5-methyl-isoxazole-4-carboxylic acid (4-diethylamino-2-ethyl-phenyl)-amide 300492 [4-(5-Fluoro-1H-indol-3-yl)-cyclohexyl]-[2-(2-methoxy-phenoxy)-ethyl]-amine 300493 3-(2,6-Dichloro-phenyl)-5-methyl-isoxazole-4-carboxylic acid {4-[ethyl-(2-hydroxy-ethyl)-amino]-phenyl}-amide 300503 (2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-[4-(5-fluoro-1H-indol-3-yl)-cyclohexyl]-amine 300510 {4-[3-Phenyl-5-(1H-tetrazol-5-yl)-pyridin-2-yl]-benzyl}-(4-[1,2,3]thiadiazol-4-yl-benzyl)-amine 300511 3-(2,6-Dichloro-phenyl)-5-methyl-isoxazole-4-carboxylic acid (4-diethylamino-2-ethyl-phenyl)-amide 300512 1-{1-[4-(2-Phenyl-quinolin-3-yl)-benzyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 300519 [4-(5-Fluoro-1H-indol-3-yl)-cyclohexyl]-[2-(2-methoxy-phenoxy)-ethyl]-amine 300521 2-Methyl-1-(1-{4-[3-phenyl-5-(1H-tetrazol-5-yl)-pyridin-2-yl]-benzyl}-piperidin-4-yl)-1H-benzoimidazole 300522 1-(1-(4-(5-(1-methyl-1H-tetrazol-5-yl)-3-phenylpyridin-2-yl)benzyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one 300524 3-(2,6-Dichloro-phenyl)-5-methyl-isoxazole-4-carboxylic acid (2-benzylcarbamoyl-phenyl)-amide 300535 6-Fluoro-2-(1-{4-[3-phenyl-5-(1H-tetrazol-5-yl)-pyridin-2-yl]-benzyl}-piperidin-4-yl)-1H-benzoimidazole 300540 3-(2,6-Dichloro-phenyl)-5-methyl-isoxazole-4-carboxylic acid {2-[(benzo[1,3]dioxol-5-ylmethyl)-carbamoyl]-phenyl}-amide 300544 [2-(2,3-Dihydro-benzo[1,4]dioxin-5-yloxy)-ethyl]-[4-(5-fluoro-1H-indol-3-yl)-cyclohexyl]-amine 300558 6-Methyl-2-(1-{4-[3-phenyl-5-(1H-tetrazol-5-yl)-pyridin-2-yl]-benzyl}-piperidin-4-yl)-1H-benzoimidazole 300562 3-(2,6-Dichloro-phenyl)-5-(2-[1,3]dioxan-2-yl-ethyl)-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 300566 3-(2,6-Dichloro-phenyl)-5-methyl-isoxazole-4-carboxylic acid [4-(ethyl-methyl-amino)-phenyl]-amide 300567 [2-(2,3-Dihydro-benzo[1,4]dioxin-5-yloxy)-ethyl]-[4-(5-fluoro-1H-indol-3-yl)-cyclohexyl]-amine 300575 1-(1-(4-(6-methyl-5-oxo-3-phenyl-4,5-dihydropyrazin-2-yl)benzyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one 300585 4-(4-Fluoro-phenyl)-2-(4-propyl-piperazin-1-yl)-5,6,7,8,9,10-hexahydro-cycloocta[b]pyridine 300586 1-{4-[4-(4-{4-[bis(4-fluorophenyl)methyl]piperazin-1-yl}butoxy)phenyl]but-3-yn-1-yl}-1-hydroxyurea 300587 N-hydroxycarbamate derivative 300588 N-hydroxycarbamate derivative 300589 N-hydroxycarbamate derivative 300591 5-[(S)-4-(Benzenesulfonyl-methyl-amino)-3-methyl-3-phenyl-butyl]-octahydro-pyrrolo[3,2-c]pyridine-1-carboxylic acid tert-butyl ester 300600 N*5*-(4-Amino-cyclohexyl)-3-chloro-N*7*-[4-(thiophene-2-sulfonyl)-phenyl]-pyrazolo[1,5-a]pyrimidine-5,7-diamine 300605 N-hydroxycarbamate derivative 300606 N-hydroxycarbamate derivative 300608 4-[5-(4-Diethylamino-cyclohexylamino)-3-isopropyl-pyrazolo[1,5-a]pyrimidin-7-ylamino]-N,N-dimethyl-benzenesulfonamide 300622 4-[5-(4-Amino-cyclohexyloxy)-3-isopropyl-pyrazolo[1,5-a]pyrimidin-7-ylamino]-N,N-dimethyl-benzenesulfonamide 300623 4-(4-Fluoro-phenyl)-2-(4-propyl-piperazin-1-yl)-5,6,7,8,9,10-hexahydro-cycloocta[b]pyridin-7-ol 300641 4-[5-(3-Amino-cyclohexylamino)-3-isopropyl-pyrazolo[1,5-a]pyrimidin-7-ylamino]-N,N-dimethyl-benzenesulfonamide 300642 (R)-4-(4-Fluoro-phenyl)-2-(4-propyl-piperazin-1-yl)-5,6,7,8,9,10-hexahydro-cycloocta[b]pyridin-7-ol 300656 (S)-4-(4-Fluoro-phenyl)-2-(4-propyl-piperazin-1-yl)-5,6,7,8,9,10-hexahydro-cycloocta[b]pyridin-8-ol 300660 5-[4-(Benzenesulfonyl-methyl-amino)-3-methyl-3-phenyl-butyl]-octahydro-pyrrolo[3,2-c]pyridine-1-carboxylic acid tert-butyl ester 300661 5-[4-(Benzenesulfonyl-methyl-amino)-3-methyl-3-phenyl-butyl]-octahydro-pyrrolo[3,2-c]pyridine-1-carboxylic acid 4-nitro-benzyl ester 300663 4-(5-Isobutoxy-3-isopropyl-pyrazolo[1,5-a]pyrimidin-7-ylamino)-N,N-dimethyl-benzenesulfonamide 300664 N-Methyl-N-{(S)-4-[4-((R)-2-oxo-5-phenyl-oxazolidin-3-yl)-piperidin-1-yl]-2-phenyl-butyl}-benzenesulfonamide 300669 4-[5-(4-Amino-cyclohexylamino)-3-chloro-pyrazolo[1,5-a]pyrimidin-7-ylamino]-N,N-dimethyl-benzenesulfonamide 300676 N-Methyl-N-[(S)-2-methyl-4-(1-methyl-2-oxo-octahydro-[1,6]naphthyridin-6-yl)-2-phenyl-butyl]-benzenesulfonamide 300678 (5-Isobutoxy-3-isopropyl-pyrazolo[1,5-a]pyrimidin-7-yl)-(4-methanesulfonyl-phenyl)-amine 300680 N-Methyl-N-{(S)-4-[4-((R)-4-methyl-2-(S)-oxo-5-phenyl-oxazolidin-3-yl)-piperidin-1-yl]-2-phenyl-butyl}-benzenesulfonamide 300686 4-[5-(4-Amino-cyclohexylamino)-3-bromo-pyrazolo[1,5-a]pyrimidin-7-ylamino]-N,N-dimethyl-benzenesulfonamide 300689 4-(4-Fluoro-phenyl)-2-(4-propyl-piperazin-1-yl)-5,6,7,8,9,10-hexahydro-cycloocta[b]pyridin-8-ol 300691 N-[(S)-4-(1-Benzyl-2-oxo-octahydro-[1,6]naphthyridin-6-yl)-2-methyl-2-phenyl-butyl]-N-methyl-benzenesulfonamide 300692 N-Methyl-N-{(S)-2-methyl-4-[1-(4-nitro-benzyl)-2-oxo-octahydro-[1,6]naphthyridin-6-yl]-2-phenyl-butyl}-benzenesulfonamide 300694 4-[5-(4-Amino-cyclohexylamino)-3-bromo-pyrazolo[1,5-a]pyrimidin-7-ylamino]-2-chloro-N,N-dimethyl-benzenesulfonamide 300700 4-[5-(4-Ethylamino-cyclohexylamino)-3-isopropyl-pyrazolo[1,5-a]pyrimidin-7-ylamino]-N,N-dimethyl-benzenesulfonamide 300701 N-Methyl-N-{(S)-4-[4-((R)-4-methyl-2-(R)-oxo-5-phenyl-oxazolidin-3-yl)-piperidin-1-yl]-2-phenyl-butyl}-benzenesulfonamide 300702 5-[(S)-4-(Benzenesulfonyl-methyl-amino)-3-phenyl-butyl]-octahydro-pyrrolo[3,2-c]pyridine-1-carboxylic acid tert-butyl ester 300707 3-{[5-(4-Chloro-phenyl)-5-oxo-pentanoyl]-methyl-amino}-pyrrolidine-1-carboxylic acid methyl-[1-(3-phenyl-propyl)-pyrrolidin-3-yl]-amide 300719 3-Imidazo[1,2-a]pyridin-3-yl-4-(2-isobutyryl-1,2,3,4-tetrahydro-[1,4]diazepino[6,7,1-hi]indol-7-yl)-pyrrole-2,5-dione 300731 3-Imidazo[1,2-a]pyrazin-3-yl-4-[2-(morpholine-4-carbonyl)-1,2,3,4-tetrahydro-[1,4]diazepino[6,7,1-hi]indol-7-yl]-pyrrole-2,5-dione 300733 3-[Methyl-(4''-trifluoromethyl-biphenyl-4-carbonyl)-amino]-pyrrolidine-1-carboxylic acid (1-butyl-pyrrolidin-3-yl)-methyl-amide 300736 3-{[2-(4-tert-Butyl-phenoxy)-acetyl]-methyl-amino}-pyrrolidine-1-carboxylic acid {1-[3-(4-chloro-phenyl)-propyl]-pyrrolidin-3-yl}-methyl-amide 300737 3-{[4-(4-Fluoro-phenoxy)-benzoyl]-methyl-amino}-pyrrolidine-1-carboxylic acid {1-[3-(4-chloro-phenyl)-propyl]-pyrrolidin-3-yl}-methyl-amide 300739 3-Imidazo[1,2-a]pyridin-3-yl-4-[2-(tetrahydro-pyran-4-carbonyl)-1,2,3,4-tetrahydro-[1,4]diazepino[6,7,1-hi]indol-7-yl]-pyrrole-2,5-dione 300753 3-Imidazo[1,2-a]pyrimidin-3-yl-4-[2-(morpholine-4-carbonyl)-1,2,3,4-tetrahydro-[1,4]diazepino[6,7,1-hi]indol-7-yl]-pyrrole-2,5-dione 300754 6-Chloro-3-[4-(2-methoxy-phenyl)-piperazin-1-ylmethyl]-3,4-dihydro-2H-benzo[1,2,4]thiadiazine 1,1-dioxide 300755 3-[Methyl-(4''-trifluoromethyl-biphenyl-4-carbonyl)-amino]-pyrrolidine-1-carboxylic acid [1-(2-hydroxy-ethyl)-pyrrolidin-3-yl]-methyl-amide 300756 3-[Methyl-(4''-trifluoromethyl-biphenyl-4-carbonyl)-amino]-pyrrolidine-1-carboxylic acid {1-[3-(4-chloro-phenyl)-propyl]-pyrrolidin-3-yl}-methyl-amide 300757 3-[Methyl-(4''-trifluoromethyl-biphenyl-4-carbonyl)-amino]-pyrrolidine-1-carboxylic acid [1-(3-cyclopentyl-propyl)-pyrrolidin-3-yl]-methyl-amide 300759 N*5*-(4-Amino-cyclohexyl)-N*7*-(4-benzenesulfonyl-phenyl)-3-bromo-pyrazolo[1,5-a]pyrimidine-5,7-diamine 300760 3-(2-Isobutyryl-1,2,3,4-tetrahydro-[1,4]diazepino[6,7,1-hi]indol-7-yl)-4-(3aH-pyrazolo[1,5-a]pyridin-3-yl)-pyrrole-2,5-dione 300765 5-[(S)-4-(Benzenesulfonyl-methyl-amino)-3-methyl-3-phenyl-butyl]-octahydro-pyrrolo[3,2-c]pyridine-1-carboxylic acid benzyl ester 300774 3-[Methyl-(4''-trifluoromethyl-biphenyl-4-carbonyl)-amino]-pyrrolidine-1-carboxylic acid {1-[2-(4-chloro-phenoxy)-ethyl]-pyrrolidin-3-yl}-methyl-amide 300775 3-[Methyl-(4''-trifluoromethyl-biphenyl-4-carbonyl)-amino]-pyrrolidine-1-carboxylic acid {1-[2-(4-chloro-benzenesulfonyl)-ethyl]-pyrrolidin-3-yl}-methyl-amide 300776 3-[Methyl-(4''-trifluoromethyl-biphenyl-4-carbonyl)-amino]-pyrrolidine-1-carboxylic acid methyl-{1-[2-(pyrrolidine-1-sulfonyl)-ethyl]-pyrrolidin-3-yl}-amide 300777 3-[Methyl-(4''-trifluoromethyl-biphenyl-4-carbonyl)-amino]-pyrrolidine-1-carboxylic acid [1-(4,4-dimethyl-cyclohexyl)-pyrrolidin-3-yl]-methyl-amide 300778 4-[5-(4-Amino-cyclohexylamino)-3-isopropyl-pyrazolo[1,5-a]pyrimidin-7-ylamino]-N,N-dimethyl-benzenesulfonamide 300785 5-[(R)-4-(Benzenesulfonyl-methyl-amino)-3-methyl-3-phenyl-butyl]-octahydro-pyrrolo[3,2-c]pyridine-1-carboxylic acid 4-nitro-benzyl ester 300788 7-(4-(H-imidazo[1,2-a]pyridin-3-yl)-2,5-dioxo-2,5-dihydro-1H-pyrrol-3-yl)-N,N-dimethyl-3,4-dihydro-[1,4]diazepino[6,7,1-hi]indole-2(1H)-carboxamide 300793 4-(5-(trans-4-aminocyclohexylamino)-3-cyclopentylpyrazolo[1,5-a]pyrimidin-7-ylamino)-N,N-dimethylbenzenesulfonamide 300799 3-Imidazo[1,2-a]pyridin-3-yl-4-[2-(piperidine-1-carbonyl)-1,2,3,4-tetrahydro-[1,4]diazepino[6,7,1-hi]indol-7-yl]-pyrrole-2,5-dione 300802 3-[Methyl-(4''-trifluoromethyl-biphenyl-4-carbonyl)-amino]-pyrrolidine-1-carboxylic acid methyl-[1-(tetrahydro-pyran-4-yl)-pyrrolidin-3-yl]-amide 300803 N-Methyl-N-[(S)-2-methyl-2-phenyl-4-(1-phenylacetyl-octahydro-pyrrolo[3,2-c]pyridin-5-yl)-butyl]-benzenesulfonamide 300805 7-(2,5-Dioxo-4-pyrrolo[1,2-b]pyridazin-5-yl-2,5-dihydro-1H-pyrrol-3-yl)-3,4-dihydro-1H-[1,4]diazepino[6,7,1-hi]indole-2-carboxylic acid dimethylamide 300815 3-(imidazo[1,2-b]pyridazin-3-yl)-4-(2-(piperidine-1-carbonyl)-1,2,3,4,7,7a-hexahydro-[1,4]diazepino[6,7,1-hi]indol-7-yl)-1H-pyrrole-2,5-dione 300825 3-(imidazo[1,2-a]pyridin-3-yl)-4-(2-(morpholine-4-carbonyl)-1,2,3,4-tetrahydro-[1,4]diazepino[6,7,1-hi]indol-7-yl)-1H-pyrrole-2,5-dione 300828 3-Imidazo[1,2-a]pyrazin-3-yl-4-[2-(piperidine-1-carbonyl)-1,2,3,4-tetrahydro-[1,4]diazepino[6,7,1-hi]indol-7-yl]-pyrrole-2,5-dione 300829 3-[Methyl-(4''-trifluoromethyl-biphenyl-4-carbonyl)-amino]-pyrrolidine-1-carboxylic acid methyl-[1-(1-methyl-piperidin-4-yl)-pyrrolidin-3-yl]-amide 300832 4-[5-(4-Amino-cyclohexylamino)-3-cyano-pyrazolo[1,5-a]pyrimidin-7-ylamino]-N,N-dimethyl-benzenesulfonamide 300846 3-(2-Acetyl-1,2,3,4-tetrahydro-[1,4]diazepino[6,7,1-hi]indol-7-yl)-4-imidazo[1,2-a]pyridin-3-yl-pyrrole-2,5-dione 300850 3-Imidazo[1,2-a]pyrimidin-3-yl-4-[2-(piperidine-1-carbonyl)-1,2,3,4-tetrahydro-[1,4]diazepino[6,7,1-hi]indol-7-yl]-pyrrole-2,5-dione 300854 3-[1-Oxo-5-(4-trifluoromethyl-phenyl)-1,3-dihydro-isoindol-2-yl]-pyrrolidine-1-carboxylic acid methyl-[1-(3-phenyl-propyl)-pyrrolidin-3-yl]-amide 300863 N*4*-(3-Bromo-phenyl)-N*6*-(2-chloro-ethyl)-quinazoline-4,6-diamine 300868 N*6*-(2-Chloro-ethyl)-N*4*-(3-chloro-phenyl)-quinazoline-4,6-diamine 300886 N-(6-((dimethylamino)methyl)-5,6,7,8-tetrahydronaphthalen-2-yl)-4'-fluorobiphenyl-4-carboxamide 300891 Biphenyl-4-carboxylic acid methyl-{3-[methyl-(1-methyl-pyrrolidin-3-yl)-carbamoyl]-propyl}-amide 300900 3-(3-Biphenyl-4-yl-1-methyl-ureido)-pyrrolidine-1-carboxylic acid {1-[3-(4-chloro-phenyl)-propyl]-pyrrolidin-3-yl}-methyl-amide 300918 3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-6-methyl-2H-benzo[1,2,4]thiadiazine 1,1-dioxide 300919 3-[Methyl-(4''-trifluoromethyl-biphenyl-4-carbonyl)-amino]-pyrrolidine-1-carboxylic acid methyl-(1-methyl-pyrrolidin-3-yl)-amide 300935 3-{[4-(6-Methoxy-pyridazin-3-yl)-benzoyl]-methyl-amino}-pyrrolidine-1-carboxylic acid [1-(4,4-dimethyl-cyclohexyl)-pyrrolidin-3-yl]-methyl-amide 300937 6-Chloro-3-[4-(2-methoxy-phenyl)-piperazin-1-ylmethyl]-2H-benzo[1,2,4]thiadiazine 1,1-dioxide 300938 3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-3,4-dihydro-2H-benzo[1,2,4]thiadiazine 1,1-dioxide 300943 3-[Methyl-(4''-trifluoromethyl-biphenyl-4-carbonyl)-amino]-pyrrolidine-1-carboxylic acid methyl-pyrrolidin-3-yl-amide 300953 2-(4-Trifluoromethyl-phenyl)-3H-imidazole-4-carboxylic acid (1-{[1-(4,4-dimethyl-cyclohexyl)-pyrrolidin-3-yl]-methyl-carbamoyl}-pyrrolidin-3-yl)-methyl-amide 300970 2-(4-Trifluoromethyl-phenyl)-thiazole-5-carboxylic acid (1-{[1-(4,4-dimethyl-cyclohexyl)-pyrrolidin-3-yl]-methyl-carbamoyl}-pyrrolidin-3-yl)-methyl-amide 301004 6-(2-Amino-2-phenyl-ethyl)-3,8-bis-(2-fluoro-phenyl)-2,3-dihydro-oxazolo[3,2-c]pyrimidine-5,7-dione 301013 2-((R)-2-Amino-2-phenyl-ethyl)-4-(2-fluoro-3-methoxy-phenyl)-7-phenyl-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidine-1,3-dione 301052 1-(2-Fluoro-phenyl)-3-[1-(1-methyl-1H-benzoimidazol-2-ylmethyl)-4-(4-pyridin-3-yl-phenyl)-piperidin-4-ylmethyl]-urea 301077 1-[1-Benzenesulfonyl-4-(4-pyridin-3-yl-phenyl)-piperidin-4-ylmethyl]-3-(2-fluoro-phenyl)-urea 301140 6-(2-Amino-2-phenyl-ethyl)-8-(2-fluoro-phenyl)-3-phenyl-2,3-dihydro-oxazolo[3,2-c]pyrimidine-5,7-dione 301153 6-(2-Amino-2-phenyl-ethyl)-8-(2-fluoro-3-methoxy-phenyl)-3-(2-fluoro-phenyl)-2,3-dihydro-thiazolo[3,2-c]pyrimidine-5,7-dione 301186 6-(2-Amino-2-phenyl-ethyl)-8-(2-chloro-phenyl)-3-(2-fluoro-phenyl)-2,3-dihydro-thiazolo[3,2-c]pyrimidine-5,7-dione 301190 6-(2-Amino-2-phenyl-ethyl)-8-(3-methoxy-phenyl)-3-phenyl-2,3-dihydro-oxazolo[3,2-c]pyrimidine-5,7-dione 301208 6-(2-Amino-2-phenyl-ethyl)-8-(2-fluoro-3-methoxy-phenyl)-3-phenyl-2,3-dihydro-oxazolo[3,2-c]pyrimidine-5,7-dione 301209 6-(2-Amino-2-phenyl-ethyl)-8-(2-chloro-3-methoxy-phenyl)-3-(2-fluoro-phenyl)-2,3-dihydro-thiazolo[3,2-c]pyrimidine-5,7-dione 301228 6-((R)-2-amino-2-phenylethyl)-8-(2-fluorophenyl)-3-phenyl-2,3-dihydro-6H-thiazolo[3,2-f]pyrimidine-5,7-dione 301251 6-(2-Amino-2-phenyl-ethyl)-3,8-bis-(2-fluoro-phenyl)-2,3-dihydro-thiazolo[3,2-c]pyrimidine-5,7-dione 301264 1-[4-(2,3-Dichloro-benzyl)-[1,4'']bipiperidinyl-1''-yl]-2-o-tolyl-ethanone 301270 [4-(3,4-Dichloro-benzyl)-[1,4'']bipiperidinyl-1''-yl]-(1H-indol-5-yl)-methanone 301271 [(3S,4S)-4-(3,4-Dichloro-benzyl)-3-methoxymethyl-[1,4'']bipiperidinyl-1''-yl]-quinolin-6-yl-methanone 301273 [4-(3,4-Dichloro-benzyl)-[1,4'']bipiperidinyl-1''-yl]-quinolin-8-yl-methanone 301274 N-[(3S,4S)-4-(3,4-Dichloro-benzyl)-1''-(quinoline-6-carbonyl)-[1,4'']bipiperidinyl-3-yl]-methanesulfonamide 301280 1-[4-(2,4-Dichloro-benzyl)-[1,4'']bipiperidinyl-1''-yl]-2-o-tolyl-ethanone 301281 1-[4-(4-Bromo-benzyl)-[1,4'']bipiperidinyl-1''-yl]-2-(2-tert-butyl-phenyl)-ethanone 301282 4-(3,4-Dichloro-benzyl)-[1,4'']bipiperidinyl-1''-carboxylic acid o-tolylamide 301286 [(3S,4S)-4-(3,4-Dichloro-benzyl)-3-methyl-[1,4'']bipiperidinyl-1''-yl]-quinolin-6-yl-methanone 301289 1-[4-(3,5-Difluoro-benzyl)-[1,4'']bipiperidinyl-1''-yl]-2-o-tolyl-ethanone 301291 4-(3-Hydroxy-phenylamino)-5-methyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid methyl ester 301295 1-[4-(4-Chloro-benzyl)-[1,4'']bipiperidinyl-1''-yl]-2-o-tolyl-ethanone 301303 1-[4-(2,5-Dichloro-benzyl)-[1,4'']bipiperidinyl-1''-yl]-2-o-tolyl-ethanone 301304 (3-Amino-phenyl)-[4-(3,4-dichloro-benzyl)-[1,4'']bipiperidinyl-1''-yl]-methanone 301307 4-[(3-Hydroxy-4-methyl-phenyl)-methyl-amino]-5-propyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid (3-pyrrolidin-1-yl-propyl)-amide 301315 [(3S,4S)-4-(3,4-Dichloro-benzyl)-3-ethyl-[1,4'']bipiperidinyl-1''-yl]-quinolin-6-yl-methanone 301323 (4-Amino-phenyl)-[4-(3,4-dichloro-benzyl)-[1,4'']bipiperidinyl-1''-yl]-methanone 301324 4-(3-Hydroxy-4-methyl-phenylamino)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid (3-pyrrolidin-1-yl-propyl)-amide 301329 1-[4-(4-Chloro-2-fluoro-benzyl)-[1,4'']bipiperidinyl-1''-yl]-2-o-tolyl-ethanone 301330 [(3S,4S)-4-(3,4-Dichloro-benzyl)-3-methoxy-[1,4'']bipiperidinyl-1''-yl]-quinolin-6-yl-methanone 301337 [(3S,4S)-4-(3,4-Dichloro-benzyl)-3-vinyl-[1,4'']bipiperidinyl-1''-yl]-quinolin-6-yl-methanone 301340 1-[4-(4-Fluoro-benzyl)-[1,4'']bipiperidinyl-1''-yl]-2-o-tolyl-ethanone 301342 xv4-(3-Hydroxy-4-methyl-phenylamino)-5-methyl-pyrrolo[2,1-f][1,2,4]tr4-(3-Hydroxy-4-methyl-phenylamino)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid (3-pyrrolidin-1-yl-propyl)-amideiazine-6-carboxylic acid (3-methox4-(3-Hydroxy-4-methyl-phenylamino)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid (3-pyrrolidin-1-yl-propyl)-amidey-propyl)-amide4-(3-Hydroxy-4-methyl-phenylamino)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid (3-pyrrolidin-1-yl-propyl)-amide 301343 [4-(3,4-Dichloro-benzyl)-[1,4'']bipiperidinyl-1''-yl]-isoquinolin-1-yl-methanone 301344 N-[(3S,4S)-4-(3,4-Dichloro-benzyl)-1''-(quinoline-6-carbonyl)-[1,4'']bipiperidinyl-3-yl]-acetamide 301348 Cinnolin-4-yl-[4-(3,4-dichloro-benzyl)-[1,4'']bipiperidinyl-1''-yl]-methanone 301352 1-[4-(3,5-Dichloro-benzyl)-[1,4'']bipiperidinyl-1''-yl]-2-o-tolyl-ethanone 301354 1-[4-(4-Chloro-3-fluoro-benzyl)-[1,4'']bipiperidinyl-1''-yl]-2-o-tolyl-ethanone 301356 1-[4-(4-Methoxy-benzyl)-[1,4'']bipiperidinyl-1''-yl]-2-o-tolyl-ethanone 301359 [4-(3,4-Dichloro-benzyl)-[1,4'']bipiperidinyl-1''-yl]-quinolin-3-yl-methanone 301360 [(3S,4S)-4-(3,4-Dichloro-benzyl)-3-hydroxymethyl-[1,4'']bipiperidinyl-1''-yl]-quinolin-6-yl-methanone 301361 [(3S,4S)-4-(3,4-Dichloro-benzyl)-3-fluoromethyl-[1,4'']bipiperidinyl-1''-yl]-quinolin-6-yl-methanone 301362 [4-(3,4-Dichloro-benzyl)-[1,4'']bipiperidinyl-1''-yl]-quinolin-6-yl-methanone 301363 [(3S,4S)-4-(3,4-Dichloro-benzyl)-3-ethoxy-[1,4'']bipiperidinyl-1''-yl]-quinolin-6-yl-methanone 301364 4-(3-Hydroxy-4-methyl-phenylamino)-5-methyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid (3-[1,2,3]triazol-2-yl-propyl)-amide 301370 1-[4-(3,4-Dichloro-benzyl)-[1,4'']bipiperidinyl-1''-yl]-2-o-tolyl-ethanone 301376 1-[4-(3-Chloro-benzyl)-[1,4'']bipiperidinyl-1''-yl]-2-o-tolyl-ethanone 301379 [4-(3,4-Dichloro-benzyl)-[1,4'']bipiperidinyl-1''-yl]-(1H-indol-4-yl)-methanone 301381 1-[4-(3-Chloro-5-fluoro-benzyl)-[1,4'']bipiperidinyl-1''-yl]-2-o-tolyl-ethanone 301382 [4-(3,4-Dichloro-benzyl)-[1,4'']bipiperidinyl-1''-yl]-quinolin-4-yl-methanone 301383 [4-(3-Hydroxy-4-methyl-phenylamino)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazin-6-yl]-carbamic acid 3-[1,2,3]triazol-2-yl-propyl ester 301393 [(3S,4S)-4-(3,4-Dichloro-benzyl)-3-methoxy-[1,4'']bipiperidinyl-1''-yl]-quinoxalin-6-yl-methanone 301396 1-Ethyl-3-{(1R,2R)-2-[(R)-2-(4-phenyl-butyl)-2,3-dihydro-benzofuran-4-yl]-cyclopropylmethyl}-urea 301397 1-{(1R,2R)-2-[(R)-5-Chloro-2-(4-phenyl-butyl)-2,3-dihydro-benzofuran-4-yl]-cyclopropylmethyl}-3-ethyl-urea 301399 N-[(3R,4S)-4-(3,4-Dichloro-benzyl)-1''-(quinoline-6-carbonyl)-[1,4'']bipiperidinyl-3-ylmethyl]-acetamide 301402 4-(3-Hydroxy-4-methyl-phenylamino)-5-propyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid ethyl ester 301404 [(3S,4S)-4-(3,4-Dichloro-benzyl)-3-methoxy-[1,4'']bipiperidinyl-1''-yl]-[1,8]naphthyridin-2-yl-methanone 301415 [(3S,4S)-4-(3,4-Dichloro-benzyl)-3-methoxy-[1,4'']bipiperidinyl-1''-yl]-quinoxalin-2-yl-methanone 301419 N-{3-[(R)-2-(4-Phenyl-butyl)-2,3-dihydro-benzofuran-4-yl]-propyl}-acetamide 301422 Cinnolin-4-yl-[(3S,4S)-4-(3,4-dichloro-benzyl)-3-methoxy-[1,4'']bipiperidinyl-1''-yl]-methanone 301425 5-Ethoxy-4-(3-hydroxy-4-methyl-phenylamino)-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid ethyl ester 301439 4-(3-Hydroxy-4-methyl-phenylamino)-5-methyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid methyl ester 301440 4-(4-Ethyl-3-hydroxy-phenylamino)-5-methyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid methyl ester 301443 N-{3-[(R)-2-(4-Phenyl-butyl)-2,3-dihydro-benzofuran-4-yl]-propyl}-propionamide 301444 N-{3-[(R)-2-(4-Phenyl-butyl)-2,3-dihydro-benzofuran-4-yl]-propyl}-butyramide 301449 4-(3-Hydroxy-4-methyl-phenylamino)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid ethyl ester 301455 4-(3-Hydroxy-4-propyl-phenylamino)-5-methyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid methyl ester 301460 [(3S,4S)-4-(3,4-Dichloro-benzyl)-3-methoxy-[1,4'']bipiperidinyl-1''-yl]-quinolin-4-yl-methanone 301462 4-(3-Hydroxy-4-isopropyl-phenylamino)-5-methyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid methyl ester 301465 5-tert-Butyl-4-[(3-hydroxy-4-methyl-phenyl)-methyl-amino]-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid methyl ester 301466 N-{3-[(R)-2-(4-Phenyl-butyl)-2,3-dihydro-benzofuran-4-yl]-propyl}-isobutyramide 301474 Cyclopropanecarboxylic acid {3-[(R)-2-(4-phenyl-butyl)-2,3-dihydro-benzofuran-4-yl]-propyl}-amide 301477 [(3S,4S)-4-(3,4-Dichloro-benzyl)-3-methoxy-[1,4'']bipiperidinyl-1''-yl]-quinolin-8-yl-methanone 301480 4-(3-Hydroxy-4-trifluoromethyl-phenylamino)-5-methyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid methyl ester 301487 4-(4-Bromo-3-hydroxy-phenylamino)-5-methyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid methyl ester 301488 4-[(3-Hydroxy-4-methyl-phenyl)-methyl-amino]-5-methyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid (3-pyrrolidin-1-yl-propyl)-amide 301492 1-Ethyl-3-{3-[(R)-2-(4-phenyl-butyl)-2,3-dihydro-benzofuran-4-yl]-propyl}-urea 301497 N-{(1R,2R)-2-[(R)-2-(4-Phenyl-butyl)-2,3-dihydro-benzofuran-4-yl]-cyclopropylmethyl}-isobutyramide 301498 Cyclopropanecarboxylic acid {(1R,2R)-2-[(R)-2-(4-phenyl-butyl)-2,3-dihydro-benzofuran-4-yl]-cyclopropylmethyl}-amide 301499 N-[(3S,4S)-4-(3,4-Dichloro-benzyl)-1''-(quinoline-6-carbonyl)-[1,4'']bipiperidinyl-3-ylmethyl]-methanesulfonamide 301501 [(3S,4S)-4-(3,4-Dichloro-benzyl)-3-methoxy-[1,4'']bipiperidinyl-1''-yl]-isoquinolin-1-yl-methanone 301524 (R,S)2-Formylamino-N-methyl-2-phenyl-N-(1-phenyl-2-pyrrolidin-1-yl-ethyl)-acetamide 301553 [(3S,4S)-4-(3,4-Dichloro-benzyl)-3-methoxy-[1,4'']bipiperidinyl-1''-yl]-[1,6]naphthyridin-2-yl-methanone 301566 N-{(1R,2R)-2-[(R)-2-(4-Phenyl-butyl)-2,3-dihydro-benzofuran-4-yl]-cyclopropylmethyl}-acetamide 301581 N-{(1R,2R)-2-[(R)-2-(4-Phenyl-butyl)-2,3-dihydro-benzofuran-4-yl]-cyclopropylmethyl}-propionamide 301585 N-{(1R,2R)-2-[(R)-2-(4-Phenyl-butyl)-2,3-dihydro-benzofuran-4-yl]-cyclopropylmethyl}-butyramide 301615 3,4-Dichloro-N-({[(S)-2-((R)-3-hydroxy-pyrrolidin-1-yl)-1-phenyl-ethyl]-methyl-carbamoyl}-methyl)-benzamide 301620 (S)N-{[Methyl-(1-phenyl-2-pyrrolidin-1-yl-ethyl)-carbamoyl]-phenyl-methyl}-benzamide 301625 (1-methyl-4,5-diphenyl-1H-imidazol-2-yl)(piperidin-1-yl)methanone 301629 3,4-Dichloro-N-({[(S)-2-((R)-3-hydroxy-pyrrolidin-1-yl)-1-phenyl-ethyl]-methyl-carbamoyl}-methyl)-N-methyl-benzamide 301630 N-cyclohexyl-1-methyl-4,5-diphenyl-1H-imidazole-2-carboxamide 301646 1-methyl-N-(piperidin-1-yl)-4,5-dip-tolyl-1H-imidazole-2-carboxamide 301651 N-({[(S)-2-((R)-3-Hydroxy-pyrrolidin-1-yl)-1-phenyl-ethyl]-methyl-carbamoyl}-methyl)-2-methoxy-benzamide 301652 N-({[(S)-2-((R)-3-Hydroxy-pyrrolidin-1-yl)-1-phenyl-ethyl]-methyl-carbamoyl}-methyl)-4-methoxy-benzamide 301655 (RorS){[Methyl-(1-phenyl-2-pyrrolidin-1-yl-ethyl)-carbamoyl]-phenyl-methyl}-carbamic acid benzyl ester 301667 {[Methyl-(1-phenyl-2-pyrrolidin-1-yl-ethyl)-carbamoyl]-methyl}-carbamic acid benzyl ester 301673 N-{[Methyl-((S)-1-phenyl-2-pyrrolidin-1-yl-ethyl)-carbamoyl]-methyl}-2-phenyl-acetamide 301676 [4-(3-Hydroxy-4-methyl-phenylamino)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazin-6-yl]-carbamic acid 3-piperidin-1-yl-propyl ester 301678 (RorS){[Methyl-(1-phenyl-2-pyrrolidin-1-yl-ethyl)-carbamoyl]-phenyl-methyl}-carbamic acid benzyl ester 301690 N-{[Methyl-((S)-1-phenyl-2-pyrrolidin-1-yl-ethyl)-carbamoyl]-methyl}-benzamide 301693 5-[5-Isopropyl-6-(3-piperidin-1-yl-propoxy)-pyrrolo[2,1-f][1,2,4]triazin-4-ylamino]-2-methyl-phenol 301696 3,4-Dichloro-N-{[methyl-((S)-1-phenyl-2-pyrrolidin-1-yl-ethyl)-carbamoyl]-methyl}-benzamide 301702 (S){1-[Methyl-(1-phenyl-2-pyrrolidin-1-yl-ethyl)-carbamoyl]-2-phenyl-ethyl}-carbamic acid benzyl ester 301708 4-(3-Hydroxy-4-methyl-phenylamino)-5-methyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid (3-morpholin-4-yl-propyl)-amide 301713 1-Oxy-benzo[1,2,5]oxadiazole-5-carboxylic acid {[methyl-((S)-1-phenyl-2-pyrrolidin-1-yl-ethyl)-carbamoyl]-methyl}-amide 301722 1-methyl-4,5-diphenyl-N-(piperidin-1-yl)-1H-imidazole-2-carboxamide 301724 1-[4-(3-Hydroxy-4-methyl-phenylamino)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazin-6-yl]-3-(3-piperidin-1-yl-propyl)-urea 301725 (S){[Methyl-(1-phenyl-2-pyrrolidin-1-yl-ethyl)-carbamoyl]-phenyl-methyl}-carbamic acid methyl ester 301735 5-(4-Chloro-phenyl)-4-(2,4-dichloro-phenyl)-1-methyl-1H-imidazole-2-carboxylic acid cyclohexyl-methyl-amide 301737 4,5-bis(4-chlorophenyl)-N-(piperidin-1-yl)-1H-imidazole-2-carboxamide 301749 5-(4-Chloro-phenyl)-4-(2,4-dichloro-phenyl)-1-methyl-1H-imidazole-2-carboxylic acid piperidin-1-ylamide 301750 4,5-Bis-(4-chloro-phenyl)-oxazole-2-carboxylic acid cyclohexylamide 301751 4,5-Bis-(4-chloro-phenyl)-1-methyl-1H-imidazole-2-carboxylic acid piperidin-1-ylamide 301752 5-(4-Chloro-phenyl)-4-(2,4-dichloro-phenyl)-1-methyl-1H-imidazole-2-carboxylic acid phenylamide 301754 4,5-Bis-(4-chloro-phenyl)-1H-imidazole-2-carboxylic acid cyclohexylamide 301758 1-(4,5-Diphenyl-1H-imidazol-2-ylsulfanyl)-1-phenyl-propan-2-one 301760 4,5-bis(4-chlorophenyl)-N-(piperidin-1-yl)oxazole-2-carboxamide 301764 5-(4-Chloro-phenyl)-4-(2,4-dichloro-phenyl)-1-methyl-1H-imidazole-2-carboxylic acid cyclohexylamide 301765 4,5-Bis-(4-chloro-phenyl)-1-methyl-1H-imidazole-2-carboxylic acid cyclohexylamide 301766 5-(4-Chloro-phenyl)-4-(2,4-dichloro-phenyl)-1-ethyl-1H-imidazole-2-carboxylic acid cyclohexylamide 301771 5-(4-Chloro-phenyl)-4-(2,4-dichloro-phenyl)-oxazole-2-carboxylic acid piperidin-1-ylamide 301783 xvx4,5-Bis-(4-chloro-phenyl)-1-methyl-1H-imidazole-2-carboxylic acid morpholin-4-ylamide[4,5-Bis-(4-chloro-phenyl)-1-methyl-1H-imidazol-24,5-Bis-(4-chloro-phenyl)-1-methyl-1H-imidazole-2-carboxylic acid morpholin-4-ylamide-yl]-piperidin-1-yl-methanone 301788 5-(4-Chloro-phenyl)-4-(2,4-dichloro-phenyl)-oxazole-2-carboxylic acid cyclohexylamide 301790 4-(4-Chloro-phenyl)-5-(2,4-dichloro-phenyl)-1-methyl-1H-imidazole-2-carboxylic acid piperidin-1-ylamide 301804 4-(4-Chloro-phenyl)-5-(2,4-dichloro-phenyl)-oxazole-2-carboxylic acid piperidin-1-ylamide 301806 4,5-Bis-(4-chloro-phenyl)-1-methyl-1H-imidazole-2-carboxylic acid morpholin-4-ylamide 301807 4-(4-Chloro-phenyl)-5-(2,4-dichloro-phenyl)-1-methyl-1H-imidazole-2-carboxylic acid cyclohexylamide 301813 5-(4-chlorophenyl)-4-(2,4-dichlorophenyl)-1-methyl-N-morpholino-1H-imidazole-2-carboxamide 301821 4-(4-Chloro-phenyl)-5-(2,4-dichloro-phenyl)-oxazole-2-carboxylic acid cyclohexylamide 301824 4,5-Bis-(4-chloro-phenyl)-1-methyl-1H-imidazole-2-carboxylic acid hexylamide 301829 1-Methyl-4,5-di-p-tolyl-1H-imidazole-2-carboxylic acid cyclohexylamide 301830 5-(4-Chloro-phenyl)-4-(2,4-dichloro-phenyl)-1-methyl-1H-imidazole-2-carboxylic acid cyclopentylamide 301831 4,5-Bis-(2,4-dichloro-phenyl)-1-methyl-1H-imidazole-2-carboxylic acid piperidin-1-ylamide 301839 4,5-Bis-(2,4-dichloro-phenyl)-oxazole-2-carboxylic acid cyclohexylamide 301847 (1-methyl-4,5-dip-tolyl-1H-imidazol-2-yl)(piperidin-1-yl)methanone 301848 5-(4-Chloro-phenyl)-4-(2,4-dichloro-phenyl)-1-methyl-1H-imidazole-2-carboxylic acid cycloheptylamide 301849 4,5-Bis-(4-chloro-phenyl)-1-methyl-1H-imidazole-2-carboxylic acid tert-butylamide 301850 4,5-Bis-(2,4-dichloro-phenyl)-1-methyl-1H-imidazole-2-carboxylic acid cyclohexylamide 301855 4,5-Bis-(2,4-dichloro-phenyl)-oxazole-2-carboxylic acid piperidin-1-ylamide 301863 3-[5-(2-Fluoro-benzoyl)-thiazol-2-ylamino]-benzonitrile 301876 3-[5-(2-Trifluoromethyl-benzoyl)-thiazol-2-ylamino]-benzonitrile 301879 3-[5-(4-Methoxy-benzoyl)-thiazol-2-ylamino]-benzonitrile 301880 3-[5-(2,5-Dimethyl-thiophene-3-carbonyl)-thiazol-2-ylamino]-benzonitrile 301893 o-Tolyl-[2-(3-trifluoromethyl-phenylamino)-thiazol-5-yl]-methanone 301964 (2-Fluoro-phenyl)-[2-(3-methoxy-phenylamino)-thiazol-5-yl]-methanone 301965 [2-(4-Chloro-phenylamino)-thiazol-5-yl]-(2-fluoro-phenyl)-methanone 301977 3-[5-(2-Methyl-benzoyl)-thiazol-2-ylamino]-benzonitrile 301981 (3-Fluoro-phenyl)-[2-(3-trifluoromethyl-phenylamino)-thiazol-5-yl]-methanone 301983 3-[5-(2-Ethyl-benzoyl)-thiazol-2-ylamino]-benzonitrile 302003 2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid {1-[3-(morpholine-4-sulfonyl)-propyl]-piperidin-4-ylmethyl}-amide 302024 (2-Ethyl-phenyl)-[2-(3-trifluoromethyl-phenylamino)-thiazol-5-yl]-methanone 302042 (2-Trifluoromethyl-phenyl)-[2-(3-trifluoromethyl-phenylamino)-thiazol-5-yl]-methanone 302048 (2,5-Dimethyl-thiophen-3-yl)-[2-(3-trifluoromethyl-phenylamino)-thiazol-5-yl]-methanone 302057 2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid {1-[3-(4,4-dimethyl-piperidine-1-sulfonyl)-propyl]-piperidin-4-ylmethyl}-amide 302080 2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid {1-[3-(4-propyl-piperidine-1-sulfonyl)-propyl]-piperidin-4-ylmethyl}-amide 302086 2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid {1-[3-(piperidine-1-sulfonyl)-propyl]-piperidin-4-ylmethyl}-amide 302099 2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid {1-[3-(8-aza-spiro[4.5]decane-8-sulfonyl)-propyl]-piperidin-4-ylmethyl}-amide 302116 2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid (1-{3-[4-(propane-2-sulfonyl)-piperazine-1-sulfonyl]-propyl}-piperidin-4-ylmethyl)-amide 302117 2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid (1-{3-[4-(4-fluoro-benzenesulfonyl)-piperazine-1-sulfonyl]-propyl}-piperidin-4-ylmethyl)-amide 302118 Naphthalene-2-carboxylic acid [4-(10-methoxy-1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-butyl]-amide 302119 2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid {1-[3-(4-cyclopentyl-piperazine-1-sulfonyl)-propyl]-piperidin-4-ylmethyl}-amide 302120 Biphenyl-4-carboxylic acid [4-(1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-butyl]-amide 302121 3-[6-(4-Chloro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid 302122 2-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-benzoic acid 302127 2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid {1-[3-(piperazine-1-sulfonyl)-propyl]-piperidin-4-ylmethyl}-amide 302132 2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid (1-{3-[4-(pyrrolidine-1-sulfonyl)-piperazine-1-sulfonyl]-propyl}-piperidin-4-ylmethyl)-amide 302133 2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid (1-{3-[4-(4-fluoro-phenyl)-piperazine-1-sulfonyl]-propyl}-piperidin-4-ylmethyl)-amide 302134 Naphthalene-2-carboxylic acid [2-(1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-ethyl]-amide 302136 3-[6-(Biphenyl-4-sulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid 302139 2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid {1-[3-(4-methyl-piperazine-1-sulfonyl)-propyl]-piperidin-4-ylmethyl}-amide 302142 3-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-benzoic acid 302144 1-(4-Fluoro-phenyl)-2-(1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-ethanone 302145 2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid {1-[3-(4-pyridin-2-yl-piperazine-1-sulfonyl)-propyl]-piperidin-4-ylmethyl}-amide 302146 Naphthalene-2-carboxylic acid [3-(1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-propyl]-amide 302158 2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid {1-[3-(4-ethyl-piperazine-1-sulfonyl)-propyl]-piperidin-4-ylmethyl}-amide 302161 N-(4-(1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl)-2-naphthamide 302170 2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid (1-{3-[4-(furan-2-carbonyl)-piperazine-1-sulfonyl]-propyl}-piperidin-4-ylmethyl)-amide 302171 Naphthalene-2-carboxylic acid [4-(7-methoxy-1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-butyl]-amide 302173 2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid {1-[3-(4-propyl-piperazine-1-sulfonyl)-propyl]-piperidin-4-ylmethyl}-amide 302175 2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid {1-[3-(4-acetyl-piperazine-1-sulfonyl)-propyl]-piperidin-4-ylmethyl}-amide 302176 2,4-Diamino-10-methyl-5,10-dihydro-benzo[b][1,8]naphthyridine-3-carbonitrile 302180 1-(4-Fluoro-phenyl)-5-(1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-pentan-1-one 302182 [6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-acetic acid 302184 2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid {1-[3-(4-pyridin-3-ylmethyl-piperazine-1-sulfonyl)-propyl]-piperidin-4-ylmethyl}-amide 302193 2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid {1-[3-(4-isopropyl-piperazine-1-sulfonyl)-propyl]-piperidin-4-ylmethyl}-amide 302194 Biphenyl-4-carboxylic acid [2-(1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-ethyl]-amide 302195 3-[6-(4-Phenoxy-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid 302196 2-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid 302198 2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid {1-[3-(4-methanesulfonyl-piperazine-1-sulfonyl)-propyl]-piperidin-4-ylmethyl}-amide 302199 Naphthalene-2-carboxylic acid [4-(8-methoxy-1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-butyl]-amide 302207 2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid {1-[3-(4-sec-butyl-piperazine-1-sulfonyl)-propyl]-piperidin-4-ylmethyl}-amide 302208 Biphenyl-4-carboxylic acid [3-(1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-propyl]-amide 302210 3-[6-(4-Methoxy-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid 302214 2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid (1-{3-[4-(propane-1-sulfonyl)-piperazine-1-sulfonyl]-propyl}-piperidin-4-ylmethyl)-amide 302215 Naphthalene-2-carboxylic acid [4-(9-methoxy-1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-butyl]-amide 302218 2-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-butyric acid 302225 3-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid 302227 3-[6-(4-Hydroxy-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid 302233 3-(6-Benzylamino-1,2,3,4-tetrahydro-carbazol-9-yl)-propionic acid 302234 [5-(4-Fluoro-benzenesulfonylamino)-2-propyl-indol-1-yl]-acetic acid 302235 4-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-butyric acid 302248 3-[6-(3-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid 302251 3-[6-(Naphthalene-2-sulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid 302256 2-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-ethanesulfonic acid 302258 5-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-pentanoic acid 302263 3-[6-(3-Chloro-4-fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid 302270 4-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-benzoic acid 302272 3-[6-(2-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid 302273 3-(6-Benzenesulfonylamino-1,2,3,4-tetrahydro-carbazol-9-yl)-propionic acid 302281 [2-(4-Fluoro-benzenesulfonylamino)-6,7,8,9,10,10a-hexahydro-5aH-cyclohepta[b]indol-5-yl]-acetic acid 302286 3-[6-(2,4-Difluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid 302287 [6-(4-Fluoro-benzenesulfonylamino)-3-methyl-1,2,3,4-tetrahydro-carbazol-9-yl]-acetic acid 302289 3-[6-(Toluene-4-sulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid 302296 (Z)-3-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-acrylic acid 302297 Ramatroban 302303 3-[6-(3,4-Difluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid 302305 3-[6-(Toluene-3-sulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid 302311 [6-(4-Fluoro-benzenesulfonylamino)-3-phenyl-1,2,3,4-tetrahydro-carbazol-9-yl]-acetic acid 302329 3-[6-(Thiophene-2-sulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid 302343 [3-tert-Butyl-6-(4-fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-acetic acid 302354 2-(benzyloxy)-6-(4-chlorophenyl)-5-phenylnicotinonitrile 302356 4-(5-Methoxy-2-methyl-phenylamino)-7-((E)-2-pyridin-4-yl-vinyl)-quinoline-3-carbonitrile 302362 4-Bromo-N-[4-(4-dimethylamino-quinazolin-2-ylamino)-cyclohexylmethyl]-2-trifluoromethoxy-benzenesulfonamide 302365 cis-4-Bromo-N-[4-(4-dimethylamino-quinazolin-2-ylamino)-cyclohexyl]-2-trifluoromethoxy-benzamide 302368 trans-4-Bromo-N-{4-[(4-dimethylamino-quinazolin-2-ylamino)-methyl]-cyclohexylmethyl}-N-methyl-2-trifluoromethoxy-benzenesulfonamide 302378 2-Benzyloxy-5-(4-chloro-phenyl)-6-(2,4-dichloro-phenyl)-nicotinonitrile 302380 4-(2,4-Dimethyl-phenylamino)-7-((E)-2-pyridin-4-yl-vinyl)-quinoline-3-carbonitrile 302384 6-(2,4-Dichloro-phenyl)-2-(3,4-difluoro-benzyloxy)-5-(4-fluoro-phenyl)-nicotinonitrile 302394 trans-4-Bromo-N-{4-[(4-dimethylamino-quinazolin-2-ylamino)-methyl]-cyclohexylmethyl}-2-trifluoromethoxy-benzamide 302405 6-(2,4-dichlorophenyl)-2-(3,4-difluorobenzyloxy)-5-p-tolylnicotinonitrile 302416 (S)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-[4-(2-methanesulfonylamino-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-amide 302419 2-(3,4-Difluoro-benzyloxy)-6-(2,4-difluoro-phenyl)-5-(4-fluoro-phenyl)-nicotinonitrile 302435 (S)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-oxo-2-[4-(2-phenylmethanesulfonylamino-phenyl)-piperazin-1-yl]-ethyl}-amide 302436 (S)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [(R)-2-[4-(2-benzenesulfonylamino-phenyl)-piperazin-1-yl]-1-(4-chloro-benzyl)-2-oxo-ethyl]-amide 302437 (S)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid ((R)-1-(4-chloro-benzyl)-2-{4-[2-(methanesulfonyl-methyl-amino)-phenyl]-piperazin-1-yl}-2-oxo-ethyl)-amide 302440 2-Benzyloxy-5-(4-chloro-phenyl)-6-(2,4-dichloro-phenyl)-nicotinamide 302452 (S)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid ((R)-1-(4-chloro-benzyl)-2-{4-[2-(cyclopropylmethyl-methanesulfonyl-amino)-phenyl]-piperazin-1-yl}-2-oxo-ethyl)-amide 302453 (S)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [(R)-2-(4-{2-[(2-amino-ethyl)-methanesulfonyl-amino]-phenyl}-piperazin-1-yl)-1-(4-chloro-benzyl)-2-oxo-ethyl]-amide 302454 (S)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid ((R)-1-(4-chloro-benzyl)-2-{4-[2-(methanesulfonyl-propyl-amino)-phenyl]-piperazin-1-yl}-2-oxo-ethyl)-amide 302455 Isoquinoline-3-carboxylic acid ((R)-1-(4-chloro-benzyl)-2-{4-[2-(cyclopropylmethyl-methanesulfonyl-amino)-phenyl]-piperazin-1-yl}-2-oxo-ethyl)-amide 302456 Naphthalene-2-carboxylic acid ((R)-1-(4-chloro-benzyl)-2-{4-[2-(cyclopropylmethyl-methanesulfonyl-amino)-phenyl]-piperazin-1-yl}-2-oxo-ethyl)-amide 302457 Quinoline-3-carboxylic acid ((R)-1-(4-chloro-benzyl)-2-{4-[2-(cyclopropylmethyl-methanesulfonyl-amino)-phenyl]-piperazin-1-yl}-2-oxo-ethyl)-amide 302458 cis-N*2*-{4-[(4-Bromo-2-trifluoromethoxy-benzylamino)-methyl]-cyclohexyl}-N*4*,N*4*-dimethyl-quinazoline-2,4-diamine 302459 4-(2-Chloro-5-methoxy-phenylamino)-7-((E)-2-pyridin-4-yl-vinyl)-quinoline-3-carbonitrile 302462 Quinoline-6-carboxylic acid ((R)-1-(4-chloro-benzyl)-2-{4-[2-(cyclopropylmethyl-methanesulfonyl-amino)-phenyl]-piperazin-1-yl}-2-oxo-ethyl)-amide 302480 4-(2,3-Dichloro-5-methoxy-phenylamino)-7-[(E)-2-(1H-imidazol-2-yl)-vinyl]-6-methoxy-quinoline-3-carbonitrile 302481 2-Benzyloxy-6-(4-dimethylamino-phenyl)-5-(4-methoxy-phenyl)-nicotinonitrile 302482 6-Methoxy-7-pyridin-3-ylethynyl-4-(3,4,5-trimethoxy-phenylamino)-quinoline-3-carbonitrile 302488 5-(4-Chloro-phenyl)-6-(2,4-dichloro-phenyl)-pyridine-2-carboxylic acid cyclopentylamide 302492 8-{4-[3-(4-Methoxy-phenyl)-[1,2,4]oxadiazol-5-ylmethoxy]-phenyl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 302494 (S)-2-{3-[4-(3-Chloro-benzyloxy)-phenyl]-ureido}-N-(3-morpholin-4-yl-propyl)-3-phenyl-propionamide 302495 4-(2,4-Dichloro-5-methoxy-phenylamino)-7-[(E)-2-(1-oxy-pyridin-4-yl)-vinyl]-quinoline-3-carbonitrile 302497 1-Benzyl-6-(4-chloro-phenyl)-2-oxo-5-phenyl-1,2-dihydro-pyridine-3-carbonitrile 302498 8-{4-[5-(3-Methoxy-phenyl)-[1,2,4]oxadiazol-3-ylmethoxy]-phenyl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 302502 5-(4-Chloro-phenyl)-6-(2,4-dichloro-phenyl)-pyridine-2-carboxylic acid cyclohexylamide 302504 4-(2,4-Dichloro-5-methoxy-phenylamino)-6-((E)-2-pyridin-4-yl-vinyl)-quinoline-3-carbonitrile 302505 (S)-2-{3-[4-(4-Methoxy-phenoxy)-phenyl]-ureido}-N-(3-morpholin-4-yl-propyl)-3-phenyl-propionamide 302506 5-(4-Chloro-phenyl)-6-(2,4-dichloro-phenyl)-2-(4-trifluoromethyl-benzyloxy)-nicotinonitrile 302510 4-(2,4-Dichloro-5-methoxy-phenylamino)-6-methoxy-7-[(E)-2-(1-oxy-pyridin-4-yl)-vinyl]-quinoline-3-carbonitrile 302514 trans-N*2*-(4-{[(4-Bromo-2-trifluoromethoxy-benzyl)-methyl-amino]-methyl}-cyclohexylmethyl)-N*4*,N*4*-dimethyl-quinazoline-2,4-diamine 302521 5-(4-Chloro-phenyl)-6-(2,4-dichloro-phenyl)-2-(4-fluoro-benzyloxy)-nicotinonitrile 302524 cis-4-Bromo-N-[4-(4-dimethylamino-quinazolin-2-ylamino)-cyclohexylmethyl]-2-trifluoromethoxy-benzamide 302525 5,6-Bis-(4-chloro-phenyl)-2-(3,4-difluoro-benzyloxy)-nicotinonitrile 302526 5-(4-Chloro-phenyl)-6-(2,4-dichloro-phenyl)-pyridine-2-carboxylic acid cycloheptylamide 302527 7-((E)-2-Pyridin-4-yl-vinyl)-4-(3,4,5-trimethoxy-phenylamino)-quinoline-3-carbonitrile 302528 1-Benzyl-5-(4-chloro-phenyl)-6-(2,4-dichloro-phenyl)-2-oxo-1,2-dihydro-pyridine-3-carbonitrile 302529 6-((E)-2-Pyridin-4-yl-vinyl)-4-(3,4,5-trimethoxy-phenylamino)-quinoline-3-carbonitrile 302538 7-[(E)-2-(1-Oxy-pyridin-4-yl)-vinyl]-4-(3,4,5-trimethoxy-phenylamino)-quinoline-3-carbonitrile 302544 5-(4-Chloro-phenyl)-6-(2,4-dichloro-phenyl)-2-(3,5-difluoro-benzyloxy)-nicotinonitrile 302550 5-(4-Chloro-phenyl)-6-(2,4-dichloro-phenyl)-pyridine-2-carboxylic acid piperidin-1-ylamide 302557 2-(3,4-difluorobenzyloxy)-6-(2-chlorophenyl)-5-(4-chlorophenyl)nicotinonitrile 302558 N*2*-[1-(4-Bromo-2-trifluoromethoxy-benzenesulfonyl)-piperidin-4-yl]-N*4*,N*4*-dimethyl-quinazoline-2,4-diamine 302559 7-Pyridin-3-ylethynyl-4-(3,4,5-trimethoxy-phenylamino)-quinoline-3-carbonitrile 302560 4-(2,3-Dichloro-5-methoxy-phenylamino)-6-pyridin-3-ylethynyl-quinoline-3-carbonitrile 302565 [5-(4-Chloro-phenyl)-6-(2,4-dichloro-phenyl)-pyridin-2-yl]-piperidin-1-yl-methanone 302572 5-(4-Chloro-phenyl)-6-(2,4-dichloro-phenyl)-2-(2,4-difluoro-benzyloxy)-nicotinonitrile 302575 4-(2,3-Dichloro-5-methoxy-phenylamino)-6-methoxy-7-((E)-2-pyrazin-2-yl-vinyl)-quinoline-3-carbonitrile 302577 5-(4-Chloro-phenyl)-6-(2,4-dichloro-phenyl)-pyridine-2-carboxylic acid phenylamide 302579 6-Pyridin-3-ylethynyl-4-(3,4,5-trimethoxy-phenylamino)-quinoline-3-carbonitrile 302581 trans-4-Bromo-N-{4-[(4-dimethylamino-quinazolin-2-ylamino)-methyl]-cyclohexylmethyl}-2-trifluoromethoxy-benzamide 302584 4-(2-Chloro-5-methoxy-phenylamino)-6-methoxy-7-((E)-2-pyridin-4-yl-vinyl)-quinoline-3-carbonitrile 302591 5-(4-Chloro-phenyl)-6-(2,4-dichloro-phenyl)-pyridine-2-carboxylic acid hexylamide 302592 (S)-2-{3-[4-(3,5-Difluoro-benzyloxy)-phenyl]-ureido}-N-(3-morpholin-4-yl-propyl)-3-phenyl-propionamide 302597 4-(2,3-Dichloro-5-methoxy-phenylamino)-7-((E)-2-pyrazin-2-yl-vinyl)-quinoline-3-carbonitrile 302598 2-(3,4-difluorobenzyloxy)-5-(4-chlorophenyl)-6-(2,4-dichlorophenyl)nicotinonitrile 302599 4-Bromo-N-[4-(4-dimethylamino-quinazolin-2-ylamino)-cyclohexyl]-2-trifluoromethoxy-benzenesulfonamide 302600 4-(2,3-Dichloro-5-methoxy-phenylamino)-7-[(E)-2-(1H-imidazol-2-yl)-vinyl]-quinoline-3-carbonitrile 302602 5-(4-Chloro-phenyl)-6-(2,4-dichloro-phenyl)-pyridine-2-carboxylic acid benzylamide 302603 6-Methoxy-7-((E)-2-pyridin-4-yl-vinyl)-4-(3,4,5-trimethoxy-phenylamino)-quinoline-3-carbonitrile 302610 5-(4-Chloro-phenyl)-6-(2,4-dichloro-phenyl)-pyridine-2-carboxylic acid (1-propyl-butyl)-amide 302621 1,3-Dipropyl-8-[4-(3-o-tolyl-[1,2,4]oxadiazol-5-ylmethoxy)-phenyl]-3,7-dihydro-purine-2,6-dione 302622 1,3-Dipropyl-8-[4-(5-p-tolyl-[1,2,4]oxadiazol-3-ylmethoxy)-phenyl]-3,7-dihydro-purine-2,6-dione 302627 8-{4-[3-(3-Fluoro-phenyl)-[1,2,4]oxadiazol-5-ylmethoxy]-phenyl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 302628 1,3-Dipropyl-8-{4-[3-(4-trifluoromethyl-phenyl)-[1,2,4]oxadiazol-5-ylmethoxy]-phenyl}-3,7-dihydro-purine-2,6-dione 302629 (S)-2-{3-[4-(3-Fluoro-phenoxy)-phenyl]-ureido}-N-(3-morpholin-4-yl-propyl)-3-phenyl-propionamide 302633 (R)-2-{3-[4-(3-Chloro-benzyloxy)-phenyl]-ureido}-N-(3-morpholin-4-yl-propyl)-3-phenyl-propionamide 302634 (S)-N-(3-Morpholin-4-yl-propyl)-3-phenyl-2-{3-[4-(4-trifluoromethyl-benzyloxy)-phenyl]-ureido}-propionamide 302635 (R)-N-(3-Morpholin-4-yl-propyl)-3-phenyl-2-{3-[4-(4-trifluoromethyl-benzyloxy)-phenyl]-ureido}-propionamide 302636 (S)-2-{3-[4-(3,5-Dimethoxy-benzyloxy)-phenyl]-ureido}-N-(3-morpholin-4-yl-propyl)-3-phenyl-propionamide 302641 (R)-2-{3-[4-(4-Ethyl-phenoxy)-phenyl]-ureido}-N-(3-morpholin-4-yl-propyl)-3-phenyl-propionamide 302643 (R)-2-{3-[4-(4-tert-Butyl-phenoxy)-phenyl]-ureido}-N-(3-morpholin-4-yl-propyl)-3-phenyl-propionamide 302644 8-{4-[3-(3-Methoxy-phenyl)-[1,2,4]oxadiazol-5-ylmethoxy]-phenyl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 302648 8-{4-[3-(4-Fluoro-phenyl)-[1,2,4]oxadiazol-5-ylmethoxy]-phenyl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 302651 8-{4-[5-(2-Methoxy-phenyl)-[1,2,4]oxadiazol-3-ylmethoxy]-phenyl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 302653 8-{4-[3-(2-Chloro-phenyl)-[1,2,4]oxadiazol-5-ylmethoxy]-phenyl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 302655 4-{5-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxymethyl]-[1,2,4]oxadiazol-3-yl}-benzonitrile 302657 8-{4-[5-(4-Methoxy-phenyl)-[1,2,4]oxadiazol-3-ylmethoxy]-phenyl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 302658 (S)-2-{3-[4-(4-Isopropyl-phenoxy)-phenyl]-ureido}-N-(3-morpholin-4-yl-propyl)-3-phenyl-propionamide 302666 1,3-Dipropyl-8-{4-[3-(2-trifluoromethyl-phenyl)-[1,2,4]oxadiazol-5-ylmethoxy]-phenyl}-3,7-dihydro-purine-2,6-dione 302667 (S)-N-(3-Morpholin-4-yl-propyl)-3-phenyl-2-{3-[4-(4-trifluoromethyl-phenoxy)-phenyl]-ureido}-propionamide 302671 8-{4-[3-(3-Chloro-phenyl)-[1,2,4]oxadiazol-5-ylmethoxy]-phenyl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 302674 1,3-Dipropyl-8-[4-(3-p-tolyl-[1,2,4]oxadiazol-5-ylmethoxy)-phenyl]-3,7-dihydro-purine-2,6-dione 302680 8-{4-[5-(2-Chloro-phenyl)-[1,2,4]oxadiazol-3-ylmethoxy]-phenyl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 302683 1,3-Dipropyl-8-[4-(5-o-tolyl-[1,2,4]oxadiazol-3-ylmethoxy)-phenyl]-3,7-dihydro-purine-2,6-dione 302685 (S)-2-{3-[4-(4-Fluoro-phenoxy)-phenyl]-ureido}-N-(3-morpholin-4-yl-propyl)-3-phenyl-propionamide 302687 1,3-Dipropyl-8-{4-[3-(3-trifluoromethyl-phenyl)-[1,2,4]oxadiazol-5-ylmethoxy]-phenyl}-3,7-dihydro-purine-2,6-dione 302696 8-{4-[3-(4-Chloro-phenyl)-[1,2,4]oxadiazol-5-ylmethoxy]-phenyl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 302698 8-{4-[3-(2-Methoxy-phenyl)-[1,2,4]oxadiazol-5-ylmethoxy]-phenyl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 302703 8-{4-[5-(3-Chloro-phenyl)-[1,2,4]oxadiazol-3-ylmethoxy]-phenyl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 302704 (R)-2-{3-[4-(4-Isopropyl-phenoxy)-phenyl]-ureido}-N-(3-morpholin-4-yl-propyl)-3-phenyl-propionamide 302706 1,3-Dipropyl-8-[4-(5-m-tolyl-[1,2,4]oxadiazol-3-ylmethoxy)-phenyl]-3,7-dihydro-purine-2,6-dione 302720 (S)-2-{3-[4-(4-Fluoro-phenylsulfanyl)-phenyl]-ureido}-N-(3-morpholin-4-yl-propyl)-3-phenyl-propionamide 302725 (S)-2-{3-[4-(4-Ethyl-phenoxy)-phenyl]-ureido}-N-(3-morpholin-4-yl-propyl)-3-phenyl-propionamide 302726 (S)-2-{3-[4-(4-tert-Butyl-phenoxy)-phenyl]-ureido}-N-(3-morpholin-4-yl-propyl)-3-phenyl-propionamide 302738 1,3-Dipropyl-8-{4-[5-(3-trifluoromethyl-phenyl)-[1,2,4]oxadiazol-3-ylmethoxy]-phenyl}-3,7-dihydro-purine-2,6-dione 302751 1-(1-(4-(6-isobutyl-5-oxo-3-phenyl-4,5-dihydropyrazin-2-yl)benzyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one 302755 1,3-Dipropyl-8-{4-[5-(4-trifluoromethyl-phenyl)-[1,2,4]oxadiazol-3-ylmethoxy]-phenyl}-3,7-dihydro-purine-2,6-dione 302758 [Tyr-Pro-Phe-Phe-NH-]2 302759 [Tyr-Pro-Phe-Phe-NH-CH2-]2 302779 8-{4-[5-(4-Chloro-phenyl)-[1,2,4]oxadiazol-3-ylmethoxy]-phenyl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 302794 4-{3-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxymethyl]-[1,2,4]oxadiazol-5-yl}-benzonitrile 302796 Tyr-Pro-Phe-Phe-OCH3 302797 Tyr-Pro-Phe-Phe-NHNH2 302805 8-{4-[5-(2-Fluoro-phenyl)-[1,2,4]oxadiazol-3-ylmethoxy]-phenyl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 302819 1-(1-{4-[6-(2-Methyl-2H-tetrazol-5-yl)-3-phenyl-quinoxalin-2-yl]-benzyl}-piperidin-4-yl)-1,3-dihydro-benzoimidazol-2-one 302820 1-(1-{4-[7-(2-Methyl-2H-tetrazol-5-yl)-3-phenyl-quinoxalin-2-yl]-benzyl}-piperidin-4-yl)-1,3-dihydro-benzoimidazol-2-one 302821 1-(1-(4-(7-phenyl-1H-pyrazolo[4,3-g]quinoxalin-6-yl)benzyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one 302825 [Tyr-Pro-Phe-NH-]2 302826 [Tyr-Pro-Phe-NH-CH2-]2 302839 1-{1-[4-(6-Benzyl-5-oxo-3-phenyl-4,5-dihydro-pyrazin-2-yl)-benzyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 302850 1-(1-(4-(6-(4-hydroxybenzyl)-5-oxo-3-phenyl-4,5-dihydropyrazin-2-yl)benzyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one 302859 1-{1-[4-(6-sec-Butyl-5-oxo-3-phenyl-4,5-dihydro-pyrazin-2-yl)-benzyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 302862 8-{4-[5-(4-Fluoro-phenyl)-[1,2,4]oxadiazol-3-ylmethoxy]-phenyl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 302879 5-(4-Chloro-phenyl)-6-(2,4-dichloro-phenyl)-2-(3,4-difluoro-benzyloxy)-N-ethyl-nicotinamide 302880 2-Butoxy-5-(4-chloro-phenyl)-6-(2,4-dichloro-phenyl)-N-methyl-nicotinamide 302881 (S)-4-(3,4-Difluoro-phenyl)-6-methoxymethyl-2-oxo-3-[3-(3'',4'',5'',6''-tetrahydro-2''H-[2,4'']bipyridinyl-1''-yl)-propylcarbamoyl]-1,2,3,4-tetrahydro-pyrimidine-5-carboxylic acid methyl ester 302882 N-((S)-1-{4-[4-Methoxy-2-(4-methoxy-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-4-methyl-benzamide 302883 SID29215557 302884 5-(4-Chloro-phenyl)-N-cyclohexyl-6-(2,4-dichloro-phenyl)-nicotinamide 302885 2-Benzyloxy-5-(4-chloro-phenyl)-N-cyclopentyl-6-(2,4-dichloro-phenyl)-nicotinamide 302886 6-{3-[4-(2-Hydroxymethyl-2,3-dihydro-benzo[1,4]dioxin-6-yl)-piperazin-1-yl]-propylamino}-1,3-dimethyl-1H-pyrimidine-2,4-dione 302888 3-Bromo-N-[4-(4-dimethylamino-quinazolin-2-ylamino)-cyclohexyl]-benzamide 302889 SID29215033 302890 2-Butoxy-5-(4-chloro-phenyl)-6-(2,4-dichloro-phenyl)-N-propyl-nicotinamide 302891 N-[4-(4-Dimethylamino-quinazolin-2-ylamino)-cyclohexyl]-2-fluoro-benzamide 302892 (S)-2-(2-Amino-ethoxymethyl)-6-ethyl-4-(4-nitro-phenyl)-1,4-dihydro-pyridine-3,5-dicarboxylic acid 5-amide 3-{[3-(4,4-diphenyl-piperidin-1-yl)-propyl]-amide} 302893 2-Butoxy-5-(4-chloro-phenyl)-6-(2,4-dichloro-phenyl)-nicotinic acid methyl ester 302894 [5-(4-Chloro-phenyl)-6-(2,4-dichloro-phenyl)-pyridin-3-yl]-piperidin-1-yl-methanone 302895 N-[4-(4-Dimethylamino-quinazolin-2-ylamino)-cyclohexyl]-3-trifluoromethyl-benzamide 302896 SID11113929 302898 5-(4-Chloro-phenyl)-6-(2,4-dichloro-phenyl)-2-(3,4-difluoro-benzyloxy)-N-propyl-nicotinamide 302899 N-[4-(4-Dimethylamino-quinazolin-2-ylamino)-cyclohexyl]-3-fluoro-benzamide 302900 SID29217472 302902 3,4-Dichloro-N-[4-(4-dimethylamino-quinazolin-2-ylamino)-cyclohexyl]-benzamide 302903 5-(4-Chloro-phenyl)-6-(2,4-dichloro-phenyl)-N-piperidin-1-yl-nicotinamide 302904 2-Benzyloxy-5-(4-chloro-phenyl)-6-(2,4-dichloro-phenyl)-N-piperidin-1-yl-nicotinamide 302905 5-(4-Chloro-phenyl)-2-cyclohexylmethoxy-6-(2,4-dichloro-phenyl)-N-methyl-nicotinamide 302909 2-(4-(3-phenylquinoxalin-2-yl)phenyl)propan-2-amine 302911 N-((S)-1-{4-[4-Methoxy-2-(4-methoxy-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-butyramide 302914 5-(4-Chloro-phenyl)-6-(2,4-dichloro-phenyl)-2-(3,4-difluoro-benzyloxy)-N-(2-fluoro-ethyl)-nicotinamide 302919 5-(4-Chloro-phenyl)-2-cyclohexylmethoxy-6-(2,4-dichloro-phenyl)-N-propyl-nicotinamide 302921 N-[4-(4-Dimethylamino-quinazolin-2-ylamino)-cyclohexyl]-3,5-dimethoxy-benzamide 302923 2-Benzyloxy-5-(4-chloro-phenyl)-6-(2,4-dichloro-phenyl)-N-methyl-nicotinamide 302924 SID11113796 302925 Cyclopropanecarboxylic acid ((S)-1-{4-[4-methoxy-2-(4-methoxy-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-amide 302926 3-Cyano-N-[4-(4-dimethylamino-quinazolin-2-ylamino)-cyclohexyl]-benzamide 302929 5-(4-Chloro-phenyl)-6-(2,4-dichloro-phenyl)-2-(3,4-difluoro-benzyloxy)-N-isopropyl-nicotinamide 302930 (R)-5-[3-(4,4-Diphenyl-piperidin-1-yl)-propylcarbamoyl]-2,6-dimethyl-4-(4-nitro-phenyl)-1,4-dihydro-pyridine-3-carboxylic acid methyl ester 302931 cis-N*2*-[4-(4-Bromo-2-trifluoromethoxy-benzylamino)-cyclohexyl]-N*4*,N*4*-dimethyl-quinazoline-2,4-diamine 302933 1-(1-(4-(5-oxo-3-phenyl-4,5-dihydropyrazin-2-yl)benzyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one 302934 (S)-1,2-Dimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-9,11-dioxa-6-aza-benzo[fg]cyclopenta[b]anthracene 302935 2-Benzyloxy-5-(4-chloro-phenyl)-6-(2,4-dichloro-phenyl)-N,N-dimethyl-nicotinamide 302936 2-Chloro-5-(4-chloro-phenyl)-6-(2,4-dichloro-phenyl)-N,N-dimethyl-nicotinamide 302937 2-Chloro-5-(4-chloro-phenyl)-6-(2,4-dichloro-phenyl)-N-propyl-nicotinamide 302939 N-((S)-1-{4-[4-Methoxy-2-(4-methoxy-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-2,2-dimethyl-propionamide 302940 5-(4-Chloro-phenyl)-2-cyclohexylmethoxy-6-(2,4-dichloro-phenyl)-nicotinic acid methyl ester 302941 2-Butoxy-5-(4-chloro-phenyl)-6-(2,4-dichloro-phenyl)-nicotinamide 302942 [(S)-1-(2,3-Dihydro-benzo[1,4]oxathiin-2-yl)methyl]-[2-(2,6-dimethoxy-phenoxy)-ethyl]-amine 302943 (5S,6R)-3-(3-{4-[4-Fluoro-2-(2,2,2-trifluoro-ethoxy)-phenyl]-piperazin-1-yl}-propyl)-5,6-dihydroxy-5-methyl-dihydro-pyrimidine-2,4-dione 302944 1-((S)-1-{4-[4-Methoxy-2-(4-methoxy-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-3-p-tolyl-urea 302946 5-(4-Chloro-phenyl)-6-(2,4-dichloro-phenyl)-N-hexyl-nicotinamide 302947 N-[4-(4-Dimethylamino-quinazolin-2-ylamino)-cyclohexyl]-4-fluoro-benzamide 302948 SID11110760 302949 2-Benzyloxy-5-(4-chloro-phenyl)-6-(2,4-dichloro-phenyl)-nicotinic acid methyl ester 302950 2-Chloro-5-(4-chloro-phenyl)-6-(2,4-dichloro-phenyl)-N-hexyl-nicotinamide 302953 4-[2-Naphthalen-1-yl-5-oxo-oxazol-(4E)-ylidenemethyl]-N-phenyl-piperazine-1-carboxamidine 302954 5-(4-Chloro-phenyl)-6-(2,4-dichloro-phenyl)-2-(3,4-difluoro-benzyloxy)-N-methyl-nicotinamide 302955 2-Benzyloxy-5-(4-chloro-phenyl)-6-(2,4-dichloro-phenyl)-N-ethyl-nicotinamide 302956 (4-Bromo-2-trifluoromethoxy-phenyl)-[4-(4-dimethylamino-quinazolin-2-ylamino)-piperidin-1-yl]-methanone 302957 2,6-Dimethyl-4-(4-nitro-phenyl)-1,4-dihydro-pyridine-3,5-dicarboxylic acid 3-amide 5-{[4-(4,4-diphenyl-piperidin-1-yl)-butyl]-amide} 302958 3-Chloro-N-[4-(4-dimethylamino-quinazolin-2-ylamino)-cyclohexyl]-benzamide 302959 N-((S)-1-{4-[4-Methoxy-2-(4-methoxy-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-2-phenyl-acetamide 302960 N*2*-[1-(4-Bromo-2-trifluoromethoxy-benzyl)-piperidin-4-yl]-N*4*,N*4*-dimethyl-quinazoline-2,4-diamine 302961 5-(4-Chloro-phenyl)-6-(2,4-dichloro-phenyl)-2-(3,4-difluoro-benzyloxy)-nicotinic acid methyl ester 302962 2-Chloro-5-(4-chloro-phenyl)-6-(2,4-dichloro-phenyl)-N-piperidin-1-yl-nicotinamide 302963 1-(4-Fluoro-phenyl)-3-((S)-1-{4-[4-methoxy-2-(4-methoxy-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-urea 302965 1-{4-[4-(2-Isopropoxy-phenyl)-piperazin-1-yl]-2-oxo-butyl}-5-oxo-pyrrolidine-2-carboxylic acid ethyl ester 302966 2-Benzyloxy-5-(4-chloro-phenyl)-6-(2,4-dichloro-phenyl)-N-propyl-nicotinamide 302971 1-((R)-2-Amino-2-phenyl-ethyl)-3-(2,6-difluoro-benzyl)-5-(2-fluoro-phenyl)-[1,3,5]triazinane-2,4,6-trione 302973 (E)-3-(2-{(E)-3-[2-(2,6-Dichloro-benzyloxy)-3-methyl-phenyl]-allyl}-phenyl)-acrylic acid 302990 Butane-1-sulfonic acid ((S)-1-{4-[4-methoxy-2-(4-methoxy-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-amide 302991 N-[4-(4-Dimethylamino-quinazolin-2-ylamino)-cyclohexyl]-3-nitro-benzamide 302992 1-((R)-2-Amino-2-phenyl-ethyl)-3-(2,6-difluoro-benzyl)-5-(2,6-difluoro-phenyl)-[1,3,5]triazinane-2,4,6-trione 302995 (E)-3-{2-[3-(2-Benzyloxy-3-methyl-phenyl)-propyl]-phenyl}-acrylic acid 303006 N-[4-(4-Dimethylamino-quinazolin-2-ylamino)-cyclohexyl]-3-methyl-benzamide 303007 N-((S)-1-{4-[4-Methoxy-2-(4-methoxy-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-benzenesulfonamide 303009 1-((R)-2-Amino-2-phenyl-ethyl)-3-benzo[1,2,5]thiadiazol-5-yl-5-(2,6-difluoro-benzyl)-[1,3,5]triazinane-2,4,6-trione 303011 (E)-3-{2-[3-(2-Benzyloxy-3-methoxy-phenyl)-propyl]-phenyl}-acrylic acid 303012 4-Methoxy-N-((S)-1-{4-[4-methoxy-2-(4-methoxy-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-benzamide 303021 N-[4-(4-Dimethylamino-quinazolin-2-ylamino)-cyclohexyl]-2,3,4-trifluoro-benzamide 303026 3-{2-[3-(2-Benzyloxy-3-methyl-phenyl)-propyl]-phenyl}-propionic acid 303030 N-((S)-1-{4-[4-Methoxy-2-(4-methoxy-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-4-methyl-benzenesulfonamide 303031 3,5-Dichloro-N-((S)-1-{4-[4-methoxy-2-(4-methoxy-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-benzenesulfonamide 303034 1-[2-Amino-3-(1H-indol-3-yl)-propyl]-3-(2,6-difluoro-benzyl)-5-(2,6-difluoro-phenyl)-[1,3,5]triazinane-2,4,6-trione 303040 3,4-Dichloro-N-((S)-1-{4-[4-methoxy-2-(4-methoxy-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-benzamide 303045 (E)-3-{2-[(E)-3-(2-Hydroxy-3-methyl-phenyl)-allyl]-phenyl}-acrylic acid 303049 3-{2-[2-(2-Benzyloxy-3-methyl-phenyl)-cyclopropyl]-phenyl}-propionic acid 303053 2,2,2-Trifluoro-N-((S)-1-{4-[4-methoxy-2-(4-methoxy-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-acetamide 303056 (E)-3-{2-[(E)-2-(2-Benzyloxy-phenyl)-vinyl]-phenyl}-acrylic acid 303061 N-((S)-1-{4-[4-Methoxy-2-(4-methoxy-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-C-phenyl-methanesulfonamide 303071 N-((S)-1-{4-[4-Methoxy-2-(4-methoxy-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-methanesulfonamide 303082 N-((S)-1-{4-[4-Methoxy-2-(4-methoxy-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-acetamide 303083 1-((S)-1-{4-[4-Methoxy-2-(4-methoxy-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-3-propyl-urea 303086 3-(2-{(E)-3-[2-(2,6-Dichloro-benzyloxy)-3-methyl-phenyl]-1-hydroxy-allyl}-phenyl)-acrylic acid 303098 (E)-3-(2-{(E)-3-[2-(4-Fluoro-benzyloxy)-3-methyl-phenyl]-allyl}-phenyl)-acrylic acid 303100 1-(2,6-Difluoro-benzyl)-3-(3-methoxy-phenyl)-5-{2-[methyl-(2-pyridin-2-yl-ethyl)-amino]-ethyl}-[1,3,5]triazinane-2,4,6-trione 303101 Ethanesulfonic acid ((S)-1-{4-[4-methoxy-2-(4-methoxy-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-amide 303102 N-((S)-1-{4-[4-Methoxy-2-(4-methoxy-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-propionamide 303107 3-(2-{(E)-3-[2-(2,6-Dichloro-benzyloxy)-3-methyl-phenyl]-3-hydroxy-propenyl}-phenyl)-acrylic acid 303108 1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3-{(S)-1-[3-(4-fluoro-phenyl)-propyl]-piperidin-3-ylmethyl}-urea 303109 1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3-{(S)-1-[2-(4-fluoro-phenyl)-ethyl]-piperidin-3-ylmethyl}-urea 303112 (S)-3-(2,3-Dichloro-phenyl)-1-(2-diethylamino-ethyl)-3-hydroxy-2-oxo-4-trifluoromethyl-2,3-dihydro-1H-indole-6-carboxylic acid amide 303114 1-{(S)-1-[2-(4-Fluoro-phenyl)-ethyl]-piperidin-3-ylmethyl}-3-[3-(1-methyl-1H-tetrazol-5-yl)-phenyl]-urea 303115 1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3-{(S)-1-[2-(4-methoxy-phenyl)-ethyl]-piperidin-3-ylmethyl}-urea 303120 (S)-3-(2-Chloro-phenyl)-1-(2-diethylamino-ethyl)-3-hydroxy-2-oxo-4-trifluoromethyl-2,3-dihydro-1H-indole-6-carboxylic acid amide 303125 1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3-{(S)-1-[2-(3-fluoro-phenyl)-ethyl]-piperidin-3-ylmethyl}-urea 303126 1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3-{(3S,4S)-1-[2-(4-fluoro-phenyl)-ethyl]-4-methyl-piperidin-3-ylmethyl}-urea 303127 (S)-3-(2,4-Dichloro-phenyl)-1-(2-diethylamino-ethyl)-3-hydroxy-2-oxo-4-trifluoromethyl-2,3-dihydro-1H-indole-6-carboxylic acid amide 303130 1-{(R)-1-[3-(4-Fluoro-phenyl)-propyl]-piperidin-3-ylmethyl}-3-[3-(1-methyl-1H-tetrazol-5-yl)-phenyl]-urea 303137 1-{(S)-1-[2-(4-Dimethylamino-phenyl)-ethyl]-piperidin-3-ylmethyl}-3-[3-ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-urea 303139 1-[1-(4-Fluoro-benzyl)-piperidin-4-ylmethyl]-3-[3-(1-methyl-1H-tetrazol-5-yl)-phenyl]-urea 303140 1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3-{(S)-1-[2-(2-fluoro-phenyl)-ethyl]-piperidin-3-ylmethyl}-urea 303141 (R)-3-(3-Chloro-phenyl)-1-(2-diethylamino-ethyl)-3-hydroxy-2-oxo-4-trifluoromethyl-2,3-dihydro-1H-indole-6-carboxylic acid amide 303144 (S)-3-(2,5-Dichloro-phenyl)-1-(2-diethylamino-ethyl)-3-hydroxy-2-oxo-4-trifluoromethyl-2,3-dihydro-1H-indole-6-carboxylic acid amide 303152 1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3-{(R)-1-[2-(4-fluoro-phenyl)-ethyl]-piperidin-3-yl}-urea 303153 1-(2-Amino-2-phenyl-ethyl)-3-(2,6-difluoro-benzyl)-5-(3-methoxy-phenyl)-[1,3,5]triazinane-2,4,6-trione 303156 (R)-3-(4-Chloro-phenyl)-1-(2-diethylamino-ethyl)-3-hydroxy-2-oxo-4-trifluoromethyl-2,3-dihydro-1H-indole-6-carboxylic acid amide 303159 (S)-3-(2,6-Dichloro-phenyl)-1-(2-diethylamino-ethyl)-3-hydroxy-2-oxo-4-trifluoromethyl-2,3-dihydro-1H-indole-6-carboxylic acid amide 303170 1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3-{(R)-1-[2-(4-fluoro-phenyl)-ethyl]-piperidin-3-ylmethyl}-urea 303185 (S)-1-(2-Diethylamino-ethyl)-3-hydroxy-3-(2-methoxy-phenyl)-2-oxo-4-trifluoromethyl-2,3-dihydro-1H-indole-6-carboxylic acid amide 303187 1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3-[(S)-1-(2-p-tolyl-ethyl)-piperidin-3-ylmethyl]-urea 303189 1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3-{(R)-1-[3-(4-fluoro-phenyl)-propyl]-piperidin-3-yl}-urea 303200 1-(2-Diethylamino-ethyl)-3-hydroxy-2-oxo-3-phenyl-4-trifluoromethyl-2,3-dihydro-1H-indole-6-carboxylic acid amide 303201 (R)-1-(2-Diethylamino-ethyl)-3-hydroxy-3-(3-methoxy-phenyl)-2-oxo-4-trifluoromethyl-2,3-dihydro-1H-indole-6-carboxylic acid amide 303203 1-{(R)-1-[2-(4-Fluoro-phenyl)-ethyl]-piperidin-3-ylmethyl}-3-[3-(1-methyl-1H-tetrazol-5-yl)-phenyl]-urea 303205 1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3-{(S)-1-[2-(4-trifluoromethyl-phenyl)-ethyl]-piperidin-3-ylmethyl}-urea 303207 1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3-{(R)-1-[3-(4-fluoro-phenyl)-propyl]-piperidin-3-ylmethyl}-urea 303214 1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3-{(R)-1-[4-(4-fluoro-phenyl)-butyl]-piperidin-3-yl}-urea 303218 (R)-1-(2-Diethylamino-ethyl)-3-hydroxy-3-(4-methoxy-phenyl)-2-oxo-4-trifluoromethyl-2,3-dihydro-1H-indole-6-carboxylic acid amide 303225 3-(2-Chloro-phenyl)-1-(2-diethylamino-ethyl)-3-hydroxy-2-oxo-4-trifluoromethyl-2,3-dihydro-1H-indole-6-carboxylic acid amide 303233 1-{(S)-1-[3-(4-Fluoro-phenyl)-propyl]-piperidin-3-ylmethyl}-3-[3-(1-methyl-1H-tetrazol-5-yl)-phenyl]-urea 303241 1-{(S)-1-[2-(2,4-Dichloro-phenyl)-ethyl]-piperidin-3-ylmethyl}-3-[3-ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-urea 303260 1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3-((S)-1-phenethyl-piperidin-3-ylmethyl)-urea 303272 1-{(3S,4S)-4-Ethyl-1-[2-(4-fluoro-phenyl)-ethyl]-piperidin-3-ylmethyl}-3-[3-ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-urea 303280 1-{1-[2-(4-Fluoro-phenyl)-ethyl]-piperidin-4-ylmethyl}-3-[3-(1-methyl-1H-tetrazol-5-yl)-phenyl]-urea 303287 1-{(S)-1-[2-(2,4-Difluoro-phenyl)-ethyl]-piperidin-3-ylmethyl}-3-[3-ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-urea 303295 1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3-{(3S,4R)-1-[2-(4-fluoro-phenyl)-ethyl]-4-isopropyl-piperidin-3-ylmethyl}-urea 303303 1-{1-[3-(4-Fluoro-phenyl)-propyl]-piperidin-4-ylmethyl}-3-[3-(1-methyl-1H-tetrazol-5-yl)-phenyl]-urea 303309 1-{(S)-1-[2-(3,4-Difluoro-phenyl)-ethyl]-piperidin-3-ylmethyl}-3-[3-ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-urea 303310 1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3-{(S)-1-[2-(4-fluoro-phenyl)-ethyl]-4,4-dimethyl-piperidin-3-ylmethyl}-urea 303324 1-{(S)-1-[2-(4-Chloro-phenyl)-ethyl]-piperidin-3-ylmethyl}-3-[3-ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-urea 303330 1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3-{(3S,4S)-1-[2-(4-fluoro-phenyl)-ethyl]-4-trifluoromethyl-piperidin-3-ylmethyl}-urea 303331 1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3-{(3S,4S)-1-[2-(4-fluoro-phenyl)-ethyl]-4-phenyl-piperidin-3-ylmethyl}-urea 303343 1-{(S)-1-[2-(4-Fluoro-phenyl)-ethyl]-piperidin-3-ylmethyl}-3-[3-(1-methyl-1H-tetrazol-5-yl)-phenyl]-urea 303353 1-{(S)-1-[2-(3-Chloro-phenyl)-ethyl]-piperidin-3-ylmethyl}-3-[3-ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-urea 303361 Biphenyl-3-carboxylic acid [(S)-1-(3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethyl]-amide 303365 1-(1-{2-[1-(2-Chloro-5-methyl-phenoxy)-cyclohexyl]-2-hydroxy-ethyl}-piperidin-4-yl)-1,3-dihydro-benzoimidazol-2-one 303371 2-(Biphenyl-4-yloxy)-2-methyl-N-[(R)-1-(3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethyl]-propionamide 303372 (S)-2-(3-Benzyl-3-methyl-ureido)-N-(3-morpholin-4-yl-propyl)-3-phenyl-propionamide 303377 (S)-N-(3-Morpholin-4-yl-propyl)-2-[3-(3-phenoxy-phenyl)-ureido]-3-phenyl-propionamide 303378 1-[1-(2-Cyclohexyl-2-hydroxy-ethyl)-piperidin-4-yl]-1,3-dihydro-benzoimidazol-2-one 303384 (R)-2-(3-Benzyl-3-methyl-ureido)-N-(3-morpholin-4-yl-propyl)-3-phenyl-propionamide 303385 (S)-2-Diphenylacetylamino-N-(3-morpholin-4-yl-propyl)-3-phenyl-propionamide 303389 2-(Biphenyl-3-yloxy)-2-methyl-N-[(S)-1-(3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethyl]-propionamide 303393 (R)-N-(3-Morpholin-4-yl-propyl)-2-[3-(3-phenoxy-phenyl)-ureido]-3-phenyl-propionamide 303394 1-(1-{2-[1-(2-Chloro-5-methyl-phenoxy)-cyclohexyl]-ethyl}-piperidin-4-yl)-1,3-dihydro-benzoimidazol-2-one 303406 2-(Biphenyl-3-yloxy)-2-methyl-N-[(R)-1-(3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethyl]-propionamide 303411 (S)-N-(3-Morpholin-4-yl-propyl)-2-[3-(2-phenoxy-phenyl)-ureido]-3-phenyl-propionamide 303412 1-{1-[3-(2-Chloro-5-methyl-phenoxy)-propyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303417 2-(Biphenyl-2-yloxy)-2-methyl-N-[(S)-1-(3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethyl]-propionamide 303426 1-{1-[3-((S)-2-Chloro-5-methyl-phenoxy)-2-hydroxy-propyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303431 2-(3-Chloro-phenoxy)-2-methyl-N-[(R)-1-(3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethyl]-propionamide 303432 2-(Biphenyl-2-yloxy)-2-methyl-N-[(R)-1-(3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethyl]-propionamide 303436 3-Hydroxy-3-phenyl-piperidine-1-carboxylic acid [1-((S)-3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethyl]-amide 303458 1-{1-[3-(4-Fluoro-2-methyl-phenoxy)-4-methyl-pentyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303468 (S)-N-(3-Morpholin-4-yl-propyl)-2-[3-(4-phenoxy-phenyl)-ureido]-3-phenyl-propionamide 303470 1-{1-[3-(2-Chloro-5-methyl-phenoxy)-4-methyl-pentyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303472 1-{1-[3-(2-Chloro-5-methyl-phenoxy)-3-cyclohexyl-2-hydroxy-propyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303475 (S)-2-{3-[4-(4-Methyl-benzyloxy)-phenyl]-ureido}-N-(3-morpholin-4-yl-propyl)-3-phenyl-propionamide 303476 1-{1-[3-(4-Fluoro-3-methyl-phenoxy)-4-methyl-pentyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303478 1-{1-[4-Methyl-3-(2-methyl-5-nitro-phenoxy)-pentyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303485 1-{1-[3-((R)-2-Chloro-5-methyl-phenoxy)-2-hydroxy-propyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303490 2-(Biphenyl-4-yloxy)-2-methyl-N-[(S)-1-(3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethyl]-propionamide 303491 1-[1-(4-Methyl-3-o-tolyloxy-pentyl)-piperidin-4-yl]-1,3-dihydro-benzoimidazol-2-one 303493 1-{1-[3-(2-Chloro-5-methyl-phenoxy)-2-hydroxy-5-methyl-hexyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303497 (R)-N-(3-Morpholin-4-yl-propyl)-2-[3-(4-phenoxy-phenyl)-ureido]-3-phenyl-propionamide 303501 (S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionamide 303503 (S)-2-[3-(4-Benzyloxy-phenyl)-ureido]-N-(3-morpholin-4-yl-propyl)-3-phenyl-propionamide 303506 1-{1-[3-(2-Ethyl-phenoxy)-4-methyl-pentyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303508 1-{1-[3-(2-Chloro-5-methyl-phenoxy)-2-hydroxy-4-phenyl-butyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303509 1-{1-[3-(5-Amino-2-methyl-phenoxy)-4-methyl-pentyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303516 1-{1-[3-(2-Chloro-5-methyl-phenoxy)-2-hydroxy-butyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303517 (S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-N-methyl-propionamide 303521 1-(1-{2-[1-(2-Chloro-5-methyl-phenoxy)-cyclohexyl]-2-imidazol-1-yl-ethyl}-piperidin-4-yl)-1,3-dihydro-benzoimidazol-2-one 303522 1-{1-[4-Methyl-3-(2-trifluoromethyl-phenoxy)-pentyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303524 1-{1-[3-(2-Chloro-5-methyl-phenoxy)-2-hydroxy-3-phenyl-propyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303525 1-{1-[3-(2,5-Dimethyl-phenoxy)-4-methyl-pentyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303526 (R)-2-[3-(4-Benzyloxy-phenyl)-ureido]-N-(3-morpholin-4-yl-propyl)-3-phenyl-propionamide 303533 1-{1-[3-(2-Chloro-5-methyl-phenoxy)-2-hydroxy-pentyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303541 1-{1-[3-(2-Isopropyl-phenoxy)-4-methyl-pentyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303546 Biphenyl-2-carboxylic acid [(R)-1-(3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethyl]-amide 303547 1-{1-[3-(2-Chloro-5-methoxy-phenoxy)-4-methyl-pentyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303550 1-[2-[(S)-(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionylamino]-3-(4-hydroxy-phenyl)-propionylamino]-cyclohexanecarboxylic acid [(S)-1-(1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-ethyl]-amide 303555 4-Benzyl-piperidine-1-carboxylic acid [(S)-1-(3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethyl]-amide 303558 1-{1-[3-(2-Chloro-5-methyl-phenoxy)-2-hydroxy-hexyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303559 1-{1-[3-(2-Fluoro-5-methyl-phenoxy)-4-methyl-pentyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303562 2-(4-Chloro-phenoxy)-2-methyl-N-[(S)-1-(3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethyl]-propionamide 303563 1-(1-{2-[1-(2-Chloro-5-methyl-phenoxy)-cyclohexyl]-2-dimethylamino-ethyl}-piperidin-4-yl)-1,3-dihydro-benzoimidazol-2-one 303564 1-{1-[3-(2-Chloro-5-fluoro-phenoxy)-4-methyl-pentyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303572 4-Benzyl-piperidine-1-carboxylic acid [(R)-1-(3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethyl]-amide 303580 2-(4-Chloro-phenoxy)-2-methyl-N-[(R)-1-(3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethyl]-propionamide 303582 1-{1-[3-(2-Chloro-5-methyl-phenoxy)-3-phenyl-propyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303583 1-{1-[3-(2-Chloro-5-methyl-phenoxy)-2-hydroxy-4-methyl-pentyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303584 1-{1-[4-Methyl-3-(5-methyl-2-nitro-phenoxy)-pentyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 303588 8-[1-(2-Bromo-phenyl)-meth-(E)-ylidene]-3-tert-butyl-7,8-dihydro-6H-pyrrolo[1,2-a]thieno[2,3-d]pyrimidin-(4Z)-ylideneamine 303595 1-[3-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-1-hydroxy-prop-2-ynyl]-cyclobutanol 303596 2-Furan-2-yl-6-(3-phenoxy-prop-1-ynyl)-[1,2,4]triazolo[1,5-a]pyrazin-8-ylamine 303602 3-[1-(2-Bromo-phenyl)-meth-(E)-ylidene]-2,3-dihydro-1H-pyrrolo[2,1-b]quinazolin-(9Z)-ylideneamine 303603 3-[1-(2-Iodo-phenyl)-meth-(E)-ylidene]-2,3-dihydro-1H-pyrrolo[2,1-b]quinazolin-(9Z)-ylideneamine 303606 3-[1-(2-Chloro-phenyl)-meth-(E)-ylidene]-1,2,3,9-tetrahydro-pyrrolo[2,1-b]quinazoline 303614 8-[1-(2-Bromo-phenyl)-meth-(E)-ylidene]-2,3-dimethyl-7,8-dihydro-6H-pyrrolo[1,2-a]thieno[2,3-d]pyrimidin-(4Z)-ylideneamine 303615 1-[1-(2-Bromo-phenyl)-meth-(E)-ylidene]-2,3,5,6,7,8-hexahydro-1H-9-thia-3a,10-diaza-cyclopenta[b]fluoren-(4Z)-ylideneamine 303624 2-Furan-2-yl-6-[3-(pyridin-3-yloxy)-prop-1-ynyl]-[1,2,4]triazolo[1,5-a]pyrazin-8-ylamine 303627 1-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-3,6-dimethyl-hept-1-yn-3-ol 303633 3-[1-(2-Ethyl-phenyl)-meth-(E)-ylidene]-2,3-dihydro-1H-pyrrolo[2,1-b]quinazolin-(9Z)-ylideneamine 303661 6-(3-tert-Butoxy-but-1-ynyl)-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-8-ylamine 303662 3-[1-(4-Methoxy-phenyl)-meth-(E)-ylidene]-2,3-dihydro-1H-pyrrolo[2,1-b]quinazolin-(9Z)-ylideneamine 303663 [3-[1-(2-Bromo-phenyl)-meth-(E)-ylidene]-2,3-dihydro-1H-pyrrolo[2,1-b]quinazolin-(9Z)-ylidene]-methyl-amine 303690 6-(1-Amino-cyclohexylethynyl)-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-8-ylamine 303698 1-[3-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-1-hydroxy-prop-2-ynyl]-cyclohexanol 303699 3-[1-(2-Bromo-phenyl)-meth-(E)-ylidene]-2,3-dihydro-1H-pyrrolo[2,1-b]quinazolin-(9Z)-ylidene-cyanamide 303700 8-[1-(2-Bromo-phenyl)-meth-(E)-ylidene]-7,8-dihydro-6H-pyrrolo[1,2-a]thieno[2,3-d]pyrimidin-(4Z)-ylideneamine 303706 3-[1-(2-Bromo-phenyl)-meth-(E)-ylidene]-1-(4-fluoro-phenyl)-1,2,3,9-tetrahydro-pyrrolo[2,1-b]quinazoline 303715 3-[1-(2-Chloro-phenyl)-meth-(E)-ylidene]-2,3-dihydro-1H-pyrrolo[2,1-b]quinazolin-(9Z)-ylideneamine 303717 6-(3-Cyclohexyl-prop-1-ynyl)-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-8-ylamine 303725 8-[1-(2-Bromo-phenyl)-meth-(E)-ylidene]-3-cyclopropyl-7,8-dihydro-6H-pyrrolo[1,2-a]thieno[2,3-d]pyrimidin-(4Z)-ylideneamine 303730 6-{2-[2-Hydroxy-3-(1H-indol-4-yloxy)-propylamino]-propoxy}-4H-benzo[1,4]oxazin-3-one 303732 3-[1-(2,6-Dichloro-phenyl)-meth-(E)-ylidene]-1,2,3,9-tetrahydro-pyrrolo[2,1-b]quinazoline 303744 (R)-N-((R)-3-(4-chlorophenyl)-1-oxo-1-(4-(2-((2-(thiophen-2-yl)ethylamino)methyl)phenyl)piperazin-1-yl)propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 303745 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [(R)-1-(4-chloro-benzyl)-2-(4-{2-[(3-isobutoxy-propylamino)-methyl]-phenyl}-piperazin-1-yl)-2-oxo-ethyl]-amide 303746 6-{1-[2-(Quinolin-5-yloxy)-ethyl]-piperidin-4-ylmethyl}-4H-benzo[1,4]oxazin-3-one 303751 4-(8-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-2-methyl-1-(pyridin-4-yl)but-3-yn-2-ol 303756 6-{1-[2-(Naphthalen-1-yloxy)-ethyl]-piperidin-4-yloxy}-4H-benzo[1,4]oxazin-3-one 303757 3-[1-(2-Chloro-4-fluoro-phenyl)-meth-(E)-ylidene]-1,2,3,9-tetrahydro-pyrrolo[2,1-b]quinazoline 303760 6-{1-[2-(2-Methyl-quinolin-5-yloxy)-ethyl]-piperidin-4-ylmethyl}-4H-benzo[1,4]oxazin-3-one 303761 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [(R)-1-(4-chloro-benzyl)-2-(4-{2-[(2-morpholin-4-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-2-oxo-ethyl]-amide 303762 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [(R)-2-(4-{2-[(3-azepan-1-yl-propylamino)-methyl]-phenyl}-piperazin-1-yl)-1-(4-chloro-benzyl)-2-oxo-ethyl]-amide 303772 6-((1-(2-(2-methylquinolin-5-yloxy)ethyl)piperidin-4-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one 303773 3-[1-(2-Bromo-phenyl)-meth-(E)-ylidene]-1,2,3,9-tetrahydro-pyrrolo[2,1-b]quinazoline 303774 3-[1-(2-Fluoro-phenyl)-meth-(E)-ylidene]-1,2,3,9-tetrahydro-pyrrolo[2,1-b]quinazoline 303775 8-[1-(2-Bromo-phenyl)-meth-(E)-ylidene]-2,3-dimethyl-7,8-dihydro-6H-furo[2,3-d]pyrrolo[1,2-a]pyrimidin-(4Z)-ylideneamine 303776 4-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-2-pyridin-4-yl-but-3-yn-2-ol 303777 4-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-2-[4-(2H-imidazol-1-yl)-phenyl]-but-3-yn-2-ol 303783 9-[1-(2-Bromo-phenyl)-meth-(E)-ylidene]-8,9-dihydro-7H-pyrido[2,3-d]pyrrolo[1,2-a]pyrimidin-(5Z)-ylideneamine 303787 6-{1-[2-(Quinolin-5-yloxy)-ethyl]-piperidin-4-yloxy}-4H-benzo[1,4]oxazin-3-one 303788 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [(R)-1-(4-chloro-benzyl)-2-(4-{2-[(3-imidazol-1-yl-propylamino)-methyl]-phenyl}-piperazin-1-yl)-2-oxo-ethyl]-amide 303789 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-oxo-2-[4-(2-{[3-(2-oxo-pyrrolidin-1-yl)-propylamino]-methyl}-phenyl)-piperazin-1-yl]-ethyl}-amide 303791 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid ((R)-1-(4-chloro-benzyl)-2-oxo-2-{4-[2-(pyridin-4-ylaminomethyl)-phenyl]-piperazin-1-yl}-ethyl)-amide 303792 1-{[2-(4-{(R)-3-(4-Chloro-phenyl)-2-[((R)-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl)-amino]-propionyl}-piperazin-1-yl)-benzylamino]-methyl}-piperidine-4-carboxylic acid ethyl ester 303797 1-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-3-isopropyl-4-methyl-pent-1-yn-3-ol 303798 1-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-3-ethyl-pent-1-yn-3-ol 303800 4-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-2-benzo[b]thiophen-3-yl-but-3-yn-2-ol 303805 3-[1-(2-Trifluoromethyl-phenyl)-meth-(E)-ylidene]-1,2,3,9-tetrahydro-pyrrolo[2,1-b]quinazoline 303806 3-[1-(2-Ethyl-phenyl)-meth-(E)-ylidene]-1,2,3,9-tetrahydro-pyrrolo[2,1-b]quinazoline 303807 3-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-1-benzo[b]thiophen-3-yl-prop-2-yn-1-ol 303810 6-{1-[2-(Quinolin-5-yloxy)-ethyl]-pyrrolidin-3-ylmethoxy}-4H-benzo[1,4]oxazin-3-one 303813 {[2-(4-{(R)-3-(4-Chloro-phenyl)-2-[((R)-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl)-amino]-propionyl}-piperazin-1-yl)-benzyl]-methyl-amino}-acetic acid ethyl ester 303814 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [(R)-2-[4-(2-{[benzyl-(2-dimethylamino-ethyl)-amino]-methyl}-phenyl)-piperazin-1-yl]-1-(4-chloro-benzyl)-2-oxo-ethyl]-amide 303820 {3-Chloro-4-[1,2-dihydro-9H-pyrrolo[2,1-b]quinazolin-(3E)-ylidenemethyl]-phenyl}-dimethyl-amine 303833 4-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-2-phenyl-but-3-yn-2-ol 303834 3-[1-(2-Ethoxy-phenyl)-meth-(E)-ylidene]-1,2,3,9-tetrahydro-pyrrolo[2,1-b]quinazoline 303835 4-[3-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-1-hydroxy-1-methyl-prop-2-ynyl]-phenol 303837 6-{1-[2-(Quinolin-5-yloxy)-ethyl]-piperidin-3-ylmethoxy}-4H-benzo[1,4]oxazin-3-one 303839 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [(R)-1-(4-chloro-benzyl)-2-(4-{2-[1-(3-isobutoxy-propylamino)-ethyl]-phenyl}-piperazin-1-yl)-2-oxo-ethyl]-amide 303840 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [(R)-1-(4-chloro-benzyl)-2-(4-{2-[1-(2-morpholin-4-yl-ethylamino)-ethyl]-phenyl}-piperazin-1-yl)-2-oxo-ethyl]-amide 303843 3-[1-Biphenyl-2-yl-meth-(E)-ylidene]-1,2,3,9-tetrahydro-pyrrolo[2,1-b]quinazoline 303845 3-[1-(2,4-Dichloro-phenyl)-meth-(E)-ylidene]-1,2,3,9-tetrahydro-pyrrolo[2,1-b]quinazoline 303846 3-[1-(3,4-Dichloro-phenyl)-meth-(E)-ylidene]-1,2,3,9-tetrahydro-pyrrolo[2,1-b]quinazoline 303860 6-{1-[2-(2,2-Dimethyl-2,7a-dihydro-benzofuran-3-yloxy)-ethyl]-piperidin-4-yloxy}-4H-benzo[1,4]oxazin-3-one 303862 3-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-1-phenyl-prop-2-yn-1-ol 303863 4-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-2-(2-fluoro-3-trifluoromethyl-phenyl)-but-3-yn-2-ol 303864 1-[3-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-1-hydroxy-prop-2-ynyl]-cyclopentanol 303865 6-{4-[2-(Quinolin-5-yloxy)-ethyl]-piperazin-1-ylmethyl}-4H-benzo[1,4]oxazin-3-one 303870 4-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-1,1,1-trifluoro-2-phenyl-but-3-yn-2-ol 303871 3-[1-(2-Trifluoromethoxy-phenyl)-meth-(E)-ylidene]-1,2,3,9-tetrahydro-pyrrolo[2,1-b]quinazoline 303872 3-[1-(2-Chloro-phenyl)-meth-(E)-ylidene]-1-ethyl-1,2,3,9-tetrahydro-pyrrolo[2,1-b]quinazoline 303873 3-[1-(2-Bromo-phenyl)-meth-(E)-ylidene]-1-butyl-1,2,3,9-tetrahydro-pyrrolo[2,1-b]quinazoline 303883 (+/-)-tert-butyl 2-({[4-(diethylamino)phenyl]amino}carbonyl)-1,2,3,4-tetrahydronaphthalen-2-ylcarbamate 303889 (+/-)-1,2,3,4-tetrahydro-naphthalene-2-carboxylic acid (4-diethylamino-phenyl)-amide 303922 6-{1-[2-(Isoquinolin-1-yloxy)-ethyl]-piperidin-4-yloxy}-4H-benzo[1,4]oxazin-3-one 303946 6-{1-[2-(Quinolin-4-yloxy)-ethyl]-piperidin-4-yloxy}-4H-benzo[1,4]oxazin-3-one 303951 (+/-)isobutyl 2-((4-(diethylamino)phenyl)carbamoyl)-8-methoxy-1,2,3,4-tetrahydronaphthalen-2-yl(methyl)carbamate 303956 (R)-N-((R)-3-(4-chlorophenyl)-1-oxo-1-(4-(2-(1-(piperidin-3-ylamino)ethyl)phenyl)piperazin-1-yl)propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 303957 1-Amino-indan-1-carboxylic acid [(R)-1-(4-chloro-benzyl)-2-oxo-2-(4-{2-[1-(piperidin-3-ylamino)-ethyl]-phenyl}-piperazin-1-yl)-ethyl]-amide 303958 2-Amino-indan-2-carboxylic acid [(R)-1-(4-chloro-benzyl)-2-oxo-2-(4-{2-[1-(piperidin-3-ylamino)-ethyl]-phenyl}-piperazin-1-yl)-ethyl]-amide 303959 2-Amino-N-[1-((R)-4-chloro-benzyl)-2-oxo-2-(4-{2-[1-(piperidin-3-ylamino)-ethyl]-phenyl}-piperazin-1-yl)-ethyl]-2-indan-1-yl-acetamide 303960 2-Amino-1,2,3,4-tetrahydro-naphthalene-2-carboxylic acid [(R)-1-(4-chloro-benzyl)-2-oxo-2-(4-{2-[1-(piperidin-3-ylamino)-ethyl]-phenyl}-piperazin-1-yl)-ethyl]-amide 303961 N-[(R)-1-(4-Chloro-benzyl)-2-oxo-2-(4-{2-[1-(piperidin-3-ylamino)-ethyl]-phenyl}-piperazin-1-yl)-ethyl]-2-(1,2,3,4-tetrahydro-isoquinolin-1-yl)-acetamide 303966 2-Amino-N-[1-((R)-4-chloro-benzyl)-2-oxo-2-(4-{2-[1-(piperidin-3-ylamino)-ethyl]-phenyl}-piperazin-1-yl)-ethyl]-3-phenyl-propionamide 303971 2-Amino-N-[1-((R)-4-chloro-benzyl)-2-oxo-2-(4-{2-[1-(piperidin-3-ylamino)-ethyl]-phenyl}-piperazin-1-yl)-ethyl]-3-pyridin-2-yl-propionamide 303978 6-{1-[2-(Quinolin-8-yloxy)-ethyl]-piperidin-4-yloxy}-4H-benzo[1,4]oxazin-3-one 303989 2-Amino-N-[1-((R)-4-chloro-benzyl)-2-oxo-2-(4-{2-[1-(piperidin-3-ylamino)-ethyl]-phenyl}-piperazin-1-yl)-ethyl]-3-pyridin-3-yl-propionamide 303990 2-Amino-N-[1-((R)-4-chloro-benzyl)-2-oxo-2-(4-{2-[1-(piperidin-3-ylamino)-ethyl]-phenyl}-piperazin-1-yl)-ethyl]-2-phenyl-acetamide 303991 N-[(R)-1-(4-Chloro-benzyl)-2-oxo-2-(4-{2-[1-(piperidin-3-ylamino)-ethyl]-phenyl}-piperazin-1-yl)-ethyl]-3-phenyl-propionamide 303992 N-[(R)-1-(4-Chloro-benzyl)-2-oxo-2-(4-{2-[1-(piperidin-3-ylamino)-ethyl]-phenyl}-piperazin-1-yl)-ethyl]-2-phenyl-acetamide 303993 Quinoline-3-carboxylic acid [(R)-1-(4-chloro-benzyl)-2-oxo-2-(4-{2-[1-(piperidin-3-ylamino)-ethyl]-phenyl}-piperazin-1-yl)-ethyl]-amide 304010 (+/-)-isobutyl 2-({[4-(diethylamino)phenyl]amino}carbonyl)-1,2,3,4-tetrahydronaphthalen-2-ylcarbamate 304146 1-Benzyl-2-(2-morpholin-4-yl-ethoxy)-1H-benzoimidazole-5-sulfonic acid 4-fluoro-benzylamide 304148 1-Benzyl-2-ethoxy-1H-benzoimidazole-5-sulfonic acid 4-fluoro-benzylamide 304162 1-Benzyl-2-ethylsulfanyl-1H-benzoimidazole-5-sulfonic acid 3-methoxy-benzylamide 304170 1-Benzyl-2-methylsulfanyl-1H-benzoimidazole-5-sulfonic acid 4-fluoro-benzylamide 304182 1-Benzyl-2-ethylsulfanyl-1H-benzoimidazole-5-sulfonic acid 4-methoxy-benzylamide 304183 1-Benzyl-2-(2-benzylamino-ethylsulfanyl)-1H-benzoimidazole-5-sulfonic acid 4-fluoro-benzylamide 304206 1-Benzyl-2-ethylsulfanyl-1H-benzoimidazole-5-sulfonic acid 4-nitro-benzylamide 304207 1-Benzyl-2-(pyridin-2-ylmethylsulfanyl)-1H-benzoimidazole-5-sulfonic acid 4-fluoro-benzylamide 304218 1-Benzyl-2-ethylsulfanyl-1H-benzoimidazole-5-sulfonic acid 4-chloro-benzylamide 304240 1-Benzyl-2-ethylsulfanyl-1H-benzoimidazole-5-sulfonic acid 4-fluoro-benzylamide 304246 [(R)-8-(2,6-Dimethoxy-phenyl)-chroman-3-yl]-dipropyl-amine 304247 (R)-8-(2,6-dimethoxyphenyl)-N,N-dimethylchroman-3-amine 304255 2-Ethoxy-1-thiophen-3-ylmethyl-1H-benzoimidazole-5-sulfonic acid 4-fluoro-benzylamide 304272 [(S)-6-(2,6-Dimethoxy-phenyl)-chroman-3-yl]-dimethyl-amine 304273 (S)-6-(2,6-dimethylphenyl)-N,N-dimethylchroman-3-amine 304281 1-Benzyl-2-(2-morpholin-4-yl-ethylsulfanyl)-1H-benzoimidazole-5-sulfonic acid 4-fluoro-benzylamide 304312 1-Benzyl-2-(2-hydroxy-ethylsulfanyl)-1H-benzoimidazole-5-sulfonic acid 4-fluoro-benzylamide 304313 2-Ethoxy-1-(2-morpholin-4-yl-ethyl)-1H-benzoimidazole-5-sulfonic acid 4-fluoro-benzylamide 304333 [(S)-6-(1-Methoxy-naphthalen-2-yl)-chroman-3-yl]-dimethyl-amine 304347 [1-Benzyl-5-(4-fluoro-benzylsulfamoyl)-1H-benzoimidazol-2-ylsulfanyl]-acetic acid ethyl ester 304397 1-(3-Chloro-benzyl)-2-ethoxy-1H-benzoimidazole-5-sulfonic acid 4-fluoro-benzylamide 304426 1-Benzyl-2-isopropyl-1H-benzoimidazole-5-sulfonic acid 4-fluoro-benzylamide 304427 1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benzoimidazole-5-sulfonic acid 3,4-difluoro-benzylamide 304428 1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benzoimidazole-5-sulfonic acid 3-fluoro-4-trifluoromethyl-benzylamide 304445 1-Benzyl-2-{2-[3-(2-fluoro-phenyl)-ureido]-ethyl}-1H-benzoimidazole-5-sulfonic acid 4-fluoro-benzylamide 304454 1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benzoimidazole-5-sulfonic acid 4-chloro-benzylamide 304460 2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid (1-butyl-piperidin-4-ylmethyl)-amide 304461 1-Benzyl-2-(pyridin-4-ylmethylsulfanyl)-1H-benzoimidazole-5-sulfonic acid 4-fluoro-benzylamide 304468 1-Benzyl-2-[2-(3-isopropyl-ureido)-ethyl]-1H-benzoimidazole-5-sulfonic acid 4-fluoro-benzylamide 304484 1-Benzyl-2-(2-pyridin-2-yl-ethylsulfanyl)-1H-benzoimidazole-5-sulfonic acid 4-fluoro-benzylamide 304490 1-Benzyl-2-[2-(3-ethyl-ureido)-ethyl]-1H-benzoimidazole-5-sulfonic acid 4-fluoro-benzylamide 304491 1-Benzyl-2-{2-[3-(2-chloro-phenyl)-ureido]-ethyl}-1H-benzoimidazole-5-sulfonic acid 4-fluoro-benzylamide 304508 N-(4-fluorobenzyl)-1-benzyl-2-(2-(pyridin-3-yl)ethylthio)-1H-benzo[d]imidazole-5-sulfonamide 304513 1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benzoimidazole-5-sulfonic acid 4-fluoro-benzylamide 304516 1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benzoimidazole-5-sulfonic acid benzylamide 304539 1-Benzyl-2-[3-(3-tert-butyl-ureido)-propyl]-1H-benzoimidazole-5-sulfonic acid 4-fluoro-benzylamide 304541 1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benzoimidazole-5-sulfonic acid 2-fluoro-benzylamide 304558 4-[1-Benzyl-5-(4-fluoro-benzylsulfamoyl)-1H-benzoimidazol-2-yl]-N-tert-butyl-butyramide 304583 1-[4-(4-Bromo-benzyl)-[1,4'']bipiperidinyl-1''-yl]-2-(2-methoxy-phenyl)-ethanone 304593 1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benzoimidazole-5-sulfonic acid 2,4-dichloro-benzylamide 304610 {2-[1-Benzyl-5-(4-fluoro-benzylsulfamoyl)-1H-benzoimidazol-2-yl]-ethyl}-carbamic acid tert-butyl ester 304618 1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benzoimidazole-5-sulfonic acid 4-methoxy-benzylamide 304633 N-{2-[1-Benzyl-5-(4-fluoro-benzylsulfamoyl)-1H-benzoimidazol-2-yl]-ethyl}-3,3-dimethyl-butyramide 304653 1-Benzyl-2-cyclopropyl-1H-benzoimidazole-5-sulfonic acid 4-fluoro-benzylamide 304898 (S)-4-Methyl-piperazine-2-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide 305031 N-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-N-methyl-2-(4-sulfamoyl-phenyl)-acetamide 305041 N-allyl-N-(1-(3,3-diphenylpropyl)piperidin-4-yl)-2-(4-(methylsulfonyl)phenyl)acetamide 305042 Thiophene-2-carboxylic acid [1-(3,3-diphenyl-propyl)-piperidin-4-yl]-methyl-amide 305046 2-(2-Chloro-phenyl)-N-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-N-methyl-acetamide 305047 2-(4-Benzyloxy-phenyl)-N-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-N-methyl-acetamide 305048 2-(3,4-Difluoro-phenyl)-N-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-N-methyl-acetamide 305058 2-(4-Dimethylsulfamoyl-phenyl)-N-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-N-ethyl-acetamide 305059 2-(4-Dimethylsulfamoyl-phenyl)-N-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-N-methyl-acetamide 305063 2-(3-Chloro-phenyl)-N-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-N-methyl-acetamide 305064 2-Biphenyl-4-yl-N-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-N-methyl-acetamide 305065 N-Allyl-N-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-2-(4-nitro-phenyl)-acetamide 305066 Furan-2-carboxylic acid [1-(3,3-diphenyl-propyl)-piperidin-4-yl]-methyl-amide 305072 N-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-N-ethyl-2-(4-methanesulfonyl-phenyl)-acetamide 305079 4-({[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-methyl-carbamoyl}-methyl)-benzoic acid methyl ester 305080 3-(3-Cyano-phenyl)-1-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-1-methyl-urea 305081 2-(4-Chloro-phenyl)-N-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-N-methyl-acetamide 305082 N-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-N-methyl-2-(4-trifluoromethyl-phenyl)-acetamide 305086 N-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-3,3,N-trimethyl-butyramide 305087 N-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-2-(4-methoxy-phenyl)-N-methyl-acetamide 305088 N-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-N-ethyl-2-(4-nitro-phenyl)-acetamide 305096 N-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-2-(4-hydroxy-phenyl)-N-methyl-acetamide 305097 1-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-1-methyl-3-m-tolyl-urea 305098 2-(3,4-Dichloro-phenyl)-N-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-N-methyl-acetamide 305099 N-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-N-methyl-2-(4-trifluoromethoxy-phenyl)-acetamide 305104 N-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-N-methyl-2-phenyl-acetamide 305105 2-(3,4-Dimethoxy-phenyl)-N-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-N-methyl-acetamide 305106 N-Cyclopropyl-N-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-2-(4-sulfamoyl-phenyl)-acetamide 305107 1-Oxo-1,3-dihydro-isoindole-2-carboxylic acid [1-(3,3-diphenyl-propyl)-piperidin-4-yl]-methyl-amide 305112 N-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-N-methyl-2-(4-nitro-phenyl)-acetamide 305113 1-Allyl-1-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-3-phenyl-urea 305114 2-(2,4-Dichloro-phenyl)-N-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-N-methyl-acetamide 305118 N-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-N-methyl-2-oxo-2-phenyl-acetamide 305119 2-(3,5-Dimethoxy-phenyl)-N-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-N-methyl-acetamide 305121 N-Cyclopropyl-N-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-2-(4-methanesulfonyl-phenyl)-acetamide 305130 N-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-N-ethyl-2-(4-trifluoromethoxy-phenyl)-acetamide 305131 3-(3,4-Dichloro-phenyl)-1-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-1-methyl-urea 305132 N-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-N-methyl-isonicotinamide 305133 N-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-2-(2-fluoro-phenyl)-N-methyl-acetamide 305140 N-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-N-methyl-2-(2,4,5-trimethoxy-phenyl)-acetamide 305141 2-(4-Acetylamino-phenyl)-N-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-N-methyl-acetamide 305142 N-Cyclopropyl-N-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-2-(4-nitro-phenyl)-acetamide 305148 2-(4-Cyano-phenyl)-N-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-N-ethyl-acetamide 305150 N-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-4-fluoro-N-methyl-benzamide 305151 N-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-2-(3-fluoro-phenyl)-N-methyl-acetamide 305158 1-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-3-(4-fluoro-phenyl)-1-methyl-urea 305159 N-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-N-methyl-2-phenyl-propionamide 305160 2-(4-Cyano-phenyl)-N-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-N-methyl-acetamide 305161 N-Allyl-N-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-2-(4-trifluoromethoxy-phenyl)-acetamide 305168 2-(4-Bromo-phenyl)-N-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-N-methyl-acetamide 305169 N-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-N-ethyl-2-(4-sulfamoyl-phenyl)-acetamide 305170 N-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-N-methyl-3-nitro-benzamide 305171 N-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-2-(4-fluoro-phenyl)-N-methyl-acetamide 305178 1-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-1-ethyl-3-(4-methanesulfonyl-benzyl)-urea 305213 1-Allyl-1-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-3-(3-methyl-benzyl)-urea 305218 N-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-2-(3-methoxy-phenyl)-N-methyl-acetamide 305219 N-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-N-methyl-2-(4-methylsulfanyl-phenyl)-acetamide 305227 3-Cyclohexyl-1-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-1-methyl-urea 305229 1-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-1-ethyl-3-p-tolyl-urea 305234 Cyclobutanecarboxylic acid [1-(3,3-diphenyl-propyl)-piperidin-4-yl]-methyl-amide 305235 N-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-3,N-dimethyl-butyramide 305238 1-Allyl-1-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-3-(4-methoxy-benzyl)-urea 305254 3-Benzyl-1-[1-(3,3-diphenyl-propyl)-piperidin-4-yl]-1-methyl-urea 305263 1-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-1-ethyl-3-(3-methyl-benzyl)-urea 305275 3-benzyl-1-(1-(3,3-diphenylpropyl)piperidin-4-yl)-1-ethylurea 305285 1-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-1-ethyl-3-(4-methoxy-benzyl)-urea 305301 1-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-1-ethyl-3-(1-phenyl-ethyl)-urea 305394 (S)-1-Cyclopropylmethyl-5-(3,4-dichloro-phenyl)-5-[2-(3-morpholin-4-yl-azetidin-1-yl)-ethyl]-piperidin-2-one 305395 (S)-1-Cyclopropylmethyl-5-(3,4-dichloro-phenyl)-5-{2-[3-(4-ethoxy-piperidin-1-yl)-azetidin-1-yl]-ethyl}-piperidin-2-one 305397 (S)-5-{2-[3-(4-Amino-piperidin-1-yl)-azetidin-1-yl]-ethyl}-1-cyclopropylmethyl-5-(3,4-dichloro-phenyl)-piperidin-2-one 305400 4-(1-{2-[(S)-1-Cyclopropylmethyl-3-(3,4-dichloro-phenyl)-6-oxo-piperidin-3-yl]-ethyl}-azetidin-3-yl)-piperazine-1-sulfonic acid dimethylamide 305403 (S)-1-Cyclopropylmethyl-5-(3,4-dichloro-phenyl)-5-{2-[3-(4-methanesulfonyl-piperazin-1-yl)-azetidin-1-yl]-ethyl}-piperidin-2-one 305408 4-(1-{2-[(S)-1-Cyclopropylmethyl-3-(3,4-dichloro-phenyl)-6-oxo-piperidin-3-yl]-ethyl}-azetidin-3-yl)-piperazine-1-sulfonic acid amide 305414 (S)-1-(1-Cyclopropyl-cyclopentyl)-5-(3,4-dichloro-phenyl)-5-[2-(3-morpholin-4-yl-azetidin-1-yl)-ethyl]-piperidin-2-one 305453 (S)-5-(3,4-Dichloro-phenyl)-1-(4,4-difluoro-cyclohexylmethyl)-5-[2-(3-morpholin-4-yl-azetidin-1-yl)-ethyl]-piperidin-2-one 305458 (S)-1-Cyclohexylmethyl-5-(3,4-dichloro-phenyl)-5-[2-(3-morpholin-4-yl-azetidin-1-yl)-ethyl]-piperidin-2-one 305462 (S)-5-(3,4-Dichloro-phenyl)-1-(4,4-difluoro-cyclohexylmethyl)-5-{2-[3-(4-methanesulfonyl-piperazin-1-yl)-azetidin-1-yl]-ethyl}-piperidin-2-one 305524 (S)-5-(3,4-Dichloro-phenyl)-1-(4,4-difluoro-cyclohexylmethyl)-5-{2-[3-(4-oxo-piperidin-1-yl)-azetidin-1-yl]-ethyl}-piperidin-2-one 305548 (S)-5-(3,4-Dichloro-phenyl)-1-(4,4-difluoro-cyclohexylmethyl)-5-{2-[3-(4-fluoro-piperidin-1-yl)-azetidin-1-yl]-ethyl}-piperidin-2-one 305581 (S)-5-(3,4-Dichloro-phenyl)-1-(4,4-difluoro-cyclohexylmethyl)-5-{2-[3-(4-hydroxy-piperidin-1-yl)-azetidin-1-yl]-ethyl}-piperidin-2-one 305588 (S)-1-Cyclopropylmethyl-5-(3,4-dichloro-phenyl)-5-{2-[3-(4-fluoro-piperidin-1-yl)-azetidin-1-yl]-ethyl}-piperidin-2-one 305589 (S)-1-(2-Cyclopropyl-ethyl)-5-(3,4-dichloro-phenyl)-5-{2-[3-(4-fluoro-piperidin-1-yl)-azetidin-1-yl]-ethyl}-piperidin-2-one 305603 N-{3-[3-(2-Benzyloxy-5-chloro-phenyl)-thiophen-2-yl]-phenyl}-2-phenyl-acetamide 305607 6-[3-(2-Benzyloxy-5-chloro-phenyl)-thiophen-2-yl]-pyridine-2-carboxylic acid 305623 2-{5-[3-(2-Benzyloxy-5-chloro-phenyl)-thiophen-2-yl]-pyridin-3-yl}-1,1,1,3,3,3-hexafluoro-propan-2-ol 305625 N-{3-[3-(2-Benzyloxy-5-chloro-phenyl)-thiophen-2-yl]-phenyl}-C-phenyl-methanesulfonamide 305636 1-{5-[3-(2-Benzyloxy-5-chloro-phenyl)-thiophen-2-yl]-pyridin-3-yl}-2,2,2-trifluoro-ethanol 305637 {4-[2-(4-Fluoro-phenyl)-6-methyl-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-(3-trifluoromethyl-phenyl)-amine 305639 (S)-5-{2-[3-(4-Amino-piperidin-1-yl)-azetidin-1-yl]-ethyl}-5-(3,4-dichloro-phenyl)-1-(4,4-difluoro-cyclohexylmethyl)-piperidin-2-one 305648 (S)-1-(1-Cyclopropyl-cyclopentyl)-5-(3,4-dichloro-phenyl)-5-{2-[3-(4-fluoro-piperidin-1-yl)-azetidin-1-yl]-ethyl}-piperidin-2-one 305651 (3,4-Difluoro-phenyl)-{4-[2-(4-fluoro-phenyl)-6-methyl-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-amine 305656 1-{5-[3-(2-Benzyloxy-5-chloro-phenyl)-thiophen-2-yl]-pyridin-3-yl}-2,2,2-trifluoro-ethane-1,1-diol 305664 (2,3-Dihydro-benzo[1,4]dioxin-6-yl)-{4-[2-(4-fluoro-phenyl)-6-methyl-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-amine 305668 {3-[3-(2-Benzyloxy-5-chloro-phenyl)-thiophen-2-yl]-phenyl}-acetic acid 305670 {5-[3-(2-Benzyloxy-5-chloro-phenyl)-thiophen-2-yl]-pyridin-3-yl}-hydroxy-acetonitrile 305673 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-oxo-2-[4-((1S,2S)-2-[1,2,4]triazol-1-yl-cyclohexyl)-piperazin-1-yl]-ethyl}-amide 305674 (4-Chloro-3-trifluoromethyl-phenyl)-{4-[2-(4-fluoro-phenyl)-6-methyl-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-amine 305683 3-(3-(2-(benzyloxy)-5-chlorophenyl)thiophen-2-yl)benzoic acid 305687 [4-(2-Cyclopropyl-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-phenyl-amine 305691 3-[3-(2-Benzyloxy-5-chloro-phenyl)-thiophen-2-yl]-N-(1-pyridin-3-yl-ethyl)-benzamide 305693 [4-(2-Cyclopropyl-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-(3,4-difluoro-phenyl)-amine 305696 5-[3-(2-Benzyloxy-5-chloro-phenyl)-thiophen-2-yl]-nicotinic acid 305702 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-oxo-2-[4-(1-[1,2,4]triazol-1-ylmethyl-cyclopentyl)-piperazin-1-yl]-ethyl}-amide 305708 2-(2-{4-[1-(2-ethoxyethyl)-1H-indol-3-yl]piperidin-1-yl}ethoxy)-4-methoxybenzoic acid 305709 N-[1-(3-Hydroxy-phenyl)-2-pyrrolidin-1-yl-ethyl]-N-methyl-2-(4-trifluoromethyl-phenyl)-acetamide 305715 N-[1-(3-Methoxy-phenyl)-2-pyrrolidin-1-yl-ethyl]-N-methyl-2-(4-trifluoromethyl-phenyl)-acetamide 305734 2-{2-[4-(1-Butyl-1H-indol-3-yl)-piperidin-1-yl]-ethoxy}-4-methoxy-benzoic acid 305745 [3-(1-{Methyl-[2-(4-trifluoromethyl-phenyl)-acetyl]-amino}-2-pyrrolidin-1-yl-ethyl)-phenoxy]-acetic acid tert-butyl ester 305792 4-(Benzhydryl-amino)-N,N-bis-(3-dimethylamino-propyl)-3-nitro-benzenesulfonamide 305804 {4-[5-(2-Methoxy-ethoxy)-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-(3-methoxy-phenyl)-amine 305847 N-[(S)-1-(3-Amino-phenyl)-2-pyrrolidin-1-yl-ethyl]-N-methyl-2-(4-trifluoromethyl-phenyl)-acetamide 305856 4-Chloro-2-(2-{4-[1-(5-chloro-thiophen-2-ylmethyl)-1H-indol-3-yl]-piperidin-1-yl}-ethoxy)-benzoic acid 305858 2-(2-(4-(1-((5-chlorothiophen-2-yl)methyl)-1H-indol-3-yl)piperidin-1-yl)ethoxy)benzoic acid 305864 5-{4-[1-(5-Chloro-thiophen-2-ylmethyl)-1H-indol-3-yl]-piperidin-1-ylmethyl}-2-methoxy-benzoic acid 305871 4-{4-[1-(2-ethoxyethyl)-1H-indol-3-yl]piperidin-1-ylmethyl}benzoic acid 305877 3-[4-(1-Butyl-1H-indol-3-yl)-piperidin-1-ylmethyl]-benzoic acid 305892 2-{2-[4-(1-Furan-3-ylmethyl-1H-indol-3-yl)-piperidin-1-yl]-ethoxy}-4-methoxy-benzoic acid 305893 [3-(1-{Methyl-[2-(4-trifluoromethyl-phenyl)-acetyl]-amino}-2-pyrrolidin-1-yl-ethyl)-phenoxy]-acetic acid 305895 3-[4-(1-Furan-3-ylmethyl-1H-indol-3-yl)-piperidin-1-ylmethyl]-benzoic acid 305897 N-[(S)-1-(3-Methanesulfonylamino-phenyl)-2-pyrrolidin-1-yl-ethyl]-N-methyl-2-(4-trifluoromethyl-phenyl)-acetamide 305905 2-(2-{4-[1-(5-Chloro-thiophen-2-ylmethyl)-1H-indol-3-yl]-piperidin-1-yl}-ethoxy)-4-methoxy-benzoic acid 305906 2-(2-{4-[1-(2-Ethoxy-ethyl)-1H-indol-3-yl]-piperidin-1-yl}-ethoxy)-benzaldehyde 305907 3-{4-[1-(5-chlorothiophen-2-ylmethyl)-1H-indol-3-yl]-piperidin-1-ylmethyl}benzoic acid 305911 N-Methyl-N-[(S)-1-(3-nitro-phenyl)-2-pyrrolidin-1-yl-ethyl]-2-(4-trifluoromethyl-phenyl)-acetamide 305915 N-[(S)-1-(3-aminosulfonylamino-phenyl)-2-pyrrolidin-1-yl-ethyl]-N-methyl-2-(4-trifluoromethyl-phenyl)-acetamide 305919 2-(2-{4-[1-(2-ethoxyethyl)-1H-indol-3-yl]piperidin-1-yl}ethoxy)benzoic acid 305926 5-{4-[1-(2-ethoxyethyl)-1H-indol-3-yl]piperidin-1-ylmethyl}-2-methoxybenzoic acid 305930 N-[3-((S)-1-{Methyl-[2-(4-trifluoromethyl-phenyl)-acetyl]-amino}-2-pyrrolidin-1-yl-ethyl)-phenyl]-succinamic acid 305934 2-{2-[4-(1-butyl-1H-indol-3-yl)piperidin-1-yl]ethoxy}-benzoic acid 305938 2-{2-[4-(1-Butyl-1H-indol-3-yl)-piperidin-1-yl]-ethoxy}-4-chloro-benzoic acid 305939 5-[4-(1-Butyl-1H-indol-3-yl)-piperidin-1-ylmethyl]-2-methoxy-benzoic acid 305943 {Carboxymethyl-[3-((S)-1-{methyl-[2-(4-trifluoromethyl-phenyl)-acetyl]-amino}-2-pyrrolidin-1-yl-ethyl)-phenyl]-amino}-acetic acid 305946 (+/-)-3-difluoromethyl-7-nitro-1,2,3,4-tetrahydroisoquinoline 305953 4-Chloro-2-{2-[4-(1-furan-3-ylmethyl-1H-indol-3-yl)-piperidin-1-yl]-ethoxy}-benzoic acid 305954 2-{2-[4-(1-Furan-3-ylmethyl-1H-indol-3-yl)-piperidin-1-yl]-ethoxy}-benzoic acid 305955 5-[4-(1-Furan-3-ylmethyl-1H-indol-3-yl)-piperidin-1-ylmethyl]-2-methoxy-benzoic acid 306078 Phosphoric acid mono-[(R)-3-[4-(4-methoxy-quinolin-2-ylmethoxy)-phenyl]-2-((Z)-octadec-9-enoylamino)-propyl] ester 306079 Phosphoric acid mono-[3-[4-(4-methoxy-quinolin-2-ylmethoxy)-phenyl]-2-((Z)-(S)-octadec-9-enoylamino)-propyl] ester 306117 Phosphoric acid mono-{(R)-2-((Z)-octadec-9-enoylamino)-3-[4-(pyridin-3-ylmethoxy)-phenyl]-propyl} ester 306128 Phosphoric acid mono-{2-((Z)-(S)-octadec-9-enoylamino)-3-[4-(pyridin-3-ylmethoxy)-phenyl]-propyl} ester 306140 Phosphoric acid mono-{(R)-2-((Z)-octadec-9-enoylamino)-3-[4-(pyridin-4-ylmethoxy)-phenyl]-propyl} ester 306155 Phosphoric acid mono-{2-((Z)-(S)-octadec-9-enoylamino)-3-[4-(pyridin-4-ylmethoxy)-phenyl]-propyl} ester 306156 Phosphoric acid mono-[(R)-3-[4-(6-methoxy-pyridin-2-ylmethoxy)-phenyl]-2-((Z)-octadec-9-enoylamino)-propyl] ester 306157 Phosphoric acid mono-[3-[4-(6-methoxy-pyridin-2-ylmethoxy)-phenyl]-2-((Z)-(S)-octadec-9-enoylamino)-propyl] ester 306170 Phosphoric acid mono-[(R)-3-[4-(4-methoxy-pyridin-2-ylmethoxy)-phenyl]-2-((Z)-octadec-9-enoylamino)-propyl] ester 306171 Phosphoric acid mono-[3-[4-(4-ethoxy-pyridin-2-ylmethoxy)-phenyl]-2-((Z)-(R)-octadec-9-enoylamino)-propyl] ester 306172 Phosphoric acid mono-((R)-2-((Z)-octadec-9-enoylamino)-3-{4-[4-(2,2,2-trifluoro-ethoxy)-pyridin-2-ylmethoxy]-phenyl}-propyl) ester 306173 Phosphoric acid mono-{2-((Z)-(R)-octadec-9-enoylamino)-3-[4-(4-propoxy-pyridin-2-ylmethoxy)-phenyl]-propyl} ester 306174 Phosphoric acid mono-[(R)-3-{4-[4-(2-methoxy-ethoxy)-pyridin-2-ylmethoxy]-phenyl}-2-((Z)-octadec-9-enoylamino)-propyl] ester 306175 Phosphoric acid mono-[3-[4-(4-methoxy-3,5-dimethyl-pyridin-2-ylmethoxy)-phenyl]-2-((Z)-(R)-octadec-9-enoylamino)-propyl] ester 306176 Phosphoric acid mono-[(S)-3-[4-(4-methoxy-3,5-dimethyl-pyridin-2-ylmethoxy)-phenyl]-2-((Z)-octadec-9-enoylamino)-propyl] ester 306177 Phosphoric acid mono-{2-((Z)-(R)-octadec-9-enoylamino)-3-[4-(quinolin-2-ylmethoxy)-phenyl]-propyl} ester 306247 {(S)-3-Hexadecanoylamino-4-[4-(pyridin-2-ylmethoxy)-phenyl]-butyl}-phosphonic acid 306248 [4-[4-(4-Methoxy-3,5-dimethyl-pyridin-2-ylmethoxy)-phenyl]-3-((Z)-(R)-octadec-9-enoylamino)-butyl]-phosphonic acid 306249 [(S)-4-[4-(4-Methoxy-3,5-dimethyl-pyridin-2-ylmethoxy)-phenyl]-3-((Z)-octadec-9-enoylamino)-butyl]-phosphonic acid 306270 [4-(4-Benzyloxy-phenyl)-1-hydroxy-3-((Z)-(S)-octadec-9-enoylamino)-butyl]-phosphonic acid 306368 (1S,4aR,5S,9aS)-4-[2-((2R,6S)-1,6-Dimethyl-piperidin-2-yl)-ethylidene]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 306391 (S)-6,6,7-Trimethyl-2-((3S,3aR,4R,4aR,9aS)-3-methyl-1-oxo-1,3,3a,4,4a,5,6,7,8,9a-decahydro-naphtho[2,3-c]furan-4-yl)-hexahydro-pyrrolo[1,2-b]isoxazol-7-ium iodide 306448 (3S,3aR,4R,4aS,8aR,9aS)-4-[(E)-2-((2R,6S)-1,6-Dimethyl-piperidin-2-yl)-vinyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 306469 (3S,3aS,4aS,8aR,9aS)-4-[2-((2R,6S)-1,6-Dimethyl-piperidin-2-yl)-eth-(Z)-ylidene]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 306489 2''-Amino-6''-(2-hydroxy-3-methyl-phenyl)-1,2,3,4,5,6-hexahydro-[3,4'']bipyridinyl-3''-carbonitrile 306490 Cyclopropanecarboxylic acid (6-pyridin-3-yl-furo[2,3-d]pyrimidin-4-yl)-amide 306491 Cyclopentanecarboxylic acid (6-phenyl-furo[2,3-d]pyrimidin-4-yl)-amide 306492 6-(4-Methoxy-phenyl)-5-pyridin-3-yl-furo[2,3-d]pyrimidin-4-ylamine 306493 Hexanoic acid [6-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-yl]-amide 306496 2''-Amino-6''-(2-hydroxy-3-methoxy-phenyl)-1,2,3,4,5,6-hexahydro-[3,4'']bipyridinyl-3''-carbonitrile 306497 2-Amino-6-(2-hydroxy-6-pentyloxy-phenyl)-1'',2'',3'',4'',5'',6''-hexahydro-[4,4'']bipyridinyl-3-carbonitrile 306499 2''-Amino-6''-(2-hydroxy-6-methoxy-phenyl)-1,2,3,4,5,6-hexahydro-[3,4'']bipyridinyl-3''-carbonitrile 306505 2''-Amino-6''-(2-ethoxy-6-hydroxy-phenyl)-1,2,3,4,5,6-hexahydro-[3,4'']bipyridinyl-3''-carbonitrile 306506 2-Amino-6-(2-hydroxy-6-isobutoxy-phenyl)-1'',2'',3'',4'',5'',6''-hexahydro-[4,4'']bipyridinyl-3-carbonitrile 306508 2''-Amino-6''-(2-cyclohexylmethoxy-6-hydroxy-phenyl)-1,2,3,4,5,6-hexahydro-[3,4'']bipyridinyl-3''-carbonitrile 306509 2-Cyclopentyl-N-[6-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-yl]-acetamide 306510 Cyclohexanecarboxylic acid [6-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-yl]-amide 306514 2-Amino-4-[1-amino-2-(4-fluoro-phenyl)-ethyl]-6-(2-hydroxy-phenyl)-nicotinonitrile 306515 2-Amino-4-(1-amino-3-phenyl-propyl)-6-(2-hydroxy-phenyl)-nicotinonitrile 306518 N-[3''-Cyano-6''-(2-hydroxy-phenyl)-1,2,3,4,5,6-hexahydro-[3,4'']bipyridinyl-2''-yl]-acetamide 306528 2-Amino-6-(2-hydroxy-6-propoxy-phenyl)-1'',2'',3'',4'',5'',6''-hexahydro-[4,4'']bipyridinyl-3-carbonitrile 306529 Cyclopropanecarboxylic acid (6-phenyl-furo[2,3-d]pyrimidin-4-yl)-amide 306530 Cyclopropanecarboxylic acid [6-(4-chloro-phenyl)-furo[2,3-d]pyrimidin-4-yl]-amide 306531 (3S,3aS,4Z,4aS,8aR,9aS)-3-methyl-4-[2-(1,5,5-trimethylpyrrolidin-2-yl)ethylidene]-dodecahydronaphtho[2,3-c]furan-1-one 306537 2''-Amino-6''-(2-hydroxy-4-methoxy-phenyl)-1,2,3,4,5,6-hexahydro-[3,4'']bipyridinyl-3''-carbonitrile 306540 N-[6-(4-Methoxy-phenyl)-furo[2,3-d]pyrimidin-4-yl]-3-methylsulfanyl-propionamide 306541 N-[6-(4-Methoxy-phenyl)-furo[2,3-d]pyrimidin-4-yl]-isobutyramide 306545 2''-Amino-6''-(2-hydroxy-6-methyl-phenyl)-1,2,3,4,5,6-hexahydro-[3,4'']bipyridinyl-3''-carbonitrile 306546 2-Amino-6-(2-hexyloxy-6-hydroxy-phenyl)-1'',2'',3'',4'',5'',6''-hexahydro-[4,4'']bipyridinyl-3-carbonitrile 306547 (3S,3aR,4aS,8aR,9aS)-3-methyl-4-[2-(1,5,5-trimethylpyrrolidin-2-yl)ethyl]-dodecahydronaphtho[2,3-c]furan-1-one 306548 (3S,3aR,4aS,8aR,9aS)-4-[2-(1-ethyl-5,5-dimethylpyrrolidin-2-yl)ethyl]-3-methyl-dodecahydronaphtho[2,3-c]furan-1-one 306556 2''-Amino-6''-(2-benzyloxy-6-hydroxy-phenyl)-1,2,3,4,5,6-hexahydro-[3,4'']bipyridinyl-3''-carbonitrile 306557 2-Amino-6-(2-hydroxy-phenyl)-1'',2'',3'',4'',5'',6''-hexahydro-[4,4'']bipyridinyl-3-carbonitrile 306563 (3S,3aS,4Z,4aS,9aS)-3-methyl-4-[2-(1,5,5-trimethylpyrrolidin-2-yl)ethylidene]-1H,3H,3aH,4H,4aH,5H,6H,7H,8H,9aH-naphtho[2,3-c]furan-1-one 306566 2''-Amino-5''-fluoro-6''-(2-hydroxy-phenyl)-1,2,3,4,5,6-hexahydro-[3,4'']bipyridinyl-3''-carbonitrile 306567 Pyrrolidine-1-carboxylic acid [6-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-yl]-amide 306572 (3S,3aS,4Z,4aS,9aS)-4-[2-(1-ethyl-5,5-dimethylpyrrolidin-2-yl)ethylidene]-3-methyl-1H,3H,3aH,4H,4aH,5H,6H,7H,8H,9aH-naphtho[2,3-c]furan-1-one 306573 2-Amino-4-(1-amino-2-phenyl-ethyl)-6-(2-hydroxy-phenyl)-nicotinonitrile 306574 2-amino-6-(2-hydroxyphenyl)-4-(piperidin-3-yl)nicotinonitrile 306575 Cyclopropanecarboxylic acid (6-p-tolyl-furo[2,3-d]pyrimidin-4-yl)-amide 306576 Cyclopropanecarboxylic acid [6-(4-fluoro-phenyl)-furo[2,3-d]pyrimidin-4-yl]-amide 306581 2-Amino-6-(2-butoxy-6-hydroxy-phenyl)-1'',2'',3'',4'',5'',6''-hexahydro-[4,4'']bipyridinyl-3-carbonitrile 306584 2''-Amino-6''-(2-amino-6-hydroxy-phenyl)-1,2,3,4,5,6-hexahydro-[3,4'']bipyridinyl-3''-carbonitrile 306585 (3S,3aR,4R,4aS,8aR,9aS)-4-[(S)-1-Hydroxy-2-(1,5,5-trimethyl-pyrrolidin-2-yl)-ethyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one iodide 306588 Cyclopropanecarboxylic acid [6-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-yl]-amide 306589 Cyclopentanecarboxylic acid [6-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-yl]-amide 306593 2''-Amino-6''-(2,6-dihydroxy-phenyl)-1,2,3,4,5,6-hexahydro-[3,4'']bipyridinyl-3''-carbonitrile 306594 2-Amino-6-(2-heptyloxy-6-hydroxy-phenyl)-1'',2'',3'',4'',5'',6''-hexahydro-[4,4'']bipyridinyl-3-carbonitrile 306601 2-Amino-4-[1-amino-2-(4-methoxy-phenyl)-ethyl]-6-(2-hydroxy-phenyl)-nicotinonitrile 306603 2-Amino-6-(2,6-dihydroxy-phenyl)-1'',2'',3'',4'',5'',6''-hexahydro-[4,4'']bipyridinyl-3-carbonitrile 306604 2-Amino-6-(2-ethoxy-6-hydroxy-phenyl)-1'',2'',3'',4'',5'',6''-hexahydro-[4,4'']bipyridinyl-3-carbonitrile 306606 Furan-2-carboxylic acid [6-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-yl]-amide 306610 2-Amino-4-(1-amino-2-methyl-propyl)-6-(2-hydroxy-phenyl)-nicotinonitrile 306611 2-Amino-4-(2-amino-ethyl)-6-(2-hydroxy-phenyl)-nicotinonitrile 306614 2''-Amino-6''-(2-hydroxy-6-isobutoxy-phenyl)-1,2,3,4,5,6-hexahydro-[3,4'']bipyridinyl-3''-carbonitrile 306625 N-(1-Phenyl-ethyl)-N''-(3-phenyl-propyl)-[1,3,5]triazine-2,4,6-triamine 306631 N-(2-Phenoxy-ethyl)-N''-(1-phenyl-ethyl)-[1,3,5]triazine-2,4,6-triamine 306632 N-(2-Phenoxy-ethyl)-N''-((S)-1-phenyl-ethyl)-pyridine-3,5-diamine 306639 N-[2-(4-Fluoro-phenoxy)-ethyl]-N''-((S)-1-phenyl-ethyl)-pyridine-3,5-diamine 306650 2''-Amino-6''-(2-heptyloxy-6-hydroxy-phenyl)-1,2,3,4,5,6-hexahydro-[3,4'']bipyridinyl-3''-carbonitrile 306651 2-Amino-6-(2-benzyloxy-6-hydroxy-phenyl)-1'',2'',3'',4'',5'',6''-hexahydro-[4,4'']bipyridinyl-3-carbonitrile 306655 2-(3-(6-methylpyridin-2-yl)-1H-pyrazol-4-yl)-1,5-naphthyridine 306658 2-Amino-4-(2-amino-propyl)-6-(2-hydroxy-phenyl)-nicotinonitrile 306659 2-Amino-4-(2-amino-2-phenyl-ethyl)-6-(2-hydroxy-phenyl)-nicotinonitrile 306661 2''-Amino-6''-(2-cyclopropylmethoxy-6-hydroxy-phenyl)-1,2,3,4,5,6-hexahydro-[3,4'']bipyridinyl-3''-carbonitrile 306667 Cyclopentanecarboxylic acid [6-(4-chloro-phenyl)-furo[2,3-d]pyrimidin-4-yl]-amide 306670 2''-Amino-6''-(2-hydroxy-phenyl)-1,2,3,4,5,6-hexahydro-[2,4'']bipyridinyl-3''-carbonitrile 306671 2''-Amino-6''-(2-hydroxy-phenyl)-[3,4'']bipyridinyl-3''-carbonitrile 306673 N-Phenethyl-N''-((S)-1-phenyl-ethyl)-pyridine-3,5-diamine 306674 N-[2-(4-Fluoro-phenyl)-ethyl]-N''-((S)-1-phenyl-ethyl)-pyridine-3,5-diamine 306675 Cyclopentanecarboxylic acid (6-p-tolyl-furo[2,3-d]pyrimidin-4-yl)-amide 306683 2''-Amino-6''-(2-hydroxy-6-propoxy-phenyl)-1,2,3,4,5,6-hexahydro-[3,4'']bipyridinyl-3''-carbonitrile 306684 2-Amino-6-(2-cyclopropylmethoxy-6-hydroxy-phenyl)-1'',2'',3'',4'',5'',6''-hexahydro-[4,4'']bipyridinyl-3-carbonitrile 306690 2-Amino-4-(1-amino-ethyl)-6-(2-hydroxy-phenyl)-nicotinonitrile 306691 2-Amino-4-(1-amino-pentyl)-6-(2-hydroxy-phenyl)-nicotinonitrile 306694 2''-Amino-6''-(2-hydroxy-6-isopropoxy-phenyl)-1,2,3,4,5,6-hexahydro-[3,4'']bipyridinyl-3''-carbonitrile 306702 2''-Amino-6''-(2-cyclobutylmethoxy-6-hydroxy-phenyl)-1,2,3,4,5,6-hexahydro-[3,4'']bipyridinyl-3''-carbonitrile 306710 2''-Amino-6''-(2-hydroxy-phenyl)-1-methyl-1,2,3,4,5,6-hexahydro-[3,4'']bipyridinyl-3''-carbonitrile 306714 Cyclopentanecarboxylic acid [6-(4-fluoro-phenyl)-furo[2,3-d]pyrimidin-4-yl]-amide 306717 6''-(2-Hydroxy-phenyl)-2''-methylamino-1,2,3,4,5,6-hexahydro-[3,4'']bipyridinyl-3''-carbonitrile 306722 N-(6-(pyridin-3-yl)furo[2,3-d]pyrimidin-4-yl)cyclopentanecarboxamide 306729 2''-Amino-6''-(2-hydroxy-6-pentyloxy-phenyl)-1,2,3,4,5,6-hexahydro-[3,4'']bipyridinyl-3''-carbonitrile 306730 2-Amino-6-(2-cyclobutylmethoxy-6-hydroxy-phenyl)-1'',2'',3'',4'',5'',6''-hexahydro-[4,4'']bipyridinyl-3-carbonitrile 306734 N-[2-(4-Fluoro-phenyl)-ethyl]-N''-[(S)-1-(4-fluoro-phenyl)-ethyl]-[1,3,5]triazine-2,4,6-triamine 306745 N-[(S)-1-(4-Fluoro-phenyl)-ethyl]-N''-(2-pyridin-2-yl-ethyl)-[1,3,5]triazine-2,4,6-triamine 306750 N,N-Dimethyl-N''-(2-phenoxy-ethyl)-N''''-((S)-1-phenyl-ethyl)-[1,3,5]triazine-2,4,6-triamine 306751 6-Methyl-N-(2-phenoxy-ethyl)-N''-((S)-1-phenyl-ethyl)-[1,3,5]triazine-2,4-diamine 306776 5-[1,8]Naphthyridin-4-yl-4-pyridin-2-yl-thiazol-2-ylamine 306783 5-(1,5-naphthyridin-2-yl)-4-(pyridin-2-yl)thiazol-2-amine 306787 N-(2-Phenoxy-ethyl)-N''-((S)-1-phenyl-ethyl)-[1,3,5]triazine-2,4-diamine 306794 6-Fluoro-N-(2-phenoxy-ethyl)-N''-((S)-1-phenyl-ethyl)-[1,3,5]triazine-2,4-diamine 306795 N*2*-(2-Phenoxy-ethyl)-N*4*-((S)-1-phenyl-ethyl)-pyridine-2,4-diamine 306798 N-[2-(4-Fluoro-phenoxy)-ethyl]-N''-[(R)-1-(4-fluoro-phenyl)-ethyl]-[1,3,5]triazine-2,4,6-triamine 306799 N-[1-(4-Fluoro-phenyl)-ethyl]-N''-phenethyl-[1,3,5]triazine-2,4,6-triamine 306802 (S)-N2-(2-(4-fluorophenoxy)ethyl)-N4-(1-phenylethyl)pyridine-2,4-diamine 306821 4-(4-chloropyridin-2-yl)-5-(quinolin-4-yl)thiazol-2-amine 306829 N-[2-(4-Fluoro-phenoxy)-ethyl]-N''-[1-(4-fluoro-phenyl)-ethyl]-[1,3,5]triazine-2,4,6-triamine 306832 N-(2-Phenoxy-ethyl)-N''-((S)-1-phenyl-ethyl)-[1,3,5]triazine-2,4,6-triamine 306836 N-[2-(4-Fluoro-phenoxy)-ethyl]-N''-[(S)-1-(4-fluoro-phenyl)-ethyl]-[1,3,5]triazine-2,4,6-triamine 306840 N*2*-Phenethyl-N*4*-((S)-1-phenyl-ethyl)-pyridine-2,4-diamine 306841 N*2*-[2-(4-Fluoro-phenyl)-ethyl]-N*4*-((S)-1-phenyl-ethyl)-pyridine-2,4-diamine 306861 5-(8-Methyl-[1,5]naphthyridin-2-yl)-4-pyridin-2-yl-thiazol-2-ylamine 306874 N-[1-(4-Fluoro-phenyl)-ethyl]-N''-(2-thiophen-2-yl-ethyl)-[1,3,5]triazine-2,4,6-triamine 306875 N-Phenethyl-N''-((S)-1-phenyl-ethyl)-pyrimidine-4,6-diamine 306887 4-(6-Methyl-pyridin-2-yl)-5-[1,5]naphthyridin-2-yl-thiazol-2-ylamine 306901 2-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)-1,5-naphthyridine 306904 N*4*-Phenethyl-N*2*-(1-phenyl-ethyl)-pyrimidine-2,4-diamine 306905 N*4*-[2-(4-Fluoro-phenoxy)-ethyl]-N*2*-(1-phenyl-ethyl)-pyrimidine-2,4-diamine 306922 4-(pyridin-2-yl)-5-(quinolin-4-yl)thiazol-2-amine 306930 4-(pyridin-3-yl)-5-(quinolin-4-yl)thiazol-2-amine 306956 N*2*-(2-Phenoxy-ethyl)-N*4*-((S)-1-phenyl-ethyl)-pyrimidine-2,4-diamine 306964 N*2*-[2-(4-Fluoro-phenoxy)-ethyl]-N*4*-((S)-1-phenyl-ethyl)-pyrimidine-2,4-diamine 306968 N-[2-(4-Fluoro-phenyl)-ethyl]-N''-((S)-1-phenyl-ethyl)-pyrimidine-4,6-diamine 306969 N-[2-(4-Fluoro-phenoxy)-ethyl]-N''-((S)-1-phenyl-ethyl)-pyrimidine-4,6-diamine 306971 4-(4-fluorophenyl)-5-(1,5-naphthyridin-2-yl)thiazol-2-amine 306984 N*2*-Phenethyl-N*4*-((S)-1-phenyl-ethyl)-pyrimidine-2,4-diamine 306985 N*2*-[2-(4-Fluoro-phenyl)-ethyl]-N*4*-(1-phenyl-ethyl)-pyrimidine-2,4-diamine 307004 N*4*-(2-Phenoxy-ethyl)-N*2*-((S)-1-phenyl-ethyl)-pyridine-2,4-diamine 307005 N*4*-[2-(4-Fluoro-phenoxy)-ethyl]-N*2*-((S)-1-phenyl-ethyl)-pyridine-2,4-diamine 307009 1-((4S,5S)-2,2-dimethyl-4-phenyl-1,3-dioxan-5-yl)-3-(2-methoxyphenyl)urea 307011 N-(4-methyl-2-(4-methylpiperazin-1-yl)quinolin-6-yl)-2-(4-(trifluoromethoxy)phenoxy)acetamide 307013 1-((4S,5S)-2,2-dimethyl-4-phenyl-1,3-dioxan-5-yl)-3-(2,4-dimethylphenyl)urea 307017 1-((4S,5S)-2,2-dimethyl-4-phenyl-1,3-dioxan-5-yl)-3-(2-(trifluoromethyl)phenyl)urea 307021 1-(2,5-dichlorophenyl)-3-((4S,5S)-2,2-dimethyl-4-phenyl-1,3-dioxan-5-yl)urea 307039 N-(2-Isopropylamino-4-methyl-quinolin-6-yl)-2-(4-trifluoromethyl-phenoxy)-acetamide 307043 1-((4S,5S)-2,2-Dimethyl-4-phenyl-[1,3]dioxan-5-yl)-3-(2-thiophen-3-yl-phenyl)-urea 307054 N*4*-Phenethyl-N*2*-((S)-1-phenyl-ethyl)-pyridine-2,4-diamine 307055 N*4*-[2-(4-Fluoro-phenyl)-ethyl]-N*2*-((S)-1-phenyl-ethyl)-pyridine-2,4-diamine 307058 1-(2-chlorophenyl)-3-((4S,5S)-2,2-dimethyl-4-phenyl-1,3-dioxan-5-yl)urea 307061 1-((4S,5S)-2,2-dimethyl-4-phenyl-1,3-dioxan-5-yl)-3-(2-fluorophenyl)urea 307081 2-(4-Chloro-phenoxy)-N-[4-methyl-2-(4-methyl-piperazin-1-yl)-quinolin-6-yl]-acetamide 307085 1-((4S,5S)-2,2-dimethyl-4-phenyl-1,3-dioxan-5-yl)-3-(2-isopropylphenyl)urea 307097 1-(2,2-Dimethyl-4-phenyl-[1,3]dioxan-5-yl)-3-(2-thiophen-2-yl-phenyl)-urea 307108 1-((4S,5S)-2,2-dimethyl-4-phenyl-1,3-dioxan-5-yl)-3-(2-iodophenyl)urea 307109 N-[4-Methyl-2-(4-methyl-piperazin-1-yl)-quinolin-6-yl]-2-(4-trifluoromethyl-phenoxy)-acetamide 307111 4-(2-fluorophenyl)-5-(quinolin-4-yl)thiazol-2-amine 307127 1-(2-Bromo-phenyl)-3-(2,2-dimethyl-4-phenyl-[1,3]dioxan-5-yl)-thiourea 307144 1-(2,2-Dimethyl-4-phenyl-[1,3]dioxan-5-yl)-3-(2-pyridin-3-yl-phenyl)-urea 307181 1-(2''-Chloro-biphenyl-2-yl)-3-((4S,5S)-2,2-dimethyl-4-phenyl-[1,3]dioxan-5-yl)-urea 307210 1-(2,4-Dichloro-phenyl)-3-((4S,5S)-2,2-dimethyl-4-phenyl-[1,3]dioxan-5-yl)-thiourea 307211 2,4-Dichloro-N-(2,2-dimethyl-4-phenyl-[1,3]dioxan-5-yl)-benzamide 307238 1-Biphenyl-2-yl-3-(2,2-dimethyl-4-phenyl-[1,3]dioxan-5-yl)-urea 307241 1-(3''-Chloro-biphenyl-2-yl)-3-((4S,5S)-2,2-dimethyl-4-phenyl-[1,3]dioxan-5-yl)-urea 307259 1-((4S,5S)-2,2-dimethyl-4-phenyl-1,3-dioxan-5-yl)-3-phenylurea 307260 1-(3-bromophenyl)-3-((4S,5S)-2,2-dimethyl-4-phenyl-1,3-dioxan-5-yl)urea 307262 5-Iodo-benzo[b]thiophene-2-carboxylic acid {4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-amide 307266 N-(2-Bromo-4-methyl-phenyl)-N''-((4S,5S)-2,2-dimethyl-4-phenyl-[1,3]dioxan-5-yl)-N''''-cyano-guanidine 307270 1-(4-bromo-2-methylphenyl)-3-((4S,5S)-2,2-dimethyl-4-phenyl-1,3-dioxan-5-yl)urea 307276 N-(4-Methyl-2-morpholin-4-yl-quinolin-6-yl)-2-(4-trifluoromethyl-phenoxy)-acetamide 307277 1-(2-chloro-5-methylphenyl)-3-((4S,5S)-2,2-dimethyl-4-phenyl-1,3-dioxan-5-yl)urea 307286 1-(2-bromophenyl)-3-((4S,5S)-2,2-dimethyl-4-phenyl-1,3-dioxan-5-yl)urea 307290 ((4S,5S)-2,2-Dimethyl-4-phenyl-[1,3]dioxan-5-yl)-carbamic acid 2-chloro-phenyl ester 307291 2-(2-Bromo-phenyl)-N-(2,2-dimethyl-4-phenyl-[1,3]dioxan-5-yl)-acetamide 307293 N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-5-iodobenzofuran-2-carboxamide 307294 1-(2,4-dichlorophenyl)-3-((4S,5S)-2,2-dimethyl-4-phenyl-1,3-dioxan-5-yl)urea 307301 1-(4-bromo-2-chlorophenyl)-3-((4S,5S)-2,2-dimethyl-4-phenyl-1,3-dioxan-5-yl)urea 307304 5-Iodo-thiophene-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide 307308 2-(2,3-Dichloro-phenoxy)-N-[4-methyl-2-(4-methyl-piperazin-1-yl)-quinolin-6-yl]-acetamide 307319 5-iodo-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)benzofuran-2-carboxamide 307322 N-(4-methyl-2-(pyrrolidin-1-yl)quinolin-6-yl)-2-(4-(trifluoromethyl)phenoxy)acetamide 307325 1-(4-bromophenyl)-3-((4S,5S)-2,2-dimethyl-4-phenyl-1,3-dioxan-5-yl)urea 307329 1-(2,4-dibromophenyl)-3-((4S,5S)-2,2-dimethyl-4-phenyl-1,3-dioxan-5-yl)urea 307331 5-Iodo-benzo[b]thiophene-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide 307336 5-Iodo-thiophene-2-carboxylic acid {4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-amide 307338 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-oxo-2-[4-(2-[1,2,4]triazol-1-ylmethyl-cyclohexyl)-piperazin-1-yl]-ethyl}-amide 307339 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-oxo-2-[4-(1-[1,2,4]triazol-1-ylmethyl-cyclohexyl)-piperazin-1-yl]-ethyl}-amide 307349 4-[(N-Cyclohexyl-4-phenyl-piperazine-1-carboximidoyl)-amino]-N-[2-(2,4-dichloro-phenyl)-ethyl]-benzamide 307352 (Z)-8-[(2R,3S,4R)-4-Hydroxy-2-((E)-(R)-3-hydroxy-4-phenoxy-but-1-enyl)-tetrahydro-furan-3-yl]-oct-4-enoic acid 307357 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [(R)-1-(4-chloro-benzyl)-2-(4-cyclohexyl-piperazin-1-yl)-2-oxo-ethyl]-amide 307359 (Z)-8-[(2R,3S,4R)-4-Hydroxy-2-((E)-(S)-3-hydroxy-4-phenoxy-but-1-enyl)-tetrahydro-furan-3-yl]-oct-4-enoic acid 307372 4-[(4-Benzyl-N-cyclohexyl-piperazine-1-carboximidoyl)-amino]-N-[2-(2,4-dichloro-phenyl)-ethyl]-benzamide 307379 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [(R)-1-(4-chloro-benzyl)-2-(4-cyclohexyl-4-oxy-piperazin-1-yl)-2-oxo-ethyl]-amide 307380 (Z)-8-{(2R,3S,4R)-4-Hydroxy-2-[(E)-(R)-3-hydroxy-4-(3-trifluoromethyl-phenoxy)-but-1-enyl]-tetrahydro-furan-3-yl}-oct-4-enoic acid 307392 4-[(N-Cyclohexyl-piperazine-1-carboximidoyl)-amino]-N-[2-(2,4-dichloro-phenyl)-ethyl]-benzamide 307394 (Z)-8-{(2R,3S,4R)-2-[(E)-(R)-4-(3-Chloro-phenoxy)-3-hydroxy-but-1-enyl]-4-hydroxy-tetrahydro-furan-3-yl}-oct-6-enoic acid 307399 (Z)-8-{(2R,3S,4R)-2-[(E)-(S)-4-(3-Chloro-phenoxy)-3-hydroxy-but-1-enyl]-4-hydroxy-tetrahydro-furan-3-yl}-oct-6-enoic acid 307409 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [(R)-1-(4-chloro-benzyl)-2-oxo-2-(4-phenyl-piperazin-1-yl)-ethyl]-amide 307425 4-[(N-Cyclohexyl-4-pyrimidin-2-yl-piperazine-1-carboximidoyl)-amino]-N-[2-(2,4-dichloro-phenyl)-ethyl]-benzamide 307428 (Z)-8-{(2R,3S,4R)-2-[(E)-(R)-4-(3-Chloro-phenoxy)-3-hydroxy-but-1-enyl]-4-hydroxy-tetrahydro-furan-3-yl}-oct-4-enoic acid 307432 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [(R)-1-(4-chloro-benzyl)-2-oxo-2-(4-oxy-4-phenyl-piperazin-1-yl)-ethyl]-amide 307434 (Z)-8-{(2R,3S,4R)-2-[(E)-(S)-4-(3-Chloro-phenoxy)-3-hydroxy-but-1-enyl]-4-hydroxy-tetrahydro-furan-3-yl}-oct-4-enoic acid 307444 4-[(N-Cyclohexyl-4-methyl-piperazine-1-carboximidoyl)-amino]-N-[2-(2,4-dichloro-phenyl)-ethyl]-benzamide 307447 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-oxo-2-[4-((1R,2R)-2-[1,2,4]triazol-1-yl-cyclohexyl)-piperazin-1-yl]-ethyl}-amide 307456 (Z)-8-{(2R,3S,4R)-4-Hydroxy-2-[(E)-(S)-3-hydroxy-4-(3-trifluoromethyl-phenoxy)-but-1-enyl]-tetrahydro-furan-3-yl}-oct-4-enoic acid 307464 4-[((R)-N-Cyclohexyl-3-methyl-piperazine-1-carboximidoyl)-amino]-N-[2-(2,4-dichloro-phenyl)-ethyl]-benzamide 307466 (Z)-8-{(2R,3S,4R)-4-Hydroxy-2-[(E)-(R)-3-hydroxy-4-(3-trifluoromethyl-phenoxy)-but-1-enyl]-tetrahydro-furan-3-yl}-oct-6-enoic acid 307492 4-{[N-Cyclohexyl-4-(2,5-dimethyl-phenyl)-piperazine-1-carboximidoyl]-amino}-N-[2-(2,4-dichloro-phenyl)-ethyl]-benzamide 307494 (Z)-7-[(2R,3S,4R)-4-Hydroxy-2-((E)-(S)-3-hydroxy-oct-1-enyl)-tetrahydro-furan-3-yl]-hept-5-enoic acid 307546 4-[((S)-N-Cyclohexyl-3-methyl-piperazine-1-carboximidoyl)-amino]-N-[2-(2,4-dichloro-phenyl)-ethyl]-benzamide 307642 {2-[5-(4-Chloro-phenyl)-isoxazol-3-yl]-phenoxymethyl}-dimethyl-amine 307643 1-[4-(5-Phenyl-isoxazol-3-yl)-phenoxymethyl]-piperidine 307646 Dimethyl-[4-(5-phenyl-isoxazol-3-yl)-phenoxymethyl]-amine 307647 3-[3-(2-Bromo-phenyl)-ureido]-6-chloro-2-hydroxy-benzamide 307655 1-(3,5-Dimethyl-phenyl)-3-[4-(1-oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-urea 307656 N-{3-Oxo-7-[4-(3-m-tolyl-ureido)-phenyl]-2,3-dihydro-1H-isoindol-4-yl}-nicotinamide 307659 1-[3-Fluoro-4-(1-oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-3-m-tolyl-urea 307660 1-{4-[7-(2-Methoxy-ethoxy)-1-oxo-2,3-dihydro-1H-isoindol-4-yl]-phenyl}-3-m-tolyl-urea 307686 2-[4-(4-Methoxy-phenyl)-piperazin-1-yl]-N-m-tolyl-acetamide 307689 Dimethyl-{4-[5-(4-nitro-phenyl)-isoxazol-3-yl]-phenoxymethyl}-amine 307690 {3-[5-(4-Chloro-phenyl)-isoxazol-3-yl]-phenoxymethyl}-dimethyl-amine 307695 1-(2-Bromo-phenyl)-3-(4-chloro-2-hydroxy-phenyl)-urea 307697 2-[4-(1-Oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-N-m-tolyl-acetamide 307701 1-(2-Bromo-phenyl)-3-(3,4-dichloro-2-hydroxy-phenyl)-urea 307702 1-(3,4-Dimethyl-phenyl)-3-[4-(1-oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-urea 307705 1-(2-Fluoro-5-trifluoromethyl-phenyl)-3-[4-(1-oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-urea 307706 1-[4-(7-Methoxy-1-oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-3-m-tolyl-urea 307709 N-{3-Oxo-7-[4-(3-m-tolyl-ureido)-phenyl]-2,3-dihydro-1H-isoindol-4-yl}-benzamide 307732 2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-N-m-tolyl-acetamide 307736 {4-[5-(4-Chloro-phenyl)-isoxazol-3-yl]-phenoxymethyl}-dimethyl-amine 307737 {4-[5-(4-Fluoro-phenyl)-isoxazol-3-yl]-phenoxymethyl}-dimethyl-amine 307738 3-[3-(2-Bromo-phenyl)-ureido]-6-chloro-2-hydroxy-benzenesulfonamide 307742 2-[4-(3-Methoxy-phenyl)-piperazin-1-yl]-N-m-tolyl-acetamide 307743 3-[3-(2-Bromo-phenyl)-ureido]-6-chloro-2-hydroxy-N,N-dimethyl-benzenesulfonamide 307744 1-Indan-5-yl-3-[4-(1-oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-urea 307749 2-Dimethylamino-N-{3-oxo-7-[4-(3-m-tolyl-ureido)-phenyl]-2,3-dihydro-1H-isoindol-4-yl}-acetamide 307753 (Z)-8-[(2R,3S,4R)-4-Hydroxy-2-((E)-(R)-3-hydroxy-4-phenoxy-but-1-enyl)-tetrahydro-furan-3-yl]-oct-6-enoic acid 307761 (Z)-8-[(R)-4-Hydroxy-2-((1R,2S,4S)-3-hydroxy-4-phenoxy-but-1-enyl)-tetrahydro-furan-3-yl]-oct-6-enoic acid 307780 1-(2-Bromo-phenyl)-3-(2,4-dihydroxy-phenyl)-urea 307781 1-[3-Chloro-4-(1-oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-3-m-tolyl-urea 307783 2-[4-(4-Fluoro-phenyl)-piperazin-1-yl]-N-m-tolyl-acetamide 307786 1-[4-(1-Oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-3-m-tolyl-urea 307789 1-(4-Butoxy-benzoyl)-5-methoxy-2-methyl-1H-indole-3-carboxylic acid 307790 3-[1-(4-Butoxy-benzoyl)-5-methoxy-2-methyl-1H-indol-3-yl]-propionic acid 307797 1-[2-Methyl-4-(1-oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-3-m-tolyl-urea 307817 [1-(2-Butoxy-benzoyl)-5-methoxy-2-methyl-1H-indol-3-yl]-acetic acid 307820 1-(3-{4-[3-(4-Chloro-phenyl)-isoxazol-5-yl]-phenoxy}-propyl)-4-methyl-piperazine 307825 1-{4-[5-(4-Chloro-phenyl)-isoxazol-3-yl]-phenoxymethyl}-4-methyl-piperazine 307827 1-(3-{4-[3-(3-Chloro-phenyl)-isoxazol-5-yl]-phenoxy}-propyl)-4-methyl-piperazine 307828 1-Methyl-3-[4-(1-oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-1-m-tolyl-urea 307830 2-[4-(4-Benzhydryl-phenyl)-piperazin-1-yl]-N-m-tolyl-acetamide 307831 1-(2-{4-[5-(4-Chloro-phenyl)-isoxazol-3-yl]-phenoxy}-ethyl)-4-methyl-piperazine 307832 1-[4-(1-Oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-3-phenyl-urea 307840 1-[4-(1-Oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-3-m-tolyl-thiourea 307841 1-[4-(1-Oxo-2,3-dihydro-1H-isoindol-4-yl)-2-trifluoromethyl-phenyl]-3-m-tolyl-urea 307844 1-[3-Methyl-4-(1-oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-3-m-tolyl-urea 307861 1-(4-Butoxy-benzoyl)-5-methoxy-1H-indole-3-carboxylic acid 307862 1-(4-Butoxy-benzoyl)-5-methoxy-2-propyl-1H-indole-3-carboxylic acid 307870 1-Methyl-4-{3-[4-(3-phenyl-isoxazol-5-yl)-phenoxy]-propyl}-piperazine 307881 (3-{4-[3-(4-Chloro-phenyl)-isoxazol-5-yl]-phenoxy}-propyl)-dimethyl-amine 307882 1-Methyl-1-[4-(1-oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-3-m-tolyl-urea 307887 1-Methyl-4-[4-(5-phenyl-isoxazol-3-yl)-phenoxymethyl]-piperazine 307888 1-[4-(1-Oxo-2,3-dihydro-1H-isoindol-4-yl)-3-trifluoromethyl-phenyl]-3-m-tolyl-urea 307892 1-Methyl-4-[4-(5-phenyl-isoxazol-3-yl)-phenoxymethyl]-piperidine 307900 [1-(3-Butoxy-benzoyl)-5-methoxy-2-methyl-1H-indol-3-yl]-acetic acid 307904 1-[2-Fluoro-4-(1-oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-3-m-tolyl-urea 307907 [1-(4-Butoxy-benzoyl)-5-methoxy-2-methyl-1H-indol-3-yl]-acetic acid 307931 1-(3-{4-[3-(4-Fluoro-phenyl)-isoxazol-5-yl]-phenoxy}-propyl)-4-methyl-piperazine 307936 1-Methyl-4-[4-(5-pyridin-2-yl-isoxazol-3-yl)-phenoxymethyl]-piperazine 307937 Dimethyl-{3-[4-(3-phenyl-isoxazol-5-yl)-phenoxy]-propyl}-amine 307940 1-[4-(1-Oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-3-o-tolyl-urea 307941 1-[4-(1-Oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-3-p-tolyl-urea 307948 2-[4-(4-Bromo-2-cyano-phenyl)-piperazin-1-yl]-N-(2,4,6-tribromo-3-methyl-phenyl)-acetamide 307965 1-Methyl-4-(3-{4-[3-(3-trifluoromethyl-phenyl)-isoxazol-5-yl]-phenoxy}-propyl)-piperazine 307979 Hymenialdisine 307984 1-[4-(1-Oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-3-(4-trifluoromethyl-phenyl)-urea 307985 1-[2-Ethyl-4-(1-oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-3-m-tolyl-urea 307989 1-(3-Cyano-phenyl)-3-[4-(1-oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-urea 307990 N-{3-Oxo-7-[4-(3-m-tolyl-ureido)-phenyl]-2,3-dihydro-1H-isoindol-4-yl}-acetamide 307994 5-[1-(4-Butoxy-benzoyl)-5-methoxy-2-methyl-1H-indol-3-yl]-pentanoic acid 308003 [1-(4-Butoxy-benzoyl)-2-methyl-1H-indol-3-yl]-acetic acid 308018 2-[4-(4-Bromo-2-cyano-phenyl)-piperazin-1-yl]-N-(4-bromo-3-methyl-phenyl)-acetamide 308033 1-(3-Fluoro-phenyl)-3-[4-(1-oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-urea 308034 1-(3-Methoxy-phenyl)-3-[4-(1-oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-urea 308039 1-[4-(7-Amino-1-oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-3-m-tolyl-urea 308045 1-Methyl-4-(3-{4-[3-(4-phenoxy-phenyl)-isoxazol-5-yl]-phenoxy}-propyl)-piperazine 308046 1-[4-(1-Oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-3-(3-trifluoromethyl-phenyl)-urea 308057 1-[2-Chloro-4-(1-oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-3-m-tolyl-urea 308066 4-[1-(4-Butoxy-benzoyl)-5-methoxy-2-methyl-1H-indol-3-yl]-butyric acid 308070 2-[4-(2-Cyano-phenyl)-piperazin-1-yl]-N-m-tolyl-acetamide 308075 1-(3-{4-[3-(4-Fluoro-phenyl)-[1,2,4]oxadiazol-5-yl]-phenoxy}-propyl)-4-methyl-piperazine 308076 1-(3-{4-[3-(4-Chloro-phenyl)-[1,2,4]oxadiazol-5-yl]-phenoxy}-propyl)-4-methyl-piperazine 308084 1-(3-Chloro-phenyl)-3-[4-(1-oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-urea 308085 1-(3-Ethyl-phenyl)-3-[4-(1-oxo-2,3-dihydro-1H-isoindol-4-yl)-phenyl]-urea 308098 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [(R)-2-(4-{2-[(2-amino-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-1-(4-chloro-benzyl)-2-oxo-ethyl]-amide 308099 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [(R)-1-(4-chloro-benzyl)-2-(4-{2-[(3-hydroxy-propylamino)-methyl]-phenyl}-piperazin-1-yl)-2-oxo-ethyl]-amide 308102 [1-(4-Butoxy-benzoyl)-2,5-dimethyl-1H-indol-3-yl]-acetic acid 308103 [1-(4-Butoxy-benzoyl)-5-hydroxy-2-methyl-1H-indol-3-yl]-acetic acid 308118 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [(R)-2-(4-{2-[(benzyl-methyl-amino)-methyl]-phenyl}-piperazin-1-yl)-1-(4-chloro-benzyl)-2-oxo-ethyl]-amide 308119 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [(R)-1-(4-chloro-benzyl)-2-(4-{2-[(methyl-pyridin-3-ylmethyl-amino)-methyl]-phenyl}-piperazin-1-yl)-2-oxo-ethyl]-amide 308120 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-[4-(2-{[methyl-(2-pyridin-2-yl-ethyl)-amino]-methyl}-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-amide 308121 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid ((R)-1-(4-chloro-benzyl)-2-oxo-2-{4-[2-(4-pyrrolidin-1-yl-piperidin-1-ylmethyl)-phenyl]-piperazin-1-yl}-ethyl)-amide 308122 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid ((R)-1-(4-chloro-benzyl)-2-oxo-2-{4-[2-(4-phenyl-piperazin-1-ylmethyl)-phenyl]-piperazin-1-yl}-ethyl)-amide 308131 N-(2-Hydroxy-5-{1-hydroxy-2-[2-(4-phenoxy-phenyl)-ethylamino]-ethyl}-phenyl)-formamide 308135 N-[2-Hydroxy-5-((R)-1-hydroxy-2-{2-[4-(4-phenyl-butoxy)-phenyl]-ethylamino}-ethyl)-phenyl]-formamide 308164 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-[4-(2-{[(2-hydroxy-ethyl)-methyl-amino]-methyl}-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-amide 308165 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-[4-(2-{[(2-methoxy-ethyl)-methyl-amino]-methyl}-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-amide 308186 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [(R)-1-(4-chloro-benzyl)-2-oxo-2-(4-{2-[1-(2-thiophen-2-yl-ethylamino)-ethyl]-phenyl}-piperazin-1-yl)-ethyl]-amide 308187 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [(R)-1-(4-chloro-benzyl)-2-oxo-2-(4-{2-[1-((S)-pyrrolidin-3-ylamino)-ethyl]-phenyl}-piperazin-1-yl)-ethyl]-amide 308188 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [(R)-2-(4-{2-[1-(4-amino-cyclohexylamino)-ethyl]-phenyl}-piperazin-1-yl)-1-(4-chloro-benzyl)-2-oxo-ethyl]-amide 308189 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [(R)-2-(4-{2-[1-((S)-2-amino-cyclohexylamino)-ethyl]-phenyl}-piperazin-1-yl)-1-(4-chloro-benzyl)-2-oxo-ethyl]-amide 308190 N-[2-Hydroxy-5-(1-hydroxy-2-{2-[4-(3-phenyl-propoxy)-phenyl]-ethylamino}-ethyl)-phenyl]-formamide 308218 3-{2-[4-((R)-3-(4-Chloro-phenyl)-2-{[(R)-oxo-(1,2,3,4-tetrahydro-isoquinolin-3-yl)-methyl]-amino}-propionyl)-piperazin-1-yl]-benzylamino}-propionic acid 308219 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-oxo-2-[4-(2-{[(piperidin-4-ylmethyl)-amino]-methyl}-phenyl)-piperazin-1-yl]-ethyl}-amide 308234 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid ((R)-1-(4-chloro-benzyl)-2-{4-[2-((S)-2-methyl-5-(S)-methyl-piperazin-1-ylmethyl)-phenyl]-piperazin-1-yl}-2-oxo-ethyl)-amide 308235 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid ((R)-1-(4-chloro-benzyl)-2-{4-[2-(1-cyclopropylamino-ethyl)-phenyl]-piperazin-1-yl}-2-oxo-ethyl)-amide 308236 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid ((R)-1-(4-chloro-benzyl)-2-{4-[2-(1-cyclopentylamino-ethyl)-phenyl]-piperazin-1-yl}-2-oxo-ethyl)-amide 308237 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-[4-(2-{1-[(furan-2-ylmethyl)-amino]-ethyl}-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-amide 308238 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-[4-(2-{1-[2-(2-fluoro-phenyl)-ethylamino]-ethyl}-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-amide 308245 N-(2-Hydroxy-5-{(R)-1-hydroxy-2-[2-(4-phenethyloxy-phenyl)-ethylamino]-ethyl}-phenyl)-formamide 308255 1N-[6-carbamoyl-9-(4-nitrobenzyl)-8,11,14-trioxo-(1R,6S,9S)-3,4-dithia-7,10,13-triazacyclotetradecanyl]-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-(2S)-propanamide 308321 N-[2-Hydroxy-5-((R)-1-hydroxy-2-{2-[3-(4-phenyl-butoxy)-phenyl]-ethylamino}-ethyl)-phenyl]-formamide 308374 N-[2-Hydroxy-5-(1-hydroxy-2-{2-[4-(indan-2-yloxy)-phenyl]-ethylamino}-ethyl)-phenyl]-formamide 308414 N-[2-Hydroxy-5-(1-hydroxy-2-{2-[3-(3-phenoxy-propoxy)-phenyl]-ethylamino}-ethyl)-phenyl]-formamide 308430 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-[4-(2-cyclopropylaminomethyl-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-amide 308431 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-[4-(2-cyclopentylaminomethyl-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-amide 308496 (R)-N-((R)-1-(4-(2-(aminomethyl)phenyl)piperazin-1-yl)-3-(4-chlorophenyl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 308527 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-[4-(2-{[(furan-2-ylmethyl)-amino]-methyl}-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-amide 308528 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-[4-(2-{[2-(2-fluoro-phenyl)-ethylamino]-methyl}-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-amide 308529 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-[4-(2-{[2-(3-fluoro-phenyl)-ethylamino]-methyl}-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-amide 308530 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-[4-(2-{[2-(4-fluoro-phenyl)-ethylamino]-methyl}-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-amide 308567 Isoindolinone Urea derivative 308583 [3-(Methyl-tetradecyl-amino)-propyl]-phosphonic acid 308584 [3-(2-Tetradecyl-pyrrolidin-1-yl)-propyl]-phosphonic acid 308606 (E)-7-{(1R,2R,3R,5S)-3,5-Dihydroxy-2-[(E)-3-hydroxy-4-(3-trifluoromethyl-phenoxy)-but-1-enyl]-cyclopentyl}-hept-5-enoic acid isopropyl ester 308636 [Hydroxy-(1-tetradecyl-pyrrolidin-3-yl)-methyl]-phosphonic acid 308644 (3-Hydroxy-1-tetradecyl-pyrrolidin-3-yl)-phosphonic acid 308648 (E)-7-[(1R,2R,3R,5S)-3,5-Dihydroxy-2-((R)-3-hydroxy-5-phenyl-pentyl)-cyclopentyl]-hept-5-enoic acid isopropyl ester 308660 [3-(2-Tridecyl-piperidin-1-yl)-propyl]-phosphonic acid 308667 [2-(1-Tetradecyl-pyrrolidin-2-yl)-ethyl]-phosphonic acid 308701 (4-Bromo-2,6-dimethyl-phenyl)-(4,5-dihydro-1H-imidazol-2-yl)-amine 308702 (4,5-Dihydro-1H-imidazol-2-yl)-(2,6-dimethyl-4-nitro-phenyl)-amine 308707 {2-[5-(4-Nonyl-phenyl)-pyrrolidin-2-yl]-ethyl}-phosphonic acid 308732 (4-Hydroxy-1-tetradecyl-piperidin-4-yl)-methyl-phosphinic acid 308733 Methyl-[2-(6-tridecyl-piperidin-2-yl)-ethyl]-phosphinic acid 308744 (4,5-Dihydro-1H-imidazol-2-yl)-(2,6-dimethyl-phenyl)-amine 308745 (3-Tetradecylamino-cyclohexyl)-phosphonic acid 308747 (4-tert-Butyl-2,6-dimethyl-phenyl)-(4,5-dihydro-1H-imidazol-2-yl)-amine 308762 1-Benzyl-2-(4-tert-butyl-2,6-dimethyl-benzyl)-4,5-dihydro-1H-imidazole 308769 2-(4-tert-Butyl-2,6-dimethyl-benzyl)-1,4,5,6-tetrahydro-pyrimidine 308778 (2-Tetradecylamino-cyclohexylmethyl)-phosphonic acid 308779 (3-Tetradecylamino-cyclopentyl)-phosphonic acid 308800 SID11111295 308807 [(1S,3S)-3-(4-Nonyl-benzylamino)-cyclohexyl]-phosphonic acid 308817 [2-((2R,5S)-5-Tetradecyl-pyrrolidin-2-yl)-ethyl]-phosphonic acid 308821 (5H-benzo[e]pyrrolo[1,2-a][1,4]diazepin-10(11H)-yl)(2-chloro-4-(3-methyl-1H-pyrazol-1-yl)phenyl)methanone 308824 1-[1-(4-Propyl-cyclohexyl)-piperidin-4-yl]-3,4-dihydro-1H-benzo[1,2,6]thiadiazine 2,2-dioxide 308825 1-[1-(1,4-Dimethyl-pentyl)-piperidin-4-yl]-3,4-dihydro-1H-benzo[1,2,6]thiadiazine 2,2-dioxide 308833 {1-[4-(Chroman-2-ylmethoxy)-benzoyl]-2-methyl-1H-indol-4-yl}-acetic acid 308852 3-Phenylamino-4-[1-(3-piperidin-1-yl-propyl)-1H-indol-3-yl]-pyrrole-2,5-dione 308870 1-[1-(4-Benzyloxy-benzyl)-piperidin-4-yl]-3,4-dihydro-1H-benzo[1,2,6]thiadiazine 2,2-dioxide 308874 1-[1-(Decahydro-naphthalen-2-yl)-piperidin-4-yl]-3,4-dihydro-1H-benzo[1,2,6]thiadiazine 2,2-dioxide 308875 Trans-1-[1-(4-Isopropyl-cyclohexyl)-piperidin-4-yl]-3,4-dihydro-1H-benzo[1,2,6]thiadiazine 2,2-dioxide 308877 1-(4-nonylbenzyl)pyrrolidin-3-ylphosphonic acid 308882 {1-[4-(Benzo[1,3]dioxol-2-ylmethoxy)-benzoyl]-2-methyl-1H-indol-4-yl}-acetic acid 308884 (4-Hydroxy-2-tetradecyl-piperidin-4-yl)-methyl-phosphinic acid 308892 1-Ethyl-3-{(S)-1-[2-(4-phenyl-butyl)-benzofuran-4-yl]-pyrrolidin-3-yl}-urea 308898 3-Phenylamino-4-[1-(3-pyrrolidin-1-yl-propyl)-1H-indol-3-yl]-pyrrole-2,5-dione 308900 1-(1-Indan-2-yl-piperidin-4-yl)-3,4-dihydro-1H-benzo[1,2,6]thiadiazine 2,2-dioxide 308901 1-[1-(1,2,3,4-Tetrahydro-naphthalen-2-yl)-piperidin-4-yl]-3,4-dihydro-1H-benzo[1,2,6]thiadiazine 2,2-dioxide 308910 {1-[4-(2,3-Dihydro-benzofuran-2-ylmethoxy)-benzoyl]-2-methyl-1H-indol-4-yl}-acetic acid 308935 3-{1-[3-(4-Methyl-piperazin-1-yl)-propyl]-1H-indol-3-yl}-4-phenylamino-pyrrole-2,5-dione 308955 1-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-3,4-dihydro-1H-benzo[1,2,6]thiadiazine 2,2-dioxide 308956 {2-Methyl-1-[4-(2-phenoxy-ethoxy)-benzoyl]-1H-indol-4-yl}-acetic acid 308963 3-(1H-Indol-3-yl)-4-p-tolylamino-pyrrole-2,5-dione 308964 3-(3-Fluoro-phenylamino)-4-(1H-indol-3-yl)-pyrrole-2,5-dione 308969 3-Butyl-1-[1-(4-isopropyl-cyclohexyl)-piperidin-4-yl]-3,4-dihydro-1H-benzo[1,2,6]thiadiazine 2,2-dioxide 308970 {1-[4-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethoxy)-benzoyl]-2-methyl-1H-indol-4-yl}-acetic acid 308973 1-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-1,3-dihydro-benzo[1,2,5]thiadiazole 2,2-dioxide 308974 2-{1-[1-(4-Isopropyl-cyclohexyl)-piperidin-4-yl]-2,2-dioxo-1,4-dihydro-2H-2lambda*6*-benzo[1,2,6]thiadiazin-3-yl}-acetamide 308979 {2-Methyl-1-[4-(4-methyl-3,4-dihydro-2H-benzo[1,4]oxazin-2-ylmethoxy)-benzoyl]-1H-indol-4-yl}-acetic acid 308991 1-cyclopropylcarboxamidomethyl-2-[2-(4-phenylbutyl)benzo[b]furan-4-yl]-(1R,2R)-cyclopropane 308992 1-Ethyl-3-{(1R,2R)-2-[2-(4-phenyl-butyl)-benzofuran-4-yl]-cyclopropylmethyl}-urea 308995 3-(1-(3-imidazol-1-ylpropyl)-1H-indol-3-yl)-4-anilino-1H-pyrrole-2,5-dione 308998 3-(1H-Indol-3-yl)-4-o-tolylamino-pyrrole-2,5-dione 308999 3-(1H-Indol-3-yl)-4-m-tolylamino-pyrrole-2,5-dione 309006 {1-[4-(Chroman-3-ylmethoxy)-benzoyl]-2-methyl-1H-indol-4-yl}-acetic acid 309017 1-[1-(4-Benzyloxy-benzyl)-piperidin-4-yl]-1,3-dihydro-benzo[1,2,5]thiadiazole 2,2-dioxide 309018 {1-[1-(4-Isopropyl-cyclohexyl)-piperidin-4-yl]-2,2-dioxo-1,4-dihydro-2H-2lambda*6*-benzo[1,2,6]thiadiazin-3-yl}-acetic acid tert-butyl ester 309031 {2-Methyl-1-[4-(4-methyl-3,4-dihydro-2H-benzo[1,4]oxazin-2-ylmethoxy)-benzoyl]-1H-indol-4-yl}-acetic acid 309035 1N-[2-[2-(4-phenylbutyl)benzo[b]furan-4-yl]-(1R,2R)-cyclopropylmethyl]butanamide 309036 1N-[2-[2-(4-phenylbutyl)benzo[b]furan-4-yl]-(1R,2R)-cyclopropylmethyl]-2-methylpropanamide 309042 1-(1-Cyclooctyl-piperidin-4-yl)-3,4-dihydro-1H-benzo[1,2,6]thiadiazine 2,2-dioxide 309043 3-(1H-Indol-3-yl)-4-phenylamino-pyrrole-2,5-dione 309044 3-(1H-Indol-3-yl)-4-(methyl-phenyl-amino)-pyrrole-2,5-dione 309058 3-(3-Chloro-phenylamino)-4-(1H-indol-3-yl)-pyrrole-2,5-dione 309059 3-(1H-Indol-3-yl)-4-(3-methoxy-phenylamino)-pyrrole-2,5-dione 309064 {1-[1-(4-Isopropyl-cyclohexyl)-piperidin-4-yl]-2,2-dioxo-1,4-dihydro-2H-2lambda*6*-benzo[1,2,6]thiadiazin-3-yl}-acetic acid methyl ester 309065 {1-[4-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethoxy)-benzoyl]-2-methyl-1H-indol-4-yl}-acetic acid 309069 1N-[2-[2-(4-phenylbutyl)benzo[b]furan-4-yl]-(1R,2R)-cyclopropylmethyl]acetamide 309074 1N-[2-[2-(4-phenylbutyl)benzo[b]furan-4-yl]-(1R,2R)-cyclopropylmethyl]propanamide 309083 3-Cyclohexylamino-4-(1H-indol-3-yl)-pyrrole-2,5-dione 309087 N-{3-[2-(4-Phenyl-butyl)-benzofuran-4-yl]-propyl}-acetamide 309088 N-{3-[2-(4-Phenyl-butyl)-benzofuran-4-yl]-propyl}-propionamide 309095 Cyclopropanecarboxylic acid {3-[2-(4-phenyl-butyl)-benzofuran-4-yl]-propyl}-amide 309099 1-Ethyl-3-{3-[2-(4-phenyl-butyl)-benzofuran-4-yl]-propyl}-urea 309106 3-[1-(2-Dimethylamino-ethyl)-1H-indol-3-yl]-4-phenylamino-pyrrole-2,5-dione 309118 N-{(S)-1-[2-(4-Phenyl-butyl)-benzofuran-4-yl]-pyrrolidin-3-yl}-isobutyramide 309123 1-[1-(4-Propyl-cyclohexyl)-piperidin-4-yl]-1,3-dihydro-benzo[1,2,5]thiadiazole 2,2-dioxide 309124 1-[1-(1,4-Dimethyl-pentyl)-piperidin-4-yl]-1,3-dihydro-benzo[1,2,5]thiadiazole 2,2-dioxide 309125 3-[1-(3-Dimethylamino-propyl)-1H-indol-3-yl]-4-m-tolylamino-pyrrole-2,5-dione 309128 8-Cyclobutylmethoxy-quinolin-2-ylamine 309131 N-(2-{1-[1-(4-Isopropyl-cyclohexyl)-piperidin-4-yl]-2,2-dioxo-1,4-dihydro-2H-2lambda*6*-benzo[1,2,6]thiadiazin-3-yl}-ethyl)-methanesulfonamide 309137 N-{3-[2-(4-Phenyl-butyl)-benzofuran-4-yl]-propyl}-butyramide 309144 N-{3-[2-(4-Phenyl-butyl)-benzofuran-4-yl]-propyl}-isobutyramide 309145 3-(1H-Indol-3-yl)-4-(3-trifluoromethyl-phenylamino)-pyrrole-2,5-dione 309151 N-{(S)-1-[2-(4-Phenyl-butyl)-benzofuran-4-yl]-pyrrolidin-3-yl}-butyramide 309153 3-(1H-Indol-3-yl)-4-(3-isopropyl-phenylamino)-pyrrole-2,5-dione 309156 1-[1-(Decahydro-naphthalen-2-yl)-piperidin-4-yl]-1,3-dihydro-benzo[1,2,5]thiadiazole 2,2-dioxide 309157 3-[1-(5-Dimethylamino-pentyl)-1H-indol-3-yl]-4-phenylamino-pyrrole-2,5-dione 309158 3-[1-(3-Hydroxy-propyl)-1H-indol-3-yl]-4-phenylamino-pyrrole-2,5-dione 309162 1-[1-(4-Isopropyl-cyclohexyl)-piperidin-4-yl]-1,3-dihydro-benzo[1,2,5]thiadiazole 2,2-dioxide 309163 2-{1-[1-(4-Isopropyl-cyclohexyl)-piperidin-4-yl]-2,2-dioxo-1,4-dihydro-2H-2lambda*6*-benzo[1,2,6]thiadiazin-3-yl}-ethanol 309179 1-(1-Biphenyl-4-ylmethyl-piperidin-4-yl)-3,4-dihydro-1H-benzo[1,2,6]thiadiazine 2,2-dioxide 309183 N-{(S)-1-[2-(4-Phenyl-butyl)-benzofuran-4-yl]-pyrrolidin-3-yl}-acetamide 309190 N-{(S)-1-[2-(4-Phenyl-butyl)-benzofuran-4-yl]-pyrrolidin-3-yl}-propionamide 309191 3-[1-(3-Dimethylamino-propyl)-1H-indol-3-yl]-4-phenylamino-pyrrole-2,5-dione 309202 1-(1-Indan-2-yl-piperidin-4-yl)-1,3-dihydro-benzo[1,2,5]thiadiazole 2,2-dioxide 309203 1-[1-(1,2,3,4-Tetrahydro-naphthalen-2-yl)-piperidin-4-yl]-1,3-dihydro-benzo[1,2,5]thiadiazole 2,2-dioxide 309204 3-[1-(4-Dimethylamino-butyl)-1H-indol-3-yl]-4-phenylamino-pyrrole-2,5-dione 309209 Cyclopropanecarboxylic acid {(S)-1-[2-(4-phenyl-butyl)-benzofuran-4-yl]-pyrrolidin-3-yl}-amide 309210 3-(3-Chloro-phenylamino)-4-[1-(3-dimethylamino-propyl)-1H-indol-3-yl]-pyrrole-2,5-dione 309211 {1-[1-(4-Isopropyl-cyclohexyl)-piperidin-4-yl]-2,2-dioxo-1,4-dihydro-2H-2lambda*6*-benzo[1,2,6]thiadiazin-3-yl}-acetonitrile 309212 {1-[4-(7-Fluoro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazin-2-ylmethoxy)-benzoyl]-2-methyl-1H-indol-4-yl}-acetic acid 309215 1-(1-Cyclooctyl-piperidin-4-yl)-1,3-dihydro-benzo[1,2,5]thiadiazole 2,2-dioxide 309216 1-(1-Naphthalen-2-ylmethyl-piperidin-4-yl)-3,4-dihydro-1H-benzo[1,2,6]thiadiazine 2,2-dioxide 309224 3-((R)-2-Amino-2-phenyl-ethyl)-5-(4-chloro-phenyl)-1-(2,6-difluoro-benzyl)-6-methyl-1H-pyrimidine-2,4-dione 309226 8-(2-Methyl-butoxy)-quinolin-2-ylamine 309227 8-(3-Methyl-butoxy)-quinolin-2-ylamine 309228 8-(1-Methyl-2-piperidin-1-yl-ethoxy)-quinolin-2-ylamine 309232 8-((S)-1-Benzo[1,3]dioxol-5-ylmethyl-pyrrolidin-3-yloxy)-quinolin-2-ylamine 309234 8-(2-Methoxy-1-methyl-ethoxy)-quinolin-2-ylamine 309235 8-Cyclohexyloxy-quinolin-2-ylamine 309236 8-(1-Methyl-2-morpholin-4-yl-ethoxy)-quinolin-2-ylamine 309237 1-Benzo[1,3]dioxol-5-yl-3-[3-(2-{[5-(2-chloro-phenyl)-furan-2-ylmethyl]-amino}-quinolin-8-yloxy)-propyl]-urea 309240 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-6-methyl-5-(2-o-tolylamino-thiazol-4-yl)-1H-pyrimidine-2,4-dione 309241 3-((R)-2-Amino-2-phenyl-ethyl)-5-[2-(4-tert-butyl-phenyl)-thiazol-4-yl]-1-(2,6-difluoro-benzyl)-6-methyl-1H-pyrimidine-2,4-dione 309242 N*7*-[(R)-1-(2,6-Dichloro-benzyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidine-5,7-diamine 309250 8-(3,3,3-trifluoropropoxy)quinolin-2-amine 309251 8-(3-Methoxy-3-methyl-butoxy)-quinolin-2-ylamine 309252 8-{2-[(Furan-3-ylmethyl)-amino]-ethoxy}-quinolin-2-ylamine 309253 2-Furan-2-yl-N*5*-[(R)-1-(5-methyl-isoxazol-3-ylmethyl)-pyrrolidin-2-ylmethyl]-[1,2,4]triazolo[1,5-a]pyrimidine-5,7-diamine 309254 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-6-methyl-5-thiophen-2-yl-1H-pyrimidine-2,4-dione 309256 (S)-N-(1-benzylpyrrolidin-3-yl)-4-(thiophen-2-yl)benzamide 309257 N-((R)-1-Benzyl-pyrrolidin-3-yl)-4-thiophen-3-yl-benzamide 309258 8-[3-(Benzo[1,3]dioxol-5-ylamino)-propoxy]-quinolin-2-ylamine 309259 N-{4-[(S)-3-(2-Amino-quinolin-8-yloxy)-pyrrolidin-1-ylmethyl]-phenyl}-acetamide 309260 2-Furan-2-yl-N*7*-methyl-N*7*-{2-[4-(2,4,6-trifluoro-phenyl)-piperazin-1-yl]-ethyl}-[1,2,4]triazolo[1,5-c]pyrimidine-5,7-diamine 309261 4''-Chloro-biphenyl-4-carboxylic acid (1-benzyl-pyrrolidin-3-yl)-amide 309263 8-Isopropoxy-quinolin-2-ylamine 309268 [(S)-3-(2-Amino-quinolin-8-yloxy)-pyrrolidin-1-yl]-benzo[1,3]dioxol-5-yl-methanone 309270 2''-Formyl-biphenyl-4-carboxylic acid (1-benzyl-pyrrolidin-3-yl)-amide 309273 8-sec-Butoxy-quinolin-2-ylamine 309274 8-Cyclopentylmethoxy-quinolin-2-ylamine 309278 8-(2-Cyclopropyl-ethoxy)-quinolin-2-ylamine 309279 8-(2-Cyclohexylamino-1-methyl-ethoxy)-quinolin-2-ylamine 309280 8-(1-Methyl-2-pyrrolidin-1-yl-ethoxy)-quinolin-2-ylamine 309283 8-{2-[(Benzo[1,3]dioxol-5-ylmethyl)-amino]-1-methyl-ethoxy}-quinolin-2-ylamine 309284 8-[2-(1H-Indazol-5-ylamino)-1-methyl-ethoxy]-quinolin-2-ylamine 309285 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-6-methyl-5-(2-p-tolylamino-thiazol-4-yl)-1H-pyrimidine-2,4-dione 309286 (R)-1-(2,6-difluorobenzyl)-3-(2-amino-2-phenylethyl)-5-(5-chlorothiophen-2-yl)-6-methylpyrimidine-2,4(1H,3H)-dione 309287 3-Chloro-N-[3-(2-{[5-(2-chloro-phenyl)-furan-2-ylmethyl]-amino}-quinolin-8-yloxy)-propyl]-benzamide 309288 {2-Methyl-1-[4-(3-phenyl-propoxy)-benzoyl]-1H-indol-4-yl}-acetic acid 309290 8-[3-(4-Chloro-3-trifluoromethyl-benzylamino)-propoxy]-quinolin-2-ylamine 309291 8-((S)-1-Benzyl-pyrrolidin-3-yloxy)-quinolin-2-ylamine 309293 N*5*-[(R)-1-(3,5-Dichloro-pyridin-4-ylmethyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrimidine-5,7-diamine 309294 3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-benzylamino-thiazol-4-yl)-1-(2,6-difluoro-benzyl)-6-methyl-1H-pyrimidine-2,4-dione 309295 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-5-[2-(2,3-dihydro-benzofuran-5-yl)-thiazol-4-yl]-6-methyl-1H-pyrimidine-2,4-dione 309296 (4-{4-[3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-6-methyl-2,4-dioxo-1,2,3,4-tetrahydro-pyrimidin-5-yl]-thiazol-2-yl}-phenyl)-carbamic acid ethyl ester 309299 8-(1,2-Dimethyl-propoxy)-quinolin-2-ylamine 309300 8-(1-Ethyl-propoxy)-quinolin-2-ylamine 309301 N7-(2-(4-(2,4-difluorophenyl)piperazin-1-yl)ethyl)-2-(furan-2-yl)-N7-methyl-[1,2,4]triazolo[1,5-c]pyrimidine-5,7-diamine 309302 4''-Fluoro-biphenyl-4-carboxylic acid (1-benzyl-pyrrolidin-3-yl)-amide 309304 2-Furan-2-yl-N*5*-methyl-N*5*-[(R)-1-(5-methyl-isoxazol-3-ylmethyl)-pyrrolidin-2-ylmethyl]-[1,2,4]triazolo[1,5-a]pyrimidine-5,7-diamine 309312 8-(3,3-Dimethyl-butoxy)-quinolin-2-ylamine 309314 8-(1,3,3-Trimethyl-butoxy)-quinolin-2-ylamine 309315 3''-Fluoro-biphenyl-4-carboxylic acid (1-benzyl-pyrrolidin-3-yl)-amide 309322 8-Cyclohexylmethoxy-quinolin-2-ylamine 309323 N-(1-Benzyl-pyrrolidin-3-yl)-4-thiophen-3-yl-benzamide 309324 N-((R)-1-Benzyl-pyrrolidin-3-yl)-4-thiophen-2-yl-benzamide 309326 8-{2-[(Benzo[1,3]dioxol-5-ylmethyl)-amino]-ethoxy}-quinolin-2-ylamine 309327 8-((R)-1-Benzo[1,3]dioxol-5-ylmethyl-pyrrolidin-3-yloxy)-quinolin-2-ylamine 309333 8-(2-Benzylamino-1-methyl-ethoxy)-quinolin-2-ylamine 309337 8-[(S)-1-(4-tert-Butyl-benzyl)-pyrrolidin-3-yloxy]-quinolin-2-ylamine 309340 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-6-methyl-5-[2-(methyl-phenyl-amino)-thiazol-4-yl]-1H-pyrimidine-2,4-dione 309341 8-[2-(3-Methoxy-benzylamino)-1-methyl-ethoxy]-quinolin-2-ylamine 309342 N-[3-(2-Amino-quinolin-8-yloxy)-propyl]-3-chloro-benzamide 309344 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-5-[2-(2,4-dimethyl-phenylamino)-thiazol-4-yl]-6-methyl-1H-pyrimidine-2,4-dione 309345 N*7*-[(R)-1-(2-Fluoro-benzyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidine-5,7-diamine 309346 2-Furan-2-yl-5-[4-(2,4,6-trifluoro-phenyl)-piperazin-1-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 309354 3-((R)-2-Amino-2-phenyl-ethyl)-5-[2-(4-chloro-phenyl)-thiazol-4-yl]-1-(2,6-difluoro-benzyl)-6-methyl-1H-pyrimidine-2,4-dione 309356 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-6-methyl-5-(5-methyl-thiophen-2-yl)-1H-pyrimidine-2,4-dione 309359 N-((S)-1-Benzyl-pyrrolidin-3-yl)-4-thiophen-3-yl-benzamide 309360 N-((R)-1-Benzyl-pyrrolidin-3-yl)-3-thiophen-3-yl-benzamide 309363 N*5*-[(R)-1-(2-Chloro-pyridin-4-ylmethyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrimidine-5,7-diamine 309366 8-(1-Methyl-butoxy)-quinolin-2-ylamine 309371 4''-Formyl-biphenyl-4-carboxylic acid (1-benzyl-pyrrolidin-3-yl)-amide 309372 8-(Tetrahydro-furan-3-ylmethoxy)-quinolin-2-ylamine 309373 8-Hexyloxy-quinolin-2-ylamine 309374 8-{2-[(Furan-3-ylmethyl)-amino]-1-methyl-ethoxy}-quinolin-2-ylamine 309379 8-Pentyloxy-quinolin-2-ylamine 309380 N-(1-Benzyl-pyrrolidin-3-yl)-4-thiophen-2-yl-benzamide 309383 8-{1-Methyl-2-[(thiophen-3-ylmethyl)-amino]-ethoxy}-quinolin-2-ylamine 309384 8-((R)-1-Benzyl-pyrrolidin-3-yloxy)-quinolin-2-ylamine 309385 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-5-[2-(2-methoxy-phenylamino)-thiazol-4-yl]-6-methyl-1H-pyrimidine-2,4-dione 309387 4-(4-Fluoro-phenyl)-5-pyridin-4-yl-1,2-dihydro-pyrazol-3-one 309388 3-(4-Fluoro-phenyl)-2-pyridin-4-yl-6,7-dihydro-5H-pyrazolo[5,1-b][1,3]oxazine 309389 2-Furan-2-yl-N*5*-[3-(4-phenyl-piperazin-1-yl)-propyl]-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 309400 N-[3-(2-Amino-quinolin-8-yloxy)-propyl]-3-cyano-benzamide 309407 8-[(R)-1-(2,2-Difluoro-benzo[1,3]dioxol-5-yl)-pyrrolidin-3-yloxy]-quinolin-2-ylamine 309413 8-(4-Methyl-cyclohexyloxy)-quinolin-2-ylamine 309415 N*7*-[(R)-1-(2-Chloro-pyridin-4-ylmethyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidine-5,7-diamine 309421 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-6-methyl-5-[2-(4-nitro-phenylamino)-thiazol-4-yl]-1H-pyrimidine-2,4-dione 309422 8-Cycloheptyloxy-quinolin-2-ylamine 309423 Methyl-[8-(1,3,3-trimethyl-butoxy)-quinolin-2-yl]-amine 309425 N*5*-{2-[4-(2,4-Difluoro-phenyl)-piperazin-1-yl]-ethyl}-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 309432 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-6-methyl-5-(2-methyl-thiazol-4-yl)-1H-pyrimidine-2,4-dione 309434 Benzo[1,3]dioxole-5-carboxylic acid [3-(2-amino-quinolin-8-yloxy)-propyl]-amide 309435 N-[3-(2-Amino-quinolin-8-yloxy)-propyl]-3-methoxy-benzamide 309437 N*7*-[(R)-1-(2-Chloro-benzyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidine-5,7-diamine 309438 2-Furan-2-yl-N*5*-[2-(4-phenyl-piperazin-1-yl)-ethyl]-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 309447 8-[1-(2,2-Difluoro-benzo[1,3]dioxol-5-yl)-pyrrolidin-3-yloxy]-quinolin-2-ylamine 309451 N-((S)-1-Benzyl-pyrrolidin-3-yl)-3-thiophen-3-yl-benzamide 309452 N-((S)-1-benzylpyrrolidin-3-yl)-3-(thiophen-2-yl)benzamide 309455 8-(2-Ethoxy-1-methyl-ethoxy)-quinolin-2-ylamine 309456 2-Furan-2-yl-N*7*-[(R)-1-(5-methyl-isoxazol-3-ylmethyl)-pyrrolidin-2-ylmethyl]-[1,2,4]triazolo[1,5-c]pyrimidine-5,7-diamine 309457 2-Furan-2-yl-N*5*-{3-[4-(2,4,6-trifluoro-phenyl)-piperazin-1-yl]-propyl}-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 309463 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-6-methyl-5-[2-(3-trifluoromethyl-phenyl)-thiazol-4-yl]-1H-pyrimidine-2,4-dione 309466 8-(3-Methyl-cyclohexyloxy)-quinolin-2-ylamine 309467 8-(Bicyclo[2.2.1]hept-2-ylmethoxy)-quinolin-2-ylamine 309475 8-[3-(4-Isopropyl-benzylamino)-propoxy]-quinolin-2-ylamine 309476 N-[3-(2-Amino-quinolin-8-yloxy)-propyl]-4-isopropyl-benzamide 309480 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-5-[2-(4-methoxy-phenylamino)-thiazol-4-yl]-6-methyl-1H-pyrimidine-2,4-dione 309481 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-5-[2-(3,4-dimethoxy-phenylamino)-thiazol-4-yl]-6-methyl-1H-pyrimidine-2,4-dione 309482 8-[1-(4-Isobutyl-phenyl)-pyrrolidin-3-yloxy]-quinolin-2-ylamine 309483 8-[1-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-pyrrolidin-3-yloxy]-quinolin-2-ylamine 309489 8-(2-tert-Butoxy-1-methyl-ethoxy)-quinolin-2-ylamine 309491 N*7*-[(R)-1-(3,5-Dichloro-pyridin-4-ylmethyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidine-5,7-diamine 309492 3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-benzyl-thiazol-4-yl)-1-(2,6-difluoro-benzyl)-6-methyl-1H-pyrimidine-2,4-dione 309493 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-6-methyl-5-[2-(4-trifluoromethyl-phenyl)-thiazol-4-yl]-1H-pyrimidine-2,4-dione 309497 2-Furan-2-yl-N*5*-{2-[4-(2,4,6-trifluoro-phenyl)-piperazin-1-yl]-ethyl}-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 309510 N-[3-(2-Amino-quinolin-8-yloxy)-propyl]-3-trifluoromethoxy-benzamide 309511 8-(3-Methyl-cyclopentyloxy)-quinolin-2-ylamine 309512 8-(2-Methyl-cyclohexyloxy)-quinolin-2-ylamine 309518 8-[1-(2-Benzo[1,3]dioxol-5-yl-1-methyl-ethyl)-pyrrolidin-3-yloxy]-quinolin-2-ylamine 309519 8-[1-(1-Phenyl-propyl)-pyrrolidin-3-yloxy]-quinolin-2-ylamine 309520 8-[2-(2-Methoxy-ethoxy)-ethoxy]-quinolin-2-ylamine 309521 8-[3-(2,2-Difluoro-benzo[1,3]dioxol-5-ylamino)-propoxy]-quinolin-2-ylamine 309526 2-Furan-2-yl-N*7*-methyl-N*7*-[(R)-1-(5-methyl-isoxazol-3-ylmethyl)-pyrrolidin-2-ylmethyl]-[1,2,4]triazolo[1,5-c]pyrimidine-5,7-diamine 309527 8-[(S)-1-(4-tert-Butyl-benzenesulfonyl)-pyrrolidin-3-yloxy]-quinolin-2-ylamine 309530 8-(2-Ethyl-1-methyl-butoxy)-quinolin-2-ylamine 309531 [5-(2-Chloro-phenyl)-furan-2-ylmethyl]-[8-(1,3,3-trimethyl-butoxy)-quinolin-2-yl]-amine 309532 N*5*-{3-[4-(2,4-Difluoro-phenyl)-piperazin-1-yl]-propyl}-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 309538 2-Furan-2-yl-N*7*-((R)-1-pyridin-4-ylmethyl-pyrrolidin-2-ylmethyl)-[1,2,4]triazolo[1,5-c]pyrimidine-5,7-diamine 309539 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-6-methyl-5-(2-phenyl-thiazol-4-yl)-1H-pyrimidine-2,4-dione 309540 2-Methoxy-4-[3-(4-phenoxy-phenyl)-ureido]-N-(3-piperidin-1-yl-propyl)-benzamide 309543 4''-Methylsulfanyl-biphenyl-4-carboxylic acid (1-benzyl-pyrrolidin-3-yl)-amide 309551 N-[3-(2-{[5-(3-Chloro-phenyl)-furan-2-ylmethyl]-amino}-quinolin-8-yloxy)-propyl]-3-cyano-benzamide 309552 Cyclopropylmethyl-{8-[1-(4-isobutyl-phenyl)-pyrrolidin-3-yloxy]-quinolin-2-yl}-amine 309553 {8-[1-(4-Isobutyl-phenyl)-pyrrolidin-3-yloxy]-quinolin-2-yl}-[5-(3-trifluoromethyl-phenyl)-furan-2-ylmethyl]-amine 309554 ((R)-sec-Butyl)-{4-[7-(4-fluoro-phenyl)-2,3-dihydro-pyrazolo[5,1-b]oxazol-6-yl]-pyrimidin-2-yl}-amine 309560 N*5*-[(R)-1-(2-Fluoro-benzyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 309561 N*5*-[(R)-1-(2-Fluoro-benzyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrimidine-5,7-diamine 309564 3-(2,6-Dichloro-phenyl)-5-[2-(2,2-dimethyl-5-oxo-pyrrolidin-1-yl)-ethyl]-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 309568 N*5*-{2-[4-(2,4-Difluoro-phenyl)-piperazin-1-yl]-ethyl}-2-furan-2-yl-N*5*-methyl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 309569 4''-Trifluoromethyl-biphenyl-4-carboxylic acid (1-benzyl-pyrrolidin-3-yl)-amide 309570 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-6-methyl-5-(2-morpholin-4-yl-thiazol-4-yl)-1H-pyrimidine-2,4-dione 309576 {4-[7-(4-Fluoro-phenyl)-2,3-dihydro-pyrazolo[5,1-b]oxazol-6-yl]-pyrimidin-2-yl}-((R)-1-phenyl-ethyl)-amine 309577 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-5-[2-(3-fluoro-4-methyl-phenyl)-thiazol-4-yl]-6-methyl-1H-pyrimidine-2,4-dione 309580 8-Propoxy-quinolin-2-ylamine 309581 {4-[7-(4-Fluoro-phenyl)-2,3-dihydro-pyrazolo[5,1-b]oxazol-6-yl]-pyrimidin-2-yl}-((R)-2-methoxy-1-methyl-ethyl)-amine 309593 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-5-(2-ethylamino-thiazol-4-yl)-6-methyl-1H-pyrimidine-2,4-dione 309595 8-(2-Methyl-cyclopropylmethoxy)-quinolin-2-ylamine 309597 N-(2-Diethylamino-ethyl)-2-ethoxy-4-[3-(4-phenoxy-phenyl)-ureido]-benzamide 309598 1-[3-(2-Amino-quinolin-8-yloxy)-propyl]-3-benzo[1,3]dioxol-5-yl-urea 309599 1-[3-(2-Amino-quinolin-8-yloxy)-propyl]-3-(3-chloro-phenyl)-urea 309600 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-6-methyl-5-(2-p-tolyl-thiazol-4-yl)-1H-pyrimidine-2,4-dione 309602 8-(2-Cyclopropylamino-1-methyl-ethoxy)-quinolin-2-ylamine 309603 8-(2-Cyclopentylamino-1-methyl-ethoxy)-quinolin-2-ylamine 309604 4-[3-(4-Acetyl-phenyl)-ureido]-N-(2-diethylamino-ethyl)-2-methoxy-benzamide 309608 {8-[1-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-pyrrolidin-3-yloxy]-quinolin-2-yl}-methyl-amine 309611 3-Chloro-N-[3-(2-propylamino-quinolin-8-yloxy)-propyl]-benzamide 309612 [2-Methyl-1-(4-phenethyloxy-benzoyl)-1H-indol-4-yl]-acetic acid 309614 N*5*-[(R)-1-(2,6-Dichloro-benzyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 309615 N*5*-[(R)-1-(2,6-Dichloro-benzyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrimidine-5,7-diamine 309618 2-Furan-2-yl-N*5*-((R)-1-pyridin-4-ylmethyl-pyrrolidin-2-ylmethyl)-[1,2,4]triazolo[1,5-a]pyrimidine-5,7-diamine 309621 2-Furan-2-yl-N*5*-methyl-N*5*-[2-(4-phenyl-piperazin-1-yl)-ethyl]-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 309629 2-Furan-2-yl-N*7*-{2-[4-(2,4,6-trifluoro-phenyl)-piperazin-1-yl]-ethyl}-[1,2,4]triazolo[1,5-c]pyrimidine-5,7-diamine 309630 Biphenyl-4-carboxylic acid (1-benzyl-pyrrolidin-3-yl)-amide 309633 3-(4-Fluoro-phenyl)-2-(2-phenoxy-pyrimidin-4-yl)-6,7-dihydro-5H-pyrazolo[5,1-b][1,3]oxazine 309636 8-[2-(Cyclopropylmethyl-amino)-1-methyl-ethoxy]-quinolin-2-ylamine 309637 Biphenyl-3-carboxylic acid (1-benzyl-pyrrolidin-3-yl)-amide 309641 7-(4-Fluoro-phenyl)-6-(2-phenoxy-pyrimidin-4-yl)-2,3-dihydro-pyrazolo[5,1-b]oxazole 309643 8-[2-(Cyclopentylmethyl-amino)-1-methyl-ethoxy]-quinolin-2-ylamine 309644 N-[3-(2-{[5-(4-Chloro-phenyl)-furan-2-ylmethyl]-amino}-quinolin-8-yloxy)-propyl]-3-cyano-benzamide 309646 3-(2,6-Dichloro-phenyl)-5-[2-(3-methyl-2-oxo-imidazolidin-1-yl)-ethyl]-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 309647 3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-amino-thiazol-4-yl)-1-(2,6-difluoro-benzyl)-6-methyl-1H-pyrimidine-2,4-dione 309648 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-5-[2-(4-fluoro-phenyl)-thiazol-4-yl]-6-methyl-1H-pyrimidine-2,4-dione 309649 [1-(4-Butoxy-benzoyl)-2-methyl-1H-indol-4-yl]-acetic acid 309650 [1-(4-Benzyloxy-benzoyl)-2-methyl-1H-indol-4-yl]-acetic acid 309652 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-6-methyl-5-(2-phenylamino-thiazol-4-yl)-1H-pyrimidine-2,4-dione 309657 N*5*-[(R)-1-(2-Chloro-benzyl)-pyrrolidin-2-ylmethyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrimidine-5,7-diamine 309658 3-((R)-2-Amino-2-phenyl-ethyl)-5-[2-(2-chloro-phenyl)-thiazol-4-yl]-1-(2,6-difluoro-benzyl)-6-methyl-1H-pyrimidine-2,4-dione 309665 8-Butoxy-quinolin-2-ylamine 309666 N7-(2-(4-(2,4-difluorophenyl)piperazin-1-yl)ethyl)-2-(furan-2-yl)-[1,2,4]triazolo[1,5-c]pyrimidine-5,7-diamine 309667 3''-Amino-biphenyl-4-carboxylic acid (1-benzyl-pyrrolidin-3-yl)-amide 309674 Biphenyl-4-carboxylic acid [4-(2-dimethylamino-ethylcarbamoyl)-3-methoxy-phenyl]-amide 309675 N-(2-Diethylamino-ethyl)-4-[3-(4-trifluoromethyl-phenyl)-ureido]-benzamide 309676 N-(2-Diethylamino-ethyl)-2-methoxy-4-[1-methyl-3-(4-phenoxy-phenyl)-ureido]-benzamide 309677 3-(2,6-Dichloro-phenyl)-5-(2-oxo-pyrrolidin-1-ylmethyl)-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 309679 2-Methoxy-N-(3-morpholin-4-yl-propyl)-4-[3-(3-phenoxy-phenyl)-ureido]-benzamide 309680 N-(2-Diethylamino-ethyl)-2-methoxy-4-[3-(3-methylsulfanyl-phenyl)-ureido]-benzamide 309686 3-(2,6-Dichloro-phenyl)-5-isopropyl-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 309687 3-(2,6-Dichloro-phenyl)-5-[2-(2-methoxy-phenyl)-ethyl]-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 309704 Biphenyl-4-carboxylic acid [4-(3-dimethylamino-propylcarbamoyl)-3-methoxy-phenyl]-amide 309705 2-Methoxy-4-[3-(3-phenoxy-phenyl)-ureido]-N-(3-piperidin-1-yl-propyl)-benzamide 309710 5-[2-(Acetyl-methyl-amino)-ethyl]-3-(2,6-dichloro-phenyl)-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 309711 4-[3-(4-Cyano-phenyl)-ureido]-N-(2-diethylamino-ethyl)-2-methoxy-benzamide 309712 N-(2-Diethylamino-ethyl)-2-methoxy-4-[3-(4-methylsulfanyl-phenyl)-ureido]-benzamide 309714 3-(2,6-Dichloro-phenyl)-5-propyl-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 309716 N-(2-Diethylamino-ethyl)-4-[3-(4-trifluoromethoxy-phenyl)-ureido]-benzamide 309721 5-(2-Benzo[1,3]dioxol-4-yl-ethyl)-3-(2,6-dichloro-phenyl)-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 309722 N-(2-Diethylamino-ethyl)-2-methoxy-4-[3-(3-trifluoromethyl-phenyl)-ureido]-benzamide 309740 Biphenyl-4-carboxylic acid [4-(2-diethylamino-ethylcarbamoyl)-3-methoxy-phenyl]-amide 309745 3-(2,6-Dichloro-phenyl)-5-(3-hydroxy-propyl)-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 309747 N-(2-Diethylamino-ethyl)-2-methoxy-4-{3-[4-(2,2,2-trifluoro-acetyl)-phenyl]-ureido}-benzamide 309750 Biphenyl-4-carboxylic acid [4-(1-benzyl-piperidin-4-ylcarbamoyl)-3-methoxy-phenyl]-amide 309751 3-(2,6-Dichloro-phenyl)-5-methyl-isoxazole-4-carboxylic acid (4-diethylamino-cyclohexyl)-amide 309756 3-(2,6-Dichloro-phenyl)-5-ethyl-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 309757 5-(2-Benzo[1,3]dioxol-5-yl-ethyl)-3-(2,6-dichloro-phenyl)-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 309758 N-(2-Diethylamino-ethyl)-2-methoxy-4-[3-(4-trifluoromethoxy-phenyl)-ureido]-benzamide 309759 N-(2-Diethylamino-ethyl)-2-methoxy-4-[3-(4-trifluoromethylsulfanyl-phenyl)-ureido]-benzamide 309786 N-(2-Diethylamino-ethyl)-2-methoxy-4-(4-phenoxy-benzoylamino)-benzamide 309787 N-(2-Diethylamino-ethyl)-2-methoxy-4-[3-(4-trifluoromethyl-phenyl)-ureido]-benzamide 309791 Biphenyl-4-carboxylic acid {4-[2-(4-benzyl-piperazin-1-yl)-ethylcarbamoyl]-3-methoxy-phenyl}-amide 309798 N-(2-Diethylamino-ethyl)-N-methyl-4-[3-(4-phenoxy-phenyl)-ureido]-benzamide 309808 N-(1-Ethyl-pyrrolidin-2-ylmethyl)-4-[3-(4-phenoxy-phenyl)-ureido]-benzamide 309809 N-(2-Diethylamino-ethyl)-2-methoxy-4-[3-(3-trifluoromethoxy-phenyl)-ureido]-benzamide 309810 N-(2-Diethylamino-ethyl)-4-[5-(4-phenoxy-phenyl)-[1,2,4]oxadiazol-3-yl]-benzamide 309811 2-Methoxy-4-[3-(3-phenylamino-phenyl)-ureido]-N-(3-piperidin-1-yl-propyl)-benzamide 309812 3-(2,6-Dichloro-phenyl)-5-[2-(tetrahydro-pyran-4-yl)-ethyl]-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 309813 5-(2-Benzo[1,3]dioxol-5-yl-ethyl)-3-(2,6-dichloro-phenyl)-isoxazole-4-carboxylic acid (4-diethylamino-cyclohexyl)-amide 309828 3-(2,6-Dichloro-phenyl)-5-[2-(tetrahydro-furan-2-yl)-ethyl]-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 309831 3-(2,6-Dichloro-phenyl)-5-(2-methoxy-ethyl)-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 309832 3-(2,6-Dichloro-phenyl)-5-(2-[1,3]dioxan-2-yl-ethyl)-isoxazole-4-carboxylic acid (4-diethylamino-cyclohexyl)-amide 309835 4-(3-Biphenyl-4-yl-ureido)-N-(3-dimethylamino-propyl)-2-methoxy-benzamide 309841 4-[3-(4-Bromo-phenyl)-ureido]-N-(2-diethylamino-ethyl)-2-methoxy-benzamide 309842 N-(2-Diethylamino-ethyl)-4-[3-(3,5-dimethoxy-phenyl)-ureido]-2-methoxy-benzamide 309856 N-(2-Diethylamino-ethyl)-4-[3-(4-phenoxy-phenyl)-ureido]-benzamide 309858 N-(1-Ethyl-pyrrolidin-2-ylmethyl)-2-methoxy-4-[3-(4-phenoxy-phenyl)-ureido]-benzamide 309859 4-[3-(3,4-Dichloro-phenyl)-ureido]-N-(2-diethylamino-ethyl)-2-methoxy-benzamide 309861 N-(3-Dimethylamino-propyl)-2-methoxy-4-(4-phenoxy-benzoylamino)-benzamide 309862 3-(2,6-Dichloro-phenyl)-5-[2-(tetrahydro-pyran-2-yl)-ethyl]-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 309865 2-Methoxy-4-[3-(4-phenylamino-phenyl)-ureido]-N-(3-piperidin-1-yl-propyl)-benzamide 309866 N-(2-Diethylamino-ethyl)-2-methoxy-4-[3-methyl-3-(4-phenoxy-phenyl)-ureido]-benzamide 309867 3-(2,6-Dichloro-phenyl)-5-[2-(2-oxo-piperidin-1-yl)-ethyl]-isoxazole-4-carboxylic acid (4-diethylamino-cyclohexyl)-amide 309880 3-(2,6-Dichloro-phenyl)-5-(2-[1,3]dioxolan-2-yl-ethyl)-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 309883 N-(1-Ethyl-pyrrolidin-2-ylmethyl)-4-[5-(4-phenoxy-phenyl)-[1,2,4]oxadiazol-3-yl]-benzamide 309891 N-(2-Diethylamino-ethyl)-4-[3-(4-fluoro-phenyl)-ureido]-2-methoxy-benzamide 309902 N-(2-Diethylamino-ethyl)-2-methoxy-4-[3-(4-phenoxy-phenyl)-ureido]-benzamide 309903 3-(2,6-Dichloro-phenyl)-5-[2-(2-oxo-piperidin-1-yl)-ethyl]-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 309904 3-(2,6-Dichloro-phenyl)-5-[2-(tetrahydro-furan-2-yl)-ethyl]-isoxazole-4-carboxylic acid (4-diethylamino-cyclohexyl)-amide 309908 4-[3-(3-Chloro-4-fluoro-phenyl)-ureido]-N-(2-diethylamino-ethyl)-2-methoxy-benzamide 309909 4-[3-(3,5-Dichloro-phenyl)-ureido]-N-(2-diethylamino-ethyl)-2-methoxy-benzamide 309916 3-{1-(4-Chloro-phenyl)-1-hydroxy-3-[4-(4-methanesulfonyl-benzyl)-[1,4]diazepan-1-yl]-propyl}-phenol 309917 N-({[1-(4-Chloro-benzyl)-pyrrolidin-2-ylmethyl]-carbamoyl}-methyl)-3-trifluoromethyl-benzamide 309919 N-{3-[6-(3-Diethylamino-propylamino)-pyrimidin-4-ylamino]-4-methyl-phenyl}-2-morpholin-4-yl-isonicotinamide 309923 1-(3-dimethylaminophenylcarboxamido)-3-(4-isopropoxyphenylcarboxamido)-4-methylbenzene 309924 N-{2-[1-(4-Chloro-benzyl)-piperidin-3-ylcarbamoyl]-ethyl}-benzamide 309931 3-Fluoro-N-{4-methyl-3-[4-(2-methyl-thiazol-4-ylmethoxy)-benzoylamino]-phenyl}-5-morpholin-4-yl-benzamide 309935 1-(3,3-Diphenyl-propyl)-4-(4-nitro-benzyl)-[1,4]diazepane 309936 4-methyl-1-[3-(1,4-oxazinan-4-yl)phenylcarboxamido]-3-[4-(2-pyridylmethoxy)phenylcarboxamido]benzene 309937 N-[5-(6,7-Dimethoxy-quinazolin-4-ylamino)-2,4-difluoro-phenyl]-benzamide 309938 N-[3-(6,7-Dimethoxy-quinazolin-4-ylamino)-4-methyl-phenyl]-3-morpholin-4-yl-benzamide 309939 N-{3-[6-(2-Diisopropylamino-ethoxy)-7-methoxy-quinazolin-4-ylamino]-4-methyl-phenyl}-2-morpholin-4-yl-isonicotinamide 309940 N-{3-[7-Methoxy-6-(2-morpholin-4-yl-ethoxy)-quinazolin-4-ylamino]-4-methyl-phenyl}-2-morpholin-4-yl-isonicotinamide 309941 N-(3-(7-methoxy-6-(2-(pyrrolidin-1-yl)ethoxy)quinazolin-4-ylamino)-4-methylphenyl)-2-morpholinoisonicotinamide 309944 4-{4-[3-Hydroxy-3-(3-hydroxy-phenyl)-3-phenyl-propyl]-[1,4]diazepan-1-ylmethyl}-benzenesulfonamide 309945 N-{4-Methyl-3-[6-(4-methyl-[1,4]diazepan-1-yl)-pyrimidin-4-ylamino]-phenyl}-2-morpholin-4-yl-isonicotinamide 309947 N-{4-Methyl-3-[2-(1-propyl-piperidin-4-yloxy)-pyrimidin-4-ylamino]-phenyl}-3-morpholin-4-yl-benzamide 309951 N-{[1-(4-Chloro-benzyl)-piperidin-3-ylcarbamoyl]-methyl}-3-trifluoromethyl-benzamide 309954 1-(3,3-Diphenyl-propyl)-4-pyridin-4-ylmethyl-[1,4]diazepane 309955 1-(3-dimethylaminophenylcarboxamido)-3-[4-(2-ethoxyethoxy)phenylcarboxamido]-4-methylbenzene 309961 1,1-di(3-hydroxyphenyl)-3-[4-(4-methylsulfonylbenzyl)-1,4-diazepan-1-yl]-1-propanol 309962 3-{1-(4-Fluoro-phenyl)-1-hydroxy-3-[4-(4-methanesulfonyl-benzyl)-[1,4]diazepan-1-yl]-propyl}-phenol 309963 N-[3-(6-Chloro-pyrimidin-4-ylamino)-4-methyl-phenyl]-2-morpholin-4-yl-isonicotinamide 309964 N-[4-Methyl-3-(pyrimidin-4-ylamino)-phenyl]-2-morpholin-4-yl-isonicotinamide 309967 3-(2,6-Dichloro-phenyl)-5-[2-(2-oxo-pyrrolidin-1-yl)-ethyl]-isoxazole-4-carboxylic acid (4-diethylamino-phenyl)-amide 309969 5-Oxo-5-phenyl-pentanoic acid [1-(4-chloro-benzyl)-piperidin-3-yl]-amide 309984 N-[3-(6,7-Dimethoxy-quinazolin-4-ylamino)-phenyl]-benzamide 309985 N-{4-Methyl-3-[6-(3-pyrrolidin-1-yl-propylamino)-pyrimidin-4-ylamino]-phenyl}-2-morpholin-4-yl-isonicotinamide 309987 N-[2-(4-Benzyl-piperazin-1-yl)-ethyl]-4-[3-(4-phenoxy-phenyl)-ureido]-benzamide 309990 3-{1-(3,5-Difluoro-phenyl)-1-hydroxy-3-[4-(4-methanesulfonyl-benzyl)-[1,4]diazepan-1-yl]-propyl}-phenol 309991 N-({[1-(4-Chloro-benzyl)-piperidin-4-ylmethyl]-carbamoyl}-methyl)-3-trifluoromethyl-benzamide 309995 4-[3-(2-Bromo-4-trifluoromethoxy-phenyl)-ureido]-N-(2-diethylamino-ethyl)-2-methoxy-benzamide 309999 1-(3-dimethylaminophenylcarboxamido)-3-[4-(2-methoxyethoxy)phenylcarboxamido]-4-methylbenzene 310000 N-{[1-(4-Chloro-benzyl)-piperidin-3-ylcarbamoyl]-methyl}-3-methyl-benzamide 310003 1,1-Bis-(4-fluoro-phenyl)-3-[4-(4-methanesulfonyl-benzyl)-[1,4]diazepan-1-yl]-propan-1-ol 310005 N-{3-[6-(2-Dimethylamino-ethoxy)-7-methoxy-quinazolin-4-ylamino]-4-methyl-phenyl}-2-morpholin-4-yl-isonicotinamide 310006 N-{3-[7-Methoxy-6-(2-piperidin-1-yl-ethoxy)-quinazolin-4-ylamino]-4-methyl-phenyl}-2-morpholin-4-yl-isonicotinamide 310009 4-Methyl-thiophene-2-carboxylic acid N''-(2-{4-[3-hydroxy-3-(3-hydroxy-phenyl)-3-phenyl-propyl]-[1,4]diazepan-1-yl}-acetyl)-hydrazide 310010 5-Oxo-5-phenyl-pentanoic acid [1-(4-chloro-benzyl)-pyrrolidin-3-yl]-amide 310011 3-{1-(3-Chloro-phenyl)-1-hydroxy-3-[4-(4-methanesulfonyl-benzyl)-[1,4]diazepan-1-yl]-propyl}-phenol 310012 N-{[1-(4-Chloro-benzyl)-pyrrolidin-3-ylcarbamoyl]-methyl}-3-trifluoromethyl-benzamide 310013 3-Fluoro-N-[4-methyl-3-(2-methylsulfanyl-pyrimidin-4-ylamino)-phenyl]-5-morpholin-4-yl-benzamide 310016 N-{2-[1-(4-Chloro-benzyl)-pyrrolidin-3-ylcarbamoyl]-ethyl}-benzamide 310017 N-({[1-(4-Chloro-benzyl)-piperidin-4-ylmethyl]-carbamoyl}-methyl)-3-methyl-benzamide 310025 1-(3-dimethylaminophenylcarboxamido)-4-methyl-3-[4-(2-pyridylmethoxy)phenylcarboxamido]benzene 310034 4-Methyl-thiophene-2-carboxylic acid N''-{2-[3-(3,3-diphenyl-propylamino)-pyrrolidin-1-yl]-acetyl}-hydrazide 310039 N-[5-(3-Dimethylamino-benzoylamino)-2-methyl-phenyl]-3,4-dimethoxy-benzamide 310045 1-(3,3-Diphenyl-propyl)-4-(4-methanesulfonyl-benzyl)-[1,4]diazepane 310046 3-Fluoro-N-{4-methyl-3-[4-(pyridin-2-ylmethoxy)-benzoylamino]-phenyl}-5-pyrrolidin-1-yl-benzamide 310047 N-[2-Chloro-5-(6,7-dimethoxy-quinazolin-4-ylamino)-4-fluoro-phenyl]-benzamide 310052 1,1-Bis-(4-chloro-phenyl)-3-[4-(4-methanesulfonyl-benzyl)-[1,4]diazepan-1-yl]-propan-1-ol 310054 N-{4-Methyl-3-[2-(3-pyrrolidin-1-yl-propylamino)-pyrimidin-4-ylamino]-phenyl}-2-morpholin-4-yl-isonicotinamide 310063 4-methyl-1-[3-(1,4-oxazinan-4-yl)phenylcarboxamido]-3-[4-(3-pyridylmethoxy)phenylcarboxamido]benzene 310064 N-[3-(6,7-Dimethoxy-quinazolin-4-ylamino)-2-fluoro-phenyl]-benzamide 310067 4-[4-(3,3-Diphenyl-propyl)-[1,4]diazepan-1-ylmethyl]-benzonitrile 310068 3-{1-Hydroxy-3-[4-(4-methanesulfonyl-benzyl)-[1,4]diazepan-1-yl]-1-phenyl-propyl}-phenol 310069 N-{3-[2-(Allyl-methyl-amino)-pyrimidin-4-ylamino]-4-methyl-phenyl}-2-morpholin-4-yl-isonicotinamide 310074 Thiophene-2-carboxylic acid N''-{2-[4-(4-chloro-benzyl)-[1,4]diazepan-1-yl]-acetyl}-hydrazide 310075 N-(2-{[1-(4-Chloro-benzyl)-pyrrolidin-2-ylmethyl]-carbamoyl}-ethyl)-benzamide 310085 1-(3-Amino-phenyl)-3-[4-(4-methanesulfonyl-benzyl)-[1,4]diazepan-1-yl]-1-phenyl-propan-1-ol 310086 1,1-Bis-(3-fluoro-phenyl)-3-[4-(4-methanesulfonyl-benzyl)-[1,4]diazepan-1-yl]-propan-1-ol 310087 Thiophene-2-carboxylic acid N''-(2-{4-[3-hydroxy-3-(3-hydroxy-phenyl)-3-phenyl-propyl]-[1,4]diazepan-1-yl}-acetyl)-hydrazide 310088 N-[5-(3-Dimethylamino-benzoylamino)-2-methyl-phenyl]-2,4-dimethoxy-benzamide 310089 3-Fluoro-N-{4-methyl-3-[4-(pyridin-2-ylmethoxy)-benzoylamino]-phenyl}-5-morpholin-4-yl-benzamide 310090 N-{4-Methyl-3-[4-(pyridin-2-ylmethoxy)-benzoylamino]-phenyl}-3-morpholin-4-yl-5-trifluoromethyl-benzamide 310093 4-Methyl-thiophene-2-carboxylic acid N''-{2-[1-(4-chloro-benzyl)-pyrrolidin-3-ylamino]-acetyl}-hydrazide 310094 N-({[1-(4-Chloro-benzyl)-pyrrolidin-2-ylmethyl]-carbamoyl}-methyl)-3-methyl-benzamide 310095 N-{[1-(4-Chloro-benzyl)-pyrrolidin-3-ylcarbamoyl]-methyl}-benzamide 310096 N-{[1-(4-Chloro-benzyl)-pyrrolidin-3-ylcarbamoyl]-methyl}-3-methyl-benzamide 310097 N-[3-(6,7-Dimethoxy-quinazolin-4-ylamino)-4-methyl-phenyl]-benzamide 310098 N-{4-Methyl-3-[2-(3-morpholin-4-yl-propylamino)-pyrimidin-4-ylamino]-phenyl}-2-morpholin-4-yl-isonicotinamide 310106 N-[5-(3-Dimethylamino-benzoylamino)-2-methyl-phenyl]-3,4,5-trimethoxy-benzamide 310113 3-(4-benzyloxyphenylcarboxamido)-4-methyl-1-[3-(1,4-oxazinan-4-yl)phenylcarboxamido]benzene 310114 N-[5-(6,7-Dimethoxy-quinazolin-4-ylamino)-2-methyl-phenyl]-benzamide 310119 N-(4-Methyl-3-{2-[methyl-(1-methyl-piperidin-4-yl)-amino]-pyrimidin-4-ylamino}-phenyl)-2-morpholin-4-yl-isonicotinamide 310122 N-[5-(3-Dimethylamino-benzoylamino)-2-fluoro-phenyl]-3,4-dimethoxy-benzamide 310124 4-Methyl-thiophene-2-carboxylic acid N''-{2-[4-(4-chloro-benzyl)-[1,4]diazepan-1-yl]-acetyl}-hydrazide 310125 5-Oxo-5-phenyl-pentanoic acid [1-(4-chloro-benzyl)-pyrrolidin-2-ylmethyl]-amide 310128 4-methyl-1-[3-(1,4-oxazinan-4-yl)phenylcarboxamido]-3-[4-(4-pyridylmethoxy)phenylcarboxamido]benzene 310129 N-[2-Chloro-5-(6,7-dimethoxy-quinazolin-4-ylamino)-phenyl]-benzamide 310130 SID26752168 310135 1-(3-Hydroxymethyl-phenyl)-3-[4-(4-methanesulfonyl-benzyl)-[1,4]diazepan-1-yl]-1-phenyl-propan-1-ol 310136 N-{3-[2-(3-Dimethylamino-2,2-dimethyl-propoxy)-pyrimidin-4-ylamino]-4-methyl-phenyl}-2-morpholin-4-yl-isonicotinamide 310138 1-(3-dimethylaminophenylcarboxamido)-3-(4-methoxyphenylcarboxamido)-4-methylbenzene 310139 N-{4-Methyl-3-[4-(pyridin-2-ylmethoxy)-benzoylamino]-phenyl}-2-morpholin-4-yl-isonicotinamide 310142 4-Methyl-thiophene-2-carboxylic acid N''-{2-[1-(3,3-diphenyl-propyl)-pyrrolidin-3-ylamino]-acetyl}-hydrazide 310143 N-({[1-(4-Chloro-benzyl)-pyrrolidin-2-ylmethyl]-carbamoyl}-methyl)-benzamide 310145 N-[4-Chloro-3-(6,7-dimethoxy-quinazolin-4-ylamino)-phenyl]-benzamide 310146 N-[3-(2-Chloro-pyrimidin-4-ylamino)-4-methyl-phenyl]-2-morpholin-4-yl-isonicotinamide 310152 3-[4-(4-Methanesulfonyl-benzyl)-[1,4]diazepan-1-yl]-1-(3-methylamino-phenyl)-1-phenyl-propan-1-ol 310153 1-Methyl-4-[2-(3-naphthalen-2-yl-8-aza-bicyclo[3.2.1]oct-2-en-8-yl)-ethoxy]-1H-indole 310156 N-[4-Chloro-3-(6,7-dimethoxy-quinazolin-4-ylamino)-phenyl]-3-dimethylamino-benzamide 310157 N-{4-Methyl-3-[2-(1-methyl-piperidin-3-ylmethoxy)-pyrimidin-4-ylamino]-phenyl}-2-morpholin-4-yl-isonicotinamide 310174 3-[4-(4-Methanesulfonyl-benzyl)-[1,4]diazepan-1-yl]-1,1-diphenyl-propan-1-ol 310183 1-(3-Fluoro-phenyl)-3-[4-(4-methanesulfonyl-benzyl)-[1,4]diazepan-1-yl]-1-phenyl-propan-1-ol 310184 4-Methyl-thiophene-2-carboxylic acid N''-(2-{2-[(3,3-diphenyl-propylamino)-methyl]-pyrrolidin-1-yl}-acetyl)-hydrazide 310186 1-(3-dimethylaminophenylcarboxamido)-3-(4-ethoxyphenylcarboxamido)-4-methylbenzene 310191 N-(2-{[1-(4-Chloro-benzyl)-piperidin-4-ylmethyl]-carbamoyl}-ethyl)-benzamide 310193 4-methyl-3-[4-(2-methyl-1,3-thiazol-4-ylmethoxy)phenylcarboxamido]-1-[3-(1,4-oxazinan-4-yl)phenylcarboxamido]benzene 310194 N-[2-Chloro-5-(6,7-dimethoxy-quinazolin-4-ylamino)-phenyl]-3-dimethylamino-benzamide 310195 4-[2-(3-Benzo[b]thiophen-3-yl-8-aza-bicyclo[3.2.1]oct-2-en-8-yl)-ethoxy]-1H-indole 310196 N-[2-Chloro-5-(3-dimethylamino-benzoylamino)-phenyl]-3,4-dimethoxy-benzamide 310197 3-Fluoro-N-{4-methyl-3-[4-(pyridin-4-ylmethoxy)-benzoylamino]-phenyl}-5-morpholin-4-yl-benzamide 310200 N-{4-Methyl-3-[2-(1-propyl-piperidin-4-yloxy)-pyrimidin-4-ylamino]-phenyl}-2-morpholin-4-yl-isonicotinamide 310204 N-[3-(6,7-Dimethoxy-quinazolin-4-ylamino)-phenyl]-3-dimethylamino-benzamide 310205 N-{3-[2-(3-Dimethylamino-propoxy)-pyrimidin-4-ylamino]-4-methyl-phenyl}-2-morpholin-4-yl-isonicotinamide 310221 1,1-di(4-hydroxyphenyl)-3-[4-(4-methylsulfonylbenzyl)-1,4-diazepan-1-yl]-1-propanol 310222 3-{1-(3-Fluoro-phenyl)-1-hydroxy-3-[4-(4-methanesulfonyl-benzyl)-[1,4]diazepan-1-yl]-propyl}-phenol 310236 3-[4-(4-Methanesulfonyl-benzyl)-[1,4]diazepan-1-yl]-1-(3-methoxy-phenyl)-1-phenyl-propan-1-ol 310238 N-[5-(3-Dimethylamino-benzoylamino)-2-methyl-phenyl]-3,4-diethoxy-benzamide 310245 4-Methyl-thiophene-2-carboxylic acid N''-{2-[3-(4-chloro-benzylamino)-pyrrolidin-1-yl]-acetyl}-hydrazide 310246 5-Oxo-5-phenyl-pentanoic acid [1-(4-chloro-benzyl)-piperidin-4-ylmethyl]-amide 310247 3-Fluoro-N-{4-methyl-3-[4-(thiazol-4-ylmethoxy)-benzoylamino]-phenyl}-5-morpholin-4-yl-benzamide 310248 N-[3-(6,7-Dimethoxy-quinazolin-4-ylamino)-4-methyl-phenyl]-3-dimethylamino-benzamide 310254 N-(4-methyl-3-(2-(1-methylpiperidin-4-yloxy)pyrimidin-4-ylamino)phenyl)-2-morpholinoisonicotinamide 310269 1,1-Bis-(4-dimethylamino-phenyl)-3-[4-(4-methanesulfonyl-benzyl)-[1,4]diazepan-1-yl]-propan-1-ol 310274 3-[4-(4-Methanesulfonyl-benzyl)-[1,4]diazepan-1-yl]-1-phenyl-1-m-tolyl-propan-1-ol 310277 4-[4-Hydroxy-4-(3-trifluoromethyl-phenyl)-piperidin-1-yl]-2,2-diphenyl-butyric acid methyl ester 310278 N-[2-Bromo-5-(3-dimethylamino-benzoylamino)-phenyl]-3,4-dimethoxy-benzamide 310279 4-methyl-1-[3-(1,4-oxazinan-4-yl)phenylcarboxamido]-3-[4-(1,3-thiazol-4-ylmethoxy)phenylcarboxamido]benzene 310280 N-({[1-(4-Chloro-benzyl)-piperidin-4-ylmethyl]-carbamoyl}-methyl)-benzamide 310282 1-(3,3-Diphenyl-propyl)-1-oxy-4-(3-trifluoromethyl-phenyl)-piperidin-4-ol 310283 4-{3-[3-(3,4-Dichloro-phenyl)-8-aza-bicyclo[3.2.1]oct-2-en-8-yl]-propoxy}-1H-indole 310289 5-Chloro-1H-indole-2-carboxylic acid (4-methyl-piperazin-1-yl)-amide 310292 4-[4-Hydroxy-4-(3-trifluoromethyl-phenyl)-piperidin-1-yl]-2,2-diphenyl-butyric acid 310293 1H-4-indolyl 3-[3-(1H-3-indolyl)-8-azabicyclo[3.2.1]oct-2-en-8-yl]propyl ether 310294 SID47201151 310312 (R)-3-(4-Chloro-phenyl)-1-(1-phenyl-2-pyrrolidin-1-yl-ethyl)-1,3,4,7-tetrahydro-azepin-2-one 310318 3-(4-Methoxy-phenyl)-1-(1-phenyl-2-pyrrolidin-1-yl-ethyl)-1,3,4,7-tetrahydro-azepin-2-one 310324 4-[4-(4-Chloro-3-trifluoromethyl-phenyl)-4-hydroxy-piperidin-1-yl]-2,2-diphenyl-butyric acid methyl ester 310334 5-Chloro-1H-indole-2-carboxylic acid (2-dimethylamino-ethyl)-methyl-amide 310337 4-[4-(4-Chloro-3-trifluoromethyl-phenyl)-4-hydroxy-piperidin-1-yl]-2,2-diphenyl-butyric acid 310346 (S)-1-(1H-Indol-4-yloxy)-3-(3-naphthalen-2-yl-8-aza-bicyclo[3.2.1]oct-2-en-8-yl)-propan-2-ol 310350 (R)-3-(3,4-Dichloro-phenyl)-1-(1-phenyl-2-pyrrolidin-1-yl-ethyl)-1,3,4,7-tetrahydro-azepin-2-one 310351 3-(4-Chloro-phenyl)-1-(1-phenyl-2-pyrrolidin-1-yl-ethyl)-1,3,4,7-tetrahydro-azepin-2-one 310358 1-(1-Phenyl-2-pyrrolidin-1-yl-ethyl)-3-(4-trifluoromethyl-phenyl)-1,3,4,7-tetrahydro-azepin-2-one 310360 4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-2,2-diphenyl-butyric acid methyl ester 310361 1H-4-indolyl 2-[3-(1H-3-indolyl)-8-azabicyclo[3.2.1]oct-2-en-8-yl]ethyl ether 310363 (5-Iodo-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone 310364 5-Chloro-1H-indole-2-carboxylic acid (2-dimethylamino-ethyl)-amide 310376 (5-Chloro-1H-indol-2-yl)-(1-methyl-piperidin-4-yl)-methanol 310383 4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-2,2-diphenyl-butyric acid 310384 4-[3-(3-Naphthalen-2-yl-8-aza-bicyclo[3.2.1]oct-2-en-8-yl)-propoxy]-1H-indole 310387 3-(3,4-Dichloro-phenyl)-1-(1-phenyl-2-pyrrolidin-1-yl-ethyl)-1,3,4,7-tetrahydro-azepin-2-one 310396 (R)-3-(4-Methoxy-phenyl)-1-(1-phenyl-2-pyrrolidin-1-yl-ethyl)-1,3,4,7-tetrahydro-azepin-2-one 310404 3-(4-Methoxy-phenyl)-acrylic acid 2-{(1S,2S)-2-[(S)-hydroxy-((R)-6-oxo-3,6-dihydro-2H-pyran-2-yl)-methyl]-cyclopropyl}-1-methyl-2-oxo-ethyl ester 310412 5-Chloro-1H-benzoimidazole-2-carboxylic acid (2-dimethylamino-ethyl)-amide 310413 5-Chloro-1H-benzoimidazole-2-carboxylic acid (2-dimethylamino-ethyl)-methyl-amide 310431 5-{2-[3-(1H-Indol-2-yl)-8-aza-bicyclo[3.2.1]oct-2-en-8-yl]-ethoxy}-quinoline 310436 (S)-3-(3,4-Dichloro-phenyl)-1-[(S)-2-((S)-3-hydroxy-pyrrolidin-1-yl)-1-phenyl-ethyl]-1,3,4,7-tetrahydro-azepin-2-one 310457 4-Methyl-piperazine-1-carboxylic acid (5-chloro-1H-benzoimidazol-2-yl)-amide 310462 (5-Chloro-1H-indol-2-yl)-(1-methyl-piperidin-4-yl)-methanone 310463 (5-chloro-1H-benzoimidazol-2-yl)(4-methylpiperazin-1-yl)methanone 310464 (Z)-1-((1S,2S)-2-((S)-hydroxy((R)-6-oxo-3,6-dihydro-2H-pyran-2-yl)methyl)cyclopropyl)-1-oxopropan-2-yl 3-(3,4-dihydroxyphenyl)acrylate 310480 8-[2-(3-Naphthalen-2-yl-8-aza-bicyclo[3.2.1]oct-2-en-8-yl)-ethoxy]-quinoline 310491 3-(3,4-Dichloro-phenoxy)-1-(1-phenyl-2-pyrrolidin-1-yl-ethyl)-1,3,4,7-tetrahydro-azepin-2-one 310503 5-[2-(3-Naphthalen-2-yl-8-aza-bicyclo[3.2.1]oct-2-en-8-yl)-ethoxy]-quinoline 310506 3-(4-Methoxy-phenyl)-acrylic acid 2-{(1S,2S)-2-[(S)-hydroxy-((R)-6-oxo-3,6-dihydro-2H-pyran-2-yl)-methyl]-cyclopropyl}-1-methyl-2-oxo-ethyl ester 310514 (S)-1-[3-(3,4-Dichloro-phenyl)-8-aza-bicyclo[3.2.1]oct-2-en-8-yl]-3-(1H-indol-4-yloxy)-propan-2-ol 310523 (S)-3-(3,4-Dichloro-phenyl)-1-((S)-1-phenyl-2-pyrrolidin-1-yl-ethyl)-1,3,4,7-tetrahydro-azepin-2-one 310533 1-(1-Phenyl-2-pyrrolidin-1-yl-ethyl)-3-[3-(pyrrolidine-1-sulfonyl)-phenyl]-1,3,4,7-tetrahydro-azepin-2-one 310544 4-(4-Chloro-phenyl)-1-(3,3-diphenyl-propyl)-piperidin-4-ol 310545 8-[2-(Indan-4-yloxy)-ethyl]-3-naphthalen-2-yl-8-aza-bicyclo[3.2.1]oct-2-ene 310552 2-Amino-3-(4-chloro-phenyl)-1-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-propan-1-one 310558 N-Ethyl-4-[phenyl-(8-pyridin-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-benzamide 310562 N-Ethyl-4-[(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-(1H-tetrazol-5-yl)-methyl]-benzamide 310564 N-Ethyl-4-(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidenemethyl)-benzamide 310565 4-[(3-Acetyl-phenyl)-(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-N-ethyl-benzamide 310568 1N-ethyl-4-{4-carbamoylphenyl[8-(3-furylmethyl)-8-azabicyclo[3.2.1]oct-3-yliden]methyl}benzamide 310569 N-Ethyl-4-[(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-(4-nitro-phenyl)-methyl]-benzamide 310571 N-Ethyl-4-{[3-(1H-tetrazol-5-yl)-phenyl]-[(1S,5R)-8-thiophen-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-(3E)-ylidene]-methyl}-benzamide 310575 4-{Bromo-[(1S,5R)-8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-(3E)-ylidene]-methyl}-N-ethyl-benzamide 310576 4-{Bromo-[(1R,5S)-8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-(3Z)-ylidene]-methyl}-N-ethyl-benzamide 310578 4-((1-methyl-1H-indol-3-yl)methylene)-3-(pyrazin-2-yl)-1H-pyrazol-5(4H)-one 310586 4-(2-Azetidin-2-yl-ethoxy)-7-chloro-2-oxo-3-((S)-3,4,5-trimethyl-phenyl)-1,2-dihydro-quinoline-6-carboxylic acid [1,2,5]thiadiazol-3-ylamide 310587 (R)-2-Amino-3-(4-chloro-phenyl)-1-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-propan-1-one 310599 4-{2-[3-(3,4-Dichloro-phenyl)-8-aza-bicyclo[3.2.1]oct-2-en-8-yl]-ethoxy}-1H-indole 310602 3-Amino-5-[(4-ethylcarbamoyl-phenyl)-(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-benzoic acid 310603 4-[(3,5-Dimethyl-isoxazol-4-yl)-(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-N-ethyl-benzamide 310609 4-[Benzo[1,3]dioxol-5-yl-(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-N-ethyl-benzamide 310610 4-{Cyano-[(1S,5R)-8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-(3E)-ylidene]-methyl}-N-ethyl-benzamide 310612 3-{(4-Ethylcarbamoyl-phenyl)-[(1S,5R)-8-(3-methyl-but-3-enyl)-8-aza-bicyclo[3.2.1]oct-(3Z)-ylidene]-methyl}-benzoic acid 310616 4-{Cyano-[(1R,5S)-8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-(3Z)-ylidene]-methyl}-N-ethyl-benzamide 310628 1-{4-[4-(2-{4-[(R)-(4-chlorophenyl)(phenyl)methyl]piperazin-1-yl}ethoxy)phenyl]but-3-yn-1-yl}-1-hydroxyurea 310630 7-Chloro-2-oxo-4-[2-((R)-6-trifluoromethyl-piperidin-2-yl)-ethoxy]-3-((S)-3,4,5-trimethyl-phenyl)-1,2-dihydro-quinoline-6-carboxylic acid pyrimidin-4-ylamide 310633 7-Chloro-2-oxo-4-(2-piperidin-2-yl-ethoxy)-3-((S)-3,4,5-trimethyl-phenyl)-1,2-dihydro-quinoline-6-carboxylic acid [1,2,5]thiadiazol-3-ylamide 310634 7-Chloro-4-[2-((R)-1-methyl-6-trifluoromethyl-piperidin-2-yl)-ethoxy]-2-oxo-3-((S)-3,4,5-trimethyl-phenyl)-1,2-dihydro-quinoline-6-carboxylic acid pyrimidin-4-ylamide 310635 2-Amino-3-(2-chloro-phenyl)-1-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-propan-1-one 310636 4-[4-Hydroxy-4-(3-trifluoromethyl-phenyl)-piperidin-1-yl]-N,N-dimethyl-2,2-diphenyl-butyramide 310637 4-[2-(3-Naphthalen-2-yl-8-aza-bicyclo[3.2.1]oct-2-en-8-yl)-ethoxy]-1H-indole 310638 2-(4-Chloro-phenyl)-2-methyl-1-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-propan-1-one 310639 1-Amino-cyclopropanecarboxylic acid [(R)-1-(4-chloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-amide 310641 4-[(3-Acetylamino-phenyl)-(8-pyridin-2-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-N-ethyl-benzamide 310649 N-Ethyl-4-[(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-pyridin-3-yl-methyl]-benzamide 310650 4-[(4-Acetyl-phenyl)-(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-N-ethyl-benzamide 310663 N-Ethyl-4-{[3-(1H-tetrazol-5-yl)-phenyl]-[(1R,5S)-8-thiophen-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-(3Z)-ylidene]-methyl}-benzamide 310670 7-Chloro-2-oxo-4-(2-pyrrolidin-2-yl-ethoxy)-3-((S)-3,4,5-trimethyl-phenyl)-1,2-dihydro-quinoline-6-carboxylic acid pyrimidin-4-ylamide 310677 1-{4-[4-(4-{4-[(R)-(4-chlorophenyl)(phenyl)methyl]piperazin-1-yl}butoxy)phenyl]but-3-yn-1-yl}-1-hydroxyurea 310684 7-Chloro-4-(2-morpholin-3-yl-ethoxy)-2-oxo-3-(3,4,5-trimethyl-phenyl)-1,2-dihydro-quinoline-6-carboxylic acid [1,2,5]thiadiazol-3-ylamide 310685 2-Aminomethyl-3-(4-chloro-phenyl)-1-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-propan-1-one 310694 N-Ethyl-4-[(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-pyrazin-2-yl-methyl]-benzamide 310695 N-Ethyl-4-{(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-[3-(1H-tetrazol-5-yl)-phenyl]-methyl}-benzamide 310696 7-Chloro-4-(2-cyclopentyl-ethoxy)-2-oxo-3-(3,4,5-trimethyl-phenyl)-1,2-dihydro-quinoline-6-carboxylic acid [1,2,5]thiadiazol-3-ylamide 310700 N-Ethyl-4-[(4-fluoro-phenyl)-(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-benzamide 310702 3-Amino-propionic acid 1-(4-chloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl ester 310711 4-[Benzo[1,3]dioxol-5-yl-(8-thiophen-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-N-ethyl-benzamide 310712 3-{3-[(4-Ethylcarbamoyl-phenyl)-(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-phenyl}-propionic acid 310722 1-{4-[4-(3-{4-[bis(4-fluorophenyl)methyl]piperazin-1-yl}propoxy)phenyl]but-3-yn-1-yl}-1-hydroxyurea 310724 1-{4-[4-(3-{4-[(R)-(4-chlorophenyl)(phenyl)methyl]piperazin-1-yl}propoxy)phenyl]but-3-yn-1-yl}-1-hydroxyurea 310726 7-Chloro-4-(2-[1,3]dioxolan-2-yl-ethoxy)-2-oxo-3-(3,4,5-trimethyl-phenyl)-1,2-dihydro-quinoline-6-carboxylic acid [1,2,5]thiadiazol-3-ylamide 310729 4-[2-(1-Aza-bicyclo[2.2.2]oct-2-yl)-ethoxy]-7-chloro-2-oxo-3-(3,4,5-trimethyl-phenyl)-1,2-dihydro-quinoline-6-carboxylic acid [1,2,5]thiadiazol-3-ylamide 310730 3-Amino-3-(4-chloro-phenyl)-1-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-propan-1-one 310732 2,2,2-Trifluoro-ethanesulfonic acid [(R)-1-(4-chloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-amide 310746 3-[(4-Ethylcarbamoyl-phenyl)-(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-5-nitro-benzoic acid 310747 N-Ethyl-4-[(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-(1-hydroxy-1,4-dihydro-pyridin-3-yl)-methyl]-benzamide 310751 N,N-Diethyl-4-[(8-phenethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-phenyl-methyl]-benzamide 310754 N-Ethyl-4-[(3-fluoro-phenyl)-(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-benzamide 310759 4-[(4-Ethylcarbamoyl-phenyl)-(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-benzoic acid 310760 N-Ethyl-4-[(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-(1-methoxy-1,4-dihydro-pyridin-3-yl)-methyl]-benzamide 310768 4-[(2,6-Dimethyl-phenyl)-(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-N-ethyl-benzamide 310772 1-{4-[4-(2-{4-[bis(4-fluorophenyl)methyl]piperazin-1-yl}ethoxy)phenyl]but-3-yn-1-yl}-1-hydroxyurea 310779 7-Chloro-2-oxo-4-[2-(tetrahydro-furan-2-yl)-ethoxy]-3-(3,4,5-trimethyl-phenyl)-1,2-dihydro-quinoline-6-carboxylic acid pyrimidin-4-ylamide 310780 3-(4-Chloro-phenyl)-1-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-propan-1-one 310785 1-(4-{4-[2-(4-{13-chloro-4-azatricyclo[9.4.0.0^{3,8}]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-ylidene}piperidin-1-yl)ethoxy]phenyl}but-3-yn-1-yl)-1-hydroxyurea 310786 4-[Cyano-(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-N-ethyl-benzamide 310787 4-[(3-Amino-phenyl)-(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-N-ethyl-benzamide 310793 N-Ethyl-4-[(8-phenethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-phenyl-methyl]-benzamide 310794 3-[(4-Ethylcarbamoyl-phenyl)-(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-benzoic acid 310795 7-Chloro-4-(2-oxetan-2-yl-ethoxy)-2-oxo-3-((R)-3,4,5-trimethyl-phenyl)-1,2-dihydro-quinoline-6-carboxylic acid [1,2,5]thiadiazol-3-ylamide 310797 N-Ethyl-4-[(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-quinolin-3-yl-methyl]-benzamide 310801 4-[Bromo-(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-N-ethyl-benzamide 310802 4-[(4-Dimethylamino-phenyl)-(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-N-ethyl-benzamide 310819 N-Ethyl-4-[(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-pyrimidin-5-yl-methyl]-benzamide 310820 N-Ethyl-4-[(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-(3-hydroxymethyl-phenyl)-methyl]-benzamide 310822 N-Ethyl-4-{(4-hydroxymethyl-phenyl)-[(1S,5R)-8-thiophen-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-(3Z)-ylidene]-methyl}-benzamide 310826 1N,1N-dimethyl-4-{4-ethylcarbamoylphenyl[8-(2-pyridylmethyl)-(1R,5S)-8-azabicyclo[3.2.1]oct-3-yliden]methyl}benzamide 310837 4-{(3-Acetyl-phenyl)-[8-(3-methyl-but-3-enyl)-8-aza-bicyclo[3.2.1]oct-3-ylidene]-methyl}-N-ethyl-benzamide 310843 2-Amino-4-methyl-pentanoic acid [(R)-1-(4-chloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-amide 310844 N-Ethyl-4-[(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-pyridin-4-yl-methyl]-benzamide 310845 4-[(3-Cyano-phenyl)-(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-N-ethyl-benzamide 310850 3-{(4-Ethylcarbamoyl-phenyl)-[(1R,5S)-8-(3-methyl-but-3-enyl)-8-aza-bicyclo[3.2.1]oct-(3E)-ylidene]-methyl}-benzoic acid 310852 7-Chloro-2-oxo-4-[2-(5-oxo-pyrrolidin-2-yl)-ethoxy]-3-((R)-3,4,5-trimethyl-phenyl)-1,2-dihydro-quinoline-6-carboxylic acid [1,2,5]thiadiazol-3-ylamide 310854 N-Ethyl-4-{furan-2-yl-[8-(3-methyl-but-3-enyl)-8-aza-bicyclo[3.2.1]oct-3-ylidene]-methyl}-benzamide 310857 4-[(3-Aminomethyl-phenyl)-(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-N-ethyl-benzamide 310858 1N,1N-dimethyl-4-{4-ethylcarbamoylphenyl[8-(2-pyridylmethyl)-(1R,5S)-8-azabicyclo[3.2.1]oct-3-yliden]methyl}benzamide 310859 4-(2R)-[3-aminopropionylamino]-3-(4-chlorophenyl)-propionyl-1-2-[2-thienyl)ethylaminomethyl]phenyl piperazine 310861 N-Ethyl-4-[(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-(4-methanesulfonyl-phenyl)-methyl]-benzamide 310862 4-[(4-Acetylamino-phenyl)-(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-N-ethyl-benzamide 310870 4-{(3-Acetyl-phenyl)-[(1S,5R)-8-(3-methyl-but-3-enyl)-8-aza-bicyclo[3.2.1]oct-(3Z)-ylidene]-methyl}-N-ethyl-benzamide 310886 1-(4-{4-[3-(4-{13-chloro-4-azatricyclo[9.4.0.0^{3,8}]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-ylidene}piperidin-1-yl)propoxy]phenyl}but-3-yn-1-yl)-1-hydroxyurea 310887 1-(4-{4-[4-(4-{13-chloro-4-azatricyclo[9.4.0.0^{3,8}]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-ylidene}piperidin-1-yl)butoxy]phenyl}but-3-yn-1-yl)-1-hydroxyurea 310890 2-Amino-2-(4-chloro-phenyl)-1-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethanone 310891 2-Amino-N-[(R)-1-(4-chloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-2-methyl-propionamide 310892 4-{(3-Acetylamino-phenyl)-[8-(1H-imidazol-4-ylmethyl)-8-aza-bicyclo[3.2.1]oct-3-ylidene]-methyl}-N-ethyl-benzamide 310893 N-Ethyl-4-[(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-pyridin-2-yl-methyl]-benzamide 310894 7-Chloro-2-oxo-4-[2-(4-oxo-azetidin-2-yl)-ethoxy]-3-((S)-3,4,5-trimethyl-phenyl)-1,2-dihydro-quinoline-6-carboxylic acid [1,2,5]thiadiazol-3-ylamide 310899 N-Ethyl-4-[(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-(4-hydroxymethyl-phenyl)-methyl]-benzamide 310900 N-Ethyl-4-{(4-hydroxymethyl-phenyl)-[(1R,5S)-8-thiophen-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-(3E)-ylidene]-methyl}-benzamide 310901 N-[(R)-1-(4-Chloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-2-dimethylamino-acetamide 310902 N-Ethyl-4-[pyrazin-2-yl-(8-thiophen-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-benzamide 310903 N-Ethyl-4-[(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-(4-sulfamoyl-phenyl)-methyl]-benzamide 310911 4-[(3-Acetylamino-phenyl)-(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-N-ethyl-benzamide 310912 4-{(3-Acetyl-phenyl)-[(1R,5S)-8-(3-methyl-but-3-enyl)-8-aza-bicyclo[3.2.1]oct-(3E)-ylidene]-methyl}-N-ethyl-benzamide 310922 N-[(R)-1-(4-Chloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-2-pyrrolidin-2-yl-acetamide 310932 7-Chloro-4-[2-(1-methyl-5-oxo-pyrrolidin-2-yl)-ethoxy]-2-oxo-3-((R)-3,4,5-trimethyl-phenyl)-1,2-dihydro-quinoline-6-carboxylic acid [1,2,5]thiadiazol-3-ylamide 310934 3-{3-[(4-Ethylcarbamoyl-phenyl)-phenyl-methylene]-8-aza-bicyclo[3.2.1]oct-8-ylmethyl}-benzoic acid 310938 N-Ethyl-4-[pyridin-2-yl-(8-thiophen-2-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-methyl]-benzamide 310939 4-Amino-N-[(R)-1-(4-chloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-butyramide 310940 1N,1N-dimethyl-4-{4-ethylcarbamoylphenyl[8-(3-furylmethyl)-8-azabicyclo[3.2.1]oct-3-yliden]methyl}benzamide 310941 N-Ethyl-4-[(8-furan-3-ylmethyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-(4-hydroxy-3-methoxy-phenyl)-methyl]-benzamide 311061 1-{(E)-4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-but-2-enyl}-pyrrolidine-2,5-dione 311070 (S)-methyl 3-(3-(4-(3-acetamidophenyl)piperidin-1-yl)propylcarbamoyl)-4-(3,4-difluorophenyl)-6-methoxy-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxylate 311086 4-Fluoro-N-[3-(1-methyl-piperidin-4-yl)-2,3-dihydro-1H-indol-5-yl]-benzamide 311100 1-{4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-cyclohexyl}-pyrrolidine-2,5-dione 311102 2-{(Z)-4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-but-2-enyl}-isoindole-1,3-dione 311131 4-Fluoro-N-[3-(1-methyl-piperidin-4-yl)-benzo[d]isoxazol-5-yl]-benzamide 311132 4-Fluoro-N-[1-(1-methyl-piperidin-4-yl)-1H-indazol-6-yl]-benzamide 311143 1-{(Z)-4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-but-2-enyl}-pyrrolidine-2,5-dione 311144 1-{2-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-benzyl}-pyrrolidine-2,5-dione 311153 2-{(E)-4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-but-2-enyl}-isoindole-1,3-dione 311175 4-Fluoro-N-[1-(1-methyl-piperidin-4-yl)-2,3-dihydro-1H-indol-6-yl]-benzamide 311176 4-Fluoro-N-[4-(1-methyl-piperidin-4-yl)-3,4-dihydro-2H-benzo[1,4]oxazin-6-yl]-benzamide 311185 4-Fluoro-N-[3-(1-methyl-piperidin-4-yl)-1H-indazol-5-yl]-benzamide 311190 2-{2-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-benzyl}-isoindole-1,3-dione 311213 4-Fluoro-N-[1-(1-methyl-piperidin-4-yl)-1H-indol-6-yl]-benzamide 311252 1-[1-(2,2-Diphenyl-ethyl)-6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl]-2,2,2-trifluoro-ethanone 311263 1-[6-Bromo-1-(2,2-diphenyl-ethyl)-7-methoxy-3,4-dihydro-1H-isoquinolin-2-yl]-ethanone 311264 Pyrrolidine-2-carboxylic acid [(R)-1-(4-chloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-amide 311292 2-{4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-cyclohexyl}-isoindole-1,3-dione 311298 [1-(2,2-Diphenyl-ethyl)-6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl]-phenyl-methanone 311302 2,4-Difluoro-N-[3-(1-methyl-piperidin-4-yl)-benzo[d]isoxazol-5-yl]-benzamide 311306 1-[1-(2,2-Diphenyl-ethyl)-6-fluoro-3,4-dihydro-1H-isoquinolin-2-yl]-ethanone 311309 2-Chloro-4-fluoro-N-[3-(1-methyl-piperidin-4-yl)-benzo[d]isoxazol-5-yl]-benzamide 311312 Azetidine-2-carboxylic acid [(R)-1-(4-chloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-amide 311325 1-[1-(2,2-Diphenyl-ethyl)-6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl]-butan-1-one 311326 1-[1-(2,2-Diphenyl-ethyl)-7-methoxy-3,4-dihydro-1H-isoquinolin-2-yl]-ethanone 311335 1-[1-(2,2-Diphenyl-ethyl)-6,8-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl]-ethanone 311344 3-Amino-N-[(R)-1-(4-chloro-benzyl)-2-oxo-2-(4-{2-[1-(2-thiophen-2-yl-ethylamino)-propyl]-phenyl}-piperazin-1-yl)-ethyl]-propionamide 311351 2,4,6-Trifluoro-N-[3-(1-methyl-piperidin-4-yl)-2,3-dihydro-1H-benzoimidazol-5-yl]-benzamide 311361 2-Chloro-4-fluoro-N-[3-(1-methyl-piperidin-4-yl)-2,3-dihydro-1H-benzoimidazol-5-yl]-benzamide 311377 1-[1-(2,2-Diphenyl-ethyl)-6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl]-hexan-1-one 311382 1-(2,2-Diphenyl-ethyl)-6,7-dimethoxy-3,4-dihydro-1H-isoquinoline-2-carboxylic acid methyl ester 311393 3-Amino-N-{(R)-1-(4-chloro-benzyl)-2-[4-(2-{[methyl-(2-thiophen-2-yl-ethyl)-amino]-methyl}-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-propionamide 311397 Piperidine-4-carboxylic acid [(R)-1-(4-chloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-amide 311439 1-(2,2-Diphenyl-ethyl)-6,7-dimethoxy-3,4-dihydro-1H-isoquinoline-2-carboxylic acid methylamide 311454 Cyclohexyl-[1-(2,2-diphenyl-ethyl)-6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl]-methanone 311458 Piperidine-3-carboxylic acid [(R)-1-(4-chloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-amide 311473 N-[(R)-1-(4-Chloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-nicotinamide 311508 1-(2,2-Diphenyl-ethyl)-6,7-dimethoxy-3,4-dihydro-1H-isoquinoline-2-carboxylic acid amide 311520 Cyclobutyl-[1-(2,2-diphenyl-ethyl)-6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl]-methanone 311523 Piperidine-2-carboxylic acid [(R)-1-(4-chloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-amide 311528 4-(2R)-[2-methoxyacetamido]3-(4-chlorophenyl)propionyl-1-2-[(2-thienyl)ethylaminomethyl]phenyl piperazine 311559 Cyclobutyl-(6,7-dimethoxy-1-phenethyl-3,4-dihydro-1H-isoquinolin-2-yl)-methanone 311560 Cyclohexyl-(6,7-dimethoxy-1-phenethyl-3,4-dihydro-1H-isoquinolin-2-yl)-methanone 311579 3-Amino-N-[(R)-2-(4-{2-[1-(2-amino-phenylamino)-ethyl]-phenyl}-piperazin-1-yl)-1-(4-chloro-benzyl)-2-oxo-ethyl]-propionamide 311580 3-Amino-N-{(R)-1-(4-chloro-benzyl)-2-[4-(2-{1-[2-(naphthalen-1-ylamino)-ethylamino]-ethyl}-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-propionamide 311581 3-Amino-N-[(R)-1-(4-chloro-benzyl)-2-oxo-2-(4-{2-[1-(4-phenyl-piperazin-1-yl)-ethyl]-phenyl}-piperazin-1-yl)-ethyl]-propionamide 311587 1-[1-(2,2-Diphenyl-ethyl)-6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl]-heptan-1-one 311588 1-(6,7-Dimethoxy-1-phenethyl-3,4-dihydro-1H-isoquinolin-2-yl)-ethanone 311597 3-Amino-N-[(R)-2-(4-{2-[1-(2-amino-benzylamino)-ethyl]-phenyl}-piperazin-1-yl)-1-(4-chloro-benzyl)-2-oxo-ethyl]-propionamide 311635 [1-(2,2-Diphenyl-ethyl)-6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl]-(4-trifluoromethyl-phenyl)-methanone 311641 3-Amino-N-{(R)-1-(4-chloro-benzyl)-2-[4-(2-{1-[(furan-2-ylmethyl)-amino]-ethyl}-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-propionamide 311661 (6,7-Dimethoxy-1-phenethyl-3,4-dihydro-1H-isoquinolin-2-yl)-(4-trifluoromethyl-phenyl)-methanone 311662 6,7-Dimethoxy-1-phenethyl-3,4-dihydro-1H-isoquinoline-2-carbaldehyde 311663 3-Amino-N-[(R)-1-(4-chloro-benzyl)-2-oxo-2-(4-{2-[1-(2-thiophen-2-yl-ethylamino)-ethyl]-phenyl}-piperazin-1-yl)-ethyl]-propionamide 311673 3-Amino-N-[(R)-1-(4-chloro-benzyl)-2-(4-{2-[1-(4-methyl-piperazin-1-yl)-ethyl]-phenyl}-piperazin-1-yl)-2-oxo-ethyl]-propionamide 311687 4-[2-(2-Benzyl-phenoxy)-ethyl]-2-methyl-morpholine 311692 2-{2-[2-(5-Bromo-2-methoxy-phenyl)-ethyl]-3-fluoro-phenyl}-1H-imidazole 311693 2-{2-[2-(5-Bromo-2-methoxy-phenyl)-ethyl]-3-chloro-phenyl}-5-methyl-1H-imidazole 311694 1-[2-(2-Benzyl-phenoxy)-ethyl]-4-phenyl-piperazine 311704 5-(5,6-Dimethyl-pyrrolo[2,1-f][1,2,4]triazin-4-ylamino)-2-methyl-phenol 311710 1-(2,2-Diphenyl-ethyl)-6,7-dimethoxy-3,4-dihydro-1H-isoquinoline-2-carbaldehyde 311711 3-Imidazo[1,2-a]pyridin-3-yl-4-[9-methyl-2-(piperidine-1-carbonyl)-1,2,3,4-tetrahydro-[1,4]diazepino[6,7,1-hi]indol-7-yl]-pyrrole-2,5-dione 311712 4-[(N-Cyclohexyl-3,5-dimethyl-piperidine-1-carboximidoyl)-amino]-N-[2-(2,4-dichloro-phenyl)-ethyl]-benzamide 311714 [(S)-5-(4-Methoxy-phenyl)-1,2,3,4-tetrahydro-naphthalen-2-yl]-dipropyl-amine 311715 3-(9-fluoro-2-(piperidine-1-carbonyl)-1,2,3,4-tetrahydro-[1,4]diazepino[6,7,1-hi]indol-7-yl)-4-(H-imidazo[1,2-a]pyridin-3-yl)-1H-pyrrole-2,5-dione 311716 1-[1-(2,2-Diphenyl-ethyl)-6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl]-propan-1-one 311718 2-benzyl-8-(2-(1-(4-(4,5-dihydro-1H-imidazol-2-yl)benzyl)piperidin-4-yl)ethoxy)-2,3,4,5-tetrahydro-1H-benzo[c]azepin-1-one 311723 1-[1-(2,2-Diphenyl-ethyl)-6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl]-ethanone 311728 (+/-)-1-(1-(4-fluorophenyl)-2-{4-[4-(2-methoxy-1-naphthyl)butyl]piperazin-1-yl}ethyl)-4-methylpiperazine 311729 3-Amino-N-[(R)-1-(4-chloro-benzyl)-2-oxo-2-(4-{2-[1-(2-piperidin-1-yl-ethylamino)-ethyl]-phenyl}-piperazin-1-yl)-ethyl]-propionamide 311733 2-Methyl-5-(6-methyl-pyrrolo[2,1-f][1,2,4]triazin-4-ylamino)-phenol 311738 2-Methyl-5-(7-methyl-pyrrolo[2,1-f][1,2,4]triazin-4-ylamino)-phenol 311739 4-[(N-Cyclohexyl-2,6-dimethyl-morpholine-4-carboximidoyl)-amino]-N-[2-(2,4-dichloro-phenyl)-ethyl]-benzamide 311741 1-[1-(2,2-Diphenyl-ethyl)-6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl]-ethanone 311748 6,7-Dimethoxy-1-phenethyl-3,4-dihydro-1H-isoquinoline-2-carboxylic acid amide 311749 1-[1-(2,2-Diphenyl-ethyl)-3,4-dihydro-1H-isoquinolin-2-yl]-ethanone 311757 3-Amino-N-[(R)-2-(4-{2-[1-((1R,2R)-2-amino-cyclohexylamino)-ethyl]-phenyl}-piperazin-1-yl)-1-(4-chloro-benzyl)-2-oxo-ethyl]-propionamide 311772 1-[3-(2-Benzyl-phenoxy)-propyl]-pyrrolidine 311773 (2-Benzyl-phenyl)-(2-pyrrolidin-1-yl-ethyl)-amine 311791 (S)-5-phenyl-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine 311792 [(S)-5-(2-Methoxy-phenyl)-1,2,3,4-tetrahydro-naphthalen-2-yl]-dipropyl-amine 311794 4-[(N-Cyclohexyl-3-oxo-piperazine-1-carboximidoyl)-amino]-N-[2-(2,4-dichloro-phenyl)-ethyl]-benzamide 311805 4-benzyl-N-(4-(2-(diisopropylamino)ethoxy)-3-methoxyphenyl)benzamide 311809 2-(2,4-Dichloro-phenoxy)-N-[2-(4-ethyl-piperazin-1-yl)-4-methyl-quinolin-6-yl]-propionamide 311817 3-(3-Phenyl-propyl)-1,2,3,4,5,6-hexahydro-benzo[f]isoquinoline 311820 4-(N''''-Cyclohexyl-N'',N''-dipropyl-guanidino)-N-[2-(2,4-dichloro-phenyl)-ethyl]-benzamide 311826 3-(4-Phenyl-butyl)-1,2,3,4,5,6-hexahydro-benzo[f]isoquinoline 311832 [(R)-8-(4-Methoxy-phenyl)-chroman-3-yl]-dipropyl-amine 311833 (2R,3R,4S,5R)-2-{6-Amino-2-[(S)-2-(4-bromo-phenyl)-1-hydroxymethyl-ethylamino]-purin-9-yl}-5-(2-ethyl-2H-tetrazol-5-yl)-tetrahydro-furan-3,4-diol 311835 3-Ethyl-1,2,3,4,5,6-hexahydro-benzo[f]isoquinoline 311836 3-Propyl-1,2,3,4,5,6-hexahydro-benzo[f]isoquinoline 311841 4-(N''-Cyclohexyl-N''''-pyrrolidin-3-yl-guanidino)-N-[2-(2,4-dichloro-phenyl)-ethyl]-benzamide 311843 N-[2-(2,4-Dichloro-phenyl)-ethyl]-4-(N'',N''''-dicyclohexyl-N''-methyl-guanidino)-benzamide 311846 2-(4-Chloro-phenoxy)-N-[2-(4-ethyl-piperazin-1-yl)-4-methyl-quinolin-6-yl]-acetamide 311855 3-Phenethyl-1,2,3,4,5,6-hexahydro-benzo[f]isoquinoline 311860 [(R)-8-(2-Methoxy-phenyl)-chroman-3-yl]-dipropyl-amine 311862 (2R,3R,4S,5R)-2-{6-Amino-2-[(S)-2-(4-chloro-phenyl)-1-hydroxymethyl-ethylamino]-purin-9-yl}-5-(2-ethyl-2H-tetrazol-5-yl)-tetrahydro-furan-3,4-diol 311866 [(S)-8-(2-Methoxy-phenyl)-chroman-3-yl]-dipropyl-amine 311869 4-[N''-(2-Amino-2-methyl-propyl)-N''''-cyclohexyl-guanidino]-N-[2-(2,4-dichloro-phenyl)-ethyl]-benzamide 311874 N-[2-(4-Ethyl-piperazin-1-yl)-4-methyl-quinolin-6-yl]-2-(pyridin-4-ylsulfanyl)-acetamide 311875 2-(2,4-Dichloro-phenoxy)-N-[4-methyl-2-(4-methyl-piperazin-1-yl)-quinolin-6-yl]-acetamide 311876 4-[(N-Cyclohexyl-2-methyl-3-oxo-piperazine-1-carboximidoyl)-amino]-N-[2-(2,4-dichloro-phenyl)-ethyl]-benzamide 311897 [(S)-5-(2,6-Dimethoxy-phenyl)-1,2,3,4-tetrahydro-naphthalen-2-yl]-dimethyl-amine 311898 (R)-8-phenyl-N,N-dipropylchroman-3-amine 311899 (2R,3R,4S,5R)-2-(6-amino-2-((S)-1-hydroxy-3-phenylpropan-2-ylamino)-9H-purin-9-yl)-5-(2-ethyl-2H-tetrazol-5-yl)tetrahydrofuran-3,4-diol 311900 (3-Chloro-4-fluoro-phenyl)-pyrrolo[2,1-f][1,2,4]triazin-4-yl-amine 311906 N-[2-(4-Ethyl-piperazin-1-yl)-4-methyl-quinolin-6-yl]-3-(4-methoxy-phenyl)-propionamide 311907 3-Pentyl-1,2,3,4,5,6-hexahydro-benzo[f]isoquinoline 311916 4-[N''-Cyclohexyl-N''''-(3,5-difluoro-benzyl)-guanidino]-N-[2-(2,4-dichloro-phenyl)-ethyl]-benzamide 311921 [(S)-5-(2,6-Dimethoxy-phenyl)-1,2,3,4-tetrahydro-naphthalen-2-yl]-dipropyl-amine 311925 {[2,2-Diphenyl-5-(4-phenyl-piperidin-1-yl)-pentylcarbamoyl]-methyl}-carbamic acid benzyl ester 311926 (S)-5-(2,6-Dimethoxy-phenyl)-1,2,3,4-tetrahydro-naphthalen-2-ylamine 311929 (3-Chloro-4-fluoro-phenyl)-(7-methyl-pyrrolo[2,1-f][1,2,4]triazin-4-yl)-amine 311930 4-[((S)-N-(R)-Cyclohexyl-2,5-dimethyl-piperazine-1-carboximidoyl)-amino]-N-[2-(2,4-dichloro-phenyl)-ethyl]-benzamide 311932 N-[2-(4-Ethyl-piperazin-1-yl)-4-methyl-quinolin-6-yl]-2-m-tolyloxy-acetamide 311934 [2-(2-Benzyl-phenoxy)-ethyl]-dimethyl-amine 311955 1-[2-(2-Benzyl-phenoxy)-ethyl]-piperidine 311956 4-[2-(2-Benzyl-phenoxy)-ethyl]-morpholine 311959 (2R,3R,4S,5R)-2-{6-Amino-2-[(S)-1-hydroxymethyl-2-(4-nitro-phenyl)-ethylamino]-purin-9-yl}-5-(2-ethyl-2H-tetrazol-5-yl)-tetrahydro-furan-3,4-diol 311961 1-(4-chlorophenyl)-4-(4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl)butan-1-one 311964 4-(4-Chloro-phenoxy)-1-{2-[(R)-1-(3H-indene-5-sulfonyl)-pyrrolidin-2-yl]-ethyl}-piperidine 311965 4-[(N-Cyclohexyl-4-pyrrolidin-1-yl-piperidine-1-carboximidoyl)-amino]-N-[2-(2,4-dichloro-phenyl)-ethyl]-benzamide 311969 3-(4-Methoxy-phenyl)-N-[4-methyl-2-(4-methyl-piperazin-1-yl)-quinolin-6-yl]-propionamide 311973 3-Butyl-1,2,3,4,5,6-hexahydro-benzo[f]isoquinoline 311974 N-(3-chloro-4-fluorophenyl)-5-methylpyrrolo[1,2-f][1,2,4]triazin-4-amine 311980 Phenyl-[2-(2-pyrrolidin-1-yl-ethoxy)-phenyl]-methanone 311981 Phenyl-[2-(2-pyrrolidin-1-yl-ethoxy)-phenyl]-methanol 311991 (2R,3R,4S,5R)-2-{6-Amino-2-[(S)-1-hydroxymethyl-2-(4-hydroxy-phenyl)-ethylamino]-purin-9-yl}-5-(2-ethyl-2H-tetrazol-5-yl)-tetrahydro-furan-3,4-diol 312000 4-[(4-Amino-N-cyclohexyl-piperidine-1-carboximidoyl)-amino]-N-[2-(2,4-dichloro-phenyl)-ethyl]-benzamide 312002 [2-(2-Benzyl-phenoxy)-ethyl]-diethyl-amine 312003 1-[2-(2-Benzyl-phenoxy)-ethyl]-pyrrolidine 312009 2-(2,4-Dichloro-phenoxy)-N-[4-methyl-2-(4-methyl-piperazin-1-yl)-quinolin-6-yl]-propionamide 312018 6-Methoxy-12-methyl-9-oxa-12-aza-tricyclo[13.4.0.0*3,8*]nonadeca-1(15),3,5,7,16,18-hexaene 312019 12-Methyl-9-oxa-12-aza-tricyclo[13.4.0.0*3,8*]nonadeca-1(15),3,5,7,16,18-hexaen-6-ol 312022 7-(4-Imidazo[1,2-a]pyridin-3-yl-2,5-dioxo-2,5-dihydro-1H-pyrrol-3-yl)-3,4-dihydro-1H-[1,4]diazepino[6,7,1-hi]indole-2-carboxylic acid isopropyl ester 312024 (2R,3R,4S,5R)-2-{6-Amino-2-[(S)-1-hydroxymethyl-2-(4-methoxy-phenyl)-ethylamino]-purin-9-yl}-5-(2-ethyl-2H-tetrazol-5-yl)-tetrahydro-furan-3,4-diol 312038 4-[(N-Cyclohexyl-3-methylamino-pyrrolidine-1-carboximidoyl)-amino]-N-[2-(2,4-dichloro-phenyl)-ethyl]-benzamide 312043 (3-Chloro-4-fluoro-phenyl)-(6-methyl-pyrrolo[2,1-f][1,2,4]triazin-4-yl)-amine 312048 N-[2-(3-Methoxy-dibenzo[b,f]azepin-5-yl)-ethyl]-acetamide 312051 2-Furan-2-yl-5-[4-(2-methoxy-benzyl)-piperazin-1-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312061 2-Furan-2-yl-5-[4-(5-methyl-3H-imidazol-4-ylmethyl)-piperazin-1-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312063 difluoro(2-{[(2Z)-1-methyl-5-(2-{[5-({4-[4-(2-oxo-2-{10-oxo-2,4,9-triazatricyclo[9.4.0.0^{3,8}]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}ethyl)piperazin-1-yl]butyl}carbamoyl)pentyl]carbamoyl}ethyl)-2H-pyrrol-1-ium-2-ylidene]methyl}-5-(thiophen-2-yl)-1H-pyrrol-1-yl)boranuide 312066 2-[6-(diethylamino)-3-(diethyliminiumyl)-3H-xanthen-9-yl]-5-[methyl(5-{[2-(2-{2-[4-(2-oxo-2-{10-oxo-2,4,9-triazatricyclo[9.4.0.0^{3,8}]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}ethyl)piperazin-1-yl]ethoxy}ethoxy)ethyl]carbamoyl}pentyl)sulfamoyl]benzene-1-sulfonate 312085 5-Phenyl-1H-pyrrole-2-carboxylic acid (1-tert-butylcarbamoyl-ethyl)-(3-diethylamino-propyl)-amide 312090 5-[4-(3-Chloro-1-methyl-1H-pyrazol-4-ylmethyl)-piperazin-1-yl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312095 2-Furan-2-yl-5-[4-(3-phenyl-propyl)-piperazin-1-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312105 2-Furan-2-yl-5-[4-(2-methyl-1H-imidazol-4-ylmethyl)-piperazin-1-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312129 5-Phenyl-1H-pyrrole-2-carboxylic acid [cyclohexylcarbamoyl-(4-hydroxy-phenyl)-methyl]-(3-diethylamino-propyl)-amide 312131 2-Methyl-5-(pyrrolo[2,1-f][1,2,4]triazin-4-ylamino)-phenol 312132 2-Methyl-5-(5-methyl-pyrrolo[2,1-f][1,2,4]triazin-4-ylamino)-phenol 312135 4-[(N-Cyclohexyl-3,5-dimethyl-piperazine-1-carboximidoyl)-amino]-N-[2-(2,4-dichloro-phenyl)-ethyl]-benzamide 312136 Naphthalene-2-carboxylic acid [4-(1,4,5,6-tetrahydro-2H-benzo[f]isoquinolin-3-yl)-butyl]-amide 312137 N-(2-Dibenzo[b,f]azepin-5-yl-2-oxo-ethyl)-acetamide 312146 5-[4-(4-Chloro-benzyl)-piperazin-1-yl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312150 5-(4-((5-chloro-1-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)methyl)piperazin-1-yl)-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-amine 312170 N-(2-Dibenzo[b,f]azepin-5-yl-ethyl)-acetamide 312173 5-Phenyl-1H-pyrrole-2-carboxylic acid (1-cyclohexylcarbamoyl-pentyl)-(3-diethylamino-propyl)-amide 312174 2-Furan-2-yl-5-(4-pyridin-4-ylmethyl-piperazin-1-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312175 2-Furan-2-yl-5-[4-(2-methyl-pyridin-3-ylmethyl)-piperazin-1-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312180 2-Furan-2-yl-5-(4-quinolin-3-ylmethyl-piperazin-1-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312193 5-Phenyl-1H-pyrrole-2-carboxylic acid (1-cyclohexylcarbamoyl-ethyl)-(3-diethylamino-propyl)-amide 312194 2-Furan-2-yl-5-[4-(2,3,6-trifluoro-benzyl)-piperazin-1-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312206 5-[4-(3,5-Dichloro-pyridin-4-ylmethyl)-piperazin-1-yl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312224 5-Phenyl-1H-pyrrole-2-carboxylic acid [cyclohexylcarbamoyl-(4-fluoro-phenyl)-methyl]-(3-diethylamino-propyl)-amide 312225 5-Phenyl-1H-pyrrole-2-carboxylic acid (cyclohexylcarbamoyl-pyridin-4-yl-methyl)-(3-diethylamino-propyl)-amide 312226 5-[4-(2,6-Dichloro-benzyl)-piperazin-1-yl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312231 5-Phenyl-1H-pyrrole-2-carboxylic acid (1-cyclohexylcarbamoyl-butyl)-(3-diethylamino-propyl)-amide 312232 2-Furan-2-yl-5-(4-pyridin-2-ylmethyl-piperazin-1-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312233 2-Furan-2-yl-5-(4-pyridin-3-ylmethyl-piperazin-1-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312239 5-[4-(6-Chloro-2,3-difluoro-benzyl)-piperazin-1-yl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312240 2-Furan-2-yl-5-(4-quinolin-4-ylmethyl-piperazin-1-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312261 5-[4-(2,6-Difluoro-benzyl)-piperazin-1-yl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312262 5-[4-(2,4-Dimethyl-pyridin-3-ylmethyl)-piperazin-1-yl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312289 5-Phenyl-1H-pyrrole-2-carboxylic acid (1-cyclohexylcarbamoyl-propyl)-(3-diethylamino-propyl)-amide 312290 (6,7-Dihydro-5H-dibenzo[a,c]cyclohepten-6-ylmethyl)-methoxymethyl-amine 312300 5-[4-(3-Chloro-2,6-difluoro-benzyl)-piperazin-1-yl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312310 2-Furan-2-yl-5-(4-quinolin-2-ylmethyl-piperazin-1-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312316 2-Furan-2-yl-5-[4-(2,3,6-trichloro-benzyl)-piperazin-1-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312321 5-Phenyl-1H-pyrrole-2-carboxylic acid [cyclohexylcarbamoyl-(4-fluoro-phenyl)-methyl]-(2-diethylamino-ethyl)-amide 312328 N-[Cyclohexylcarbamoyl-(4-fluoro-phenyl)-methyl]-N-(3-diethylamino-propyl)-3-(3,4-dihydro-2H-quinolin-1-yl)-propionamide 312329 2-Furan-2-yl-5-(4-phenyl-piperazin-1-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312337 5-(4-Benzyl-piperazin-1-yl)-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312338 5-(4-Benzofuran-2-ylmethyl-piperazin-1-yl)-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312343 (4-Methoxy-6,7-dihydro-5H-dibenzo[a,c]cyclohepten-6-ylmethyl)-propoxymethyl-amine 312344 (5H-Dibenzo[a,c]cyclohepten-6-yl)-methoxymethyl-amine 312357 Acetic acid 4-{4-[4-(5-methoxy-1H-indol-3-yl)-butyl]-piperazin-1-yl}-phenyl ester 312368 N-(4-{4-[4-(5-Methoxy-1H-indol-3-yl)-butyl]-piperazin-1-yl}-phenyl)-acetamide 312378 N-(8-Methoxy-10,11-dihydro-5H-dibenzo[a,d]cyclohepten-10-ylmethyl)-acetamide 312379 N-(8-Methoxy-10,11-dihydro-5H-dibenzo[a,d]cyclohepten-10-ylmethyl)-propionamide 312380 2-Furan-2-yl-5-(4-furan-2-ylmethyl-piperazin-1-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312381 [2-(4-Methoxy-6,7-dihydro-5H-dibenzo[a,c]cyclohepten-6-yl)-ethyl]-methoxymethyl-amine 312382 [2-(10,11-Dihydro-dibenzo[b,f]azepin-5-yl)-ethyl]-methoxymethyl-amine 312384 N-(2-chloro-6-methylphenyl)-2-[(4-pyridinyl)amino]-1,3-thiazole- 312390 2-Furan-2-yl-5-(4-thiazol-4-ylmethyl-piperazin-1-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312391 5-[4-(2-Chloro-6-methyl-quinolin-3-ylmethyl)-piperazin-1-yl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312396 N-(2-chloro-6-methylphenyl)-2-[(4-methyl-2-pyridinyl)amino]-1,3-thiazole-5-carboxamide 312412 5-Phenyl-1H-pyrrole-2-carboxylic acid [1-cyclohexylcarbamoyl-2-(5-methyl-furan-2-yl)-ethyl]-(3-diethylamino-propyl)-amide 312418 2-Methoxy-11-[(methoxymethyl-amino)-methyl]-10,11-dihydro-dibenzo[a,d]cyclohepten-5-one 312420 2-Furan-2-yl-5-(4-phenethyl-piperazin-1-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312423 5-Phenyl-1H-pyrrole-2-carboxylic acid (3-diethylamino-propyl)-[(4-fluoro-benzylcarbamoyl)-(4-fluoro-phenyl)-methyl]-amide 312424 2-Furan-2-yl-5-[4-(1H-imidazol-4-ylmethyl)-piperazin-1-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312425 [2-(6,7-Dihydro-5H-dibenzo[a,c]cyclohepten-6-yl)-ethyl]-methoxymethyl-amine 312428 2-Furan-2-yl-5-(4-thiophen-3-ylmethyl-piperazin-1-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312429 2-Furan-2-yl-5-[4-(2-methylsulfanyl-thiophen-3-ylmethyl)-piperazin-1-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312433 2-Furan-2-yl-5-(4-[1,2,3]thiadiazol-4-ylmethyl-piperazin-1-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312434 5-[4-(2-Chloro-quinolin-3-ylmethyl)-piperazin-1-yl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 312446 5-Phenyl-1H-pyrrole-2-carboxylic acid [cyclohexylcarbamoyl-(3,4-dimethoxy-phenyl)-methyl]-(3-diethylamino-propyl)-amide 312456 (2-chloro-6-methyl-phenyl)-[8-((S)-3-methyl-piperazin-1-yl)-3,3a-dihydro-2,5,9,9b-tetraaza-cyclopenta[a]naphthalen-4-yl]-amine 312468 4-{1-[4-(5-Methoxy-1H-indol-3-yl)-butyl]-1,2,3,6-tetrahydro-pyridin-4-yl}-phenol 312479 N-(2-chloro-6-methylphenyl)-2-(2,6-dimethylpyrimidin-4-ylamino)thiazole-5-carboxamide 312480 3-[4-(4-Phenyl-piperidin-1-yl)-butyl]-1H-indol-5-ol 312482 5'-(quinolin-4-yl)-2,4'-bithiazol-2'-amine 312483 4-(5-Chloro-pyridin-2-yl)-5-quinolin-4-yl-thiazol-2-ylamine 312484 N-(2-chloro-6-methylphenyl)-2-[(3-pyridinyl)amino]-1,3-thiazole-5-carboxamide 312493 N-(2-chloro-6-methylphenyl)-2-[(6-methyl-2-pyridinyl)amino]-1,3-thiazole-5-carboxamide 312500 5-(6-methyl-1,5-naphthyridin-4-yl)-4-(pyridin-2-yl)thiazol-2-amine 312519 4-(3-chlorophenyl)-5-(1,5-naphthyridin-2-yl)thiazol-2-amine 312520 N-(2-chloro-6-methylphenyl)-2-(4,6-dimethylpyrimidin-2-ylamino)thiazole-5-carboxamide 312533 5-Methoxy-3-{4-[4-(4-methoxy-phenyl)-3,6-dihydro-2H-pyridin-1-yl]-butyl}-1H-indole 312534 3-[4-(4-Benzo[1,3]dioxol-5-yl-3,6-dihydro-2H-pyridin-1-yl)-butyl]-5-methoxy-1H-indole 312553 3-[4-(4-Phenyl-piperazin-1-yl)-butyl]-1H-indol-5-ol 312554 3-[4-(4-Phenyl-piperidin-1-yl)-butyl]-1H-indole-5-carboxylic acid methyl ester 312556 5-(naphthalen-1-yl)-4-(pyridin-2-yl)thiazol-2-amine 312557 4-Pyridin-2-yl-5-quinolin-2-yl-thiazol-2-ylamine 312580 5-Methoxy-3-(4-{4-[4-(2-methoxy-ethoxy)-phenyl]-piperazin-1-yl}-butyl)-1H-indole 312581 2,2-Dimethyl-propionic acid 4-{4-[4-(5-methoxy-1H-indol-3-yl)-butyl]-piperazin-1-yl}-phenyl ester 312582 3-[4-(4-Benzo[1,3]dioxol-5-yl-piperazin-1-yl)-butyl]-1H-indole-5-carboxylic acid amide 312584 (4-Chloro-3-trifluoromethyl-phenyl)-[4-(6-methyl-2-phenyl-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-amine 312587 5-Ethoxy-3-{4-[4-(4-methoxy-phenyl)-piperazin-1-yl]-butyl}-1H-indole 312588 3-[4-(4-{2-Cyano-3-[2-(2-ethoxy-ethoxy)-ethoxy]-phenyl}-piperazin-1-yl)-butyl]-1H-indole-5-carboxylic acid amide 312592 4-{4-[4-(5-Methoxy-1H-indol-3-yl)-butyl]-piperazin-1-yl}-phenol 312597 3-{4-[4-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-piperazin-1-yl]-butyl}-1H-indole-5-carboxylic acid 312598 3-{4-[4-(4-Cyano-3-methoxy-phenyl)-piperazin-1-yl]-butyl}-1H-indole-5-carbonitrile 312601 (2,3-Dihydro-benzo[1,4]dioxin-6-yl)-(4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-yl)-amine 312602 (3,4-Difluoro-phenyl)-(4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-yl)-amine 312603 3-[4-(4-Benzo[1,3]dioxol-5-yl-piperazin-1-yl)-butyl]-5-fluoro-1H-indole 312604 3-[4-(4-Benzo[1,3]dioxol-5-yl-piperazin-1-yl)-butyl]-1H-indole-5-carbonitrile 312618 [4-(6-Methoxy-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-(3-methoxy-5-trifluoromethyl-phenyl)-amine 312620 3-[4-(4-Phenyl-piperazin-1-yl)-butyl]-1H-indole-5-carboxylic acid methyl ester 312621 3-[4-(4-Phenyl-piperidin-1-yl)-butyl]-1H-indole-5-carboxylic acid 312634 3-{4-[4-(3,4-Dimethoxy-phenyl)-piperazin-1-yl]-butyl}-5-methoxy-1H-indole 312635 3-{4-[4-(4-Carbamoyl-phenyl)-piperazin-1-yl]-butyl}-1H-indole-5-carboxylic acid amide 312637 {4-[6-Methyl-2-(3-trifluoromethyl-phenyl)-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-phenyl-amine 312648 [4-(6-Methoxy-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-(3-trifluoromethoxy-phenyl)-amine 312649 3-{4-[4-(2-Carbamoyl-phenyl)-piperazin-1-yl]-butyl}-1H-indole-5-carboxylic acid amide 312650 3-{4-[4-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-piperazin-1-yl]-butyl}-1H-indole-5-carboxylic acid amide 312652 2-Hydroxymethyl-5-[6-methylamino-2-(4-quinolin-2-yl-pyrazol-1-yl)-purin-9-yl]-tetrahydro-furan-3,4-diol 312661 [4-(6-Methyl-2-phenyl-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-phenyl-amine 312663 (3,4-Difluoro-phenyl)-[4-(2-phenyl-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-amine 312665 3-{4-[4-(2-Cyano-3-methoxy-phenyl)-piperazin-1-yl]-butyl}-1H-indole-5-carbonitrile 312666 7-{4-[4-(5-Cyano-1H-indol-3-yl)-butyl]-piperazin-1-yl}-benzofuran-2-carboxylic acid amide 312668 3-[4-(4-Benzo[1,3]dioxol-5-yl-piperazin-1-yl)-butyl]-5-methoxy-1H-indole 312675 3-{4-[4-(4-Benzyloxy-phenyl)-piperazin-1-yl]-butyl}-5-methoxy-1H-indole 312678 2-Hydroxymethyl-5-[6-methylamino-2-(4-pyridin-4-yl-pyrazol-1-yl)-purin-9-yl]-tetrahydro-furan-3,4-diol 312679 (3,4-Difluoro-phenyl)-[4-(6-methyl-2-phenyl-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-amine 312683 3-{4-[4-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-piperazin-1-yl]-butyl}-5-methoxy-1H-indole 312684 3-{4-[4-(2-Cyano-phenyl)-piperazin-1-yl]-butyl}-1H-indole-5-carboxylic acid amide 312687 3-[4-(4-Phenyl-piperazin-1-yl)-butyl]-1H-indole-5-carboxylic acid amide 312697 N-(3,4-dimethoxyphenyl)-4-(pyrazolo[1,5-b]pyridazin-3-yl)pyrimidin-2-amine 312698 3-{4-[4-(2-Cyano-3-fluoro-phenyl)-piperazin-1-yl]-butyl}-1H-indole-5-carboxylic acid amide 312699 3-{4-[4-(4-Cyano-phenyl)-piperazin-1-yl]-butyl}-1H-indole-5-carbonitrile 312701 5-Methoxy-3-[4-(4-phenyl-piperazin-1-yl)-butyl]-1H-indole 312706 3-{4-[4-(2,4-Dimethoxy-phenyl)-piperazin-1-yl]-butyl}-1H-indole-5-carboxylic acid amide 312707 3-{4-[4-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-piperazin-1-yl]-butyl}-1H-indole-5-carbaldehyde oxime 312709 3-{4-[4-(2,3-Dihydro-benzofuran-5-yl)-piperazin-1-yl]-butyl}-5-methoxy-1H-indole 312710 Benzo[1,3]dioxol-5-yl-(4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-yl)-amine 312711 (3,5-Dimethoxy-phenyl)-[4-(6-methoxy-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-amine 312712 3-{4-[4-(3-Cyano-4-hydroxy-phenyl)-piperazin-1-yl]-butyl}-1H-indole-5-carbonitrile 312713 4-{4-[4-(5-Cyano-1H-indol-3-yl)-butyl]-piperazin-1-yl}-benzofuran-2-carboxylic acid amide 312724 2-{4-[4-(5-Cyano-1H-indol-3-yl)-butyl]-piperazin-1-yl}-isophthalonitrile 312725 3-{4-[4-(1H-Indol-5-yl)-piperazin-1-yl]-butyl}-1H-indole-5-carbonitrile 312726 3-[4-(4-Chroman-6-yl-piperazin-1-yl)-butyl]-5-methoxy-1H-indole 312727 (4-Chloro-3-trifluoromethyl-phenyl)-[4-(2-phenyl-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-amine 312737 5-Methoxy-3-{4-[4-(4-methoxy-phenyl)-piperazin-1-yl]-butyl}-1H-indole 312742 3-{4-[4-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-piperazin-1-yl]-butyl}-1H-indole-5-carboxylic acid methyl ester 312743 3-{4-[4-(4-Cyano-2-methoxy-phenyl)-piperazin-1-yl]-butyl}-1H-indole-5-carbonitrile 312744 (2,3-Dihydro-benzo[1,4]dioxin-6-yl)-[4-(6-methyl-2-phenyl-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-amine 312753 3-{4-[4-(4-Ethoxy-phenyl)-piperazin-1-yl]-butyl}-5-methoxy-1H-indole 312758 N-(4-isopropylphenyl)-4-(pyrazolo[1,5-b]pyridazin-3-yl)pyrimidin-2-amine 312759 3-[4-(4-Benzofuran-5-yl-piperazin-1-yl)-butyl]-1H-indole-5-carbonitrile 312761 2-Hydroxymethyl-5-[6-(3-iodo-benzylamino)-2-(4-pyridin-2-yl-pyrazol-1-yl)-purin-9-yl]-tetrahydro-furan-3,4-diol 312762 (3,4-Dihydro-2H-benzo[b][1,4]dioxepin-7-yl)-(4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-yl)-amine 312763 (3,4-Dichloro-phenyl)-(4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-yl)-amine 312774 [4-(2-Phenyl-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-(3-trifluoromethyl-phenyl)-amine 312779 [4-(6-Ethoxy-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-(3-methoxy-5-trifluoromethyl-phenyl)-amine 312788 [4-(6-Methyl-2-phenyl-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-(3-trifluoromethyl-phenyl)-amine 312790 (4-sec-Butyl-phenyl)-(4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-yl)-amine 312791 3-{4-[4-(4-Acetylamino-phenyl)-piperazin-1-yl]-butyl}-1H-indole-5-carboxylic acid amide 312792 3-{4-[4-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-piperazin-1-yl]-butyl}-1H-indole-5-carbonitrile 312795 3-[4-(4-Phenyl-piperazin-1-yl)-butyl]-1H-indole-5-carboxylic acid 312796 3-[4-(4-Phenyl-piperidin-1-yl)-butyl]-1H-indole-5-carboxylic acid amide 312804 (4-tert-Butyl-phenyl)-(4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-yl)-amine 312805 4-[4-(6-Methoxy-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-ylamino]-benzonitrile 312806 4-{4-[4-(5-Fluoro-1H-indol-3-yl)-butyl]-piperazin-1-yl}-benzonitrile 312807 3-[4-(4-{2-Cyano-3-[2-(2-ethoxy-ethoxy)-ethoxy]-phenyl}-piperazin-1-yl)-butyl]-1H-indole-5-carbonitrile 312809 2-Hydroxymethyl-5-[6-methylamino-2-(4-pyridin-3-yl-pyrazol-1-yl)-purin-9-yl]-tetrahydro-furan-3,4-diol 312822 [4-(6-Methoxy-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-(4-nitro-phenyl)-amine 312823 (3,5-Difluoro-phenyl)-[4-(2-phenyl-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-amine 312824 6-{4-[4-(5-Cyano-1H-indol-3-yl)-butyl]-piperazin-1-yl}-benzofuran-2-carboxylic acid amide 312827 5-Methoxy-3-{4-[4-(3,4,5-trimethoxy-phenyl)-piperazin-1-yl]-butyl}-1H-indole 312828 N-(2-chloro-6-methylphenyl)-2-(pyridin-2-ylamino)thiazole-5-carboxamide 312833 N-(2-chloro-6-methylphenyl)-2-[(4,6-dimethyl-2-pyridinyl)-amino]-1,3-thiazole-5-carboxamide 312839 2-Amino-1-[3-(1H-benzoimidazol-2-yl)-3,4-dihydro-1H-isoquinolin-2-yl]-3-(4-hydroxy-phenyl)-propan-1-one 312844 5-Cyclopentyloxy-3-{4-[4-(4-methoxy-phenyl)-piperazin-1-yl]-butyl}-1H-indole 312845 (4-Chloro-3-trifluoromethyl-phenyl)-{4-[2-(3-trifluoromethyl-phenyl)-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-amine 312848 3-{4-[4-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-piperazin-1-yl]-butyl}-5-fluoro-1H-indole 312849 3-{4-[4-(4-Hydroxy-phenyl)-piperazin-1-yl]-butyl}-1H-indole-5-carbonitrile 312851 2-Hydroxymethyl-5-{6-(3-iodo-benzylamino)-2-[4-(4-methoxy-phenyl)-pyrazol-1-yl]-purin-9-yl}-tetrahydro-furan-3,4-diol 312877 2-Amino-3-(4-hydroxy-phenyl)-1-[2-(5-methyl-4-phenyl-1H-imidazol-2-yl)-pyrrolidin-1-yl]-propan-1-one 312879 5-{4-[4-(5-Cyano-1H-indol-3-yl)-butyl]-piperazin-1-yl}-2,3-dihydro-benzofuran-2-carboxylic acid amide 312880 3-(4-{4-[4-(tert-Butyl-dimethyl-silanyloxy)-phenyl]-piperazin-1-yl}-butyl)-5-methoxy-1H-indole 312881 3-{4-[4-(2-Cyano-benzofuran-5-yl)-piperazin-1-yl]-butyl}-1H-indole-5-carbonitrile 312882 1-[9-(3,4-Dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-6-methylamino-9H-purin-2-yl]-1H-pyrazole-4-carboxylic acid 4-chloro-benzylamide 312883 3-[2-(3-Trifluoromethyl-phenylamino)-pyrimidin-4-yl]-pyrazolo[1,5-b]pyridazin-6-ol 312884 (3-Methoxy-5-trifluoromethyl-phenyl)-[4-(6-methyl-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-amine 312885 3-{4-[4-(2,3-Dihydro-benzofuran-5-yl)-piperazin-1-yl]-butyl}-1H-indole-5-carbonitrile 312896 2-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid phenethyl-amide 312909 3-{4-[4-(4-Cyano-3,5-difluoro-phenyl)-piperazin-1-yl]-butyl}-1H-indole-5-carbonitrile 312910 5-{4-[4-(5-Cyano-1H-indol-3-yl)-butyl]-piperazin-1-yl}-benzo[b]thiophene-2-carboxylic acid amide 312912 Acetic acid 3-{4-[4-(4-methoxy-phenyl)-piperazin-1-yl]-butyl}-1H-indol-5-yl ester 312913 {4-[2-(4-Methoxy-phenyl)-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-phenyl-amine 312916 3-[4-(4-Chroman-6-yl-piperazin-1-yl)-butyl]-1H-indole-5-carboxylic acid amide 312917 3-{4-[4-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-piperazin-1-yl]-butyl}-1H-indole-5-carbaldehyde 312937 (4-Chloro-3-trifluoromethyl-phenyl)-(4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-yl)-amine 312940 3-{4-[4-(4-Methoxy-phenyl)-piperazin-1-yl]-butyl}-1H-indole-5-carboxylic acid methyl ester 312941 3-{4-[4-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-piperazin-1-yl]-butyl}-1H-indol-5-ol 312942 {4-[2-(4-Fluoro-phenyl)-6-methyl-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-phenyl-amine 312945 N-phenyl-4-(pyrazolo[1,5-b]pyridazin-3-yl)pyrimidin-2-amine 312946 3-{4-[4-(4-Fluoro-phenyl)-piperazin-1-yl]-butyl}-1H-indole-5-carbonitrile 312947 4-{4-[4-(5-Cyano-1H-indol-3-yl)-butyl]-piperazin-1-yl}-phthalonitrile 312968 (3,5-Dimethoxy-phenyl)-(4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-yl)-amine 312969 (3,5-Bis-trifluoromethyl-phenyl)-[4-(6-methoxy-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-amine 312971 5-{4-[4-(5-Cyano-1H-indol-3-yl)-butyl]-piperazin-1-yl}-benzofuran-2-carboxylic acid amide 312972 2-{4-[4-(5-Cyano-1H-indol-3-yl)-butyl]-piperazin-1-yl}-benzamide 312973 2-{2-[4-(4-Chloro-phenyl)-pyrazol-1-yl]-6-methylamino-purin-9-yl}-5-hydroxymethyl-tetrahydro-furan-3,4-diol 312975 Methyl-phenyl-(4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-yl)-amine 312976 2-Hydroxymethyl-5-[6-(3-iodo-benzylamino)-2-(4-isoquinolin-1-yl-pyrazol-1-yl)-purin-9-yl]-tetrahydro-furan-3,4-diol 312977 [4-(6-Ethoxy-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-(3-trifluoromethyl-phenyl)-amine 312978 3-[4-(4-Benzo[1,2,5]thiadiazol-4-yl-piperazin-1-yl)-butyl]-1H-indole-5-carbonitrile 312981 2-Amino-3-(4-hydroxy-phenyl)-1-[3-(5-methyl-4-propyl-1H-imidazol-2-yl)-3,4-dihydro-1H-isoquinolin-2-yl]-propan-1-one 312999 {4-[2-(4-Fluoro-phenyl)-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-phenyl-amine 313000 Phenyl-{4-[2-(3-trifluoromethyl-phenyl)-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-amine 313001 (3-Methoxy-5-trifluoromethyl-phenyl)-(4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-yl)-amine 313002 [4-(6-Methyl-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-(3-trifluoromethyl-phenyl)-amine 313005 3-{4-[4-(4-Hydroxy-phenyl)-piperazin-1-yl]-butyl}-1H-indole-5-carboxylic acid amide 313006 [4-(6-Phenyl-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-(3-trifluoromethyl-phenyl)-amine 313007 (3,4-Difluoro-phenyl)-{4-[2-(4-methoxy-phenyl)-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-amine 313022 Thiophene-2-sulfonic acid (3-{(R)-1-hydroxy-2-[(R)-2-(1H-indol-3-yl)-1-methyl-ethylamino]-ethyl}-phenyl)-amide 313030 (3,4-Difluoro-phenyl)-{4-[6-methyl-2-(3-trifluoromethyl-phenyl)-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-amine 313032 (3,4-Difluoro-phenyl)-{4-[2-(4-fluoro-phenyl)-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-amine 313033 (2,3-Dihydro-benzo[1,4]dioxin-6-yl)-{4-[2-(3-trifluoromethyl-phenyl)-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-amine 313037 3-{4-[4-(2-Oxo-2H-chromen-6-yl)-piperazin-1-yl]-butyl}-1H-indole-5-carbonitrile 313038 {4-[2-(4-Chloro-phenyl)-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-(3,4-difluoro-phenyl)-amine 313040 4-(4-(pyrazolo[1,5-b]pyridazin-3-yl)pyrimidin-2-ylamino)benzonitrile 313041 N-(4-nitrophenyl)-4-(pyrazolo[1,5-b]pyridazin-3-yl)pyrimidin-2-amine 313058 (S)-2-amino-3-(4-hydroxyphenyl)-1-((S)-3-(5-methyl-4-phenyl-1H-imidazol-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)propan-1-one 313066 2-[2-(4-Benzooxazol-2-yl-pyrazol-1-yl)-6-methylamino-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 313068 (2,3-Dihydro-benzo[1,4]dioxin-6-yl)-{4-[6-methyl-2-(3-trifluoromethyl-phenyl)-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-amine 313069 1-[9-(3,4-Dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-6-methylamino-9H-purin-2-yl]-1H-pyrazole-4-carboxylic acid propylamide 313071 (3,5-Dichloro-phenyl)-(4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-yl)-amine 313072 3-[4-(4-Phenyl-piperazin-1-yl)-butyl]-1H-indole-5-carbonitrile 313073 3-[4-(4-Chroman-6-yl-piperazin-1-yl)-butyl]-1H-indole-5-carbonitrile 313074 2-Hydroxymethyl-5-{2-[4-(4-methoxy-phenyl)-pyrazol-1-yl]-6-propylamino-purin-9-yl}-tetrahydro-furan-3,4-diol 313075 (3-Methoxy-phenyl)-[4-(6-methoxy-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-amine 313076 Phenyl-[4-(2-phenyl-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-amine 313098 3-{4-[4-(4-Methoxy-phenyl)-piperazin-1-yl]-butyl}-5-pentyloxy-1H-indole 313099 2-[2-(1-Benzyl-1H-pyrazol-4-yl)-6-propylamino-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 313101 (3,5-Dimethyl-phenyl)-(4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-yl)-amine 313106 3-{4-[4-(2,3-Dihydro-benzofuran-5-yl)-piperazin-1-yl]-butyl}-1H-indole-5-carboxylic acid amide 313107 (2,3-Dihydro-benzo[1,4]dioxin-6-yl)-{4-[2-(4-methoxy-phenyl)-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-amine 313108 {4-[2-(4-Chloro-phenyl)-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-(2,3-dihydro-benzo[1,4]dioxin-6-yl)-amine 313117 Macrolide derivative 313118 Macrolide derivative 313130 5-{4-[4-(5-Fluoro-1H-indol-3-yl)-butyl]-piperazin-1-yl}-benzofuran-2-carbonitrile 313131 3-{4-[4-(5-Chloro-2-methoxy-phenyl)-piperazin-1-yl]-butyl}-1H-indole-5-carbonitrile 313132 5-Benzyloxy-3-{4-[4-(4-methoxy-phenyl)-piperazin-1-yl]-butyl}-1H-indole 313133 5-Methoxy-3-{4-[4-(4-methoxy-3,5-dimethyl-phenyl)-piperazin-1-yl]-butyl}-1H-indole 313134 (2,3-Dihydro-benzo[1,4]dioxin-6-yl)-{4-[2-(4-fluoro-phenyl)-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-amine 313135 {4-[2-(4-Chloro-phenyl)-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-phenyl-amine 313138 5-Chloro-3-{4-[4-(2,3-dihydro-benzo[1,4]dioxin-6-yl)-piperazin-1-yl]-butyl}-1H-indole 313139 3-{4-[4-(4-Methoxy-phenyl)-piperazin-1-yl]-butyl}-1H-indole-5-carbonitrile 313142 N-(2-chloro-6-methylphenyl)-2-(6-morpholinopyrimidin-4-ylamino)thiazole-5-carboxamide 313156 (S)-2-amino-3-(4-hydroxyphenyl)-1-((S)-2-(5-methyl-4-phenyl-1H-imidazol-2-yl)piperidin-1-yl)propan-1-one 313160 5-{4-[4-(5-Cyano-1H-indol-3-yl)-butyl]-piperazin-1-yl}-1H-indole-2-carboxylic acid amide 313162 3-{4-[4-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-piperazin-1-yl]-butyl}-1H-indole 313163 5-{4-[4-(5-Fluoro-1H-indol-3-yl)-butyl]-piperazin-1-yl}-benzofuran-2-carboxylic acid amide 313167 [4-(6-Methoxy-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-(3-trifluoromethyl-phenyl)-amine 313168 3-{4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-butyl}-1H-indole-5-carbonitrile 313169 3-[4-(4-Benzo[1,2,5]thiadiazol-5-yl-piperazin-1-yl)-butyl]-1H-indole-5-carbonitrile 313176 [3-(2-{(R)-(R)-2-Hydroxy-2-[3-(thiophene-2-sulfonylamino)-phenyl]-ethylamino}-propyl)-1H-indol-7-yloxy]-acetic acid 313182 Methanesulfonic acid 3-(2-{(R)-(R)-2-hydroxy-2-[3-(thiophene-2-sulfonylamino)-phenyl]-ethylamino}-propyl)-1H-indol-7-yl ester 313187 2-Amino-1-[3-(5-bromo-4-phenyl-1H-imidazol-2-yl)-3,4-dihydro-1H-isoquinolin-2-yl]-3-(4-hydroxy-phenyl)-propan-1-one 313198 4-{4-[4-(5-Cyano-1H-indol-3-yl)-butyl]-piperazin-1-yl}-benzamide 313199 5-{4-[4-(5-Cyano-1H-indol-3-yl)-butyl]-piperazin-1-yl}-benzofuran-4-carboxylic acid amide 313202 (2,3-Dihydro-benzo[1,4]dioxin-6-yl)-[4-(6-methyl-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-amine 313203 {4-[2-(4-Methoxy-phenyl)-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-(3-trifluoromethyl-phenyl)-amine 313216 (S)-2-amino-3-(4-hydroxyphenyl)-1-((S)-3-(4-phenyl-1H-imidazol-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)propan-1-one 313231 3-{4-[4-(4-Methoxy-phenyl)-piperazin-1-yl]-butyl}-1H-indole-5-carboxylic acid amide 313232 {4-[2-(4-Chloro-phenyl)-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-(3-trifluoromethyl-phenyl)-amine 313262 (2,3-Dihydro-benzo[1,4]dioxin-6-yl)-[4-(6-methoxy-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-amine 313263 {4-[2-(4-Fluoro-phenyl)-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-(3-trifluoromethyl-phenyl)-amine 313266 6-{4-[4-(5-Fluoro-1H-indol-3-yl)-butyl]-piperazin-1-yl}-chromen-2-one 313269 (4-Pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-yl)-o-tolyl-amine 313270 N-(3-methoxyphenyl)-4-(pyrazolo[1,5-b]pyridazin-3-yl)pyrimidin-2-amine 313296 (3,4-Difluoro-phenyl)-{4-[2-(3-trifluoromethyl-phenyl)-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-amine 313297 (4-Chloro-3-trifluoromethyl-phenyl)-{4-[6-methyl-2-(3-trifluoromethyl-phenyl)-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-amine 313298 (3-Bromo-5-trifluoromethyl-phenyl)-(4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-yl)-amine 313299 (3,5-Difluoro-phenyl)-(4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-yl)-amine 313300 3-{4-[4-(3,4-Dimethoxy-phenyl)-piperazin-1-yl]-butyl}-1H-indole-5-carbonitrile 313303 [4-(6-Propoxy-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-(3-trifluoromethyl-phenyl)-amine 313304 (2,3-Dihydro-benzo[1,4]dioxin-6-yl)-[4-(6-phenyl-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-amine 313315 Thiophene-2-sulfonic acid (3-{(R)-1-hydroxy-2-[(R)-2-(7-methoxy-1H-indol-3-yl)-1-methyl-ethylamino]-ethyl}-phenyl)-amide 313323 1-[9-(3,4-Dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-6-methylamino-9H-purin-2-yl]-1H-pyrazole-4-carboxylic acid ethylamide 313324 2-[2-(1-Benzyl-1H-pyrazol-4-yl)-6-methylamino-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 313325 [4-(6-Methyl-pyrazolo[1,5-b]pyridazin-3-yl)-pyrimidin-2-yl]-(4-trifluoromethyl-phenyl)-amine 313326 (4-Chloro-3-trifluoromethyl-phenyl)-{4-[2-(4-fluoro-phenyl)-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-amine 313329 3-{4-[4-(3,5-Dichloro-4-methoxy-phenyl)-piperazin-1-yl]-butyl}-1H-indole-5-carboxylic acid amide 313330 3-{4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-butyl}-1H-indole-5-carboxylic acid amide 313331 (4-Chloro-3-trifluoromethyl-phenyl)-{4-[2-(4-methoxy-phenyl)-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-amine 313332 {4-[2-(4-Chloro-phenyl)-pyrazolo[1,5-b]pyridazin-3-yl]-pyrimidin-2-yl}-(4-chloro-3-trifluoromethyl-phenyl)-amine 313341 Naphthalene-1-sulfonic acid [3-(6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-propyl]-amide 313393 (S)-2-((S)-2-Benzyl-1,3-dioxo-octahydro-pyrido[1,2-c]pyrimidin-5-ylamino)-3-(1H-indol-3-yl)-propionic acid tert-butyl ester 313408 (S)-2-[(4R,5R)-2-(4-Dimethylamino-phenyl)-4-methyl-1,3-dioxo-octahydro-pyrido[1,2-c]pyrimidin-5-ylamino]-3-(1H-indol-3-yl)-propionic acid tert-butyl ester 313428 [(5S,9S,12S,14aR)-9-Benzyl-5-(4-hydroxy-benzyl)-12-(1H-indol-3-ylmethyl)-4,8,11,14-tetraoxo-dodecahydro-3a,6,7,10,13-pentaaza-cyclopentacyclotridecen-7-yl]-acetic acid 313429 [(5R,9R,12R,14aS)-9-Benzyl-5-(4-hydroxy-benzyl)-12-(1H-indol-3-ylmethyl)-4,8,11,14-tetraoxo-dodecahydro-3a,6,7,10,13-pentaaza-cyclopentacyclotridecen-7-yl]-acetic acid 313441 7-[(cyclopropylmethyl)(methyl)amino]-8,8-dimethyl-5,6,7,8-tetrahydronaphthalen-2-ol 313454 8,8-dimethyl-7-{[(2E)-3-phenylprop-2-enyl]amino}-5,6,7,8-tetrahydronaphthalen-2-ol 313477 7-(Bis-cyclopropylmethyl-amino)-8,8-dimethyl-5,6,7,8-tetrahydro-naphthalen-2-ol 313484 4-Methoxy-N-[3-(6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-propyl]-benzenesulfonamide 313492 8,8-Dimethyl-7-[methyl-((E)-3-phenyl-allyl)-amino]-5,6,7,8-tetrahydro-naphthalen-2-ol 313495 (S)-2-((4R,5R)-2-Benzyl-4-methyl-1,3-dioxo-octahydro-pyrido[1,2-c]pyrimidin-5-ylamino)-3-(1H-indol-3-yl)-propionic acid adamantan-2-yl ester 313501 Methanesulfonic acid 3-(2-{2-hydroxy-2-[(R)-3-(thiophene-2-sulfonylamino)-phenyl]-ethylamino}-ethyl)-1H-indol-7-yl ester 313507 7-(dimethylamino)-8,8-dimethyl-5,6,7,8-tetrahydronaphthalen-2-ol 313518 N-Ethyl-4-methoxy-N-[3-(6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-propyl]-benzenesulfonamide 313523 TCMDC-139048 313544 (S)-2-[(S)-2-(4-Dimethylamino-phenyl)-1,3-dioxo-octahydro-pyrido[1,2-c]pyrimidin-5-ylamino]-3-(1H-indol-3-yl)-propionic acid tert-butyl ester 313552 4-Methoxy-N-{3-[4-(o-methoxyphenyl)-piperazin-1-yl]-propyl}-benzenesulfonamide 313553 N-[3-(6-Methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-propyl]-benzenesulfonamide 313577 [(5S,9R,12S,14aR)-9-Benzyl-5-(4-hydroxy-benzyl)-12-(1H-indol-3-ylmethyl)-4,8,11,14-tetraoxo-dodecahydro-3a,6,7,10,13-pentaaza-cyclopentacyclotridecen-7-yl]-acetic acid 313578 [(5R,9S,12R,14aS)-9-Benzyl-5-(4-hydroxy-benzyl)-12-(1H-indol-3-ylmethyl)-4,8,11,14-tetraoxo-dodecahydro-3a,6,7,10,13-pentaaza-cyclopentacyclotridecen-7-yl]-acetic acid 313579 [(5R,9S,12R,14aR)-9-Benzyl-5-(4-hydroxy-benzyl)-12-(1H-indol-3-ylmethyl)-4,8,11,14-tetraoxo-dodecahydro-3a,6,7,10,13-pentaaza-cyclopentacyclotridecen-7-yl]-acetic acid 313580 [(5S,9R,12S,14aS)-9-Benzyl-5-(4-hydroxy-benzyl)-12-(1H-indol-3-ylmethyl)-4,8,11,14-tetraoxo-dodecahydro-3a,6,7,10,13-pentaaza-cyclopentacyclotridecen-7-yl]-acetic acid 313581 [(5R,9R,12S,14aR)-9-Benzyl-5-(4-hydroxy-benzyl)-12-(1H-indol-3-ylmethyl)-4,8,11,14-tetraoxo-dodecahydro-3a,6,7,10,13-pentaaza-cyclopentacyclotridecen-7-yl]-acetic acid 313582 [(5S,9S,12R,14aS)-9-Benzyl-5-(4-hydroxy-benzyl)-12-(1H-indol-3-ylmethyl)-4,8,11,14-tetraoxo-dodecahydro-3a,6,7,10,13-pentaaza-cyclopentacyclotridecen-7-yl]-acetic acid 313608 6-Methoxy-8,8-dimethyl-7-((E)-3-phenyl-allylamino)-5,6,7,8-tetrahydro-naphthalen-2-ol 313656 7-(dipropylamino)-8,8-dimethyl-5,6,7,8-tetrahydronaphthalen-2-ol 313657 7-[(cyclopropylmethyl)amino]-8,8-dimethyl-5,6,7,8-tetrahydronaphthalen-2-ol 313687 (S)-2-((4S,5S)-2-Benzyl-4-methyl-1,3-dioxo-octahydro-pyrido[1,2-c]pyrimidin-5-ylamino)-3-(1H-indol-3-yl)-propionic acid tert-butyl ester 313734 N-Ethyl-N-[3-(6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-propyl]-4-methyl-benzenesulfonamide 313738 Naphthalene-1-sulfonic acid ethyl-[3-(6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-propyl]-amide 313743 3-Amino-N-(3-{(R)-1-hydroxy-2-[2-(7-methanesulfonyl-1H-indol-3-yl)-ethylamino]-ethyl}-phenyl)-benzenesulfonamide 313747 (S)-2-[(R)-2-(4-Dimethylamino-phenyl)-1,3-dioxo-octahydro-pyrido[1,2-c]pyrimidin-5-ylamino]-3-(1H-indol-3-yl)-propionic acid tert-butyl ester 313780 (S)-2-((R)-2-Benzyl-1,3-dioxo-octahydro-pyrido[1,2-c]pyrimidin-5-ylamino)-3-(1H-indol-3-yl)-propionic acid tert-butyl ester 313781 (S)-2-[(R)-2-(4-Dimethylamino-phenyl)-1,3-dioxo-octahydro-pyrido[1,2-c]pyrimidin-5-ylamino]-3-(1H-indol-3-yl)-propionic acid adamantan-2-yl ester 313782 (S)-2-[(4R,5R)-2-(4-Dimethylamino-phenyl)-4-methyl-1,3-dioxo-octahydro-pyrido[1,2-c]pyrimidin-5-ylamino]-3-(1H-indol-3-yl)-propionic acid adamantan-2-yl ester 313788 [(5R,9S,12S,14aR)-9-Benzyl-5-(4-hydroxy-benzyl)-12-(1H-indol-3-ylmethyl)-4,8,11,14-tetraoxo-dodecahydro-3a,6,7,10,13-pentaaza-cyclopentacyclotridecen-7-yl]-acetic acid 313789 [(5S,9R,12R,14aS)-9-Benzyl-5-(4-hydroxy-benzyl)-12-(1H-indol-3-ylmethyl)-4,8,11,14-tetraoxo-dodecahydro-3a,6,7,10,13-pentaaza-cyclopentacyclotridecen-7-yl]-acetic acid 313790 [(5S,9S,12S,14aS)-9-Benzyl-5-(4-hydroxy-benzyl)-12-(1H-indol-3-ylmethyl)-4,8,11,14-tetraoxo-dodecahydro-3a,6,7,10,13-pentaaza-cyclopentacyclotridecen-7-yl]-acetic acid 313791 [(5R,9R,12R,14aR)-9-Benzyl-5-(4-hydroxy-benzyl)-12-(1H-indol-3-ylmethyl)-4,8,11,14-tetraoxo-dodecahydro-3a,6,7,10,13-pentaaza-cyclopentacyclotridecen-7-yl]-acetic acid 313792 [(5S,9S,12R,14aR)-9-Benzyl-5-(4-hydroxy-benzyl)-12-(1H-indol-3-ylmethyl)-4,8,11,14-tetraoxo-dodecahydro-3a,6,7,10,13-pentaaza-cyclopentacyclotridecen-7-yl]-acetic acid 313793 [(5R,9R,12S,14aS)-9-Benzyl-5-(4-hydroxy-benzyl)-12-(1H-indol-3-ylmethyl)-4,8,11,14-tetraoxo-dodecahydro-3a,6,7,10,13-pentaaza-cyclopentacyclotridecen-7-yl]-acetic acid 313825 (S)-2-((R)-2-Benzyl-1,3-dioxo-octahydro-pyrido[1,2-c]pyrimidin-5-ylamino)-3-(1H-indol-3-yl)-propionic acid adamantan-2-yl ester 313845 7-(allylamino)-8,8-dimethyl-5,6,7,8-tetrahydronaphthalen-2-ol 313846 7-[allyl(methyl)amino]-8,8-dimethyl-5,6,7,8-tetrahydronaphthalen-2-ol 313860 7-[Bis-((E)-3-phenyl-allyl)-amino]-8,8-dimethyl-5,6,7,8-tetrahydro-naphthalen-2-ol 313861 7-amino-6-methoxy-8,8-dimethyl-5,6,7,8-tetrahydronaphthalen-2-ol 313876 8,8-dimethyl-7-(propylamino)-5,6,7,8-tetrahydronaphthalen-2-ol 313877 8,8-dimethyl-7-[methyl(propyl)amino]-5,6,7,8-tetrahydronaphthalen-2-ol 313880 7-(diallylamino)-8,8-dimethyl-5,6,7,8-tetrahydronaphthalen-2-ol 313883 N-Ethyl-N-[3-(6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-propyl]-benzenesulfonamide 313902 (S)-2-((4R,5R)-2-Benzyl-4-methyl-1,3-dioxo-octahydro-pyrido[1,2-c]pyrimidin-5-ylamino)-3-(1H-indol-3-yl)-propionic acid tert-butyl ester 313909 N-[3-(6-Methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-propyl]-4-methyl-benzenesulfonamide 313913 4-[3-(3-{2-[1-(3-Chloro-phenyl)-piperidin-4-ylamino]-ethyl}-ureido)-phenyl]-2,6-dimethyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid dimethyl ester 313914 2,6-Dimethyl-4-[3-(3-{2-[1-(2-methylsulfanyl-phenyl)-piperidin-4-ylamino]-ethyl}-ureido)-phenyl]-1,4-dihydro-pyridine-3,5-dicarboxylic acid dimethyl ester 313950 3-Amino-N-(3-{(R)-1-hydroxy-2-[(R)-2-(7-methanesulfonyl-1H-indol-3-yl)-1-methyl-ethylamino]-ethyl}-phenyl)-benzenesulfonamide 313956 (S)-3-{[5-(2,4-Dimethyl-phenyl)-thiophene-2-carbonyl]-methyl-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 313983 4-((E)-2,4-Dihydroxy-phenylazo)-3-hydroxy-naphthalene-1-sulfonic acid 313984 2-Hydrazino-3-(1H-indol-3-yl)-propionic acid 313987 (S)-3-{[5-(2-Chloro-4-ethoxy-phenyl)-thiophene-2-carbonyl]-methyl-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 314006 2-[6-(3-Chloro-phenylamino)-9-isopropyl-9H-purin-2-ylamino]-2-methyl-propan-1-ol 314015 2-Chloro-N-(4-chloro-benzothiazol-2-yl)-acetamide 314016 1-(3-nitrophenyl)-3-phenylprop-2-en-1-one 314017 N-arylpiperazine derivative 314032 3-[1-(2-Hydroxy-phenyl)-meth-(Z)-ylidene]-5-nitro-1,3-dihydro-indol-2-one 314033 5-Methoxy-3-[4-oxo-2-thioxo-thiazolidin-(5E)-ylidene]-1,3-dihydro-indol-2-one 314046 2,6-Dimethyl-4-(3-{3-[2-(1-phenyl-piperidin-4-ylamino)-ethyl]-ureido}-phenyl)-1,4-dihydro-pyridine-3,5-dicarboxylic acid dimethyl ester 314047 2,6-Dimethyl-4-[3-(3-{2-[1-(2-nitro-phenyl)-piperidin-4-ylamino]-ethyl}-ureido)-phenyl]-1,4-dihydro-pyridine-3,5-dicarboxylic acid dimethyl ester 314062 N-Ethyl-N-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]-propyl}-4-methyl-benzenesulfonamide 314063 (Z)-2-(4-Nitro-benzoyl)-3-pyridin-2-yl-acrylic acid ethyl ester 314070 N-arylpiperazine derivative 314071 N-arylpiperazine derivative 314072 N-arylpiperazine derivative 314073 N-arylpiperazine derivative 314074 2,6-Dimethyl-4-(3-{3-[2-(1-o-tolyl-piperidin-4-ylamino)-ethyl]-ureido}-phenyl)-1,4-dihydro-pyridine-3,5-dicarboxylic acid dimethyl ester 314075 2,6-Dimethyl-4-[3-(3-{2-[1-(2-trifluoromethyl-phenyl)-piperidin-4-ylamino]-ethyl}-ureido)-phenyl]-1,4-dihydro-pyridine-3,5-dicarboxylic acid dimethyl ester 314077 4-[3-(3-{2-[1-(2-Cyano-phenyl)-piperidin-4-ylamino]-ethyl}-ureido)-phenyl]-2,6-dimethyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid dimethyl ester 314078 4-[3-(3-{2-[1-(2-Methoxy-phenyl)-piperidin-4-ylamino]-ethyl}-ureido)-phenyl]-2,6-dimethyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid dimethyl ester 314079 2,6-Dimethyl-4-[3-(3-{2-[1-(2-trifluoromethoxy-phenyl)-piperidin-4-ylamino]-ethyl}-ureido)-phenyl]-1,4-dihydro-pyridine-3,5-dicarboxylic acid dimethyl ester 314123 5-bromo-3-(2-oxo-2-phenylethylidene)indolin-2-one 314153 5-Methyl-3-(2-oxo-2-phenyl-ethylidene)-1,3-dihydro-indol-2-one 314154 3,9,11-Trichloro-5,6-dihydro-benzo[c]acridine-7-carbonyl chloride 314155 (4-Chloro-phenyl)-[3-(4-chloro-phenyl)-2,4-dioxo-oxazolidin-(5Z)-ylidene]-acetonitrile 314176 2-{(2-Hydroxy-ethyl)-[5-(4-methoxy-phenyl)-[1,3,4]oxadiazol-2-yl]-amino}-ethanol 314193 5-bromo-3-(2-oxo-2-p-tolylethylidene)indolin-2-one 314194 1-Methyl-3-[2-oxo-2-phenyl-eth-(Z)-ylidene]-1,3-dihydro-indol-2-one 314207 5-Methyl-4-nitro-3-phenyl-4,5-dihydro-1H-pyrazole 314211 (3-Oxo-1-phenyl-1,3-dihydro-isobenzofuran-1-yl)-thiourea 314225 N-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-4-methyl-benzenesulfonamide 314226 N-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyl}-4-methyl-benzenesulfonamide 314228 2-Chloro-5-nitro-benzoic acid ethyl ester 314231 N-(4-cinnamoylphenyl)acetamide 314245 N-arylpiperazine derivative 314246 N-arylpiperazine derivative 314247 N-arylpiperazine derivative 314248 N-arylpiperazine derivative 314249 N-arylpiperazine derivative 314263 4-aza-8-fluorotryptanthrin 314316 (S)-3-{[5-(2,6-Dimethyl-phenyl)-thiophene-2-carbonyl]-methyl-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 314345 2-Nitro-4b,9,10-triaza-benzo[b]fluorene-5,11-dione 314347 3-(2-oxo-2-phenylethylidene)indolin-2-one 314348 5-Chloro-4-nitro-thiophene-2-sulfonic acid (4-trifluoromethyl-phenyl)-amide 314349 (E)-1-(4-Nitro-phenyl)-3-pyridin-2-yl-propenone 314352 3-Fluoro-N-{3-[5-(2-methyl-benzoyl)-thiazol-2-ylamino]-propyl}-benzenesulfonamide 314380 3-Chloro-4b,9,10-triaza-benzo[b]fluorene-5,11-dione 314399 1-(2,4-Dichloro-benzoyl)-3-(2-hydroxy-5-nitro-phenyl)-thiourea 314400 N-(4-Chloro-2-methyl-phenyl)-3-nitro-benzamide 314408 5-[5-Fluoro-2-oxo-1,2-dihydro-indol-(3Z)-ylidene]-thiazolidine-2,4-dione 314446 4-[3-(3-{2-[1-(2-Hydroxy-phenyl)-piperidin-4-ylamino]-ethyl}-ureido)-phenyl]-2,6-dimethyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid dimethyl ester 314447 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-2-(2'-methoxy-biphenyl-4-yl)-acetamide 314448 N-(1-{4-[(R)-2-(3-Amino-propionylamino)-3-(2,4-dichloro-phenyl)-propionyl]-piperazin-1-yl}-cyclohexylmethyl)-4-trifluoromethoxy-benzamide 314449 N-(1-{4-[(R)-2-(3-Amino-propionylamino)-3-(2,4-dichloro-phenyl)-propionyl]-piperazin-1-yl}-cyclohexylmethyl)-4-methyl-benzamide 314450 N-(1-{4-[(R)-2-(3-Amino-propionylamino)-3-(2,4-dichloro-phenyl)-propionyl]-piperazin-1-yl}-cyclohexylmethyl)-4-trifluoromethyl-benzamide 314451 N-(1-{4-[(R)-2-(3-Amino-propionylamino)-3-(2,4-dichloro-phenyl)-propionyl]-piperazin-1-yl}-cyclohexylmethyl)-4-tert-butyl-benzamide 314452 Furan-2-carboxylic acid (1-{4-[(R)-2-(3-amino-propionylamino)-3-(2,4-dichloro-phenyl)-propionyl]-piperazin-1-yl}-cyclohexylmethyl)-amide 314457 2-(4-Amino-furazan-3-yl)-1-ethyl-1H-benzoimidazol-5-ol 314462 1-(2-Fluoro-5-trifluoromethyl-phenyl)-3-(4-{[2-(4-methanesulfonylmethyl-phenylamino)-pyrimidin-4-yl]-methyl-amino}-phenyl)-urea 314463 3-[4-({4-[3-(2-Fluoro-5-trifluoromethyl-phenyl)-ureido]-phenyl}-methyl-amino)-pyrimidin-2-ylamino]-benzenesulfonamide 314464 4-[4-({4-[3-(2-Fluoro-5-trifluoromethyl-phenyl)-ureido]-phenyl}-methyl-amino)-pyrimidin-2-ylamino]-benzenesulfonamide 314465 TCMDC-138736 314466 1-(4-{[2-(3-Methanesulfonylmethyl-phenylamino)-pyrimidin-4-yl]-methyl-amino}-phenyl)-3-(4-trifluoromethoxy-phenyl)-urea 314467 3-[4-(Methyl-{4-[3-(4-trifluoromethoxy-phenyl)-ureido]-phenyl}-amino)-pyrimidin-2-ylamino]-benzenesulfonamide 314468 4-[4-(Methyl-{4-[3-(4-trifluoromethoxy-phenyl)-ureido]-phenyl}-amino)-pyrimidin-2-ylamino]-benzenesulfonamide 314469 3-Methoxy-N-{3-[5-(2-methyl-benzoyl)-thiazol-2-ylamino]-propyl}-benzenesulfonamide 314483 (S)-3-{[5-(4-Ethoxy-phenyl)-thiophene-2-carbonyl]-methyl-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 314499 (S)-3-{Methyl-[5-(2-trifluoromethyl-phenyl)-thiophene-2-carbonyl]-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 314500 (1S,4R,6S)-2-Aza-bicyclo[2.2.2]octane-6-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide 314501 (1S,4S,6S)-2-Aza-bicyclo[2.2.2]octane-6-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide 314503 4-(1-Ethyl-6-fluoro-1H-benzoimidazol-2-yl)-furazan-3-ylamine 314504 4-(1-Ethyl-4-methoxy-1H-imidazo[4,5-c]pyridin-2-yl)-furazan-3-ylamine 314505 4-(4-Ethoxy-1-ethyl-1H-imidazo[4,5-c]pyridin-2-yl)-furazan-3-ylamine 314515 2,5-Dimethoxy-N-{3-[4-(2-methyl-benzoyl)-thiazol-2-ylamino]-propyl}-benzenesulfonamide 314518 (S)-3-{[5-(4-Ethyl-phenyl)-thiophene-2-carbonyl]-methyl-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 314533 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-3-yl)-3-methoxy-benzamide 314535 4-(3-Ethyl-3H-imidazo[4,5-c]pyridin-2-yl)-furazan-3-ylamine 314537 4-(1-Ethyl-4-phenyl-1H-imidazo[4,5-c]pyridin-2-yl)-furazan-3-ylamine 314546 Thiophene-2-sulfonic acid {3-[5-(2-methyl-benzoyl)-thiazol-2-ylamino]-propyl}-amide 314551 2-Chloro-N-{3-[4-(2-methyl-benzoyl)-thiazol-2-ylamino]-propyl}-5-trifluoromethyl-benzenesulfonamide 314553 (S)-3-{[5-(2,4-Dichloro-phenyl)-thiophene-2-carbonyl]-methyl-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 314558 4-(1H-Imidazo[4,5-c]pyridin-2-yl)-furazan-3-ylamine 314561 N-arylpiperazine derivative 314563 N-(4-{[2-(3-Methanesulfonylmethyl-phenylamino)-pyrimidin-4-yl]-methyl-amino}-phenyl)-2-phenyl-acetamide 314564 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-2-(4'-methoxy-biphenyl-4-yl)-acetamide 314565 3-Amino-N-[(R)-2-[4-(1-{[2-(4-chloro-phenyl)-acetylamino]-methyl}-cyclohexyl)-piperazin-1-yl]-1-(2,4-dichloro-benzyl)-2-oxo-ethyl]-propionamide 314566 3-Amino-N-{(R)-1-(2,4-dichloro-benzyl)-2-[4-(1-{[2-(3-methoxy-phenyl)-acetylamino]-methyl}-cyclohexyl)-piperazin-1-yl]-2-oxo-ethyl}-propionamide 314567 (R)-3-amino-N-(3-(2,4-dichlorophenyl)-1-(4-(1-((2-(4-methoxyphenyl)acetamido)methyl)cyclohexyl)piperazin-1-yl)-1-oxopropan-2-yl)propanamide 314568 3-Amino-N-{(R)-1-(2,4-dichloro-benzyl)-2-[4-(1-{[2-(3,4-dimethoxy-phenyl)-acetylamino]-methyl}-cyclohexyl)-piperazin-1-yl]-2-oxo-ethyl}-propionamide 314569 3-Amino-N-[(R)-1-(2,4-dichloro-benzyl)-2-oxo-2-(4-{1-[(2-thiophen-2-yl-acetylamino)-methyl]-cyclohexyl}-piperazin-1-yl)-ethyl]-propionamide 314570 (S)-3-{[5-(2-Chloro-phenyl)-thiophene-2-carbonyl]-methyl-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 314571 4-(1-Cyclohexyl-1H-imidazo[4,5-c]pyridin-2-yl)-furazan-3-ylamine 314596 8-(4-methoxyphenyl)-2-morpholin-4-yl-chromen-4-one 314597 8-(4-hydroxymethylphenyl)-2-morpholin-4-ylchromen-4-one 314602 4-[3-(1-{4-[(R)-2-(3-Amino-propionylamino)-3-(2,4-dichloro-phenyl)-propionyl]-piperazin-1-yl}-cyclohexylmethyl)-ureido]-benzoic acid methyl ester 314603 3-Amino-N-[(R)-1-(2,4-dichloro-benzyl)-2-oxo-2-(4-{1-[(2,2,2-trifluoro-acetylamino)-methyl]-cyclohexyl}-piperazin-1-yl)-ethyl]-propionamide 314635 1-Ethyl-3-(4-{[2-(4-methanesulfonylmethyl-phenylamino)-pyrimidin-4-yl]-methyl-amino}-phenyl)-urea 314637 3-Amino-N-((R)-1-(2,4-dichloro-benzyl)-2-{4-[1-(isobutylamino-methyl)-cyclohexyl]-piperazin-1-yl}-2-oxo-ethyl)-propionamide 314638 3-Amino-N-[(R)-1-(2,4-dichloro-benzyl)-2-(4-{1-[(3,3-dimethyl-butylamino)-methyl]-cyclohexyl}-piperazin-1-yl)-2-oxo-ethyl]-propionamide 314642 4-(1-Ethyl-5-methoxy-1H-benzoimidazol-2-yl)-furazan-3-ylamine 314645 1-(4-{[2-(3-Methanesulfonylmethyl-phenylamino)-pyrimidin-4-yl]-methyl-amino}-phenyl)-3-phenyl-thiourea 314652 (S)-3-[Methyl-(5-p-tolyl-thiophene-2-carbonyl)-amino]-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 314653 (S)-3-{[5-(4-Dimethylamino-phenyl)-thiophene-2-carbonyl]-methyl-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 314670 (S)-3-{[5-(4-Methoxy-2-methyl-phenyl)-thiophene-2-carbonyl]-methyl-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 314674 1-[2-(4-Amino-furazan-3-yl)-1-ethyl-1H-imidazo[4,5-c]pyridin-7-ylmethyl]-piperidin-4-ylamine 314675 4-(1-Piperidin-4-yl-1H-imidazo[4,5-c]pyridin-2-yl)-furazan-3-ylamine 314676 4-[1-(1-Amino-butyl)-1H-imidazo[4,5-c]pyridin-2-yl]-furazan-3-ylamine 314678 8-(5-acetylthiophen-2-yl)-2-morpholin-4-ylchromen-4-one 314679 8-benzo[b]thiophen-2-yl-2-morpholin-4-ylchromen-4-one 314684 (S)-3-{[5-(4-Methanesulfonyl-phenyl)-thiophene-2-carbonyl]-methyl-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 314685 4-Fluoro-N-{3-[5-(2-methyl-benzoyl)-thiazol-2-ylamino]-propyl}-benzenesulfonamide 314704 (S)-3-{[5-(2-Chloro-4-methyl-phenyl)-thiophene-2-carbonyl]-methyl-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 314713 3-Amino-N-[(R)-1-(2,4-dichloro-benzyl)-2-(4-{1-[(4-fluoro-benzylamino)-methyl]-cyclohexyl}-piperazin-1-yl)-2-oxo-ethyl]-propionamide 314714 3-Amino-N-[(R)-2-(4-{1-[(4-cyano-benzylamino)-methyl]-cyclohexyl}-piperazin-1-yl)-1-(2,4-dichloro-benzyl)-2-oxo-ethyl]-propionamide 314715 3-Amino-N-[(R)-1-(2,4-dichloro-benzyl)-2-(4-{1-[(4-dimethylamino-benzylamino)-methyl]-cyclohexyl}-piperazin-1-yl)-2-oxo-ethyl]-propionamide 314716 3-Amino-N-[(R)-1-(2,4-dichloro-benzyl)-2-oxo-2-(4-{1-[(4-trifluoromethyl-benzylamino)-methyl]-cyclohexyl}-piperazin-1-yl)-ethyl]-propionamide 314717 3-Amino-N-[(R)-1-(2,4-dichloro-benzyl)-2-oxo-2-(4-{1-[(4-trifluoromethoxy-benzylamino)-methyl]-cyclohexyl}-piperazin-1-yl)-ethyl]-propionamide 314718 (R)-3-{Methyl-[5-(4-trifluoromethyl-phenyl)-thiophene-2-carbonyl]-amino}-pyrrolidine-1-carboxylic acid methyl-((S)-1-methyl-pyrrolidin-3-yl)-amide 314719 3-Methoxy-N-[1-((E)-3-phenyl-allyl)-piperidin-4-yl]-benzamide 314720 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-2-biphenyl-4-yl-acetamide 314721 N-(1-{4-[(R)-2-(3-Amino-propionylamino)-3-(2,4-dichloro-phenyl)-propionyl]-piperazin-1-yl}-cyclohexylmethyl)-4-chloro-benzamide 314722 N-(1-{4-[(R)-2-(3-Amino-propionylamino)-3-(2,4-dichloro-phenyl)-propionyl]-piperazin-1-yl}-cyclohexylmethyl)-4-bromo-benzamide 314723 (R)-N-((1-(4-(2-(3-aminopropanamido)-3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)cyclohexyl)methyl)-4-methoxybenzamide 314724 N-(1-{4-[(R)-2-(3-Amino-propionylamino)-3-(2,4-dichloro-phenyl)-propionyl]-piperazin-1-yl}-cyclohexylmethyl)-2-methoxy-benzamide 314725 N-(1-{4-[(R)-2-(3-Amino-propionylamino)-3-(2,4-dichloro-phenyl)-propionyl]-piperazin-1-yl}-cyclohexylmethyl)-4-trifluoromethoxy-benzamide 314727 [2-(4-Amino-furazan-3-yl)-1-ethyl-1H-benzoimidazol-5-yl]-methanol 314730 N-(4-{[2-(3-Methanesulfonylmethyl-phenylamino)-pyrimidin-4-yl]-methyl-amino}-phenyl)-N'-phenyl-guanidine 314731 1-(2-Fluoro-5-trifluoromethyl-phenyl)-3-(4-{[2-(3-methanesulfonylmethyl-phenylamino)-pyrimidin-4-yl]-methyl-amino}-phenyl)-urea 314754 (S)-3-{Methyl-[5-(3-trifluoromethyl-phenyl)-thiophene-2-carbonyl]-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 314756 (1R,4S,6R)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide 314757 (1R,4S,6S)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide 314758 4-(1-Ethyl-5-fluoro-1H-benzoimidazol-2-yl)-furazan-3-ylamine 314759 4-(4-Chloro-1-ethyl-1H-imidazo[4,5-c]pyridin-2-yl)-furazan-3-ylamine 314760 4-(1,4-Diethyl-1H-imidazo[4,5-c]pyridin-2-yl)-furazan-3-ylamine 314761 8-dibenzofuran-4-yl-2-morpholin-4-ylchromen-4-one 314770 1-Cyclopentyl-3-(4-{[2-(3-methanesulfonylmethyl-phenylamino)-pyrimidin-4-yl]-methyl-amino}-phenyl)-urea 314777 (S)-3-{[5-(4-Fluoro-phenyl)-thiophene-2-carbonyl]-methyl-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 314778 2-Chloro-N-{3-[5-(2-methyl-benzoyl)-thiazol-2-ylamino]-propyl}-5-trifluoromethyl-benzenesulfonamide 314783 (S)-3-[Methyl-(5-o-tolyl-thiophene-2-carbonyl)-amino]-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 314784 (S)-3-{[5-(4-Isopropoxy-phenyl)-thiophene-2-carbonyl]-methyl-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 314789 4-(1-Ethyl-1H-imidazo[4,5-c]pyridin-2-yl)-1,5-dimethyl-1H-pyrazol-3-ylamine 314793 1-(4-{[2-(3-Methanesulfonylmethyl-phenylamino)-pyrimidin-4-yl]-methyl-amino}-phenyl)-3-phenyl-urea 314796 2-(4-Amino-furazan-3-yl)-3-ethyl-3H-benzoimidazol-5-ol 314797 4-(1-ethyl-1H-imidazo[4,5-c]pyridin-2-yl)-1,2,5-oxadiazol-3-amine 314798 4-(1-Ethyl-4-phenoxy-1H-imidazo[4,5-c]pyridin-2-yl)-furazan-3-ylamine 314823 N-[4-(1-Ethyl-1H-imidazo[4,5-c]pyridin-2-yl)-furazan-3-yl]-acetamide 314824 4-(7-Bromo-1-ethyl-1H-imidazo[4,5-c]pyridin-2-yl)-furazan-3-ylamine 314828 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-2-(3'-methoxy-biphenyl-4-yl)-acetamide 314829 Thiophene-2-carboxylic acid (1-{4-[(R)-2-(3-amino-propionylamino)-3-(2,4-dichloro-phenyl)-propionyl]-piperazin-1-yl}-cyclohexylmethyl)-amide 314830 1,6-Dihydro-pyridine-3-carboxylic acid (1-{4-[2-((R)-3-amino-propionylamino)-3-(2,4-dichloro-phenyl)-propionyl]-piperazin-1-yl}-cyclohexylmethyl)-amide 314832 3-Amino-N-((R)-1-(2,4-dichloro-benzyl)-2-oxo-2-{4-[1-(phenylacetylamino-methyl)-cyclohexyl]-piperazin-1-yl}-ethyl)-propionamide 314833 3-Amino-N-{(R)-1-(2,4-dichloro-benzyl)-2-[4-(1-{[2-(4-fluoro-phenyl)-acetylamino]-methyl}-cyclohexyl)-piperazin-1-yl]-2-oxo-ethyl}-propionamide 314834 (S)-3-{[5-(3-Chloro-phenyl)-thiophene-2-carbonyl]-methyl-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 314836 4-(1-Ethyl-4-pyrrolidin-1-yl-1H-imidazo[4,5-c]pyridin-2-yl)-furazan-3-ylamine 314837 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-3-yl)-3,5-dimethoxy-benzamide 314841 2-Methoxy-5-methyl-N-{3-[5-(2-methyl-benzoyl)-thiazol-2-ylamino]-propyl}-benzenesulfonamide 314851 2-Methoxy-5-methyl-N-{3-[4-(2-methyl-benzoyl)-thiazol-2-ylamino]-propyl}-benzenesulfonamide 314858 3-Amino-N-[2-[4-(1-aminomethyl-cyclohexyl)-piperazin-1-yl]-1-(2,4-dichloro-benzyl)-2-oxo-ethyl]-propionamide 314864 (1S,4R,6S)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide 314865 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-2-(3'-cyano-biphenyl-4-yl)-acetamide 314866 3-Amino-N-[(R)-1-(2,4-dichloro-benzyl)-2-(4-{1-[3-(4-fluoro-phenyl)-ureidomethyl]-cyclohexyl}-piperazin-1-yl)-2-oxo-ethyl]-propionamide 314867 3-Amino-N-[(R)-2-(4-{1-[3-(4-chloro-phenyl)-ureidomethyl]-cyclohexyl}-piperazin-1-yl)-1-(2,4-dichloro-benzyl)-2-oxo-ethyl]-propionamide 314868 (R)-1-((1-(4-(2-(3-aminopropanamido)-3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)cyclohexyl)methyl)-3-(4-methoxyphenyl)urea 314869 3-Amino-N-[(R)-1-(2,4-dichloro-benzyl)-2-(4-{1-[3-(4-dimethylamino-phenyl)-ureidomethyl]-cyclohexyl}-piperazin-1-yl)-2-oxo-ethyl]-propionamide 314870 3-Amino-N-[(R)-1-(2,4-dichloro-benzyl)-2-(4-{1-[3-(4-nitro-phenyl)-ureidomethyl]-cyclohexyl}-piperazin-1-yl)-2-oxo-ethyl]-propionamide 314871 (S)-3-{[5-(3-Methoxy-phenyl)-thiophene-2-carbonyl]-methyl-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 314895 (S)-3-{[5-(2-Methoxy-phenyl)-thiophene-2-carbonyl]-methyl-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 314899 (S)-3-{[5-(4-Methoxy-phenyl)-thiophene-2-carbonyl]-methyl-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 314910 2-morpholin-4-yl-8-thiophen-2-ylchromen-4-one 314913 (4-{[2-(3-Methanesulfonylmethyl-phenylamino)-pyrimidin-4-yl]-methyl-amino}-phenyl)-carbamic acid phenyl ester 314914 4-(1-Cyclopropyl-1H-imidazo[4,5-c]pyridin-2-yl)-furazan-3-ylamine 314929 (S)-3-{[5-(4-Chloro-2-methyl-phenyl)-thiophene-2-carbonyl]-methyl-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 314933 4-(1-Methyl-1H-imidazo[4,5-c]pyridin-2-yl)-furazan-3-ylamine 314934 4-(1-Ethyl-7-piperidin-1-ylmethyl-1H-imidazo[4,5-c]pyridin-2-yl)-furazan-3-ylamine 314938 2-morpholin-4-yl-8-thiophen-3-ylchromen-4-one 314939 1-Butyl-3-(4-{[2-(3-methanesulfonylmethyl-phenylamino)-pyrimidin-4-yl]-methyl-amino}-phenyl)-urea 314943 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-3-yl)-3,5-dichloro-benzamide 314954 (S)-3-{[5-(4-Isopropyl-phenyl)-thiophene-2-carbonyl]-methyl-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 314960 3-Fluoro-N-{3-[4-(2-methyl-benzoyl)-thiazol-2-ylamino]-propyl}-benzenesulfonamide 314966 4-(1-Ethyl-7-piperazin-1-ylmethyl-1H-imidazo[4,5-c]pyridin-2-yl)-furazan-3-ylamine 314968 3-Amino-N-[(R)-2-(4-{1-[(cyclohexylmethyl-amino)-methyl]-cyclohexyl}-piperazin-1-yl)-1-(2,4-dichloro-benzyl)-2-oxo-ethyl]-propionamide 314969 3-Amino-N-[(R)-1-(2,4-dichloro-benzyl)-2-oxo-2-(4-{1-[(3-phenyl-propylamino)-methyl]-cyclohexyl}-piperazin-1-yl)-ethyl]-propionamide 314970 3-Amino-N-((R)-1-(2,4-dichloro-benzyl)-2-oxo-2-{4-[1-(phenethylamino-methyl)-cyclohexyl]-piperazin-1-yl}-ethyl)-propionamide 314971 3-Amino-N-[(R)-2-{4-[1-(benzylamino-methyl)-cyclohexyl]-piperazin-1-yl}-1-(2,4-dichloro-benzyl)-2-oxo-ethyl]-propionamide 314972 3-Amino-N-[(R)-1-(2,4-dichloro-benzyl)-2-(4-{1-[(2-fluoro-benzylamino)-methyl]-cyclohexyl}-piperazin-1-yl)-2-oxo-ethyl]-propionamide 314973 4-(1-ethyl-1H-benzo[d]imidazol-2-yl)-1,2,5-oxadiazol-3-amine 314974 4-(1-Phenyl-1H-imidazo[4,5-c]pyridin-2-yl)-furazan-3-ylamine 314975 N-((2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-1H-imidazo[4,5-c]pyridin-7-yl)methyl)piperidin-4-amine 314976 1-[2-(4-Amino-furazan-3-yl)-1-ethyl-1H-benzoimidazol-5-yl]-ethanone 314977 4-(1-Ethyl-4-methyl-1H-imidazo[4,5-c]pyridin-2-yl)-furazan-3-ylamine 314980 N-(4-{[2-(3-Methanesulfonylmethyl-phenylamino)-pyrimidin-4-yl]-methyl-amino}-phenyl)-C-phenyl-methanesulfonamide 314982 (S)-3-[(4'-Chloro-biphenyl-4-carbonyl)-methyl-amino]-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 314995 (S)-3-{Methyl-[5-(4-trifluoromethoxy-phenyl)-thiophene-2-carbonyl]-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 315010 (S)-3-{Methyl-[5-(4-trifluoromethyl-phenyl)-thiophene-2-carbonyl]-amino}-pyrrolidine-1-carboxylic acid methyl-((S)-1-methyl-pyrrolidin-3-yl)-amide 315015 3-Amino-N-{(R)-1-(2,4-dichloro-benzyl)-2-oxo-2-[4-(1-{[(thiophen-2-ylmethyl)-amino]-methyl}-cyclohexyl)-piperazin-1-yl]-ethyl}-propionamide 315017 3-Amino-N-{1-(2,4-dichloro-benzyl)-2-[4-(1-{[(1,6-dihydro-pyridin-2-ylmethyl)-amino]-methyl}-cyclohexyl)-piperazin-1-yl]-2-oxo-ethyl}-propionamide 315018 N-(1-{4-[(R)-2-(3-Amino-propionylamino)-3-(2,4-dichloro-phenyl)-propionyl]-piperazin-1-yl}-cyclohexylmethyl)-benzamide 315019 N-(1-{4-[(R)-2-(3-Amino-propionylamino)-3-(2,4-dichloro-phenyl)-propionyl]-piperazin-1-yl}-cyclohexylmethyl)-4-fluoro-benzamide 315020 (E)-N-(1-cinnamylpiperidin-4-yl)-3,5-dimethoxybenzamide 315023 8-(dibenzo[b,d]thiophen-4-yl)-2-morpholino-4H-chromen-4-one 315027 (S)-3-{[5-(4-Cyano-phenyl)-thiophene-2-carbonyl]-methyl-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 315030 2,5-Dimethoxy-N-{3-[5-(2-methyl-benzoyl)-thiazol-2-ylamino]-propyl}-benzenesulfonamide 315052 (R)-3-{Methyl-[5-(4-trifluoromethyl-phenyl)-thiophene-2-carbonyl]-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 315067 2-(3-chlorophenyl)-1-(2-methyl-1-pentyl-1H-indol-3-yl)ethanone 315069 2-(2-bromophenyl)-1-(1-pentyl-1H-indol-3-yl)ethanone 315070 2-(2-bromophenyl)-1-(2-methyl-1-pentyl-1H-indol-3-yl)ethanone 315073 (S)-1-(4-Fluoro-phenyl)-piperazine-2-carboxylic acid {(S)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315074 6-(4-Chloro-phenylsulfanyl)-4-((R)-3-{[(4R,5S)-4-(4-fluoro-phenyl)-piperidin-3-ylmethyl]-amino}-butyl)-2-(4-methoxy-phenyl)-2H-pyridazin-3-one 315075 6-(4-Chloro-phenylsulfanyl)-4-((R)-3-{[(4S,5R)-4-(4-fluoro-phenyl)-piperidin-3-ylmethyl]-amino}-butyl)-2-(4-methoxy-phenyl)-2H-pyridazin-3-one 315094 1-(2-Dimethylamino-ethyl)-3-(4-{[2-(3-methanesulfonylmethyl-phenylamino)-pyrimidin-4-yl]-methyl-amino}-phenyl)-urea 315096 (S)-3-[(4'-Methoxy-2'-methyl-biphenyl-4-carbonyl)-methyl-amino]-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 315101 Trans 4-(4-Fluoro-phenyl)-piperidine-3-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-methyl-amide 315102 (4R,5S)-4-(4-Fluoro-phenyl)-1-methyl-piperidine-3-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315111 3-Cyclopentyl-N-(2-dimethylamino-ethyl)-N-{4'-[(2-pyridin-2-yl-ethylamino)-methyl]-biphenyl-4-ylmethyl}-propionamide TFA 315112 3-Cyclopentyl-N-(2-dimethylamino-ethyl)-N-{4'-[(2-phenoxy-ethylamino)-methyl]-biphenyl-4-ylmethyl}-propionamide TFA 315113 3-Cyclopentyl-N-[4'-(phenethylamino-methyl)-biphenyl-4-ylmethyl]-N-piperidin-2-ylmethyl-propionamide TFA 315117 (E)-N-(2-Dimethylamino-ethyl)-N-{4-[5-(phenethylamino-methyl)-pyridin-2-yl]-benzyl}-3-phenyl-acrylamide 315143 2-(3-methoxyphenyl)-1-(1-pentyl-1H-indol-3-yl)ethanone 315148 2-(3-fluorophenyl)-1-(1-pentyl-1H-indol-3-yl)ethanone 315151 4-{3-[2-(1H-Indol-3-yl)-ethylsulfanyl]-5-quinoxalin-2-yl-[1,2,4]triazol-4-yl}-butylamine 315156 4-{3-[2-(6-Fluoro-1H-indol-3-yl)-ethylsulfanyl]-5-quinolin-2-yl-[1,2,4]triazol-4-yl}-butylamine 315177 2-(3-methoxyphenyl)-1-(2-methyl-1-pentyl-1H-indol-3-yl)ethanone 315180 2-(3-fluorophenyl)-1-(2-methyl-1-pentyl-1H-indol-3-yl)ethanone 315185 (4R,5S)-4-(2,4-Dichloro-phenyl)-piperidine-3-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315186 (4R,5S)-4-(4-Fluoro-phenyl)-piperidine-3-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315187 (4R,5S)-4-(3-Fluoro-phenyl)-piperidine-3-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315188 (4R,5S)-4-(2-Fluoro-phenyl)-piperidine-3-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315196 N-(2,5-Dimethoxy-benzyl)-2-phenoxy-nicotinamide 315202 4-(1-Ethyl-1H-imidazo[4,5-c]pyridin-2-yl)-5-methyl-1H-pyrazol-3-ylamine 315203 4-[1-(3-Aminomethyl-phenyl)-1H-imidazo[4,5-c]pyridin-2-yl]-furazan-3-ylamine 315208 2-(4-Bromo-phenyl)-1-(2-methyl-1-pentyl-1H-indol-3-yl)-ethanone 315209 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-3-yl)-3-trifluoromethoxy-benzamide 315211 (E)-N-[2-(3-Methoxy-phenyl)-ethyl]-N-[4'-(phenethylamino-methyl)-biphenyl-4-ylmethyl]-3-phenyl-acrylamide TFA 315212 (E)-N-{4'-[(2-Methoxy-ethylamino)-methyl]-biphenyl-4-ylmethyl}-3-phenyl-N-pyridin-3-ylmethyl-acrylamide TFA 315213 (E)-N-(4'-{[(Benzo[1,3]dioxol-5-ylmethyl)-amino]-methyl}-biphenyl-4-ylmethyl)-3-phenyl-N-pyridin-3-ylmethyl-acrylamide TFA 315214 N-(2-Dimethylamino-ethyl)-N-[4'-(phenethylamino-methyl)-biphenyl-4-ylmethyl]-benzamide TFA 315215 1-(2-Dimethylamino-ethyl)-1-[4'-(phenethylamino-methyl)-biphenyl-4-ylmethyl]-3-phenyl-urea TFA 315216 1-(2-methyl-1-pentyl-1H-indol-3-yl)-2-phenylethanone 315225 (4R,5S)-4-(4-Trifluoromethyl-phenyl)-piperidine-3-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315226 (4R,5S)-4-(3-Trifluoromethyl-phenyl)-piperidine-3-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315230 (2-Chloro-benzyl)-(5-nitro-4-phenoxy-1H-indazol-3-yl)-amine 315234 N-(2-Chloro-benzyl)-2-(2-fluoro-phenoxy)-nicotinamide 315237 4-[1-(4-Amino-butyl)-1H-imidazo[4,5-c]pyridin-2-yl]-furazan-3-ylamine 315238 4-[1-(3-Amino-propyl)-1H-imidazo[4,5-c]pyridin-2-yl]-furazan-3-ylamine 315239 1-(4-{[2-(3-Methanesulfonylmethyl-phenylamino)-pyrimidin-4-yl]-methyl-amino}-phenyl)-3-phenethyl-urea 315240 4-[1-(4-Aminomethyl-phenyl)-1H-imidazo[4,5-c]pyridin-2-yl]-furazan-3-ylamine 315242 1-[2-[((R)-1-Amino-indane-2-carbonyl)-amino]-3-(4-chloro-phenyl)-propionyl]-4-cyclohexyl-piperidine-4-carboxylic acid tert-butylamide 315243 1-[2-[((R)-3-Amino-1,2,3,4-tetrahydro-naphthalene-2-carbonyl)-amino]-3-(4-chloro-phenyl)-propionyl]-4-cyclohexyl-piperidine-4-carboxylic acid tert-butylamide 315245 1-[(R)-2-[((1R,2R)-1-Amino-1,2,3,4-tetrahydro-naphthalene-2-carbonyl)-amino]-3-(4-chloro-phenyl)-propionyl]-4-cyclohexyl-piperidine-4-carboxylic acid tert-butylamide 315246 1-[(R)-2-[((1S,2S)-1-Amino-1-methyl-1,2,3,4-tetrahydro-naphthalene-2-carbonyl)-amino]-3-(4-chloro-phenyl)-propionyl]-4-cyclohexyl-piperidine-4-carboxylic acid tert-butylamide 315249 (2R,3S)-3-Benzyl-piperidine-4-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315250 (2R,3S)-3-(4-Fluoro-benzyl)-piperidine-4-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315251 (4R,5S)-4-(2-Fluoro-phenyl)-pyrrolidine-3-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315252 (4R,5S)-4-(4-Fluoro-phenyl)-pyrrolidine-3-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315257 1-(1-pentyl-1H-indol-3-yl)-2-p-tolylethanone 315258 1-(2-methyl-1-pentyl-1H-indol-3-yl)-2-p-tolylethanone 315266 N-(2-Dimethylamino-ethyl)-N-{6-[4-(phenethylamino-methyl)-phenyl]-pyridin-3-ylmethyl}-3-phenyl-acrylamide 315271 4-{3-(6-Fluoro-quinolin-2-yl)-5-[2-(1H-indol-3-yl)-ethylsulfanyl]-[1,2,4]triazol-4-yl}-butylamine 315275 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-3-yl)-3,5-dimethoxy-4-methyl-benzamide 315277 1-(4-{[2-(4-Methanesulfonylmethyl-phenylamino)-pyrimidin-4-yl]-methyl-amino}-phenyl)-3-(2-morpholin-4-yl-ethyl)-urea 315278 4-(3-Morpholin-4-yl-propyl)-piperazine-1-carboxylic acid (4-{[2-(4-methanesulfonylmethyl-phenylamino)-pyrimidin-4-yl]-methyl-amino}-phenyl)-amide 315279 1-(4-{[2-(4-Methanesulfonylmethyl-phenylamino)-pyrimidin-4-yl]-methyl-amino}-phenyl)-3-[4-(4-methyl-piperazin-1-ylmethyl)-phenyl]-urea 315281 (S)-3-{[5-(4-Chloro-phenyl)-thiophene-2-carbonyl]-methyl-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 315294 (1-Benzyl-piperidin-4-yl)-[4'-(phenethylamino-methyl)-biphenyl-3-ylmethyl]-amine 315299 2-(4-fluorophenyl)-1-(1-pentyl-1H-indol-3-yl)ethanone 315303 N-(2-Chloro-benzyl)-2-phenoxy-nicotinamide 315308 (S)-3-[(4'-Methoxy-biphenyl-4-carbonyl)-methyl-amino]-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 315314 2-(2-chlorophenyl)-1-(1-pentyl-1H-indol-3-yl)ethanone 315315 2-(2-chlorophenyl)-1-(2-methyl-1-pentyl-1H-indol-3-yl)ethanone 315316 1-(1-pentyl-1H-indol-3-yl)-2-phenylethanone 315328 N-(4'-Aminomethyl-biphenyl-4-ylmethyl)-3-cyclopentyl-N-(2-dimethylamino-ethyl)-propionamide TFA 315329 3-Cyclopentyl-N-(2-dimethylamino-ethyl)-N-[4'-(indan-2-ylaminomethyl)-biphenyl-4-ylmethyl]-propionamide TFA 315334 2-(2-fluorophenyl)-1-(1-pentyl-1H-indol-3-yl)ethanone 315338 2-(4-Fluoro-phenyl)-1-(2-methyl-1-pentyl-1H-indol-3-yl)-ethanone 315342 N-{4-[(4-Phenoxy-1H-pyrazolo[4,3-c]pyridin-3-ylamino)-methyl]-phenyl}-acetamide 315355 2-(4-chlorophenyl)-1-(1-pentyl-1H-indol-3-yl)ethanone 315356 2-(4-chlorophenyl)-1-(2-methyl-1-pentyl-1H-indol-3-yl)ethanone 315358 (S)-1-(4-Fluoro-phenyl)-piperazine-2-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315359 (R)-1-(4-Fluoro-phenyl)-piperazine-2-carboxylic acid {(S)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315365 2-(2-methoxyphenyl)-1-(1-pentyl-1H-indol-3-yl)ethanone 315368 2-(2-fluorophenyl)-1-(2-methyl-1-pentyl-1H-indol-3-yl)ethanone 315394 2-(2-methoxyphenyl)-1-(2-methyl-1-pentyl-1H-indol-3-yl)ethanone 315405 (4R,5S)-4-Phenyl-piperidine-3-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315406 (4R,5S)-4-(4-Chloro-phenyl)-piperidine-3-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315407 (4R,5S)-4-(3-Chloro-phenyl)-piperidine-3-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315416 1-(2,6-Dichloro-phenyl)-3-(4-{[2-(3-methanesulfonylmethyl-phenylamino)-pyrimidin-4-yl]-methyl-amino}-phenyl)-urea 315417 3-(1-Ethyl-1H-imidazo[4,5-c]pyridin-2-yl)-pyrazin-2-ylamine 315418 (R,S)-4-[1-(2-Amino-1-methyl-ethyl)-1H-imidazo[4,5-c]pyridin-2-yl]-furazan-3-ylamine 315432 (E)-N-(2-Dimethylamino-ethyl)-N-[4'-(phenethylamino-methyl)-biphenyl-4-ylmethyl]-3-phenyl-acrylamide TFA 315433 (E)-N-[4'-(Phenethylamino-methyl)-biphenyl-4-ylmethyl]-3-phenyl-N-pyridin-3-ylmethyl-acrylamide TFA 315439 (E)-2-Phenyl-ethenesulfonic acid (2-dimethylamino-ethyl)-[4'-(phenethylamino-methyl)-biphenyl-4-ylmethyl]-amide TFA 315449 2-Phenoxy-N-((S)-1-phenyl-ethyl)-nicotinamide 315454 1-(2-Dimethylamino-ethyl)-3-(4-{[2-(4-methanesulfonylmethyl-phenylamino)-pyrimidin-4-yl]-methyl-amino}-phenyl)-urea 315458 1-[(R)-2-[((1S,2S)-1-Amino-1,2,3,4-tetrahydro-naphthalene-2-carbonyl)-amino]-3-(4-chloro-phenyl)-propionyl]-4-cyclohexyl-piperidine-4-carboxylic acid tert-butylamide 315467 2-(4-bromophenyl)-1-(1-pentyl-1H-indol-3-yl)ethanone 315474 (1-Benzyl-piperidin-4-yl)-[4'-(phenethylamino-methyl)-biphenyl-4-ylmethyl]-amine 315478 3-Cyclopentyl-N-(2-dimethylamino-ethyl)-N-{4-[5-(phenethylamino-methyl)-pyridin-2-yl]-benzyl}-propionamide 315481 4-{3-[2-(1H-Indol-3-yl)-ethylsulfanyl]-5-quinolin-2-yl-[1,2,4]triazol-4-yl}-butylamine 315491 4-{3-[2-(1H-Indol-3-yl)-ethylsulfanyl]-5-naphthalen-2-yl-[1,2,4]triazol-4-yl}-butylamine 315493 (S)-3-{Methyl-[5-(4-trifluoromethyl-phenyl)-thiophene-2-carbonyl]-amino}-pyrrolidine-1-carboxylic acid methyl-((R)-1-methyl-pyrrolidin-3-yl)-amide 315497 (2S,3S)-3-(4-Chloro-phenyl)-piperidine-4-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315501 1-(2-methyl-1-pentyl-1H-indol-3-yl)-2-o-tolylethanone 315509 2-(4-methoxyphenyl)-1-(1-pentyl-1H-indol-3-yl)ethanone 315515 Thiophene-2-sulfonic acid {3-[4-(2-methyl-benzoyl)-thiazol-2-ylamino]-propyl}-amide 315521 4-{3-[2-(7-Chloro-1H-indol-3-yl)-ethylsulfanyl]-5-quinolin-2-yl-[1,2,4]triazol-4-yl}-butylamine 315524 (2S,3S)-3-(2,4-Dichloro-phenyl)-piperidine-4-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315525 (2S,3S)-3-(4-Fluoro-phenyl)-piperidine-4-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315526 (2S,3S)-3-(2-Fluoro-phenyl)-piperidine-4-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315527 (2S,3S)-3-(4-Trifluoromethyl-phenyl)-piperidine-4-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315528 (2S,3S)-3-(4-Cyano-phenyl)-piperidine-4-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315532 (4R,5S)-4-(2,4-Difluoro-phenyl)-pyrrolidine-3-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315533 (4R,5S)-4-(4-Chloro-phenyl)-pyrrolidine-3-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315534 (4R,5S)-4-p-Tolyl-pyrrolidine-3-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315535 (4R,5S)-4-(4-Methoxy-phenyl)-pyrrolidine-3-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315536 (R)-1-(4-Fluoro-phenyl)-piperazine-2-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315543 Benzo[1,3]dioxole-5-carboxylic acid [4'-(phenethylamino-methyl)-biphenyl-4-ylmethyl]-pyridin-3-ylmethyl-amide TFA 315544 2-Phenyl-cyclopropanecarboxylic acid (2-dimethylamino-ethyl)-[4'-(phenethylamino-methyl)-biphenyl-4-ylmethyl]-amide TFA 315545 3-Cyclopentyl-N-(2-dimethylamino-ethyl)-N-[4'-(phenethylamino-methyl)-biphenyl-4-ylmethyl]-propionamide with di TFA 315549 2-(4-methoxyphenyl)-1-(2-methyl-1-pentyl-1H-indol-3-yl)ethanone 315562 SID17432479 315563 N*3*-(2-Chloro-benzyl)-4-phenoxy-1H-indazole-3,5-diamine 315568 N-(2-Chloro-benzyl)-2-(4-methoxy-phenoxy)-nicotinamide 315570 3-(1-Ethyl-1H-imidazo[4,5-c]pyridin-2-yl)-pyridin-2-ylamine 315574 3-Cyclopentyl-N-(2-dimethylamino-ethyl)-N-{6-[4-(phenethylamino-methyl)-phenyl]-pyridin-3-ylmethyl}-propionamide 315588 (4R,5S)-4-p-Tolyl-piperidine-3-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315590 (4R,5S)-4-Naphthalen-2-yl-piperidine-3-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315591 (4R,5S)-4-Naphthalen-1-yl-piperidine-3-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315592 (4R,5S)-4-Thiophen-3-yl-piperidine-3-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315593 (2S,3S)-3-Phenyl-piperidine-4-carboxylic acid {(R)-3-[6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-1-methyl-propyl}-amide 315598 4-{3-[2-(7-Methyl-1H-indol-3-yl)-ethylsulfanyl]-5-quinolin-2-yl-[1,2,4]triazol-4-yl}-butylamine 315604 4-[1-(3-Dimethylamino-propyl)-1H-imidazo[4,5-c]pyridin-2-yl]-furazan-3-ylamine 315605 (R,S)-4-(1-Piperidin-3-yl-1H-imidazo[4,5-c]pyridin-2-yl)-furazan-3-ylamine 315606 1-Ethyl-3-(4-{[2-(3-methanesulfonylmethyl-phenylamino)-pyrimidin-4-yl]-methyl-amino}-phenyl)-urea 315607 1-(4-{[2-(4-Methanesulfonylmethyl-phenylamino)-pyrimidin-4-yl]-methyl-amino}-phenyl)-3-[4-(4-methyl-piperazin-1-ylmethyl)-phenyl]-urea 315609 2-(3-chlorophenyl)-1-(1-pentyl-1H-indol-3-yl)ethanone 315610 1-(1-pentyl-1H-indol-3-yl)-2-o-tolylethanone 315620 N*6*-Cyclohexyl-N*2*-(2-ethyl-phenyl)-9H-purine-2,6-diamine 315631 5-{3-[2-(1H-Indol-3-yl)-ethylsulfanyl]-5-naphthalen-2-yl-[1,2,4]triazol-4-yl}-pentylamine 315640 (4R,10aR)-4-Methyl-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole-7-carbonitrile 315641 N-((4R,10aR)-4-Methyl-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indol-7-yl)-acetamide 315663 N*6*-Cycloheptyl-N*2*-phenyl-9H-purine-2,6-diamine 315665 Decyl-phosphonic acid 315668 3-[4-(4-Amino-butyl)-5-quinolin-2-yl-4H-[1,2,4]triazol-3-ylsulfanyl]-1-(7-methyl-1H-indol-3-yl)-propan-1-one 315673 4-{3-(3-Bromo-phenyl)-5-[2-(1H-indol-3-yl)-ethylsulfanyl]-[1,2,4]triazol-4-yl}-butylamine 315677 N*6*-Cyclobutyl-N*2*-(4-morpholin-4-yl-phenyl)-9H-purine-2,6-diamine 315678 N*6*-Cyclohexyl-N*2*-ethyl-9H-purine-2,6-diamine 315680 (4R,10aS)-4,6,7-Trimethyl-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole 315681 (4R,10aR)-7-chloro-4,6-dimethyl-1,2,3,4,10,10a-hexahydropyrazino[1,2-a]indole 315699 (2,5-Dichloro-benzyl)-(4-phenoxy-1H-indazol-3-yl)-amine 315710 N*6*-Cyclohexyl-9-methyl-N*2*-phenyl-9H-purine-2,6-diamine 315711 (1,1-Difluoro-pentadecyl)-phosphonic acid 315718 N*6*-Bicyclo[2.2.1]hept-2-yl-N*2*-(4-morpholin-4-yl-phenyl)-9H-purine-2,6-diamine 315719 Phosphoric acid monododecyl ester 315729 (3-Chloro-benzyl)-(4-phenoxy-1H-indazol-3-yl)-amine 315735 N-(4-{[4-(4-Methanesulfonyl-phenoxy)-1H-indazol-3-ylamino]-methyl}-phenyl)-acetamide 315738 4-{3-(1H-Indol-7-yl)-5-[2-(1H-indol-3-yl)-ethylsulfanyl]-[1,2,4]triazol-4-yl}-butylamine 315748 Phosphoric acid monotetradecyl ester 315754 N*2*-Biphenyl-4-yl-N*6*-cyclohexyl-9H-purine-2,6-diamine 315755 Thiophosphoric acid decyl ester 315756 Thiophosphoric acid dodecyl ester 315778 (S)-7-Chloro-6-methyl-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole 315789 (4R,10aR)-4,7-Dimethyl-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole 315795 (4-{3-[2-(1H-Indol-3-yl)-ethylsulfanyl]-5-naphthalen-2-yl-[1,2,4]triazol-4-yl}-butyl)-dimethyl-amine 315801 (2,5-Dimethoxy-benzyl)-(5-nitro-4-phenoxy-1H-indazol-3-yl)-amine 315803 N*6*-Cyclopropyl-N*2*-(4-morpholin-4-yl-phenyl)-9H-purine-2,6-diamine 315813 SID29217638 315830 (4R,10aR)-4-Methyl-7-trifluoromethyl-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole 315832 3-{3-[2-(1H-Indol-3-yl)-ethylsulfanyl]-5-naphthalen-2-yl-[1,2,4]triazol-4-yl}-propylamine 315833 4-{3-[2-(5-Chloro-1H-indol-3-yl)-ethylsulfanyl]-5-quinolin-2-yl-[1,2,4]triazol-4-yl}-butylamine 315849 Cyclohexyl-(2-phenylsulfanyl-9H-purin-6-yl)-amine 315850 Tetradecyl-phosphonic acid 315853 (4R,10aR)-4,6-Dimethyl-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole 315854 N*6*-Cycloheptyl-9-methyl-N*2*-phenyl-9H-purine-2,6-diamine 315860 N*2*-Benzyl-N*6*-cyclohexyl-9H-purine-2,6-diamine 315861 Phosphoric acid mono-((E)-dodec-9-enyl) ester 315862 Phosphoric acid mono-((E)-tetradec-9-enyl) ester 315868 N*6*-Cyclohexyl-N*2*-(4-dimethylamino-phenyl)-9H-purine-2,6-diamine 315869 Thiophosphoric acid (E)-dodec-9-enyl ester 315876 N-(4-{[4-(4-Fluoro-phenoxy)-1H-indazol-3-ylamino]-methyl}-phenyl)-acetamide 315885 (4R,10aR)-4,6,7-Trimethyl-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole 315899 Thiophosphoric acid (E)-tetradec-9-enyl ester 315901 N-{4-[(4-Phenoxy-1H-indazol-3-ylamino)-methyl]-phenyl}-acetamide 315908 4-{3-(4-Ethyl-phenyl)-5-[2-(1H-indol-3-yl)-ethylsulfanyl]-[1,2,4]triazol-4-yl}-butylamine 315919 N*6*-Cyclooctyl-N*2*-(4-morpholin-4-yl-phenyl)-9H-purine-2,6-diamine 315926 7-Chloro-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole 315950 Phosphoric acid monodecyl ester 315955 6-N-cyclohexyl-2-N-(naphthalen-2-yl)-1H-purine-2,6-diamine 315968 (2,5-Dimethoxy-benzyl)-[4-(4-fluoro-phenoxy)-1H-indazol-3-yl]-amine 315970 4-{3-Benzo[b]thiophen-2-yl-5-[2-(1H-indol-3-yl)-ethylsulfanyl]-[1,2,4]triazol-4-yl}-butylamine 315980 (4R,10aS)-7-chloro-4,6-dimethyl-1,2,3,4,10,10a-hexahydropyrazino[1,2-a]indole 315987 Phosphoric acid mono-((E)-tetradec-11-enyl) ester 315993 N*6*-Ethyl-N*2*-(4-morpholin-4-yl-phenyl)-9H-purine-2,6-diamine 315994 N*6*-Cyclooctyl-N*2*-phenyl-9H-purine-2,6-diamine 315998 3-[4-(4-Amino-butyl)-5-quinolin-2-yl-4H-[1,2,4]triazol-3-ylsulfanyl]-2,2-dimethyl-1-(7-methyl-1H-indol-3-yl)-propan-1-one 316004 SID29215538 316009 (R)-7-Chloro-6-methyl-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole 316021 SID29216411 316032 (2,5-Dimethoxy-benzyl)-[4-(4-methanesulfonyl-phenoxy)-1H-indazol-3-yl]-amine 316033 Dodecyl-phosphonic acid 316035 ((4R,10aR)-4-Methyl-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indol-7-yl)-methanol 316037 N*6*-Cyclopentyl-N*2*-(4-morpholin-4-yl-phenyl)-9H-purine-2,6-diamine 316050 N*6*-Cyclohexyl-N*2*-(4-phenyl-piperidin-1-yl)-9H-purine-2,6-diamine 316058 (2,5-Dimethoxy-benzyl)-(4-phenoxy-1H-indazol-3-yl)-amine 316076 Octanoic acid (S)-1-methyl-2-octanoyloxy-diphosphoric acid 316077 Phosphoric acid mono-[(S)-3-(4-benzyloxy-phenyl)-2-octadecanoylamino-propyl] ester 316084 N*6*-Cyclohexyl-N*2*-phenyl-9H-purine-2,6-diamine 316085 Phosphoric acid monodec-9-enyl ester 316086 Phosphoric acid mono-((E)-dec-4-enyl) ester 316092 Thiophosphoric acid tetradecyl ester 316093 Thiophosphoric acid dec-9-enyl ester 316112 N*6*-Cycloheptyl-N*2*-(4-morpholin-4-yl-phenyl)-9H-purine-2,6-diamine 316115 3-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonylamino)-3-methylisoxazol-5-yl)benzylthio)propanoic acid 316129 4-{3-[2-(1H-Indol-3-yl)-ethylsulfanyl]-5-naphthalen-1-yl-[1,2,4]triazol-4-yl}-butylamine 316137 5-[8-(Isopropyl-methyl-amino)-9-methyl-9H-purin-6-ylamino]-bicyclo[2.2.1]heptan-2-ol 316138 2-Hexadecanoylamino-3-(4-phosphonooxy-phenyl)-propionic acid 316151 Degarelix analogue 316159 2-Phenyl-2,5-dihydro-pyrazolo[4,3-c]quinolin-4-one 316171 (3S,4aR,4bS,6S,8R,8aR,10aR)-3-Furan-3-yl-4a,8a-dimethyl-1,5-dioxo-6-phenylcarbamoyloxy-dodecahydro-2-oxa-phenanthrene-8-carboxylic acid methyl ester 316173 1-(3'-Cyano-biphenyl-4-yl)-3-(3,4-dichloro-phenyl)-1-(2-dimethylamino-ethyl)-urea 316183 1-(3'-Cyano-biphenyl-4-yl)-1-(1-cyclopentyl-piperidin-4-yl)-3-(4-methoxy-phenyl)-urea 316193 4-Methoxy-2-phenyl-2H-pyrazolo[4,3-c]quinoline 316215 1-(3'-Cyano-biphenyl-4-yl)-1-(1-cyclopentyl-piperidin-4-yl)-3-phenyl-urea 316217 2-Phenyl-2,5-dihydro-pyrazolo[4,3-c]quinoline-4-thione 316243 1-(3'-Cyano-biphenyl-4-yl)-3-(3-fluoro-4-trifluoromethyl-phenyl)-1-[2-(4-methyl-piperazin-1-yl)-ethyl]-urea 316247 (3S,4aR,4bS,6S,8R,8aR,10aR)-3-Furan-3-yl-4a,8a-dimethyl-1,5-dioxo-6-trimethylsilanyloxy-dodecahydro-2-oxa-phenanthrene-8-carboxylic acid methyl ester 316253 Degarelix analogue 316261 Degarelix analogue 316262 Degarelix analogue 316263 Degarelix analogue 316264 Degarelix analogue 316265 Degarelix analogue 316268 1-(3'-Cyano-biphenyl-4-yl)-1-(1-cyclopentyl-piperidin-4-yl)-3-(4-fluoro-3-trifluoromethyl-phenyl)-urea 316274 3-(3-Chloro-4-fluoro-phenyl)-1-(3'-cyano-biphenyl-4-yl)-1-(2-methylamino-ethyl)-urea 316298 3-(3-Chloro-4-fluoro-phenyl)-1-(3'-cyano-biphenyl-4-yl)-1-[2-((R)-3-hydroxy-pyrrolidin-1-yl)-ethyl]-urea 316300 (3S,4aR,4bS,6S,8R,8aR,10aR)-3-Furan-3-yl-4a,8a-dimethyl-1,5-dioxo-6-(2,2,2-trichloro-acetimidoyloxy)-dodecahydro-2-oxa-phenanthrene-8-carboxylic acid methyl ester 316308 Herkinorin 316318 Degarelix analogue 316319 Degarelix analogue 316320 Degarelix analogue 316321 Degarelix analogue 316339 (3S,4aR,4bS,6S,8R,8aR,10aR)-3-Furan-3-yl-6-isobutyryloxy-4a,8a-dimethyl-1,5-dioxo-dodecahydro-2-oxa-phenanthrene-8-carboxylic acid methyl ester 316359 Degarelix analogue 316362 (3S,4aR,4bS,5R,6S,8R,8aR,10aR)-3-Furan-3-yl-5,6-dihydroxy-4a,8a-dimethyl-1-oxo-dodecahydro-2-oxa-phenanthrene-8-carboxylic acid methyl ester 316372 1-(3'-Cyano-biphenyl-4-yl)-3-(4-fluoro-3-trifluoromethyl-phenyl)-1-(1-isobutyryl-piperidin-4-yl)-urea 316405 1-(3'-Chloro-biphenyl-4-yl)-1-(1-cyclopentyl-piperidin-4-yl)-3-(3,4-dichloro-phenyl)-urea 316408 1-(3'-Cyano-biphenyl-4-yl)-1-(1-cyclopentyl-piperidin-4-yl)-3-(3-methoxy-phenyl)-urea 316423 1-(3'-Cyano-biphenyl-4-yl)-1-(1-cyclopropylmethyl-piperidin-4-yl)-3-(4-fluoro-3-trifluoromethyl-phenyl)-urea 316429 1-(3'-Cyano-biphenyl-4-yl)-3-(3-fluoro-4-trifluoromethyl-phenyl)-1-(2-pyrrolidin-1-yl-ethyl)-urea 316432 1-(3'-Cyano-biphenyl-4-yl)-3-(3-fluoro-4-trifluoromethyl-phenyl)-1-[2-((R)-3-hydroxy-pyrrolidin-1-yl)-ethyl]-urea 316436 3-(3-Chloro-4-fluoro-phenyl)-1-(3'-cyano-biphenyl-4-yl)-1-(1-cyclopentyl-piperidin-4-yl)-urea 316437 Degarelix analogue 316438 Degarelix analogue 316439 Degarelix analogue 316440 Degarelix analogue 316441 Degarelix analogue 316455 (3S,4aR,4bS,6S,8R,8aR,10aR)-6-Allylcarbamoyloxy-3-furan-3-yl-4a,8a-dimethyl-1,5-dioxo-dodecahydro-2-oxa-phenanthrene-8-carboxylic acid methyl ester 316457 1-(1-Cyclopentyl-piperidin-4-yl)-3-(3,4-dichloro-phenyl)-1-(3'-trifluoromethoxy-biphenyl-4-yl)-urea 316463 1-(3'-Cyano-biphenyl-4-yl)-3-(3,4-dichloro-phenyl)-1-[2-((R)-3-hydroxy-pyrrolidin-1-yl)-ethyl]-urea 316476 Degarelix analogue 316482 (3S,4aR,4bS,5R,6S,8R,8aR,10aR)-5,6-Diacetoxy-3-furan-3-yl-4a,8a-dimethyl-1-oxo-dodecahydro-2-oxa-phenanthrene-8-carboxylic acid methyl ester 316486 3-(3-Chloro-4-fluoro-phenyl)-1-(3'-cyano-biphenyl-4-yl)-1-(2-dimethylamino-ethyl)-urea 316490 Oxalic acid (3S,4aR,4bS,6S,8R,8aR,10aR)-3-furan-3-yl-8-methoxycarbonyl-4a,8a-dimethyl-1,5-dioxo-dodecahydro-2-oxa-phenanthren-6-yl ester methyl ester 316494 (2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 2-(furan-3-yl)-6a,10b-dimethyl-9-(methylsulfonyloxy)-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 316519 3-(3-Chloro-phenyl)-1-(3'-cyano-biphenyl-4-yl)-1-(1-cyclopentyl-piperidin-4-yl)-urea 316537 1-(3'-Cyano-biphenyl-4-yl)-1-(1-ethanesulfonyl-piperidin-4-yl)-3-(4-fluoro-3-trifluoromethyl-phenyl)-urea 316540 1-(1-Cyclopentyl-piperidin-4-yl)-3-(3,4-dichloro-phenyl)-1-(3'-trifluoromethyl-biphenyl-4-yl)-urea 316542 1-(3'-Cyano-biphenyl-4-yl)-3-(3-fluoro-4-trifluoromethyl-phenyl)-1-[2-((S)-3-hydroxy-pyrrolidin-1-yl)-ethyl]-urea 316551 Degarelix analogue 316552 Degarelix analogue 316553 Degarelix analogue 316554 Degarelix analogue 316565 1-(3'-Cyano-biphenyl-4-yl)-1-(1-ethyl-piperidin-4-yl)-3-(4-fluoro-3-trifluoromethyl-phenyl)-urea 316568 (2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 2-(furan-3-yl)-6a,10b-dimethyl-4,10-dioxo-9-(propionyloxy)-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 316570 1-(3'-Cyano-biphenyl-4-yl)-1-(2-dimethylamino-ethyl)-3-(3-fluoro-4-trifluoromethyl-phenyl)-urea 316592 (R)-1-(3'-cyanobiphenyl-4-yl)-3-(4-fluoro-3-(trifluoromethyl)phenyl)-1-(2-(3-hydroxypyrrolidin-1-yl)ethyl)urea 316627 1-(3'-cyano-biphenyl-4-yl)-1-(1-cyclopentyl-piperidin-4-yl)-3-(3,5-dichloro-phenyl)-urea 316631 (3S,4aR,4bS,6S,8R,8aR,10aR)-3-Furan-3-yl-4a,8a-dimethyl-6-(2-methyl-acryloyloxy)-1,5-dioxo-dodecahydro-2-oxa-phenanthrene-8-carboxylic acid methyl ester 316634 Nicotinic acid (3S,4aR,4bS,6S,8R,8aR,10aR)-3-furan-3-yl-8-methoxycarbonyl-4a,8a-dimethyl-1,5-dioxo-dodecahydro-2-oxa-phenanthren-6-yl ester 316640 Degarelix analogue 316641 Degarelix analogue 316642 Degarelix analogue 316643 Degarelix analogue 316644 Degarelix analogue 316670 1-(4-Bromo-2,5-dimethoxy-benzyl)-propylamine 316671 (1R,2S)-2-Amino-1-(4-bromo-2,5-dimethoxy-phenyl)-butan-1-ol 316743 2-(4-Chloro-phenyl)-2,5-dihydro-pyrazolo[4,3-c]quinolin-4-one 316781 2-p-Tolyl-2,5-dihydro-pyrazolo[4,3-c]quinolin-4-one 316791 (1R,2R)-2-Amino-1-(4-bromo-2,5-dimethoxy-phenyl)-propan-1-ol 316792 (1S,2R)-2-(4-Bromo-2,5-dimethoxy-phenyl)-2-methoxy-1-methyl-ethylamine 316806 2-{(R)-2-[(S)-2-(Acetyl-butyl-amino)-acetylamino]-acetylamino}-6-amino-hexanoic acid (1-{1-[(S)-1-((S)-carbamoylmethyl-carbamoyl)-2-(1H-indol-3-yl)-ethylcarbamoyl]-4-guanidino-butylcarbamoyl}-2-phenyl-ethyl)-amide 316807 (S)-2-Acetylamino-hexanoic acid ({(4-amino-butyl)-[((S,R)-1-{(S)-4-amino-1-[1-(carbamoylmethyl-carbamoyl)-2-(1H-indol-3-yl)-ethylcarbamoyl]-butylcarbamoyl}-2-phenyl-ethylcarbamoyl)-methyl]-carbamoyl}-methyl)-amide 316815 [(S)-1-((4aS,5R)-2-Benzyl-1-mercapto-3-oxo-octahydro-pyrido[1,2-c]pyrimidin-5-ylcarbamoyl)-2-(1H-indol-3-yl)-ethyl]-carbamic acid tert-butyl ester 316816 [(S)-2-(1H-Indol-3-yl)-1-((4aS,5R)-2-naphthalen-1-yl-1,3-dioxo-octahydro-pyrido[1,2-c]pyrimidin-5-ylcarbamoyl)-ethyl]-carbamic acid tert-butyl ester 316820 2-(2-Chloro-phenyl)-2,5-dihydro-pyrazolo[4,3-c]quinolin-4-one 316856 2-(4-Ethyl-phenyl)-2,5-dihydro-pyrazolo[4,3-c]quinolin-4-one 316892 2-(4-Bromo-2,5-dimethoxy-phenyl)-morpholine 316893 2-Amino-1-(4-bromo-2,5-dimethoxy-phenyl)-ethanol 316894 2-(4-Bromo-2,5-dimethoxy-phenyl)-2-methoxy-ethylamine 316900 (1R,2R)-2-(4-Bromo-2,5-dimethoxy-phenyl)-2-methoxy-1-methyl-ethylamine 316992 2-{(R)-2-[(S)-2-((S)-Acetylamino)-hexanoylamino]-acetylamino}-6-amino-hexanoic acid (1-{1-[(S)-1-((S)-carbamoylmethyl-carbamoyl)-2-(1H-indol-3-yl)-ethylcarbamoyl]-4-guanidino-butylcarbamoyl}-2-phenyl-ethyl)-amide 317041 (1S,2R)-2-Amino-1-(4-bromo-2,5-dimethoxy-phenyl)-propan-1-ol 317042 (1R,2S)-2-Amino-1-(4-bromo-2,5-dimethoxy-phenyl)-propan-1-ol 317043 (1S,2S)-2-Amino-1-(4-bromo-2,5-dimethoxy-phenyl)-propan-1-ol 317097 (2S)-6-amino-N-[(1R)-1-[({[(1S)-1-[(carbamoylmethyl)carbamoyl]-2-(1H-indol-3-yl)ethyl]carbamoyl}methyl)({3-[(diaminomethylidene)amino]propyl})carbamoyl]-2-phenylethyl]-2-{2-[(2S)-2-acetamidohexanamido]acetamido}hexanamide 317098 2-{(R)-2-[(S)-2-((S)-Acetylamino)-hexanoylamino]-acetylamino}-6-amino-hexanoic acid [1-((S)-1-{[(carbamoylmethyl-carbamoyl)-methyl]-[2-(1H-indol-3-yl)-ethyl]-carbamoyl}-4-guanidino-butylcarbamoyl)-2-phenyl-ethyl]-amide 317099 2-((S)-2-{(S)-(R)-2-[{2-[2-(Acetyl-butyl-amino)-acetylamino]-acetyl}-(4-amino-butyl)-amino]-acetylamino}-3-phenyl-propionylamino)-5-guanidino-pentanoic acid [1-(carbamoylmethyl-carbamoyl)-2-(1H-indol-3-yl)-ethyl]-amide 317106 [(S)-1-((4aS,5R)-1,3-Dioxo-2-phenyl-octahydro-pyrido[1,2-c]pyrimidin-5-ylcarbamoyl)-2-(1H-indol-3-yl)-ethyl]-carbamic acid tert-butyl ester 317110 2-(4-Methoxy-phenyl)-2,5-dihydro-pyrazolo[4,3-c]quinolin-4-one 317115 Degarelix analogue 317116 Degarelix analogue 317142 2-(4-Fluoro-phenyl)-2,5-dihydro-pyrazolo[4,3-c]quinolin-4-one 317151 (1R,2S)-2-(4-Bromo-2,5-dimethoxy-phenyl)-2-methoxy-1-methyl-ethylamine 317152 (1S,2S)-2-(4-Bromo-2,5-dimethoxy-phenyl)-2-methoxy-1-methyl-ethylamine 317179 2-Phenyl-2H-pyrazolo[4,3-c]quinoline 317180 Benzyl-(2-phenyl-2H-pyrazolo[4,3-c]quinolin-4-yl)-amine 317205 2-[(S)-2-((S)-2-Acetylamino-hexanoylamino)-1-oxo-ethylamino]-6-amino-hexanoic acid {1-[({[(carbamoylmethyl-carbamoyl)-methyl]-[2-(1H-indol-3-yl)-ethyl]-carbamoyl}-methyl)-(3-guanidino-propyl)-carbamoyl]-2-phenyl-ethyl}-amide 317207 2-((S)-2-{(R)-2-[{2-[2-(Acetyl-butyl-amino)-acetylamino]-acetyl}-(4-amino-butyl)-amino]-acetylamino}-3-phenyl-propionylamino)-5-guanidino-pentanoic acid [(carbamoylmethyl-carbamoyl)-methyl]-[2-(1H-indol-3-yl)-ethyl]-amide 317246 (6aR,10aR)-3-Adamantan-2-ylmethyl-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol 317286 2-{(R)-2-[(S)-2-((S)-Acetylamino)-hexanoylamino]-acetylamino}-6-amino-hexanoic acid (1-{(S)-1-[[(carbamoylmethyl-carbamoyl)-methyl]-(1H-indol-3-ylmethyl)-carbamoyl]-4-guanidino-butylcarbamoyl}-2-phenyl-ethyl)-amide 317287 (S)-2-{2-[2-(Acetyl-butyl-amino)-acetylamino]-acetylamino}-6-amino-hexanoic acid ((R)-1-{1-[(S)-[(carbamoylmethyl-carbamoyl)-methyl]-(1H-indol-3-ylmethyl)-carbamoyl]-4-guanidino-butylcarbamoyl}-2-phenyl-ethyl)-amide 317326 2-[(S)-2-((S)-2-Acetylamino-hexanoylamino)-1-oxo-ethylamino]-6-amino-hexanoic acid {1-[({[(carbamoylmethyl-carbamoyl)-methyl]-[2-(1H-indol-3-yl)-ethyl]-carbamoyl}-methyl)-(4-guanidino-butyl)-carbamoyl]-2-phenyl-ethyl}-amide 317507 4-(5-amino-1-(2,6-difluorobenzoyl)-1H-1,2,4-triazol-3-ylamino)benzenesulfonamide 317529 2-{(S)-2-[2-(Acetyl-butyl-amino)-acetylamino]-1-oxo-ethylamino}-6-amino-hexanoic acid {1-[({[(carbamoylmethyl-carbamoyl)-methyl]-[2-(1H-indol-3-yl)-ethyl]-carbamoyl}-methyl)-(3-guanidino-propyl)-carbamoyl]-2-phenyl-ethyl}-amide 317530 2-Acetylamino-hexanoic acid {[(4-amino-butyl)-({(S)-1-[({[(carbamoylmethyl-carbamoyl)-methyl]-[2-(1H-indol-3-yl)-ethyl]-carbamoyl}-methyl)-(3-guanidino-propyl)-carbamoyl]-2-phenyl-ethylcarbamoyl}-methyl)-carbamoyl]-methyl}-amide 317531 2-{(R)-2-[{2-[2-(Acetyl-butyl-amino)-acetylamino]-acetyl}-(4-amino-butyl)-amino]-1-oxo-ethylamino}-N-({[(carbamoylmethyl-carbamoyl)-methyl]-[2-(1H-indol-3-yl)-ethyl]-carbamoyl}-methyl)-N-(3-guanidino-propyl)-3-phenyl-propionamide 317604 (S)-2-Acetylamino-hexanoic acid ({(4-amino-butyl)-[((R)-(S)-1-{1-[[(carbamoylmethyl-carbamoyl)-methyl]-(1H-indol-3-ylmethyl)-carbamoyl]-4-guanidino-butylcarbamoyl}-2-phenyl-ethylcarbamoyl)-methyl]-carbamoyl}-methyl)-amide 317605 2-[(S)-2-((S)-2-Acetylamino-hexanoylamino)-1-oxo-ethylamino]-6-amino-hexanoic acid {1-[{[[(carbamoylmethyl-carbamoyl)-methyl]-(1H-indol-3-ylmethyl)-carbamoyl]-methyl}-(3-guanidino-propyl)-carbamoyl]-2-phenyl-ethyl}-amide 317606 2-(2-{(S)-(R)-2-[{2-[2-(Acetyl-butyl-amino)-acetylamino]-acetyl}-(4-amino-butyl)-amino]-acetylamino}-3-phenyl-propionylamino)-5-guanidino-pentanoic acid [(carbamoylmethyl-carbamoyl)-methyl]-(1H-indol-3-ylmethyl)-amide 317607 2-{2-[2-(Acetyl-butyl-amino)-acetylamino]-acetylamino}-6-amino-hexanoic acid {1-[(R)-({[(carbamoylmethyl-carbamoyl)-methyl]-[(Z)-1-(1H-indol-3-yl)methyl]-carbamoyl}-methyl)-(3-guanidino-propyl)-carbamoyl]-2-phenyl-ethyl}-amide 317608 2-Acetylamino-hexanoic acid {[(4-amino-butyl)-({(S)-1-[{[[(carbamoylmethyl-carbamoyl)-methyl]-(1H-indol-3-ylmethyl)-carbamoyl]-methyl}-(3-guanidino-propyl)-carbamoyl]-2-phenyl-ethylcarbamoyl}-methyl)-carbamoyl]-methyl}-amide 317609 2-{2-[{(R)-2-[2-(Acetyl-butyl-amino)-acetylamino]-acetyl}-(4-amino-butyl)-amino]-acetylamino}-N-{[[(carbamoylmethyl-carbamoyl)-methyl]-(1H-indol-3-ylmethyl)-carbamoyl]-methyl}-N-(3-guanidino-propyl)-3-phenyl-propionamide 317640 1-tert-Butyl-3-[7-(4-diethylamino-butylamino)-3-phenyl-[1,6]naphthyridin-2-yl]-urea 317802 1-tert-Butyl-3-{3-(2,6-dichloro-phenyl)-7-[3-(4-methyl-piperazin-1-yl)-propylamino]-[1,6]naphthyridin-2-yl}-urea 317803 (2Z)-1,3-benzothiazol-2(3H)-ylidene(2-chloropyrimidin-4-yl)acetonitrile 317804 [3H-Benzothiazol-(2Z)-ylidene]-[2-(2-hydroxy-ethylamino)-pyrimidin-4-yl]-acetonitrile 317805 1-tert-Butyl-3-[6-(3,5-dimethoxy-phenyl)-2-(3-hydroxy-propylamino)-pyrido[2,3-d]pyrimidin-7-yl]-urea 317811 [3H-Benzothiazol-(2Z)-ylidene]-[2-(2-pyridin-2-yl-ethylamino)-pyrimidin-4-yl]-acetonitrile 317813 1-tert-Butyl-3-[7-(5-diethylamino-pentylamino)-3-(3,5-dimethoxy-phenyl)-[1,6]naphthyridin-2-yl]-urea 317816 [3H-Benzothiazol-(2Z)-ylidene]-[2-(2-[1,2,4]triazol-1-yl-ethylamino)-pyrimidin-4-yl]-acetonitrile 317829 [3H-Benzothiazol-(2Z)-ylidene]-{2-[methyl-(3-methylamino-propyl)-amino]-pyrimidin-4-yl}-acetonitrile 317832 1-{6-(3,5-Dimethoxy-phenyl)-2-[3-(4-methyl-piperazin-1-yl)-propylamino]-pyrido[2,3-d]pyrimidin-7-yl}-3-ethyl-urea 317833 [3H-Benzothiazol-(2Z)-ylidene]-{2-[(pyridin-4-ylmethyl)-amino]-pyrimidin-4-yl}-acetonitrile 317834 [3H-Benzothiazol-(2Z)-ylidene]-{2-[2-(4-nitro-phenyl)-ethylamino]-pyrimidin-4-yl}-acetonitrile 317837 [3H-Benzothiazol-(2Z)-ylidene]-[2-(2-piperidin-1-yl-ethylamino)-pyrimidin-4-yl]-acetonitrile 317839 N*7*-[3-(4-Methyl-piperazin-1-yl)-propyl]-3-phenyl-[1,6]naphthyridine-2,7-diamine 317840 1-tert-Butyl-3-[3-(3,5-dimethoxy-phenyl)-7-(4-phenoxy-butylamino)-[1,6]naphthyridin-2-yl]-urea 317841 1-tert-Butyl-3-[3-(3,5-dimethoxy-phenyl)-7-(5-phenoxy-pentylamino)-[1,6]naphthyridin-2-yl]-urea 317854 1-benzyl-7-cyclohexyl-3-propyl-1H-imidazo[1,2-a]purine-2,4(3H,8H)-dione 317856 [3H-Benzothiazol-(2Z)-ylidene]-[2-(3-pyrazol-1-yl-propylamino)-pyrimidin-4-yl]-acetonitrile 317859 [3H-Benzothiazol-(2Z)-ylidene]-[2-(2-dimethylamino-ethylamino)-pyrimidin-4-yl]-acetonitrile 317867 [3H-Benzothiazol-(2Z)-ylidene]-{2-[2-(2-fluoro-phenyl)-ethylamino]-pyrimidin-4-yl}-acetonitrile 317868 [3H-Benzothiazol-(2Z)-ylidene]-{2-[2-(1-methyl-1H-imidazol-4-yl)-ethylamino]-pyrimidin-4-yl}-acetonitrile 317875 N*2*,N*7*-Bis-[3-(4-methyl-piperazin-1-yl)-propyl]-3-phenyl-[1,6]naphthyridine-2,7-diamine 317876 [3H-Benzothiazol-(2Z)-ylidene]-(2-morpholin-4-yl-pyrimidin-4-yl)-acetonitrile 317877 N-[3-(4-{[3H-Benzothiazol-(2Z)-ylidene]-cyano-methyl}-pyrimidin-2-ylamino)-propyl]-N-propyl-propionamide 317882 1-benzyl-7-isopropyl-3-propyl-1H-imidazo[1,2-a]purine-2,4(3H,8H)-dione 317886 2-[(5,6-Diphenyl-furo[2,3-d]pyrimidin-4-yl)-methyl-amino]-ethanol 317887 (5,6-Diphenyl-furo[2,3-d]pyrimidin-4-ylamino)-acetic acid 317894 2-(2-(4-methoxyphenethylamino)pyrimidin-4-yl)-2-(benzo[d]thiazol-2(3H)-ylidene)acetonitrile 317897 1-{3-(3,5-Dimethoxy-phenyl)-7-[3-(4-methyl-piperazin-1-yl)-propylamino]-[1,6]naphthyridin-2-yl}-3-ethyl-urea 317904 1-tert-Butyl-3-[3-(3,5-dimethoxy-phenyl)-7-(4-hydroxy-butylamino)-[1,6]naphthyridin-2-yl]-urea 317905 N-(4-Benzyloxy-butyl)-N-[2-(3-tert-butyl-ureido)-3-(3,5-dimethoxy-phenyl)-3,4-dihydro-[1,6]naphthyridin-7-yl]-acetamide 317908 1-benzyl-7-(4-fluorophenyl)-3-propyl-1H-imidazo[1,2-a]purine-2,4(3H,8H)-dione 317922 N-[2-(3-tert-Butyl-ureido)-3-(3,5-dimethoxy-phenyl)-3,4-dihydro-[1,6]naphthyridin-7-yl]-N-(3-hydroxy-propyl)-acetamide 317923 1-tert-Butyl-3-{6-(3,5-dimethoxy-phenyl)-2-[3-(4-methyl-piperazin-1-yl)-propylamino]-pyrido[2,3-d]pyrimidin-7-yl}-urea 317927 1-tert-Butyl-3-{3-(3,5-dimethoxy-phenyl)-7-[4-(4-methyl-piperazin-1-yl)-butylamino]-[1,6]naphthyridin-2-yl}-urea 317928 1-[3-(2,6-Dichloro-phenyl)-7-(4-diethylamino-butylamino)-[1,6]naphthyridin-2-yl]-3-ethyl-urea 317951 1-{3-(2,6-Dichloro-phenyl)-7-[3-(4-methyl-piperazin-1-yl)-propylamino]-[1,6]naphthyridin-2-yl}-3-ethyl-urea 317952 N-(4-Benzyloxy-butyl)-N-[2-(3-tert-butyl-ureido)-3-(3,5-dimethoxy-phenyl)-[1,6]naphthyridin-7-yl]-acetamide 317955 SID29217621 317958 N-[2-(3-tert-Butyl-ureido)-3-(3,5-dimethoxy-phenyl)-[1,6]naphthyridin-7-yl]-N-(4-hydroxy-butyl)-acetamide 317960 (2Z)-1,3-benzothiazol-2(3H)-ylidene(2-hydrazinopyrimidin-4-yl)acetonitrile 317962 (6aR,10aR)-3-Adamantan-1-yl-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol 317977 1-benzyl-7-ethyl-6-methyl-3-propyl-1H-imidazo[1,2-a]purine-2,4(3H,8H)-dione 317980 N-[2-(3-tert-Butyl-ureido)-3-(3,5-dimethoxy-phenyl)-3,4-dihydro-[1,6]naphthyridin-7-yl]-N-(5-hydroxy-pentyl)-acetamide 317985 (2Z)-(2-chloropyrimidin-4-yl)[5-(trifluoromethyl)-1,3-benzothiazol-2(3H)-ylidene]acetonitrile 317988 (2Z)-1,3-benzothiazol-2(3H)-ylidene[2-(methylamino)pyrimidin-4-yl]acetonitrile 317989 [3H-Benzothiazol-(2Z)-ylidene]-[2-(3-dimethylamino-propylamino)-pyrimidin-4-yl]-acetonitrile 317991 [3H-Benzothiazol-(2Z)-ylidene]-[2-(3-hydroxy-propylamino)-pyrimidin-4-yl]-acetonitrile 318004 3-(5,6-Diphenyl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)-propane-1,2-diol 318009 (2Z)-1,3-benzothiazol-2(3H)-ylidene(6-bromo-2-chloropyrimidin-4-yl)acetonitrile 318010 [3H-Benzothiazol-(2Z)-ylidene]-[2-(2-methoxy-ethylamino)-pyrimidin-4-yl]-acetonitrile 318013 [3H-Benzothiazol-(2Z)-ylidene]-{2-[2-(1H-imidazol-4-yl)-ethylamino]-pyrimidin-4-yl}-acetonitrile 318016 [3H-Benzothiazol-(2Z)-ylidene]-{2-[2-(3-methyl-3H-imidazol-4-yl)-ethylamino]-pyrimidin-4-yl}-acetonitrile 318019 2-(benzo[d]thiazol-2(3H)-ylidene)-2-(2-(2-(pyridin-3-yl)ethylamino)pyrimidin-4-yl)acetonitrile 318029 1-benzyl-7-cyclopropyl-3-propyl-1H-imidazo[1,2-a]purine-2,4(3H,8H)-dione 318035 (6aR,10aR)-3-Adamantan-1-ylmethyl-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol 318037 [3H-Benzothiazol-(2Z)-ylidene]-{2-[(pyridin-3-ylmethyl)-amino]-pyrimidin-4-yl}-acetonitrile 318038 4-(2-(4-(benzo[d]thiazol-2(3H)-ylidene(cyano)methyl)pyrimidin-2-ylamino)ethyl)benzenesulfonamide 318043 1-tert-Butyl-3-[7-(4-diethylamino-butylamino)-3-(3,5-dimethoxy-phenyl)-[1,6]naphthyridin-2-yl]-urea 318044 1-tert-Butyl-3-{3-(3,5-dimethoxy-phenyl)-7-[5-(4-methyl-piperazin-1-yl)-pentylamino]-[1,6]naphthyridin-2-yl}-urea 318047 (6aR,10aR)-3-Adamantan-2-ylidenemethyl-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol 318055 2-[5,6-Bis-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-ylamino]-ethanol 318056 2-(5,6-diphenylfuro[2,3-d]pyrimidin-4-ylamino)ethanol 318060 5-(4-Bromo-phenyl)-1-(2,4-dichloro-phenyl)-4-ethyl-1H-pyrazole-3-carboxylic acid piperidin-1-ylamide 318061 [3H-Benzothiazol-(2Z)-ylidene]-[2-(4-methoxy-piperidin-1-yl)-pyrimidin-4-yl]-acetonitrile 318062 [3H-Benzothiazol-(2Z)-ylidene]-(2-benzylamino-pyrimidin-4-yl)-acetonitrile 318071 N-[2-(3-tert-Butyl-ureido)-3-(3,5-dimethoxy-phenyl)-[1,6]naphthyridin-7-yl]-N-(5-hydroxy-pentyl)-acetamide 318072 1-tert-Butyl-3-[3-(3,5-dimethoxy-phenyl)-7-(3-phenoxy-propylamino)-[1,6]naphthyridin-2-yl]-urea 318073 1-tert-Butyl-3-{7-[3-(4-methyl-piperazin-1-yl)-propylamino]-3-phenyl-[1,6]naphthyridin-2-yl}-urea 318074 [3H-Benzothiazol-(2Z)-ylidene]-[2-(4-methyl-piperazin-1-yl)-pyrimidin-4-yl]-acetonitrile 318075 [3H-Benzothiazol-(2Z)-ylidene]-{2-[3-(4-methyl-piperazin-1-yl)-propylamino]-pyrimidin-4-yl}-acetonitrile 318089 [3H-Benzothiazol-(2Z)-ylidene]-{2-[2-(4-hydroxy-phenyl)-ethylamino]-pyrimidin-4-yl}-acetonitrile 318092 3-(3,5-Dimethoxy-phenyl)-N*7*-[3-(4-methyl-piperazin-1-yl)-propyl]-[1,6]naphthyridine-2,7-diamine 318093 1-tert-Butyl-3-[3-(3,5-dimethoxy-phenyl)-7-(4-morpholin-4-yl-butylamino)-[1,6]naphthyridin-2-yl]-urea 318094 3-(2,6-Dichloro-phenyl)-N*7*-(4-diethylamino-butyl)-[1,6]naphthyridine-2,7-diamine 318097 N*7*-(4-Diethylamino-butyl)-3-(3,5-dimethoxy-phenyl)-[1,6]naphthyridine-2,7-diamine 318098 N-[2-(3-tert-Butyl-ureido)-3-(3,5-dimethoxy-phenyl)-[1,6]naphthyridin-7-yl]-N-(3-hydroxy-propyl)-acetamide 318102 1-tert-Butyl-3-[3-(3,5-dimethoxy-phenyl)-7-(3-hydroxy-propylamino)-[1,6]naphthyridin-2-yl]-urea 318103 N-(3-Benzyloxy-propyl)-N-[2-(3-tert-butyl-ureido)-3-(3,5-dimethoxy-phenyl)-3,4-dihydro-[1,6]naphthyridin-7-yl]-acetamide 318105 [3H-Benzothiazol-(2Z)-ylidene]-[2-(3-imidazol-1-yl-propylamino)-pyrimidin-4-yl]-acetonitrile 318112 1-benzyl-7-ethyl-3-propyl-1H-imidazo[1,2-a]purine-2,4(3H,8H)-dione 318125 1-[2-(4-Diethylamino-butylamino)-6-(3,5-dimethoxy-phenyl)-pyrido[2,3-d]pyrimidin-7-yl]-3-ethyl-urea 318147 1-benzyl-6,7-dimethyl-3-propyl-1H-imidazo[1,2-a]purine-2,4(3H,8H)-dione 318148 2-(5,6-Diphenyl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)-ethanol 318150 3-(2,6-Dichloro-phenyl)-N*7*-[3-(4-methyl-piperazin-1-yl)-propyl]-[1,6]naphthyridine-2,7-diamine 318151 N-(3-Benzyloxy-propyl)-N-[2-(3-tert-butyl-ureido)-3-(3,5-dimethoxy-phenyl)-[1,6]naphthyridin-7-yl]-acetamide 318154 [2-(2-Amino-ethylamino)-pyrimidin-4-yl]-[3H-benzothiazol-(2Z)-ylidene]-acetonitrile 318158 [3H-Benzothiazol-(2Z)-ylidene]-[2-(2-indol-1-yl-ethylamino)-pyrimidin-4-yl]-acetonitrile 318160 (2Z)-(2-aminopyrimidin-4-yl)(1,3-benzothiazol-2(3H)-ylidene)acetonitrile 318161 [3H-Benzothiazol-(2Z)-ylidene]-[2-(2-morpholin-4-yl-ethylamino)-pyrimidin-4-yl]-acetonitrile 318165 N*7*-(4-Diethylamino-butyl)-3-phenyl-[1,6]naphthyridine-2,7-diamine 318166 1-tert-Butyl-3-[3-(3,5-dimethoxy-phenyl)-7-(5-hydroxy-pentylamino)-[1,6]naphthyridin-2-yl]-urea 318167 N-(5-Benzyloxy-pentyl)-N-[2-(3-tert-butyl-ureido)-3-(3,5-dimethoxy-phenyl)-3,4-dihydro-[1,6]naphthyridin-7-yl]-acetamide 318171 1-benzyl-7-tert-butyl-3-propyl-1H-imidazo[1,2-a]purine-2,4(3H,8H)-dione 318175 1-(5,6-Diphenyl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)-propan-2-ol 318181 N-[2-(3-tert-Butyl-ureido)-3-(3,5-dimethoxy-phenyl)-3,4-dihydro-[1,6]naphthyridin-7-yl]-N-(4-hydroxy-butyl)-acetamide 318182 [3H-Benzothiazol-(2Z)-ylidene]-{2-[(pyridin-2-ylmethyl)-amino]-pyrimidin-4-yl}-acetonitrile 318183 {2-[2-(4-Amino-phenyl)-ethylamino]-pyrimidin-4-yl}-[3H-benzothiazol-(2Z)-ylidene]-acetonitrile 318190 [3H-Benzothiazol-(2Z)-ylidene]-{2-[2-(3-fluoro-phenyl)-ethylamino]-pyrimidin-4-yl}-acetonitrile 318216 1-tert-Butyl-3-[7-(3-diethylamino-propylamino)-3-(3,5-dimethoxy-phenyl)-[1,6]naphthyridin-2-yl]-urea 318222 (2Z)-1,3-benzothiazol-2(3H)-ylidene[2-(dimethylamino)pyrimidin-4-yl]acetonitrile 318223 (6aR,10aR)-3-Adamantan-2-yl-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol 318241 1-tert-Butyl-3-{3-(3,5-dimethoxy-phenyl)-7-[3-(4-methyl-piperazin-1-yl)-propylamino]-[1,6]naphthyridin-2-yl}-urea 318245 1-tert-Butyl-3-[3-(2,6-dichloro-phenyl)-7-(4-diethylamino-butylamino)-[1,6]naphthyridin-2-yl]-urea 318247 1-[7-(4-Diethylamino-butylamino)-3-(3,5-dimethoxy-phenyl)-[1,6]naphthyridin-2-yl]-3-ethyl-urea 318248 1-tert-Butyl-3-[3-(3,5-dimethoxy-phenyl)-7-(5-morpholin-4-yl-pentylamino)-[1,6]naphthyridin-2-yl]-urea 318249 [2-(3-Amino-propylamino)-pyrimidin-4-yl]-[3H-benzothiazol-(2Z)-ylidene]-acetonitrile 318251 [3H-Benzothiazol-(2Z)-ylidene]-(2-piperazin-1-yl-pyrimidin-4-yl)-acetonitrile 318252 [3H-Benzothiazol-(2Z)-ylidene]-[2-(3-morpholin-4-yl-propylamino)-pyrimidin-4-yl]-acetonitrile 318257 1-benzyl-7-methyl-3-propyl-1H,8H-imidazo[2,1-f]purine-2,4-dione 318266 4-{2-[4-(3-Trifluoromethyl-phenyl)-piperazin-1-yl]-ethoxy}-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-ene-3,5-dione 318275 1-benzyl-7-(4-methoxyphenyl)-3-propyl-1H-imidazo[1,2-a]purine-2,4(3H,8H)-dione 318299 1-benzyl-7-phenyl-3-propyl-1H-pyrrolo[1,2-a]purine-2,4(3H,6H)-dione 318307 {3-[2-(1,1-Diphenyl-propylsulfanyl)-ethyl]-2-hydroxymethyl-benzofuran-7-yloxy}-acetic acid 318317 {3-[2-(2,2-Diphenyl-ethylsulfanyl)-ethyl]-benzofuran-7-yloxy}-acetic acid 318318 [3-(3-Benzhydrylsulfanyl-propyl)-benzofuran-7-yloxy]-acetic acid 318339 {2-Hydroxymethyl-3-[2-(2,2,2-trifluoro-1,1-diphenyl-ethylsulfanyl)-ethyl]-benzofuran-7-yloxy}-acetic acid 318382 4-[2-(4-Pyridin-2-yl-piperazin-1-yl)-ethoxy]-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-ene-3,5-dione 318386 1-benzyl-7-ethyl-3-propyl-1H-pyrrolo[1,2-a]purine-2,4(3H,6H)-dione 318390 Cannabidiol 318400 {3-[2-(Diphenyl-ethanesulfonyl)-ethyl]-2-hydroxymethyl-benzofuran-7-yloxy}-acetic acid 318425 [3-(2,2-Diphenyl-ethylsulfanylmethyl)-benzofuran-7-yloxy]-acetic acid 318436 {3-[3-(3,3-Diphenyl-propylsulfanyl)-propyl]-benzofuran-7-yloxy}-acetic acid 318440 [3-(2-Benzhydrylsulfanyl-ethyl)-2-hydroxymethyl-benzofuran-7-yloxy]-acetic acid 318473 4-{2-[4-(3-Chloro-phenyl)-piperazin-1-yl]-ethoxy}-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-ene-3,5-dione 318481 1-benzyl-7-phenyl-3-propyl-1H-imidazo[1,2-a]purine-2,4(3H,8H)-dione 318514 {3-[2-(1,1-Diphenyl-ethylsulfanyl)-ethyl]-2-hydroxymethyl-benzofuran-7-yloxy}-acetic acid 318520 [3-(2-Benzhydrylsulfanyl-ethyl)-benzofuran-7-yloxy]-acetic acid 318521 {3-[2-(Diphenyl-ethanesulfinyl)-ethyl]-2-hydroxymethyl-benzofuran-7-yloxy}-acetic acid 318568 4-[2-(4-Pyrimidin-2-yl-piperazin-1-yl)-ethoxy]-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-ene-3,5-dione 318604 1-benzyl-7-methyl-3-propyl-1H-pyrrolo[1,2-a]purine-2,4(3H,6H)-dione 318613 (3-Benzhydrylsulfanylmethyl-benzofuran-7-yloxy)-acetic acid 318614 [3-[2-(1,1-Diphenyl-ethylsulfanyl)-ethyl]-2-(2-hydroxy-ethyl)-benzofuran-7-yloxy]-acetic acid 318623 {3-[3-(2,2-Diphenyl-ethylsulfanyl)-propyl]-benzofuran-7-yloxy}-acetic acid 318662 4-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propoxy}-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-ene-3,5-dione 318664 1-benzyl-6,7-dimethyl-3-propyl-1H-pyrrolo[1,2-a]purine-2,4(3H,6H)-dione 318686 {3-[2-(1,1-Diphenyl-ethylsulfanyl)-ethyl]-benzofuran-7-yloxy}-acetic acid 318708 [3-(3,3-Diphenyl-propylsulfanylmethyl)-benzofuran-7-yloxy]-acetic acid 318710 {3-[2-(3,3-Diphenyl-propylsulfanyl)-ethyl]-benzofuran-7-yloxy}-acetic acid 318740 [3-[2-(1,1-Diphenyl-ethylsulfanyl)-ethyl]-2-(3-hydroxy-propyl)-benzofuran-7-yloxy]-acetic acid 318765 N-[4-(3-Bromo-phenylamino)-quinazolin-6-yl]-2-chloro-acetamide 318766 2-Chloro-N-[4-(3-iodo-phenylamino)-quinazolin-6-yl]-acetamide 318773 N-[4-(3-Bromo-phenylamino)-7-(4-methyl-piperazin-1-yl)-quinazolin-6-yl]-acrylamide 318798 4-{3-[4-(3-Chloro-phenyl)-piperazin-1-yl]-propoxy}-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-ene-3,5-dione 318804 H-Dmt-D-Arg(NO2)-Phe-Lys(Z)-OH 318828 Benzofuran-2-carboxylic acid ((S)-1-{(R)-1-[4-(3-dimethylamino-propoxy)-benzyl]-pyrrolidin-3-ylcarbamoyl}-3-methyl-butyl)-amide 318861 N-[4-(4,5-Dichloro-2-fluoro-phenylamino)-quinazolin-6-yl]-2-methoxy-acetamide 318875 (S)-2-(2-Benzo[1,3]dioxol-5-yl-acetylamino)-4-methyl-pentanoic acid {(S)-1-[4-(3-dimethylamino-propoxy)-benzyl]-pyrrolidin-3-yl}-amide 318876 3,4-Dichloro-N-((S)-1-{(S)-1-[4-(3-dimethylamino-propoxy)-benzyl]-pyrrolidin-3-ylcarbamoyl}-3-methyl-butyl)-benzamide 318900 (4,5-Dichloro-2-fluoro-phenyl)-(6,7-dimethoxy-quinazolin-4-yl)-amine 318901 N-[4-(4,5-Dichloro-2-fluoro-phenylamino)-quinazolin-6-yl]-acrylamide 318909 N-((S)-1-{(S)-1-[4-(3-Dimethylamino-propoxy)-benzyl]-pyrrolidin-3-ylcarbamoyl}-3-methyl-butyl)-benzamide 318913 (S)-2-Acetylamino-4-methyl-pentanoic acid {(S)-1-[4-(3-dimethylamino-propoxy)-benzyl]-pyrrolidin-3-yl}-amide 318914 3,4-Dichloro-N-((S)-1-{(S)-1-[4-(3-dimethylamino-propoxy)-benzyl]-pyrrolidin-3-ylcarbamoyl}-2-phenyl-ethyl)-benzamide 318927 N-[4-(4,5-Dichloro-2-fluoro-phenylamino)-7-(4-methyl-piperazin-1-yl)-quinazolin-6-yl]-acrylamide 318937 Thiophene-2-carboxylic acid ((S)-1-{(S)-1-[4-(3-dimethylamino-propoxy)-benzyl]-pyrrolidin-3-ylcarbamoyl}-3-methyl-butyl)-amide 318938 4-Bromo-N-{(S)-1-[4-(3-dimethylamino-propoxy)-benzyl]-pyrrolidin-3-yl}-3-methyl-benzamide 318947 7,11,14,15-tetramethyl-(4S,5R,7S,14S,15R,17R)-3,6-dioxatetracyclo[12.4.0.04,18.05,7]octadeca-1(18),10-diene-4,17-diol 318948 7,11,14,15-tetramethyl-(4S,5S,7R,14S,15R)-3,6-dioxatetracyclo[12.4.0.04,18.05,7]octadeca-1(18),10-dien-4-ol 318951 N-[4-(3-Iodo-phenylamino)-quinazolin-6-yl]-2-methoxy-acetamide 318952 2-Chloro-N-[4-(4,5-dichloro-2-fluoro-phenylamino)-quinazolin-6-yl]-acetamide 318956 4-[3-(4-Pyridin-2-yl-piperazin-1-yl)-propoxy]-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-ene-3,5-dione 318982 4-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propoxy}-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-ene-3,5-dione 318996 4-{2-[4-(2-Chloro-phenyl)-piperazin-1-yl]-ethoxy}-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-ene-3,5-dione 319011 Sodium salt {3-[(S)-2-(4,5-diphenyl-oxazol-2-yl)-cyclopent-2-enylmethyl]-phenoxy}-acetate 319018 H-Dmt-D-Arg(NO2)-Phe-Lys(Z)-NH2 319049 (E)-4-Dimethylamino-but-2-enoic acid [4-(4,5-dichloro-2-fluoro-phenylamino)-quinazolin-6-yl]-amide 319059 4-Bromo-N-((S)-1-{(S)-1-[4-(3-dimethylamino-propoxy)-benzyl]-pyrrolidin-3-ylcarbamoyl}-3-methyl-butyl)-benzamide 319060 (S)-N-(1-(4-(3-(dimethylamino)propoxy)benzyl)pyrrolidin-3-yl)-4-bromobenzamide 319063 N-((S)-1-{(S)-1-[4-(3-Dimethylamino-propoxy)-benzyl]-pyrrolidin-3-ylcarbamoyl}-3-methyl-butyl)-isonicotinamide 319067 ((S)-1-{(S)-1-[4-(3-Dimethylamino-propoxy)-benzyl]-pyrrolidin-3-ylcarbamoyl}-3-methyl-butyl)-carbamic acid phenyl ester 319068 N-{(S)-1-[4-(3-Dimethylamino-propoxy)-benzyl]-pyrrolidin-3-yl}-benzamide 319078 4-{3-[4-(3-Trifluoromethyl-phenyl)-piperazin-1-yl]-propoxy}-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-ene-3,5-dione 319105 3,4,7,11-tetramethyl-(1R,3R,4S,11S,12S,13R,16S,18S)-14,17,19-trioxapentacyclo[9.7.1.04,16.013,18.016,18]nonadec-7-ene-12,13-diol 319116 (E)-4-Dimethylamino-but-2-enoic acid [4-(3-iodo-phenylamino)-quinazolin-6-yl]-amide 319139 7,11,14,15-tetramethyl-(4S,5S,7R,14S,15R,17S)-3,6-dioxatetracyclo[12.4.0.04,18.05,7]octadeca-1(18),10-diene-4,17-diol 319170 N-[4-(3-Bromo-phenylamino)-quinazolin-6-yl]-2-methoxy-acetamide 319174 4-[3-(4-Pyrimidin-2-yl-piperazin-1-yl)-propoxy]-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-ene-3,5-dione 319193 N-((S)-1-((S)-1-(4-(3-(dimethylamino)propoxy)benzyl)pyrrolidin-3-ylamino)-4-methyl-1-oxopentan-2-yl)benzo[b]thiophene-2-carboxamide 319196 (S)-3,4-dichloro-N-(1-(4-(3-(dimethylamino)propoxy)benzyl)pyrrolidin-3-yl)benzamide 319197 Benzofuran-2-carboxylic acid {(S)-1-[4-(3-dimethylamino-propoxy)-benzyl]-pyrrolidin-3-yl}-amide 319210 4-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethoxy}-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-ene-3,5-dione 319213 4-[4-Bromo-2-(4-fluoro-phenyl)-5-(1-methyl-piperidin-4-yl)-1H-pyrrol-3-yl]-pyridine 319224 (S)-4-Methyl-2-(3-phenyl-ureido)-pentanoic acid {(S)-1-[4-(3-dimethylamino-propoxy)-benzyl]-pyrrolidin-3-yl}-amide 319226 3,4-Dichloro-N-((S)-1-{(S)-1-[4-(3-dimethylamino-propoxy)-benzyl]-pyrrolidin-3-ylcarbamoyl}-2-methyl-propyl)-benzamide 319250 Furan-2-carboxylic acid ((S)-1-{(S)-1-[4-(3-dimethylamino-propoxy)-benzyl]-pyrrolidin-3-ylcarbamoyl}-3-methyl-butyl)-amide 319256 Isoquinoline-1-carboxylic acid [1'-(3,4-dichloro-benzyl)-[1,4']bipiperidinyl-3-ylmethyl]-amide 319257 2-[4-(Benzenesulfonylamino-methyl)-phenyl]-N-[(S)-2-((S)-3-hydroxy-pyrrolidin-1-yl)-1-phenyl-ethyl]-N-methyl-acetamide 319260 6-[2-(1-Isobutyl-piperidin-4-yl)-5-phenyl-3H-imidazol-4-yl]-1-(propane-2-sulfonyl)-1H-benzoimidazol-2-ylamine 319261 2-(4-Aminomethyl-phenyl)-N-methyl-N-((S)-1-phenyl-2-pyrrolidin-1-yl-ethyl)-acetamide 319262 2-[2-(Acetylamino-methyl)-phenyl]-N-methyl-N-((S)-1-phenyl-2-pyrrolidin-1-yl-ethyl)-acetamide 319266 4-[4-Chloro-2-(4-fluoro-phenyl)-5-(1-methyl-piperidin-4-yl)-1H-pyrrol-3-yl]-pyridine 319287 Quinoline-6-carboxylic acid {1'-[2-(3,4-dichloro-phenyl)-acetyl]-[1,4']bipiperidinyl-3-ylmethyl}-amide 319289 4-[2-(4-Fluoro-phenyl)-4-methyl-5-(1-methyl-piperidin-4-yl)-1H-pyrrol-3-yl]-pyridine 319290 3-(3-Chloro-4-fluoro-phenyl)-1-[(1S,3R,6R)-6-(3-cyano-phenyl)-bicyclo[4.1.0]hept-3-yl]-1-[2-((R)-3-hydroxy-pyrrolidin-1-yl)-ethyl]-urea 319291 N-[(S)-2-((S)-3-Hydroxy-pyrrolidin-1-yl)-1-phenyl-ethyl]-N-methyl-2-{4-[(toluene-4-sulfonylamino)-methyl]-phenyl}-acetamide 319312 Quinoline-6-carboxylic acid [1'-(3,4-dichloro-benzyl)-3'-methyl-[1,4']bipiperidinyl-3-ylmethyl]-amide 319318 1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-ylmethyl}-cyclopropylamine 319319 4-[5-(1-Methyl-piperidin-4-yl)-2-(4-trifluoromethoxy-phenyl)-1H-pyrrol-3-yl]-pyridine 319322 4-[2-(4-Fluoro-phenyl)-5-(1-methyl-piperidin-4-yl)-furan-3-yl]-pyridine 319323 7,11,14,15-tetramethyl-(4S,5R,7S,14S,15R)-3,6-dioxatetracyclo[12.4.0.04,18.05,7]octadeca-1(18),10-dien-4-ol 319351 Naphthalene-2-carboxylic acid [1'-(3,4-dichloro-benzyl)-[1,4']bipiperidinyl-3-ylmethyl]-amide 319352 Quinoline-6-carboxylic acid {1'-[1-(3,4-dichloro-phenyl)-ethyl]-[1,4']bipiperidinyl-3-ylmethyl}-amide 319357 3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-((R)-3-hydroxypyrrolidin-1-yl)ethyl)urea 319365 4-[2-(4-Fluoro-phenyl)-5-(1-methyl-piperidin-4-yl)-thiophen-3-yl]-pyridine 319366 4-[2-(4-Fluoro-phenyl)-5-(1-methyl-piperidin-4-yl)-1H-pyrrol-3-yl]-2-methyl-pyridine 319367 Sodium salt {(R)-5-[(R)-2-(4,5-diphenyl-oxazol-2-yl)-pyrrolidin-1-yl]-5,6,7,8-tetrahydro-naphthalen-1-yloxy}-acetate 319388 Quinoline-8-carboxylic acid [1'-(3,4-dichloro-benzyl)-[1,4']bipiperidinyl-3-ylmethyl]-amide 319393 4-[2-(3-Chloro-4-fluoro-phenyl)-5-(1-methyl-piperidin-4-yl)-1H-pyrrol-3-yl]-pyridine 319395 4-(2-(4-fluorophenyl)-5-(1-methylpiperidin-4-yl)-1H-pyrrol-3-yl)pyridine 319405 N-[1'-(3,4-Dichloro-benzyl)-[1,4']bipiperidinyl-3-ylmethyl]-2-methyl-benzamide 319419 6-(5-Phenyl-2-piperidin-4-yl-3H-imidazol-4-yl)-1-(propane-2-sulfonyl)-1H-benzoimidazol-2-ylamine 319420 2-Amino-6-[2-(2,6-difluoro-phenyl)-5-phenyl-3H-imidazol-4-yl]-benzoimidazole-1-sulfonic acid dimethylamide; Bismesylate salt 319421 2-(2-Aminomethyl-phenyl)-N-methyl-N-((S)-1-phenyl-2-pyrrolidin-1-yl-ethyl)-acetamide 319422 2-(3-Aminomethyl-phenyl)-N-methyl-N-((S)-1-phenyl-2-pyrrolidin-1-yl-ethyl)-acetamide 319428 Quinoline-2-carboxylic acid ((S)-1-{(S)-1-[4-(3-dimethylamino-propoxy)-benzyl]-pyrrolidin-3-ylcarbamoyl}-3-methyl-butyl)-amide 319429 Benzo[1,3]dioxole-5-carboxylic acid ((S)-1-{(S)-1-[4-(3-dimethylamino-propoxy)-benzyl]-pyrrolidin-3-ylcarbamoyl}-3-methyl-butyl)-amide 319433 1H-Indole-5-carboxylic acid [1'-(3,4-dichloro-benzyl)-[1,4']bipiperidinyl-3-ylmethyl]-amide 319437 1H-Benzoimidazole-5-carboxylic acid [1'-(3,4-dichloro-benzyl)-[1,4']bipiperidinyl-3-ylmethyl]-amide 319448 Quinoline-6-carboxylic acid [1'-(3,4-dichloro-benzyl)-4'-methyl-[1,4']bipiperidinyl-3-ylmethyl]-amide 319451 2-{4-[(Butane-1-sulfonylamino)-methyl]-phenyl}-N-[(S)-2-((S)-3-hydroxy-pyrrolidin-1-yl)-1-phenyl-ethyl]-N-methyl-acetamide 319456 4-Chloro-N-{(S)-1-[4-(3-dimethylamino-propoxy)-benzyl]-pyrrolidin-3-yl}-3-methyl-benzamide 319471 N-[1'-(3,4-Dichloro-benzyl)-[1,4']bipiperidinyl-3-ylmethyl]-2-o-tolyl-acetamide 319484 6-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imidazol-4-yl]-1-(propane-2-sulfonyl)-1H-benzoimidazol-2-ylamine 319485 1-[(1S,2R,5S)-5-(4-Cyano-phenyl)-bicyclo[3.1.0]hex-2-yl]-3-(3,5-dichloro-phenyl)-1-(2-pyrrolidin-1-yl-ethyl)-urea 319512 1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-ylmethyl}-cyclopropanol 319515 4-[2-(4-Fluoro-phenyl)-5-(1-methyl-piperidin-4-yl)-1H-pyrrol-3-yl]-3-methyl-pyridine 319528 N-[1'-(3,4-Dichloro-benzyl)-[1,4']bipiperidinyl-3-ylmethyl]-2-methoxy-benzamide 319529 Quinoline-6-carboxylic acid [1'-(2,5-dichloro-benzyl)-[1,4']bipiperidinyl-3-ylmethyl]-amide 319541 4-[5-(1-Methyl-piperidin-4-yl)-3-pyridin-4-yl-1H-pyrrol-2-yl]-phenol 319543 4-[2-(3,4-Difluoro-phenyl)-5-(1-methyl-piperidin-4-yl)-1H-pyrrol-3-yl]-pyridine 319546 Benzofuran-2-carboxylic acid ((R)-1-{(R)-1-[4-(3-dimethylamino-propoxy)-benzyl]-pyrrolidin-3-ylcarbamoyl}-3-methyl-butyl)-amide 319547 1H-Indole-2-carboxylic acid ((S)-1-{(S)-1-[4-(3-dimethylamino-propoxy)-benzyl]-pyrrolidin-3-ylcarbamoyl}-3-methyl-butyl)-amide 319565 SID26756760 319567 Quinoline-6-carboxylic acid [1'-(3,4-dichloro-benzyl)-[1,4']bipiperidinyl-3-ylmethyl]-amide 319572 2-{4-[(4-Fluoro-benzenesulfonylamino)-methyl]-phenyl}-N-[(S)-2-((S)-3-hydroxy-pyrrolidin-1-yl)-1-phenyl-ethyl]-N-methyl-acetamide 319575 3,5-Dichloro-N-{(S)-1-[4-(3-dimethylamino-propoxy)-benzyl]-pyrrolidin-3-yl}-benzamide 319576 Benzo[1,3]dioxole-5-carboxylic acid {(S)-1-[4-(3-dimethylamino-propoxy)-benzyl]-pyrrolidin-3-yl}-amide 319579 Cinnoline-4-carboxylic acid [1'-(3,4-dichloro-benzyl)-[1,4']bipiperidinyl-3-ylmethyl]-amide 319585 1H-Indole-4-carboxylic acid [1'-(3,4-dichloro-benzyl)-[1,4']bipiperidinyl-3-ylmethyl]-amide 319603 6-(2-(2,6-dichlorophenyl)-4-phenyl-1H-imidazol-5-yl)-1-(isopropylsulfonyl)-1H-benzo[d]imidazol-2-amine monomesylate 319604 1-Cyclopentanesulfonyl-6-[2-(2,6-difluoro-phenyl)-5-phenyl-3H-imidazol-4-yl]-1H-benzoimidazol-2-ylamine; Bismesylate salt 319608 2-[3-(Acetylamino-methyl)-phenyl]-N-methyl-N-((S)-1-phenyl-2-pyrrolidin-1-yl-ethyl)-acetamide 319609 N-[(S)-2-((S)-3-Hydroxy-pyrrolidin-1-yl)-1-phenyl-ethyl]-N-methyl-2-[4-(phenylmethanesulfonylamino-methyl)-phenyl]-acetamide 319635 3-(3-Chloro-4-fluoro-phenyl)-1-[(1R,3R,6S)-6-(3-cyano-phenyl)-bicyclo[4.1.0]hept-3-yl]-1-[2-((R)-3-hydroxy-pyrrolidin-1-yl)-ethyl]-urea 319638 4-[5-(4-Fluoro-phenyl)-2-(1-methyl-piperidin-4-yl)-1H-imidazol-4-yl]-pyridine 319639 6-[5-(4-Fluoro-phenyl)-3-methyl-3H-imidazol-4-yl]-1-(propane-2-sulfonyl)-1H-benzoimidazol-2-ylamine 319640 1-[(1S,2R,5S)-5-(2-Cyano-phenyl)-bicyclo[3.1.0]hex-2-yl]-3-(4-fluoro-3-trifluoromethyl-phenyl)-1-[2-((R)-3-hydroxy-pyrrolidin-1-yl)-ethyl]-urea 319662 Naphthalene-1-carboxylic acid [1'-(3,4-dichloro-benzyl)-[1,4']bipiperidinyl-3-ylmethyl]-amide 319667 4-{2-(4-Fluoro-phenyl)-5-[1-(1-methyl-azetidin-2-ylmethyl)-piperidin-4-yl]-1H-pyrrol-3-yl}-pyridine 319668 4-[2-(4-Methanesulfonyl-phenyl)-5-(1-methyl-piperidin-4-yl)-1H-pyrrol-3-yl]-pyridine 319671 4-[4-(4-Fluoro-phenyl)-2-(1-methyl-piperidin-4-yl)-oxazol-5-yl]-pyridine 319686 Quinoline-6-carboxylic acid [1'-(4-chloro-benzyl)-[1,4']bipiperidinyl-3-ylmethyl]-amide 319688 Quinoline-6-carboxylic acid {1'-[2-(3,4-dichloro-phenyl)-ethyl]-[1,4']bipiperidinyl-3-ylmethyl}-amide 319698 4-[4-(4-Fluoro-phenyl)-2-(1-methyl-piperidin-4-yl)-thiazol-5-yl]-pyridine 319699 3-[2-(4-Fluoro-phenyl)-5-(1-methyl-piperidin-4-yl)-1H-pyrrol-3-yl]-pyridine 319710 N-[1'-(3,4-Dichloro-benzyl)-[1,4']bipiperidinyl-3-ylmethyl]-acetamide 319727 4-[2-(3-Bromo-4-fluoro-phenyl)-5-(1-methyl-piperidin-4-yl)-1H-pyrrol-3-yl]-pyridine 319731 Quinoline-4-carboxylic acid [1'-(3,4-dichloro-benzyl)-[1,4']bipiperidinyl-3-ylmethyl]-amide 319738 Cyclohexanecarboxylic acid [1'-(3,4-dichloro-benzyl)-[1,4']bipiperidinyl-3-ylmethyl]-amide 319739 Quinoline-6-carboxylic acid [1'-(3,5-dichloro-benzyl)-[1,4']bipiperidinyl-3-ylmethyl]-amide 319749 3-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-6-p-tolyl-1,5-dihydro-pyrrolo[3,2-d]pyrimidine-2,4-dione 319752 N-[(S)-2-((S)-3-Hydroxy-pyrrolidin-1-yl)-1-phenyl-ethyl]-2-(4-methanesulfonylamino-phenyl)-N-methyl-acetamide 319755 1-[4-(3-Cyano-phenyl)-cyclohexyl]-3-(4-fluoro-3-trifluoromethyl-phenyl)-1-[2-((R)-3-hydroxy-pyrrolidin-1-yl)-ethyl]-urea 319756 4-[5-(1-Methyl-piperidin-4-yl)-2-thiophen-3-yl-1H-pyrrol-3-yl]-pyridine 319757 4-[2-Furan-3-yl-5-(1-methyl-piperidin-4-yl)-1H-pyrrol-3-yl]-pyridine 319764 6-(4-Methoxy-phenyl)-3-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]-propyl}-1,5-dihydro-pyrrolo[3,2-d]pyrimidine-2,4-dione 319782 4-[5-(1-Ethyl-piperidin-4-yl)-2-(4-fluoro-phenyl)-1H-pyrrol-3-yl]-pyridine 319783 2-[2-(Methanesulfonylamino-methyl)-phenyl]-N-methyl-N-((S)-1-phenyl-2-pyrrolidin-1-yl-ethyl)-acetamide 319784 N-[(S)-2-((S)-3-Hydroxy-pyrrolidin-1-yl)-1-phenyl-ethyl]-2-[4-(3-methanesulfonylamino-propyl)-phenyl]-N-methyl-acetamide 319805 6-(2-Chloro-phenyl)-3-{2-[4-(2-chloro-phenyl)-piperazin-1-yl]-ethyl}-1,5-dihydro-pyrrolo[3,2-d]pyrimidine-2,4-dione 319823 N-[(S)-2-((S)-3-Hydroxy-pyrrolidin-1-yl)-1-phenyl-ethyl]-N-methyl-2-{4-[(propane-2-sulfonylamino)-methyl]-phenyl}-acetamide 319827 6-[5-(4-Fluoro-phenyl)-2-isopropyl-3H-imidazol-4-yl]-1-(propane-2-sulfonyl)-1H-benzoimidazol-2-ylamine; compound with methanesulfonic acid 319828 6-[2-tert-Butyl-5-(2,4-difluoro-phenyl)-3H-imidazol-4-yl]-1-(2-methyl-propane-2-sulfonyl)-1H-benzoimidazol-2-ylamine; compound with methanesulfonic acid 319845 1-[(1S,2R,5S)-5-(4-Cyano-phenyl)-bicyclo[3.1.0]hex-2-yl]-3-(4-fluoro-3-trifluoromethyl-phenyl)-1-[4-(4-methyl-piperazin-1-yl)-butyl]-urea 319848 2-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-ethylamine 319852 6-(2-(2,6-difluorophenyl)-4-phenyl-1H-imidazol-5-yl)-1-(isopropylsulfonyl)-1H-benzo[d]imidazol-2-amine 319855 3-(3-Chloro-4-fluoro-phenyl)-1-[(3R,6R)-6-(3-cyano-phenyl)-bicyclo[4.1.0]hept-3-yl]-1-[2-((R)-3-hydroxy-pyrrolidin-1-yl)-ethyl]-urea 319879 4-[5-(1-Methyl-piperidin-4-yl)-2-phenyl-1H-pyrrol-3-yl]-pyridine 319881 2-[4-(Methanesulfonylamino-methyl)-phenyl]-N-methyl-N-((S)-1-phenyl-2-pyrrolidin-1-yl-ethyl)-acetamide 319884 3-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-propan-1-ol 319885 4-[5-(1-Methyl-piperidin-4-yl)-2-(4-trifluoromethyl-phenyl)-1H-pyrrol-3-yl]-pyridine 319891 3-{2-[4-(2-Chloro-phenyl)-piperazin-1-yl]-ethyl}-6-phenyl-1,5-dihydro-pyrrolo[3,2-d]pyrimidine-2,4-dione 319920 3-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyl}-1,5-dihydro-pyrrolo[3,2-d]pyrimidine-2,4-dione 319933 2-[4-(Acetylamino-methyl)-phenyl]-N-methyl-N-((S)-1-phenyl-2-pyrrolidin-1-yl-ethyl)-acetamide 319937 1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-propan-2-one 319960 N-[(S)-2-((S)-3-Hydroxy-pyrrolidin-1-yl)-1-phenyl-ethyl]-N-methyl-2-{4-[(thiophen-2-ylmethanesulfonylamino)-methyl]-phenyl}-acetamide 319966 4-[2-(4-Chloro-phenyl)-5-(1-methyl-piperidin-4-yl)-1H-pyrrol-3-yl]-pyridine 319967 4-[2-Furan-2-yl-5-(1-methyl-piperidin-4-yl)-1H-pyrrol-3-yl]-pyridine 319970 6-[2-Ethyl-5-(4-fluoro-phenyl)-3H-imidazol-4-yl]-1-(propane-2-sulfonyl)-1H-benzoimidazol-2-ylamine; compound with methanesulfonic acid 319971 6-[2-tert-Butyl-5-(2,4-difluoro-phenyl)-3H-imidazol-4-yl]-1-(propane-2-sulfonyl)-1H-benzoimidazol-2-ylamine; compound with methanesulfonic acid 319980 3-{3-[4-(2-Chloro-phenyl)-piperazin-1-yl]-propyl}-6-phenyl-1,5-dihydro-pyrrolo[3,2-d]pyrimidine-2,4-dione 319991 3-(4-Fluoro-phenyl)-6-(1-methyl-piperidin-4-yl)-4-pyridin-4-yl-pyridazine 319992 2-[2-(4-Fluoro-phenyl)-5-(1-methyl-piperidin-4-yl)-1H-pyrrol-3-yl]-pyridine 319997 2-[4-(Ethanesulfonylamino-methyl)-phenyl]-N-[(S)-2-((S)-3-hydroxy-pyrrolidin-1-yl)-1-phenyl-ethyl]-N-methyl-acetamide 320002 3-(3-Chloro-4-fluoro-phenyl)-1-[4-(3-cyano-phenyl)-cyclohex-3-enyl]-1-(2-pyrrolidin-1-yl-ethyl)-urea 320018 3-{2-[4-(2-Chloro-phenyl)-piperazin-1-yl]-ethyl}-1,5-dihydro-pyrrolo[3,2-d]pyrimidine-2,4-dione 320022 N-[(S)-2-((S)-3-Hydroxy-pyrrolidin-1-yl)-1-phenyl-ethyl]-2-[4-(2-methanesulfonylamino-ethyl)-phenyl]-N-methyl-acetamide 320039 6-(2-Chloro-phenyl)-3-{2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-1,5-dihydro-pyrrolo[3,2-d]pyrimidine-2,4-dione 320052 2-[3-(Methanesulfonylamino-methyl)-phenyl]-N-methyl-N-((S)-1-phenyl-2-pyrrolidin-1-yl-ethyl)-acetamide 320053 2-(2-Methanesulfonyl-2,3-dihydro-1H-isoindol-5-yl)-N-methyl-N-((S)-1-phenyl-2-pyrrolidin-1-yl-ethyl)-acetamide 320058 1-[4-(3-Cyano-phenyl)-cyclohexyl]-3-(4-fluoro-3-trifluoromethyl-phenyl)-1-[2-((R)-3-hydroxy-pyrrolidin-1-yl)-ethyl]-urea 320059 2-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-1-methyl-ethylamine 320060 4-[5-(1-Methyl-piperidin-4-yl)-2-thiazol-2-yl-1H-pyrrol-3-yl]-pyridine 320074 6-(3-Chloro-phenyl)-3-{2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-1,5-dihydro-pyrrolo[3,2-d]pyrimidine-2,4-dione 320078 2-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-ethanol 320079 4-[4,5-Bis-(4-fluoro-phenyl)-1H-pyrrol-2-yl]-1-methyl-piperidine 320087 3-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-6-phenyl-1,5-dihydro-pyrrolo[3,2-d]pyrimidine-2,4-dione 320109 4-[2-(4-Fluoro-phenyl)-5-(1-propyl-piperidin-4-yl)-1H-pyrrol-3-yl]-pyridine 320115 N-[(S)-2-((S)-3-Hydroxy-pyrrolidin-1-yl)-1-phenyl-ethyl]-N-methyl-2-{4-[(propane-1-sulfonylamino)-methyl]-phenyl}-acetamide 320116 3-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyl}-6-p-tolyl-1,5-dihydro-pyrrolo[3,2-d]pyrimidine-2,4-dione 320130 6-(4-Chloro-phenyl)-3-{2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-1,5-dihydro-pyrrolo[3,2-d]pyrimidine-2,4-dione 320137 4-[2-(3-Fluoro-phenyl)-5-(1-methyl-piperidin-4-yl)-1H-pyrrol-3-yl]-pyridine 320141 1-(isopropylsulfonyl)-6-(4-phenyl-1H-imidazol-5-yl)-1H-benzo[d]imidazol-2-amine 320142 6-[5-(4-Fluoro-phenyl)-3H-imidazol-4-yl]-1-(propane-2-sulfonyl)-1H-benzoimidazol-2-ylamine; Bismesylate salt 320143 6-[2-tert-Butyl-5-(4-fluoro-phenyl)-3H-imidazol-4-yl]-1-(propane-2-sulfonyl)-1H-benzoimidazol-2-ylamine; Bismesylate salt 320166 N-(2-((2-(dimethylamino)ethyl)(methyl)amino)-4-methylquinolin-6-yl)-3-(4-(trifluoromethoxy)phenyl)acrylamide 320173 N-[(S)-2-((S)-3-Hydroxy-pyrrolidin-1-yl)-1-phenyl-ethyl]-2-[4-(methanesulfonylamino-methyl)-phenyl]-N-methyl-acetamide 320182 1-[4-(3-Cyano-phenyl)-4-methyl-cyclohexyl]-3-(4-fluoro-3-trifluoromethyl-phenyl)-1-[2-((R)-3-hydroxy-pyrrolidin-1-yl)-ethyl]-urea 320184 3-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-propylamine 320202 3-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-1,5-dihydro-pyrrolo[3,2-d]pyrimidine-2,4-dione 320205 N-Methyl-2-{4-[(3-methyl-ureido)-methyl]-phenyl}-N-((S)-1-phenyl-2-pyrrolidin-1-yl-ethyl)-acetamide 320216 3-{3-[4-(2-Chloro-phenyl)-piperazin-1-yl]-propyl}-1,5-dihydro-pyrrolo[3,2-d]pyrimidine-2,4-dione 320219 3-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyl}-6-phenyl-1,5-dihydro-pyrrolo[3,2-d]pyrimidine-2,4-dione 320236 5,5-Bis-(4-bromo-phenyl)-3-ethyl-2-thioxo-imidazolidin-4-one 320237 3-Allyl-5,5-bis-(4-iodo-phenyl)-imidazolidine-2,4-dione 320246 (S)-2-((R)-2-Methyl-4-naphthalen-1-yl-piperazin-1-ylmethyl)-hexahydro-pyrrolo[1,2-a]pyrazine-1,4-dione 320263 1-((S)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizin-3-yl)-ethanone 320266 (S)-2-[4-((S)-2-Methyl-4-naphthalen-1-yl-piperazin-1-yl)-butyl]-hexahydro-pyrrolo[1,2-a]pyrazine-1,4-dione 320267 2-[4-(9H-5,6-Dioxa-benzocyclohepten-1-yl)-piperazin-1-ylmethyl]-hexahydro-pyrrolo[1,2-a]pyrazine-1,4-dione 320288 ((R)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizin-3-yl)-phenyl-methanone 320289 ((R)-3-Dimethylaminomethyl-5,6,7,8-tetrahydro-indolizin-7-yl)-dipropyl-amine 320290 ((S)-3-Dimethylaminomethyl-5,6,7,8-tetrahydro-indolizin-7-yl)-dipropyl-amine 320317 5,5-bis(4-bromophenyl)-3-butylimidazolidine-2,4-dione 320323 Dipropyl-(S)-5,6,7,8-tetrahydro-indolizin-7-yl-amine 320327 3-Allyl-5,5-bis-(4-bromo-phenyl)-2-thioxo-imidazolidin-4-one 320341 (7R)-3-[(1E)-(hydroxyimino)methyl]-N,N-dipropyl-5,6,7,8-tetrahydroindolizin-7-amine 320342 (S)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizine-3-carbaldehyde oxime 320346 SID11112643 320350 (S)-2-(4-Naphthalen-1-yl-piperazin-1-ylmethyl)-hexahydro-pyrrolo[1,2-a]pyrazine-1,4-dione 320372 1-((S)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizin-3-yl)-2,2,2-trifluoro-ethanone 320376 5,5-bis(4-bromophenyl)-3-butyl-2-thioxoimidazolidin-4-one 320400 5,5-Bis-(4-chloro-phenyl)-3-phenethyl-2-thioxo-imidazolidin-4-one 320428 3-Butyl-5,5-bis-(4-iodo-phenyl)-imidazolidine-2,4-dione 320439 (S)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizine-3-carbonitrile 320440 1-((R)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizin-3-yl)-ethanone 320441 2-((R)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizin-3-ylmethylene)-malononitrile 320456 (R)-2-[4-((R)-2-Methyl-4-naphthalen-1-yl-piperazin-1-yl)-butyl]-hexahydro-pyrrolo[1,2-a]pyrazine-1,4-dione 320471 (S)-2-((S)-2-Methyl-4-naphthalen-1-yl-piperazin-1-ylmethyl)-hexahydro-pyrrolo[1,2-a]pyrazine-1,4-dione 320473 2-((S)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizin-3-ylmethylene)-malononitrile 320494 (R)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizine-3-carboxylic acid ethyl ester 320495 (S)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizine-3-carboxylic acid ethyl ester 320500 (R)-5,6,6a,7-Tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol 320511 3-Allyl-5,5-bis-(4-iodo-phenyl)-2-thioxo-imidazolidin-4-one 320531 5,5-Bis-(4-bromo-phenyl)-3-isopropyl-2-thioxo-imidazolidin-4-one 320538 (R)-2-(4-Naphthalen-1-yl-piperazin-1-ylmethyl)-hexahydro-pyrrolo[1,2-a]pyrazine-1,4-dione 320543 (R)-2-((S)-2-Methyl-4-naphthalen-1-yl-piperazin-1-ylmethyl)-hexahydro-pyrrolo[1,2-a]pyrazine-1,4-dione 320556 ((S)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizin-3-yl)-phenyl-methanone 320584 1-((R)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizin-3-yl)-2,2,2-trifluoro-ethanone 320585 (R)-5-Dipropylamino-4,5,6,7-tetrahydro-indole-1-carbaldehyde 320586 (S)-5-Dipropylamino-4,5,6,7-tetrahydro-indole-1-carbaldehyde 320590 (S)-2-[4-(9H-5,6-Dioxa-benzocyclohepten-1-yl)-piperazin-1-ylmethyl]-hexahydro-pyrrolo[1,2-a]pyrazine-1,4-dione 320599 ((R)-3-Phenyl-5,6,7,8-tetrahydro-indolizin-7-yl)-dipropyl-amine 320616 3-benzyl-5,5-bis(4-chlorophenyl)-2-thioxoimidazolidin-4-one 320617 3-Benzyl-5,5-bis-(4-bromo-phenyl)-imidazolidine-2,4-dione 320626 3-Benzyl-5,5-bis-(4-bromo-phenyl)-2-thioxo-imidazolidin-4-one 320645 2-[4-(4-Naphthalen-1-yl-piperazin-1-yl)-butyl]-hexahydro-pyrrolo[1,2-a]pyrazine-1,4-dione 320654 (7R)-3-[(1Z)-(hydroxyimino)methyl]-N,N-dipropyl-5,6,7,8-tetrahydroindolizin-7-amine 320655 (S)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizine-3-carbaldehyde oxime 320664 (R)-2-((R)-2-Methyl-4-naphthalen-1-yl-piperazin-1-ylmethyl)-hexahydro-pyrrolo[1,2-a]pyrazine-1,4-dione 320666 (R)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizine-3-carbonitrile 320667 ((S)-3-Phenyl-5,6,7,8-tetrahydro-indolizin-7-yl)-dipropyl-amine 320681 2,2,2-Trichloro-1-((R)-7-dipropylamino-5,6,7,8-tetrahydro-indolizin-3-yl)-ethanone 320682 2,2,2-Trichloro-1-((S)-7-dipropylamino-5,6,7,8-tetrahydro-indolizin-3-yl)-ethanone 320686 5,5-Bis-(4-bromo-phenyl)-3-isobutyl-2-thioxo-imidazolidin-4-one 320694 5,5-Bis-(4-chloro-phenyl)-3-isobutyl-2-thioxo-imidazolidin-4-one 320695 3-Butyl-5,5-bis-(4-iodo-phenyl)-2-thioxo-imidazolidin-4-one 320713 (R)-3-(2-amino-2-phenylethyl)-1-(2,6-difluorobenzyl)-5-(2-fluoro-3-methoxyphenyl)pyrimidine-2,4(1H,3H)-dione 320723 8-(2-chloro-3,4,5-trimethoxyphenylthio)-2-fluoro-9-(pent-4-ynyl)-9H-purin-6-amine 320747 3-((S)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-1H-pyrimidine-2,4-dione 320844 Naphthalene-2-carboxylic acid {1-[2-((S)-8-methoxy-1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-ethyl]-piperidin-4-yl}-amide 320848 Radiolabeled octreotide derivative 320849 Radiolabeled octreotide derivative 320850 Radiolabeled octreotide derivative 320997 8-{2-[4-(3,4-Difluoro-phenyl)-piperazin-1-yl]-ethyl}-8-aza-spiro[4.5]decane-7,9-dione 321054 Naphthalene-2-carboxylic acid {1-[2-((R)-8-methoxy-1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-ethyl]-piperidin-4-yl}-amide 321070 8-(2-iodo-5-methoxyphenylthio)-9-(pent-4-ynyl)-9H-purin-6-amine 321095 3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-fluoro-3-methoxy-phenyl)-1-(2-fluoro-6-methylsulfanyl-benzyl)-1H-pyrimidine-2,4-dione 321133 (R)-1-(2-fluoro-6-(trifluoromethyl)benzyl)-3-(2-amino-2-phenylethyl)-5-phenylpyrimidine-2,4(1H,3H)-dione 321135 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-5-(2-fluoro-3-hydroxy-phenyl)-1H-pyrimidine-2,4-dione 321170 Radiolabeled octreotide derivative 321171 Radiolabeled octreotide derivative 321172 Radiolabeled octreotide derivative 321201 8-{2-[4-(2,4-Difluoro-phenyl)-piperazin-1-yl]-ethyl}-8-aza-spiro[4.5]decane-7,9-dione 321202 2-[3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-fluoro-3-methoxy-phenyl)-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-ylmethyl]-3-fluoro-N,N-dimethyl-benzenesulfonamide 321203 3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-fluoro-3-methoxy-phenyl)-1-[2-fluoro-6-(morpholine-4-sulfonyl)-benzyl]-1H-pyrimidine-2,4-dione 321271 2-((1R,5S)-3-3-Aza-bicyclo[3.1.0]hex-3-yl-1-phenyl-propyl)-4-methyl-phenol 321276 Naphthalene-2-carboxylic acid [4-((S)-7-methoxy-1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-butyl]-amide 321288 Bis-(4-fluoro-phenyl)-hydroxy-acetic acid 4-(3-aza-bicyclo[3.1.0]hex-3-yl)-but-2-ynyl ester 321299 4-Methyl-2-[3-((1R,5S)-1-methyl-3-aza-bicyclo[3.1.0]hex-3-yl)-1-phenyl-propyl]-phenol 321304 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2-fluoro-6-trifluoromethyl-benzyl)-5-(2-trifluoromethyl-phenyl)-1H-pyrimidine-2,4-dione 321307 3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-fluoro-phenyl)-1-(2-fluoro-6-trifluoromethyl-benzyl)-1H-pyrimidine-2,4-dione 321309 4-(4-methylpiperazin-1-yl)-N-(5-(2-phenylacetyl)-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl)benzamide 321311 {3-[(S)-2-(4,5-Diphenyl-oxazol-2-yl)-cyclohex-2-enylmethyl]-phenyl}-acetic acid 321312 6-{(S)-2-[(Benzofuran-2-carbonyl)-amino]-6-benzyloxycarbonylamino-hexanoylamino}-hexanoic acid 321313 6-{(R)-2-[(Benzofuran-2-carbonyl)-amino]-6-benzyloxycarbonylamino-hexanoylamino}-hexanoic acid 321317 (1S,2R)-2-[2-Amino-3-((S)-4-hydroxy-2,6-dimethyl-phenyl)-propionylamino]-cyclopentanecarboxylic acid [(S)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-ethyl]-amide 321318 (1R,2S)-2-[2-Amino-3-((S)-4-hydroxy-2,6-dimethyl-phenyl)-propionylamino]-cyclopentanecarboxylic acid [(S)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-ethyl]-amide 321319 2-[2-Amino-3-((S)-4-hydroxy-2,6-dimethyl-phenyl)-propionylamino]-cyclohexanecarboxylic acid [(S)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-ethyl]-amide 321320 2-[2-Amino-3-((S)-4-hydroxy-2,6-dimethyl-phenyl)-propionylamino]-cyclohexanecarboxylic acid [(S)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-ethyl]-amide 321321 (1S,2R)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-ylamino)-1-oxo-3-phenylpropan-2-yl)-2-((S)-2-amino-3-(4-hydroxyphenyl)propanamido)cyclohexanecarboxamide 321330 NDP-SYSMEHFRWGKPVG 321333 Naphthalene-2-carboxylic acid [(R)-4-(1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-butyl]-amide 321334 3-((S)-2-Amino-2-phenyl-ethyl)-5-(2-fluoro-3-methoxy-phenyl)-1-(2-fluoro-6-trifluoromethyl-benzyl)-1H-pyrimidine-2,4-dione 321344 (S)-1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid [(S)-1-((1S,2S)-1-carbamoyl-2-phenyl-propylcarbamoyl)-2-phenyl-ethyl]-amide 321345 (S)-1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid {(S)-1-[(S)-1-carbamoyl-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-phenyl-ethyl}-amide 321357 8-{2-[4-(2,4,5-Trifluoro-phenyl)-piperazin-1-yl]-ethyl}-8-aza-spiro[4.5]decane-7,9-dione 321359 3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-fluoro-3-hydroxy-phenyl)-1-(2-fluoro-6-trifluoromethyl-benzyl)-1H-pyrimidine-2,4-dione 321361 Naphthalene-2-carboxylic acid [4-((S)-8-methoxy-1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-butyl]-amide 321367 4-Methyl-2-[3-((1R,5S)-2-methyl-3-aza-bicyclo[3.1.0]hex-3-yl)-1-phenyl-propyl]-phenol 321388 Naphthalene-2-carboxylic acid [4-((S)-9-methoxy-1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-butyl]-amide 321391 2-[(R)-1-Amino-2-((S)-4-hydroxy-phenyl)-ethyl]-thiazolidine-4-carboxylic acid [(S)-1-benzyl-2-((S)-2-carbamoyl-pyrrolidin-1-yl)-2-oxo-ethyl]-amide 321397 Cyclopentyl-hydroxy-(4-methoxy-phenyl)-acetic acid 4-(3-aza-bicyclo[3.1.0]hex-3-yl)-but-2-ynyl ester 321415 (R)-1-(2-fluoro-6-(trifluoromethyl)benzyl)-3-(2-amino-2-phenylethyl)-5-(2-chlorophenyl)pyrimidine-2,4(1H,3H)-dione 321416 3-[(S)-2-(4,5-Diphenyl-oxazol-2-yl)-cyclohex-2-enylmethyl]-benzoic acid 321417 6-{(S)-2-[(Benzofuran-2-carbonyl)-amino]-5-benzyloxycarbonylamino-pentanoylamino}-hexanoic acid 321418 {(S)-4-[(S)-1-(Benzyl-methyl-carbamoyl)-2-phenyl-ethylcarbamoyl]-4-[(1H-indole-2-carbonyl)-amino]-butyl}-carbamic acid benzyl ester 321431 Naphthalene-2-carboxylic acid [4-((R)-7-methoxy-1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-butyl]-amide 321434 3-((R)-2-Amino-2-phenyl-ethyl)-1-(2-chloro-6-fluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-1H-pyrimidine-2,4-dione 321435 (R)-1-(2,6-difluorobenzyl)-3-(2-amino-2-phenylethyl)-5-(2-chlorophenyl)pyrimidine-2,4(1H,3H)-dione 321441 (R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid [(S)-1-((R)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-ethyl]-amide 321442 (R)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid [(S)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-ethyl]-amide 321458 (R)-3-(2-amino-2-phenylethyl)-5-(2-fluoro-3-methoxyphenyl)-1-(2-fluoro-6-(trifluoromethyl)benzyl)pyrimidine-2,4(1H,3H)-dione 321474 (1R,2R)-1-[2-Amino-3-((S)-4-hydroxy-phenyl)-propionylamino]-indan-2-carboxylic acid [(S)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-ethyl]-amide 321475 (1S,2S)-1-[2-Amino-3-((S)-4-hydroxy-phenyl)-propionylamino]-indan-2-carboxylic acid [(S)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-ethyl]-amide 321476 (1R,2S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-ylamino)-1-oxo-3-phenylpropan-2-yl)-2-((S)-2-amino-3-(4-hydroxyphenyl)propanamido)cyclopentanecarboxamide 321477 (1S,2R)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-ylamino)-1-oxo-3-phenylpropan-2-yl)-2-((S)-2-amino-3-(4-hydroxyphenyl)propanamido)cyclopentanecarboxamide 321478 (1R,2S)-2-[2-Amino-3-((S)-4-hydroxy-phenyl)-propionylamino]-cyclopentanecarboxylic acid {(S)-1-[(S)-1-carbamoyl-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-phenyl-ethyl}-amide 321479 (1S,2R)-2-[2-Amino-3-((S)-4-hydroxy-phenyl)-propionylamino]-cyclopentanecarboxylic acid {(S)-1-[(S)-1-carbamoyl-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-phenyl-ethyl}-amide 321490 (R)-1-(2-fluoro-6-(methylsulfonyl)benzyl)-3-(2-amino-2-phenylethyl)-5-(2-fluoro-3-methoxyphenyl)pyrimidine-2,4(1H,3H)-dione 321491 3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-fluoro-3-methoxy-phenyl)-1-[2-fluoro-6-(propane-2-sulfonyl)-benzyl]-1H-pyrimidine-2,4-dione 321492 3-((R)-2-Amino-2-phenyl-ethyl)-1-[2-fluoro-6-(2-hydroxy-ethanesulfonyl)-benzyl]-5-(2-fluoro-3-methoxy-phenyl)-1H-pyrimidine-2,4-dione 321493 Naphthalene-2-carboxylic acid [4-((S)-10-methoxy-1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-butyl]-amide 321511 3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-chloro-phenyl)-1-(2-methanesulfonyl-6-trifluoromethyl-benzyl)-1H-pyrimidine-2,4-dione 321531 Naphthalene-2-carboxylic acid [4-((R)-8-methoxy-1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-butyl]-amide 321551 Naphthalene-2-carboxylic acid [(S)-4-(1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-butyl]-amide 321553 (R)-1-(2-fluoro-6-(methylsulfonyl)benzyl)-3-(2-amino-2-phenylethyl)-5-(2-chlorophenyl)pyrimidine-2,4(1H,3H)-dione 321561 Naphthalene-2-carboxylic acid {4-[2-((S)-8-methoxy-1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-ethyl]-cyclohexyl}-amide 321572 (1R,2S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-ylamino)-1-oxo-3-phenylpropan-2-yl)-2-((S)-2-amino-3-(4-hydroxyphenyl)propanamido)cyclohexanecarboxamide 321573 2-[2-Amino-3-((S)-4-hydroxy-phenyl)-propionylamino]-cyclohexanecarboxylic acid {1-[(S)-(S)-1-carbamoyl-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-phenyl-ethyl}-amide 321574 2-[2-Amino-3-((S)-4-hydroxy-phenyl)-propionylamino]-cyclohexanecarboxylic acid {1-[(S)-(S)-1-carbamoyl-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-phenyl-ethyl}-amide 321587 3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-chloro-3-methoxy-phenyl)-1-(2,6-difluoro-benzyl)-1H-pyrimidine-2,4-dione 321589 Naphthalene-2-carboxylic acid [4-((R)-9-methoxy-1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-butyl]-amide 321594 N-(2,6-diethylphenyl)-3-(4-(4-methylpiperazin-1-yl)benzamido)-4,6-dihydropyrrolo[3,4-c]pyrazole-5(1H)-carboxamide 321619 Naphthalene-2-carboxylic acid [4-((R)-10-methoxy-1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-butyl]-amide 321626 (S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid [(S)-2-((S)-1-carbamoyl-2-(S)-phenyl-ethylcarbamoyl)-indan-1-yl]-amide 321627 (S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid [(R)-2-((R)-1-carbamoyl-2-(S)-phenyl-ethylcarbamoyl)-indan-1-yl]-amide 321634 AEKKDEGPYRMEHFRWGSPPKD 321635 GPYRMEHFRWGSPPKD-NH2 321706 5-{2-[4-(1H-Benzoimidazol-4-ylmethyl)-piperazin-1-yl]-ethoxy}-2-methyl-quinoline 321722 N-{(R)-2-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-4-nitro-N-pyridin-2-yl-benzamide 321723 5-{2-[4-(4-Chloro-3-nitro-benzyl)-piperazin-1-yl]-ethoxy}-2-methyl-quinoline 321727 4-Cyano-N-{(S)-2-[4-(2,3-dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-N-pyridin-2-yl-benzamide 321747 2-Amino-4-{4-[2-(2-methyl-quinolin-5-yloxy)-ethyl]-piperazin-1-ylmethyl}-phenol 321749 (R)-1-(2-fluoro-6-(trifluoromethyl)benzyl)-3-(2-amino-2-phenylethyl)-5-(2-chloro-3-methoxyphenyl)pyrimidine-2,4(1H,3H)-dione 321752 5-{2-[4-(3,4-Dichloro-benzyl)-piperazin-1-yl]-ethoxy}-2-methyl-quinoline 321756 2-Methyl-5-[2-(4-quinolin-5-ylmethyl-piperazin-1-yl)-ethoxy]-quinoline 321771 Ac-YR[CEH(pCl-dF)RWC]-NH2 321772 Ac-YR[CEH(pF-dF)RWC]-NH2 321773 Ac-YR[CE(1-Me-H)dFRWC]-NH2 321774 Hydroxy-diphenyl-acetic acid 4-(3-aza-bicyclo[3.1.0]hex-3-yl)-but-2-ynyl ester 321792 Vasopressin Analogue 321793 Vasopressin Analogue 321822 4-Chloro-N-{(R)-2-[4-(2,3-dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-N-pyridin-2-yl-benzamide 321836 N-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propyl]-3-oxo-2,3,4,5-tetrahydro-1H-benzo[c]azepin-4-yl}-2-phenyl-acetamide 321837 H-Tyr-Tic-Phe-Phe-OH 321848 5-{2-[4-(4-Methoxy-3-nitro-benzyl)-piperazin-1-yl]-ethoxy}-2-methyl-quinoline 321873 5-{2-[4-(1H-Indol-7-ylmethyl)-piperazin-1-yl]-ethoxy}-2-methyl-quinoline 321876 3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-chloro-4-methyl-phenyl)-1-(2-fluoro-6-trifluoromethyl-benzyl)-1H-pyrimidine-2,4-dione 321877 3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-chloro-4-trifluoromethyl-phenyl)-1-(2-fluoro-6-trifluoromethyl-benzyl)-1H-pyrimidine-2,4-dione 321894 N-{(S)-2-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-N-pyridin-2-yl-4-trifluoromethyl-benzamide 321896 3-((R)-2-Amino-2-phenyl-ethyl)-5-(3-ethoxy-2-fluoro-phenyl)-1-(2-fluoro-6-trifluoromethyl-benzyl)-1H-pyrimidine-2,4-dione 321897 3-((R)-2-Amino-2-phenyl-ethyl)-5-[2-fluoro-3-(2,2,2-trifluoro-ethoxy)-phenyl]-1-(2-fluoro-6-trifluoromethyl-benzyl)-1H-pyrimidine-2,4-dione 321898 3-((R)-2-Amino-2-phenyl-ethyl)-5-(2-fluoro-3-isopropoxy-phenyl)-1-(2-fluoro-6-trifluoromethyl-benzyl)-1H-pyrimidine-2,4-dione 321906 N-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propyl]-3-oxo-2,3,4,5-tetrahydro-1H-benzo[c]azepin-4-yl}-2-phenyl-acetamide 321909 C-Phenyl-N-{3-[2-((S)-5-phenyl-4-phenyl-oxazol-2-yl)-cyclohex-2-enylmethyl]-benzoyl}-methanesulfonamide 321910 (S)-2-{(S)-5-Benzyloxycarbonylamino-2-[(1H-indole-2-carbonyl)-amino]-pentanoylamino}-3-phenyl-propionic acid 321917 4-Cyano-N-{(R)-2-[4-(2,3-dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-N-pyridin-2-yl-benzamide 321927 2-{4-[2-(2-Methyl-quinolin-5-yloxy)-ethyl]-piperazin-1-ylmethyl}-2H,7H-benzo[e][1,2]oxazin-6-one 321947 2-Methyl-5-{2-[4-(4-methyl-3-nitro-benzyl)-piperazin-1-yl]-ethoxy}-quinoline 321949 Vasopressin Analogue 321950 Vasopressin Analogue 321964 SID29215497 321965 Ac-YRMEHdFRWGSPPKD-NH2 321967 Ac-YR[CEHdFRWC]-NH2 321968 Ac-YR[CEHFRWC]-NH2 321969 Ac-YRMEHdFRWG-NH2 321970 Ac-YRC(Me)*EHdFRWC(Me)NH2 321971 Ac-YR[CEH(d-2alpha-Nal)RWC]-NH2 321977 4-{4-[2-(2-Methyl-quinolin-5-yloxy)-ethyl]-piperazin-1-ylmethyl}-2-nitro-phenol 321985 8-((4-(2-(2-methylquinolin-5-yloxy)ethyl)piperazin-1-yl)methyl)quinoline 321998 Cyclopentyl-hydroxy-phenyl-acetic acid 4-(3-aza-bicyclo[3.1.0]hex-3-yl)-but-2-ynyl ester 321999 Cyclohexyl-hydroxy-phenyl-acetic acid 4-(3-aza-bicyclo[3.1.0]hex-3-yl)-but-2-ynyl ester 322069 4-Chloro-N-{(S)-2-[4-(2,3-dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-N-pyridin-2-yl-benzamide 322086 Ac-[CEHdFRWC]-NH2 322087 Ac-YCit[CEHdFRWC]-NH2 322088 Ac-YK[CEHdFRWC]-NH2 322089 Ac-R[CEHdFRWC]-NH2 322090 Ac-dR[CEHdFRWC]-NH2 322091 N-Benzyloxy-3-[(S)-2-(4,5-diphenyl-oxazol-2-yl)-cyclohex-2-enylmethyl]-benzamide 322111 5-{2-[4-(2,5-Dichloro-benzyl)-piperazin-1-yl]-ethoxy}-2-methyl-quinoline 322116 Vasopressin Analogue 322117 Vasopressin Analogue 322122 5-Chloro-6-(4-methyl-piperazin-1-yl)-2,3-dihydro-indole-1-carboxylic acid (4-pyridin-4-yl-naphthalen-1-yl)-amide 322128 N-{(S)-2-[(R)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propyl]-3-oxo-2,3,4,5-tetrahydro-1H-benzo[c]azepin-4-yl}-2-phenyl-acetamide 322133 (S)-N-((S)-1-((S)-1-amino-3-(1H-indol-3-yl)-1-oxopropan-2-ylamino)-1-oxo-3-phenylpropan-2-yl)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)pyrrolidine-2-carboxamide 322134 Tyr-Pro-Phe-Pro-NH2 322142 N-{(R)-2-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-N-pyridin-2-yl-4-trifluoromethyl-benzamide 322147 N-{(S)-2-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-4-nitro-N-pyridin-2-yl-benzamide 322148 5-{4-[2-(2-Methyl-quinolin-5-yloxy)-ethyl]-piperazin-1-ylmethyl}-quinazoline 322170 5-{2-[4-(4-Fluoro-3-nitro-benzyl)-piperazin-1-yl]-ethoxy}-2-methyl-quinoline 322180 Vasopressin Analogue 322200 K-252a analogue 322244 N-{(R)-2-[(R)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propyl]-3-oxo-2,3,4,5-tetrahydro-1H-benzo[c]azepin-4-yl}-2-phenyl-acetamide 322247 N-{4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-4-hydroxy-benzamide 322383 2-{1-ferra-1,1'-spirobi[pentacyclo[2.2.0.0^{1,3}.0^{1,5}.0^{2,6}]hexane]-2,2',4,4'-tetraen-6-yl}-N-{4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl}acetamide 322388 K-252a analogue 322426 N-{(E)-4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-4-nitro-benzamide 322444 N-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl}-1-ruthena-1,1'-spirobi[pentacyclo[2.2.0.0^{1,3}.0^{1,5}.0^{2,6}]hexane]-2,2',4,4'-tetraene-6-carboxamide 322534 N-{4-[4-(3-chloro-2-methoxyphenyl)piperazin-1-yl]butyl}-1-ferra-1,1'-spirobi[pentacyclo[2.2.0.0^{1,3}.0^{1,5}.0^{2,6}]hexane]-2,2',4,4'-tetraene-6-carboxamide 322629 N-{4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-4-methoxy-benzamide 322642 N-{4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl}-1-ruthena-1,1'-spirobi[pentacyclo[2.2.0.0^{1,3}.0^{1,5}.0^{2,6}]hexane]-2,2',4,4'-tetraene-6-carboxamide 322674 (2E)-3-{1-ferra-1,1'-spirobi[pentacyclo[2.2.0.0^{1,3}.0^{1,5}.0^{2,6}]hexane]-2,2',4,4'-tetraen-6-yl}-N-{4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl}but-2-enamide 322703 4-(4-Fluoro-3-methoxycarbamoyl-phenylamino)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid ethyl ester 322704 2,4-Difluoro-5-[5-isopropyl-6-(3-methyl-[1,2,4]oxadiazol-5-yl)-pyrrolo[2,1-f][1,2,4]triazin-4-ylamino]-N-methoxy-benzamide 322714 (R)-3-(2,4-Dichloro-phenyl)-2-isobutylamino-1-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-propan-1-one 322735 ethyl 5-isopropyl-4-(3-(methoxycarbamoyl)phenylamino)pyrrolo[1,2-f][1,2,4]triazine-6-carboxylate 322736 [4-(2,4-Difluoro-5-methoxycarbamoyl-phenylamino)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazin-6-yl]-carbamic acid tetrahydro-furan-2-ylmethyl ester 322739 2,4-Difluoro-5-[5-isopropyl-6-(5-methanesulfonylmethyl-[1,3,4]oxadiazol-2-yl)-pyrrolo[2,1-f][1,2,4]triazin-4-ylamino]-N-methoxy-benzamide 322740 N-(1-Benzenesulfonyl-4-methoxy-1H-indol-2-ylmethyl)-propionamide 322745 4-(2,4-Difluoro-5-isopropoxycarbamoyl-phenylamino)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid ethyl ester 322746 2,4-Difluoro-5-[5-isopropyl-6-(5-isopropyl-[1,3,4]oxadiazol-2-yl)-pyrrolo[2,1-f][1,2,4]triazin-4-ylamino]-N-methoxy-benzamide 322771 2,4-Difluoro-5-{5-isopropyl-6-[5-(2,2,2-trifluoro-ethyl)-[1,3,4]oxadiazol-2-yl]-pyrrolo[2,1-f][1,2,4]triazin-4-ylamino}-N-methoxy-benzamide 322777 4-(2-Fluoro-5-methoxycarbamoyl-phenylamino)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid ethyl ester 322799 N-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl}-1-ferra-1,1'-spirobi[pentacyclo[2.2.0.0^{1,3}.0^{1,5}.0^{2,6}]hexane]-2,2',4,4'-tetraene-6-carboxamide 322804 [4-(2,4-Difluoro-5-methoxycarbamoyl-phenylamino)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazin-6-yl]-carbamic acid butyl ester 322813 2,4-difluoro-5-(5-isopropyl-6-(5-methyl-1,3,4-oxadiazol-2-yl)pyrrolo[1,2-f][1,2,4]triazin-4-ylamino)-N-methoxybenzamide 322814 2,4-Difluoro-5-[5-isopropyl-6-(5-methyl-4H-[1,2,4]triazol-3-yl)-pyrrolo[2,1-f][1,2,4]triazin-4-ylamino]-N-methoxy-benzamide 322827 4-(2,4-Difluoro-5-isobutoxycarbamoyl-phenylamino)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid ethyl ester 322828 2,4-Difluoro-5-[6-(5-isobutyl-[1,3,4]oxadiazol-2-yl)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazin-4-ylamino]-N-methoxy-benzamide 322830 5-[6-(5-Cyclopropylmethyl-[1,3,4]oxadiazol-2-yl)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazin-4-ylamino]-2,4-difluoro-N-methoxy-benzamide 322853 7-[(2,4-dichloro-5-methoxyphenyl)amino]-2-[4-(4-morpholinylmethyl)phenyl]thieno[3,2-b]pyridine-6-carbonitrile 322887 7-[(2,4-dichlorophenyl)amino]-2-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}thieno[3,2-b]pyridine-6-carbonitrile 322908 ethyl 5-isopropyl-4-(3-(methoxycarbamoyl)phenoxy)pyrrolo[1,2-f][1,2,4]triazine-6-carboxylate 322909 [4-(2,4-Difluoro-5-methoxycarbamoyl-phenylamino)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazin-6-yl]-carbamic acid 3-piperidin-1-yl-propyl ester 322910 7-(2,4-Dichloro-5-methoxy-phenylamino)-2-[5-(4-methyl-piperazin-1-ylmethyl)-thiophen-2-yl]-thieno[3,2-b]pyridine-6-carbonitrile 322911 ethyl 4-(4-bromo-3-(methoxycarbamoyl)phenylamino)-5-isopropylpyrrolo[1,2-f][1,2,4]triazine-6-carboxylate 322912 2,4-difluoro-5-(5-isopropyl-6-(5-methyloxazol-2-yl)pyrrolo[1,2-f][1,2,4]triazin-4-ylamino)-N-methoxybenzamide 322927 4-(5-Ethoxycarbamoyl-2,4-difluoro-phenylamino)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid ethyl ester 322928 5-[6-(5-Ethyl-[1,3,4]oxadiazol-2-yl)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazin-4-ylamino]-2,4-difluoro-N-methoxy-benzamide 322932 (R)-2-(2-Amino-ethylamino)-3-(2,4-dichloro-phenyl)-1-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-propan-1-one 322936 (R)-N-(3-(2,4-dichlorophenyl)-1-oxo-1-(4-(2-((2-(thiophen-2-yl)ethylamino)methyl)phenyl)piperazin-1-yl)propan-2-yl)acetamide 322937 N-[(R)-1-(2,4-Dichloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-benzamide 322938 4-Amino-N-[(R)-1-(2,4-dichloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-butyramide 322951 2,4-Difluoro-5-[5-isopropyl-6-(5-trifluoromethyl-[1,3,4]oxadiazol-2-yl)-pyrrolo[2,1-f][1,2,4]triazin-4-ylamino]-N-methoxy-benzamide 322954 5-[6-(5-Dimethylaminomethyl-[1,3,4]oxadiazol-2-yl)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazin-4-ylamino]-2,4-difluoro-N-methoxy-benzamide 322974 N-{4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl}-1-ferra-1,1'-spirobi[pentacyclo[2.2.0.0^{1,3}.0^{1,5}.0^{2,6}]hexane]-2,2',4,4'-tetraene-6-carboxamide 322980 [4-(2,4-Difluoro-5-methoxycarbamoyl-phenylamino)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazin-6-yl]-carbamic acid ethyl ester 322981 5-[6-(5-Cyclopropyl-[1,3,4]oxadiazol-2-yl)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazin-4-ylamino]-2,4-difluoro-N-methoxy-benzamide 323018 2,4-Difluoro-5-[5-isopropyl-6-(5-methyl-[1,2,4]oxadiazol-3-yl)-pyrrolo[2,1-f][1,2,4]triazin-4-ylamino]-N-methoxy-benzamide 323053 5-{6-[5-(Difluoro-methanesulfonyl-methyl)-[1,3,4]oxadiazol-2-yl]-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazin-4-ylamino}-2,4-difluoro-N-methoxy-benzamide 323098 (R)-2-(Cyclopropylmethyl-amino)-3-(2,4-dichloro-phenyl)-1-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-propan-1-one 323099 (R)-3-(2,4-Dichloro-phenyl)-2-[(thiazol-2-ylmethyl)-amino]-1-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-propan-1-one 323100 (R)-2-Benzylamino-3-(2,4-dichloro-phenyl)-1-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-propan-1-one 323104 N-[(R)-1-(2,4-Dichloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-methanesulfonamide 323117 5-Isopropyl-4-(3-methoxycarbamoyl-4-methyl-phenylamino)-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid ethyl ester 323118 [4-(2,4-Difluoro-5-methoxycarbamoyl-phenylamino)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazin-6-yl]-carbamic acid 1-methyl-piperidin-4-yl ester 323122 4-(2,4-Difluoro-5-methoxycarbamoyl-phenylamino)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid ethyl ester 323123 2,4-Difluoro-5-(5-isopropyl-6-[1,3,4]oxadiazol-2-yl-pyrrolo[2,1-f][1,2,4]triazin-4-ylamino)-N-methoxy-benzamide 323142 7-(2,4-Dichloro-5-methoxy-phenylamino)-2-[5-(4-methyl-piperazin-1-ylmethyl)-thiophen-3-yl]-thieno[3,2-b]pyridine-6-carbonitrile 323144 [4-(2,4-Difluoro-5-methoxycarbamoyl-phenylamino)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazin-6-yl]-carbamic acid 3-methanesulfonyl-propyl ester 323146 5-[6-(5-Dimethylamino-[1,3,4]oxadiazol-2-yl)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazin-4-ylamino]-2,4-difluoro-N-methoxy-benzamide 323147 N-[1-(2,6-Dimethyl-benzyl)-4-methoxy-1H-indol-2-ylmethyl]-propionamide 323173 7-(2,4-Dichloro-5-methoxy-phenylamino)-2-[4-(4-methyl-piperazin-1-ylmethyl)-phenyl]-thieno[3,2-b]pyridine-6-carbonitrile 323178 5-[6-(5-Difluoromethyl-[1,3,4]oxadiazol-2-yl)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazin-4-ylamino]-2,4-difluoro-N-methoxy-benzamide 323182 N-[1-(4-Chloro-benzoyl)-4-methoxy-1H-indol-2-ylmethyl]-propionamide 323209 4-(5-Cyclopropylmethoxycarbamoyl-2,4-difluoro-phenylamino)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid ethyl ester 323262 (2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 9-acetoxy-6a,10b-dimethyl-4,10-dioxo-2-(tetrahydrofuran-3-yl)-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 323263 N-[4-(3-Aza-bicyclo[3.1.0]hex-3-yl)-but-2-ynyl]-2,2-bis-(4-fluoro-phenyl)-2-hydroxy-acetamide 323268 (3S,4aR,4bS,6S,8R,8aR)-6-Acetoxy-3-furan-3-yl-4a,8a-dimethyl-5-oxo-4,4a,4b,5,6,7,8,8a,9,10-decahydro-3H-2-oxa-phenanthrene-8-carboxylic acid methyl ester 323279 (R)-3-amino-N-(3-(2,4-dichlorophenyl)-1-oxo-1-(4-(2-((2-(thiophen-2-yl)ethylamino)methyl)phenyl)piperazin-1-yl)propan-2-yl)propanamide 323280 [(R)-1-(2,4-Dichloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-carbamic acid benzyl ester 323281 [(R)-1-Naphthalen-1-ylmethyl-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-carbamic acid benzyl ester 323282 [(R)-1-(4-Hydroxy-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-carbamic acid benzyl ester 323304 N-[(R)-1-(2,4-Dichloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-succinamic acid methyl ester 323305 [(R)-1-(2,4-Dichloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-carbamic acid methyl ester 323376 N-{4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-2-hydroxy-benzamide 323377 N-[4-(3-Aza-bicyclo[3.1.0]hex-3-yl)-but-2-ynyl]-2-cyclohexyl-2-hydroxy-2-phenyl-acetamide 323400 1-Cyclopropyl-3-[(R)-1-(2,4-dichloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-urea 323401 1-[(R)-1-(2,4-Dichloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-3-isopropyl-urea 323402 1-tert-Butyl-3-[(R)-1-(2,4-dichloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-urea 323403 1-[(R)-1-(2,4-Dichloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-3-(2-fluoro-benzyl)-urea 323404 1-[(R)-1-(2,4-Dichloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-3-(2-hydroxy-ethyl)-urea 323405 1-Cyclopentyl-3-[(R)-1-(2,4-dichloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-urea 323418 [(R)-1-(1H-Indol-3-ylmethyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-carbamic acid benzyl ester 323419 [(R)-1-Benzo[b]thiophen-3-ylmethyl-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-carbamic acid benzyl ester 323421 Salvinorin A (ester) 323429 (3S,4aS,4bR,6S,8R,8aR,10aR)-6-Acetoxy-3-furan-3-yl-4a,8a-dimethyl-5-oxo-dodecahydro-2-oxa-phenanthrene-8-carboxylic acid methyl ester 323433 N*1*,N*1*-Diethyl-N*4*-(2-naphthalen-2-yl-quinazolin-4-yl)-pentane-1,4-diamine 323434 N*4*-(2-Benzyl-quinazolin-4-yl)-N*1*,N*1*-diethyl-pentane-1,4-diamine 323439 N*1*,N*1*-Diethyl-N*4*-(2-phenoxymethyl-quinazolin-4-yl)-pentane-1,4-diamine 323442 (R)-2-Amino-3-(2,4-dichloro-phenyl)-1-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-propan-1-one 323446 N-{(E)-4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-3-nitro-benzamide 323520 [(R)-1-(2,4-Dichloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-carbamic acid isopropyl ester 323521 1-[(R)-1-(2,4-Dichloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-3-ethyl-urea 323523 (-)-1-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-yl)ethyl]-4-[4-(2-methoxy-1-naphthyl)butyl]piperazine 323537 2-Amino-N-{(E)-4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-benzamide 323557 N*4*-[2-(3,5-Dichloro-phenoxymethyl)-pyrimidin-4-yl]-N*1*,N*1*-diethyl-pentane-1,4-diamine 323569 3-Amino-N-{(E)-4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-benzamide 323572 N-[4-(3-Aza-bicyclo[3.1.0]hex-3-yl)-but-2-ynyl]-2-hydroxy-2,2-diphenyl-acetamide 323576 (3S,4aS,4bR,6S,8R,8aR,10aR)-6-Acetoxy-3-furan-3-yl-1-hydroxy-4a,8a-dimethyl-5-oxo-dodecahydro-2-oxa-phenanthrene-8-carboxylic acid methyl ester 323578 (2S,4aR,6aS,7R,9S,10aS,10bR)-2-(furan-3-yl)-7-(hydroxymethyl)-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-benzo[f]isochromen-9-yl acetate 323609 N*1*,N*1*-Diethyl-N*4*-(2-phenethyl-quinazolin-4-yl)-pentane-1,4-diamine 323614 [(R)-1-(1H-Imidazol-4-ylmethyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-carbamic acid benzyl ester 323651 N-{(E)-4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-2-nitro-benzamide 323673 N*4*-[2-(3-Chloro-phenoxymethyl)-pyrimidin-4-yl]-N*1*,N*1*-diethyl-pentane-1,4-diamine 323681 (3S,4aR,4bS,6S,8R,8aR,10aR)-6-Formyloxy-3-furan-3-yl-4a,8a-dimethyl-1,5-dioxo-dodecahydro-2-oxa-phenanthrene-8-carboxylic acid methyl ester 323686 (3S,4aR,4bR,5R,6S,8aR,10aR)-5,6-Diacetoxy-3-furan-3-yl-4a,8a-dimethyl-1-oxo-3,4,4a,4b,5,6,8a,9,10,10a-decahydro-1H-2-oxa-phenanthrene-8-carboxylic acid methyl ester 323697 [(R)-1-(2,4-Dichloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-carbamic acid ethyl ester 323698 [(R)-1-(2,4-Dichloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-carbamic acid 2-fluoro-ethyl ester 323702 3-[(R)-1-(2,4-Dichloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-1,1-dimethyl-urea 323703 Pyrrolidine-1-carboxylic acid [(R)-1-(2,4-dichloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-amide 323710 1-(1,2-Dihydro-pyridin-2-yl)-3-{(1R,2S)-2-[(S)-3-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-urea 323711 Naltrindole analogue 323713 1-((1R,2S)-2-(((S)-3-(4-fluorobenzyl)piperidin-1-yl)methyl)cyclohexyl)-3-(3-(1-methyl-1H-tetrazol-5-yl)phenyl)urea 323717 Dimethyl-{4-[1-(4-phenyl-piperazin-1-yl)-2-(2-p-tolyl-ethylamino)-ethyl]-phenyl}-amine 323718 N-[2-(4-tert-Butyl-phenyl)-2-(4-phenyl-piperazin-1-yl)-ethyl]-2-phenyl-acetamide 323720 N'-[4-(2,4-Dichloro-benzyloxy)-pyrimidin-2-yl]-N,N-diethyl-butane-1,4-diamine 323723 1-[2-Biphenyl-4-yl-2-(4-cyclohexyl-piperazin-1-yl)-ethyl]-3-(3,5-dimethyl-phenyl)-urea 323724 [2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethyl]-[2-(4-fluoro-phenyl)-ethyl]-amine 323726 [5-(2''-Chloro-biphenyl-3-yl)-oxazol-2-yl]-(5-ethanesulfonyl-2-methoxy-phenyl)-amine 323727 1-(3,5-Dichloro-phenyl)-3-[2-(4-dimethylamino-phenyl)-2-(4-methyl-piperazin-1-yl)-ethyl]-urea 323730 [2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-methoxy-phenyl)-ethyl]-[2-(3,5-dimethyl-phenyl)-ethyl]-amine 323732 [5-(4-Chloro-phenyl)-oxazol-2-yl]-(5-ethanesulfonyl-2-methoxy-phenyl)-amine 323733 1-[2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethyl]-3-p-tolyl-urea 323734 1-(4-tert-Butyl-phenyl)-3-[2-(4-tert-butyl-phenyl)-2-(4-cyclohexyl-piperazin-1-yl)-ethyl]-urea 323743 Cyclopropyl-[4-(1-isopropyl-piperidin-4-yloxy)-benzyl]-amine 323744 Naltrindole analogue 323745 Naltrindole analogue 323746 Biphenyl-4-carboxylic acid (1-acetyl-2,2,4-trimethyl-4-phenyl-1,2,3,4-tetrahydro-quinolin-6-yl)-amide 323754 4-[1-(2-Hydroxy-1-methyl-ethyl)-piperidin-4-yloxy]-benzonitrile 323758 [2-(4-Methyl-piperazin-1-yl)-2-phenyl-ethyl]-(2-p-tolyl-ethyl)-amine 323764 1-[2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-methoxy-phenyl)-ethyl]-3-(4-trifluoromethyl-phenyl)-urea 323765 N-[2-(4-tert-Butyl-phenyl)-2-(4-phenyl-piperazin-1-yl)-ethyl]-2-(2-methoxy-phenyl)-acetamide 323770 1-(4-Chloro-phenyl)-3-[2-(4-cyclohexyl-piperazin-1-yl)-4-methyl-pentyl]-urea 323771 1-[2-(4-tert-Butyl-phenyl)-2-(4-cyclohexyl-piperazin-1-yl)-ethyl]-3-(4-trifluoromethyl-phenyl)-urea 323772 (5-Ethanesulfonyl-2-methoxy-phenyl)-[5-(4-fluoro-phenyl)-oxazol-2-yl]-amine 323775 [2-(4-tert-Butyl-phenyl)-2-(4-cyclohexyl-piperazin-1-yl)-ethyl]-[2-(2-methoxy-phenyl)-ethyl]-amine 323776 1-[2-(4-Cyclohexyl-piperazin-1-yl)-2-phenyl-ethyl]-3-(4-methoxy-phenyl)-urea 323777 [4-(1-Isopropyl-piperidin-4-yloxy)-benzyl]-phenyl-amine 323779 Naltrindole analogue 323783 4-(1-sec-Butyl-piperidin-4-yloxy)-benzonitrile 323788 (5-Ethanesulfonyl-2-methoxy-phenyl)-[5-(3-thiophen-2-yl-phenyl)-oxazol-2-yl]-amine 323792 1-[2-(4-Cyclohexyl-piperazin-1-yl)-4-methyl-pentyl]-3-(3,5-dichloro-phenyl)-urea 323793 [2-(4-tert-Butyl-phenyl)-2-(4-phenyl-piperazin-1-yl)-ethyl]-[2-(4-methoxy-phenyl)-ethyl]-amine 323795 1-[2-(4-Cyclohexyl-piperazin-1-yl)-2-phenyl-ethyl]-3-(3,5-dichloro-phenyl)-urea 323802 1-[2-(4-tert-Butyl-phenyl)-2-(4-cyclohexyl-piperazin-1-yl)-ethyl]-3-(4-dimethylamino-phenyl)-urea 323808 1-{(1R,2S)-2-[(S)-3-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-(4-[1,2,4]triazol-1-yl-phenyl)-urea 323814 Naltrindole analogue 323818 [2-(4-Fluoro-phenyl)-ethyl]-[2-(4-phenyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethyl]-amine 323819 2-(2-Methoxy-phenyl)-N-[2-(2-methoxy-phenyl)-2-(4-phenyl-piperazin-1-yl)-ethyl]-acetamide 323820 (5-Ethanesulfonyl-2-methoxy-phenyl)-{5-[3-(3-methyl-3H-imidazol-4-yl)-phenyl]-oxazol-2-yl}-amine 323823 N*4*-[2-(2,4-Dichloro-benzyloxy)-pyrimidin-4-yl]-N*1*,N*1*-diethyl-pentane-1,4-diamine 323828 (3-Ethanesulfonyl-phenyl)-(5-phenyl-oxazol-2-yl)-amine 323829 (5-Phenyl-oxazol-2-yl)-m-tolyl-amine 323830 N-[2-(4-Dimethylamino-phenyl)-2-(4-phenyl-piperazin-1-yl)-ethyl]-2-(4-trifluoromethyl-phenyl)-acetamide 323831 1-[2-(4-Cyclohexyl-piperazin-1-yl)-2-(2-methoxy-phenyl)-ethyl]-3-(4-fluoro-phenyl)-urea 323837 2-[4-(4-Chloro-phenylsulfanyl)-phenyl]-1H-benzoimidazole-5-carboxylic acid amide 323845 Naltrindole analogue 323846 Naltrindole analogue 323847 2-Dibenzofuran-2-yl-1H-benzoimidazole-5-carboxylic acid amide 323852 Naltrindole analogue 323856 Dimethyl-(4-{2-[2-(4-phenyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethylamino]-ethyl}-phenyl)-amine 323858 N*4*-[4-(2,4-Dichloro-benzyloxy)-pyrimidin-2-yl]-N*1*,N*1*-diethyl-pentane-1,4-diamine 323863 [2-(4-tert-Butyl-phenyl)-2-(4-cyclohexyl-piperazin-1-yl)-ethyl]-[2-(4-tert-butyl-phenyl)-ethyl]-amine 323864 1-(4-tert-Butyl-phenyl)-3-[2-(4-cyclohexyl-piperazin-1-yl)-2-(4-methoxy-phenyl)-ethyl]-urea 323869 [2-(4-Cyclohexyl-piperazin-1-yl)-2-phenyl-ethyl]-[2-(3,5-dichloro-phenyl)-ethyl]-amine 323870 1-[2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethyl]-3-phenyl-urea 323876 Naltrindole analogue 323877 (11-Fluoro-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-dimethyl-amine 323878 (11-Chloro-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-dimethyl-amine 323879 1-[4-(1-Isopropyl-piperidin-4-yloxy)-benzyl]-4-phenyl-piperazine 323880 Naltrindole analogue 323881 [3-((R)-4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-acetic acid 323885 2-[4-(4-Nitro-phenoxy)-phenyl]-1H-benzoimidazole-5-carboxylic acid amide 323886 3-[4-(5-Carbamoyl-1H-benzoimidazol-2-yl)-phenoxy]-benzoic acid 323888 1-deoxosalvinorin 323889 1-{2-[4-(3,4-Dichloro-phenyl)-piperazin-1-yl]-4-methyl-pentyl}-3-p-tolyl-urea 323890 [2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethyl]-(2-p-tolyl-ethyl)-amine 323892 (5-Ethanesulfonyl-2-methoxy-phenyl)-[5-(3-pyridin-2-yl-phenyl)-oxazol-2-yl]-amine 323897 5-(2-Chloro-6-cyclopentylamino-purin-9-yl)-tetrahydro-furan-2,3,4-triol 323899 Dimethyl-(4-{1-(4-phenyl-piperazin-1-yl)-2-[2-(4-trifluoromethyl-phenyl)-ethylamino]-ethyl}-phenyl)-amine 323900 [2-(4-Fluoro-phenyl)-ethyl]-[2-(4-methoxy-phenyl)-2-(4-methyl-piperazin-1-yl)-ethyl]-amine 323906 1-[2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-methoxy-phenyl)-ethyl]-3-(4-fluoro-phenyl)-urea 323907 1-[2-(4-tert-Butyl-phenyl)-2-(4-cyclohexyl-piperazin-1-yl)-ethyl]-3-(4-methoxy-phenyl)-urea 323909 (5-Ethanesulfonyl-2-methoxy-phenyl)-[5-(3-ethyl-phenyl)-oxazol-2-yl]-amine 323910 Naltrindole analogue 323912 Naltrindole analogue 323916 1-{(1R,2S)-2-[(S)-3-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-[2-(1-methyl-1H-tetrazol-5-yl)-phenyl]-urea 323917 Naltrindole analogue 323920 (4-{2-[2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethylamino]-ethyl}-phenyl)-dimethyl-amine 323921 1-[2-(2-Methoxy-phenyl)-2-(4-phenyl-piperazin-1-yl)-ethyl]-3-p-tolyl-urea 323926 1-[2-Biphenyl-4-yl-2-(4-cyclohexyl-piperazin-1-yl)-ethyl]-3-p-tolyl-urea 323930 N'-[4-(2,4-Dichloro-benzyloxy)-pyrimidin-2-yl]-N,N-dimethyl-pentane-1,5-diamine 323931 1-[2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-methoxy-phenyl)-ethyl]-3-p-tolyl-urea 323936 (5-Ethanesulfonyl-2-methoxy-phenyl)-[5-(4-methoxy-phenyl)-oxazol-2-yl]-amine 323937 N-[2-(4-Cyclohexyl-piperazin-1-yl)-2-phenyl-ethyl]-2-(3,5-dichloro-phenyl)-acetamide 323938 1-[2-Phenyl-2-(4-phenyl-piperazin-1-yl)-ethyl]-3-p-tolyl-urea 323939 1-{3-[2-(5-Ethanesulfonyl-2-methoxy-phenylamino)-oxazol-5-yl]-phenyl}-ethanone 323943 Naltrindole analogue 323944 Naltrindole analogue 323951 Naltrindole analogue 323954 [2-(4-Cyclohexyl-piperazin-1-yl)-2-(2-methoxy-phenyl)-ethyl]-[2-(3,5-dichloro-phenyl)-ethyl]-amine 323961 [2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethyl]-[2-(4-trifluoromethyl-phenyl)-ethyl]-amine 323962 1-[2-(4-Cyclohexyl-piperazin-1-yl)-2-phenyl-ethyl]-3-(4-trifluoromethyl-phenyl)-urea 323963 2-(5-Phenyl-oxazol-2-ylamino)-benzonitrile 323964 (5-Ethanesulfonyl-2-methoxy-phenyl)-[5-(2''-fluoro-biphenyl-3-yl)-oxazol-2-yl]-amine 323965 N'-[4-(2,4-Dichloro-benzyloxy)-pyrimidin-2-yl]-N,N-diethyl-propane-1,3-diamine 323967 [2-(4-Methoxy-phenyl)-ethyl]-[2-(4-phenyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethyl]-amine 323968 [2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-methoxy-phenyl)-ethyl]-[2-(4-trifluoromethyl-phenyl)-ethyl]-amine 323972 [2-(4-Methyl-piperazin-1-yl)-2-phenyl-ethyl]-[2-(4-trifluoromethyl-phenyl)-ethyl]-amine 323985 (11-Bromo-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-dimethyl-amine 323986 {[(2S,4S)-17-fluoro-3-oxa-13-thiatetracyclo[12.4.0.0^{2,6}.0^{7,12}]octadeca-1(14),7(12),8,10,15,17-hexaen-4-yl]methyl}dimethylamine 323987 4-(1-Propyl-piperidin-4-yloxy)-benzonitrile 323988 4-(1-Isopropyl-piperidin-4-yloxy)-benzonitrile 323989 N-[4-(1-Isopropyl-piperidin-4-yloxy)-benzyl]-N,N'',N''-trimethyl-ethane-1,2-diamine 323990 1-{(1R,2S)-2-[(S)-3-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-(2-fluoro-phenyl)-urea 323994 1-[2-(4-Methyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethyl]-3-p-tolyl-urea 323996 [2-(4-tert-Butyl-phenyl)-2-(4-cyclohexyl-piperazin-1-yl)-ethyl]-[2-(4-trifluoromethyl-phenyl)-ethyl]-amine 323997 [2-(4-tert-Butyl-phenyl)-ethyl]-[2-(4-cyclohexyl-piperazin-1-yl)-2-(4-methoxy-phenyl)-ethyl]-amine 324000 1-[2-(4-Dimethylamino-phenyl)-2-(4-methyl-piperazin-1-yl)-ethyl]-3-(4-fluoro-phenyl)-urea 324001 1-[2-(4-tert-Butyl-phenyl)-2-(4-cyclohexyl-piperazin-1-yl)-ethyl]-3-(4-fluoro-phenyl)-urea 324011 N-[2-Phenyl-2-(4-phenyl-piperazin-1-yl)-ethyl]-2-p-tolyl-acetamide 324012 N*1*,N*1*-Diethyl-N*4*-(2-styryl-quinazolin-4-yl)-pentane-1,4-diamine 324018 1-(3-Cyano-4-pyrazol-1-yl-cyclohexa-2,4-dienyl)-3-{(1R,2S)-2-[(S)-3-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-urea 324019 Naltrindole analogue 324020 Naltrindole analogue 324023 1-{(1R,2S)-2-[(S)-3-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-[4-(1-methyl-1H-tetrazol-5-yl)-phenyl]-urea 324026 1-[2-(4-tert-Butyl-phenyl)-2-(4-cyclohexyl-piperazin-1-yl)-ethyl]-3-phenyl-urea 324027 [2-(4-Methyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethyl]-phenethyl-amine 324028 (5-Ethanesulfonyl-2-methoxy-phenyl)-[5-(3-pyridin-4-yl-phenyl)-oxazol-2-yl]-amine 324035 (3-Phenoxy-phenyl)-(5-phenyl-oxazol-2-yl)-amine 324036 1-(3,5-Dichloro-phenyl)-3-[2-(4-methyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethyl]-urea 324043 [2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethyl]-[2-(3,5-dichloro-phenyl)-ethyl]-amine 324044 [2-Biphenyl-4-yl-2-(4-cyclohexyl-piperazin-1-yl)-ethyl]-[2-(3,5-dimethyl-phenyl)-ethyl]-amine 324048 Naltrindole analogue 324060 1-[2-(4-Cyclohexyl-piperazin-1-yl)-2-phenyl-ethyl]-3-p-tolyl-urea 324061 [2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethyl]-phenethyl-amine 324068 3,4-Dihydroxy-5-[6-(3-iodo-benzylamino)-purin-9-yl]-4-methyl-tetrahydro-furan-2-carboxylic acid methylamide 324069 N'-[4-(2,4-Dichloro-benzyloxy)-pyrimidin-2-yl]-N,N-diethyl-ethane-1,2-diamine 324070 [2-(4-tert-Butyl-phenyl)-2-(4-cyclohexyl-piperazin-1-yl)-ethyl]-[2-(4-methoxy-phenyl)-ethyl]-amine 324071 1-[2-(4-Cyclohexyl-piperazin-1-yl)-2-(2-methoxy-phenyl)-ethyl]-3-(3,5-dichloro-phenyl)-urea 324072 [3-(5-Phenyl-oxazol-2-ylamino)-phenyl]-methanol 324078 [2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-methoxy-phenyl)-ethyl]-[2-(3,5-dichloro-phenyl)-ethyl]-amine 324083 1-(2-Methoxy-phenyl)-3-[2-(4-methyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethyl]-urea 324090 4-(1-Methyl-piperidin-4-yloxy)-benzonitrile 324091 3-{(R)-3-[(4-Fluoro-benzenesulfonyl)-methyl-amino]-1,2,3,4-tetrahydro-carbazol-9-yl}-propionic acid 324093 (-)-{[(2S,4R)-17-fluoro-3-oxa-13-thiatetracyclo[12.4.0.0^{2,6}.0^{7,12}]octadeca-1(14),7(12),8,10,15,17-hexaen-4-yl]methyl}dimethylamine 324094 4-(1-Isobutyl-piperidin-4-yloxy)-benzonitrile 324095 4-(1-Cyclopentyl-piperidin-4-yloxy)-benzonitrile 324102 (5-Ethanesulfonyl-2-methoxy-phenyl)-[5-(3-thiophen-3-yl-phenyl)-oxazol-2-yl]-amine 324105 5-Hydroxymethyl-2-[6-(3-iodo-benzylamino)-purin-9-yl]-3-methyl-tetrahydro-furan-3,4-diol 324112 [2-(2-Methoxy-phenyl)-ethyl]-[2-(2-methoxy-phenyl)-2-(4-phenyl-piperazin-1-yl)-ethyl]-amine 324113 1-[2-(4-Cyclohexyl-piperazin-1-yl)-2-(2-methoxy-phenyl)-ethyl]-3-(4-methoxy-phenyl)-urea 324118 [2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethyl]-[2-(4-methoxy-phenyl)-ethyl]-amine 324119 1-[2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-dimethylamino-phenyl)-ethyl]-3-(3,5-dichloro-phenyl)-urea 324120 4-[2-(5-Ethanesulfonyl-2-methoxy-phenylamino)-oxazol-5-yl]-benzonitrile 324121 4-[2-(5-Ethanesulfonyl-2-methoxy-phenylamino)-oxazol-5-yl]-benzamide 324122 (4-{2-[2-(4-tert-Butyl-phenyl)-2-(4-cyclohexyl-piperazin-1-yl)-ethylamino]-ethyl}-phenyl)-dimethyl-amine 324123 [4-(1-Isopropyl-piperidin-4-yloxy)-benzyl]-pyridin-2-yl-amine 324124 1-[4-(1-Isopropyl-piperidin-4-yloxy)-benzyl]-4-methyl-piperazine 324127 1-{(1R,2S)-2-[(S)-3-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-[3-(5-methyl-tetrazol-1-yl)-phenyl]-urea 324128 Naltrindole analogue 324136 1-{2-[4-(3,4-Dichloro-phenyl)-piperazin-1-yl]-4-methyl-pentyl}-3-(3,5-dimethyl-phenyl)-urea 324138 [2-(4-Cyclohexyl-piperazin-1-yl)-2-phenyl-ethyl]-[2-(4-trifluoromethyl-phenyl)-ethyl]-amine 324143 4-(5-Phenyl-oxazol-2-ylamino)-benzenesulfonamide 324146 Dimethyl-(4-{2-[2-phenyl-2-(4-phenyl-piperazin-1-yl)-ethylamino]-ethyl}-phenyl)-amine 324147 N-[2-(4-Methoxy-phenyl)-2-(4-phenyl-piperazin-1-yl)-ethyl]-2-phenyl-acetamide 324150 N-[2-(4-tert-Butyl-phenyl)-2-(4-cyclohexyl-piperazin-1-yl)-ethyl]-2-(4-trifluoromethyl-phenyl)-acetamide 324152 N-(5-Benzyloxy-pentyl)-N-[2-(3-tert-butyl-ureido)-3-(3,5-dimethoxy-phenyl)-[1,6]naphthyridin-7-yl]-acetamide 324153 (11-Fluoro-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-dimethyl-amine 324154 Naltrindole analogue 324160 Naltrindole analogue 324167 1-[2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethyl]-3-(4-trifluoromethyl-phenyl)-urea 324168 1-[2-(4-Cyclohexyl-piperazin-1-yl)-2-phenyl-ethyl]-3-(4-fluoro-phenyl)-urea 324169 (5-Biphenyl-3-yl-oxazol-2-yl)-(5-ethanesulfonyl-2-methoxy-phenyl)-amine 324175 [2-(4-tert-Butyl-phenyl)-2-(4-cyclohexyl-piperazin-1-yl)-ethyl]-phenethyl-amine 324178 1-(4-Fluoro-phenyl)-3-[2-phenyl-2-(4-phenyl-piperazin-1-yl)-ethyl]-urea 324186 Naltrindole analogue 324188 4-(1-Ethyl-piperidin-4-yloxy)-benzonitrile 324189 1-Benzyl-4-[4-(1-isopropyl-piperidin-4-yloxy)-benzyl]-piperazine 324190 Naltrindole analogue 324191 Naltrindole analogue 324199 [2-(4-tert-Butyl-phenyl)-2-(4-cyclohexyl-piperazin-1-yl)-ethyl]-[2-(3,5-dichloro-phenyl)-ethyl]-amine 324200 [2-(4-Methoxy-phenyl)-2-(4-phenyl-piperazin-1-yl)-ethyl]-(2-p-tolyl-ethyl)-amine 324202 (5-Ethanesulfonyl-2-methoxy-phenyl)-[5-(3-pyridin-3-yl-phenyl)-oxazol-2-yl]-amine 324203 [2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-methoxy-phenyl)-ethyl]-phenethyl-amine 324214 [2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-methoxy-phenyl)-ethyl]-(2-p-tolyl-ethyl)-amine 324215 1-[2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethyl]-3-(4-methoxy-phenyl)-urea 324228 Naltrindole analogue 324231 (11-Chloro-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-dimethyl-amine 324232 (11-Bromo-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-dimethyl-amine 324233 1-[4-(1-Isopropyl-piperidin-4-yloxy)-benzyl]-4-methyl-[1,4]diazepane 324235 1-{(1R,2S)-2-[(S)-3-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-(4-methoxy-phenyl)-urea 324237 2-[4-(3-Diethylcarbamoyl-phenoxy)-phenyl]-1H-benzoimidazole-5-carboxylic acid amide 324238 Naltrindole analogue 324241 1-[2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethyl]-3-(4-fluoro-phenyl)-urea 324242 1-[2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethyl]-3-(2-methoxy-phenyl)-urea 324243 N*4*-(2,4-Dichloro-benzyl)-N*2*-(4-diethylamino-1-methyl-butyl)-pyrimidine-2,4-diamine 324250 1-[3,5-Bis-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3-{(1R,2S)-2-[(S)-3-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-urea 324252 1-(4-Methoxy-phenyl)-3-[2-(4-phenyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethyl]-urea 324253 [2-(4-Methyl-piperazin-1-yl)-2-phenyl-ethyl]-phenethyl-amine 324259 [2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethyl]-[2-(2-methoxy-phenyl)-ethyl]-amine 324260 [2-(4-tert-Butyl-phenyl)-2-(4-phenyl-piperazin-1-yl)-ethyl]-[2-(2-methoxy-phenyl)-ethyl]-amine 324274 1-{(1R,2S)-2-[(S)-3-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-(4-methyl-thiazol-2-yl)-urea 324275 1-(3-Acetyl-4-fluoro-phenyl)-3-{(1R,2S)-2-[(S)-3-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-urea 324287 N*2*-(3H-Benzoimidazol-5-yl)-5-bromo-N*4*-(2,3-dichloro-benzyl)-pyrimidine-2,4-diamine 324290 (S)-4-Benzoyl-1-[5-guanidino-2-((S)-2-naphthalen-2-yl-acetylamino)-pentanoyl]-piperazine-2-carboxylic acid benzylamide 324300 N*2*-(3H-Benzoimidazol-5-yl)-5-bromo-N*4*-(1,2,3,4-tetrahydro-naphthalen-1-yl)-pyrimidine-2,4-diamine 324301 (3H-Benzoimidazol-5-yl)-(4-ethoxy-5-trifluoromethyl-pyrimidin-2-yl)-amine 324302 N*2*-(3H-Benzoimidazol-5-yl)-5-bromo-N*4*-(4-fluoro-phenyl)-pyrimidine-2,4-diamine 324303 (2S,4R)-4-Benzyl-1-{(S)-2-[2-(3,4-dichloro-phenyl)-acetylamino]-5-guanidino-pentanoyl}-pyrrolidine-2-carboxylic acid benzylamide 324304 (3H-Benzoimidazol-5-yl)-(4-cyclohexyloxy-5-trifluoromethyl-pyrimidin-2-yl)-amine 324310 Naltrindole analogue 324313 Butyl-[4-(1-isopropyl-piperidin-4-yloxy)-benzyl]-methyl-amine 324314 1-Isopropyl-4-(4-pyrrolidin-1-ylmethyl-phenoxy)-piperidine 324323 1-{(1R,2S)-2-[(S)-3-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-(5-fluoro-2-methyl-phenyl)-urea 324324 1-(4-Chloro-benzothiazol-2-yl)-3-{(1R,2S)-2-[(S)-3-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-urea 324325 2-[4-(3,4-Dichloro-phenylsulfamoyl)-phenyl]-1H-benzoimidazole-5-carboxylic acid amide 324336 4-Bromo-N-[4-(4-dimethylamino-quinazolin-2-ylamino)-cyclohexyl]-2-trifluoromethoxy-benzenesulfonamide 324352 (2S,4R)-4-Benzyl-1-[(S)-5-guanidino-2-(2-naphthalen-1-yl-acetylamino)-pentanoyl]-pyrrolidine-2-carboxylic acid benzylamide 324357 1-{(1R,2S)-2-[(S)-3-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-(3-fluoro-phenyl)-urea 324360 2-(4-Phenylcarbamoyl-phenyl)-1H-benzoimidazole-5-carboxylic acid amide 324362 1-{(1R,2S)-2-[3-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-(1H-indol-5-yl)-urea 324370 Naltrindole analogue 324371 Naltrindole analogue 324372 2-[4-(4-Chloro-benzenesulfinyl)-phenyl]-1H-benzoimidazole-5-carboxylic acid amide 324373 2-[4-(4-Chloro-benzenesulfonyl)-phenyl]-1H-benzoimidazole-5-carboxylic acid amide 324376 N*4*-(3H-Benzoimidazol-5-yl)-N*2*-(3-chloro-phenyl)-5-trifluoromethyl-pyrimidine-2,4-diamine 324377 (2S,4R)-4-Benzyl-1-{(S)-2-[(biphenyl-2-carbonyl)-amino]-5-guanidino-pentanoyl}-pyrrolidine-2-carboxylic acid benzylamide 324380 N6-Methyladenosine 324393 1-(4-Bromo-phenyl)-3-{(1R,2S)-2-[(S)-3-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-urea 324395 2-Biphenyl-4-yl-1H-benzoimidazole-5-carboxylic acid amide 324398 4-(4-(1-isopropylpiperidin-4-yloxy)benzyl)morpholine 324399 1-[4-(1-Isopropyl-piperidin-4-yloxy)-benzyl]-piperidin-4-ol 324414 (3H-Benzoimidazol-5-yl)-(4-o-tolylsulfanyl-5-trifluoromethyl-pyrimidin-2-yl)-amine 324416 (2S,4R)-4-Benzyl-1-{(S)-2-[2-(4-chloro-phenyl)-acetylamino]-5-guanidino-pentanoyl}-pyrrolidine-2-carboxylic acid benzylamide 324417 Octane-1-sulfonic acid {4-[(4-dimethylamino-quinazolin-2-ylamino)-methyl]-cyclohexylmethyl}-amide 324420 N*4*-(3H-Benzoimidazol-5-yl)-5-trifluoromethyl-N*2*-(4-trifluoromethyl-phenyl)-pyrimidine-2,4-diamine 324421 (S)-4-Benzyl-1-[5-guanidino-2-((S)-2-naphthalen-2-yl-acetylamino)-pentanoyl]-piperazine-2-carboxylic acid benzylamide 324425 N-Dibenzofuran-2-yl-2-[4-(8-methoxy-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide 324438 4-(1-Cyclohexyl-piperidin-4-yloxy)-benzonitrile 324439 4-(1-Benzyl-piperidin-4-yloxy)-benzonitrile 324444 1-{(1R,2S)-2-[(S)-3-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-(5-methyl-isoxazol-3-yl)-urea 324445 1-(3-Acetyl-phenyl)-3-{(1R,2S)-2-[(R)-3-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-urea 324450 (2S,4R)-4-Benzyl-1-[(S)-5-guanidino-2-(2-1H-indol-3-yl-acetylamino)-pentanoyl]-pyrrolidine-2-carboxylic acid phenylamide 324455 (3H-Benzoimidazol-5-yl)-[4-(3-methoxy-phenoxy)-5-trifluoromethyl-pyrimidin-2-yl]-amine 324460 4-Bromo-N-[4-(quinazolin-2-ylaminomethyl)-cyclohexyl]-2-trifluoromethoxy-benzenesulfonamide 324463 (2R,3R,4S,5R)-2-(6-(3-chlorobenzylamino)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 324464 N*4*-Benzo[1,3]dioxol-5-yl-N*2*-(3H-benzoimidazol-5-yl)-5-bromo-pyrimidine-2,4-diamine 324470 17-cyclopropylmethyl-10-hydroxy-3-methoxy-13-oxo-(1R,9R,10S)-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-triene-4-carboxamide 324478 Naltrindole analogue 324481 N*4*-[4-(3H-Benzoimidazol-5-ylamino)-5-trifluoromethyl-pyrimidin-2-yl]-benzene-1,2,4-triamine derivative 324485 N*4*-(3H-Benzoimidazol-5-yl)-5-bromo-N*2*-(3-chloro-phenyl)-pyrimidine-2,4-diamine 324486 (3H-Benzoimidazol-5-yl)-[4-(4-chloro-phenoxy)-5-trifluoromethyl-pyrimidin-2-yl]-amine 324495 (2S,4R)-4-Benzyl-1-[(S)-5-guanidino-2-(2-1H-indol-3-yl-acetylamino)-pentanoyl]-pyrrolidine-2-carboxylic acid phenethyl-amide 324496 N*2*,N*4*-Bis-(1H-benzoimidazol-5-yl)-5-bromo-pyrimidine-2,4-diamine 324497 (2S,4R)-4-Benzyl-1-[(S)-5-guanidino-2-(3-phenyl-propionylamino)-pentanoyl]-pyrrolidine-2-carboxylic acid benzylamide 324511 1-{(1R,2S)-2-[(S)-3-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-thiazol-2-yl-urea 324512 Naltrindole analogue 324513 Naltrindole analogue 324514 N*2*-(3H-Benzoimidazol-5-yl)-5-bromo-N*4*-[4-(pyridin-3-yloxy)-phenyl]-pyrimidine-2,4-diamine 324523 4-Bromo-N-[4-(4-dimethylamino-quinazolin-2-ylamino)-cyclohexylmethyl]-2-trifluoromethoxy-benzenesulfonamide 324526 N2-(1H-benzo[d]imidazol-6-yl)-N4-(2-chlorophenyl)-5-(trifluoromethyl)pyrimidine-2,4-diamine 324527 N*2*-(3H-Benzoimidazol-5-yl)-5-bromo-N*4*-indan-1-yl-pyrimidine-2,4-diamine 324529 (2S,4R)-4-Benzyl-1-[(S)-5-guanidino-2-(2-naphthalen-2-yl-acetylamino)-pentanoyl]-pyrrolidine-2-carboxylic acid benzylamide 324535 4-Bromo-N-[4-(quinazolin-2-ylamino)-cyclohexyl]-2-trifluoromethoxy-benzenesulfonamide 324538 2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-carbonitrile 324544 17-cyclopropylmethyl-3,10-dihydroxy-13-oxo-(1R,9R,10S)-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-triene-4-carboxamide 324548 17-cyclobutylmethyl-3,10-dihydroxy-13-oxo-(1R,9R,10S)-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-triene-4-carboxamide 324553 2-[4-(4-Chloro-phenylcarbamoyl)-phenyl]-1H-benzoimidazole-5-carboxylic acid amide 324554 2-(4''-Chloro-biphenyl-4-yl)-1H-benzoimidazole-5-carboxylic acid amide 324557 N-{4-[(4-Dimethylamino-quinazolin-2-ylamino)-methyl]-cyclohexylmethyl}-methanesulfonamide 324569 4-Bromo-N-{4-[(4-dimethylamino-quinazolin-2-ylamino)-methyl]-cyclohexylmethyl}-2-trifluoromethoxy-benzenesulfonamide 324577 (R)-2-((3S,4S)-3-((4-(3H-imidazo[4,5-b]pyridin-3-yl)piperidin-1-yl)methyl)-4-phenylpyrrolidin-1-yl)-2-cyclohexylacetic acid 324578 [4-(1-Isopropyl-piperidin-4-yloxy)-benzyl]-dimethyl-amine 324579 Diethyl-[4-(1-isopropyl-piperidin-4-yloxy)-benzyl]-amine 324589 1-{(1R,2S)-2-[(S)-3-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-(3-fluoro-4-methyl-phenyl)-urea 324590 1-((1R,2S)-2-(((S)-3-(4-fluorobenzyl)piperidin-1-yl)methyl)cyclohexyl)-3-(5-acetyl-4-methylthiazol-2-yl)urea 324591 Naltrindole analogue 324592 Naltrindole analogue 324611 N*2*-(3H-Benzoimidazol-5-yl)-N*4*-(4-chloro-phenyl)-5-trifluoromethyl-pyrimidine-2,4-diamine 324613 (2R,3S,4R,5R)-2-Hydroxymethyl-5-[6-(2-phenyl-cyclopropylamino)-purin-9-yl]-tetrahydro-furan-3,4-diol 324616 (R)-3-Cyclobutyl-2-[(3S,4S)-3-[4-(7-ethyl-imidazo[1,2-a]pyridin-3-yl)-piperidin-1-ylmethyl]-4-(3-fluoro-phenyl)-pyrrolidin-1-yl]-propionic acid 324625 2-[4-(4-Methanesulfonylamino-phenoxy)-phenyl]-1H-benzoimidazole-5-carboxylic acid amide 324626 2-(4-Phenylsulfamoyl-phenyl)-1H-benzoimidazole-5-carboxylic acid amide 324637 N*4*-(3H-Benzoimidazol-5-yl)-N*2*-(4-bromo-phenyl)-5-trifluoromethyl-pyrimidine-2,4-diamine 324638 (3H-Benzoimidazol-5-yl)-(4-o-tolyloxy-5-trifluoromethyl-pyrimidin-2-yl)-amine 324639 Butane-1-sulfonic acid {4-[(4-dimethylamino-quinazolin-2-ylamino)-methyl]-cyclohexylmethyl}-amide 324642 N*4*-(3H-Benzoimidazol-5-yl)-N*2*-m-tolyl-5-trifluoromethyl-pyrimidine-2,4-diamine 324644 (2S,4R)-1-[(S)-2-(2-Benzo[1,3]dioxol-5-yl-acetylamino)-5-guanidino-pentanoyl]-4-benzyl-pyrrolidine-2-carboxylic acid benzylamide 324649 (3H-Benzoimidazol-5-yl)-(4-isopropoxy-5-trifluoromethyl-pyrimidin-2-yl)-amine 324650 (3H-Benzoimidazol-5-yl)-(4-isobutoxy-5-trifluoromethyl-pyrimidin-2-yl)-amine 324668 1-Isopropyl-4-(4-piperidin-1-ylmethyl-phenoxy)-piperidine 324669 1-[4-(1-Isopropyl-piperidin-4-yloxy)-benzyl]-azepane 324681 (2R,3S,4R,5R)-2-Hydroxymethyl-5-{6-[(pyridin-3-ylmethyl)-amino]-purin-9-yl}-tetrahydro-furan-3,4-diol 324691 4-Bromo-N-[4-(quinazolin-2-ylaminomethyl)-cyclohexylmethyl]-2-trifluoromethoxy-benzenesulfonamide 324692 (2S,4R)-4-Benzyl-1-[(S)-5-guanidino-2-(2-naphthalen-1-yl-acetylamino)-pentanoyl]-pyrrolidine-2-carboxylic acid 4-methoxy-benzylamide 324698 N*2*-(3H-Benzoimidazol-5-yl)-N*4*-(4-methoxy-phenyl)-5-trifluoromethyl-pyrimidine-2,4-diamine 324701 9-(2-Benzenesulfonylmethyl-benzyl)-6-furan-2-yl-9H-purin-2-ylamine 324705 1-{(1R,2S)-2-[(S)-3-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-(1-methyl-1H-pyrazol-3-yl)-urea 324706 1-{(1R,2S)-2-[3-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-(1H-indazol-5-yl)-urea 324719 2-(4-Benzyloxy-phenyl)-1H-benzoimidazole-5-carboxylic acid amide 324721 (2S,4R)-4-Benzyl-1-((S)-5-guanidino-2-phenylacetylamino-pentanoyl)-pyrrolidine-2-carboxylic acid benzylamide 324726 N*2*,N*4*-Bis-(1H-benzoimidazol-5-yl)-5-trifluoromethyl-pyrimidine-2,4-diamine 324732 (2S,4R)-4-Benzyl-1-{(S)-2-[2-(2-chloro-phenyl)-acetylamino]-5-guanidino-pentanoyl}-pyrrolidine-2-carboxylic acid benzylamide 324740 N-{4-[(4-Amino-quinazolin-2-ylamino)-methyl]-cyclohexylmethyl}-4-bromo-2-trifluoromethoxy-benzenesulfonamide 324742 (2S,4R)-4-Benzyl-1-[(S)-5-guanidino-2-(2-1H-indol-3-yl-acetylamino)-pentanoyl]-pyrrolidine-2-carboxylic acid benzylamide 324743 (R)-2-cyclohexyl-2-((3S,4S)-3-((4-(2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)methyl)-4-phenylpyrrolidin-1-yl)acetic acid 324746 2-[4-(4-Chloro-phenylsulfamoyl)-phenyl]-1H-benzoimidazole-5-carboxylic acid amide 324747 Naltrindole analogue 324749 {1-[4-(1-Isopropyl-piperidin-4-yloxy)-benzyl]-piperidin-4-yl}-methanol 324750 4-[4-(4-benzylhexahydro-1-pyridinylmethyl)phenoxy]-1-isopropylhexahydropyridine 324753 2-(4-(4-hydroxyphenylthio)phenyl)-1H-benzo[d]imidazole-5-carboxamide 324755 (3H-Benzoimidazol-5-yl)-[4-(4-fluoro-phenoxy)-5-trifluoromethyl-pyrimidin-2-yl]-amine 324761 N*4*-(3H-Benzoimidazol-5-yl)-5-bromo-N*2*-[4-(pyridin-3-yloxy)-phenyl]-pyrimidine-2,4-diamine 324764 (2R,3R,4S,5R)-2-(2-Amino-6-methylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 324766 4-(5-Pyrrolidin-1-yl-pentyloxy)-benzonitrile 324768 (2S,4R)-4-Benzyl-1-[(S)-5-guanidino-2-(2-1H-indol-3-yl-acetylamino)-pentanoyl]-pyrrolidine-2-carboxylic acid (3-phenyl-propyl)-amide 324770 (R)-3-Cyclobutyl-2-[(3S,4S)-3-(4-imidazo[1,2-a]pyrimidin-2-yl-piperidin-1-ylmethyl)-4-phenyl-pyrrolidin-1-yl]-propionic acid 324771 (R)-3-Cyclobutyl-2-{(3S,4S)-3-(3-fluoro-phenyl)-4-[4-(6-phenyl-imidazo[1,2-a]pyridin-3-yl)-piperidin-1-ylmethyl]-pyrrolidin-1-yl}-propionic acid 324773 1-{(1R,2S)-2-[(S)-3-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-(4-fluoro-phenyl)-urea 324774 1-{(1R,2S)-2-[(S)-3-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-[1,3,4]thiadiazol-2-yl-urea 324775 Naltrindole analogue 324777 {[(2S,4R,6R)-17-fluoro-3-oxa-13-thiatetracyclo[12.4.0.0^{2,6}.0^{7,12}]octadeca-1(14),7(12),8,10,15,17-hexaen-4-yl]methyl}dimethylamine 324782 2-[4-(6-Chloro-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-quinolin-6-yl-acetamide 324785 4-Bromo-N-{4-[(4-dimethylamino-quinazolin-2-ylamino)-methyl]-cyclohexyl}-2-trifluoromethoxy-benzenesulfonamide 324793 (S)-N-{(S)-1-[(S)-1-(Carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-3-((S)-2-{(R)-2-[((S)-6-hydroxy-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl)-amino]-propionylamino}-3-phenyl-propionylamino)-succinamic acid 324794 (S)-1-((S)-6-Hydroxy-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl)-pyrrolidine-2-carboxylic acid [(S)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-ethyl]-amide 324795 4-Bromo-N-[4-(quinazolin-2-ylamino)-cyclohexylmethyl]-2-trifluoromethoxy-benzenesulfonamide 324798 1-(4-(4-(piperidin-1-ylmethyl)benzyloxy)benzyl)piperidine 324801 6-Furan-2-yl-9-naphthalen-2-ylmethyl-9H-purin-2-ylamine 324807 1-(3,5-Diacetyl-phenyl)-3-{(1R,2S)-2-[(S)-3-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-urea 324813 Naltrindole analogue 324820 (2R,3R,4S,5R)-2-[6-(2,2-Diphenyl-ethylamino)-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 324833 2-Amino-N-((S)-1-{[(1-{(S)-4-[(R)-2-(2-{2-[1-amino-2-((R)-4-hydroxy-phenyl)-ethylamino]-propionylamino}-acetylamino)-3-(S)-phenyl-propionylamino]-phenylcarbamoyl}-2-phenyl-ethylcarbamoyl)-methyl]-carbamoyl}-ethyl)-3-(4-hydroxy-phenyl)-propionamide; ditrifluoroacetic acid 324834 2-Amino-N-(1-{[(2-{(S)-4-[(R)-2-(2-{(S)-2-[1-amino-2-((R)-4-hydroxy-phenyl)-ethylamino]-propionylamino}-acetylamino)-3-phenyl-propionyl]-piperazin-1-yl}-1-benzyl-2-oxo-ethylcarbamoyl)-methyl]-carbamoyl}-ethyl)-3-((R)-4-hydroxy-phenyl)-propionamide; ditrifluoroacetic acid 324835 2-Amino-N-(1-{[(1-{(S)-2-[(R)-2-(2-{(S)-2-[1-amino-2-((R)-4-hydroxy-phenyl)-ethylamino]-propionylamino}-acetylamino)-3-phenyl-propionylamino]-phenylcarbamoyl}-2-phenyl-ethylcarbamoyl)-methyl]-carbamoyl}-ethyl)-3-((R)-4-hydroxy-phenyl)-propionamide; ditrifluoroacetic acid 324837 (2R,3R,4S,5R)-2-[6-(5-Chloro-2-methoxy-benzylamino)-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 324841 17-cyclopropylmethyl-3,4,10-trihydroxy-(1R,9R,10S)-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-13-one 324851 1-(3,4-Difluoro-phenyl)-3-{(1R,2S)-2-[(S)-3-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-urea 324852 Naltrindole analogue 324853 Naltrindole analogue 324855 4-[4-(3H-Benzoimidazol-5-ylamino)-5-trifluoromethyl-pyrimidin-2-ylamino]-benzenesulfonamide 324861 (3H-Benzoimidazol-5-yl)-[4-(4-bromo-phenoxy)-5-trifluoromethyl-pyrimidin-2-yl]-amine 324867 N*2*,N*4*-Bis-(1H-benzoimidazol-5-yl)-5-fluoro-pyrimidine-2,4-diamine 324868 N*2*-(3H-Benzoimidazol-5-yl)-N*4*-(3-chloro-phenyl)-5-trifluoromethyl-pyrimidine-2,4-diamine 324869 N*2*-[1-(4-Bromo-2-trifluoromethoxy-benzenesulfonyl)-piperidin-4-ylmethyl]-N*4*,N*4*-dimethyl-quinazoline-2,4-diamine 324890 9-(2-Fluoro-4-trifluoromethyl-benzyl)-6-furan-2-yl-9H-purin-2-ylamine 324891 (R)-{(3S,4S)-3-[4-(2-Benzoimidazol-1-yl-ethyl)-piperidin-1-ylmethyl]-4-phenyl-pyrrolidin-1-yl}-cyclohexyl-acetic acid 324947 6-Furan-2-yl-9-(1-phenyl-ethyl)-9H-purin-2-ylamine 324968 (R)-Cyclohexyl-{(3S,4S)-3-[4-(1H-indol-3-yl)-piperidin-1-ylmethyl]-4-phenyl-pyrrolidin-1-yl}-acetic acid 324971 (R)-Cyclohexyl-{(3S,4S)-3-[4-(4-oxo-4H-quinazolin-1-yl)-piperidin-1-ylmethyl]-4-phenyl-pyrrolidin-1-yl}-acetic acid 324975 6-Furan-2-yl-9-(2-methoxy-benzyl)-9H-purin-2-ylamine 324981 9-(2,6-difluorobenzyl)-6-(furan-2-yl)-9H-purin-2-amine 324997 (R)-2-[(3S,4S)-3-[4-(6-Chloro-imidazo[1,2-a]pyridin-3-yl)-piperidin-1-ylmethyl]-4-(3-fluoro-phenyl)-pyrrolidin-1-yl]-3-cyclobutyl-propionic acid 325006 (R)-3-Cyclobutyl-2-[(3S,4S)-3-[4-(6-fluoro-imidazo[1,2-a]pyridin-3-yl)-piperidin-1-ylmethyl]-4-(3-fluoro-phenyl)-pyrrolidin-1-yl]-propionic acid 325007 (R)-3-Cyclobutyl-2-{(3S,4S)-3-(3-fluoro-phenyl)-4-[4-(6-trifluoromethyl-imidazo[1,2-a]pyridin-3-yl)-piperidin-1-ylmethyl]-pyrrolidin-1-yl}-propionic acid 325012 (R)-3-Cyclobutyl-2-[(3S,4S)-3-phenyl-4-(4-[1,2,4]triazolo[4,3-a]pyridin-3-yl-piperidin-1-ylmethyl)-pyrrolidin-1-yl]-propionic acid 325018 6-Furan-2-yl-9-(2,4,6-trifluoro-benzyl)-9H-purin-2-ylamine 325019 (R)-[(3S,4S)-3-(4-Benzoimidazol-1-ylmethyl-piperidin-1-ylmethyl)-4-phenyl-pyrrolidin-1-yl]-cyclohexyl-acetic acid 325070 6-Furan-2-yl-9-phenethyl-9H-purin-2-ylamine 325077 9-(4-Chloro-benzyl)-6-furan-2-yl-9H-purin-2-ylamine 325081 9-(2,6-Dichloro-benzyl)-6-furan-2-yl-9H-purin-2-ylamine 325082 6-Furan-2-yl-9-naphthalen-1-ylmethyl-9H-purin-2-ylamine 325097 6-Furan-2-yl-9-(3-phenyl-propyl)-9H-purin-2-ylamine 325102 9-(4-(trifluoromethyl)benzyl)-6-(furan-2-yl)-9H-purin-2-amine 325103 (R)-2-((3S,4S)-3-((4-(1H-benzo[d]imidazol-1-yl)piperidin-1-yl)methyl)-4-phenylpyrrolidin-1-yl)-2-cyclohexylacetic acid 325157 (R)-Cyclohexyl-{(3S,4S)-3-[4-(4-oxo-4H-quinazolin-3-yl)-piperidin-1-ylmethyl]-4-phenyl-pyrrolidin-1-yl}-acetic acid 325192 2-amino-6-(2-furyl)-9-(4-methoxyphenylmethyl)-9Hpurine 325193 6-Furan-2-yl-9-(4-isopropyl-benzyl)-9H-purin-2-ylamine 325221 9-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-6-furan-2-yl-9H-purin-2-ylamine 325223 (R)-{(3S,4S)-3-[4-(3-Benzoimidazol-1-yl-propyl)-piperidin-1-ylmethyl]-4-phenyl-pyrrolidin-1-yl}-cyclohexyl-acetic acid 325275 (R)-[(3S,4S)-3-(4-Benzotriazol-1-yl-piperidin-1-ylmethyl)-4-phenyl-pyrrolidin-1-yl]-cyclohexyl-acetic acid 325279 6-Furan-2-yl-9-phenyl-9H-purin-2-ylamine 325280 9-benzyl-6-(furan-2-yl)-9H-purin-2-amine 325307 (R)-3-Cyclobutyl-2-[(3S,4S)-3-[4-(6,8-dichloro-imidazo[1,2-a]pyridin-3-yl)-piperidin-1-ylmethyl]-4-(3-fluoro-phenyl)-pyrrolidin-1-yl]-propionic acid 325318 (R)-3-Cyclobutyl-2-{(3S,4S)-3-(3-fluoro-phenyl)-4-[4-(6-nitro-imidazo[1,2-a]pyridin-3-yl)-piperidin-1-ylmethyl]-pyrrolidin-1-yl}-propionic acid 325322 9-(3-methoxybenzyl)-6-(furan-2-yl)-9H-purin-2-amine 325343 (R)-2-((3S,4S)-3-((4-(1H-imidazo[4,5-b]pyridin-1-yl)piperidin-1-yl)methyl)-4-phenylpyrrolidin-1-yl)-2-cyclohexylacetic acid 325351 9-(3-Fluoro-4-trifluoromethyl-benzyl)-6-furan-2-yl-9H-purin-2-ylamine 325384 1-(4-(4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimidin-5-yl)phenyl)urea 325423 5-(4-(dimethylamino)phenyl)-6-(4-methoxyphenyl)furo[2,3-d]pyrimidin-4-amine 325428 2-Ethoxymethyl-4-(4-fluoro-phenyl)-3-[2-((R)-1-phenyl-ethylamino)-pyrimidin-4-yl]-2H-isoxazol-5-one 325429 [1-Isopropyl-2-(2-methoxy-5-nitro-benzylsulfanyl)-1H-benzoimidazol-5-yl]-carbamic acid tert-butyl ester 325442 1-(4-(4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimidin-5-yl)phenyl)-3-phenylurea 325443 1-(4-(4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimidin-5-yl)phenyl)-3-(2-fluoro-5-(trifluoromethyl)phenyl)urea 325445 [4-(4-Fluoro-phenyl)-5-oxo-3-(2-phenoxy-pyrimidin-4-yl)-5H-isoxazol-2-yl]-acetaldehyde 325462 1-tert-Butyl-3-[1-(2-methoxy-ethyl)-2-(2-methoxy-5-nitro-benzylsulfanyl)-1H-benzoimidazol-5-yl]-urea 325486 4-[6-Amino-5-(2,6-difluoro-benzoyl)-pyridin-2-ylamino]-N,N-dimethyl-benzenesulfonamide 325502 N-[1-Isopropyl-2-(2-methoxy-5-nitro-benzylsulfanyl)-1H-benzoimidazol-5-yl]-isobutyramide 325516 6-(3,4-dichlorophenyl)-5-(4-methoxyphenyl)furo[2,3-d]pyrimidin-4-amine 325539 1-tert-Butyl-3-[2-(2-methoxy-5-nitro-benzylsulfanyl)-1-phenethyl-1H-benzoimidazol-5-yl]-urea 325550 1-(4-(4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimidin-5-yl)phenyl)-3-cyclohexylurea 325590 N-(3-(4-amino-5-(4-methoxyphenyl)furo[2,3-d]pyrimidin-6-yl)phenyl)methanesulfonamide 325613 5,6-bis(4-methoxyphenyl)furo[2,3-d]pyrimidin-4-amine 325614 5-(4-methoxyphenyl)furo[2,3-d]pyrimidin-4-amine 325638 N-(4-(4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimidin-5-yl)phenyl)-3-chlorobenzenesulfonamide 325699 2-Ethoxymethyl-4-(4-fluoro-phenyl)-3-[2-((S)-1-phenyl-ethylamino)-pyrimidin-4-yl]-2H-isoxazol-5-one 325722 2-Ethoxymethyl-4-(4-fluoro-phenyl)-3-[2-(2-hydroxy-phenoxy)-pyrimidin-4-yl]-2H-isoxazol-5-one 325724 3-(4-amino-5-(4-methoxyphenyl)furo[2,3-d]pyrimidin-6-yl)-N,N-dimethylbenzamide 325735 Cyclobutanecarboxylic acid [1-isopropyl-2-(2-methoxy-5-nitro-benzylsulfanyl)-1H-benzoimidazol-5-yl]-amide 325765 N-(4-(4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimidin-5-yl)phenyl)-3-fluorobenzamide 325767 1-[1-Benzyl-2-(2-methoxy-5-nitro-benzylsulfanyl)-1H-benzoimidazol-5-yl]-3-tert-butyl-urea 325775 1-(4-(4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimidin-5-yl)phenyl)-3-(4-chlorophenyl)urea 325790 N-(3-(4-amino-5-(biphenyl-4-yl)furo[2,3-d]pyrimidin-6-yl)phenyl)methanesulfonamide 325797 N-[1-Isopropyl-2-(2-methoxy-5-nitro-benzylsulfanyl)-1H-benzoimidazol-5-yl]-2,2-dimethyl-propionamide 325832 1-tert-Butyl-3-[2-(2-methoxy-5-nitro-benzylsulfanyl)-1-pyridin-2-ylmethyl-1H-benzoimidazol-5-yl]-urea 325839 2-Ethoxymethyl-4-(4-fluoro-phenyl)-3-[2-(3-hydroxy-phenoxy)-pyrimidin-4-yl]-2H-isoxazol-5-one 325851 3-(4-amino-5-(4-methoxyphenyl)furo[2,3-d]pyrimidin-6-yl)benzamide 325857 4-[6-Amino-5-(2,6-difluoro-benzoyl)-pyridin-2-ylamino]-benzenesulfonamide 325887 N-(4-phenoxyphenyl)-N'-[1-(2-pyrrolidin-1-ylethyl)-1H-indazol-5-yl]urea 325888 1-[1-(3-Cyclopentylamino-propyl)-1H-indazol-5-yl]-3-(4-phenoxy-phenyl)-urea 325890 N-[3-(4-Carbamoyl-5-ureido-thiophen-2-ylethynyl)-phenyl]-isonicotinamide 325896 N-[1-Isopropyl-2-(2-methoxy-5-nitro-benzylsulfanyl)-1H-benzoimidazol-5-yl]-3,3-dimethyl-butyramide 325907 Decanoic acid (2-dimethylamino-ethyl)-{1-[3-(4-methoxy-phenyl)-4-oxo-3,4-dihydro-quinazolin-2-yl]-ethyl}-amide 325910 (1R,2S,4aR,13bS)-2-Hydroxy-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydro-indolo[2',3':3,4]pyrido[1,2-b]isoquinoline-1-carboxylic acid 325911 4-[((1R,2S,4aR,13bS)-2-Hydroxy-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydro-indolo[2',3':3,4]pyrido[1,2-b]isoquinoline-1-carbonyl)-amino]-butyric acid benzyl ester 325912 {3-[((1R,2S,4aR,13bS)-2-Hydroxy-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydro-indolo[2',3':3,4]pyrido[1,2-b]isoquinoline-1-carbonyl)-amino]-propyl}-carbamic acid tert-butyl ester 325913 {3-[((1R,2S,4aR,13bS)-2-Hydroxy-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydro-indolo[2',3':3,4]pyrido[1,2-b]isoquinoline-1-carbonyl)-amino]-propyl}-carbamic acid benzyl ester 325916 8-((2S,3aS,12bS)-11-Bromo-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-7-oxa-8-aza-bicyclo[4.2.0]octa-1(6),2,4-trien-3-ylamine 325917 1-(3-{5-[3-(4-Phenoxy-phenyl)-ureido]-indazol-1-yl}-propyl)-piperidine-4-carboxylic acid amide 325919 (1R,2S,4aR,13bS)-2-Hydroxy-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydro-indolo[2',3':3,4]pyrido[1,2-b]isoquinoline-1-carboxylic acid (3-amino-propyl)-amide 325925 1-tert-Butyl-3-[2-(2-methoxy-5-nitro-benzylsulfanyl)-1-phenyl-1H-benzoimidazol-5-yl]-urea 325938 5-[5-(1-Hydroxy-2-methyl-propyl)-thiophen-3-ylethynyl]-2-ureido-thiophene-3-carboxylic acid amide 325944 Decanoic acid {1-[3-(2-cyano-phenyl)-4-oxo-3,4-dihydro-quinazolin-2-yl]-ethyl}-(2-dimethylamino-ethyl)-amide 325948 5-(3-Amino-phenylethynyl)-2-ureido-thiophene-3-carboxylic acid amide 325952 ((2R,3aS,12bS)-11-Fluoro-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-dimethyl-amine 325957 Cyclopropanecarboxylic acid [1-isopropyl-2-(3-methyl-benzylsulfanyl)-1H-benzoimidazol-5-yl]-amide 325958 1-Isopropyl-3-[1-isopropyl-2-(2-methoxy-5-nitro-benzylsulfanyl)-1H-benzoimidazol-5-yl]-urea 325979 Azaline B derivative 325980 Azaline B derivative 325981 Azaline B derivative 325982 Azaline B derivative 325987 6-(3-tert-Butyl-ureido)-2-(2-methoxy-5-nitro-benzylsulfanyl)-3-propyl-3H-benzoimidazole-4-carboxylic acid 325988 1-tert-Butyl-3-[2-(2-methoxy-5-nitro-benzylsulfanyl)-1-propyl-7-(pyrrolidine-1-carbonyl)-1H-benzoimidazol-5-yl]-urea 325990 Cyclopropanecarboxylic acid [1-isopropyl-2-(2-methoxy-benzylsulfanyl)-1H-benzoimidazol-5-yl]-amide 325999 8-((2S,3aS,12bS)-11-Bromo-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-7-oxa-8-aza-bicyclo[4.2.0]octa-1(6),2,4-triene-3-carbonitrile 326000 1-{1-[2-(4-Hydroxy-piperidin-1-yl)-ethyl]-1H-indazol-5-yl}-3-(4-phenoxy-phenyl)-urea 326001 8-((2S,3aS,12bS)-11-Bromo-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-3-morpholin-4-yl-7-oxa-8-aza-bicyclo[4.2.0]octa-1(6),2,4-triene 326005 1-[2-(4-Phenoxy-phenyl)-ethyl]-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-5-yl]-urea 326007 5-(3-Acetylamino-phenylethynyl)-2-ureido-thiophene-3-carboxylic acid amide 326008 1-(4-Phenoxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-4-yl]-urea 326016 1-Cyclopropyl-3-[1-isopropyl-2-(2-methoxy-5-nitro-benzylsulfanyl)-1H-benzoimidazol-5-yl]-urea 326023 Cyclopropanecarboxylic acid [1-isopropyl-2-(2-methoxy-5-nitro-benzylsulfanyl)-1H-benzoimidazol-5-yl]-amide 326025 1-(4-Phenoxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-6-yl]-urea 326026 Decanoic acid {1-[3-(4-cyano-phenyl)-4-oxo-3,4-dihydro-quinazolin-2-yl]-ethyl}-(2-dimethylamino-ethyl)-amide 326050 8-((2S,3aS,12bS)-11-Bromo-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-7-oxa-8-aza-bicyclo[4.2.0]octa-1(6),2,4-triene-3-carboxylic acid ethyl ester 326051 1-{1-[2-((S)-2-Methoxymethyl-pyrrolidin-1-yl)-ethyl]-1H-indazol-5-yl}-3-(4-phenoxy-phenyl)-urea 326053 5-(2-Fluoro-phenylethynyl)-2-ureido-thiophene-3-carboxylic acid amide 326054 5-(2-Chloro-phenylethynyl)-2-ureido-thiophene-3-carboxylic acid amide 326057 N-[3-(4-Carbamoyl-5-ureido-thiophen-2-ylethynyl)-phenyl]-nicotinamide 326072 Cyclopropanecarboxylic acid [2-(2-chloro-benzylsulfanyl)-1-isopropyl-1H-benzoimidazol-5-yl]-amide 326073 1-tert-Butyl-3-[1-ethyl-2-(2-methoxy-5-nitro-benzylsulfanyl)-1H-benzoimidazol-5-yl]-urea 326074 6-(3-tert-Butyl-ureido)-2-(2-methoxy-5-nitro-benzylsulfanyl)-3-propyl-3H-benzoimidazole-4-carboxylic acid (pyridin-4-ylmethyl)-amide 326075 6-(3-tert-Butyl-ureido)-2-(2-methoxy-5-nitro-benzylsulfanyl)-3-propyl-3H-benzoimidazole-4-carboxylic acid (pyridin-3-ylmethyl)-amide 326076 6-(3-tert-Butyl-ureido)-2-(2-methoxy-5-nitro-benzylsulfanyl)-3-propyl-3H-benzoimidazole-4-carboxylic acid (pyridin-2-ylmethyl)-amide 326077 6-(3-tert-Butyl-ureido)-2-(2-methoxy-5-nitro-benzylsulfanyl)-3-propyl-3H-benzoimidazole-4-carboxylic acid (2-pyridin-4-yl-ethyl)-amide 326078 6-(3-tert-Butyl-ureido)-2-(2-methoxy-5-nitro-benzylsulfanyl)-3-propyl-3H-benzoimidazole-4-carboxylic acid (2-pyridin-3-yl-ethyl)-amide 326079 6-(3-tert-Butyl-ureido)-2-(2-methoxy-5-nitro-benzylsulfanyl)-3-propyl-3H-benzoimidazole-4-carboxylic acid (3-dimethylamino-propyl)-amide 326080 Cyclopropanecarboxylic acid [2-(5-acetyl-2-methoxy-benzylsulfanyl)-1-isopropyl-1H-benzoimidazol-5-yl]-amide 326081 1-tert-Butyl-3-[1-butyl-2-(2-methoxy-5-nitro-benzylsulfanyl)-1H-benzoimidazol-5-yl]-urea 326082 6-(3-tert-Butyl-ureido)-2-(2-methoxy-5-nitro-benzylsulfanyl)-3-propyl-3H-benzoimidazole-4-carboxylic acid (2-pyridin-2-yl-ethyl)-amide 326086 Decanoic acid (2-dimethylamino-ethyl)-[1-(4-oxo-3-phenyl-3,4-dihydro-quinazolin-2-yl)-ethyl]-amide 326088 1N-{3-[2-hydroxy-(1R,2S,4aR,13bS)-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroisoquino[3,2-a]b-carbolin-1-ylcarboxamido]propyl}-2-hydroxy-(1S,2R,4aS,13bR,14aR)-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroisoquino[3,2-a] 326093 8-((2S,3aS,12bS)-11-Bromo-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-3-morpholin-4-ylmethyl-7-oxa-8-aza-bicyclo[4.2.0]octa-1(6),2,4-triene 326095 1-(4-Benzyloxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-5-yl]-urea 326098 ((2S,3aS,12bS)-11-Chloro-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-dimethyl-amine 326099 ((2R,3aS,12bS)-11-Bromo-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-dimethyl-amine 326105 1-tert-Butyl-3-[2-(2-methoxy-5-nitro-benzylsulfanyl)-1-pyridin-3-ylmethyl-1H-benzoimidazol-5-yl]-urea 326114 1-tert-Butyl-3-[2-(2-methoxy-5-nitro-benzylsulfanyl)-1-pyridin-4-ylmethyl-1H-benzoimidazol-5-yl]-urea 326118 5-[5-(1-Hydroxy-propyl)-thiophen-3-ylethynyl]-2-ureido-thiophene-3-carboxylic acid amide 326124 1-{1-[3-((S)-2-Methoxymethyl-pyrrolidin-1-yl)-propyl]-1H-indazol-5-yl}-3-(4-phenoxy-phenyl)-urea 326128 Dimethyl-[(2R,3aS,12bR)-1-(2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-yl)methyl]-amine 326136 Azaline B derivative 326137 Azaline B derivative 326155 5-(3-Methanesulfonylamino-phenylethynyl)-2-ureido-thiophene-3-carboxylic acid amide 326158 5-(3-Hydroxy-phenylethynyl)-2-ureido-thiophene-3-carboxylic acid amide 326159 5-Cyclopropylethynyl-2-ureido-thiophene-3-carboxylic acid amide 326160 {2-[((1R,2S,4aR,13bS)-2-Hydroxy-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydro-indolo[2',3':3,4]pyrido[1,2-b]isoquinoline-1-carbonyl)-amino]-acetylamino}-acetic acid methyl ester 326165 1-(4-Benzyloxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-4-yl]-urea 326170 1-tert-Butyl-3-[1-isopropyl-2-(2-methoxy-5-nitro-benzylsulfanyl)-1H-benzoimidazol-5-yl]-urea 326181 8-((2S,3aS,12bS)-11-Bromo-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-3-phenyl-7-oxa-8-aza-bicyclo[4.2.0]octa-1(6),2,4-triene 326182 N-(2-(dimethylamino)ethyl)-N-(1-(3-(4-fluorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)decanamide 326184 1-[2-(4-Phenoxy-phenyl)-ethyl]-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-6-yl]-urea 326188 1-(4-Phenoxy-benzyl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-5-yl]-urea 326190 5-(3-Benzoylamino-phenylethynyl)-2-ureido-thiophene-3-carboxylic acid amide 326193 5-[3-(2-Dimethylamino-acetylamino)-phenylethynyl]-2-ureido-thiophene-3-carboxylic acid amide 326195 6-(3-tert-Butyl-ureido)-2-(2-methoxy-5-nitro-benzylsulfanyl)-3-propyl-3H-benzoimidazole-4-carboxylic acid methyl ester 326205 Cyclopropanecarboxylic acid [2-(5-chloro-2-methoxy-benzylsulfanyl)-1-isopropyl-1H-benzoimidazol-5-yl]-amide 326208 5-(5-Cyano-thiophen-3-ylethynyl)-2-ureido-thiophene-3-carboxylic acid amide 326209 1-[1-(2-Isobutylamino-ethyl)-1H-indazol-5-yl]-3-(4-phenoxy-phenyl)-urea 326213 [8-((2S,3aS,12bS)-11-Bromo-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-7-oxa-8-aza-bicyclo[4.2.0]octa-1(6),2,4-trien-3-yl]-dimethyl-amine 326214 1-{1-[3-(4-Hydroxy-piperidin-1-yl)-propyl]-1H-indazol-5-yl}-3-(4-phenoxy-phenyl)-urea 326222 Cyclopropanecarboxylic acid [1-isopropyl-2-(2-methyl-benzylsulfanyl)-1H-benzoimidazol-5-yl]-amide 326223 1-[1-Isopropyl-2-(2-methoxy-5-nitro-benzylsulfanyl)-1H-benzoimidazol-5-yl]-3-methyl-urea 326232 1-(4-Benzyloxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-6-yl]-urea 326233 5-(3-Fluoro-phenylethynyl)-2-ureido-thiophene-3-carboxylic acid amide 326235 [((1R,2S,4aR,13bS)-2-Hydroxy-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydro-indolo[2',3':3,4]pyrido[1,2-b]isoquinoline-1-carbonyl)-amino]-acetic acid methyl ester 326238 Decanoic acid {1-[3-(3-cyano-phenyl)-4-oxo-3,4-dihydro-quinazolin-2-yl]-ethyl}-(2-dimethylamino-ethyl)-amide 326239 4-[((1R,2S,4aR,13bS)-2-Hydroxy-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydro-indolo[2',3':3,4]pyrido[1,2-b]isoquinoline-1-carbonyl)-amino]-butyric acid 326243 ((2S,3aS,12bS)-11-Fluoro-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-dimethyl-amine 326247 6-(3-tert-Butyl-ureido)-2-(2-methoxy-5-nitro-benzylsulfanyl)-3-propyl-3H-benzoimidazole-4-carboxylic acid dimethylamide 326254 1-{1-[2-(3,3-Difluoro-pyrrolidin-1-yl)-ethyl]-1H-indazol-5-yl}-3-(4-phenoxy-phenyl)-urea 326259 1-(1-Benzyl-piperidin-4-yl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-6-yl]-urea 326264 ((2R,3aS,12bS)-11-Chloro-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-dimethyl-amine 326278 1-tert-Butyl-3-[1-cyclopropyl-2-(2-methoxy-5-nitro-benzylsulfanyl)-1H-benzoimidazol-5-yl]-urea 326289 1-[8-((2S,3aS,12bS)-11-Bromo-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-7-oxa-8-aza-bicyclo[4.2.0]octa-1(6),2,4-trien-3-yl]-azetidin-2-one 326290 1-(2-{5-[3-(4-Phenoxy-phenyl)-ureido]-indazol-1-yl}-ethyl)-piperidine-4-carboxylic acid amide 326299 1-(1-Benzyl-piperidin-4-yl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-5-yl]-urea 326303 Azaline B derivative 326304 Azaline B derivative 326305 Azaline B derivative 326306 1-(4-Phenoxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-5-yl]-1,3-dihydro-imidazol-2-one 326311 6-(3-tert-Butyl-ureido)-2-(2-methoxy-5-nitro-benzylsulfanyl)-3-propyl-3H-benzoimidazole-4-carboxylic acid methylamide 326312 6-(3-tert-Butyl-ureido)-2-(2-methoxy-5-nitro-benzylsulfanyl)-3-propyl-3H-benzoimidazole-4-carboxylic acid tert-butylamide 326313 6-(3-tert-Butyl-ureido)-2-(2-methoxy-5-nitro-benzylsulfanyl)-3-propyl-3H-benzoimidazole-4-carboxylic acid benzylamide 326314 3-[5-(Cyclopropanecarbonyl-amino)-1-isopropyl-1H-benzoimidazol-2-ylsulfanylmethyl]-4-methoxy-benzoic acid methyl ester 326315 1-tert-Butyl-3-[2-(2-methoxy-5-nitro-benzylsulfanyl)-1-propyl-1H-benzoimidazol-5-yl]-urea 326316 6-(3-tert-Butyl-ureido)-2-(2-methoxy-5-nitro-benzylsulfanyl)-3-propyl-3H-benzoimidazole-4-carboxylic acid [3-(benzyl-methyl-amino)-propyl]-amide 326325 Decanoic acid (2-dimethylamino-ethyl)-[1-(4-oxo-3-p-tolyl-3,4-dihydro-quinazolin-2-yl)-ethyl]-amide 326334 5-[3-(2,2,2-Trifluoro-acetylamino)-phenylethynyl]-2-ureido-thiophene-3-carboxylic acid amide 326345 6-(3-tert-Butyl-ureido)-2-(2-methoxy-5-nitro-benzylsulfanyl)-3-propyl-3H-benzoimidazole-4-carboxylic acid (2-amino-ethyl)-amide 326347 Cyclopropanecarboxylic acid [2-(5-cyano-2-methoxy-benzylsulfanyl)-1-isopropyl-1H-benzoimidazol-5-yl]-amide 326348 1-tert-Butyl-3-[2-(2-methoxy-5-nitro-benzylsulfanyl)-1-pentyl-1H-benzoimidazol-5-yl]-urea 326352 8-((2S,3aS,12bS)-11-Bromo-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-3-methyl-7-oxa-8-aza-bicyclo[4.2.0]octa-1(6),2,4-triene 326353 1-(4-Phenoxy-benzyl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-6-yl]-urea 326354 1-[1-(2-Cyclopentylamino-ethyl)-1H-indazol-5-yl]-3-(4-phenoxy-phenyl)-urea 326355 5-o-Tolylethynyl-2-ureido-thiophene-3-carboxylic acid amide 326358 {2-[3-(4-Carbamoyl-5-ureido-thiophen-2-ylethynyl)-phenylcarbamoyl]-ethyl}-carbamic acid methyl ester 326395 ((2S,3aS,12bS)-11-Bromo-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-dimethyl-amine 326404 {6-[(Diphenylcarbamoyloxy)-methyl]-5,6,7,8-tetrahydro-naphthalen-1-yloxy}-acetic acid 326407 (R)-2-{(S)-1-[2-Amino-3-((S)-4-hydroxy-phenyl)-propionyl]-pyrrolidin-2-ylmethyleneaminooxy}-N-((S)-1-carbamoyl-2-phenyl-ethyl)-3-phenyl-propionamide 326409 ((2R,3aS,12bS)-11-Methoxy-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-dimethyl-amine 326413 3-[2-(Pyridin-4-ylamino)-5-[1,2,4]triazol-1-yl-thiazol-4-yl]-benzonitrile 326447 5-Thiophen-3-ylethynyl-2-ureido-thiophene-3-carboxylic acid amide 326482 3-[5-Imidazol-1-yl-2-(pyridin-3-ylamino)-thiazol-4-yl]-benzonitrile 326491 Azaline B derivative 326506 2-(4-Phenoxy-benzylamino)-N-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indol-6-yl]-acetamide 326507 1-(4-Phenoxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-5-yl]-imidazolidin-2-one 326510 3-[2-(3-Methyl-pyridin-2-ylamino)-5-[1,2,4]triazol-1-yl-thiazol-4-yl]-benzonitrile 326531 3-[5-(2-Methyl-imidazol-1-yl)-2-(pyrazin-2-ylamino)-thiazol-4-yl]-benzonitrile 326544 3-[2-(Pyridin-3-ylamino)-5-[1,2,4]triazol-1-yl-thiazol-4-yl]-benzonitrile 326570 (S)-2-{(S)-1-[2-Amino-3-((S)-4-hydroxy-phenyl)-propionyl]-pyrrolidin-2-ylmethyleneaminooxy}-N-((S)-1-carbamoyl-2-phenyl-ethyl)-3-phenyl-propionamide 326577 ((2S,3aS,12bS)-11-Methoxy-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-dimethyl-amine 326590 {(S)-6-[(Diphenylcarbamoyloxy)-methyl]-5,6-dihydroxy-5,6,7,8-tetrahydro-naphthalen-1-yloxy}-acetic acid 326593 3-[2-(Pyridin-2-ylamino)-5-[1,2,4]triazol-1-yl-thiazol-4-yl]-benzonitrile 326603 1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrrolidine-3-carboxylic acid [(S)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-ethyl]-amide 326604 (S)-2-{(R)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrrolidin-2-yloxyamino}-N-((S)-1-carbamoyl-2-phenyl-ethyl)-3-phenyl-propionamide 326605 (R)-2-{(R)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrrolidin-2-yloxyamino}-N-((S)-1-carbamoyl-2-phenyl-ethyl)-3-phenyl-propionamide 326615 5-(5-Hydroxymethyl-thiophen-3-ylethynyl)-2-ureido-thiophene-3-carboxylic acid amide 326619 (R)-2-(6-((diphenylcarbamoyloxy)methyl)-6-hydroxy-5,6,7,8-tetrahydronaphthalen-1-yloxy)acetic acid 326633 2-[5-Methyl-5-(1H-tetrazol-5-yl)-hexyloxy]-4,6-diphenyl-pyridine 326637 7-(2,4-Dichloro-5-methoxy-phenylamino)-2-[5-(4-methyl-piperazin-1-ylmethyl)-pyridin-2-yl]-thieno[3,2-b]pyridine-6-carbonitrile 326638 7-(2,4-Dichloro-5-methoxy-phenylamino)-2-[6-(4-methyl-piperazin-1-ylmethyl)-pyridin-2-yl]-thieno[3,2-b]pyridine-6-carbonitrile 326639 7-(2,4-Dichloro-5-methoxy-phenylamino)-2-[3-(4-methyl-piperazin-1-yl)-prop-1-ynyl]-thieno[3,2-b]pyridine-6-carbonitrile 326640 7-(2,4-Dichloro-5-methoxy-phenylamino)-2-(5-dimethylaminomethyl-pyridin-2-yl)-thieno[3,2-b]pyridine-6-carbonitrile 326641 7-(2,4-Dichloro-5-methoxy-phenylamino)-2-[5-(4-methyl-piperazine-1-carbonyl)-pyridin-2-yl]-thieno[3,2-b]pyridine-6-carbonitrile 326642 7-(2,4-Dichloro-phenylamino)-2-[5-(4-methyl-piperazin-1-ylmethyl)-pyridin-2-yl]-thieno[3,2-b]pyridine-6-carbonitrile 326643 4-(4-(4-(chlorodifluoromethoxy)phenylamino)phthalazin-1-yl)benzamide 326644 7-(2,4-Dichloro-5-methoxy-phenylamino)-2-[3-(4-methyl-piperazin-1-ylmethyl)-phenyl]-thieno[3,2-b]pyridine-6-carbonitrile 326645 7-(2,4-Dichloro-5-methoxy-phenylamino)-2-(5-piperazin-1-ylmethyl-furan-3-yl)-thieno[3,2-b]pyridine-6-carbonitrile 326646 7-(2,4-Dichloro-5-methoxy-phenylamino)-2-(5-piperazin-1-ylmethyl-furan-2-yl)-thieno[3,2-b]pyridine-6-carbonitrile 326647 7-(2,4-Dichloro-5-methoxy-phenylamino)-2-[2-(4-methyl-piperazin-1-ylmethyl)-thiazol-4-yl]-thieno[3,2-b]pyridine-6-carbonitrile 326648 4-(4-(3-tert-butylphenylamino)phthalazin-1-yl)benzamide 326649 4-(4-(m-tolylamino)phthalazin-1-yl)benzamide 326650 4-(4-(3-bromophenylamino)phthalazin-1-yl)benzamide 326651 4-(4-(4-chlorophenylamino)phthalazin-1-yl)benzamide 326652 4-(4-(p-tolylamino)phthalazin-1-yl)benzamide 326653 4-(4-(4-methoxyphenylamino)phthalazin-1-yl)benzamide 326655 methyl 4-(4-(4-carbamoylphenyl)phthalazin-1-ylamino)benzoate 326657 4-(4-(4-tert-butylphenylamino)phthalazin-1-yl)benzamide 326658 4-(4-(4-bromophenylamino)phthalazin-1-yl)benzamide 326659 4-(4-(3,4-dichlorophenylamino)phthalazin-1-yl)benzamide 326660 4-(4-(3-chlorophenylamino)phthalazin-1-yl)benzamide 326661 3-(4-(4-tert-butylphenylamino)phthalazin-1-yl)benzamide 326662 3-(4-(4-(chlorodifluoromethoxy)phenylamino)phthalazin-1-yl)benzamide 326663 4-(4-(4-tert-butylphenylamino)phthalazin-1-yl)-N-methylbenzamide 326664 4-(4-(4-chlorophenylamino)phthalazin-1-yl)-N-methylbenzamide 326666 (4-(4-(4-(chlorodifluoromethoxy)phenylamino)phthalazin-1-yl)phenyl)(morpholino)methanone 326667 4-[4-(2,4-Dimethyl-phenylamino)-phthalazin-1-yl]-benzamide 326675 SID24276146 326676 4-[4-(4-Chloro-phenylamino)-phthalazin-1-yl]-benzoic acid methyl ester 326686 methyl 4-(4-(4-(chlorodifluoromethoxy)phenylamino)phthalazin-1-yl)benzoate 326709 [6-((3S,5R)-4-Ethyl-3,5-dimethyl-piperazin-1-yl)-5-methoxy-2,3-dihydro-indol-1-yl]-[4-(6-methyl-pyridin-2-yl)-naphthalen-1-yl]-methanone 326710 [6-((3S,5R)-3,5-Dimethyl-4-propyl-piperazin-1-yl)-5-methoxy-2,3-dihydro-indol-1-yl]-[4-(6-methyl-pyridin-2-yl)-naphthalen-1-yl]-methanone 326711 5-Methoxy-6-(4-methyl-piperazin-1-yl)-2,3-dihydro-indole-1-carboxylic acid (2,3-dichloro-phenyl)-amide 326712 5-Methoxy-6-((3S,5R)-3,4,5-trimethyl-piperazin-1-yl)-2,3-dihydro-indole-1-carboxylic acid (2,3-dichloro-phenyl)-amide 326715 (2,3-Dichloro-phenyl)-[5-methoxy-6-((3R,5S)-3,4,5-trimethyl-piperazin-1-yl)-2,3-dihydro-indol-1-yl]-methanone 326716 (3-Chloro-phenyl)-[5-methoxy-6-((3R,5S)-3,4,5-trimethyl-piperazin-1-yl)-2,3-dihydro-indol-1-yl]-methanone 326717 [5-Methoxy-6-(4-methyl-piperazin-1-yl)-2,3-dihydro-indol-1-yl]-[4-(6-methyl-pyridin-2-yl)-naphthalen-1-yl]-methanone 326718 [5-Methoxy-6-((3S,5R)-3,4,5-trimethyl-piperazin-1-yl)-2,3-dihydro-indol-1-yl]-[4-(6-methyl-pyridin-2-yl)-naphthalen-1-yl]-methanone 326719 [6-((3S,5R)-3,5-Dimethyl-piperazin-1-yl)-5-methoxy-2,3-dihydro-indol-1-yl]-[4-(6-methyl-pyridin-2-yl)-naphthalen-1-yl]-methanone 326720 2-(3-Chloro-2-fluoro-phenyl)-1-[5-methoxy-6-((3R,5S)-3,4,5-trimethyl-piperazin-1-yl)-2,3-dihydro-indol-1-yl]-ethanone 326721 2-(3-Fluoro-2-trifluoromethyl-phenyl)-1-[5-methoxy-6-((3S,5R)-3,4,5-trimethyl-piperazin-1-yl)-2,3-dihydro-indol-1-yl]-ethanone 326722 5-Methoxy-6-((3R,5S)-3,4,5-trimethyl-piperazin-1-yl)-2,3-dihydro-indole-1-carboxylic acid (2-fluoro-3-trifluoromethyl-phenyl)-amide 326723 5-Methoxy-6-((3R,5S)-3,4,5-trimethyl-piperazin-1-yl)-2,3-dihydro-indole-1-carboxylic acid (2-chloro-3-trifluoromethyl-phenyl)-amide 326724 5-Methoxy-6-((3R,5S)-3,4,5-trimethyl-piperazin-1-yl)-2,3-dihydro-indole-1-carboxylic acid 2-fluoro-3-trifluoromethyl-phenyl ester 326725 5-Methoxy-6-((3R,5S)-3,4,5-trimethyl-piperazin-1-yl)-2,3-dihydro-indole-1-carboxylic acid 2-chloro-3-trifluoromethyl-phenyl ester 326726 [5-Methoxy-6-((3R,5S)-3,4,5-trimethyl-piperazin-1-yl)-2,3-dihydro-indol-1-yl]-(2'-methyl-biphenyl-4-yl)-methanone 326727 1-{4'-[6-((3R,5S)-3,5-Dimethyl-piperazin-1-yl)-5-methoxy-2,3-dihydro-indole-1-carbonyl]-2-methyl-biphenyl-4-yl}-ethanone 326728 2-(2-Fluoro-3-trifluoromethyl-phenyl)-1-[5-methoxy-6-((3S,5R)-3,4,5-trimethyl-piperazin-1-yl)-2,3-dihydro-indol-1-yl]-ethanone 326730 5-Methoxy-6-((3S,5R)-3,4,5-trimethyl-piperazin-1-yl)-2,3-dihydro-indole-1-carboxylic acid (3-chloro-2-fluoro-phenyl)-amide 326735 [6-((3R,5S)-3,5-Dimethyl-piperazin-1-yl)-5-methoxy-2,3-dihydro-indol-1-yl]-[4-(2,5-dimethyl-pyridin-4-yl)-phenyl]-methanone 326736 [5-Methoxy-6-((3S,5R)-3,4,5-trimethyl-piperazin-1-yl)-2,3-dihydro-indol-1-yl]-[2'-methyl-4'-(5-methyl-[1,2,4]oxadiazol-3-yl)-biphenyl-4-yl]-methanone 326737 [6-((3S,5R)-3,5-Dimethyl-piperazin-1-yl)-5-methoxy-2,3-dihydro-indol-1-yl]-[2'-methyl-4'-(5-methyl-[1,2,4]oxadiazol-3-yl)-biphenyl-4-yl]-methanone 326738 1-(5-{4-[6-((3R,5S)-3,5-Dimethyl-piperazin-1-yl)-5-methoxy-2,3-dihydro-indole-1-carbonyl]-phenyl}-6-methyl-pyridin-2-yl)-pyrrolidin-2-one 326739 [6-((3S,5R)-3,5-Dimethyl-piperazin-1-yl)-5-methoxy-2,3-dihydro-indol-1-yl]-(2'-methyl-4'-pyrimidin-2-yl-biphenyl-4-yl)-methanone 326784 N-[(E)-(R)-1-(4-Chloro-benzyl)-3-(2-piperidin-1-yl-ethylcarbamoyl)-allyl]-N-methyl-3,5-bis-trifluoromethyl-benzamide 326965 4-(1-Benzyl-1H-indazol-5-ylamino)-5-ethyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid dimethylamide 326966 [4-(1-Benzyl-1H-indazol-5-ylamino)-5-ethyl-pyrrolo[2,1-f][1,2,4]triazin-6-yl]-carbamic acid benzyl ester 326967 [4-(1-Benzyl-1H-indazol-5-ylamino)-5-ethyl-pyrrolo[2,1-f][1,2,4]triazin-6-yl]-methanol 326973 (1-Benzyl-1H-indazol-5-yl)-(5-ethyl-6-ethylaminomethyl-pyrrolo[2,1-f][1,2,4]triazin-4-yl)-amine 326974 (1-Benzyl-1H-indazol-5-yl)-(6-ethoxymethyl-5-ethyl-pyrrolo[2,1-f][1,2,4]triazin-4-yl)-amine 326983 2-[4-(1-Benzyl-1H-indazol-5-ylamino)-5-ethyl-pyrrolo[2,1-f][1,2,4]triazin-6-yl]-acetamide 326991 [4-(1-Benzyl-1H-indazol-5-ylamino)-5-ethyl-pyrrolo[2,1-f][1,2,4]triazin-6-yl]-acetic acid 326992 4-(1-Benzyl-1H-indazol-5-ylamino)-5-ethyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid (3-imidazol-1-yl-propyl)-amide 326999 4-(1-Benzyl-1H-indazol-5-ylamino)-5-ethyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid 3-imidazol-1-yl-propyl ester 327000 [4-(1-Benzyl-1H-indazol-5-ylamino)-5-ethyl-pyrrolo[2,1-f][1,2,4]triazin-6-yl]-carbamic acid 2-imidazol-1-yl-ethyl ester 327032 4-(3-Chloro-4-fluoro-phenylamino)-5-ethyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid ethyl ester 327039 4-(3-Bromo-phenylamino)-5-ethyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid ethyl ester 327040 5-Ethyl-4-(1H-indazol-5-ylamino)-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid ethyl ester 327047 4-Benzylamino-5-ethyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid ethyl ester 327048 4-(1-Benzyl-1H-indazol-5-ylamino)-5-ethyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid ethyl ester 327055 5-Ethyl-4-(4-phenoxy-phenylamino)-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid ethyl ester 327056 4-(1-Benzyl-1H-indazol-5-ylamino)-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid ethyl ester 327061 4-(1-Benzyl-1H-indazol-5-ylamino)-5-methyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid ethyl ester 327062 4-(1-Benzyl-1H-indazol-5-ylamino)-5-isopropyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid ethyl ester 327069 4-(4-Chloro-phenyl)-piperazine-1-carboxylic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide 327070 4-(1-Benzyl-1H-indazol-5-ylamino)-5-propyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid ethyl ester 327077 4-(4-Fluoro-phenyl)-piperazine-1-carboxylic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide 327079 4-(1-Benzyl-1H-indazol-5-ylamino)-5-ethyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid 327082 4-Biphenyl-4-yl-piperazine-1-carboxylic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide 327083 4-(4-Trifluoromethyl-phenyl)-piperazine-1-carboxylic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide 327084 4-(1-Benzyl-1H-indazol-5-ylamino)-5-ethyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid amide 327085 4-(1-Benzyl-1H-indazol-5-ylamino)-5-ethyl-pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid methylamide 327090 4-(4-Methylsulfanyl-phenyl)-piperazine-1-carboxylic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide 327091 1-(2-Methoxy-phenyl)-piperidine-4-carboxylic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide 327098 2-Furan-2-yl-6-(3-methanesulfonyl-phenyl)-[1,2,4]triazolo[1,5-a]pyrazin-8-ylamine 327099 3-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-benzamide 327104 3,4-diarylpyrazoline derivative 327107 2-Furan-2-yl-6-pyridin-3-yl-[1,2,4]triazolo[1,5-a]pyrazin-8-ylamine 327111 3,4-diarylpyrazoline derivative 327112 3,4-diarylpyrazoline derivative 327115 2,6-Di-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-8-ylamine 327116 2-Furan-2-yl-6-naphthalen-1-yl-[1,2,4]triazolo[1,5-a]pyrazin-8-ylamine 327120 3,4-diarylpyrazoline derivative 327125 2-Furan-2-yl-6-quinolin-8-yl-[1,2,4]triazolo[1,5-a]pyrazin-8-ylamine 327126 2-Furan-2-yl-6-pyrimidin-5-yl-[1,2,4]triazolo[1,5-a]pyrazin-8-ylamine 327129 3,4-diarylpyrazoline derivative 327130 3,4-diarylpyrazoline derivative 327134 3-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-N-isopropyl-benzamide 327138 3,4-diarylpyrazoline derivative 327139 3,4-diarylpyrazoline derivative 327141 3-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-N,N-dimethyl-benzamide 327142 3-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-N,N-diethyl-benzamide 327146 3,4-diarylpyrazoline derivative 327147 3,4-diarylpyrazoline derivative 327148 2-Furan-2-yl-6-(3-isopropyl-phenyl)-[1,2,4]triazolo[1,5-a]pyrazin-8-ylamine 327149 6-(3-Amino-phenyl)-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-8-ylamine 327150 [3-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-phenyl]-(4-benzyl-piperazin-1-yl)-methanone 327153 3,4-diarylpyrazoline derivative 327154 3-(4-chlorophenyl)-N-methyl-4-phenyl-N'-(piperidin-1-ylsulfonyl)-4,5-dihydro-1H-pyrazole-1-carboximidamide 327156 N-[3-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-phenyl]-acetamide 327157 [3-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-phenyl]-(4-pyridin-4-yl-piperazin-1-yl)-methanone 327158 [3-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-phenyl]-morpholin-4-yl-methanone 327161 3,4-diarylpyrazoline derivative 327162 3,4-diarylpyrazoline derivative 327163 1-[3-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-phenyl]-ethanone 327164 2-Furan-2-yl-6-(3-nitro-phenyl)-[1,2,4]triazolo[1,5-a]pyrazin-8-ylamine 327165 [4-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-phenyl]-morpholin-4-yl-methanone 327166 3-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-N-[2-(4-hydroxy-phenyl)-ethyl]-benzamide 327171 6-(3-Dimethylamino-phenyl)-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-8-ylamine 327172 4-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-N-[2-(4-hydroxy-phenyl)-ethyl]-benzamide 327173 4-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-N-(3-imidazol-1-yl-propyl)-benzamide 327177 3-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-benzoic acid ethyl ester 327178 8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazine-6-carboxylic acid butylamide 327179 8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazine-6-carboxylic acid benzylamide 327186 3-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-benzonitrile 327187 8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazine-6-carboxylic acid benzyl-methyl-amide 327188 N-(4-hydroxyphenethyl)-8-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a]pyrazine-6-carboxamide 327195 2-Furan-2-yl-6-(3-trifluoromethyl-phenyl)-[1,2,4]triazolo[1,5-a]pyrazin-8-ylamine 327196 8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazine-6-carboxylic acid (3-phenyl-propyl)-amide 327204 [3-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-phenyl]-methanol 327214 2-Furan-2-yl-6-(3-methoxy-phenyl)-[1,2,4]triazolo[1,5-a]pyrazin-8-ylamine 327232 (4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Thr-NH2 327248 (4-amino)-D-Phe-c[Cys-(3-iodo)-Tyr-D-Trp-Lys-Val-Cys]-Thr-NH2 327251 (4-amino-3-iodo)-D-Phe-c[Cys-(3-iodo)-Tyr-D-Trp-Lys-Val-Cys]-Thr-NH2 327272 (4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Asp-NH2 327277 (4-amino-3-iodo)-D-Phe-c[Cys-(3-iodo)-Tyr-D-Trp-Lys-Val-Cys]-Asp-NH2 327286 4-fluoro-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)benzamide 327291 N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-4-fluorobenzamide 327292 6-fluoro-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)nicotinamide 327296 (4-amino-3-iodo)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Thr-NH2 327299 N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-6-fluoronicotinamide 327300 6-Fluoro-pyridine-2-carboxylic acid {4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-amide 327307 6-Fluoro-pyridine-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide 327308 4-Fluoro-N-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-benzenesulfonamide 327310 (4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-D-Thr-NH2 327316 H-D-Phe-Cys-Tyr-D-Trp-Lys-Val-Cys-Thr-NH2 327318 D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Asp-NH2 327319 N-{4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-butyl}-4-fluoro-benzenesulfonamide 327333 (4-amino-3-iodo)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Asp-NH2 327339 (4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-D-Asp-NH2 327503 5-Methoxy-2-methyl-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole 327513 SID26755027 327527 (LTB4-(Csa)4)2-Glu-H Conjugate 327551 (2S,4aS,6aR,7R,9S,10aS,10bR)-9-acetoxy-2-(furan-3-yl)-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylic acid 327552 (3S,4aR,4bS,6S,8R,8aR,10aR)-6-Acetoxy-3-furan-3-yl-4a,8a-dimethyl-1,5-dioxo-dodecahydro-2-oxa-phenanthrene-8-carboxylic acid ethyl ester 327591 (6,7-Dimethoxy-quinazolin-4-yl)-[3-methyl-4-(pyridin-2-ylmethoxy)-phenyl]-amine 327598 [3-Chloro-4-(pyridin-2-ylmethoxy)-phenyl]-[7-methoxy-5-(4-methyl-piperidin-1-yloxy)-quinazolin-4-yl]-amine 327605 [3-Chloro-4-(3-fluoro-benzyloxy)-phenyl]-[5-(1-methyl-piperidin-4-yloxy)-quinazolin-4-yl]-amine 327606 (3-Chloro-4-methoxy-phenyl)-[5-(1-methyl-piperidin-4-yloxy)-quinazolin-4-yl]-amine 327619 [3-Chloro-4-(pyridin-2-ylmethoxy)-phenyl]-[5-(tetrahydro-pyran-4-yloxy)-quinazolin-4-yl]-amine 327620 N-(3-chloro-4-(pyridin-2-ylmethoxy)phenyl)-5-(1-methylpiperidin-4-yloxy)quinazolin-4-amine 327627 [3-Chloro-4-(pyrazin-2-ylmethoxy)-phenyl]-[5-(1-methyl-piperidin-4-yloxy)-quinazolin-4-yl]-amine 327628 [3-Chloro-4-(thiazol-4-ylmethoxy)-phenyl]-[5-(1-methyl-piperidin-4-yloxy)-quinazolin-4-yl]-amine 327632 [5-(1-Methyl-piperidin-4-yloxy)-quinazolin-4-yl]-[4-(pyridin-2-ylmethoxy)-phenyl]-amine 327633 [3-Chloro-4-(pyridin-2-ylmethoxy)-phenyl]-(5-methoxy-quinazolin-4-yl)-amine 327642 Acetic acid (3S,4aR,4bS,6S,8R,8aR,10aS)-8-cyclopropylcarbamoyl-3-furan-3-yl-4a,8a-dimethyl-1,5-dioxo-dodecahydro-2-oxa-phenanthren-6-yl ester 327643 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-5-methoxy-2-[(pyridin-2-ylmethyl)-amino]-benzamide 327653 Pyridine-2-carboxylic acid [2-(1-benzo[1,3]dioxol-5-ylmethyl-piperidin-4-ylcarbamoyl)-4-chloro-phenyl]-amide 327654 N-(1-benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-5-chloro-2-[(thiazol-2-ylmethyl)amino]benzamide 327660 2-[((3S,4aR,4bS,6S,8R,8aR,10aR)-6-Acetoxy-3-furan-3-yl-4a,8a-dimethyl-1,5-dioxo-dodecahydro-2-oxa-phenanthrene-8-carbonyl)-amino]-propionic acid benzyl ester 327662 [((3S,4aR,4bS,6S,8R,8aR,10aR)-6-Acetoxy-3-furan-3-yl-4a,8a-dimethyl-1,5-dioxo-dodecahydro-2-oxa-phenanthrene-8-carbonyl)-amino]-acetic acid benzyl ester 327666 1-((3S,4aR,4bS,6S,8R,8aR,10aR)-6-Acetoxy-3-furan-3-yl-4a,8a-dimethyl-1,5-dioxo-dodecahydro-2-oxa-phenanthrene-8-carbonyl)-pyrrolidine-2-carboxylic acid benzyl ester 327669 5-Chloro-N-(1-naphthalen-2-ylmethyl-piperidin-4-yl)-2-[(thiazol-2-ylmethyl)-amino]-benzamide 327670 5-Chloro-N-(1-quinolin-6-ylmethyl-piperidin-4-yl)-2-[(thiazol-2-ylmethyl)-amino]-benzamide 327676 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-3-chloro-benzamide 327677 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-5-chloro-2-hydroxy-benzamide 327678 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-2,5-dichloro-nicotinamide 327679 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-5-chloro-2-isopropylamino-nicotinamide 327683 2-Amino-N-(1-benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-5-chloro-benzamide 327684 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-5-chloro-2-methylamino-benzamide 327685 5-Chloro-N-[1-(2,3-dihydro-benzofuran-5-ylmethyl)-piperidin-4-yl]-2-isopropylamino-nicotinamide 327686 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-5-chloro-2-cyclobutylamino-nicotinamide 327690 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-5-chloro-2-methanesulfonylamino-benzamide 327691 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-2-methanesulfonylamino-5-methoxy-benzamide 327693 5-Chloro-N-[1-(4-chloro-benzyl)-piperidin-4-yl]-2-cyclobutylamino-nicotinamide 327694 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-5-chloro-2-isobutylamino-nicotinamide 327699 N-[1-(4-Chloro-benzyl)-piperidin-4-yl]-2-methanesulfonylamino-5-methoxy-benzamide 327700 N-[1-(4-Chloro-benzyl)-piperidin-4-yl]-2-(3-isopropyl-ureido)-5-methoxy-benzamide 327701 5-Chloro-N-[1-(3-fluoro-4-methoxy-benzyl)-piperidin-4-yl]-2-isobutylamino-nicotinamide 327702 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-5-chloro-2-(cyclopropylmethyl-amino)-nicotinamide 327707 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-2-(cyclopropylmethyl-amino)-5-methoxy-benzamide 327708 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-2-(cyclohexylmethyl-amino)-5-methoxy-benzamide 327709 5-Chloro-N-[1-(4-chloro-benzyl)-piperidin-4-yl]-2-(cyclopropylmethyl-amino)-nicotinamide 327710 5-Chloro-N-[1-(4-chloro-benzyl)-piperidin-4-yl]-2-[(furan-2-ylmethyl)-amino]-nicotinamide 327713 (3S,4aR,4bS,6S,8R,8aR,10aR)-6-Acetoxy-3-furan-3-yl-4a,8a-dimethyl-1,5-dioxo-dodecahydro-2-oxa-phenanthrene-8-carboxylic acid pent-4-ynyl ester 327714 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-5-methoxy-2-[(tetrahydro-furan-3-ylmethyl)-amino]-benzamide 327715 N-(1-Benzyl-piperidin-4-yl)-5-chloro-2-(4-methoxy-benzylamino)-nicotinamide 327716 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-5-chloro-2-[(1H-imidazol-2-ylmethyl)-amino]-nicotinamide 327720 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-5-methoxy-2-[(pyrimidin-5-ylmethyl)-amino]-benzamide 327723 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-5-chloro-2-[(1H-imidazol-4-ylmethyl)-amino]-nicotinamide 327727 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-2-[(1H-imidazol-2-ylmethyl)-amino]-5-methoxy-benzamide 327728 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-5-chloro-2-[(thiazol-4-ylmethyl)-amino]-nicotinamide 327729 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-5-chloro-2-[(thiazol-2-ylmethyl)-amino]-nicotinamide 327731 (3S,4aR,4bS,6S,8R,8aR,10aR)-6-Acetoxy-3-furan-3-yl-4a,8a-dimethyl-1,5-dioxo-dodecahydro-2-oxa-phenanthrene-8-carboxylic acid methoxymethyl ester 327732 (3S,4aR,4bS,6S,8R,8aR,10aS)-6-Acetoxy-3-furan-3-yl-4a,8a-dimethyl-1,5-dioxo-dodecahydro-2-oxa-phenanthrene-8-carboxylic acid methoxymethyl ester 327733 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-2-[(3H-imidazol-4-ylmethyl)-amino]-5-methoxy-benzamide 327734 N-(1-benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-5-chloro-2-(2-isopropoxyethylamino)nicotinamide 327735 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-5-chloro-2-(3-isopropoxy-propylamino)-nicotinamide 327738 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-5-methoxy-2-[(3-methyl-3H-imidazol-4-ylmethyl)-amino]-benzamide 327739 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-5-chloro-2-{[(R)-1-(tetrahydro-furan-2-yl)methyl]-amino}-nicotinamide 327744 2-[(3H-Imidazol-4-ylmethyl)-amino]-5-methoxy-N-(1-naphthalen-2-ylmethyl-piperidin-4-yl)-benzamide 327746 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-2-(2-isopropoxy-ethylamino)-5-thiophen-2-yl-nicotinamide 327749 2-[(3H-Imidazol-4-ylmethyl)-amino]-5-methoxy-N-(1-quinolin-6-ylmethyl-piperidin-4-yl)-benzamide 327750 6-(2-Isopropoxy-ethylamino)-[3,4']bipyridinyl-5-carboxylic acid (1-benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-amide 327791 N-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)-2-[(3H-imidazol-4-ylmethyl)-amino]-benzamide 327792 N-[1-(4-Acetyl-benzyl)-piperidin-4-yl]-5-chloro-2-[(3H-imidazol-4-ylmethyl)-amino]-benzamide 327793 N-Cyclohexyl-2-(7-methyl-4-oxo-1,4-dihydro-[1,8]naphthyridin-3-yl)-acetamide 327794 N-Benzyl-2-(7-methyl-4-oxo-1,4-dihydro-[1,8]naphthyridin-3-yl)-acetamide 327802 7-Amino-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid 4-chloro-benzylamide 327803 7-Amino-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid benzylamide 327818 7-Chloro-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid benzylamide 327820 7-Bromo-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid benzylamide 327834 3-Benzyl-7-methyl-[1,8]naphthyridin-4-ol 327835 4-Oxo-7-phenethylamino-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid benzylamide 327841 5-Azido-6-benzyl-2-methyl-[1,8]naphthyridine 327843 3-Benzyl-7-methyl-[1,8]naphthyridine-4-thiol 327844 7-Dimethylamino-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid benzylamide 327849 (3-Benzyl-7-methyl-[1,8]naphthyridin-4-yl)-hydrazine 327850 3-(2-Chloro-benzyl)-7-methyl-[1,8]naphthyridin-4-ol 327851 4-Oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid benzylamide 327852 7-Benzylamino-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid benzylamide 327860 7-Methyl-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid benzylamide 327865 7-Methyl-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid 4-chloro-benzylamide 327878 7-Methyl-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid (4-methyl-piperazin-1-yl)-amide 327885 7-Methyl-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid cyclohexylamide 327886 7-Methyl-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid (4-methyl-cyclohexyl)-amide 327887 7-Methyl-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid (3-methyl-butyl)-amide 327894 7-Methyl-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid 4-fluoro-benzylamide 327895 7-Methyl-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid 4-methoxy-benzylamide 327903 7-Methyl-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid 4-methyl-benzylamide 327904 7-Methyl-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid phenethyl-amide 327912 7-Methyl-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid (furan-2-ylmethyl)-amide 327913 7-Methyl-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid (1-phenyl-ethyl)-amide 327921 7-Methyl-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid 4-nitro-benzylamide 327929 7-Methyl-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid 4-amino-benzylamide 327937 7-Methyl-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid 4-benzoylamino-benzylamide 327942 1-(4-{5-[4-(2,2-Dimethyl-propyl)-phenyl]-[1,2,4]oxadiazol-3-yl}-benzyl)-azetidine-3-carboxylic acid 327956 1-{4-[5-(4-Ethoxy-phenyl)-[1,2,4]oxadiazol-3-yl]-benzyl}-azetidine-3-carboxylic acid 327962 1-{4-[5-(4-tert-Butyl-phenyl)-[1,2,4]oxadiazol-3-yl]-benzyl}-azetidine-3-carboxylic acid 327964 1-{4-[5-(4-Butyl-phenyl)-[1,2,4]oxadiazol-3-yl]-benzyl}-azetidine-3-carboxylic acid 327983 1-{4-[5-(4-Isopropoxy-phenyl)-[1,2,4]oxadiazol-3-yl]-benzyl}-azetidine-3-carboxylic acid 327986 1-{4-[5-(4-Cyclohexyl-phenyl)-[1,2,4]oxadiazol-3-yl]-benzyl}-azetidine-3-carboxylic acid 328004 1-{4-[5-(4-Hexyl-phenyl)-[1,2,4]oxadiazol-3-yl]-benzyl}-azetidine-3-carboxylic acid 328016 1-{4-[5-(4-Cyclopropyl-phenyl)-[1,2,4]oxadiazol-3-yl]-benzyl}-azetidine-3-carboxylic acid 328031 1-(4-{5-[4-(1,1-Dimethyl-propyl)-phenyl]-[1,2,4]oxadiazol-3-yl}-benzyl)-azetidine-3-carboxylic acid 328064 1-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)benzyl)azetidine-3-carboxylic acid 328068 1-{4-[5-(4-Cyclobutyl-phenyl)-[1,2,4]oxadiazol-3-yl]-benzyl}-azetidine-3-carboxylic acid 328071 1-{4-[5-(4-tert-Butyl-phenyl)-[1,3,4]oxadiazol-2-yl]-benzyl}-azetidine-3-carboxylic acid 328082 1-{4-[3-(4-tert-Butyl-phenyl)-[1,2,4]oxadiazol-5-yl]-benzyl}-azetidine-3-carboxylic acid 328100 1-{4-[5-(4-Propyl-phenyl)-[1,2,4]oxadiazol-3-yl]-benzyl}-azetidine-3-carboxylic acid 328106 1-{4-[5-(4-Cyclopentyl-phenyl)-[1,2,4]oxadiazol-3-yl]-benzyl}-azetidine-3-carboxylic acid 328110 (E)-N-(2-{[(2-Dimethylamino-ethyl)-methyl-amino]-methyl}-3-methyl-quinolin-6-yl)-3-(4-trifluoromethoxy-phenyl)-acrylamide 328111 (E)-N-(2-{[(2-Dimethylamino-ethyl)-methyl-amino]-methyl}-4-ethyl-quinolin-6-yl)-3-(4-trifluoromethoxy-phenyl)-acrylamide 328114 N-[4-Methyl-2-(4-methyl-piperazin-1-yl)-quinolin-6-yl]-3-p-tolyl-acrylamide 328115 SID24267169 328116 (E)-N-[2-(4-Ethyl-piperazin-1-ylmethyl)-4-methyl-quinolin-6-yl]-N-methyl-3-(4-trifluoromethoxy-phenyl)-acrylamide 328117 (E)-N-(3,4-Difluoro-benzyl)-N-{2-[(2-dimethylamino-ethyl)-methyl-amino]-4-methyl-quinolin-6-yl}-3-(4-trifluoromethoxy-phenyl)-acrylamide 328118 2-(2,4-Dichloro-phenoxy)-N-(4-methyl-2-morpholin-4-yl-quinolin-6-yl)-acetamide 328122 (E)-3-(3-Chloro-phenyl)-N-[4-methyl-2-(4-methyl-piperazin-1-yl)-quinolin-6-yl]-acrylamide 328123 N-(4-Methyl-2-morpholin-4-yl-quinolin-6-yl)-2-(4-trifluoromethoxy-phenoxy)-acetamide 328124 1-(4-{5-[4-((S)-3,3-Difluoro-cyclopentyl)-phenyl]-[1,2,4]oxadiazol-3-yl}-benzyl)-azetidine-3-carboxylic acid 328128 [5-Fluoro-1-(3-fluoro-benzenesulfonyl)-2-methyl-1H-indol-3-yl]-acetic acid 328129 2-(2,4-Dichloro-phenoxy)-N-(4-methyl-2-piperazin-1-yl-quinolin-6-yl)-acetamide 328133 [5-Fluoro-1-(4-methanesulfonyl-benzenesulfonyl)-2-methyl-1H-indol-3-yl]-acetic acid 328135 (E)-N-[2-((3S,5R)-3,5-Dimethyl-piperazin-1-yl)-4-methyl-quinolin-6-yl]-3-(4-trifluoromethoxy-phenyl)-acrylamide 328136 N-[2-(2,5-Diaza-bicyclo[2.2.1]hept-2-yl)-4-methyl-quinolin-6-yl]-2-(4-trifluoromethoxy-phenoxy)-acetamide 328143 N-[4-Methyl-2-(4-pyrrolidin-1-yl-piperidin-1-yl)-quinolin-6-yl]-2-(4-trifluoromethoxy-phenoxy)-acetamide 328149 2-(3,4-Dichloro-phenyl)-N-[2-(4-ethyl-piperazin-1-yl)-4-methyl-quinolin-6-yl]-acetamide 328150 SID24267167 328151 (E)-N-(4-Methyl-2-piperazin-1-yl-quinolin-6-yl)-3-(4-trifluoromethoxy-phenyl)-acrylamide 328152 (E)-N-(2-[1,4]Diazepan-1-yl-4-methyl-quinolin-6-yl)-3-(4-trifluoromethoxy-phenyl)-acrylamide 328160 2-Thiophen-2-yl-quinoline-4-carboxylic acid [2-(4-ethyl-piperazin-1-yl)-4-methyl-quinolin-6-yl]-amide 328165 1-(4-{5-[4-((R)-3,3-Difluoro-cyclopentyl)-phenyl]-[1,2,4]oxadiazol-3-yl}-benzyl)-azetidine-3-carboxylic acid 328168 GNF-Pf-1550 328170 1-[4-(5-Biphenyl-4-yl-[1,2,4]oxadiazol-3-yl)-benzyl]-azetidine-3-carboxylic acid 328178 (1-Benzenesulfonyl-5-fluoro-2-methyl-1H-indol-3-yl)-acetic acid 328184 (E)-N-[2-(4-Ethyl-piperazin-1-yl)-4-methyl-quinolin-6-yl]-3-(4-isopropoxy-phenyl)-acrylamide 328185 (E)-3-[4-(3-Methyl-butoxy)-phenyl]-N-[4-methyl-2-(4-methyl-piperazin-1-yl)-quinolin-6-yl]-acrylamide 328192 1-[2-(4-Ethyl-piperazin-1-yl)-4-methyl-quinolin-6-yl]-3-(4-methoxy-benzyl)-urea 328197 N-(4-Fluoro-phenyl)-N-methyl-N'-[4-methyl-2-(4-methyl-piperazin-1-yl)-quinolin-6-yl]-succinamide 328198 N-(3-Chloro-4-fluoro-phenyl)-N'-[2-(4-ethyl-piperazin-1-yl)-4-methyl-quinolin-6-yl]-succinamide 328200 1-(4-{5-[4-(3,3,3-Trifluoro-propyl)-phenyl]-[1,2,4]oxadiazol-3-yl}-benzyl)-azetidine-3-carboxylic acid 328204 2-(2,4-Dichloro-phenoxy)-N-(4-methyl-2-piperidin-1-yl-quinolin-6-yl)-acetamide 328205 (E)-3-(4-Methoxy-phenyl)-N-(4-methyl-2-morpholin-4-yl-quinolin-6-yl)-acrylamide 328211 (E)-N-[2-(4-Ethyl-piperazin-1-yl)-4-methyl-quinolin-6-yl]-3-(4-trifluoromethoxy-phenyl)-acrylamide 328212 (E)-N-[2-(4-Ethyl-piperazin-1-ylmethyl)-quinolin-6-yl]-3-(4-trifluoromethoxy-phenyl)-acrylamide 328215 [5-Fluoro-1-(4-fluoro-benzenesulfonyl)-2-methyl-1H-indol-3-yl]-acetic acid 328217 [5-Fluoro-2-methyl-1-(toluene-4-sulfonyl)-1H-indol-3-yl]-acetic acid 328218 (E)-N-(2-{[(2-Dimethylamino-ethyl)-methyl-amino]-methyl}-quinolin-6-yl)-3-(4-trifluoromethoxy-phenyl)-acrylamide 328221 (E)-N-{2-[(2-Dimethylamino-ethyl)-methyl-amino]-quinolin-6-yl}-3-p-tolyl-acrylamide 328222 (E)-N-[2-(4-Ethyl-piperazin-1-ylmethyl)-3-methyl-quinolin-6-yl]-3-(4-trifluoromethoxy-phenyl)-acrylamide 328262 [1-(1,2-Dimethyl-1H-imidazole-4-sulfonyl)-5-fluoro-2-methyl-1H-indol-3-yl]-acetic acid 328291 N-[2-(4-Amino-piperidin-1-yl)-4-methyl-quinolin-6-yl]-2-(4-trifluoromethoxy-phenoxy)-acetamide 328292 N-(4-Methyl-2-piperidin-1-yl-quinolin-6-yl)-2-(4-trifluoromethoxy-phenoxy)-acetamide 328295 [(S)-9-(4-Chloro-phenylsulfanyl)-6-fluoro-2,3-dihydro-1H-pyrrolo[1,2-a]indol-1-yl]-acetic acid 328298 2-(2,4-Dichloro-phenoxy)-N-{2-[(2-dimethylamino-ethyl)-methyl-amino]-4-methyl-quinolin-6-yl}-acetamide 328299 2-(2,4-Dichloro-phenoxy)-N-{4-methyl-2-[methyl-(2-methylamino-ethyl)-amino]-quinolin-6-yl}-acetamide 328300 [1-(Butane-1-sulfonyl)-5-fluoro-2-methyl-1H-indol-3-yl]-acetic acid 328304 [1-(2,5-Dichloro-benzenesulfonyl)-5-fluoro-2-methyl-1H-indol-3-yl]-acetic acid 328305 (E)-N-[2-(2-Dimethylamino-ethylamino)-4-methyl-quinolin-6-yl]-3-(4-trifluoromethoxy-phenyl)-acrylamide 328311 (E)-N-[2-(2-Dimethylamino-1-methyl-ethylamino)-4-methyl-quinolin-6-yl]-3-(4-trifluoromethoxy-phenyl)-acrylamide 328317 N-{2-[(1-Ethyl-pyrrolidin-2-ylmethyl)-amino]-4-methyl-quinolin-6-yl}-2-(4-trifluoromethoxy-phenoxy)-acetamide 328324 N-[2-(3-Dimethylamino-propylamino)-4-methyl-quinolin-6-yl]-2-(4-trifluoromethoxy-phenoxy)-acetamide 328325 2-(2,4-Dichloro-phenoxy)-N-[2-(2-dimethylamino-ethoxy)-4-methyl-quinolin-6-yl]-acetamide 328332 (E)-N-[2-(2-Dimethylamino-ethoxy)-4-methyl-quinolin-6-yl]-3-(4-trifluoromethoxy-phenyl)-acrylamide 328333 2-(2,4-Dichloro-phenoxy)-N-{2-[(2-hydroxy-ethyl)-methyl-amino]-4-methyl-quinolin-6-yl}-acetamide 328340 (E)-N-{2-[(2-Hydroxy-ethyl)-methyl-amino]-4-methyl-quinolin-6-yl}-3-(4-trifluoromethoxy-phenyl)-acrylamide 328341 Acetic acid 2-({6-[2-(3,4-dichloro-phenoxy)-acetylamino]-4-methyl-quinolin-2-yl}-methyl-amino)-ethyl ester 328348 [5-Fluoro-1-(4-methoxy-benzenesulfonyl)-2-methyl-1H-indol-3-yl]-acetic acid 328351 (4-Fluoro-naphthalen-1-yl)-[1-(1-methyl-piperidin-2-ylmethyl)-1H-indol-3-yl]-methanone 328352 (4-Bromo-naphthalen-1-yl)-[1-(1-methyl-piperidin-2-ylmethyl)-1H-indol-3-yl]-methanone 328359 (4-Methoxy-naphthalen-1-yl)-[1-(1-methyl-piperidin-2-ylmethyl)-1H-indol-3-yl]-methanone 328367 (4-Hydroxy-naphthalen-1-yl)-[1-(1-methyl-piperidin-2-ylmethyl)-1H-indol-3-yl]-methanone 328368 4-[1-(1-Methyl-piperidin-2-ylmethyl)-1H-indole-3-carbonyl]-naphthalene-1-carbonitrile 328375 [4-(2-Hydroxy-ethyl)-naphthalen-1-yl]-[1-(1-methyl-piperidin-2-ylmethyl)-1H-indol-3-yl]-methanone 328376 (6-Hydroxy-naphthalen-1-yl)-[1-(1-methyl-piperidin-2-ylmethyl)-1H-indol-3-yl]-methanone 328383 1-(1-Methyl-piperidin-2-ylmethyl)-1H-indole-3-carboxylic acid naphthalen-1-ylamide 328384 [1-(1-Methyl-piperidin-2-ylmethyl)-1H-indol-3-yl]-(octahydro-quinolin-1-yl)-methanone 328389 [1-(1-Methyl-piperidin-2-ylmethyl)-1H-indazol-3-yl]-naphthalen-1-yl-methanone 328390 [1-(1-Methyl-piperidin-2-ylmethyl)-1H-indol-3-yl]-(4-nitro-naphthalen-1-yl)-methanone 328397 (2-Methyl-naphthalen-1-yl)-[1-(1-methyl-piperidin-2-ylmethyl)-1H-indol-3-yl]-methanone 328398 (2-Iodo-phenyl)-[1-(1-methyl-piperidin-2-ylmethyl)-1H-indol-3-yl]-methanone 328426 6-(4-(4-fluorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 328432 2,2-Dimethyl-propionic acid 2-hydroxymethyl-4-[3-isobutyl-5-methyl-hex-(E)-ylidene]-tetrahydro-furan-2-ylmethyl ester 328438 5-(2,2-Dimethyl-propoxymethyl)-5-hydroxymethyl-3-[3-isobutyl-5-methyl-hex-(E)-ylidene]-dihydro-furan-2-one 328439 5-(2,2-Dimethyl-propoxymethyl)-5-hydroxymethyl-3-[3-isobutyl-5-methyl-hex-(Z)-ylidene]-dihydro-furan-2-one 328446 2,2-Dimethyl-propionic acid 2-hydroxymethyl-4-[3-isobutyl-5-methyl-hex-(E)-ylidene]-5-thioxo-tetrahydro-furan-2-ylmethyl ester 328454 2,2-Dimethyl-thiopropionic acid O-{2-hydroxymethyl-4-[3-isobutyl-5-methyl-hex-(E)-ylidene]-5-oxo-tetrahydro-furan-2-ylmethyl} ester 328469 (4-Methyl-naphthalen-1-yl)-[1-(1-methyl-piperidin-2-ylmethyl)-1H-indol-3-yl]-methanone 328589 (3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(4-methyl-pyridin-2-yl)-vinyl]-decahydro-naphtho[2,3-c]furan-1-one 328590 2-{6-[(E)-2-((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-1-oxo-dodecahydro-naphtho[2,3-c]furan-4-yl)-vinyl]-pyridin-3-yl}-benzoic acid ethyl ester 328596 (3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(5-methyl-pyridin-2-yl)-vinyl]-decahydro-naphtho[2,3-c]furan-1-one 328597 (3R,3aS,4S,4aR,8aS,9aR)-4-(2-(6-ethylpyridin-2-yl)vinyl)-3-methyl-decahydronaphtho[2,3-c]furan-1(3H)-one 328598 (3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(2-Methoxy-phenyl)-pyridin-2-yl]-vinyl}-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 328599 (3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(2-Fluoro-phenyl)-pyridin-2-yl]-vinyl}-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 328605 (3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(6-vinyl-pyridin-2-yl)-vinyl]-decahydro-naphtho[2,3-c]furan-1-one 328606 (3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(6-propyl-pyridin-2-yl)-vinyl]-decahydro-naphtho[2,3-c]furan-1-one 328607 (3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(2-Chloro-phenyl)-pyridin-2-yl]-vinyl}-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 328608 (3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(3-Fluoro-phenyl)-pyridin-2-yl]-vinyl}-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 328613 (3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(6-Butyl-pyridin-2-yl)-vinyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 328614 (3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(6-Hexyl-pyridin-2-yl)-vinyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 328615 (3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(3-Chloro-phenyl)-pyridin-2-yl]-vinyl}-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 328617 (3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(3-Bromo-phenyl)-pyridin-2-yl]-vinyl}-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 328622 (3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(6-Isopropyl-pyridin-2-yl)-vinyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 328623 (3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(6-Isobutyl-pyridin-2-yl)-vinyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 328624 3-{6-[(E)-2-((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-1-oxo-dodecahydro-naphtho[2,3-c]furan-4-yl)-vinyl]-pyridin-3-yl}-benzonitrile 328625 (3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(5-m-tolyl-pyridin-2-yl)-vinyl]-decahydro-naphtho[2,3-c]furan-1-one 328630 (3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(6-Cyclopropyl-pyridin-2-yl)-vinyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 328631 (3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(6-methylamino-pyridin-2-yl)-vinyl]-decahydro-naphtho[2,3-c]furan-1-one 328632 (3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(3-Isopropyl-phenyl)-pyridin-2-yl]-vinyl}-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 328633 (3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(3-Methoxy-phenyl)-pyridin-2-yl]-vinyl}-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 328639 (3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(6-Hydroxymethyl-pyridin-2-yl)-vinyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 328640 (3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(6-Methoxymethyl-pyridin-2-yl)-vinyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 328641 3-{6-[(E)-2-((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-1-oxo-dodecahydro-naphtho[2,3-c]furan-4-yl)-vinyl]-pyridin-3-yl}-benzenesulfonamide 328643 DTPA Conjugate 328646 (3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(6-Benzyl-pyridin-2-yl)-vinyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 328648 (3R,3aS,4S,4aR,8aS,9aR,E)-3-methyl-4-(2-(5-(3-(trifluoromethyl)phenyl)pyridin-2-yl)vinyl)-decahydronaphtho[2,3-c]furan-1(3H)-one 328649 4-{1-[((E)-3-Phenyl)-allyl]-piperidin-4-ylamino}-chromen-2-one 328655 (3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(5-Benzyl-pyridin-2-yl)-vinyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 328657 6-Chloro-4-[1-(3-phenyl-allyl)-piperidin-4-ylamino]-chromen-2-one 328658 6-Methoxy-4-[1-(3-phenyl-allyl)-piperidin-4-ylamino]-chromen-2-one 328664 (3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(5-Methoxy-pyridin-2-yl)-vinyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 328665 (3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(5-Benzyloxy-pyridin-2-yl)-vinyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 328666 6-Chloro-4-(1-naphthalen-2-ylmethyl-piperidin-4-ylamino)-chromen-2-one 328667 4-(1-Benzo[1,3]dioxol-5-ylmethyl-piperidin-4-ylamino)-6-chloro-chromen-2-one 328672 (3R,3aS,4S,4aR,8aS,9aR)-3-methyl-4-(2-(6-methylpyridin-2-yl)vinyl)-decahydronaphtho[2,3-c]furan-1(3H)-one 328673 (3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[(E)-2-(6-methyl-pyridin-2-yl)-vinyl]-decahydro-naphtho[2,3-c]furan-1-one 328674 6-Chloro-4-[1-(2,3-dihydro-benzofuran-5-ylmethyl)-piperidin-4-ylamino]-chromen-2-one 328675 6-Chloro-4-[1-(2,2-difluoro-benzo[1,3]dioxol-5-ylmethyl)-piperidin-4-ylamino]-chromen-2-one 328679 Dipropyl-(4,5,6,7-tetrahydro-pyrazolo[1,5-a]pyridin-5-yl)-amine 328680 Dipropyl-(R)-4,5,6,7-tetrahydro-pyrazolo[1,5-a]pyridin-5-yl-amine 328681 (3S,3aR,4R,4aS,8aR,9aS)-4-[(E)-2-(6-Ethyl-pyridin-2-yl)-vinyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 328682 4-(1-Benzooxazol-5-ylmethyl-piperidin-4-ylamino)-6-chloro-chromen-2-one 328683 4-(1-Benzooxazol-6-ylmethyl-piperidin-4-ylamino)-6-chloro-chromen-2-one 328686 Dipropyl-(S)-4,5,6,7-tetrahydro-pyrazolo[1,5-a]pyridin-5-yl-amine 328687 (3-Chloro-4,5,6,7-tetrahydro-pyrazolo[1,5-a]pyridin-5-yl)-dipropyl-amine 328688 5-Propylamino-4,5,6,7-tetrahydro-pyrazolo[1,5-a]pyridine-3-carboxylic acid methyl ester 328689 (3R,3aS,4S,4aR,8aS,9aR,E)-3-methyl-4-(2-(5-phenylpyridin-2-yl)vinyl)-decahydronaphtho[2,3-c]furan-1(3H)-one 328690 (3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(5-p-tolyl-pyridin-2-yl)-vinyl]-decahydro-naphtho[2,3-c]furan-1-one 328691 6-Chloro-4-[1-(1H-indol-5-ylmethyl)-piperidin-4-ylamino]-chromen-2-one 328692 4-(1-Benzo[b]thiophen-5-ylmethyl-piperidin-4-ylamino)-6-chloro-chromen-2-one 328696 5-Dipropylamino-4,5,6,7-tetrahydro-pyrazolo[1,5-a]pyridine-3-carboxylic acid methyl ester 328697 (5-Dipropylamino-4,5,6,7-tetrahydro-pyrazolo[1,5-a]pyridin-3-yl)-methanol 328698 5-Dipropylamino-4,5,6,7-tetrahydro-pyrazolo[1,5-a]pyridine-3-carbaldehyde 328699 (3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(4-Methoxy-phenyl)-pyridin-2-yl]-vinyl}-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 328700 (3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(4-Fluoro-phenyl)-pyridin-2-yl]-vinyl}-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 328702 6-Chloro-4-[1-(1H-indol-6-ylmethyl)-piperidin-4-ylamino]-chromen-2-one 328703 6-Chloro-4-[1-(1-methyl-1H-indol-6-ylmethyl)-piperidin-4-ylamino]-chromen-2-one 328708 (3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(4-Chloro-phenyl)-pyridin-2-yl]-vinyl}-3-methyl-decahydro-naphtho[2,3-c]furan-1-one 328710 4-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-ylamino)-6-methoxy-2H-chromen-2-one 328714 (3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-((E)-2-pyridin-2-yl-vinyl)-decahydro-naphtho[2,3-c]furan-1-one 328715 (3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(5-o-tolyl-pyridin-2-yl)-vinyl]-decahydro-naphtho[2,3-c]furan-1-one 328716 (3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-{(E)-2-[5-(2-trifluoromethyl-phenyl)-pyridin-2-yl]-vinyl}-decahydro-naphtho[2,3-c]furan-1-one 328720 4-(2,4-Dichloro-5-methoxy-phenylamino)-8-methoxy-7-(2-morpholin-4-yl-ethoxy)-benzo[g]quinoline-3-carbonitrile 328721 [6-Iodo-1-(1-methyl-piperidin-2-ylmethyl)-1H-indol-3-yl]-naphthalen-1-yl-methanone 328732 (4-Iodo-naphthalen-1-yl)-[1-(1-methyl-piperidin-2-ylmethyl)-1H-indol-3-yl]-methanone 328737 4-(2,4-Dichloro-5-methoxy-phenylamino)-8-methoxy-7-[2-(4-methyl-piperazin-1-yl)-ethoxy]-benzo[g]quinoline-3-carbonitrile 328741 (3-Iodo-phenyl)-[2-methyl-1-(1-methyl-piperidin-2-ylmethyl)-1H-indol-3-yl]-methanone 328744 4-(2,4-Dichloro-5-methoxy-phenylamino)-7-[2-(4-hydroxy-piperidin-1-yl)-ethoxy]-8-methoxy-benzo[g]quinoline-3-carbonitrile 328752 4-(2-Chloro-5-methoxy-4-methyl-phenylamino)-8-methoxy-7-(2-morpholin-4-yl-ethoxy)-benzo[g]quinoline-3-carbonitrile 328753 8-Methoxy-7-[2-(4-methyl-piperazin-1-yl)-ethoxy]-4-(3,4,5-trimethoxy-phenylamino)-benzo[g]quinoline-3-carbonitrile 328760 8-Methoxy-7-(2-morpholin-4-yl-ethoxy)-4-(3,4,5-trimethoxy-phenylamino)-benzo[g]quinoline-3-carbonitrile 328763 (2-Iodo-phenyl)-[2-methyl-1-(1-methyl-piperidin-2-ylmethyl)-1H-indol-3-yl]-methanone 328767 4-(2,4-Dichloro-phenylamino)-8-methoxy-7-(2-morpholin-4-yl-ethoxy)-benzo[g]quinoline-3-carbonitrile 328778 4-(4-Chloro-5-methoxy-2-methyl-phenylamino)-7-methoxy-8-(2-morpholin-4-yl-ethoxy)-benzo[g]quinoline-3-carbonitrile 328784 (4-Iodo-phenyl)-[2-methyl-1-(1-methyl-piperidin-2-ylmethyl)-1H-indol-3-yl]-methanone 328787 4-(4-Chloro-5-methoxy-2-methyl-phenylamino)-7-methoxy-8-[2-(4-methyl-piperazin-1-yl)-ethoxy]-benzo[g]quinoline-3-carbonitrile 328794 4-(2,4-Dichloro-5-methoxy-phenylamino)-7-methoxy-8-(2-morpholin-4-yl-ethoxy)-benzo[g]quinoline-3-carbonitrile 328801 4-(2,4-Dichloro-5-methoxy-phenylamino)-7-methoxy-8-[2-(4-methyl-piperazin-1-yl)-ethoxy]-benzo[g]quinoline-3-carbonitrile 328809 4-(2,4-Dichloro-5-methoxy-phenylamino)-8-[2-(4-hydroxy-piperidin-1-yl)-ethoxy]-7-methoxy-benzo[g]quinoline-3-carbonitrile 328817 4-(2-Chloro-5-methoxy-4-methyl-phenylamino)-7-methoxy-8-(2-morpholin-4-yl-ethoxy)-benzo[g]quinoline-3-carbonitrile 328825 4-(2-Chloro-5-methoxy-4-methyl-phenylamino)-8-[2-(4-hydroxy-piperidin-1-yl)-ethoxy]-7-methoxy-benzo[g]quinoline-3-carbonitrile 328830 4-(2-Chloro-4-fluoro-5-methoxy-phenylamino)-7-methoxy-8-(2-morpholin-4-yl-ethoxy)-benzo[g]quinoline-3-carbonitrile 328831 7-Methoxy-8-[2-(4-methyl-piperazin-1-yl)-ethoxy]-4-(3,4,5-trimethoxy-phenylamino)-benzo[g]quinoline-3-carbonitrile 328837 4-(4-Chloro-5-methoxy-2-methyl-phenylamino)-8-methoxy-7-(2-morpholin-4-yl-ethoxy)-benzo[g]quinoline-3-carbonitrile 328838 7-Methoxy-8-(2-morpholin-4-yl-ethoxy)-4-(3,4,5-trimethoxy-phenylamino)-benzo[g]quinoline-3-carbonitrile 328843 4-(4-Chloro-5-methoxy-2-methyl-phenylamino)-8-methoxy-7-[2-(4-methyl-piperazin-1-yl)-ethoxy]-benzo[g]quinoline-3-carbonitrile 328844 4-(2,4-Dichloro-phenylamino)-7-methoxy-8-(2-morpholin-4-yl-ethoxy)-benzo[g]quinoline-3-carbonitrile 328856 N-[4-(2-Ethyl-4-m-tolyl-thiazol-5-yl)-pyridin-2-yl]-propionamide 328857 N-[4-(2-Ethyl-4-m-tolyl-thiazol-5-yl)-pyridin-2-yl]-butyramide 328858 Benzyl-{4-[2-(4-methanesulfonyl-phenyl)-4-m-tolyl-thiazol-5-yl]-pyridin-2-yl}-amine 328861 Cyclohexanecarboxylic acid [4-(2-ethyl-4-m-tolyl-thiazol-5-yl)-pyridin-2-yl]-amide 328862 N-[4-(2-Ethyl-4-m-tolyl-thiazol-5-yl)-pyridin-2-yl]-2-phenyl-acetamide 328863 {4-[2-(4-Methanesulfonyl-phenyl)-4-m-tolyl-thiazol-5-yl]-pyridin-2-yl}-phenethyl-amine 328871 N-[4-(2-Ethyl-4-m-tolyl-thiazol-5-yl)-pyridin-2-yl]-3-phenyl-propionamide 328880 N-[4-(2-Ethyl-4-m-tolyl-thiazol-5-yl)-pyridin-2-yl]-benzamide 328881 N-{4-[4-(3-Chloro-phenyl)-2-ethyl-thiazol-5-yl]-pyridin-2-yl}-benzamide 328889 N-[4-(2-Ethyl-4-phenyl-thiazol-5-yl)-pyridin-2-yl]-benzamide 328890 N-{4-[2-Ethyl-4-(4-fluoro-phenyl)-thiazol-5-yl]-pyridin-2-yl}-benzamide 328898 N-{4-[2-Ethyl-4-(3-trifluoromethyl-phenyl)-thiazol-5-yl]-pyridin-2-yl}-benzamide 328899 N-[4-(2-Ethyl-4-o-tolyl-thiazol-5-yl)-pyridin-2-yl]-benzamide 328907 N-[4-(2-Ethyl-4-p-tolyl-thiazol-5-yl)-pyridin-2-yl]-benzamide 328908 N-{4-[2-Ethyl-4-(3-methoxy-phenyl)-thiazol-5-yl]-pyridin-2-yl}-benzamide 328914 N-{4-[2-Ethyl-4-(4-methoxy-phenyl)-thiazol-5-yl]-pyridin-2-yl}-benzamide 328921 N-[4-(2-Methyl-4-m-tolyl-thiazol-5-yl)-pyridin-2-yl]-benzamide 328922 N-[4-(2-Propyl-4-m-tolyl-thiazol-5-yl)-pyridin-2-yl]-benzamide 328929 Benzyl-[4-(2-ethyl-4-m-tolyl-thiazol-5-yl)-pyridin-2-yl]-amine 328930 [4-(2-Ethyl-4-m-tolyl-thiazol-5-yl)-pyridin-2-yl]-phenethyl-amine 328937 [4-(2-Ethyl-4-m-tolyl-thiazol-5-yl)-pyridin-2-yl]-(3-phenyl-propyl)-amine 328943 Cyclopentyl-[4-(2-ethyl-4-m-tolyl-thiazol-5-yl)-pyridin-2-yl]-amine 328944 4-(2-Ethyl-4-m-tolyl-thiazol-5-yl)-2-pyrrolidin-1-yl-pyridine 328950 4-[2-(4-Methanesulfonyl-phenyl)-4-m-tolyl-thiazol-5-yl]-pyridine 328951 4-[2-(4-Methanesulfonyl-phenyl)-4-m-tolyl-thiazol-5-yl]-2-methyl-pyridine 328955 N-(4-Guanidino-butyl)-N-(1-phenethyl-piperidin-4-yl)-propionamide 328962 4-(2-Ethyl-4-m-tolyl-thiazol-5-yl)-pyridine 328963 4-(2-Ethyl-4-m-tolyl-thiazol-5-yl)-2-methyl-pyridine 328964 4-(2-Ethyl-4-m-tolyl-thiazol-5-yl)-2-fluoro-pyridine 328965 N-{4-[2-(4-Methanesulfonyl-phenyl)-4-m-tolyl-thiazol-5-yl]-pyridin-2-yl}-benzamide 328970 4-(2-Ethyl-4-m-tolyl-thiazol-5-yl)-pyridin-2-ylamine 328971 2-Chloro-4-(2-ethyl-4-m-tolyl-thiazol-5-yl)-pyridine 328972 N-[4-(2-Ethyl-4-m-tolyl-thiazol-5-yl)-pyridin-2-yl]-acetamide 328973 N-{4-[2-(4-Methanesulfonyl-phenyl)-4-m-tolyl-thiazol-5-yl]-pyridin-2-yl}-2-phenyl-acetamide 328976 1-(4-(4-amino-6-(2-methoxyethyl)thieno[2,3-d]pyrimidin-5-yl)phenyl)-3-m-tolylurea 328977 1-(4-(4-amino-6-(3-hydroxypropyl)thieno[2,3-d]pyrimidin-5-yl)phenyl)-3-m-tolylurea 328981 N-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-methylbenzamide 328983 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-(2-chlorophenyl)urea 328984 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-(3-chlorophenyl)urea 328985 1-(4-(4-amino-6-(2-(dimethylamino)ethyl)thieno[2,3-d]pyrimidin-5-yl)phenyl)-3-m-tolylurea 328990 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-phenylurea 328991 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-(4-chlorophenyl)urea 328992 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-(3-bromophenyl)urea 328993 1-(4-(4-aminothieno[2,3-d]pyrimidin-5-yl)-3-fluorophenyl)-3-m-tolylurea 328994 1-(4-(4-aminothieno[2,3-d]pyrimidin-5-yl)-3-chlorophenyl)-3-m-tolylurea 328998 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-m-tolylurea 329000 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-(4-bromophenyl)urea 329001 1-(4-(4-aminothieno[2,3-d]pyrimidin-5-yl)-3-methoxyphenyl)-3-m-tolylurea 329002 1-(4-(4-aminothieno[2,3-d]pyrimidin-5-yl)-2-fluorophenyl)-3-m-tolylurea 329005 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-m-tolylthiourea 329006 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-2-cyano-3-m-tolylguanidine 329007 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-(3-(trifluoromethyl)phenyl)urea 329008 ethyl 3-(3-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)ureido)benzoate 329014 N-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)benzo[d]oxazol-2-amine 329015 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-(3,5-dimethylphenyl)urea 329016 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-(3,5-dichlorophenyl)urea 329020 N-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-2-m-tolylacetamide 329021 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-1-methyl-3-m-tolylurea 329022 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-(2-fluoro-5-(trifluoromethyl)phenyl)urea 329023 1-(4-(4-aminothieno[2,3-d]pyrimidin-5-yl)-2-chlorophenyl)-3-m-tolylurea 329029 3-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-1-methyl-1-m-tolylurea 329030 3-(4-amino-5-(4-(3-m-tolylureido)phenyl)thieno[2,3-d]pyrimidin-6-yl)propanamide 329046 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-benzylurea 329047 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-(cyclohexylmethyl)urea 329048 3-(4-amino-5-(4-(3-m-tolylureido)phenyl)thieno[2,3-d]pyrimidin-6-yl)-N-methylpropanamide 329054 1-(4-(4-amino-6-ethylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-m-tolylurea 329055 1-(4-(4-amino-6-ethylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-cyclohexylurea 329056 3-(4-amino-5-(4-(3-m-tolylureido)phenyl)thieno[2,3-d]pyrimidin-6-yl)-N,N-dimethylpropanamide 329061 1-(4-(4-aminothieno[2,3-d]pyrimidin-5-yl)phenyl)-3-m-tolylurea 329062 1-(4-(4-aminothieno[2,3-d]pyrimidin-5-yl)phenyl)-3-butylurea 329063 1-(4-(4-amino-6-(morpholinomethyl)thieno[2,3-d]pyrimidin-5-yl)phenyl)-3-m-tolylurea 329069 1-(4-(4-aminothieno[2,3-d]pyrimidin-5-yl)phenyl)-3-isobutylurea 329070 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-o-tolylurea 329071 1-(4-(4-amino-6-((4-methylpiperazin-1-yl)methyl)thieno[2,3-d]pyrimidin-5-yl)phenyl)-3-m-tolylurea 329078 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-p-tolylurea 329080 1-(4-(4-amino-6-((dimethylamino)methyl)thieno[2,3-d]pyrimidin-5-yl)phenyl)-3-m-tolylurea 329081 1-(4-(4-amino-6-propylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-m-tolylurea 329086 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-(2-methoxyphenyl)urea 329087 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-(3-methoxyphenyl)urea 329088 1-(4-(4-amino-6-isopropylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-m-tolylurea 329089 1-(4-(4-amino-6-benzylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-m-tolylurea 329092 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-(4-methoxyphenyl)urea 329093 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-(2-fluorophenyl)urea 329094 1-(4-(4-amino-6-(pyridin-3-ylmethyl)thieno[2,3-d]pyrimidin-5-yl)phenyl)-3-m-tolylurea 329109 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-(3-fluorophenyl)urea 329110 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-(4-fluorophenyl)urea 329111 1-(4-(4-amino-6-(pyridin-4-ylmethyl)thieno[2,3-d]pyrimidin-5-yl)phenyl)-3-m-tolylurea 329112 1-(4-(4-amino-6-(2-hydroxyethyl)thieno[2,3-d]pyrimidin-5-yl)phenyl)-3-m-tolylurea 329115 5-(4-aminophenyl)-6-methylthieno[2,3-d]pyrimidin-4-amine 329154 3-[(2-Cycloheptylmethyl-5-naphthalen-2-yl-2,3-dihydro-1H-pyrrole-3-carbonyl)-amino]-benzoic acid 329157 3-[(5-Cycloheptylmethyl-2-naphthalen-2-yl-4,5-dihydro-1H-imidazole-4-carbonyl)-amino]-benzoic acid 329160 1-{2-[1-Benzoyl-3-((S)-3,4-dichloro-phenyl)-pyrrolidin-3-yl]-ethyl}-4-phenyl-piperidine-4-carboxylic acid amide 329162 3-{[5-(2-Adamantan-1-yl-ethyl)-2-phenyl-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-benzoic acid 329168 3-{[2-(2-Adamantan-1-yl-ethyl)-5-o-tolyl-2,3-dihydro-1H-pyrrole-3-carbonyl]-amino}-benzoic acid 329175 3-{[2-(2-Adamantan-1-yl-ethyl)-5-phenyl-2,3-dihydro-1H-pyrrole-3-carbonyl]-amino}-benzoic acid 329258 (S)-8-{4-[3-(1H-Indol-3-yl)-propyl]-piperazin-1-yl}-2-methyl-4H-benzo[1,4]oxazin-3-one 329259 5-{[5-(2-Adamantan-1-yl-ethyl)-2-o-tolyl-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-2-fluoro-benzoic acid 329260 5-{[5-(2-Adamantan-1-yl-ethyl)-2-o-tolyl-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-2-dimethylamino-benzoic acid 329261 5-{[5-(2-Adamantan-1-yl-ethyl)-2-o-tolyl-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-2-methoxy-benzoic acid 329262 [5-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-isoxazol-3-yloxy]-acetic acid 329264 3-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-ylmethyl]-1H-indole 329265 (R)-8-(4-(3-(5-fluoro-1H-indol-3-yl)propyl)piperazin-1-yl)-2-methyl-2H-benzo[b][1,4]oxazin-3(4H)-one 329266 (S)-8-{4-[3-(5-Fluoro-1H-indol-3-yl)-propyl]-piperazin-1-yl}-2-methyl-4H-benzo[1,4]oxazin-3-one 329267 3-{[5-(2-Adamantan-1-yl-ethyl)-2-(2,4-dimethyl-phenyl)-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-benzoic acid 329270 3-{2-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-ethyl}-1H-indole 329271 3-{3-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-1H-indole 329272 (R)-8-{4-[3-(7-Fluoro-1H-indol-3-yl)-propyl]-piperazin-1-yl}-2-methyl-4H-benzo[1,4]oxazin-3-one 329273 (S)-8-{4-[3-(7-Fluoro-1H-indol-3-yl)-propyl]-piperazin-1-yl}-2-methyl-4H-benzo[1,4]oxazin-3-one 329274 3-{[5-(2-Adamantan-1-yl-ethyl)-2-(2,6-dimethyl-phenyl)-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-benzoic acid 329275 3-{[5-(2-Adamantan-1-yl-ethyl)-2-(2,4,6-trimethyl-phenyl)-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-benzoic acid 329276 1-{2-[3-((S)-3,4-Dichloro-phenyl)-1-(3,4,5-trimethoxy-benzoyl)-pyrrolidin-3-yl]-ethyl}-4-phenyl-piperidine-4-carboxylic acid amide 329280 3-{4-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-butyl}-1H-indole 329281 3-{5-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-pentyl}-1H-indole 329282 5-{[5-(2-Adamantan-1-yl-ethyl)-2-(2,4,6-trimethyl-phenyl)-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-2-methyl-benzoic acid 329283 3-{[5-(2-Adamantan-1-yl-ethyl)-2-methyl-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-benzoic acid 329284 3-{[5-(2-Adamantan-1-yl-ethyl)-2-propyl-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-benzoic acid 329287 3-{3-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-4-fluoro-1H-indole 329288 3-{3-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-5-fluoro-1H-indole 329290 3-{[5-(2-Adamantan-1-yl-ethyl)-2-isopropyl-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-benzoic acid 329291 3-{[5-(2-Adamantan-1-yl-ethyl)-2-tert-butyl-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-benzoic acid 329295 3-{3-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-6-fluoro-1H-indole 329298 3-{[5-(2-Adamantan-1-yl-ethyl)-2-cyclopropyl-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-benzoic acid 329299 3-{[5-(2-Adamantan-1-yl-ethyl)-2-cyclopentyl-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-benzoic acid 329302 3-{3-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-7-fluoro-1H-indole 329303 3-{3-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-5-methoxy-1H-indole 329304 3-{[5-(2-Adamantan-1-yl-ethyl)-2-cyclohexyl-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-benzoic acid 329308 4-Chloro-3-{3-[4-(2,3-dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-1H-indole 329309 5-Chloro-3-{3-[4-(2,3-dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-1H-indole 329310 3-{[5-(2-Adamantan-1-yl-ethyl)-2-o-tolyl-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-benzoic acid 329311 3-{[5-(3-Methyl-butyl)-2-o-tolyl-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-benzoic acid 329312 3-{[5-(2-Adamantan-1-yl-ethyl)-2-cycloheptyl-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-benzoic acid 329315 6-Chloro-3-{3-[4-(2,3-dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-1H-indole 329316 7-Chloro-3-{3-[4-(2,3-dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-1H-indole 329317 3-{[5-(3,3-Dimethyl-butyl)-2-o-tolyl-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-benzoic acid 329318 3-{[5-(2-Cyclohexyl-ethyl)-2-o-tolyl-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-benzoic acid 329319 3-{[5-(2-Adamantan-1-yl-ethyl)-2-bicyclo[2.2.2]oct-1-yl-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-benzoic acid 329324 3-{3-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-5-methyl-1H-indole 329325 3-{3-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-7-methyl-1H-indole 329326 3-[(5-Phenethyl-2-o-tolyl-4,5-dihydro-1H-imidazole-4-carbonyl)-amino]-benzoic acid 329327 3-{[5-(2-Adamantan-1-yl-ethyl)-2-(1-methyl-cyclohexyl)-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-benzoic acid 329330 3-[3-(4-Chroman-5-yl-piperazin-1-yl)-propyl]-1H-indole 329332 3-[(5-Adamantan-1-ylmethyl-2-o-tolyl-4,5-dihydro-1H-imidazole-4-carbonyl)-amino]-benzoic acid 329333 5-{[5-(2-Adamantan-1-yl-ethyl)-2-(1-methyl-cyclohexyl)-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-2-methyl-benzoic acid 329336 5-{4-[3-(1H-Indol-3-yl)-propyl]-piperazin-1-yl}-1,2,3,4-tetrahydro-quinoline 329337 5-{4-[3-(1H-Indol-3-yl)-propyl]-piperazin-1-yl}-1-methyl-1,2,3,4-tetrahydro-quinoline 329342 5-{4-[3-(1H-Indol-3-yl)-propyl]-piperazin-1-yl}-3-methyl-1,2,3,4-tetrahydro-quinoline 329343 5-{4-[3-(1H-Indol-3-yl)-propyl]-piperazin-1-yl}-3,4-dihydro-1H-quinolin-2-one 329346 3-{[5-(Adamantan-1-yloxymethyl)-2-bicyclo[2.2.2]oct-1-yl-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-benzoic acid 329347 3-{[5-(Adamantan-1-yloxymethyl)-2-(2,4,6-trimethyl-phenyl)-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-benzoic acid 329349 8-{4-[3-(1H-Indol-3-yl)-propyl]-piperazin-1-yl}-4H-benzo[1,4]oxazin-3-one 329350 8-{4-[3-(1H-Indol-3-yl)-propyl]-piperazin-1-yl}-2-methyl-4H-benzo[1,4]oxazin-3-one 329351 5-(2-Adamantan-1-yl-ethyl)-2-o-tolyl-4,5-dihydro-1H-imidazole-4-carboxylic acid (3-methylamino-phenyl)-amide 329353 8-{4-[3-(1H-Indol-3-yl)-propyl]-piperazin-1-yl}-2,2-dimethyl-4H-benzo[1,4]oxazin-3-one 329354 8-{4-[3-(1H-Indol-3-yl)-propyl]-piperazin-1-yl}-2,4-dimethyl-4H-benzo[1,4]oxazin-3-one 329355 (3-{[5-(2-Adamantan-1-yl-ethyl)-2-o-tolyl-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-phenyl)-acetic acid 329356 3-(3-{[5-(2-Adamantan-1-yl-ethyl)-2-o-tolyl-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-phenyl)-propionic acid 329357 2-[5-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-pyridin-2-yloxy]-N-(4-fluoro-phenyl)-acetamide 329361 8-{4-[3-(1H-Indol-3-yl)-propyl]-piperazin-1-yl}-3,4-dihydro-2H-benzo[1,4]oxazine 329362 (R)-8-{4-[3-(1H-Indol-3-yl)-propyl]-piperazin-1-yl}-2-methyl-4H-benzo[1,4]oxazin-3-one 329363 5-{[5-(2-Adamantan-1-yl-ethyl)-2-o-tolyl-4,5-dihydro-1H-imidazole-4-carbonyl]-amino}-2-methyl-benzoic acid 329364 8-(6-Hydroxy-pyridin-3-yl)-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 329367 (R)-2-((R)-3-(R)-Indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-N-isopropyl-2-(4-methanesulfonyl-phenyl)-acetamide 329368 (R)-2-((R)-4-(R)-Allyl-3-indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-N-isopropyl-2-phenyl-acetamide 329369 (R)-2-((R)-3-(R)-Indan-2-yl-6-isobutyl-2-oxo-piperazin-1-yl)-N-isopropyl-2-phenyl-acetamide 329371 4-[(R)-((R)-3-(R)-Indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-isopropylcarbamoyl-methyl]-benzamide 329373 (R)-2-(2,4-difluorophenyl)-2-((3R,6R)-3-(2,3-dihydro-1H-inden-2-yl)-6-isobutyl-2,5-dioxopiperazin-1-yl)-N-isopropylacetamide 329379 (R)-N-tert-Butyl-2-((R)-3-(R)-indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-2-phenyl-acetamide 329382 (R)-N-tert-Butyl-2-(4-chloro-phenyl)-2-((R)-3-(R)-indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-acetamide 329389 (R)-N-tert-Butyl-2-((R)-3-(R)-indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-2-(4-methoxy-phenyl)-acetamide 329390 (R)-N-tert-Butyl-2-((R)-3-(R)-indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-2-(4-trifluoromethoxy-phenyl)-acetamide 329392 (R)-2-(4-Acetylamino-phenyl)-N-tert-butyl-2-((R)-3-(R)-indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-acetamide 329393 (R)-2-(3-Acetylamino-phenyl)-N-tert-butyl-2-((R)-3-(R)-indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-acetamide 329394 (R)-N-tert-Butyl-2-((R)-3-(R)-indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-2-[4-(4-methyl-piperazin-1-yl)-phenyl]-acetamide 329395 (R)-N-tert-Butyl-2-((R)-3-(R)-indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-2-[3-(4-methyl-piperazin-1-yl)-phenyl]-acetamide 329398 3,4-Dihydro-2H-benzo[e][1,3]oxazine 329399 (S)-2-(4-Acetylamino-phenyl)-2-((R)-3-(R)-indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-N-isopropyl-acetamide 329404 (S)-2-((R)-3-(R)-Indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-N-isopropyl-2-phenyl-acetamide 329405 (S)-2-(4-Fluoro-phenyl)-2-((R)-3-(R)-indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-N-isopropyl-acetamide 329414 (S)-2-((R)-3-(R)-Indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-N-isopropyl-2-(4-trifluoromethyl-phenyl)-acetamide 329417 (S)-2-((R)-3-(R)-Indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-N-isopropyl-2-p-tolyl-acetamide 329424 (S)-2-(4-Dimethylamino-phenyl)-2-((R)-3-(R)-indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-N-isopropyl-acetamide 329431 (R)-2-(4-Acetylamino-phenyl)-2-((R)-3-(R)-indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-N-isopropyl-acetamide 329432 (S)-2-((R)-3-(R)-Indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-N-isopropyl-2-(4-methanesulfonyl-phenyl)-acetamide 329439 (R)-2-((R)-3-(R)-Indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-N-isopropyl-2-phenyl-acetamide 329440 4-[(S)-((R)-3-(R)-Indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-isopropylcarbamoyl-methyl]-benzamide 329441 N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-7-methoxybenzofuran-2-carboxamide 329444 (R)-2-((3R,6R)-3-(2,3-dihydro-1H-inden-2-yl)-6-isobutyl-2,5-dioxopiperazin-1-yl)-2-(4-fluorophenyl)-N-isopropylacetamide 329445 (S)-N-tert-Butyl-2-((R)-3-(R)-indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-2-phenyl-acetamide 329446 (R)-2-((R)-3-(R)-Indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-N-isopropyl-2-(4-trifluoromethyl-phenyl)-acetamide 329447 (S)-N-tert-Butyl-2-(4-chloro-phenyl)-2-((R)-3-(R)-indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-acetamide 329450 Urea derivative 329453 (R)-2-((R)-3-(R)-Indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-N-isopropyl-2-p-tolyl-acetamide 329454 (S)-N-tert-Butyl-2-((R)-3-(R)-indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-2-(4-methoxy-phenyl)-acetamide 329455 (S)-N-tert-Butyl-2-((R)-3-(R)-indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-2-(4-trifluoromethoxy-phenyl)-acetamide 329463 Urea derivative 329464 Urea derivative 329466 Urea derivative 329467 Urea derivative 329468 Urea derivative 329469 Urea derivative 329470 Urea derivative 329473 (R)-2-((3R,6R)-3-(2,3-dihydro-1H-inden-2-yl)-6-isobutyl-2,5-dioxopiperazin-1-yl)-2-(4-(dimethylamino)phenyl)-N-isopropylacetamide 329474 (R)-2-((3R,6R)-3-Indan-2-yl-6-isobutyl-2,5-dioxo-piperazin-1-yl)-N-isopropyl-N-methyl-2-phenyl-acetamide 329520 HYNIC Conjugate 329537 9-Methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine 329540 2,9-Dimethyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine 329541 2-butyl-9-methyl-8-(2H-1,2,3-triazol-2-yl)-9H-purin-6-amine 329545 9-Methyl-2-pentyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine 329546 9-Methyl-2-phenethyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine 329547 2-Isopropyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine 329553 9-Methyl-2-propyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine 329554 1-Methyl-2-[1,2,3]triazol-2-yl-1H-imidazo[4,5-c]pyridin-4-ylamine 329555 1,6-Dimethyl-2-[1,2,3]triazol-2-yl-1H-imidazo[4,5-c]pyridin-4-ylamine 329715 1-(4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)benzyl)azetidine-3-carboxylic acid 329722 [1-(4-Chloro-benzenesulfonyl)-5-fluoro-2-methyl-1H-indol-3-yl]-acetic acid 329822 HYNIC Analogue 329823 2-[5-(4-tert-Butyl-phenyl)-[1,3,4]oxadiazol-2-yl]-phenylamine 329852 {2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-ylmethyl}-(5-nitro-thiazol-2-yl)-amine 329854 4-({2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-ylmethyl}-amino)-pyridine-2,6-dicarbonitrile 329856 1-Thiophen-2-yl-3,4-dihydro-1H-isoquinoline-2-carboxylic acid (R)-(1-aza-bicyclo[2.2.2]oct-3-yl) ester 329860 2,2,2-Trifluoro-1-[4-({2-[2-((R)-2-methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-ylmethyl}-amino)-phenyl]-ethanone 329870 {2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-ylmethyl}-pyrimidin-5-yl-amine 329875 3-({2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-ylmethyl}-amino)-benzonitrile 329892 (6-Chloro-pyridazin-3-yl)-{2-[2-((R)-2-methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-ylmethyl}-amine 329903 3-({2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-ylmethyl}-amino)-pyrazine-2-carbonitrile 329914 1-(4-(4-aminothieno[2,3-d]pyrimidin-5-yl)-2-methoxyphenyl)-3-m-tolylurea 329915 1-(11-Amino-5,6,6a,11b-tetrahydro-7-thia-8,10-diaza-benzo[c]fluoren-3-yl)-3-m-tolyl-urea 329919 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-(4-(trifluoromethyl)phenyl)urea 329920 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-(2-fluoro-5-methylphenyl)urea 329921 (5-Ethyl-pyrimidin-2-yl)-{2-[2-((R)-2-methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-ylmethyl}-amine 329923 {2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-ylmethyl}-(3-nitro-pyridin-2-yl)-amine 329928 1-(4-(4-amino-6-ethylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-(3-(trifluoromethyl)phenyl)urea 329929 {2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-ylmethyl}-pyrazin-2-yl-amine 329935 1-(4-(4-aminothieno[2,3-d]pyrimidin-5-yl)phenyl)-3-(3-chlorophenyl)urea 329963 (S)-3-Amino-N-((S)-1-{(S)-1-[(S)-3-[2-[2-((S)-(S)-1-carboxy-2-phenyl-ethylcarbamoyl)-pyrrolidin-1-yl]-1-(3H-imidazol-4-ylmethyl)-2-oxo-ethylcarbamoyl]-5-(4-hydroxy-benzyl)-phenylcarbamoyl]-2-methyl-propylcarbamoyl}-4-guanidino-butyl)-succinamic acid 329969 {2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-ylmethyl}-pyrimidin-2-yl-amine 329981 {2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-ylmethyl}-(2-nitro-phenyl)-amine 329993 (3,5-Dinitro-pyridin-2-yl)-{2-[2-((R)-2-methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-ylmethyl}-amine 329994 1-Phenyl-1,2,3,4-tetrahydro-quinoline-2-carboxylic acid (R)-(1-aza-bicyclo[2.2.2]oct-3-yl) ester 329995 Benzhydryl-carbamic acid 1-aza-bicyclo[2.2.2]oct-3-yl ester 329996 (5-Bromo-pyrimidin-2-yl)-{2-[2-((R)-2-methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-ylmethyl}-amine 330001 {2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-ylmethyl}-(4-nitro-phenyl)-amine 330011 (4-Chloro-phenyl)-[8-(4-methyl-piperazin-1-yl)-2,3-dihydro-pyrrolo[3,2-g]isoquinolin-1-yl]-methanone 330016 4-[8-(4-Methyl-piperazin-1-yl)-2,3-dihydro-pyrrolo[3,2-g]isoquinoline-1-carbonyl]-benzonitrile 330017 [8-(4-Methyl-piperazin-1-yl)-2,3-dihydro-pyrrolo[3,2-g]isoquinolin-1-yl]-(2-trifluoromethyl-phenyl)-methanone 330022 {2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-ylmethyl}-(5-nitro-pyridin-2-yl)-amine 330024 (2-Chloro-phenyl)-[8-(4-methyl-piperazin-1-yl)-2,3-dihydro-pyrrolo[3,2-g]isoquinolin-1-yl]-methanone 330025 3-{2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-ylamino}-benzonitrile 330032 [8-(4-Methyl-piperazin-1-yl)-2,3-dihydro-pyrrolo[3,2-g]isoquinolin-1-yl]-(6-trifluoromethyl-pyridin-3-yl)-methanone 330033 [8-(4-Methyl-piperazin-1-yl)-2,3-dihydro-pyrrolo[3,2-g]isoquinolin-1-yl]-quinolin-5-yl-methanone 330034 {2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-pyrimidin-5-yl-amine 330045 {2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-pyrazin-2-yl-amine 330049 {2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-(3-nitro-pyridin-2-yl)-amine 330054 [8-(4-Methyl-piperazin-1-yl)-2,3-dihydro-pyrrolo[3,2-g]isoquinolin-1-yl]-(5-methyl-2-trifluoromethyl-furan-3-yl)-methanone 330055 (2,4-Dimethyl-oxazol-5-yl)-[8-(4-methyl-piperazin-1-yl)-2,3-dihydro-pyrrolo[3,2-g]isoquinolin-1-yl]-methanone 330060 [8-(4-Methyl-piperazin-1-yl)-2,3-dihydro-pyrrolo[3,2-g]isoquinolin-1-yl]-(1-methyl-5-trifluoromethyl-1H-pyrazol-4-yl)-methanone 330061 [8-(4-Methyl-piperazin-1-yl)-2,3-dihydro-pyrrolo[3,2-g]isoquinolin-1-yl]-pyrazolo[1,5-a]pyridin-3-yl-methanone 330066 (5-Methyl-1-phenyl-1H-pyrazol-4-yl)-[8-(4-methyl-piperazin-1-yl)-2,3-dihydro-pyrrolo[3,2-g]isoquinolin-1-yl]-methanone 330067 4-{5-Ethyl-4-[8-(4-methyl-piperazin-1-yl)-2,3-dihydro-pyrrolo[3,2-g]isoquinoline-1-carbonyl]-pyrazol-1-yl}-benzonitrile 330069 2-({2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-ylmethyl}-amino)-nicotinonitrile 330072 {2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-(2-nitro-phenyl)-amine 330073 4-[5-Ethyl-4-(8-piperazin-1-yl-2,3-dihydro-pyrrolo[3,2-g]isoquinoline-1-carbonyl)-pyrazol-1-yl]-benzonitrile 330080 4-{5-Ethyl-4-[8-(4-ethyl-piperazin-1-yl)-2,3-dihydro-pyrrolo[3,2-g]isoquinoline-1-carbonyl]-pyrazol-1-yl}-benzonitrile 330081 (5-Ethyl-pyrimidin-2-yl)-{2-[2-((R)-2-methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-amine 330087 4-{5-Ethyl-4-[8-(4-isopropyl-piperazin-1-yl)-2,3-dihydro-pyrrolo[3,2-g]isoquinoline-1-carbonyl]-pyrazol-1-yl}-benzonitrile 330093 4-{4-[8-((3R,5S)-3,5-Dimethyl-piperazin-1-yl)-2,3-dihydro-pyrrolo[3,2-g]isoquinoline-1-carbonyl]-5-ethyl-pyrazol-1-yl}-benzonitrile 330095 {2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-(5-nitro-pyridin-2-yl)-amine 330100 4-{5-Ethyl-4-[(R)-8-(hexahydro-pyrrolo[1,2-a]pyrazin-2-yl)-2,3-dihydro-pyrrolo[3,2-g]isoquinoline-1-carbonyl]-pyrazol-1-yl}-benzonitrile 330103 6-({2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-ylmethyl}-amino)-nicotinonitrile 330106 4-{5-Ethyl-4-[(S)-8-(hexahydro-pyrrolo[1,2-a]pyrazin-2-yl)-2,3-dihydro-pyrrolo[3,2-g]isoquinoline-1-carbonyl]-pyrazol-1-yl}-benzonitrile 330110 4-{2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-ylamino}-benzonitrile 330121 {2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-pyrimidin-2-yl-amine 330129 1-tert-Butoxy-3-{4-[5-(4-fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-propan-2-ol 330130 1-Allyloxy-3-{4-[5-(4-fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-propan-2-ol 330143 1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-3-phenoxy-propan-2-ol 330152 1-Benzyloxy-3-{4-[5-(4-fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-propan-2-ol 330168 1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-3-(furan-2-ylmethoxy)-propan-2-ol 330169 3-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-propane-1,2-diol 330174 N'-(4,5-Dihydro-oxazol-2-yl)-N-(3-methoxy-phenyl)-N-p-tolyl-hydrazine 330176 (S)-2-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-butane-1,3-diol 330181 3-[N'-(4,5-Dihydro-oxazol-2-yl)-N-p-tolyl-hydrazino]-phenol 330183 (R)-2-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-butane-1,3-diol 330188 N'-(4,5-Dihydro-1H-imidazol-2-yl)-N-(3-methoxy-phenyl)-N-p-tolyl-hydrazine 330189 3-[N'-(4,5-Dihydro-1H-imidazol-2-yl)-N-p-tolyl-hydrazino]-phenol 330191 1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-butane-2,3-diol 330197 4-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-butan-1-ol 330198 (S,R)-3-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-butan-2-ol 330199 (R,S)-3-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-butan-2-ol 330203 5-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-pentan-1-ol 330204 Acetic acid 2-{4-[5-(4-fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-ethyl ester 330205 (R)-5-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-ylmethyl}-pyrrolidin-3-ol 330206 1-((R)-2-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-ylmethyl}-4-hydroxy-pyrrolidin-1-yl)-ethanone 330209 (R)-1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-propan-2-ol 330214 6-Methyl-2-{2-[2-((R)-2-methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-ylamino}-nicotinonitrile 330215 (S)-1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-propan-2-ol 330221 1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-butan-2-ol 330222 1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-pentan-2-ol 330230 1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-hexan-2-ol 330231 1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-octan-2-ol 330238 1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-3-phenyl-propan-2-ol 330244 1-Ethoxy-3-{4-[5-(4-fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-propan-2-ol 330249 1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-3-isopropoxy-propan-2-ol 330250 {2-[2-((R)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-(5-trifluoromethyl-pyridin-2-yl)-amine 330282 4-(2-Methoxy-phenyl)-piperazine-1-carboxylic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide 330283 4-(2-Chloro-phenyl)-piperazine-1-carboxylic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide 330287 4-(2-Fluoro-phenyl)-piperazine-1-carboxylic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide 330313 {8-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-4-methyl-3,4-dihydro-2H-quinolin-1-yl}-cyclohexyl-methanone 330314 1-{8-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-6-fluoro-4-methyl-3,4-dihydro-2H-quinolin-1-yl}-ethanone 330322 1-{8-[2-(4-Benzo[d]isoxazol-3-yl-piperazin-1-yl)-ethyl]-4,5-dimethyl-3,4-dihydro-2H-quinolin-1-yl}-ethanone 330323 1-{8-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-6-chloro-4-methyl-3,4-dihydro-2H-quinolin-1-yl}-ethanone 330330 1-{8-[2-(4-Benzo[d]isoxazol-3-yl-piperazin-1-yl)-ethyl]-6-fluoro-4-methyl-3,4-dihydro-2H-quinolin-1-yl}-ethanone 330331 1-{8-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-4-phenyl-3,4-dihydro-2H-quinolin-1-yl}-ethanone 330338 1-{8-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-4,5-dimethyl-3,4-dihydro-2H-quinolin-1-yl}-ethanone 330339 4-[(S)-2-(4-Fluoro-phenyl)-5-(4-methoxy-benzyloxymethyl)-6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-3-yl]-pyrimidin-2-ylamine 330346 4-[(R)-2-(4-Fluoro-phenyl)-5-(4-methoxy-benzyloxymethyl)-6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-3-yl]-pyrimidin-2-ylamine 330351 {4-[(S)-2-(4-Fluoro-phenyl)-5-(4-methoxy-benzyloxymethyl)-6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-3-yl]-pyrimidin-2-yl}-propyl-amine 330357 8-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-3,4-dihydro-1H-quinolin-2-one 330358 8-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-4-methyl-3,4-dihydro-1H-quinolin-2-one 330359 {4-[(R)-2-(4-Fluoro-phenyl)-5-(4-methoxy-benzyloxymethyl)-6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-3-yl]-pyrimidin-2-yl}-propyl-amine 330360 (S)-(2-(4-fluorophenyl)-3-(2-(propylamino)pyrimidin-4-yl)-6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-5-yl)methanol 330367 8-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-6-fluoro-4-methyl-3,4-dihydro-1H-quinolin-2-one 330368 8-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-3-methyl-3,4-dihydro-1H-quinolin-2-one 330369 [(R)-2-(4-Fluoro-phenyl)-3-(2-propylamino-pyrimidin-4-yl)-6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-5-yl]-methanol 330370 N-{3-[4-(3-Azido-phenyl)-5-pyridin-4-yl-imidazol-1-yl]-propyl}-4-iodo-benzamide 330377 8-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-1,4-dimethyl-3,4-dihydro-1H-quinolin-2-one 330378 8-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-4-phenyl-3,4-dihydro-1H-quinolin-2-one 330379 N-(3-(4-(4-fluorophenyl)-5-(pyridin-4-yl)-1H-imidazol-1-yl)propyl)benzamide 330388 8-[2-(4-Benzo[d]isoxazol-3-yl-piperazin-1-yl)-ethyl]-4-methyl-3,4-dihydro-1H-quinolin-2-one 330390 HYNIC Conjugate 330396 8-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-4,5-dimethyl-3,4-dihydro-1H-quinolin-2-one 330397 6-Fluoro-4-methyl-8-{2-[4-(1-oxo-1H-1lambda*4*-benzo[d]isothiazol-3-yl)-piperazin-1-yl]-ethyl}-3,4-dihydro-1H-quinolin-2-one 330406 8-[2-(4-Benzo[d]isoxazol-3-yl-piperazin-1-yl)-ethyl]-4,6-dimethyl-3,4-dihydro-1H-quinolin-2-one 330407 8-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-6-chloro-4-methyl-3,4-dihydro-1H-quinolin-2-one 330414 8-[2-(4-Benzo[d]isoxazol-3-yl-piperazin-1-yl)-ethyl]-6-fluoro-4-methyl-3,4-dihydro-1H-quinolin-2-one 330415 8-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-4,4-dimethyl-1,2,3,4-tetrahydro-quinoline 330426 8-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-6-fluoro-4,4-dimethyl-1,2,3,4-tetrahydro-quinoline 330427 {8-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-4-methyl-3,4-dihydro-2H-quinolin-1-yl}-phenyl-methanone 330438 1-{8-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-4-methyl-3,4-dihydro-2H-quinolin-1-yl}-ethanone 330440 1-{8-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-4-methyl-3,4-dihydro-2H-quinolin-1-yl}-2-(2,6-dimethoxy-phenyl)-ethanone 330449 1-{8-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-4-methyl-3,4-dihydro-2H-quinolin-1-yl}-2-(3-methoxy-phenyl)-ethanone 330554 Penta-Apc-DPhe-Arg-Trp-Gly-NH2 330560 4-(4-Ethoxy-phenyl)-1-pentanoylamino-cyclohexanecarboxylic acid ((R)-1-{(S)-1-[(S)-1-(carbamoylmethyl-carbamoyl)-2-(1H-indol-3-yl)-ethylcarbamoyl]-4-guanidino-butylcarbamoyl}-2-phenyl-ethyl)-amide 330584 N-[2-(2-Fluoro-phenyl)-2-(4-methyl-piperazin-1-yl)-ethyl]-methanesulfonamide 330586 N-[2-(2-Fluoro-phenyl)-2-(4-methyl-piperazin-1-yl)-ethyl]-acetamide 330589 Ethyl-[2-(2-fluoro-phenyl)-2-(4-methyl-piperazin-1-yl)-ethyl]-carbamic acid methyl ester 330590 N-Ethyl-N-[2-(2-fluoro-phenyl)-2-(4-methyl-piperazin-1-yl)-ethyl]-methanesulfonamide 330591 N-Ethyl-N-[2-(2-fluoro-phenyl)-2-(4-methyl-piperazin-1-yl)-ethyl]-acetamide 330593 N,N-Diethyl-2-(2-fluoro-phenyl)-2-(4-methyl-piperazin-1-yl)-acetamide 330594 Diethyl-[(S)-2-(4-methyl-piperazin-1-yl)-2-phenyl-ethyl]-amine 330595 Diethyl-[(R)-2-(4-methyl-piperazin-1-yl)-2-phenyl-ethyl]-amine 330598 Diethyl-[(S)-2-(2-fluoro-phenyl)-2-(4-methyl-piperazin-1-yl)-ethyl]-amine 330599 Diethyl-[(R)-2-(2-fluoro-phenyl)-2-(4-methyl-piperazin-1-yl)-ethyl]-amine 330601 1N,1N-diethyl-2-[2-hydroxy-3-(1H-4-indolyloxy)propylaminomethyl]-1-phenyl-(1S,2R)-cyclopropane-1-carboxamide 330620 1-Benzyl-4-methyl-piperazine 330621 1-Methyl-4-(1-phenyl-ethyl)-piperazine 330624 Diethyl-[2-(4-methyl-piperazin-1-yl)-2-phenyl-ethyl]-amine 330625 Diethyl-[2-(4-methyl-piperazin-1-yl)-3-phenyl-propyl]-amine 330626 Diethyl-[2-(4-methyl-piperazin-1-yl)-4-phenyl-butyl]-amine 330628 Diethyl-[2-(4-methyl-piperazin-1-yl)-5-phenyl-pentyl]-amine 330629 Diethyl-[2-(4-methyl-piperazin-1-yl)-2-(2-trifluoromethyl-phenyl)-ethyl]-amine 330632 Diethyl-[2-(4-methyl-piperazin-1-yl)-2-(3-trifluoromethyl-phenyl)-ethyl]-amine 330633 Diethyl-[2-(4-methyl-piperazin-1-yl)-2-(4-trifluoromethyl-phenyl)-ethyl]-amine 330634 [2-(2-Chloro-phenyl)-2-(4-methyl-piperazin-1-yl)-ethyl]-diethyl-amine 330638 Diethyl-[2-(4-methyl-piperazin-1-yl)-2-o-tolyl-ethyl]-amine 330639 Diethyl-[2-(2-fluoro-phenyl)-2-(4-methyl-piperazin-1-yl)-ethyl]-amine 330640 Diethyl-[2-(2-methoxy-phenyl)-2-(4-methyl-piperazin-1-yl)-ethyl]-amine 330643 [2-(2,6-Difluoro-phenyl)-2-(4-methyl-piperazin-1-yl)-ethyl]-diethyl-amine 330644 [2-(2,4-Difluoro-phenyl)-2-(4-methyl-piperazin-1-yl)-ethyl]-diethyl-amine 330645 [2-(2-Fluoro-phenyl)-2-(4-methyl-piperazin-1-yl)-ethyl]-carbamic acid methyl ester 330654 3-(2-chlorophenyl)-1-(5-methoxy-6-(2-(piperidin-1-yl)ethoxy)indolin-1-yl)prop-2-en-1-one 330655 1-[4-Methoxy-3-(2-piperidin-1-yl-ethoxy)-phenyl]-3-(4-methyl-3-trifluoromethyl-phenyl)-imidazolidin-2-one 330661 1-(2-Chloro-phenyl)-3-[4-methoxy-3-(2-piperidin-1-yl-ethoxy)-phenyl]-imidazolidin-2-one 330664 N-(1-(3,3-bis(4-fluorophenyl)propyl)piperidin-4-yl)-N-ethyl-2-(4-(methylsulfonyl)phenyl)acetamide 330667 1-(2,3-Dichloro-phenyl)-3-[4-methoxy-3-(2-piperidin-1-yl-ethoxy)-phenyl]-imidazolidin-2-one 330668 1-(3,4-Dichloro-phenyl)-3-[4-methoxy-3-(2-piperidin-1-yl-ethoxy)-phenyl]-imidazolidin-2-one 330673 1-Phenyl-3,4-dihydro-1H-isoquinoline-2-carboxylic acid (R)-(1-aza-bicyclo[2.2.2]oct-3-yl) ester 330675 N-{1-[3-(4-Chloro-phenyl)-3-phenyl-propyl]-piperidin-4-yl}-N-ethyl-2-(4-methanesulfonyl-phenyl)-acetamide 330678 1-[4-Methoxy-3-(2-piperidin-1-yl-ethoxy)-phenyl]-3-phenyl-imidazolidin-2-one 330679 1-(3-Fluoro-phenyl)-3-[4-methoxy-3-(2-piperidin-1-yl-ethoxy)-phenyl]-imidazolidin-2-one 330682 N-{1-[3,3-Bis-(4-chloro-phenyl)-propyl]-piperidin-4-yl}-N-ethyl-2-(4-methanesulfonyl-phenyl)-acetamide 330685 1-(3-Fluoro-phenyl)-3-[4-methoxy-3-(2-morpholin-4-yl-ethoxy)-phenyl]-imidazolidin-2-one 330686 1-[3-(2-Dimethylamino-ethoxy)-4-methoxy-phenyl]-3-(3-fluoro-phenyl)-imidazolidin-2-one 330688 N-Ethyl-N-{1-[3-(4-fluoro-phenyl)-3-phenyl-propyl]-piperidin-4-yl}-2-(4-methanesulfonyl-phenyl)-acetamide 330691 1-(3-Fluoro-phenyl)-3-[3-(2-hydroxy-ethoxy)-4-methoxy-phenyl]-imidazolidin-2-one 330692 1-(3,4-Dichloro-phenyl)-3-[4-methoxy-3-(2-morpholin-4-yl-ethoxy)-phenyl]-imidazolidin-2-one 330693 (5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepin-10-yl)-biphenyl-4-yl-methanone 330694 (5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepin-10-yl)-(2'-methyl-biphenyl-4-yl)-methanone 330698 1-(3,4-Dichloro-phenyl)-3-[3-(2-dimethylamino-ethoxy)-4-methoxy-phenyl]-imidazolidin-2-one 330699 1-[4-Methoxy-3-(2-morpholin-4-yl-ethoxy)-phenyl]-3-(4-methyl-3-trifluoromethyl-phenyl)-imidazolidin-2-one 330700 (5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepin-10-yl)-(2'-nitro-biphenyl-4-yl)-methanone 330701 (5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepin-10-yl)-(3',5'-difluoro-biphenyl-4-yl)-methanone 330706 1-(3,4-Dichloro-phenyl)-3-[6-(2-piperidin-1-yl-ethoxy)-pyridin-3-yl]-imidazolidin-2-one 330707 (5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepin-10-yl)-(4'-methyl-biphenyl-4-yl)-methanone 330708 1-Phenyl-1,3-dihydro-isoindole-2-carboxylic acid (R)-(1-aza-bicyclo[2.2.2]oct-3-yl) ester 330712 1-(3,4-Dichloro-phenyl)-3-[6-(pyridin-2-ylmethoxy)-pyridin-3-yl]-imidazolidin-2-one 330713 1-(3-Fluoro-phenyl)-3-[4-methoxy-3-(2-piperidin-1-yl-ethoxy)-phenyl]-1,3-dihydro-imidazol-2-one 330715 (5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepin-10-yl)-(4'-propyl-biphenyl-4-yl)-methanone 330719 1-(3,5-Difluoro-phenyl)-3-[4-methoxy-3-(2-piperidin-1-yl-ethoxy)-phenyl]-1,3-dihydro-imidazol-2-one 330720 3-(3-Fluoro-phenyl)-1-[4-methoxy-3-(2-piperidin-1-yl-ethoxy)-phenyl]-imidazolidine-2,4-dione 330722 (5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepin-10-yl)-(4-p-tolyloxy-phenyl)-methanone 330727 1-(3,5-Difluoro-phenyl)-3-[4-methoxy-3-(2-piperidin-1-yl-ethoxy)-phenyl]-imidazolidin-2-one 330740 (5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepin-10-yl)-[4-(toluene-4-sulfonyl)-phenyl]-methanone 330747 (5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepin-10-yl)-(4-thiophen-2-yl-phenyl)-methanone 330748 Biphenyl-4-yl-(3-dimethylaminomethyl-5H,11H-benzo[e]pyrrolo[1,2-a][1,4]diazepin-10-yl)-methanone 330755 4-Phenyl-3,4-dihydro-1H-isoquinoline-2-carboxylic acid (R)-(1-aza-bicyclo[2.2.2]oct-3-yl) ester 330756 (3-Dimethylaminomethyl-5H,11H-benzo[e]pyrrolo[1,2-a][1,4]diazepin-10-yl)-(4-thiophen-2-yl-phenyl)-methanone 330761 N-{1-[3-(4-Amino-phenyl)-3-phenyl-propyl]-piperidin-4-yl}-N-ethyl-2-(4-methanesulfonyl-phenyl)-acetamide 330762 N-{1-[3-(4-Acetylamino-phenyl)-3-phenyl-propyl]-piperidin-4-yl}-N-ethyl-2-(4-methanesulfonyl-phenyl)-acetamide 330763 N-Ethyl-2-(4-methanesulfonyl-phenyl)-N-{1-[3-phenyl-3-(4-phenylacetylamino-phenyl)-propyl]-piperidin-4-yl}-acetamide 330764 N-{4-[3-(4-{Ethyl-[2-(4-methanesulfonyl-phenyl)-acetyl]-amino}-piperidin-1-yl)-1-phenyl-propyl]-phenyl}-benzamide 330765 N-{4-[3-(4-{Ethyl-[2-(4-methanesulfonyl-phenyl)-acetyl]-amino}-piperidin-1-yl)-1-phenyl-propyl]-phenyl}-2,2-dimethyl-propionamide 330766 N-Ethyl-N-{1-[3-(4-methanesulfonylamino-phenyl)-3-phenyl-propyl]-piperidin-4-yl}-2-(4-methanesulfonyl-phenyl)-acetamide 330767 N-Ethyl-2-(4-methanesulfonyl-phenyl)-N-{1-[3-phenyl-3-(4-phenylmethanesulfonylamino-phenyl)-propyl]-piperidin-4-yl}-acetamide 330768 N-{1-[3-(4-Benzenesulfonylamino-phenyl)-3-phenyl-propyl]-piperidin-4-yl}-N-ethyl-2-(4-methanesulfonyl-phenyl)-acetamide 330769 1'-cyclooctylmethyl-1-(2-hydroxyethyl)spiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-2-one 330770 1-cyclohexylmethyl-1'-cyclooctylmethylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-2-one 330775 N-{1-[3-(4-Chloro-phenyl)-3-(3-fluoro-phenyl)-propyl]-piperidin-4-yl}-N-ethyl-2-(4-methanesulfonyl-phenyl)-acetamide 330778 1'-cyclooctylmethylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-2-one 330779 1'-cyclooctylmethyl-1-(4-methoxybenzyl)spiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-2-one 330782 N-{1-[3-(4-Amino-phenyl)-3-(3-fluoro-phenyl)-propyl]-piperidin-4-yl}-N-ethyl-2-(4-methanesulfonyl-phenyl)-acetamide 330783 N-{1-[3-(4-Acetylamino-phenyl)-3-(3-fluoro-phenyl)-propyl]-piperidin-4-yl}-N-ethyl-2-(4-methanesulfonyl-phenyl)-acetamide 330784 N-Ethyl-N-{1-[3-(3-fluoro-phenyl)-3-(4-methanesulfonylamino-phenyl)-propyl]-piperidin-4-yl}-2-(4-methanesulfonyl-phenyl)-acetamide 330799 1-benzyl-1'-cyclooctylmethylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-2-one 330800 1'-cyclooctylmethyl-1-(2-oxiranylmethyl)spiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-2-one 330801 1-Cyclohexyl-3,4-dihydro-1H-isoquinoline-2-carboxylic acid (R)-(1-aza-bicyclo[2.2.2]oct-3-yl) ester 330810 methyl [1'-(cyclopropylmethyl)-2-oxospiro[indole-3,4'-piperidin]-1(2H)-yl]acetate 330811 methyl 2-[1'-cyclohexylmethyl-2-oxospiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]acetate 330812 1'-cyclooctylmethyl-1-{2-hydroxy-3-[2-(1,4-oxazinan-4-yl)ethylamino]propyl}spiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-2-one 330818 methyl 2-[1'-cycloheptylmethyl-2-oxospiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]acetate 330819 methyl 2-[1'-cyclooctylmethyl-2-oxospiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]acetate 330820 1'-cyclooctylmethyl-1-[3-ethyl(4-methylbenzyl)amino-2-hydroxypropyl]spiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-2-one 330821 1'-cyclooctylmethyl-1-cyclopropylmethyl-6-methoxyspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-2-one 330826 methyl 2-[1'-cyclododecylmethyl-2-oxospiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]acetate 330827 methyl 2-[1'-hexyl-2-oxospiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]acetate 330828 1'-cyclooctylmethyl-6-methoxy-1-methylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-2-one 330829 1'-cyclooctylmethyl-1-ethyl-6-methoxyspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-2-one 330835 methyl 2-[1'-(2-butyloctyl)-2-oxospiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]acetate 330837 1'-cyclooctylmethyl-6-hydroxy-1-methylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-2-one 330838 1'-cyclooctylmethyl-1-methylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-2-one 330841 N-{1-[3-(3-Chloro-phenyl)-3-phenyl-propyl]-piperidin-4-yl}-N-ethyl-2-(4-methanesulfonyl-phenyl)-acetamide 330842 methyl 2-[1'-(4-chlorobenzyl)-2-oxospiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]acetate 330843 methyl 2-[1'-(1-naphthylmethyl)-2-oxospiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]acetate 330844 1'-cyclooctylmethyl-1,6-dimethylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-2-one 330846 1-Benzyl-3,4-dihydro-1H-isoquinoline-2-carboxylic acid (R)-(1-aza-bicyclo[2.2.2]oct-3-yl) ester 330847 N-{1-[3-(3,4-Dichloro-phenyl)-3-phenyl-propyl]-piperidin-4-yl}-N-ethyl-2-(4-methanesulfonyl-phenyl)-acetamide 330848 methyl 2-[1'-(2-naphthylmethyl)-2-oxospiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]acetate 330849 methyl 2-[2-oxo-1'-(4-trifluoromethylbenzyl)spiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]acetate 330850 1'-cyclooctylmethyl-1,5-dimethylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-2-one 330851 1'-cyclooctylmethyl-1,4-dimethylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-2-one 330854 N-Ethyl-2-(4-methanesulfonyl-phenyl)-N-[1-(3-phenyl-3-p-tolyl-propyl)-piperidin-4-yl]-acetamide 330855 methyl 2-[2-oxo-1'-(3-trifluoromethylbenzyl)spiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]acetate 330856 methyl 2-[2-oxo-1'-(4-phenylbenzyl)spiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]acetate 330857 1'-cyclooctylmethyl-1-methyl-5-trifluoromethylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-2-one 330858 1'-cyclooctylmethyl-5-fluoro-1-methylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-2-one 330861 N-Ethyl-2-(4-methanesulfonyl-phenyl)-N-{1-[3-phenyl-3-(4-trifluoromethyl-phenyl)-propyl]-piperidin-4-yl}-acetamide 330862 methyl 2-[2-oxo-1'-(1-phenylethyl)spiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]acetate 330863 methyl 2-[2-oxo-1'-[2-(3-thienyl)benzyl]spiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]acetate 330864 1'-cyclooctylmethyl-5-isopropyl-1-propylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-2-one 330865 1'-cyclooctylmethyl-5-isopropyl-1-methylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-2-one 330867 4-[3-(4-{Ethyl-[2-(4-methanesulfonyl-phenyl)-acetyl]-amino}-piperidin-1-yl)-1-phenyl-propyl]-benzoic acid methyl ester 330868 4-[3-(4-{Ethyl-[2-(4-methanesulfonyl-phenyl)-acetyl]-amino}-piperidin-1-yl)-1-phenyl-propyl]-benzamide 330869 methyl 2-[2-oxo-1'-(1,2,3,4-tetrahydro-2-naphthalenyl)spiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]acetate 330870 methyl 2-[2-oxo-1'-perhydro-2-naphthalenylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]acetate 330881 N-Ethyl-2-(4-methanesulfonyl-phenyl)-N-{1-[3-(4-methoxy-phenyl)-3-phenyl-propyl]-piperidin-4-yl}-acetamide 330882 N-[1-(3-Biphenyl-4-yl-3-phenyl-propyl)-piperidin-4-yl]-N-ethyl-2-(4-methanesulfonyl-phenyl)-acetamide 330883 methyl 2-[1'-(1,2-dihydro-5-acenaphthylenyl)-2-oxospiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]acetate 330884 methyl 2-[1'-[4-(tert-butyl)cyclohexylmethyl]-2-oxospiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]acetate 330888 4-Hydroxy-1-phenyl-3,4-dihydro-1H-isoquinoline-2-carboxylic acid (R)-(1-aza-bicyclo[2.2.2]oct-3-yl) ester 330889 N-Ethyl-2-(4-methanesulfonyl-phenyl)-N-{1-[3-(4-methylsulfanyl-phenyl)-3-phenyl-propyl]-piperidin-4-yl}-acetamide 330897 N-ethyl-2-(4-(methylsulfonyl)phenyl)-N-(1-(3-(4-(methylsulfonyl)phenyl)-3-phenylpropyl)piperidin-4-yl)acetamide 330898 N-{1-[3-(4-tert-Butoxyamino-phenyl)-3-phenyl-propyl]-piperidin-4-yl}-N-ethyl-2-(4-methanesulfonyl-phenyl)-acetamide 330900 2-[1'-cyclooctylmethyl-2-oxospiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]ethyl acetate 330983 N,3-diphenyl-1H-indazol-6-amine 330984 (2-Chloro-phenyl)-(3-phenyl-1H-indazol-6-yl)-amine 330994 4-[6-(2-Chloro-phenylamino)-1H-indazol-3-yl]-benzoic acid 331002 3-[6-(2-Chloro-phenylamino)-1H-indazol-3-yl]-benzamide 331003 3-Chloro-7-{2-[(R)-4-(6-fluoro-naphthalen-1-yl)-2-methyl-piperazin-1-yl]-ethyl}-4,7-dihydro-5H-thieno[2,3-c]pyran-2-carboxylic acid amide 331009 3-[6-(2-Chloro-phenylamino)-1H-indazol-3-yl]-benzoic acid 331010 3-[6-(2-Chloro-phenylamino)-1H-indazol-3-yl]-N-(3-morpholin-4-yl-propyl)-benzamide 331023 3-[6-(2-Chloro-phenylamino)-1H-indazol-3-yl]-N-(2-dimethylamino-ethyl)-benzamide 331024 3-(6-(2-chlorophenylamino)-1H-indazol-3-yl)-N-(piperidin-4-yl)benzamide 331033 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {1-(4-chloro-benzyl)-2-[4-(1-methanesulfonyl-1,2,3,4-tetrahydro-quinolin-8-yl)-piperazin-1-yl]-2-oxo-ethyl}-amide 331034 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {1-(4-chloro-benzyl)-2-[4-(1-methanesulfonyl-2,3-dihydro-1H-indol-7-yl)-piperazin-1-yl]-2-oxo-ethyl}-amide 331072 [2-(3-Fluoro-phenyl)-ethyl]-(5-methoxy-1,2,3,4-tetrahydro-naphthalen-1-ylmethyl)-methyl-amine 331085 N-((S)-1-{4-[2-(2,6-Difluoro-benzenesulfonyl)-4-trifluoromethyl-benzyl]-phenyl}-ethyl)-methanesulfonamide 331086 N-((S)-1-{4-[4-Chloro-2-(4-chloro-benzoyl)-benzenesulfonyl]-phenyl}-ethyl)-methanesulfonamide 331087 N-[(S)-1-(4-{4-Chloro-2-[1-(2-fluoro-phenyl)-1-hydroxy-ethyl]-benzenesulfonyl}-phenyl)-ethyl]-methanesulfonamide 331094 N-((S)-1-{4-[4-Trifluoromethoxy-2-(2-trifluoromethoxy-benzenesulfonyl)-benzyl]-phenyl}-ethyl)-methanesulfonamide 331095 N-[1-(4-{(S)-4-Chloro-2-[1-(4-chloro-phenyl)-1-hydroxy-ethyl]-benzenesulfonyl}-phenyl)-ethyl]-methanesulfonamide 331096 N-[(S)-1-(4-{1-[4-Chloro-2-(4-chloro-benzenesulfonyl)-phenyl]-propyl}-phenyl)-ethyl]-methanesulfonamide 331101 N-((S)-1-{4-[2-(3-Fluoro-benzenesulfonyl)-4-trifluoromethyl-benzyl]-phenyl}-ethyl)-methanesulfonamide 331102 N-[(S)-1-(4-{[4-Chloro-2-(4-chloro-benzenesulfonyl)-phenyl]-[(E)-methoxyimino]-methyl}-phenyl)-ethyl]-methanesulfonamide 331106 N-((S)-1-{4-[4-Trifluoromethoxy-2-(3-trifluoromethyl-benzenesulfonyl)-benzyl]-phenyl}-ethyl)-methanesulfonamide 331107 N-((S)-1-{4-[2-(2-Fluoro-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-methanesulfonamide 331108 N-[(S)-1-(4-{1-[2-(2-Fluoro-benzenesulfonyl)-4-trifluoromethoxy-phenyl]-vinyl}-phenyl)-ethyl]-methanesulfonamide 331109 3-(2-Dimethylamino-ethyl)-1-methyl-1H-indol-4-ol 331112 N-{(S)-1-[4-(2-Benzenesulfonyl-4-chloro-benzenesulfonyl)-phenyl]-ethyl}-methanesulfonamide 331113 N-((S)-1-{4-[4-Chloro-2-(2-chloro-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-methanesulfonamide 331114 Phosphoric acid mono-[3-(2-dimethylamino-ethyl)-1-methyl-1H-indol-4-yl] ester 331115 1-Butyl-3-(2-dimethylamino-ethyl)-1H-indol-4-ol 331116 Phosphoric acid mono-[1-butyl-3-(2-dimethylamino-ethyl)-1H-indol-4-yl] ester 331120 N-((S)-1-{4-[4-Chloro-2-(3-chloro-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-methanesulfonamide 331121 N-((S)-1-{4-[4-Chloro-2-(4-chloro-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-methanesulfonamide 331122 3-(2-Dimethylamino-ethyl)-1H-indol-6-ol 331123 3-(2-Dimethylamino-ethyl)-2-methyl-1H-indol-4-ol 331124 [2-(4-Fluoro-1H-indol-3-yl)-ethyl]-dimethyl-amine 331126 (S)-N-(1-(4-(4-chloro-2-(2-fluorophenylsulfonyl)phenylsulfonyl)phenyl)ethyl)methanesulfonamide 331127 N-((S)-1-{4-[4-Chloro-2-(2-trifluoromethoxy-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-methanesulfonamide 331128 3-[2-(4-Methyl-piperazin-1-yl)-ethyl]-1H-indol-4-ol 331129 3-[2-(3,4-Dihydro-2H-quinolin-1-yl)-ethyl]-1H-indol-4-ol 331132 N-{(S)-1-[4-(2-Benzenesulfonyl-4-methoxy-benzenesulfonyl)-phenyl]-ethyl}-methanesulfonamide 331133 3-(2-Pyrrolidin-1-yl-ethyl)-1H-indol-4-ol 331134 3-Dimethylaminomethyl-1H-indol-4-ol 331137 N-((S)-1-{4-[2-(4-Chloro-benzenesulfonyl)-4-methoxy-benzenesulfonyl]-phenyl}-ethyl)-methanesulfonamide 331138 N-((S)-1-{4-[2-(4-Chloro-benzenesulfonyl)-4-hydroxy-benzenesulfonyl]-phenyl}-ethyl)-methanesulfonamide 331139 3-Dimethylaminomethyl-1-methyl-1H-indol-4-ol 331140 3-(3-Dimethylamino-propyl)-1H-indol-4-ol 331141 3-(2-Dimethylamino-propyl)-1H-indol-4-ol 331142 1-(2-Dimethylamino-ethyl)-1H-indol-4-ol 331145 N-((S)-1-{4-[2-(4-Chloro-benzenesulfonyl)-4-cyclopentyloxy-benzenesulfonyl]-phenyl}-ethyl)-methanesulfonamide 331150 N-((S)-1-{4-[2-(4-Chloro-benzenesulfonyl)-4-trifluoromethyl-benzenesulfonyl]-phenyl}-ethyl)-methanesulfonamide 331151 N-((S)-1-{4-[2-(4-Chloro-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-methanesulfonamide 331153 N-((S)-1-{4-[2-(2-Fluoro-benzenesulfonyl)-4-methyl-benzenesulfonyl]-phenyl}-ethyl)-methanesulfonamide 331154 N-((S)-1-{4-[2-(2-Fluoro-benzenesulfonyl)-4-trifluoromethyl-benzenesulfonyl]-phenyl}-ethyl)-methanesulfonamide 331156 N-((R)-1-{4-[4-Methoxy-2-(4-methoxy-benzenesulfonyl)-benzenesulfonyl]-phenyl}-ethyl)-methanesulfonamide 331158 N-(1-{4-[2-(2-Fluoro-benzenesulfonyl)-4-trifluoromethoxy-benzoyl]-phenyl}-ethyl)-methanesulfonamide 331160 N-(1-{4-[4-Methoxy-2-(4-methoxy-benzenesulfonyl)-benzenesulfonyl]-phenyl}-1-methyl-ethyl)-methanesulfonamide 331161 N-{4-[4-Methoxy-2-(4-methoxy-benzenesulfonyl)-benzenesulfonyl]-benzyl}-methanesulfonamide 331162 N-(1-{4-[4-Chloro-2-(4-chloro-benzenesulfonyl)-benzoyl]-phenyl}-ethyl)-methanesulfonamide 331168 N-((S)-1-{4-[4-Methoxy-2-(4-methoxy-benzenesulfonyl)-benzyl]-phenyl}-ethyl)-methanesulfonamide 331169 N-((S)-1-{4-[4-Chloro-2-(4-chloro-benzenesulfonyl)-benzyl]-phenyl}-ethyl)-methanesulfonamide 331170 N-[(S)-1-(4-{4-Chloro-2-[1-(2-fluoro-phenyl)-vinyl]-benzenesulfonyl}-phenyl)-ethyl]-methanesulfonamide 331171 N-((S)-1-{4-[4-Chloro-2-(4-chloro-phenylamino)-benzenesulfonyl]-phenyl}-ethyl)-methanesulfonamide 331176 N-((S)-1-{4-[2-(2-Fluoro-benzenesulfonyl)-4-trifluoromethoxy-benzyl]-phenyl}-ethyl)-methanesulfonamide 331177 N-((S)-1-{4-[2-(2-Fluoro-benzenesulfonyl)-4-trifluoromethyl-benzyl]-phenyl}-ethyl)-methanesulfonamide 331178 N-((S)-1-{4-[4-Chloro-2-(4-chloro-phenoxy)-benzenesulfonyl]-phenyl}-ethyl)-methanesulfonamide 331179 N-((S)-1-{4-[4-Chloro-2-(4-chloro-benzyl)-benzenesulfonyl]-phenyl}-ethyl)-methanesulfonamide 331277 11-[2-Benzoimidazol-1-yl-eth-(E)-ylidene]-6,11-dihydro-dibenzo[b,e]oxepine-2-carboxylic acid 331319 {11-[2-(4-Benzyl-piperidin-1-yl)-eth-(E)-ylidene]-6,11-dihydro-dibenzo[b,e]oxepin-2-yl}-acetic acid 331330 1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]-4-[2-(2-{1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydro-4-pyridinylcarboxamido}ethoxy)ethylcarbamoyl]hexahydropyridine 331331 1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]-4-{2-[2-(2-{1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydro-4-pyridinylcarboxamido}ethoxy)ethoxy]ethylcarbamoyl}hexahydropyridine 331332 1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]-4-{2-[2-(3-{1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydro-4-pyridinylcarboxamido}propoxy)ethoxy]ethoxymethylcarbamoyl}hexahydropyridine 331333 4-Amino-5-chloro-2-methoxy-benzoic acid 2-[4-(11-amino-undecanoylamino)-piperidin-1-yl]-ethyl ester 331336 1-[2-(4-amino-5-chloro-2-hydroxyphenylcarbonyloxy)ethyl]-4-(5-{1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydro-4-pyridinylcarboxamido}pentylcarboxamido)hexahydropyridine 331338 4-(2-{1-[2-(4-amino-5-chloro-2-hydroxyphenylcarbonyloxy)ethyl]hexahydro-4-pyridinylcarbamoyl}ethylcarboxamido)-1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydropyridine 331339 4-(3-{1-[2-(4-amino-5-chloro-2-hydroxyphenylcarbonyloxy)ethyl]hexahydro-4-pyridinylcarbamoyl}propylcarboxamido)-1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydropyridine 331340 1-[2-(4-amino-5-chloro-2-hydroxyphenylcarbonyloxy)ethyl]-4-(5-{1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydro-4-pyridinylcarbamoyl}pentylcarboxamido)hexahydropyridine 331341 4-(10-{1-[2-(4-amino-5-chloro-2-hydroxyphenylcarbonyloxy)ethyl]hexahydro-4-pyridinylcarbamoyl}decylcarboxamido)-1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydropyridine 331343 1-[2-(4-amino-5-chloro-2-hydroxyphenylcarbonyloxy)ethyl]-4-(3-{1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydro-4-pyridinylcarboxamido}propylcarbamoyl)hexahydropyridine 331344 1-[2-(4-amino-5-chloro-2-hydroxyphenylcarbonyloxy)ethyl]-4-(5-{1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydro-4-pyridinylcarboxamido}pentylcarbamoyl)hexahydropyridine 331345 1-[2-(4-amino-5-chloro-2-hydroxyphenylcarbonyloxy)ethyl]-4-(10-{1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydro-4-pyridinylcarboxamido}decylcarbamoyl)hexahydropyridine 331346 1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]-4-(2-{1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydro-4-pyridinylmethylcarbamoyl}ethylcarboxamidomethyl)hexahydropyridine 331347 1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]-4-(3-{1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydro-4-pyridinylmethylcarbamoyl}propylcarboxamidomethyl)hexahydropyridine 331348 1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]-4-(5-{1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydro-4-pyridinylmethylcarbamoyl}pentylcarboxamidomethyl)hexahydropyridine 331349 1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]-4-(10-{1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydro-4-pyridinylmethylcarbamoyl}decylcarboxamidomethyl)hexahydropyridine 331350 N-{2-(2,3-Dihydro-benzofuran-6-yl)-2-[4-(2-ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-2-propyl-phenoxy]-acetyl}-4-isopropyl-benzenesulfonamide 331351 1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]-4-{2-[2-(2-{1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydro-4-pyridinyl}ethylcarbamoyl)ethylcarboxamido]ethyl}hexahydropyridine 331352 1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]-4-{2-[3-(2-{1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydro-4-pyridinyl}ethylcarbamoyl)propylcarboxamido]ethyl}hexahydropyridine 331353 1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]-4-{2-[5-(2-{1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydro-4-pyridinyl}ethylcarbamoyl)pentylcarboxamido]ethyl}hexahydropyridine 331354 2-{4-[2-(11-{[2-(1-{2-[(4-amino-5-chloro-2-methoxyphenyl)carbonyloxy]ethyl}piperidin-4-yl)ethyl]carbamoyl}undecanamido)ethyl]piperidin-1-yl}ethyl 4-amino-5-chloro-2-methoxybenzoate 331355 1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]-4-[10-(1-benzylhexahydro-4-pyridinylcarbamoyl)decylcarboxamido]hexahydropyridine 331356 1-[2-(3-amino-4-chloro-2-methoxyphenylcarbonyloxy)ethyl]-4-(7-{4-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydro-1-pyrazinyl}-7-oxoheptanoyl)hexahydropyrazine 331357 1-[2-(3-amino-4-chloro-2-methoxyphenylcarbonyloxy)ethyl]-4-(12-{4-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydro-1-pyrazinyl}-12-oxododecanoyl)hexahydropyrazine 331358 1-[2-(3-amino-4-chloro-2-methoxyphenylcarbonyloxy)ethyl]-4-(3-{1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydro-4-pyridinylcarboxamidomethyl}benzylcarbamoyl)hexahydropyridine 331359 1-[2-(3-amino-4-chloro-2-methoxyphenylcarbonyloxy)ethyl]-4-{2-[7-(2-{1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydro-4-pyridinylcarbamoyl}ethyl)dibenzo[b,d]furan-3-yl]ethylcarboxamido}hexahydropyridine 331361 2-{4-[11-({10-[(1-{2-[(4-amino-5-chloro-2-methoxyphenyl)carbonyloxy]ethyl}piperidin-4-yl)carbamoyl]decyl}({[(piperidin-4-ylmethyl)carbamoyl]methyl})amino)undecanamido]piperidin-1-yl}ethyl 4-amino-5-chloro-2-methoxybenzoate 331379 N-[2'-(4,5-Dimethyl-isoxazol-3-ylsulfamoyl)-4-oxazol-2-yl-biphenyl-2-ylmethyl]-3,3,N-trimethyl-butyramide 331536 ethyl 8-chloro-4-imino-4,5-dihydro-[1,2,4]triazolo[1,5-a]quinoxaline-2-carboxylate 331537 ethyl 8-methyl-4-oxo-4,5-dihydro-1,2,4-triazolo[1,5-a]quinoxaline-2-carboxylate 331538 ethyl 8-acetamido-4-oxo-4,5-dihydro-[1,2,4]triazolo[1,5-a]quinoxaline-2-carboxylate 331541 (5-fluoro-4-methyl-1H-indol-2-yl)-(4-methylpiperazin-1-yl)methanone 331542 (S)-N-((1-(2-amino-2-oxoethyl)-1H-benzo[d]imidazol-2-yl)methyl)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 331559 N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-9H-fluorene-2-carboxamide 331561 (S)-N-((1H-benzo[d]imidazol-2-yl)methyl)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 331579 Biphenyl-4-carboxylic acid {4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-amide 331580 N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)benzamide 331592 isopropyl 4,5-dihydro-4-oxo-1,2,4-triazolo[1,5-a]quinoxaline-2-carboxylate 331593 benzyl 4,5-dihydro-4-oxo-1,2,4-triazolo[1,5-a]quinoxaline-2-carboxylate 331594 4,5-dihydro-4-oxo-1,2,4-triazolo[1,5-a]quinoxaline-2-benzylcarboxamide 331613 (5-fluoro-1H-benzoimidazol-2-yl)(4-methylpiperazin-1-yl)methanone 331623 (5-methyl-1H-benzoimidazol-2-yl)(4-methylpiperazin-1-yl)methanone 331624 (4-methylpiperazin-1-yl)(5-trifluoromethyl-1H-benzoimidazol-2-yl)methanone 331625 (5-fluoro-4-methyl-1H-benzoimidazol-2-yl)(4-methylpiperazin-1-yl)methanone 331626 (4,5-difluoro-1H-benzoimidazol-2-yl)(4-methylpiperazin-1-yl)methanone 331628 3-fluoro-N-(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenylamine 331633 (4-chloro-6-methyl-1H-benzoimidazol-2-yl)(4-methylpiperazin-1-yl)methanone 331634 (4,6-dichloro-1H-benzoimidazol-2-yl)(4-methylpiperazin-1-yl)methanone 331646 2-(2-(((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamido)methyl)-1H-benzo[d]imidazol-1-yl)acetic acid 331647 N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-1-naphthamide 331648 cis-N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-4-phenylcyclohexanecarboxamide 331649 (S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-N-((1-methyl-1H-benzo[d]imidazol-2-yl)methyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 331650 (S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-N-((1-benzyl-1H-benzo[d]imidazol-2-yl)methyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 331655 N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-1-naphthamide 331659 (S)-N-((1-allyl-1H-benzo[d]imidazol-2-yl)methyl)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 331667 (S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-N-((1-(cyclopropylmethyl)-1H-benzo[d]imidazol-2-yl)methyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 331668 cis-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-4-phenylcyclohexanecarboxamide 331669 trans-N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-4-phenylcyclohexanecarboxamide 331670 trans-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-4-phenylcyclohexanecarboxamide 331688 (2R,3R,4S,5R)-2-(6-(bicyclo[2.2.1]heptan-7-ylamino)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 331716 ethyl 5-methyl-4-oxo-4,5-dihydro-1,2,4-triazolo[1,5-a]quinoxaline-2-carboxylate 331719 diethyl 4,5-dihydro-4-oxo-1,2,4-triazolo[1,5-a]quinoxaline-2,5-dicarboxylate 331732 (7-chloro-5-methyl-1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone 331733 (4-methylpiperazin-1-yl)(6H-thieno[2,3-b]pyrrol-5-yl)methanone 331734 (2-chloro-6H-thieno[2,3-b]pyrrol-5-yl)(4-methylpiperazin-1-yl)methanone 331744 (4-methylpiperazin-1-yl)(4H-thieno[3,2-b]pyrrol-5-yl)methanone 331745 (2-chloro-4H-thieno[3,2-b]pyrrol-5-yl)(4-methylpiperazin-1-yl)methanone 331746 (4-methylpiperazin-1-yl)-(3-methyl-4H-thieno[3,2-b]pyrrol-5-yl)-methanone 331747 (2-chloro-3-methyl-4H-thieno[3,2-b]pyrrol-5-yl)(4-methylpiperazin-1-yl)methanone 331748 (1H-benzoimidazol-2-yl)(4-methylpiperazin-1-yl)methanone 331749 (4-methyl-1H-benzoimidazol-2-yl)(4-methylpiperazin-1-yl)methanone 331756 2-(5-chloro-1H-benzo[d]imidazol-2-yl)quinoxaline 331760 (5-trifluoromethyl-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone 331762 7,8-Dihydro-3H,6H-5-thia-1,2,3,4,8a-pentaaza-cyclopenta[b]naphthalen-9-one 331771 2-(1H-imidazo[4,5-c]pyridin-2-yl)quinoxaline 331780 2-(4-methyl-1H-benzo[d]imidazol-2-yl)quinoxaline 331781 2-(4-chloro-1H-benzo[d]imidazol-2-yl)quinoxaline 331782 2-(4-(methylthio)-1H-benzo[d]imidazol-2-yl)quinoxaline 331789 2-(4-(ethylthio)-1H-benzo[d]imidazol-2-yl)quinoxaline 331790 2-(4-nitro-1H-benzo[d]imidazol-2-yl)quinoxaline 331800 8-methyl-2-phenyl-[1,2,4]triazolo[1,5-a]quinoxalin-4(5H)-one 331805 4,5-dihydro-8-methyl-2-(4-methoxyphenyl)-1,2,4-triazolo[1,5-a]quinoxalin-4-one 331812 8-chloro-2-phenyl-[1,2,4]triazolo[1,5-a]quinoxalin-4(5H)-one 331823 2-(1H-benzo[d]imidazol-2-yl)quinoxaline 331824 5-methyl-2-phenyl-[1,2,4]triazolo[1,5-a]quinoxalin-4(5H)-one 331829 4,5-dihydro-5,8-dimethyl-2-phenyl-1,2,4-triazolo[1,5-a]quinoxalin-4-one 331830 8-chloro-2-phenyl-[1,2,4]triazolo[1,5-a]quinoxalin-4-amine 331835 8-chloro-2-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-a]quinoxalin-4-amine 331836 2,5,8-trimethyl-4,7-dihydro-1H-1,3,4,6,7,9-hexaaza-trindene 331837 7-methyl-6,7-dihydro-3H-thiazolo[3,2-a][1,2,3]triazolo[4,5-d]pyrimidin-9-one 331841 2-phenyl-[1,2,4]triazolo[1,5-a]quinoxalin-4(5H)-one 331842 2-ethyl-5,8-dimethyl-4,7-dihydro-1H-benzo[1,2-d:3,4-d':5,6-d'']-triimidazole 331843 2,5-diethyl-8-methyl-4,7-dihydro-1H-benzo[1,2-d:3,4-d':5,6-d'']-triimidazole 331844 2,5,8-triethyl-4,7-dihydro-1H-benzo[1,2-d:3,4-d':5,6-d'']-triimidazole 331857 ethyl 2-(2-(((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamido)methyl)-1H-benzo[d]imidazol-1-yl)acetate 331865 2-(5,6-dimethyl-1H-benzo[d]imidazol-2-yl)quinoxaline 331866 2-(6-chloro-4-methyl-1H-benzo[d]imidazol-2-yl)quinoxaline 331867 2-(4,6-dichloro-1H-benzo[d]imidazol-2-yl)quinoxaline 331921 (R)-N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methyl-2,3-dihydrobenzofuran-2-carboxamide 331928 N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methyl-6-(methylsulfonamido)chroman-2-carboxamide 331929 (S)-N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methyl-2,3-dihydrobenzofuran-2-carboxamide 331937 (R)-N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methylchroman-2-carboxamide 331943 N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methylbenzofuran-2-carboxamide 331948 5-acetamido-N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methyl-2,3-dihydrobenzofuran-2-carboxamide 331949 methyl (R)-2-(((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)(methyl)carbamoyl)-2,3-dihydrobenzofuran-5-ylcarbamate 331956 methyl ((S)-2-(((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)(methyl)carbamoyl)chroman-6-yl)methylcarbamate 331961 (S)-N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methylchroman-2-carboxamide 331962 6-acetamido-N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methylchroman-2-carboxamide 331979 3-(Dmt-Tic-NH-propyl)-6-(Dmt-Tic-NH-butyl)-2-(1H)-pyrazinone 331980 3-(Dmt-Tic-NH-butyl)-6-(Dmt-Tic-NH-propyl)-2-(1H)-pyrazinone 331981 1,6-bis-(N,N-dimethyl-Dmt-Tic-NH)hexane 331982 3,6-bis-(N,N-dimethyl-Dmt-Tic-NH-propyl)-2(1H)-pyrazinone 331983 3-(Dmt-Tic-NH-ethyl)-6-(Dmt-Tic-NH-butyl)-2-(1H)-pyrazinone 332012 1,4-bis-(Dmt-Tic-amino)butane 332013 1,6-bis-(Dmt-Tic-amino)hexane 332014 1,10-bis-(Dmt-Tic-amino)decane 332018 6-Methylsulfamoyl-chroman-2-carboxylic acid [(S)-2-((S)-3-hydroxy-pyrrolidin-1-yl)-1-phenyl-ethyl]-methyl-amide 332024 (R)-N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methyl-6-(propylsulfonamido)chroman-2-carboxamide 332025 (S)-N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methyl-5-(methylsulfonamido)-2,3-dihydrobenzofuran-2-carboxamide 332032 (R)-N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methyl-7-(methylsulfonamido)-2,3-dihydrobenzofuran-2-carboxamide 332053 (S)-N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methyl-6-(propylsulfonamido)chroman-2-carboxamide 332060 (R)-N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methyl-6-(methylsulfonamidomethyl)chroman-2-carboxamide 332061 (S)-N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methyl-6-(methylsulfonamidomethyl)chroman-2-carboxamide 332068 (S)-N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methyl-7-(methylsulfonamido)-2,3-dihydrobenzofuran-2-carboxamide 332069 5-Methylsulfamoyl-2,3-dihydro-benzofuran-2-carboxylic acid [(S)-2-((S)-3-hydroxy-pyrrolidin-1-yl)-1-phenyl-ethyl]-methyl-amide 332075 (R)-N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methyl-5-(propylsulfonamidomethyl)-2,3-dihydrobenzofuran-2-carboxamide 332101 (R)-N-(2-(3-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-3-oxoprop-1-enyl)-5-chlorophenyl)acetamide 332104 methyl ((R)-2-(((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)(methyl)carbamoyl)chroman-6-yl)methylcarbamate 332116 (S)-N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methyl-5-(propylsulfonamidomethyl)-2,3-dihydrobenzofuran-2-carboxamide 332126 methyl 2-(((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)(methyl)carbamoyl)chroman-6-ylcarbamate 332127 6-Sulfamoyl-chroman-2-carboxylic acid [(S)-2-((S)-3-hydroxy-pyrrolidin-1-yl)-1-phenyl-ethyl]-methyl-amide 332136 methyl (S)-2-(((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)(methyl)carbamoyl)-2,3-dihydrobenzofuran-5-ylcarbamate 332137 (R)-N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methyl-5-(methylsulfonamido)-2,3-dihydrobenzofuran-2-carboxamide 332139 N-[1-[2-phenylethyl]-4-piperidinyl]-N-phenyl-2-[(+/-)-[18F]fluoropropanamide 332140 N-[1-[2-(2-thienyl)ethyl]-4-piperidinyl]-N-phenyl-2-[(+/-)-[18F]fluoropropanamide 332149 N-(2-(3-(3-(4-fluorobenzyl)-3,8-diaza-bicyclo[3.2.1]octan-8-yl)-3-oxoprop-1-enyl)-5-chloro-4-methoxyphenyl)acetamide 332156 N-(2-(3-(3-(4-fluorobenzyl)-3,8-diaza-bicyclo[3.2.1]octan-8-yl)-3-oxoprop-1-enyl)-5-chlorophenyl)-2-(dimethylamino)acetamide 332167 (R)-N-(2-(3-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-3-oxopropyl)-5-chlorophenyl)acetamide 332172 {2-[2-(2-chlorobenzyloxy)phenoxy]ethyl}-2-[2,6-dimethoxyphenoxy)ethyl]amine 332175 (R)-N-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethylamino)-5-chlorophenyl)acetamide 332178 3,6-bis(Dmt-Tic-NH-butyl)-2(1H)-pyrazinone 332191 {2-[2-(3-chlorobenzyloxy)phenoxy]ethyl}-[2-(2,6-dimethoxyphenoxy)ethyl]amine 332200 3,6-bis(Dmt-Tic-NH-ethyl)-2(1H)-pyrazinone 332203 N-(2-(3-((2R,5S)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl)-3-oxoprop-1-enyl)-5-chlorophenyl)acetamide 332204 N-(2-(3-((2S,5R)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl)-3-oxoprop-1-enyl)-5-chlorophenyl)acetamide 332207 N-(2-(3-((1R,4R)-5-(4-fluorobenzyl)-2,5-diaza-bicyclo[2.2.1]heptan-2-yl)-3-oxoprop-1-enyl)-5-chlorophenyl)acetamide 332212 N-(2-(3-(4-(4-fluorobenzyl)piperazin-1-yl)-3-oxoprop-1-enyl)-5-chlorophenyl)acetamide 332213 4-(2-((R)-4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethyl)-7-chloro-6-methoxy-3,4-dihydroquinazolin-2(1H)-one 332214 N-(2-(3-(3-(4-fluorobenzyl)-3,8-diaza-bicyclo[3.2.1]octan-8-yl)-3-oxoprop-1-enyl)-5-chlorophenyl)acetamide 332219 (2S,5S,11bR,1'S)-2-[Nalpha-(tert-butoxycarbonyl)-L-tryptophyl)amino]-5-[(1'-carbamoyl-2'-phenyl)ethyl]carbamoyl-3-oxo-2,3,5,6,11,11b-hexahydro-1H-indolizino-[8,7-b]indole 332224 fluoromethyl 1-(2-phenylethyl)-4-(N-phenylpropanamido)piperidine-4-carboxylate 332225 (R)-N-(2-(1-(4-fluorobenzyl)-3-methylpiperazine-4-carbonyl)-5-chloro-1H-indol-7-yl)acetamide 332226 (R)-N-(2-(1-(4-fluorobenzyl)-3-methylpiperazine-4-carbonyl)-5-chlorobenzofuran-7-yl)acetamide 332231 2-fluoroethyl 1-(2-phenylethyl)-4-(N-phenylpropanamido)piperidine-4-carboxylate 332232 N[1-(5-[18F]fluoropentyl)-4-piperidinyl]-N-phenylpropanamide 332246 3,6-bis(Dmt-Tic-NH-propyl)-2(1H)-pyrazinone 332258 N-(2-(3-(8-(4-fluorobenzyl)-3,8-diaza-bicyclo[3.2.1]octan-3-yl)-3-oxoprop-1-enyl)-5-chlorophenyl)acetamide 332259 (R)-1-(2-(3-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-3-oxoprop-1-enyl)-5-chlorophenyl)urea 332264 methyl 4-[(N-1-oxopropyl)-N-phenylamino]-1-(5-[18F]-fluoropentyl)-4-piperidinecarboxylate 332268 (R)-N-(2-(3-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-3-oxoprop-1-enyl)-5-chloro-4-methoxyphenyl)acetamide 332269 N-(6-(3-(3-(4-fluorobenzyl)-3,8-diaza-bicyclo[3.2.1]octan-8-yl)-3-oxoprop-1-enyl)quinolin-7-yl)acetamide 332270 clopenphendioxan 332278 (R)-N-(3-(3-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-3-oxoprop-1-enyl)naphthalen-2-yl)acetamide 332279 (R)-N-(6-(3-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-3-oxoprop-1-enyl)quinolin-7-yl)acetamide 332282 (2S,5S,11bR,1'S)-2-[Nalpha-(tert-butoxycarbonyl)-D-tryptophyl)amino]-5-[(1'-carbamoyl-2'-phenyl)ethyl]carbamoyl-3-oxo-2,3,5,6,11,11b-hexahydro-1H-indolizino-[8,7-b]indole 332283 (2S,5S,11bR,1'R)-2-[Nalpha-(tert-butoxycarbonyl)-L-tryptophyl)amino]-5-[(1'-carbamoyl-2'-phenyl)ethyl]carbamoyl-3-oxo-2,3,5,6,11,11b-hexahydro-1H-indolizino-[8,7-b]indole 332295 (2S,5S,11bR,1'R)-2-[Nalpha-(tert-butoxycarbonyl)-D-tryptophyl)amino]-5-[(1'-carbamoyl-2'-phenyl)ethyl]carbamoyl-3-oxo-2,3,5,6,11,11b-hexahydro-1H-indolizino-[8,7-b]indole 332296 (2R,5R,11bS,1'S)-2-[Nalpha-(tert-butoxycarbonyl)-L-tryptophyl)amino]-5-[(1'-carbamoyl-2'-phenyl)ethyl]carbamoyl-3-oxo-2,3,5,6,11,11b-hexahydro-1H-indolizino-[8,7-b]indole 332333 3-Chloro-2-ethoxy-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 332337 2-(4-Ethylpiperazin-1-yl)-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 332352 (2R,5R,11bS,1'S)-2-[Nalpha-(tert-butoxycarbonyl)-D-tryptophyl)amino]-5-[(1'-carbamoyl-2'-phenyl)ethyl]carbamoyl-3-oxo-2,3,5,6,11,11b-hexahydro-1H-indolizino-[8,7-b]indole 332354 (2R,5R,11bS,1'R)-2-[Nalpha-(tert-butoxycarbonyl)-D-tryptophyl)amino]-5-[(1'-carbamoyl-2'-phenyl)ethyl]carbamoyl-3-oxo-2,3,5,6,11,11b-hexahydro-1H-indolizino-[8,7-b]indole 332390 2-(2-methoxyethoxy)-5-{[6-methoxy-7-(2-methoxyethoxy)-quinazolin-4-yl]amino}benzo-1,4-quinone 332394 3,6-bis(Dmt-Tic-NH-methyl)-2(1H)-pyrazinone 332400 (R)-N-(2-(3-(4-(4-fluorobenzyl)-2-methyl-1,4-diazepan-1-yl)-3-oxoprop-1-enyl)-5-chlorophenyl)acetamide 332444 2-{[4-(diethylamino)phenyl][4-(diethyliminio)cyclohexa-2,5-dien-1-ylidene]methyl}-5-({[6-oxo-6-({2-[2-(2-{4-[2-oxo-2-(6-oxo-5,6-dihydro-11H-pyrido[2,3-b][1,4]-benzodiazepin-11-yl)ethylpiperazin-1-yl}ethoxy)ethoxy]ethyl}amino)hexyl]amino}sulfonyl)]-benzene 332465 7-(naphthalen-2-yloxyethoxy)-2-morpholin-4-yl-chromen-4-one 332472 2-(2-(benzenesulfonyl)ethoxy)-2-morpholin-4-yl-chromen-4-one 332474 2-[3-(Ethylamino)phenoxy]-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 332491 4-ethoxy-N-{2-oxo-2-[2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}-N-phenylbenzenesulfonamide 332510 1-(3-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridazin-3-yl)phenyl)ethanone 332520 2-Methoxy-5-({6-methoxy-7-[(1-methylpiperidin-4-yl)methoxy]quinazolin-4-yl}amino)benzo-1,4-quinone 332532 7-(1-oxypyridin-2-ylmethoxy)-2-morpholin-4-yl-chromen-4-one 332563 8-biphenyl-2-yl-2-morpholin-4-ylchromen-4-one 332567 3-(2-morpholin-4-yl-4-oxo-4H-chromen-8-yl)benzoic acid ethyl ester 332580 2-morpholin-4-yl-8-(4-trifluoromethoxyphenyl)chromen-4-one 332581 2-morpholin-4-yl-8-naphthalen-2-ylchromen-4-one 332587 8-furan-2-yl-2-morpholin-4-ylchromen-4-one 332589 2-morpholin-4-yl-8-(2-trifluoromethylphenyl)chromen-4-one 332591 2-Methoxy-5-{[6-methoxy-7-(3-pyrrolidin-1-ylpropoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 332596 2-[3-(2-morpholin-4-yl-4-oxo-4H-chromen-8-yl)-benzyl]-isoindole-1,3-dione 332600 1-ethyl-2-[(1E,3E)-3-(1-ethylquinolin-2-(1H)-ylidene)prop-1-enyl]-6-{[6-oxo-6-({2-[2-(2-{4-[2-oxo-2-(6-oxo-5,6-dihydro-11H-pyrido[2,3-b][1,4]benzodiazepin-11-yl)ethyl]-piperazin-1-yl}ethoxy)ethoxy]ethyl}amino)hexanoyl]-amino}]quinolinium iodide 332603 N-[4-(2-morpholin-4-yl-4-oxo-4H-chromen-8-yl)phenyl]acetamide 332615 atosiban 332622 8-[2-(4-fluorophenyl)vinyl]-2-morpholin-4-ylchromen-4-one 332635 2-morpholin-4-yl-8-(3-trifluoromethoxyphenyl)-chromen-4-one 332640 7-(2-(ethanesulfonyl)ethoxy)-2-morpholin-4-yl-chromen-4-one 332646 7-(1-oxypyridin-4-ylmethoxy)-2-morpholin-4-yl-chromen-4-one 332647 7-(2-(phenylmethanesulfonyl)ethoxy)-2-morpholin-4-yl-chromen-4-one 332651 [2-(2,6-dimethoxyphenoxy)ethyl]-{2-[2-(4-methoxy-benzyloxy)phenoxy]ethyl}amine 332653 N-[3-(2-morpholin-4-yl-4-oxo-4H-chromen-8-yl)phenyl]acetamide 332660 N-(4-chloro-2-methylphenyl)-2-(N-(4-methoxyphenyl)phenylsulfonamido)acetamide 332661 8-(4-chlorophenyl)-2-morpholin-4-ylchromen-4-one 332668 8-(2-hydroxymethylphenyl)-2-morpholin-4-ylchromen-4-one 332669 8-(3-hydroxymethylphenyl)-2-morpholin-4-ylchromen-4-one 332691 N-(4-chlorophenyl)-4-ethoxy-N-{2-[(2E)-2-(2-hydroxybenzylidene)hydrazino]-2-oxoethyl}benzenesulfonamide 332710 N-(3-chloro-2-methylphenyl)-2-(3,4-dimethoxy-N-p-tolylphenylsulfonamido)acetamide 332714 [2-(2,6-dimethoxyphenoxy)ethyl]-{2-[2-(3-methyl-benzyloxy)phenoxy]ethyl}amine 332718 SID24802020 332722 [2-(2,6-dimethoxyphenoxy)ethyl]-{2-[2-(2-methoxy-benzyloxy)phenoxy]ethyl}amine 332725 N-(2-(3,4-dihydroisoquinolin-2(1H)-yl)-2-oxoethyl)-N-p-tolylbenzenesulfonamide 332726 8-(3-hydroxyphenyl)-2-morpholin-4-ylchromen-4-one 332729 [2-(2,6-dimethoxyphenoxy)ethyl]-{2-[2-(3-methoxy-benzyloxy)phenoxy]ethyl}amine 332733 8-(4-hydroxyphenyl)-2-morpholin-4-ylchromen-4-one 332734 8-(1H-indol-5-yl)-2-morpholin-4-ylchromen-4-one 332745 N-(4-chlorophenyl)-4-ethoxy-N-{2-oxo-2-[(2E)-2-(2-pyridinylmethylene)hydrazino]ethyl}benzenesulfonamide 332754 [2-(2,6-dimethoxyphenoxy)ethyl]-{2-[2-(2-methyl-benzyloxy)phenoxy]ethyl}amine 332768 Bo(15)PZ 332825 [2-(2,6-dimethoxyphenoxy)ethyl]-{2-[2-(3-nitro-benzyloxy)phenoxy]ethyl}amine 332833 [2-(2,6-dimethoxyphenoxy)ethyl]-{2-[2-(4-nitro-benzyloxy)phenoxy]ethyl}amine 332864 2-[(2-hydroxyethyl)methylamino]benzo[h]chromen-4-one 332870 7-propoxy-2-(morpholin-4-yl)-chromen-4-one 332887 RR(17)PZ 332890 4-ethoxy-N-{2-[2-(2-hydroxybenzylidene)hydrazino]-2-oxoethyl}-N-(4-methylphenyl)benzenesulfonamide 332893 7-(4-bromobenzyloxy)-2-morpholin-4-yl-chromen-4-one 332900 7-(4-methylsulfanylbenzyloxy)-2-(morpholin-4-yl)-chromen-4-one 332902 N-[2-(2-(morpholin-4-yl)-4-oxo-4H-chromen-7-yloxy)ethyl]phthalimide 332905 [2-(2,6-dimethoxyphenoxy)ethyl]-{2-[2-(4-methyl-benzyloxy)phenoxy]ethyl}amine 332906 [2-(2,6-dimethoxyphenoxy)ethyl]-{2-[2-(2-nitro-benzyloxy)phenoxy]ethyl}amine 332912 7-(4-bromophenylethoxy)-2-morpholin-4-yl-chromen-4-one 332924 N'-(2-hydroxybenzylidene)-2-(N-(4-chlorophenyl)phenylsulfonamido)acetohydrazide 332930 7-(2-chlorobenzyloxy)-2-(morpholin-4-yl)-chromen-4-one 332931 7-(4-chlorobenzyloxy)-2-(morpholin-4-yl)-chromen-4-one 332944 7-(3-methylbenzyloxy)-2-morpholin-4-yl-chromen-4-one 332946 7-(3-fluorobenzyloxy)-2-morpholin-4-yl-chromen-4-one 332948 (S)-N-((R)-3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 332951 2-amino-N-((R)-1-(4-chloro-benzyl)-2-oxo-2-{4-[1-(phenylacetylamino-methyl)-cyclohexyl]-piperazin-1-yl}-ethyl)-2-phenyl-acetamide 332952 N-((R)-3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)isoindoline-1-carboxamide 332953 4-(2-morpholin-4-yl-4-oxo-4H-chromen-8-yl)benzoic acid benzyl ester 332956 7-(4-fluorobenzyloxy)-2-morpholin-4-yl-chromen-4-one 332960 8-(2-benzyloxyphenyl)-2-morpholin-4-ylchromen-4-one 332961 8-(3-benzyloxyphenyl)-2-morpholin-4-ylchromen-4-one 332963 (R)-N-(3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)furan-2-carboxamide 332965 N-((R)-3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)indoline-2-carboxamide 332966 3-amino-N-((R)-3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)-3-phenylpropanamide 332970 2-amino-N-((R)-3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)-3-phenylpropanamide 332976 7-(4-methoxyphenylethoxy)-2-morpholin-4-yl-chromen-4-one 332977 7-ethyloxyethoxy-2-morpholin-4-yl-chromen-4-one 332984 7-phenyloxyethoxy-2-morpholin-4-yl-chromen-4-one 332988 4-(2-morpholin-4-yl-4-oxo-4H-chromen-8-yl)benzonitrile 332993 N-((R)-1-(4-Chloro-benzyl)-2-oxo-2-{4-[1-(phenylacetylamino-methyl)-cyclohexyl]-piperazin-1-yl}-ethyl)-2-(2-fluoro-phenyl)-acetamide 332994 1-amino-N-((R)-3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)-2,3-dihydro-1H-indene-1-carboxamide 332995 (R)-N-((R)-3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 332996 7-(3,4-difluorobenzyloxy)-2-morpholin-4-yl-chromen-4-one 332997 7-(3-bromobenzyloxy)-2-morpholin-4-yl-chromen-4-one 332998 N-((R)-1-(4-chloro-benzyl)-2-oxo-2-{4-[1-(phenylacetylamino-methyl)-cyclohexyl]-piperazin-1-yl}-ethyl)-2-thiophen-2-yl-acetamide 333002 2-amino-N-((R)-3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)-3-(pyridin-4-yl)propanamide 333003 (R)-2-amino-N-(3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)-2,3-dihydro-1H-indene-2-carboxamide 333006 N-(4-methylphenyl)-N-{2-oxo-2-[2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}-2-naphthalenesulfonamide 333011 7-(2-chlorophenyloxyethoxy)-2-morpholin-4-yl-chromen-4-one 333012 (R)-N-(3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)quinoline-3-carboxamide 333017 2-(N-(3-chlorophenyl)phenylsulfonamido)-N'-(1-(2-hydroxyphenyl)ethylidene)acetohydrazide 333018 N-(4-methylphenyl)-N-{2-oxo-2-[2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}[1,1'-biphenyl]-4-sulfonamide 333019 7-(4-chlorophenyloxyethoxy)-2-morpholin-4-yl-chromen-4-one 333020 8-(4-methylnaphthalen-1-yl)-2-morpholin-4-ylchromen-4-one 333037 7-cyclohexylmethoxy-2-(morpholin-4-yl)-chromen-4-one 333038 N-(3-chloro-2-methylphenyl)-2-(N-p-tolylphenylsulfonamido)acetamide 333039 N-(3-chloro-2-methylphenyl)-2-(N-(4-chlorophenyl)phenylsulfonamido)acetamide 333040 4-(2-hydroxybenzylamino)-N-(3-phenoxyphenyl)piperidine-1-sulfonamide 333044 (R)-isobutyl 3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-ylcarbamate 333051 2-morpholin-4-yl-8-styrylchromen-4-one 333052 (R)-N-(3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)nicotinamide 333057 7-(3-chlorobenzyloxy)-2-morpholin-4-yl-chromen-4-one 333059 8-(2-acetylphenyl)-2-morpholin-4-ylchromen-4-one 333060 8-benzo[b]thiophen-3-yl-2-morpholin-4-ylchromen-4-one 333066 4-(3-chloro-4-fluorophenylamino)-6-(3-(4-methylpiperazin-1-yl)propylamino)-1,7-naphthyridine-3-carbonitrile 333067 3-(3-chloro-4-fluoro-phenyl)-1-(3'-cyano-biphenyl-4-ylmethyl)-1-(2-pyrrolidin-1-yl-ethyl)-urea 333069 2-(2-(2-(4-ethoxy-N-p-tolylphenylsulfonamido)acetyl)-1,2,3,4-tetrahydroisoquinolin-3-yl)acetamide 333072 N-[3-(2-(morpholin-4-yl)-4-oxo-4H-chromen-7-yloxy)propyl]phthalimide 333073 (R)-N-(3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)benzamide 333074 (R)-N-(3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)-4-fluorobenzamide 333075 N-[2-(3'-cyano-biphenyl-4-yl)-ethyl]-N-[(3,5-dichloro-phenylcarbamoyl)-methyl]-2-pyrrolidin-1-yl-acetamide 333080 2-(2-(2-(4-ethoxy-N-(4-methoxyphenyl)phenylsulfonamido)acetyl)-1,2,3,4-tetrahydroisoquinolin-3-yl)acetamide 333081 7-(naphthalen-2-ylmethoxy)-2-(morpholin-4-yl)-chromen-4-one 333082 7-benzoyloxy-2-(morpholin-4-yl)-chromen-4-one 333083 N-[2-(3'-cyano-biphenyl-4-yl)-ethyl]-N-[(3,5-dichloro-phenylcarbamoyl)-methyl]-2-((R)-3-hydroxy-pyrrolidin-1-yl)-acetamide 333084 N-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-yl)-5-methoxy-1H-indazol-3-amine 333085 2-(2-(4-ethoxy-N-(4-methoxyphenyl)phenylsulfonamido)acetyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 333087 7-(4-cyanobenzyloxy)-2-morpholin-4-yl-chromen-4-one 333089 N-(3'-cyano-biphenyl-4-ylmethyl)-N-[(3,5-dichloro-phenylcarbamoyl)-methyl]-3-pyrrolidin-1-yl-propionamide 333090 N-(1-((1H-indazol-6-yl)methyl)piperidin-4-yl)-5-methoxy-1H-indazol-3-amine 333091 N-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-yl)-4-methoxy-1H-indazol-3-amine 333094 7-(3-methoxybenzyloxy)-2-morpholin-4-yl-chromen-4-one 333095 7-(4-tert-butylbenzyloxy)-2-morpholin-4-yl-chromen-4-one 333097 N-(1-(2-fluoro-4-methoxybenzyl)piperidin-4-yl)-5-chloro-1H-indazol-3-amine 333098 N-[2-(3'-cyano-biphenyl-4-yl)-ethyl]-N-[(3,5-dichloro-phenylcarbamoyl)-methyl]-3-((S)-3-hydroxy-pyrrolidin-1-yl)-propionamide 333099 N-(3-(trifluoromethyl)benzyl)-4-phenoxybenzamide 333100 N-(3-hydroxy-4-(1-hydroxy-2-methylpropan-2-yl)benzyl)-4-(4-chlorophenoxy)benzamide 333104 (S)-N-(1-(2-fluorobenzyl)pyrrolidin-3-yl)-4-(thiophen-2-yl)benzamide 333105 (S)-N-(1-(4-fluorobenzyl)pyrrolidin-3-yl)-4-(thiophen-2-yl)benzamide 333106 N-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-yl)-5-methoxy-1-methyl-1H-indazol-3-amine 333107 6-(4-cyanobenzyloxy)-2-morpholin-4-yl-chromen-4-one 333108 4-(2-hydroxybenzylamino)-N-(3-(4-fluorophenoxy)phenyl)piperidine-1-sulfonamide 333113 1-(3'-cyano-biphenyl-4-ylmethyl)-3-(4-fluoro-3-trifluoromethyl-phenyl)-1-(2-pyrrolidin-1-yl-ethyl)-urea 333114 1-(3'-cyano-biphenyl-4-ylmethyl)-3-(3,5-dichloro-phenyl)-1-(3-pyrrolidin-1-yl-propyl)-urea 333119 methyl 3-(2-(morpholin-4-yl)-4-oxo-4H-chromen-7-yloxymethyl)-benzoate 333120 3-(3-chloro-4-fluoro-phenyl)-1-(3'-cyano-biphenyl-4-ylmethyl)-1-(3-pyrrolidin-1-yl-propyl)-urea 333122 N-[2-(3'-cyano-biphenyl-4-yl)-ethyl]-N-[(3,5-dichloro-phenylcarbamoyl)-methyl]-2-((S)-3-hydroxy-pyrrolidin-1-yl)-acetamide 333125 2-(2-(4-ethoxy-N-(4-methoxyphenyl)phenylsulfonamido)acetyl)isoindoline-1-carboxamide 333126 methyl 4-(2-(morpholin-4-yl)-4-oxo-4H-chromen-7-yloxymethyl)-benzoate 333128 2-amino-N-((R)-3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)-1,2,3,4-tetrahydronaphthalene-2-carboxamide 333129 N-((R)-1-(4-chloro-benzyl)-2-oxo-2-{4-[1-(phenylacetylamino-methyl)-cyclohexyl]-piperazin-1-yl}-ethyl)-2-(1,2,3,4-tetrahydro-isoquinolin-3-yl)-acetamide 333133 N-[2-(2-(morpholin-4-yl)-4-oxo-4H-chromen-6-yloxy)-methyl]-phthalimide 333134 7-hydroxy-2-(morpholin-4-yl)chromen-4-one 333135 N-(4-chlorophenyl)-3,4-dimethoxy-N-{2-oxo-2-[(2E)-2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}benzenesulfonamide 333138 7-phenylethoxy-2-morpholin-4-yl-chromen-4-one 333141 N-(1-(3-methoxybenzyl)piperidin-4-yl)-5-chloro-1H-indazol-3-amine 333142 N-(1-(3,4-dimethylbenzyl)piperidin-4-yl)-5-chloro-1H-indazol-3-amine 333153 7-(4-methylbenzyloxy)-2-morpholin-4-yl-chromen-4-one 333154 N-[(R)-1-(3'-cyano-biphenyl-4-yl)-ethyl]-N-[(3,5-dichloro-phenylcarbamoyl)-methyl]-3-((S)-3-hydroxy-pyrrolidin-1-yl)-propionamide 333155 1-(3'-cyano-biphenyl-4-ylmethyl)-3-(4-fluoro-3-trifluoromethyl-phenyl)-1-(3-pyrrolidin-1-yl-propyl)-urea 333156 1-(3'-cyano-biphenyl-4-ylmethyl)-3-(3,5-dichloro-phenyl)-1-(2-pyrrolidin-1-yl-ethyl)-urea 333158 4-(2-hydroxybenzylamino)-N-(3-(2,4-difluorophenoxy)phenyl)piperidine-1-sulfonamide 333159 N-[(S)-1-(3'-cyano-biphenyl-4-yl)-ethyl]-N-[(3,5-dichloro-phenylcarbamoyl)-methyl]-3-((S)-3-hydroxy-pyrrolidin-1-yl)-propionamide 333164 N'-(1-(2-hydroxyphenyl)ethylidene)-2-(N-phenylphenylsulfonamido)acetohydrazide 333166 N-((R)-1-(4-chloro-benzyl)-2-oxo-2-{4-[1-(phenylacetylamino-methyl)-cyclohexyl]-piperazin-1-yl}-ethyl)-2-methoxy-acetamide 333167 N-[(R)-1-(3'-cyano-biphenyl-4-yl)-ethyl]-N-[(3,5-dichloro-phenylcarbamoyl)-methyl]-4-((S)-3-hydroxy-pyrrolidin-1-yl)-butyramide 333168 N-((S)-1-(4-(trifluoromethoxy)benzyl)pyrrolidin-3-yl)-3-(thiophen-2-yl)benzamide 333171 N-(4-(trifluoromethyl)benzyl)-4-phenoxybenzamide 333172 N-((2,3-dihydro-1H-inden-5-yl)methyl)-4-phenoxybenzamide 333173 N-((R)-1-(4-chloro-benzyl)-2-oxo-2-{4-[1-(phenylacetylamino-methyl)-cyclohexyl]-piperazin-1-yl}-ethyl)-2-dimethylamino-acetamide 333174 (S)-N-(1-(3-(trifluoromethyl)benzyl)pyrrolidin-3-yl)-4-(thiophen-2-yl)benzamide 333175 (S)-N-(1-(3,4-dichlorobenzyl)pyrrolidin-3-yl)-4-(thiophen-2-yl)benzamide 333179 N-(3-(trifluoromethoxy)benzyl)-4-phenoxybenzamide 333184 (S)-N-(1-(3,4-difluorobenzyl)pyrrolidin-3-yl)-4-(thiophen-2-yl)benzamide 333185 4-(3-chloro-4-fluorophenylamino)-6-(3-morpholinopropylamino)-1,7-naphthyridine-3-carbonitrile 333188 2-morpholinobenzo[h]quinolin-4(1H)-one 333193 8-(4-acetylphenyl)-2-morpholin-4-ylchromen-4-one 333194 (1-benzo{1,3}dioxol-5-ylmethyl-piperidin-4-yl)(5-chloro-1Hindazol-3-yl)amine 333195 N-(1-(4-chlorobenzyl)piperidin-4-yl)-5-chloro-1H-indazol-3-amine 333197 N-[(S)-1-(3'-cyano-biphenyl-4-yl)-ethyl]-N-[(3,5-dichloro-phenylcarbamoyl)-methyl]-2-((S)-3-hydroxy-pyrrolidin-1-yl)-acetamide 333201 N-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-yl)-5-chloro-1-phenyl-1H-indazol-3-amine 333202 N-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-yl)-1-benzyl-5-nitro-1H-indazol-3-amine 333204 (S)-N-(1-(3-methoxybenzyl)pyrrolidin-3-yl)-4-(thiophen-2-yl)benzamide 333205 N-[1-(3'-cyano-biphenyl-4-yl)-1-methyl-ethyl]-N-[(3,5-dichloro-phenylcarbamoyl)-methyl]-2-pyrrolidin-1-yl-acetamide 333207 N-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-yl)-1-benzyl-5-chloro-1H-indazol-3-amine 333209 N-((S)-1-(4-chlorobenzyl)pyrrolidin-3-yl)-3-(thiophen-2-yl)benzamide 333210 (R)-4-(3-chloro-4-fluorophenylamino)-6-(1-phenylpropylamino)-1,7-naphthyridine-3-carbonitrile 333219 N-(3'-cyano-biphenyl-4-ylmethyl)-N-[(3,5-dichloro-phenylcarbamoyl)-methyl]-2-pyrrolidin-1-yl-acetamide 333223 N-(1-benzylpiperidin-4-yl)-5-chloro-1H-indazol-3-amine 333230 N-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-yl)-5-methyl-1H-indazol-3-amine 333231 N-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-yl)-5-nitro-1H-indazol-3-amine 333237 N-(1-((2,3-dihydrobenzo[b][1,4]dioxin-6-yl)methyl)piperidin-4-yl)-5-nitro-1H-indazol-3-amine 333238 3-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-ylamino)-1H-indazole-5-carbonitrile 333239 6-(2-morpholinoethylamino)-4-(4-(phenylthio)phenylamino)-1,7-naphthyridine-3-carbonitrile 333240 5-chloro-N-(1-((7-methoxybenzo[d][1,3]dioxol-5-yl)methyl)piperidin-4-yl)-1H-indazol-3-amine 333241 (S)-N-(1-(4-(trifluoromethyl)benzyl)pyrrolidin-3-yl)-4-(thiophen-2-yl)benzamide 333242 N-((S)-1-(4-(trifluoromethyl)benzyl)pyrrolidin-3-yl)-3-(thiophen-2-yl)benzamide 333245 4-(3-chloro-4-fluorophenylamino)-6-(pyridin-3-ylmethylamino)-[1,7]naphthyridine-3-carbonitrile 333246 6-(benzylamino)-4-(3-chloro-4-fluorophenylamino)-1,7-naphthyridine-3-carbonitrile 333247 N-[(S)-1-(4-Methyl-benzyl)-pyrrolidin-3-yl]-3-thiophen-2-yl-benzamide 333256 N-(3'-cyano-biphenyl-4-ylmethyl)-N-[(3,5-dichloro-phenylcarbamoyl)-methyl]-2-((R)-3-hydroxy-pyrrolidin-1-yl)-acetamide 333265 N-(3'-cyano-biphenyl-4-ylmethyl)-N-[(3,5-dichloro-phenylcarbamoyl)-methyl]-2-((S)-3-hydroxy-pyrrolidin-1-yl)-acetamide 333266 2-morpholin-4-yl-8-phenoxathiin-4-ylchromen-4-one 333267 8-(4-benzyloxyphenyl)-2-morpholin-4-ylchromen-4-one 333272 N-[(R)-1-(3'-cyano-biphenyl-4-yl)-ethyl]-N-[(3,5-dichloro-phenylcarbamoyl)-methyl]-2-((S)-3-hydroxy-pyrrolidin-1-yl)-acetamide 333276 4-(4-chloro-2-fluorophenylamino)-6-(2-morpholinoethylamino)-1,7-naphthyridine-3-carbonitrile 333277 6-[(2-morpholin-4-ylethyl)amino]-4-[(4-phenoxyphenyl)amino]-[1,7]naphthyridine-3-carbonitrile 333279 2-((R)-3-acetylamino-pyrrolidin-1-yl)-N-[2-(3'-cyano-biphenyl-4-yl)-ethyl]-N-[(3,5-dichloro-phenylcarbamoyl)-methyl]-acetamide 333284 4-(4-benzoylphenylamino)-6-(2-morpholinoethylamino)-1,7-naphthyridine-3-carbonitrile 333285 4-(3-chloro-4-fluorophenylamino)-6-(2-morpholino-1-phenylethylamino)-1,7-naphthyridine-3-carbonitrile 333286 N-[2-(3'-cyano-biphenyl-4-yl)-ethyl]-N-[(3,5-dichloro-phenylcarbamoyl)-methyl]-3-pyrrolidin-1-yl-propionamide 333289 (S)-4-(3-chloro-4-fluorophenylamino)-6-(1-phenylethylamino)-1,7-naphthyridine-3-carbonitrile 333290 (R)-4-(3-chloro-4-fluorophenylamino)-6-(1-phenylethylamino)-1,7-naphthyridine-3-carbonitrile 333291 N-[2-(3'-cyano-biphenyl-4-yl)-ethyl]-N-[(3,5-dichloro-phenylcarbamoyl)-methyl]-3-((R)-3-hydroxy-pyrrolidin-1-yl)-propionamide 333299 N-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-yl)-1H-indazol-3-amine 333300 5-chloro-N-(1-(naphthalen-2-ylmethyl)piperidin-4-yl)-1H-indazol-3-amine 333301 5-chloro-N-(1-((2,3-dihydrobenzo[b][1,4]dioxin-6-yl)methyl)piperidin-4-yl)-1H-indazol-3-amine 333304 (S)-N-(1-(benzo[d][1,3]dioxol-5-ylmethyl)pyrrolidin-3-yl)-4-(thiophen-2-yl)benzamide 333305 1-(4-amino-2,3-dihydro-1,2,5-oxadiazol-3-yl)-5-(piperidin-1-ylmethyl)-N'-(pyridin-4-ylmethylene)-4,5-dihydro-1H-1,2,3-triazole-4-carbohydrazide 333306 4-(5-(piperidin-1-ylmethyl)-4-(5-(pyridin-4-yl)-4H-1,2,4-triazol-3-yl)-4,5-dihydro-1,2,3-triazol-1-yl)-4,5-dihydro-1,2,5-oxadiazol-3-amine 333313 (R)-N-(3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)-3,3-dimethylbutanamide 333315 4-(3-chloro-4-fluorophenylamino)-6-(2-morpholinoethylamino)-1,7-naphthyridine-3-carbonitrile 333316 4-(4-benzylphenylamino)-6-(2-morpholinoethylamino)-1,7-naphthyridine-3-carbonitrile 333324 (S)-N-(1-(4-(trifluoromethoxy)benzyl)pyrrolidin-3-yl)-4-(thiophen-2-yl)benzamide 333325 4-(3,4-dichlorophenylamino)-6-(2-morpholinoethylamino)-1,7-naphthyridine-3-carbonitrile 333330 4-phenoxy-N-(pyridin-2-ylmethyl)benzamide 333331 N-(3-hydroxy-4-(1-hydroxy-2-methylpropan-2-yl)benzyl)-4-phenoxybenzamide 333335 4-(3,5-dichlorophenylamino)-6-(2-morpholinoethylamino)-1,7-naphthyridine-3-carbonitrile 333337 N-(4-methyl-benzyl)-4-phenoxy-benzamide 333353 N-(2-chloro-5-methoxyphenyl)-7-(3-morpholin-4-ylpropoxy)-5-(tetrahydro-2H-pyran-4-yloxy)quinazolin-4-amine 333360 N-(2-chloro-5-methoxyphenyl)-5-isopropoxy-7-(3-morpholinopropoxy)quinazolin-4-amine 333362 N-(3-chloro-6-methoxypyridin-2-yl)-7-(3-morpholinopropoxy)-5-(tetrahydro-2H-pyran-4-yloxy)quinazolin-4-amine 333363 (R)-N-(3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)cyclobutanecarboxamide 333368 N-(2-chloro-5-methoxypyridin-3-yl)-7-(3-morpholinopropoxy)-5-(tetrahydro-2H-pyran-4-yloxy)quinazolin-4-amine 333369 N-(2-chloro-5-methoxypyridin-3-yl)-5-isopropoxy-7-(3-morpholinopropoxy)quinazolin-4-amine 333370 Cocaine 333372 (R)-N-(3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)propionamide 333380 N-(5-chloro-2-methoxypyridin-4-yl)-7-(3-morpholinopropoxy)-5-(tetrahydro-2H-pyran-4-yloxy)quinazolin-4-amine 333381 (3-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-ylamino)-5-chloro-1H-indazol-1-yl)(pyridin-3-yl)methanone 333382 (R)-N-(3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)pentanamide 333385 3-[2-(4-isoquinolin-1-yl-piperazin-1-yl)-ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333386 3-{2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-7-methyl-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333387 (3-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-ylamino)-5-chloro-1H-indazol-1-yl)(thiazol-4-yl)methanone 333388 2-morpholin-4-yl-8-(6,7,8,9-tetrahydro-dibenzothiophen-4-yl)-chromen-4-one 333389 (R)-N-(3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)-3-methylbutanamide 333392 (R)-N-(3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)cyclopentanecarboxamide 333393 (R)-N-(3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)-2-ethylbutanamide 333395 2-{4-[2-(7-methyl-4-oxo-5,6,7,8-tetrahydro-4H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-3-yl)-ethyl]-piperazin-1-yl}-benzonitrile 333396 7-methyl-3-[2-(4-o-tolyl-piperazin-1-yl)-ethyl]-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333410 N-(1-(benzo[c][1,2,5]thiadiazol-5-ylmethyl)piperidin-4-yl)-5-chloro-1H-indazol-3-amine 333413 3-[2-(4-biphenyl-2-yl-piperazin-1-yl)-ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333416 7-methyl-3-{2-[4-(2-phenoxy-phenyl)-piperazin-1-yl]-ethyl}-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333417 3-{2-[4-(2-benzyloxy-phenyl)-piperazin-1-yl]-ethyl}-7-methyl-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333419 4-(3-chloro-4-fluorophenylamino)-6-(3-(pyrrolidin-1-yl)propylamino)-1,7-naphthyridine-3-carbonitrile 333420 3-{2-[4-(2-chloro-phenyl)-piperazin-1-yl]-ethyl}-7-methyl-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333432 (R)-N-(3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)cyclopropanecarboxamide 333435 3-{2-[4-(5-chloro-2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-7-methyl-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333436 7-methyl-3-[2-(4-quinolin-4-yl-piperazin-1-yl)-ethyl]-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333437 N-(3-chloro-6-methoxypyridin-2-yl)-5-isopropoxy-7-(2-(4-methylpiperazin-1-yl)ethoxy)quinazolin-4-amine 333438 1-(4-(3-(4-(3-chloro-6-methoxypyridin-2-ylamino)-5-isopropoxyquinazolin-7-yloxy)propyl)piperazin-1-yl)ethanone 333439 3-{2-[4-(2-isopropoxy-phenyl)-piperazin-1-yl]-ethyl}-7-methyl-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333440 3-(2-{4-[2-(2,2-dimethyl-propoxy)-phenyl]-piperazin-1-yl}-ethyl)-7-methyl-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333451 (R)-N-(3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)butyramide 333475 1-(4-(2-(4-(3-chloro-6-methoxypyridin-2-ylamino)-5-isopropoxyquinazolin-7-yloxy)ethyl)piperazin-1-yl)ethanone 333476 1-(4-(2-(4-(3-chloro-6-methoxypyrazin-2-ylamino)-5-isopropoxyquinazolin-7-yloxy)ethyl)piperazin-1-yl)ethanone 333478 5-chloro-N-(1-(naphthalen-2-ylmethyl)piperidin-4-yl)-1-(pyridin-2-ylmethyl)-1H-indazol-3-amine 333479 N-(1-{4-[(R)-2-acetylamino-3-(4-chloro-phenyl)-propionyl]-piperazin-1-yl}-cyclohexylmethyl)-2-phenyl-acetamide 333485 N-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-yl)-5-chloro-1-(pyridin-3-ylmethyl)-1H-indazol-3-amine 333486 N-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-yl)-5-chloro-1-(pyridin-4-ylmethyl)-1H-indazol-3-amine 333487 (R)-N-(3-(4-chlorophenyl)-1-oxo-1-(4-(1-((2-phenylacetamido)methyl)cyclohexyl)piperazin-1-yl)propan-2-yl)isobutyramide 333499 1-(4-(2-(4-(5-chloro-2-methoxypyrimidin-4-ylamino)-5-isopropoxyquinazolin-7-yloxy)ethyl)piperazin-1-yl)ethanone 333527 (3-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-ylamino)-5-chloro-1H-indazol-1-yl)(cyclopropyl)methanone 333528 1-(3-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-ylamino)-5-chloro-1H-indazol-1-yl)-2-morpholinoethanone 333535 N-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-yl)-5-chloro-1-(pyridin-2-ylmethyl)-1H-indazol-3-amine 333537 7-methyl-3-[2-(4-naphthalen-1-yl-piperazin-1-yl)-ethyl]-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333538 H-Dmt-Tic-NH-(CH2)6-NH-Dmt-H 333539 H-Dmt-Tic-NH-(CH2)6-NH-Tic-H 333547 3-{2-[4-(2,5-dimethoxy-phenyl)-piperazin-1-yl]-ethyl}-7-methyl-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333548 3-{2-[4-(2-methoxy-5-methyl-phenyl)-piperazin-1-yl]-ethyl}-7-methyl-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333551 H-Dmt-Tic-NH-(CH2)6-NH-Phe-H 333565 3-{2-[4-(2-methoxy-5-trifluoromethyl-phenyl)-piperazin-1-yl]-ethyl}-7-methyl-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333566 3-{2-[4-(2,3-dihydro-benzofuran-7-yl)-piperazin-1-yl]-ethyl}-7-methyl-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333573 3-[2-(4-benzo[b]thiophen-7-yl-piperazin-1-yl)-ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333574 3-[2-(4-isoquinolin-4-yl-piperazin-1-yl)-ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333592 3-{2-[4-(4-methoxy-biphenyl-3-yl)-piperazin-1-yl]-ethyl}-7-methyl-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333593 3-{2-[4-(4-chloro-2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-7-methyl-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333609 (1R,2R,4S)-4-[(2R)-2-[(1R,9S,15R,16E,18R,19R,21R,23S,24E,26E,28E,30S,32S,35R)-1,18-dihydroxy-19,30-dimethoxy-15,17,21,23,29,35-hexamethyl-2,3,10,14,20-pentaoxo-11,36-dioxa-4-azatricyclo[30.3.1.0^{4,9}]hexatriaconta-16,24,26,28-tetraen-12-yl]propyl]-2-methoxycyclohexyl N-methoxy-N-methylcarbamate 333630 N-(3-chloro-6-methoxypyridin-2-yl)-5-isopropoxy-7-(2-(pyrrolidin-1-yl)ethoxy)quinazolin-4-amine 333633 7-methyl-3-[2-(4-quinolin-5-yl-piperazin-1-yl)-ethyl]-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333634 3-[2-(4-isoquinolin-5-yl-piperazin-1-yl)-ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333641 N-(3-chloro-6-methoxypyridin-2-yl)-5-isopropoxy-7-(3-(4-methylpiperazin-1-yl)propoxy)quinazolin-4-amine 333667 3-{2-[4-(3-chloro-2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-7-methyl-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333668 3-{2-[4-(4,5-dichloro-2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-7-methyl-5,6,7,8-tetrahydro-3H-pyrido[4',3a':4,5]thieno[2,3-d]pyrimidin-4-one 333669 N-(5-chloro-2-methoxypyridin-4-yl)-5-isopropoxy-7-(3-morpholinopropoxy)quinazolin-4-amine 333675 3-[2-(4-isoquinolin-8-yl-piperazin-1-yl)-ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333676 7-methyl-3-[2-(4-quinolin-8-yl-piperazin-1-yl)-ethyl]-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333682 7-methyl-3-[2-(4-quinazolin-4-yl-piperazin-1-yl)-ethyl]-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333697 3-{2-[4-(3,5-dichloro-2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-7-methyl-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333709 3-{2-[4-(2-methoxy-naphthalen-1-yl)-piperazin-1-yl]-ethyl}-7-methyl-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333710 7-methyl-3-[2-(4-quinolin-2-yl-piperazin-1-yl)-ethyl]-5,6,7,8-tetrahydro-3H-pyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-one 333712 N-(3-chloro-6-methoxypyridin-2-yl)-5-isopropoxy-7-(3-morpholinopropoxy)quinazolin-4-amine 333718 N-(3-chloro-6-methoxypyridin-2-yl)-5-isopropoxy-7-(2-morpholinoethoxy)quinazolin-4-amine 333719 N-(3-chloro-6-methoxypyridin-2-yl)-5-isopropoxy-7-(3-(pyrrolidin-1-yl)propoxy)quinazolin-4-amine 333742 (1R,9S,12S,15R,16E,18R,19R,21R,23S,24E,26E,28E,30S,32S,35R)-1,18-dihydroxy-19,30-dimethoxy-12-[(2R)-1-[(1S,3R,4S)-3-methoxy-4-(2H-1,2,3,4-tetrazol-2-yl)cyclohexyl]propan-2-yl]-15,17,21,23,29,35-hexamethyl-11,36-dioxa-4-azatricyclo[30.3.1.0^{4,9}]hexatriaconta-16,24,26,28-tetraene-2,3,10,14,20-pentone 333796 N-[5-(7-methoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-ylamino)-pyrimidin-2-yl]-benzamide 333801 (1R,9S,12S,15R,16E,18R,19R,21R,23S,24E,26E,28E,30S,32S,35R)-1,18-dihydroxy-19,30-dimethoxy-12-[(2R)-1-[(1S,3R,4S)-3-methoxy-4-(1H-1,2,3,4-tetrazol-1-yl)cyclohexyl]propan-2-yl]-15,17,21,23,29,35-hexamethyl-11,36-dioxa-4-azatricyclo[30.3.1.0^{4,9}]hexatriaconta-16,24,26,28-tetraene-2,3,10,14,20-pentone 333875 N-[5-(8-methoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-ylamino)-pyrimidin-2-yl]-4-methyl-benzamide 333876 3-fluoro-N-[5-(8-methoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-ylamino)-pyrimidin-2-yl]-benzamide 333877 3-fluoro-N-[5-(7-methoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-ylamino)-pyrimidin-2-yl]-benzamide 333913 N-[5-(7,8-dimethoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-ylamino)-pyrimidin-2-yl]-3-fluoro-benzamide 333914 4-fluoro-N-[5-(7-methoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-ylamino)-pyrimidin-2-yl]-benzamide 333919 N-[5-(10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-ylamino)-pyrimidin-2-yl]-benzamide 333924 1-(1-chloro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-8-yl)-3-(4-chloro-3-trifluoromethyl-phenyl)-urea 333927 N-[5-(8-methoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-ylamino)-pyrimidin-2-yl]-benzamide 333941 N-[5-(9-methoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-ylamino)-pyrimidin-2-yl]-benzamide 333977 N-[5-(7,8-dimethoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-ylamino)-pyrimidin-2-yl]-benzamide 333978 N-[5-(7-diethylamino-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-ylamino)-pyrimidin-2-yl]-benzamide 333985 N-[5-(10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-ylamino)-pyrimidin-2-yl]-4-methyl-benzamide 333996 N-[5-(7,8-dimethoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-ylamino)-pyrimidin-2-yl]-4-methyl-benzamide 334019 N-(4-(4-amino-1-(1-(tetrahydro-2H-pyran-4-yl)piperidin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-2-methoxyphenyl)-4-(trifluoromethoxy)benzamide 334020 N-(4-(4-amino-1-(1-benzylpiperidin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-2-methoxyphenyl)-2-fluoro-4-(trifluoromethyl)benzamide 334021 N-(4-(4-amino-1-(1-(tetrahydro-2H-pyran-4-yl)piperidin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-2-methoxyphenyl)-5-cyano-1-methyl-1H-indole-2-carboxamide 334023 4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3-methoxybenzamido)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334024 4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3-cyanobenzamido)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334030 6-(4-methoxyphenyl)-3-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-1H-pyrrolo[2,3-d]pyrimidine-2,4(3H,7H)-dione 334035 7-(1-tert-butylpiperidin-4-yloxy)-5-(2,4-difluorophenyl)-1-(2,6-difluorophenyl)quinolin-2(1H)-one 334036 6-(2-methoxyphenyl)-3-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-1H-pyrrolo[2,3-d]pyrimidine-2,4(3H,7H)-dione 334044 N-butyl-3-methyl-1H-thieno[2,3-c]pyrazole-5-carboxamide 334047 N-benzyl-3-methyl-1H-thieno[2,3-c]pyrazole-5-carboxamide 334055 N-butyl-N-methyl-3-phenyl-1H-thieno[2,3-c]pyrazole-5-carboxamide 334064 1-(5-carbamoyl-3-methyl-1H-thieno[2,3-c]pyrazol-4-yl)-3-phenylurea 334065 2-(4-(5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-2-oxo-1,2-dihydroquinolin-7-yl)piperidin-1-yl)-2-methylpropanoic acid 334072 (5Z,8Z,11Z,14Z)-N-(2,5-dimethoxybenzyl)icosa-5,8,11,14-tetraenamide 334073 (2R)-2-(4-(5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-2-oxo-1,2-dihydroquinolin-7-yl)piperidin-1-yl)propanoic acid 334082 (5Z,8Z,11Z,14Z)-N-(2,4-dimethoxybenzyl)icosa-5,8,11,14-tetraenamide 334083 (5Z,8Z,11Z,14Z)-1-(4-(3,4-dimethylphenyl)piperazin-1-yl)icosa-5,8,11,14-tetraen-1-one 334084 7-(1-tert-butylpiperidin-4-yloxy)-5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)quinolin-2(1H)-one 334085 (5Z,8Z,11Z,14Z)-1-(4-(4-chlorophenyl)piperazin-1-yl)icosa-5,8,11,14-tetraen-1-one 334092 3-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-6-phenyl-1H-pyrrolo[2,3-d]pyrimidine-2,4(3H,7H)-dione 334095 3-(2-(4-(2-chlorophenyl)piperazin-1-yl)ethyl)-6-phenyl-1H-pyrrolo[2,3-d]pyrimidine-2,4(3H,7H)-dione 334100 N-(4-(4-amino-1-(piperidin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-2-methoxyphenyl)-2-fluoro-4-(trifluoromethyl)benzamide 334120 N-(4-(4-amino-1-(1-(tetrahydro-2H-pyran-4-yl)piperidin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-2-methoxyphenyl)-4-methylbenzamide 334128 3-(2-(4-(2-chlorophenyl)piperazin-1-yl)ethyl)-6-(2-methoxyphenyl)-1H-pyrrolo[2,3-d]pyrimidine-2,4(3H,7H)-dione 334129 6-(2-chlorophenyl)-3-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-1H-pyrrolo[2,3-d]pyrimidine-2,4(3H,7H)-dione 334131 methyl 3-methyl-1H-thieno[2,3-c]pyrazole-5-carboxylate 334132 methyl 3-(phenylamino)-1H-thieno[2,3-c]pyrazole-5-carboxylate 334137 6-(2-chlorophenyl)-3-(2-(4-(2-chlorophenyl)piperazin-1-yl)ethyl)-1H-pyrrolo[2,3-d]pyrimidine-2,4(3H,7H)-dione 334140 3-methyl-1H-thieno[2,3-c]pyrazole-5-carboxamide 334145 (5Z,8Z,11Z,14Z)-1-(4-(4-fluorophenyl)piperazin-1-yl)icosa-5,8,11,14-tetraen-1-one 334146 3-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-6-o-tolyl-1H-pyrrolo[2,3-d]pyrimidine-2,4(3H,7H)-dione 334152 3-(2-(4-(2-chlorophenyl)piperazin-1-yl)ethyl)-6-o-tolyl-1H-pyrrolo[2,3-d]pyrimidine-2,4(3H,7H)-dione 334157 4-(2-chlorobenzamido)-3-methyl-1H-thieno[2,3-c]pyrazole-5-carboxamide 334167 (2S)-2-(4-(5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-2-oxo-1,2-dihydroquinolin-7-yl)piperidin-1-yl)propanoic acid 334168 N-(4-(4-amino-1-(1-(tetrahydro-2H-pyran-4-yl)piperidin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-2-methoxyphenyl)-3-hydroxybenzamide 334172 7-(1-tert-butylpiperidin-4-yloxy)-5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)quinolin-2(1H)-one 334173 3-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-6-p-tolyl-1H-pyrrolo[2,3-d]pyrimidine-2,4(3H,7H)-dione 334174 3-[2-[4-(2-chlorophenyl)-1-piperazinyl]ethyl]-6-(4-methylphenyl)-1H-pyrrolo[2,3-d]pyrimidine-2,4(3H,7H)-dione 334192 N-benzyl-3-phenyl-1H-thieno[2,3-c]pyrazole-5-carboxamide 334195 3-(5-(3-amino-3-methylbut-1-ynyl)-2-methoxyphenyl)-N-(2,4-difluorophenyl)-1H-pyrazolo[3,4-b]pyridin-6-amine 334198 6-(4-chlorophenyl)-3-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-1H-pyrrolo[2,3-d]pyrimidine-2,4(3H,7H)-dione 334199 6-(4-chlorophenyl)-3-(2-(4-(2-chlorophenyl)piperazin-1-yl)ethyl)-1H-pyrrolo[2,3-d]pyrimidine-2,4(3H,7H)-dione 334200 N-phenethyl-3-phenyl-1H-thieno[2,3-c]pyrazole-5-carboxamide 334201 N-(4-methoxybenzyl)-3-phenyl-1H-thieno[2,3-c]pyrazole-5-carboxamide 334202 7-(1-tert-butylpiperidin-4-yloxy)-1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)quinolin-2(1H)-one 334210 (4-methylpiperazin-1-yl)(3-phenyl-1H-thieno[2,3-c]pyrazol-5-yl)methanone 334211 4-acetamido-3-methyl-1H-thieno[2,3-c]pyrazole-5-carboxamide 334214 4-azido-N-(1-(2-(2-(4-(4-chloro-2-fluorophenylamino)-6-methoxyquinazolin-7-yloxy)ethoxy)ethylamino)-1-oxo-6-(5-(2-oxo-hexahydro-1H-thieno[3,4-d]imidazol-4-yl)pentanamido)hexan-2-yl)-2,3,5,6-tetrafluorobenzamide 334215 N-(2-(4-(4-chloro-2-fluorophenylamino)-6-methoxyquinazolin-7-yloxy)ethyl)-5-(2-oxo-hexahydro-1H-thieno[3,4-d]imidazol-4-yl)pentanamide 334227 3-(5-(3-amino-3-methylbutyl)-2-methoxyphenyl)-N-(2,4-difluorophenyl)-1H-pyrazolo[3,4-b]pyridin-6-amine 334240 N-(4-(1-(1-(1-acetylpiperidin-4-yl)piperidin-4-yl)-4-amino-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-2-methoxyphenyl)-2-fluoro-4-(trifluoromethyl)benzamide 334249 N-(4-(4-amino-1-(1-(tetrahydro-2H-pyran-4-yl)piperidin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-2-methoxyphenyl)-4-(dimethylamino)benzamide 334266 N-(2-(2-(4-(4-chloro-2-fluorophenylamino)-6-methoxyquinazolin-7-yloxy)ethoxy)ethyl)-5-(2-oxo-hexahydro-1H-thieno[3,4-d]imidazol-4-yl)pentanamide 334267 3-(6-(2,4-difluorophenylamino)-1H-pyrazolo[3,4-b]pyridin-3-yl)-4-methoxybenzoic acid 334268 3-(6-(2,4-difluorophenylamino)-1H-pyrazolo[3,4-b]pyridin-3-yl)-4-methoxy-N-(tetrahydro-2H-pyran-4-yl)benzamide 334275 methyl 2-(5-carbamoyl-3-methyl-1H-thieno[2,3-c]pyrazol-4-ylamino)-2-oxoacetate 334276 3-methyl-4-(2-phenoxyacetamido)-1H-thieno[2,3-c]pyrazole-5-carboxamide 334283 4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3-chlorobenzamido)phenyl)-N-butyl-1,4-diazepane-1-carboxamide 334286 3-methyl-4-(thiophene-2-carboxamido)-1H-thieno[2,3-c]pyrazole-5-carboxamide 334299 N-(4-(4-amino-1-(1-(tetrahydro-2H-pyran-4-yl)piperidin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-2-methoxyphenyl)-4-hydroxyquinoline-2-carboxamide 334300 N-(4-(1-(1-(1-acetylpiperidin-4-yl)piperidin-4-yl)-4-amino-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-2-methoxyphenyl)-1-methyl-1H-indole-2-carboxamide 334310 (E)-N-(3,5-dimethoxyphenethyl)undec-2-enamide 334313 N-(4-(1-(4-(4-acetylpiperazin-1-yl)cyclohexyl)-4-amino-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-2-methoxyphenyl)-1-methyl-1H-indole-2-carboxamide 334322 N-(4-(4-amino-1-(1-methylpiperidin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-2-methoxyphenyl)-2-fluoro-4-(trifluoromethyl)benzamide 334343 N-cyclohexyl-3-phenyl-1H-thieno[2,3-c]pyrazole-5-carboxamide 334349 N-(4-methoxyphenethyl)oleamide 334350 N-(3,5-dimethoxyphenethyl)oleamide 334352 3-(2-(4-(2-chlorophenyl)piperazin-1-yl)ethyl)-6-(4-methoxyphenyl)-1H-pyrrolo[2,3-d]pyrimidine-2,4(3H,7H)-dione 334353 N-(4-(4-amino-1-(1-(tetrahydro-2H-pyran-4-yl)piperidin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-2-methoxyphenyl)-2-fluoro-4-(trifluoromethyl)benzamide 334354 N-(4-(4-amino-1-(1-(1-methylpiperidin-4-yl)piperidin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-2-methoxyphenyl)-2-fluoro-4-(trifluoromethyl)benzamide 334355 N-(4-(4-amino-1-(1-(tetrahydro-2H-pyran-4-yl)piperidin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-2-methoxyphenyl)-1-methyl-1H-benzo[d]imidazole-2-carboxamide 334357 N-(4-(4-amino-1-(1-(tetrahydro-2H-pyran-4-yl)piperidin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-2-methoxyphenyl)-1-methyl-1H-indole-2-carboxamide 334358 N-(4-(4-amino-1-(1-(tetrahydro-2H-pyran-4-yl)piperidin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-2-methoxyphenyl)-5-chloro-1-methyl-1H-indole-2-carboxamide 334363 N-(2,4-dimethoxyphenethyl)oleamide 334373 7-(1-tert-butylpiperidin-4-yl)-5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-1,6-naphthyridin-2(1H)-one 334374 N-cyclopentyl-3-(6-(2,4-difluorophenylamino)-1H-pyrazolo[3,4-b]pyridin-3-yl)-4-methoxybenzamide 334376 N-(3,5-dimethoxyphenethyl)docos-13-enamide 334383 (3-(6-(2,4-difluorophenylamino)-1H-pyrazolo[3,4-b]pyridin-3-yl)-4-methoxyphenyl)(piperazin-1-yl)methanone 334385 N-(2,4-dimethoxyphenethyl)docos-13-enamide 334386 4-Methoxyphenethylarachidonoylamide 334391 (E)-N-(4-methoxyphenethyl)undec-2-enamide 334395 (5Z,8Z,11Z,14Z)-N-(2,4-dimethoxyphenethyl)icosa-5,8,11,14-tetraenamide 334398 N-(4-morpholinophenyl)docos-13-enamide 334399 N-(4-methoxyphenyl)oleamide 334404 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-(8-methyl-8-aza-bicyclo[3.2.1]octan-3-yl)quinolin-2(1H)-one 334405 N-(4-methoxybenzyl)oleamide 334407 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-(2,2,6,6-tetramethyl-1,2,3,6-tetrahydropyridin-4-yl)quinolin-2(1H)-one 334408 7-(8-aza-bicyclo[3.2.1]octan-3-yl)-5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)quinolin-2(1H)-one 334411 (E)-N-(4-methoxyphenyl)undec-2-enamide 334414 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-(8-isopropyl-8-aza-bicyclo[3.2.1]octan-3-yl)quinolin-2(1H)-one 334418 7-(1-tert-butylpiperidin-4-yl)-1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-1,6-naphthyridin-2(1H)-one 334419 7-(1-tert-butylpiperidin-4-yl)-5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)-1,6-naphthyridin-2(1H)-one 334421 (5Z,8Z,11Z,14Z)-N-(4-morpholinophenyl)icosa-5,8,11,14-tetraenamide 334423 7-(1-tert-butyl-1,2,3,6-tetrahydropyridin-4-yl)-5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)quinolin-2(1H)-one 334425 4-(1-benzyl-1H-imidazol-2-yl)-N-ethyl-4-phenylpiperidine-1-carboxamide 334426 (4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidin-1-yl)(4-methylpiperazin-1-yl)methanone 334427 methyl 2-(4-(5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-2-oxo-1,2-dihydroquinolin-7-yl)piperidin-1-yl)propanoate 334434 4-(1-benzyl-1H-imidazol-2-yl)-N-(2-fluorophenyl)-4-phenylpiperidine-1-carboxamide 334473 1-methyl-5-(2-phenylH-pyrazolo[1,5-a]pyridin-3-yl)-1H-pyrazolo[3,4-c]pyridazin-3-amine 334474 1-allyl-5-(2-phenylH-pyrazolo[1,5-a]pyridin-3-yl)-1H-pyrazolo[3,4-c]pyridazin-3-amine 334478 4-(1-(3-fluorobenzyl)-1H-imidazol-2-yl)-N,4-diphenylpiperidine-1-carboxamide 334487 7-(1-tert-butylpiperidin-4-yl)-5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)quinolin-2(1H)-one 334494 methyl 2-(4-(5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-2-oxo-1,2-dihydroquinolin-7-yl)piperidin-1-yl)-2-methylpropanoate 334499 7-(1-tert-butylpiperidin-4-yl)-1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)quinolin-2(1H)-one 334500 7-(1-tert-butylpiperidin-4-yl)-5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)quinolin-2(1H)-one 334503 (5Z,8Z,11Z,14Z)-N-(4-methoxyphenyl)icosa-5,8,11,14-tetraenamide 334504 (5Z,8Z,11Z,14Z)-N-(4-methoxybenzyl)icosa-5,8,11,14-tetraenamide 334516 2-(3-amino-5-(2-phenylH-pyrazolo[1,5-a]pyridin-3-yl)-1H-pyrazolo[3,4-c]pyridazin-1-yl)ethanol 334521 7-(1-tert-butylpiperidin-4-yl)-5-(2-chloro-4-fluorophenyl)-1-(2,6-difluorophenyl)quinolin-2(1H)-one 334530 4-(1-benzoyl-1H-imidazol-2-yl)-N,4-diphenylpiperidine-1-carboxamide 334536 4-(3-(6-(2,4-difluorophenylamino)-1H-pyrazolo[3,4-b]pyrazin-3-yl)-4-methoxyphenyl)-2-methylbut-3-yn-2-ol 334542 4-(1-benzyl-1H-imidazol-2-yl)-N-(3-fluorophenyl)-4-phenylpiperidine-1-carboxamide 334549 4-(1-benzyl-1H-imidazol-2-yl)-N-(4-fluorophenyl)-4-phenylpiperidine-1-carboxamide 334550 3-(5-(3-amino-3-methylbutyl)-2-methoxyphenyl)-N-(2,4-difluorophenyl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine 334557 4-(3-(6-(2,4-difluorophenylamino)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-4-methoxyphenyl)-2-methylbutan-2-ol 334566 4-(1-(4-fluorobenzyl)-1H-imidazol-2-yl)-N,4-diphenylpiperidine-1-carboxamide 334567 4-(1-(3-methoxybenzyl)-1H-imidazol-2-yl)-N,4-diphenylpiperidine-1-carboxamide 334574 4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3-fluorobenzamido)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334581 4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(4-fluorobenzamido)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334606 N-(2,4-difluorophenyl)-3-(5-(3-(dimethylamino)propyl)-2-methoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine 334607 N-(2,4-difluorophenyl)-3-(2-methoxy-5-(3-(4-methylpiperazin-1-yl)propyl)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine 334609 N,4-diphenyl-4-(1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl)piperidine-1-carboxamide 334614 3-(5-(3-amino-3-methylbut-1-ynyl)-2-methoxyphenyl)-N-(2,4-difluorophenyl)-1H-pyrazolo[3,4-b]pyrazin-6-amine 334616 N,4-diphenyl-4-(1-(1-phenylethyl)-1H-imidazol-2-yl)piperidine-1-carboxamide 334619 4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3,4-difluorobenzamido)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334620 4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3,5-difluorobenzamido)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334625 4-(1-benzyl-1H-imidazol-2-yl)-N-(2-methoxyphenyl)-4-phenylpiperidine-1-carboxamide 334626 4-(1-benzyl-1H-imidazol-2-yl)-N-(3-methoxyphenyl)-4-phenylpiperidine-1-carboxamide 334635 4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-benzamidophenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334642 4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(2-chlorobenzamido)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334649 4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3-chlorobenzamido)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334651 4-(2-(3-chlorobenzamido)-4-(phenethylcarbamoyl)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334658 4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3-chlorobenzamido)phenyl)-N,N-dimethyl-1,4-diazepane-1-carboxamide 334660 N-((S)-1-(4-(2,4-dichlorobenzyloxy)pyrimidin-2-ylamino)-3-methylbutan-2-yl)-1-methylpiperidine-3-carboxamide 334661 (4-(4-(2,4-dichlorobenzyloxy)pyrimidin-2-yl)piperazin-1-yl)(1-methylpiperidin-3-yl)methanone 334672 N-(2,4-difluorophenyl)-3-(2-methoxy-5-((tetrahydro-2H-pyran-4-ylamino)methyl)phenyl)-1H-pyrazolo[3,4-b]pyridin-6-amine 334675 4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(thiophene-2-carboxamido)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334682 4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(nicotinamido)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334685 3-(5-((cyclopentylamino)methyl)-2-methoxyphenyl)-N-(2,4-difluorophenyl)-1H-pyrazolo[3,4-b]pyridin-6-amine 334686 3-(5-(3-amino-3-methylbut-1-ynyl)-2-methoxyphenyl)-N-(2,4-difluorophenyl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine 334689 4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(isonicotinamido)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334691 (R)-1,1-bis(4-fluorophenyl)-3-(3-methoxyquinuclidin-3-yl)prop-2-yn-1-ol 334695 4-(4-(benzylcarbamoyl)-2-(3-chlorobenzamido)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334698 3-(5-(3-amino-3-methylbutyl)-2-methoxyphenyl)-N-(2,4-difluorophenyl)-1H-pyrazolo[3,4-b]pyrazin-6-amine 334699 4-(3-(6-(2,4-difluorophenylamino)-1H-pyrazolo[3,4-b]pyrazin-3-yl)-4-methoxyphenyl)-2-methylbutan-2-ol 334700 4-phenyl-4-[1H-imidazol-2-yl]-piperidine 334701 4-(1-(2-fluorobenzyl)-1H-imidazol-2-yl)-N,4-diphenylpiperidine-1-carboxamide 334702 4-(4-((4-chlorobenzyl)carbamoyl)-2-(3-chlorobenzamido)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334711 (4-(4-(2,4-dichlorobenzylamino)pyrimidin-2-yl)piperazin-1-yl)(1-methylpiperidin-3-yl)methanone 334715 4-(1-benzyl-1H-imidazol-2-yl)-N-methyl-N,4-diphenylpiperidine-1-carboxamide 334716 4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidine-1-carboxamide 334725 4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(thiophene-3-carboxamido)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334732 4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(furan-2-carboxamido)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334736 4-(3-(6-(2,4-difluorophenylamino)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-4-methoxyphenyl)-2-methylbut-3-yn-2-ol 334737 N-(2,4-difluorophenyl)-3-(5-(3-(dimethylamino)prop-1-ynyl)-2-methoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine 334742 4-(2-(3-chlorobenzamido)-4-(isopropylcarbamoyl)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334746 N-(2,4-difluorophenyl)-3-(2-methoxy-5-(3-(4-methylpiperazin-1-yl)prop-1-ynyl)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine 334748 4-(4-((3,4-dimethoxyphenethyl)carbamoyl)-2-(3-chlorobenzamido)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334764 4-(1-benzyl-1H-imidazol-2-yl)-N-(4-methoxyphenyl)-4-phenylpiperidine-1-carboxamide 334769 2-(4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidin-1-yl)pyrimidine 334770 4-(1-benzyl-1H-imidazol-2-yl)-4-phenyl-1-(thiazol-2-yl)piperidine 334773 4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(2-fluorobenzamido)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334778 4-(4-((4-fluorophenethyl)carbamoyl)-2-(3-chlorobenzamido)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334779 (4-(2-(2,4-dichlorobenzylamino)pyrimidin-4-yl)piperazin-1-yl)(1-methylpiperidin-3-yl)methanone 334791 1-(3-methoxyquinuclidin-3-yl)-3-phenyloct-1-yn-3-ol 334798 4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3-chlorobenzamido)phenyl)-N-propyl-1,4-diazepane-1-carboxamide 334799 4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3-chlorobenzamido)phenyl)-N-isopropyl-1,4-diazepane-1-carboxamide 334803 1-(3-methoxyquinuclidin-3-yl)-3-phenylhept-1-yn-3-ol 334808 4-(4-((2-chlorophenethyl)carbamoyl)-2-(3-chlorobenzamido)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334813 (R)-1,1-bis(4-chlorophenyl)-3-(3-methoxyquinuclidin-3-yl)prop-2-yn-1-ol 334824 8-(1-((5-(4-methoxyphenyl)isoxazol-3-yl)methyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 334831 8-(1-((5-(2-methoxyphenyl)isoxazol-3-yl)methyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 334832 (S)-(4-(4-(2,4-dichlorobenzylamino)pyrimidin-2-yl)piperazin-1-yl)(piperidin-2-yl)methanone 334833 (R)-(4-(4-(2,4-dichlorobenzylamino)pyrimidin-2-yl)piperazin-1-yl)(piperidin-2-yl)methanone 334838 (R)-(4-(4-(2,4-dichlorobenzylamino)pyrimidin-2-yl)piperazin-1-yl)(pyrrolidin-2-yl)methanone 334844 4-(4-((3-chlorophenethyl)carbamoyl)-2-(3-chlorobenzamido)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334847 2-benzyl-4-(3-methoxyquinuclidin-3-yl)-1-phenylbut-3-yn-2-ol 334850 methyl 4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3-chlorobenzamido)phenyl)-1,4-diazepane-1-carboxylate 334851 4-(4-((4-chlorophenethyl)carbamoyl)-2-(3-chlorobenzamido)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334858 4-(4-((2-fluorophenethyl)carbamoyl)-2-(3-chlorobenzamido)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334861 4-(3-methoxyquinuclidin-3-yl)-1,2-diphenylbut-3-yn-2-ol 334863 ethyl 4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3-chlorobenzamido)phenyl)-1,4-diazepane-1-carboxylate 334870 2-(4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidin-1-yl)benzo[d]thiazole 334876 2-(4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidin-1-yl)-1-methyl-1H-benzo[d]imidazole 334879 (4-(4-(2,4-dichlorobenzylamino)pyrimidin-2-yl)piperazin-1-yl)(piperidin-3-yl)methanone 334890 4-(2-(3-chlorobenzamido)-4-((cyclopropylmethyl)carbamoyl)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334893 4-(4-((3-fluorophenethyl)carbamoyl)-2-(3-chlorobenzamido)phenyl)-N-ethyl-1,4-diazepane-1-carboxamide 334900 1-(2-(4-(4-chloro-3-hydroxyphenyl)-5-(pyridin-4-yl)-1H-imidazol-2-yl)-2-methylpropyl)-3-(4-chlorophenyl)urea 334902 1,3-dipropyl-8-(1-((5-(4-(trifluoromethyl)phenyl)isoxazol-3-yl)methyl)-1H-pyrazol-4-yl)-1H-purine-2,6(3H,7H)-dione 334903 4-(1-benzyl-1H-imidazol-2-yl)-1-(methylsulfonyl)-4-phenylpiperidine 334910 4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidine-1-sulfonamide 334914 4-(4-(benzo[b]thiophen-2-yl)pyrimidin-2-ylamino)-N-(2-(dimethylamino)ethyl)benzamide 334918 4-(1-benzyl-1H-imidazol-2-yl)-N,4-diphenylpiperidine-1-sulfonamide 334923 4-(4-(benzo[b]thiophen-2-yl)pyrimidin-2-ylamino)-N-(2-(pyrrolidin-1-yl)ethyl)benzamide 334924 (R)-3-(3-methoxyquinuclidin-3-yl)-1,1-dip-tolylprop-2-yn-1-ol 334926 4-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(4-chlorophenyl)-4-oxobutanamide 334931 N-(2-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)ethyl)-4-chlorobenzamide 334933 (R)-1,1-bis(3-fluorophenyl)-3-(3-methoxyquinuclidin-3-yl)prop-2-yn-1-ol 334934 4-((1H-imidazol-4-yl)methyl)-1-(3-phenoxypropyl)piperidine 334935 4-((1H-imidazol-4-yl)methyl)-1-(3-(3-chlorophenoxy)propyl)piperidine 334936 4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3-chlorobenzamido)phenyl)-N-methyl-1,4-diazepane-1-carboxamide 334937 N-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propyl)-4-chlorobenzamide 334938 N-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propyl)-3-chlorobenzenamine 334939 (R)-3-(3-methoxyquinuclidin-3-yl)-1,1-dim-tolylprop-2-yn-1-ol 334940 (R)-3-(3-methoxyquinuclidin-3-yl)-1,1-di(thiophen-2-yl)prop-2-yn-1-ol 334943 8-(1-((5-(3-chlorophenyl)isoxazol-3-yl)methyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 334944 1,3-dipropyl-8-(1-((5-(2-(trifluoromethyl)phenyl)isoxazol-3-yl)methyl)-1H-pyrazol-4-yl)-1H-purine-2,6(3H,7H)-dione 334945 2-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(4-chlorophenyl)ethanesulfonamide 334947 (R)-3-(3-methoxyquinuclidin-3-yl)-1,1-di(thiophen-3-yl)prop-2-yn-1-ol 334950 8-(1-((5-(3-methoxyphenyl)isoxazol-3-yl)methyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 334954 1-cyclopentyl-3-(3-methoxyquinuclidin-3-yl)-1-(pyridin-2-yl)prop-2-yn-1-ol 334969 4-((1H-imidazol-4-yl)methyl)-1-(3-(phenylsulfonyl)propyl)piperidine 334975 4-((1H-imidazol-4-yl)methyl)-N-(4-chlorophenyl)piperidine-1-carboxamide 334976 2-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(4-chlorophenyl)acetamide 334979 (4-(4-(benzo[b]thiophen-2-yl)pyrimidin-2-ylamino)phenyl)(4-(dimethylamino)piperidin-1-yl)methanone 334985 (R)-3-(3-methoxyquinuclidin-3-yl)-1,1-bis(3-(trifluoromethyl)phenyl)prop-2-yn-1-ol 334990 3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(3-chlorophenyl)-3-oxopropanamide 334991 2-chloro-5-(2-(furan-2-yl)-5-(pyridin-4-yl)-1H-imidazol-4-yl)phenol 334992 2-chloro-5-(5-(pyridin-4-yl)-1H-imidazol-4-yl)phenol 335003 5-(2-(4-(aminomethyl)phenyl)-5-(pyridin-4-yl)-1H-imidazol-4-yl)-2-chlorophenol 335011 methyl 4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propanamido)benzoate 335014 5-(2-(1-amino-2-methylpropan-2-yl)-5-(pyridin-4-yl)-1H-imidazol-4-yl)-2-chlorophenol 335017 3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-cyclohexylpropanamide 335018 3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(4-chlorobenzyl)propanamide 335020 1-(5H-dibenzo[a,d]cyclohepten-5-yl)-3-((R)-3-methoxy-1-aza-bicyclo[2.2.2]oct-3-yl)-prop-2-yn-1-ol 335021 4-(4-chloro-3-hydroxyphenyl)-N-(3-(dimethylamino)propyl)-5-(pyridin-4-yl)-1H-imidazole-2-carboxamide 335022 N-(2-(4-(4-chloro-3-hydroxyphenyl)-5-(pyridin-4-yl)-1H-imidazol-2-yl)-2-methylpropyl)methanesulfonamide 335023 8-(1-((5-(2-chlorophenyl)isoxazol-3-yl)methyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 335024 8-(1-((5-(4-chlorophenyl)isoxazol-3-yl)methyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 335031 8-((cis, rac)-2-hydroxy-2-p-tolyl-cyclohexyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 335032 8-((cis, rac)-2-hydroxy-2-pyridin-4-yl-cyclohexyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 335033 4-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(4-chlorophenyl)butanamide 335034 2-chloro-5-(2-(pyridin-3-yl)-5-(pyridin-4-yl)-1H-imidazol-4-yl)phenol 335041 2-(4-(4-(benzo[b]thiophen-2-yl)pyrimidin-2-ylamino)phenyl)acetic acid 335042 (4-(4-(benzo[b]thiophen-2-yl)pyrimidin-2-ylamino)phenyl)(pyrrolidin-1-yl)methanone 335049 N-(2-aminoethyl)-4-(4-(benzo[b]thiophen-2-yl)pyrimidin-2-ylamino)benzamide 335055 ((2S,3S,4R,5R)-5-(2-chloro-6-(cyclopropylamino)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrothiophen-2-yl)(morpholino)methanone 335056 (2S,3S,4R,5R)-5-(2-chloro-6-(cyclopentylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyl-tetrahydrothiophene-2-carboxamide 335060 1-cyclobutyl-3-(3-methoxyquinuclidin-3-yl)-1-(pyridin-2-yl)prop-2-yn-1-ol 335063 (2S,3S,4R,5R)-5-(2-chloro-6-(cyclopentylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrothiophene-2-carboxamide 335067 3-(3-methoxyquinuclidin-3-yl)-1-phenyl-1-(pyridin-2-yl)prop-2-yn-1-ol 335068 3-(3-methoxyquinuclidin-3-yl)-1-phenyl-1-(pyridin-3-yl)prop-2-yn-1-ol 335070 1-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-4-phenylbutan-1-one 335071 4-((1H-imidazol-4-yl)methyl)-1-(4-(4-chlorophenyl)butyl)piperidine 335072 4-((1H-imidazol-4-yl)methyl)-1-heptylpiperidine 335076 4-(4-(benzo[b]thiophen-2-yl)pyrimidin-2-ylamino)benzoic acid 335077 3-(4-(benzo[b]thiophen-2-yl)pyrimidin-2-ylamino)benzoic acid 335078 1-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)heptan-1-one 335079 cis-1-phenyl-8-(2-phenyl-cyclohexyl)-1,3,8-triaza-spiro[4.5]decan-4-one 335081 5-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(4-chlorophenyl)pentanamide 335090 8-[(cis, rac)-2-(4-chloro-phenyl)-2-hydroxy-cyclohexyl]-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 335093 3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(4-chlorophenyl)-N-methylpropanamide 335094 3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(3-chlorophenyl)propanamide 335096 4-(2-tert-butyl-4-(4-fluorophenyl)-1H-imidazol-5-yl)pyridine 335098 1-(4-fluoro-phenyl)-8-[(cis, rac)-2-(4-fluoro-phenyl)-2-hydroxy-cyclohexyl]-1,3,8-triaza-spiro[4.5]decan-4-one 335099 3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(3-fluorophenyl)propanamide 335100 4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propoxy)benzonitrile 335101 2-chloro-5-(2-phenyl-5-(pyridin-4-yl)-1H-imidazol-4-yl)phenol 335105 (2S,3S,4R,5R)-5-(2-chloro-6-(3-iodobenzylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrothiophene-2-carboxamide 335106 (2S,3S,4R,5R)-5-(6-(3-iodobenzylamino)-2-chloro-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrothiophene-2-carboxamide 335107 Biphalin 335111 4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propoxy)benzaldehyde oxime 335112 1-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-3-phenoxypropan-1-one 335117 (2S,3S,4R,5R)-5-(6-(3-iodobenzylamino)-2-chloro-9H-purin-9-yl)-3,4-dihydroxy-N-isopentyl-tetrahydrothiophene-2-carboxamide 335118 4-((1H-imidazol-4-yl)methyl)-1-(4-phenylbutyl)piperidine 335119 methyl 4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-3-oxopropoxy)benzoate 335122 (R)-3-((R)-3-methoxyquinuclidin-3-yl)-1-phenyl-1-(pyridin-3-yl)prop-2-yn-1-ol 335128 (S)-3-((R)-3-methoxyquinuclidin-3-yl)-1-phenyl-1-(pyridin-3-yl)prop-2-yn-1-ol 335129 3-(3-methoxyquinuclidin-3-yl)-1-phenyl-1-(pyridin-4-yl)prop-2-yn-1-ol 335135 (R)-3-(8-methoxyquinuclidin-8-yl)-1,1-di(pyridin-3-yl)prop-2-yn-1-ol 335148 3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-phenylpropanamide 335149 3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(4-methoxyphenyl)propanamide 335150 5-(2-tert-butyl-5-(pyridin-4-yl)-1H-imidazol-4-yl)-2-chlorophenol 335151 8-((cis, rac)-2-hydroxy-2-phenyl-cyclohexyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 335152 8-[(cis, rac)-2-hydroxy-2-(4-methoxy-phenyl)-cyclohexyl]-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 335154 3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(4-chlorophenyl)propanamide 335155 8-[(cis, rac)-2-(3-chloro-phenyl)-2-hydroxy-cyclohexyl]-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 335156 1-(4-chloro-phenyl)-8-[(cis, rac)-2-(4-fluoro-phenyl)-2-hydroxy-cyclohexyl]-1,3,8-triaza-spiro[4.5]decan-4-one 335164 8-[(cis, rac)-2-(4-chloro-phenyl)-2-hydroxy-cyclohexyl]-1-(4-fluoro-phenyl)-1,3,8-triaza-spiro[4.5]decan-4-one 335165 8-[(cis, rac)-2-(4-chloro-phenyl)-2-hydroxy-cyclohexyl]-1-(4-methoxy-phenyl)-1,3,8-triaza-spiro[4.5]decan-4-one 335170 8-(1-((3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl)methyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 335178 (4-(4-(5-(3-amino-3-methylbut-1-ynyl)thiophen-2-yl)pyrimidin-2-ylamino)phenyl)(4-(pyrrolidin-1-yl)piperidin-1-yl)methanone 335180 8-[(cis, rac)-2-hydroxy-2-(3-methoxy-phenyl)-cyclohexyl]-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 335181 8-((cis, rac)-2-hydroxy-2-pyridin-2-yl-cyclohexyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 335186 8-(1-((3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl)methyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 335187 8-(1-((3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl)methyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 335188 8-((cis, rac)-2-hydroxy-2-pyridin-3-yl-cyclohexyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 335193 8-(1-((3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl)methyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 335196 (4-(4-(benzo[b]thiophen-2-yl)pyrimidin-2-ylamino)phenyl)(4-(pyrrolidin-1-yl)piperidin-1-yl)methanone 335197 (4-(4-(benzo[b]thiophen-2-yl)pyrimidin-2-ylamino)-2-chlorophenyl)(4-(pyrrolidin-1-yl)piperidin-1-yl)methanone 335198 (4-(4-(5-(3-amino-3-methylbutyl)thiophen-2-yl)pyrimidin-2-ylamino)phenyl)(4-(pyrrolidin-1-yl)piperidin-1-yl)methanone 335200 1,3-dipropyl-8-(1-((5-(3-(trifluoromethyl)phenyl)-1,2,4-oxadiazol-3-yl)methyl)-1H-pyrazol-4-yl)-1H-purine-2,6(3H,7H)-dione 335202 [O-methyl-11C]2-{4-[4-(7-methoxynaphthalen-1-yl)piperazin-1-yl]butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione 335208 1,3-dipropyl-8-(1-((5-(2-(trifluoromethyl)phenyl)-1,2,4-oxadiazol-3-yl)methyl)-1H-pyrazol-4-yl)-1H-purine-2,6(3H,7H)-dione 335209 (S)-2-amino-N-{(4S,10S,15S,21S)-21-[(S)-2-amino-3-(4-hydroxy-phenyl)-propionylamino]-10,15-dibenzyl-5,8,11,14,17,20-hexaoxo-1,2-dithia-6,9,12,13,16,19-hexaaza-cyclodocos-4-yl}-3-(4-hydroxy-phenyl)-propionamide 335212 (2S,3S,4R,5R)-N-(3-fluorobenzyl)-5-(2-chloro-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrothiophene-2-carboxamide 335213 8-(1-((3-phenyl-1,2,4-oxadiazol-5-yl)methyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 335214 8-(1-((3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl)methyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 335217 (R)-3-(3-methoxyquinuclidin-3-yl)-1,1-diphenylprop-2-yn-1-ol 335219 8-(1-((5-(4-methoxyphenyl)-1,2,4-oxadiazol-3-yl)methyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 335221 (2S,3S,4R,5R)-N-(3-fluorophenethyl)-5-(2-chloro-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrothiophene-2-carboxamide 335222 (2S,3S,4R,5R)-5-(2-chloro-6-(methylamino)-9H-purin-9-yl)-N-(3,3-diphenylpropyl)-3,4-dihydroxy-tetrahydrothiophene-2-carboxamide 335228 (S)-3-(3-methoxyquinuclidin-3-yl)-1,1-diphenylprop-2-yn-1-ol 335229 1-cyclohexyl-3-((R)-3-methoxyquinuclidin-3-yl)-1-phenylprop-2-yn-1-ol 335232 (2S,3S,4R,5R)-N-(3-chlorobenzyl)-5-(6-(3-iodobenzylamino)-2-chloro-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrothiophene-2-carboxamide 335237 (2S,3S,4R,5R)-5-(6-(3-iodobenzylamino)-2-chloro-9H-purin-9-yl)-N-(cyclopropylmethyl)-3,4-dihydroxy-tetrahydrothiophene-2-carboxamide 335244 (2S,3S,4R,5R)-5-(6-(3-iodobenzylamino)-2-chloro-9H-purin-9-yl)-N-cyclobutyl-3,4-dihydroxy-tetrahydrothiophene-2-carboxamide 335245 N-(2-methyl-4-(5-(2-(4-(4-(pyrrolidin-1-yl)piperidine-1-carbonyl)phenylamino)pyrimidin-4-yl)thiophen-2-yl)butan-2-yl)acetamide 335246 1,3-dipropyl-8-(1-((3-p-tolyl-1,2,4-oxadiazol-5-yl)methyl)-1H-pyrazol-4-yl)-1H-purine-2,6(3H,7H)-dione 335247 1,3-dipropyl-8-(1-((3-m-tolyl-1,2,4-oxadiazol-5-yl)methyl)-1H-pyrazol-4-yl)-1H-purine-2,6(3H,7H)-dione 335250 1-pentyl-8-((1S,2S)-2-phenyl-cyclohexyl)-1,3,8-triaza-spiro[4.5]decan-4-one 335251 (4-(4-(5-(3-amino-3-ethylpentyl)thiophen-2-yl)pyrimidin-2-ylamino)phenyl)(4-(pyrrolidin-1-yl)piperidin-1-yl)methanone 335252 N-(2-chlorophenyl)-2-(4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-1H-pyrazol-1-yl)acetamide 335253 ((2S,3S,4R,5R)-5-(6-(3-iodobenzylamino)-2-chloro-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrothiophen-2-yl)(4-benzylpiperidin-1-yl)methanone 335254 ((2S,3S,4R,5R)-5-(6-(3-iodobenzylamino)-2-chloro-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrothiophen-2-yl)(4-(4-fluorophenyl)piperazin-1-yl)methanone 335255 8-[(cis, rac)-2-(3,4-dichloro-phenyl)-2-hydroxy-cyclohexyl]-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 335256 8-(1-((5-(3-methoxyphenyl)-1,2,4-oxadiazol-3-yl)methyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 335257 (2S,3S,4R,5R)-5-(2-chloro-6-(cyclopropylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyl-tetrahydrothiophene-2-carboxamide 335258 (2S,3S,4R,5R)-5-(2-chloro-6-(cyclopropylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrothiophene-2-carboxamide 335259 (2S,3S,4R,5R)-5-(6-(3-iodobenzylamino)-2-chloro-9H-purin-9-yl)-N-cyclopropyl-3,4-dihydroxy-tetrahydrothiophene-2-carboxamide 335264 8-(1-((5-(2-methoxyphenyl)-1,2,4-oxadiazol-3-yl)methyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 335266 (2S,3S,4R,5R)-5-(2-chloro-6-(cyclopropylamino)-9H-purin-9-yl)-N-cyclopropyl-3,4-dihydroxy-tetrahydrothiophene-2-carboxamide 335267 (4-benzylpiperidin-1-yl)((2S,3S,4R,5R)-5-(2-chloro-6-(cyclopropylamino)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrothiophen-2-yl)methanone 335270 1,3-dipropyl-8-(1-((3-(2-(trifluoromethyl)phenyl)-1,2,4-oxadiazol-5-yl)methyl)-1H-pyrazol-4-yl)-1H-purine-2,6(3H,7H)-dione 335271 (S)-1-cyclohexyl-3-((R)-3-methoxyquinuclidin-3-yl)-1-phenylprop-2-yn-1-ol 335272 ((2S,3S,4R,5R)-5-(6-(3-iodobenzylamino)-2-chloro-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrothiophen-2-yl)(morpholino)methanone 335276 (3-(2-phenyl-5-(pyridin-4-yl)-1H-imidazol-4-yl)phenyl)methanol 335278 1-cyclopentyl-3-(3-methoxyquinuclidin-3-yl)-1-phenylprop-2-yn-1-ol 335279 1-cyclobutyl-3-(3-methoxyquinuclidin-3-yl)-1-phenylprop-2-yn-1-ol 335285 8-[(cis, rac)-2-(4-fluoro-phenyl)-2-hydroxy-cyclohexyl]-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 335286 8-((cis, rac)-2-hydroxy-2-o-tolyl-cyclohexyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 335287 (S)-2-Amino-N-{(4R,10S,15S,21R)-21-[(S)-2-amino-3-(4-hydroxy-phenyl)-propionylamino]-10,15-dibenzyl-5,8,11,14,17,20-hexaoxo-1,2-dithia-6,9,12,13,16,19-hexaaza-cyclodocos-4-yl}-3-(4-hydroxy-phenyl)-propionamide 335289 (2S,3S,4R,5R)-5-[2-chloro-6-(2-methyl-benzylamino)-purin-9-yl]-3,4-dihydroxy-tetrahydro-thiophene-2-carboxylic acid ethylamide 335290 N3-(1-naphthyl)-1-hexyl-4-oxo-1,4-dihydroquinoline-3-carboxamide 335292 8-(1-((5-(2-chlorophenyl)-1,2,4-oxadiazol-3-yl)methyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 335293 8-(1-((5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl)methyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 335295 (2S,3S,4R,5R)-5-[2-chloro-6-(2-methyl-benzylamino)-purin-9-yl]-3,4-dihydroxy-tetrahydro-thiophene-2-carboxylic acid dimethylamide 335297 4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid (3,5-dimethyl-adamantan-1-yl)-amide 335298 N3-(1-(3,5-dimethyl)adamantyl)-4-oxo-1-benzyl-1,4-dihydroquinoline-3-carboxamide 335299 4-(3-((4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-1H-pyrazol-1-yl)methyl)-1,2,4-oxadiazol-5-yl)benzonitrile 335302 3-((1H-pyrrol-3-yl)methylene)-6-(4-hydroxyphenyl)indolin-2-one 335305 (RS)-N3-(1-phenylethyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide 335309 3-((1H-pyrrol-3-yl)methylene)-6-(4-aminophenyl)indolin-2-one 335310 3-((1H-pyrrol-2-yl)methylene)-6-(4-hydroxy-2-methoxyphenyl)indolin-2-one 335312 (6aR,10aR)-6,6,9-trimethyl-3-(2-methylpentan-2-yl)-6a,7,10,10a-tetrahydro-6H-benzo[c]chromene 335314 (4-(4-(5-(3-hydroxy-3-methylbutyl)thiophen-2-yl)pyrimidin-2-ylamino)phenyl)(4-(pyrrolidin-1-yl)piperidin-1-yl)methanone 335315 (2S,3S,4R,5R)-N-(3-(trifluoromethyl)benzyl)-5-(6-(3-iodobenzylamino)-2-chloro-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrothiophene-2-carboxamide 335321 (2S,3S,4R,5R)-5-[2-chloro-6-(2-methyl-benzylamino)-purin-9-yl]-3,4-dihydroxy-tetrahydro-thiophene-2-carboxylic acid cyclopropylamide 335325 N-(trans-4-(2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl)cyclohexyl)quinoline-4-carboxamide 335326 1,3-dipropyl-8-(1-((3-(3-(trifluoromethyl)phenyl)-1,2,4-oxadiazol-5-yl)methyl)-1H-pyrazol-4-yl)-1H-purine-2,6(3H,7H)-dione 335327 1-phenyl-8-((trans,rac)-2-phenyl-cyclohexyl)-1,3,8-triaza-spiro[4.5]decan-4-one 335328 (2S,3S,4R,5R)-5-[2-chloro-6-(2-methyl-benzylamino)-purin-9-yl]-3,4-dihydroxy-tetrahydro-thiophene-2-carboxylic acid cyclopropylmethyl-amide 335330 N-(trans-4-(2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl)cyclohexyl)quinoline-2-carboxamide 335334 8-((trans, rac)-2-hydroxy-2-phenyl-cyclohexyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 335335 1,3-dipropyl-8-(1-((5-(4-(trifluoromethyl)phenyl)-1,2,4-oxadiazol-3-yl)methyl)-1H-pyrazol-4-yl)-1H-purine-2,6(3H,7H)-dione 335340 (2S,3S,4R,5R)-5-(6-(3-iodobenzylamino)-2-chloro-9H-purin-9-yl)-N-(3,3-diphenylpropyl)-3,4-dihydroxy-tetrahydrothiophene-2-carboxamide 335341 (4-benzyl-piperidin-1-yl)-{(2S,3S,4R,5R)-5-[2-chloro-6-(2-methyl-benzylamino)-purin-9-yl]-3,4-dihydroxy-tetrahydro-thiophen-2-yl}-methanone 335346 8-(1-((5-(3-chlorophenyl)-1,2,4-oxadiazol-3-yl)methyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 335351 (R)-N3-(1-phenylethyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide 335352 (S)-N3-(1-phenylethyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide 335361 (R)-N3-(1-(2-naphthyl)ethyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide 335364 3-((3,5-dimethyl-1H-pyrrol-2-yl)methylene)-6-(4-hydroxy-3-methoxyphenyl)indolin-2-one 335365 (2S,3S,4R,5R)-5-(6-(3-iodobenzylamino)-2-chloro-9H-purin-9-yl)-3,4-dihydroxy-N-phenethyl-tetrahydrothiophene-2-carboxamide 335367 potassium (2-dodecyl-1,3-dioxolan-4-yl)methyl hydrogenphosphate 335371 (2S,3S,4R,5R)-5-[2-chloro-6-(2-methyl-benzylamino)-purin-9-yl]-3,4-dihydroxy-tetrahydro-thiophene-2-carboxylic acid methylamide 335372 {(2S,3S,4R,5R)-5-[2-chloro-6-(2-methyl-benzylamino)-purin-9-yl]-3,4-dihydroxy-tetrahydro-thiophen-2-yl}-morpholin-4-yl-methanone 335376 potassium (2-(heptadec-9-enyl)-1,3-dioxolan-4-yl)methyl hydrogenphosphate 335385 (4-(4-(benzo[b]thiophen-2-yl)pyrimidin-2-ylamino)-2-methoxyphenyl)(4-(pyrrolidin-1-yl)piperidin-1-yl)methanone 335386 (4-(4-(5-(4-hydroxybutyl)thiophen-2-yl)pyrimidin-2-ylamino)phenyl)(4-(pyrrolidin-1-yl)piperidin-1-yl)methanone 335390 (4-(4-(5-(3-methoxypropyl)thiophen-2-yl)pyrimidin-2-ylamino)phenyl)(4-(pyrrolidin-1-yl)piperidin-1-yl)methanone 335392 3-((1H-pyrrol-2-yl)methylene)-5-(4-hydroxy-3-methoxyphenyl)indolin-2-one 335393 6-(4-hydroxy-3-methoxyphenyl)-3-((3-isopropyl-5-methyl-1H-pyrrol-2-yl)methylene)indolin-2-one 335394 N-(trans-4-(2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl)cyclohexyl)quinoxaline-2-carboxamide 335396 1,3-dipropyl-8-(1-((3-(4-(trifluoromethyl)phenyl)-1,2,4-oxadiazol-5-yl)methyl)-1H-pyrazol-4-yl)-1H-purine-2,6(3H,7H)-dione 335399 N-(trans-4-(2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl)cyclohexyl)quinoline-3-carboxamide 335400 1-phenethyl-8-((1S,2S)-2-phenyl-cyclohexyl)-1,3,8-triaza-spiro[4.5]decan-4-one 335401 N3-(1-naphthyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide 335402 4-(5-((4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-1H-pyrazol-1-yl)methyl)-1,2,4-oxadiazol-3-yl)benzonitrile 335403 8-(1-((3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl)methyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 335407 potassium ((2R,4R)-2-(heptadec-9-enyl)-1,3-dioxolan-4-yl)methyl hydrogenphosphate 335409 3-((1H-indol-3-yl)methylene)-6-(4-hydroxy-3-methoxyphenyl)indolin-2-one 335410 6-(4-hydroxy-3-methoxyphenyl)-3-((7-methyl-1H-indol-3-yl)methylene)indolin-2-one 335418 methyl 3-(5-((6-(4-hydroxy-3-methoxyphenyl)-2-oxoindolin-3-ylidene)methyl)-2,4-dimethyl-1H-pyrrol-3-yl)propanoate 335422 N3-(1-naphthyl)-1-butyl-4-oxo-1,4-dihydroquinoline-3-carboxamide 335428 3-((4-((dimethylamino)methyl)-3-isopropyl-5-methyl-1H-pyrrol-2-yl)methylene)-6-(4-hydroxy-3-methoxyphenyl)indolin-2-one 335429 6-(4-hydroxy-3-methoxyphenyl)-3-((4-(2-hydroxyethyl)-3,5-dimethyl-1H-pyrrol-2-yl)methylene)indolin-2-one 335431 N-(trans-4-(2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl)cyclohexyl)isoquinoline-3-carboxamide 335433 N3-(2-adamantyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide 335457 bis-((+)-N-cyclobutylmethylmorphinan-3-yl) sebacoylate 335458 bis-((-)-N-[(S)-tetrahydrofurfuryl]morphinan-3-yl) sebacoylate 335459 1-((-)-N-cyclobutylmethylmorphinan-3-yl) 10-((-)-N-cyclobutylmethylmorphinan-3-yl) sebacoylate 335471 N3-(4-cyanophenyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide 335472 (RS)-N3-(1-(1-naphthyl)ethyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide 335476 1-(6-fluoropyridin-3-yl)-3-(3-methoxyquinuclidin-3-yl)-1-phenylprop-2-yn-1-ol 335479 (1R,9R)-17-[(2S)-oxolan-2-ylmethyl]-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-trien-4-ol 335482 (R)-N3-(1-(1-naphthyl)ethyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide 335486 5-(4-hydroxy-3-methoxyphenyl)-3-((7-methyl-1H-indol-3-yl)methylene)indolin-2-one 335488 7-methoxy-N-(4-(4-(5-methoxybenzo[d]isoxazol-3-yl)piperazin-1-yl)butyl)benzofuran-2-carboxamide 335490 potassium (2-(6-(4-octylphenyl)hexyl)-1,3-dioxolan-4-yl)methyl hydrogenphosphate 335496 potassium ((2R,4S)-2-(heptadec-9-enyl)-1,3-dioxolan-4-yl)methyl hydrogenphosphate 335502 3-((1H-pyrrol-3-yl)methylene)-6-(4-hydroxy-3-methoxyphenyl)indolin-2-one 335504 potassium ((2S,4S)-2-(heptadec-9-enyl)-1,3-dioxolan-4-yl)methyl hydrogenphosphate 335511 6-(4-hydroxy-3-methoxyphenyl)-3-(pyrrolidin-2-ylmethylene)indolin-2-one 335514 8-((cis, rac)-4-hydroxy-4-phenyl-tetrahydro-pyran-3-yl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 335517 N3-(2-(benzo[1,3]dioxol-5-yl)ethyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide 335518 3-((1H-pyrrolo[2,3-b]pyridin-3-yl)methylene)-6-(4-hydroxy-3-methoxyphenyl)indolin-2-one 335519 (Z)-3-((1H-imidazol-2-yl)methylene)-6-(4-hydroxy-3-methoxyphenyl)indolin-2-one 335520 8-((cis, rac)-3-hydroxy-3-phenyl-tetrahydro-pyran-4-yl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 335521 1-(2-fluoropyridin-3-yl)-3-(3-methoxyquinuclidin-3-yl)-1-phenylprop-2-yn-1-ol 335522 N-(trans-4-(2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl)cyclohexyl)-2-naphthamide 335524 4-Oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide 335525 (-)-N3-(1-(1,2,3,4-tetrahydronaphthyl))-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide 335527 N3-(phenethyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide 335528 3-(3-methoxyquinuclidin-3-yl)-1-phenyl-1-(pyridazin-3-yl)prop-2-yn-1-ol 335529 3-(3-methoxyquinuclidin-3-yl)-1-phenyl-1-(pyrimidin-5-yl)prop-2-yn-1-ol 335533 5-(4-chloro-3-methylphenyl)-1-(4-methylbenzyl)-N-((1S,2S,4R)-1,3,3-trimethylbicyclo[2.2.1]heptan-2-yl)-1H-pyrazole-3-carboxamide 335535 (Z)-3-((1H-pyrrol-2-yl)methylene)-6-(4-hydroxy-3-methoxyphenyl)indolin-2-one 335540 bis-((-)-N-cyclobutylmethylmorphinan-3-yl) muconate 335541 10-{[(1R,9R)-17-(cyclobutylmethyl)-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2,4,6-trien-4-yl]oxy}-10-oxodecanoic acid 335542 MCL-139 335553 1-phenyl-8-((cis,1R,2R)-2-phenyl-cyclohexyl)-1,3,8-triaza-spiro[4.5]decan-4-one 335557 2-(2-Methoxyphenylamino)-6-(3-acetamidophenyl)pyrazine 335563 ((2S,3S,4R,5R)-5-(2-chloro-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrothiophen-2-yl)(4-(4-fluorophenyl)piperazin-1-yl)methanone 335581 2-(3-Hydroxyphenylamino)-6-(3-acetamidophenyl)pyrazine 335582 2-[4-(Trifluoromethoxy)phenylamino]-6-(3-acetamidophenyl)-pyrazine 335592 1-((-)-N-cyclobutylmethylmorphinan-3-yl) 10-((+)-N-cyclobutylmethylmorphinan-3-yl) sebacoylate 335593 bis-((-)-N-propargylmorphinan-3-yl) sebacoylate 335599 2-(3-Methoxyphenylamino)-6-(3-acetamidophenyl)pyrazine 335604 2-[4-(Morpholinosulfonyl)phenylamino]-6-(3-acetamidophenyl)pyrazine 335605 2-(4-Morpholinophenylamino)-6-(3-acetamidophenyl)pyrazine 335606 2-[3-(2-Aminoethoxy)phenylamino]-6-(3-acetamidophenyl)-pyrazine 335607 N-(3-(6-(4-methoxyphenylamino)pyrazin-2-yl)phenyl)acetamide 335618 2-(3,5-Dimethoxyphenylamino)-6-(3-acetamidophenyl)pyrazine 335622 bis-(3-amino-(-)-N-cyclobutylmethylmorphinan) succinamide 335624 (2S,3S,4R,5R)-5-(2-chloro-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N,N-dimethyl-tetrahydrothiophene-2-carboxamide 335631 (2S,3S,4R,5R)-5-(2-chloro-6-(methylamino)-9H-purin-9-yl)-N-cyclopropyl-3,4-dihydroxy-tetrahydrothiophene-2-carboxamide 335634 2-(3,4-Methylenedioxyphenylamino)-6-(3-acetamidophenyl)-pyrazine 335650 2-[3-(Oxazol-5-yl)phenylamino]-6-(3-acetamidophenyl)pyrazine 335655 bis-(3-amino-(-)-N-cyclobutylmethylmorphinan) sebacamide 335656 bis-((-)-N-cyclobutylmethylmorphinan-3-amino) furamide 335657 (2S,3S,4R,5R)-5-(2-chloro-6-(methylamino)-9H-purin-9-yl)-N-(cyclopropylmethyl)-3,4-dihydroxy-tetrahydrothiophene-2-carboxamide 335660 3-((6-(4-hydroxy-3-methoxyphenyl)-2-oxoindolin-3-ylidene)methyl)-1H-pyrrolo[2,3-b]pyridine-6-carbonitrile 335663 2-(3,4-Dimethoxyphenylamino)-6-(3-acetamidophenyl)pyrazine 335664 (2S,3S,4R,5R)-5-(2-chloro-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-isopentyl-tetrahydrothiophene-2-carboxamide 335665 ((2S,3S,4R,5R)-5-(2-chloro-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrothiophen-2-yl)(morpholino)methanone 335669 2-(2,4-Dimethoxyphenylamino)-6-(3-acetamidophenyl)pyrazine 335670 2-(3-Chlorophenylamino)-6-(3-acetamidophenyl)pyrazine 335671 (4-benzylpiperidin-1-yl)((2S,3S,4R,5R)-5-(2-chloro-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrothiophen-2-yl)methanone 335675 1-(4-chloro-phenyl)-8-((1S,2S)-2-phenyl-cyclohexyl)-1,3,8-triaza-spiro[4.5]decan-4-one 335690 (+)-3-hydroxy-N-cyclobutylmethylmorphinan mandelate 335691 (+)-3-hydroxy-N-cyclopropylmethylmorphinan mandelate 335692 1-((-)-N-cyclobutylmethylmorphinan-3-yl) 10-(3,6-diol-7,8-didehydro-4,5-epoxy-17-methyl-(5alpha,6alpha)morphinan-3-yl) sebacoylate 335693 1-phenyl 10-((-)-N-cyclobutylmethylmorphinan-3-yl) sebacoylate 335694 2-Phenoxyethylamino-6-(3-acetamidophenyl)pyrazine 335712 (2S)-1-(6-methoxy-1H-indazol-1-yl)propan-2-amine 335713 1-((S)-2-aminopropyl)-7-methyl-1H-indazol-6-ol 335714 1-((S)-2-aminopropyl)-7-fluoro-1H-indazol-6-ol 335715 2-(3,4,5-Trimethoxyphenylamino)-6-(3-acetamidophenyl)-pyrazine 335716 2-(Phenylamino)-6-(3-acetamidophenyl)pyrazine 335719 2-(3,4-Dihydro-2H-benzo[b][1,4]dioxepin-7-ylamino)-6-(3-acetamidophenyl)pyrazine 335723 5-(furan-2-yl)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-1H-pyrazole-3-carboxamide 335724 2-(2,2,3,3-Tetrafluoro-2,3-dihydrobenzo[b][1,4]dioxin-6-ylamino)-6-(3-acetamidophenyl)pyrazine 335725 2-(2,2-Difluorobenzo[d][1,3]dioxol-5-ylamino)-6-(3-acetamidophenyl)pyrazine 335729 1-(2-aminoethyl)-1H-indazol-6-ol 335730 1-((S)-2-aminopropyl)-1H-indazol-6-ol 335732 2-(4-Methoxyphenyloxyethylamino)-6-(3-acetamidophenyl)-pyrazine 335738 2-(3,4,5-Trimethoxybenzylamino)-6-(3-acetamidophenyl)pyrazine 335739 2-(3-Fluorophenylmethylamino)-6-(3'-acetamidophenyl)pyrazine 335746 2-(3-Furylmethylamino)-6-(3-acetamidophenyl)pyrazine 335750 2-(Phenyl-N-methylamino)-6-(3-acetamidophenyl)pyrazine 335762 N-(4-(4-(5-methoxybenzo[d]isoxazol-3-yl)piperazin-1-yl)butyl)-3-(pyrimidin-2-yl)benzamide 335776 2-(3-Oxo-1,3-dihydroisobenzofuran-5-ylamino)-6-(3-acetamidophenyl)pyrazine 335777 2-(2,6-Dichloropyridin-4-ylamino)-6-(3-acetamidophenyl)-pyrazine 335782 1-((-)-N-cyclopropylmethylmorphinan-3-yl) 10-(N-cyclobutylmethylmorphinan-3-yl) sebacoylate 335783 (2-chloropurin-9-yl)-3,4-dihydroxytetrahydrothiphene-2-carboxylic acid methyl amide 335786 2-(4-tert-Butylthiazol-2-ylamino)-6-(3-acetamidophenyl)pyrazine 335789 N-(trans-4-(2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl)cyclohexyl)quinoline-6-carboxamide 335790 (2S,3S,4R,5R)-5-(2-chloro-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrothiophene-2-carboxamide 335795 2-(3-Chloro-4-fluorobenzylamino)-6-(3-acetamidophenyl)-pyrazine 335797 N-(trans-4-(2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl)cyclohexyl)quinoline-8-carboxamide 335829 1-((R)-2-aminopropyl)-1H-indazol-6-ol 335838 7-methoxy-N-(4-(4-(quinoxalin-5-yl)piperazin-1-yl)butyl)benzofuran-2-carboxamide 335839 7-methoxy-N-(4-(4-(7-methoxyisoquinolin-1-yl)piperazin-1-yl)butyl)benzofuran-2-carboxamide 335844 2-(Benzylamino)-6-(3-acetamidophenyl)pyrazine 335845 N-(4-(4-(5-methoxybenzo[d]isoxazol-3-yl)piperazin-1-yl)butyl)benzo[c][1,2,5]oxadiazole-5-carboxamide 335846 7-methoxy-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)benzofuran-2-carboxamide 335847 N-(4-(4-(5-methoxybenzo[d]isoxazol-3-yl)piperazin-1-yl)butyl)-3-(5-methyl-1,2,4-oxadiazol-3-yl)benzamide 335849 2-(Phenylethylamino)-6-(3-acetamidophenyl)pyrazine 335850 2-(3-Phenylpropylamino)-6-(3-acetamidophenyl)pyrazine 335854 N-(4-(4-(5-methoxybenzo[d]isoxazol-3-yl)piperazin-1-yl)butyl)-3-morpholinobenzamide 335855 3-(1H-imidazol-1-yl)-N-(4-(4-(5-methoxybenzo[d]isoxazol-3-yl)piperazin-1-yl)butyl)benzamide 335876 N-[4-[4-(5-methoxy-2-benisooazolyl)piperazin-1-yl]butyl]-5-(2-furanyl)-1H-pyrazole-3-carboxamide 335877 N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)benzo[c][1,2,5]oxadiazole-5-carboxamide 335883 2-(2,3-Dihydrobenzo[b][1,4]dioxin-6-ylamino)-6-(3-acetamidophenyl)pyrazine 335887 N-(4-(4-(5-methoxybenzo[d]isoxazol-3-yl)piperazin-1-yl)butyl)quinoxaline-6-carboxamide 335888 N-(4-(4-(5-methoxybenzo[d]isoxazol-3-yl)piperazin-1-yl)butyl)benzo[d][1,3]dioxole-5-carboxamide 335891 N-[4-[4-(5-methoxy-2-benzisoxazolyl)piperazin-1-yl]butyl]-4-(4-morpholinyl)benzamide 335892 N-[4-[4-(5-methoxy-2-benzisoxazolyl)piperazin-1-yl]butyl]-4-(1H-imidazol-1-yl)benzamide 335894 N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]quinoxaline-6-carboxamide 335901 N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)benzo[d][1,3]dioxole-5-carboxamide 335908 1-((S)-2-aminopropyl)-7-chloro-1H-indazol-6-ol 335909 1-((S)-2-aminopropyl)-7-iodo-1H-indazol-6-ol 335913 N-(4-(4-(1H-indazol-3-yl)piperazin-1-yl)butyl)-7-methoxybenzofuran-2-carboxamide 335916 2-(2,3-Dehydro-1,4-benzodioxin-6-methylamino)-6-(3'-acetamidophenyl)pyrazine 335917 2-(3,4-Methylenedioxyphenylaminomethyl)-6-(3-acetamidophenyl)pyrazine 335922 2-[(5-Methyl-3-isoxazolyl)methylamino]-6-(3-acetamidophenyl)pyrazine 335923 2-[(1,5-Dimethyl-1H-pyrazol-3-yl)methylamino]-6-(3-acetamidophenyl)pyrazine 335952 4-(4-bromo-2-fluorophenylamino)-N-(cyclopropylmethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 335953 4-(4-bromo-2-fluorophenylamino)-5-chloro-N-(cyclopropylmethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 336025 N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-4-morpholinobenzamide 336026 4-(1H-imidazol-1-yl)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)benzamide 336059 4-(4-bromo-2-fluorophenylamino)-N-(cyclopropylmethoxy)-5-fluoro-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 336060 4-(4-bromo-2-fluorophenylamino)-N-(cyclopropylmethoxy)-1,5-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide 336098 4-(4-bromo-2-fluorophenylamino)-N-(2-hydroxyethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 336099 4-(4-bromo-2-fluorophenylamino)-5-chloro-N-(2-hydroxyethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 336102 4-(4-bromo-2-fluorophenylamino)-5-fluoro-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 336104 4-(4-bromo-2-fluorophenylamino)-5-fluoro-N-(2-hydroxyethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 336105 4-(4-bromo-2-fluorophenylamino)-N-(2-hydroxyethoxy)-1,5-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide 336113 (S)-N,N-diisobutyl-2-(2-(4-methoxy-3,5-dimethylphenyl)-3-(1-(phenethylamino)propan-2-yl)-1H-indol-5-yl)-2-methylpropanamide 336142 9-[3-(1-Ethyl-propylamino)-propyl]-8-2-iodo-5-methoxy-phenylsulfanyl)-9H-purin-6-ylamine 336144 4-(4-bromo-2-fluorophenylamino)-5-fluoro-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxylic acid 336145 4-(4-bromo-2-fluorophenylamino)-5-fluoro-N,1-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide 336152 4-(4-bromo-2-fluorophenylamino)-N-(cyclopropylmethyl)-5-fluoro-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 336153 4-(4-bromo-2-fluorophenylamino)-5-fluoro-N-hydroxy-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 336154 4-(4-bromo-2-fluorophenylamino)-5-fluoro-N-methoxy-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 336169 pGlu-His-Trp-Ser-His-D-Tyr-Leu-Arg-Pro-Gly-NH2 336190 4-(4-bromo-2-fluorophenylamino)-N-ethoxy-5-fluoro-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 336191 4-(4-bromo-2-fluorophenylamino)-N-methoxy-1,5-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide 336199 4-(4-bromo-2-fluorophenylamino)-N-ethoxy-1,5-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide 336209 9-Butyl-8-(2-chloro-5-methoxy-benzyl)-9H-purin-6-ylamine 336223 8-(2-Iodo-5-methoxy-phenylsulfanyl)-9-(2-isobutylamino-ethyl)-9H-purin-6-ylamine 336234 8-(2-Iodo-5-methoxy-phenylsulfanyl)-9-(4-methyl-pent-3-enyl)-9H-purin-6-ylamine 336235 8-(2-Iodo-5-methoxy-phenylsulfanyl)-9-(3-isopropylaminopropyl)-9H-purin-6-ylamine 336258 9-Butyl-8-(2-iodo-5-methoxy-benzyl)-9H-purin-6-ylamine 336259 9-Butyl-8-(2,5-dimethoxy-phenylsulfanyl)-9H-purin-6-ylamine 336278 2-Fluoro-8-(2-iodo-5-methoxy-phenylsulfanyl)-9-pent-4-ynyl-9H-purin-6-ylamine 336286 9-(3-sec-Butylamino-propyl)-8-(2-iodo-5-methoxy-phenylsulfanyl)-9H-purin-6-ylamine 336297 4-(4-bromo-2-chlorophenylamino)-5-chloro-N-(2-hydroxyethoxy)-6-methoxynicotinamide 336300 8-(2-iodo-5-methoxyphenylthio)-9-(2-(neopentylamino)ethyl)-9H-purin-6-amine 336303 4-(4-bromo-2-chlorophenylamino)-5,6-dichloro-N-(2-hydroxyethoxy)nicotinamide 336324 8-(2-Bromo-5-methoxy-benzyl)-9-butyl-9H-purin-6-ylamine 336326 9-(3-(tert-butylamino)propyl)-8-(2-iodo-5-methoxyphenylthio)-9H-purin-6-amine 336537 7-ethyl-6,7,8,9,14,15-hexahydro-5H-benz[d]indolo[2,3-g]azecine 336538 2,3-dimethoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 336544 7-cyclopropylmethyl-6,7,8,9,14,15-hexahydro-5H-benz[d]indolo[2,3-g]azecine 336546 3,6-dimethyl-4,5,6,7,8,13-hexahydro-3H-pyrrolo[2,3-f][3]benzazecine 336559 6-methyl-4,5,6,7,8,13-hexahydrothieno[2,3-f][3]benzazecine 336628 3-methyl-6-phenyl-1,2,3,4,5,6,7,8-octahydroazonino[5,4-b]indole 336646 7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 336666 7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecin-3-ol 336674 N-(4-benzoylphenyl)-2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336675 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(4-((pyrrolidin-1-ylsulfonyl)methyl)phenyl)acetamide 336676 N-(4-(benzyloxy)phenyl)-2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336677 N-(4-methoxyphenethyl)-4-(2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamido)benzamide 336678 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(4-(phenylsulfonyl)phenyl)acetamide 336681 c[Thr-Tyr-Thr-His-DNaf-Arg-Trp-Thr-Ile-Pro] 336685 2-(4-(2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamido)phenyl)acetic acid 336686 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(4-hydroxyphenyl)acetamide 336687 N-(4-(4,4-dimethyl-4,5-dihydrooxazol-2-yl)phenyl)-2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336688 N-(4-chlorophenyl)-2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336691 N-biphenyl-4-yl-2-[4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-phenoxy]-acetamide 336692 N-(4-bromophenyl)-2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)propanamide 336693 4-(azetidin-1-yl)-1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)pyrimidin-2(1H)-one 336694 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-4-(piperidin-1-yl)pyrimidin-2(1H)-one 336695 ethyl 2-(4-(2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamido)phenyl)acetate 336696 2-[4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-phenoxy]-N-(4-sulfamoyl-phenyl)-acetamide 336697 N-(4-bromophenyl)-2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336698 2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(4-fluorophenyl)acetamide 336699 8-{5-[2-(4-fluoro-phenyl)-2-oxo-ethoxy]-2-methyl-2H-pyrazol-3-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 336700 2-(4-(7-chloro-2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(3-fluorophenyl)acetamide 336701 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(4-formylphenyl)acetamide 336703 2-(4-(1,3-diethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-phenylacetamide 336704 N-(4-fluorophenyl)-2-(4-(3-methyl-2,4-dioxo-1-propyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336705 8-{5-[2-(4-bromo-phenyl)-2-oxo-ethoxy]-2-methyl-2H-pyrazol-3-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 336709 N-benzyl-2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336710 ethyl 4-(2-(4-(1-methyl-2,4-dioxo-3-propyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamido)benzoate 336711 2-(4-(7-chloro-2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-p-tolylacetamide 336714 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(4-fluorophenyl)propanamide 336715 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(4-fluorophenyl)acetamide 336716 N-(4-tert-butylphenyl)-2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336717 N-(4-bromophenyl)-2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-3-methoxyphenoxy)acetamide 336718 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(2-hydroxyphenyl)acetamide 336719 2-(4-(1-methyl-2,4-dioxo-3-propyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-phenylacetamide 336721 2-(3-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)propylthio)pyrimidin-4-ol 336722 4-(2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamido)-N,N,N-trimethylbenzenaminium 336723 N-(4-acetylphenyl)-2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336724 N-(4-cyanophenyl)-2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336725 N-(4-fluorophenyl)-2-(4-(1-methyl-2,4-dioxo-3-propyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336726 N-(4-cyanophenyl)-2-(4-(1,3-diethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336727 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-4-hydroxy-5-methylpyrimidin-2(1H)-one 336729 2-(4-(7-chloro-2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(2-fluorophenyl)acetamide 336730 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(4-fluorophenyl)butanamide 336731 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-2-methyl-N-phenylpropanamide 336732 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(4-fluorophenyl)-2-methylpropanamide 336733 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(4-iodophenyl)acetamide 336734 2-(4-(7-chloro-2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(4-chlorophenyl)acetamide 336735 8-[2-methyl-5-(2-oxo-2-p-tolyl-ethoxy)-2H-pyrazol-3-yl]-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 336737 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-phenylpropanamide 336738 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(4-methoxyphenyl)propanamide 336740 N-(4-bromophenyl)-2-(4-(7-chloro-2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336741 2-(4-(1-(3-methoxypropyl)-3-methyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-phenylacetamide 336749 2-(4-(3-methyl-2,4-dioxo-1-propyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-phenylacetamide 336750 ethyl 2-(4-(2-(4-(1-methyl-2,4-dioxo-3-propyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamido)phenyl)acetate 336754 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-phenylacetamide 336755 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-phenylbutanamide 336756 2-(4-(7-bromo-2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-phenylacetamide 336757 4-(2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamido)benzamide 336761 N-(4-bromophenyl)-2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)butanamide 336762 N-(4-(cyanomethyl)phenyl)-2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336763 2-(4-(7-chloro-2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(2-chlorophenyl)acetamide 336764 2-(4-(7-chloro-2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(4-methoxyphenyl)acetamide 336765 N-cyclopentyl-2-(4-(1-(3-methoxypropyl)-3-methyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336772 N-(4-bromophenyl)-2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336776 2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-phenylacetamide 336777 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(4-methoxyphenyl)acetamide 336778 2-(4-(7-bromo-2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(4-fluorophenyl)acetamide 336779 N-(4-acetylphenyl)-2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336780 2-(4-(7-chloro-2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(4-fluorophenyl)acetamide 336781 2-(4-(7-chloro-2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-phenylacetamide 336782 N-(4-acetylphenyl)-2-(4-(7-chloro-2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336783 N-(2,3-dihydro-1H-inden-1-yl)-2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336784 2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-3-methoxyphenoxy)-N-(4-fluorophenyl)acetamide 336785 2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(4-fluorophenyl)propanamide 336786 2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-phenylpropanamide 336789 ethyl 4-(2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamido)benzoate 336793 2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(4-nitrophenyl)acetamide 336794 N-(4-iodophenyl)-2-(4-(1-methyl-2,4-dioxo-3-propyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336799 N-(4-acetylamino-phenyl)-2-[4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-phenoxy]-acetamide 336800 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-p-tolylacetamide 336802 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-4-phenylpyrimidin-2(1H)-one 336804 8-{5-[2-(4-fluoro-phenyl)-2-oxo-ethoxy]-1-methyl-1H-pyrazol-3-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 336808 N-(4-bromophenyl)-2-(N-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenyl)formamido)acetamide 336811 N-(4-chlorobenzyl)-2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-3-methoxyphenoxy)acetamide 336819 N-(4-fluorobenzyl)-2-(4-(7-chloro-2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336820 N-(4-chlorobenzyl)-2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-2-methoxyphenoxy)acetamide 336822 N-(4-bromophenyl)-2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-2-methoxyphenoxy)acetamide 336823 2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-3-methoxyphenoxy)-N-phenylacetamide 336826 2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(1,3,4-thiadiazol-2-yl)acetamide 336827 N-benzyl-2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-methylacetamide 336831 N-cyclopentyl-2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336836 (R)-2-{3-[3-(4-Benzoylphenyl)ureido]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl}-N-(4-methoxyphenyl)-N-methylacetamide 336838 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(4-(trifluoromethoxy)phenyl)acetamide 336839 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-5-chloro-4-hydroxypyrimidin-2(1H)-one 336840 8-{5-[2-(4-bromo-phenyl)-2-oxo-ethoxy]-1-methyl-1H-pyrazol-3-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 336845 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-4-hydroxy-5-(trifluoromethyl)pyrimidin-2(1H)-one 336846 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-4-hydroxy-2-oxo-1,2-dihydropyrimidine-5-carbonitrile 336850 (4-((1H-1,2,4-triazol-1-yl)methyl)-4-cyclohexylpiperidin-1-yl)((1R,2R,4R)-2-(4-chlorophenyl)-4-(dimethylamino)cyclopentyl)methanone 336854 (R)-2-{3-[3-(4-Benzoylphenyl)ureido]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-benzo[b][1,4]diazepin-1-yl}-N-isopropyl-N-(4-methoxyphenyl)acetamide 336855 (S)-2-{3-[3-(4-Benzoylphenyl)ureido]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-benzo[b][1,4]diazepin-1-yl}-N-isopropyl-N-(4-methoxyphenyl)acetamide 336856 2-benzoyl-N-(3-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}propyl)benzamide 336857 N-(3-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}propyl)-3-phenoxybenzamide 336860 N-(4-chlorobenzyl)-2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)propanamide 336861 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(6-methoxypyridin-3-yl)acetamide 336867 N-(2,6-dimethoxypyrimidin-4-yl)-2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336868 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(5-methylpyridin-2-yl)acetamide 336882 2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-2-methoxyphenoxy)-N-(4-fluorophenyl)acetamide 336883 2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-2-methoxyphenoxy)-N-phenylacetamide 336886 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-3-methylpyrimidine-2,4(1H,3H)-dione 336891 c[Ser-Tyr-Thr-His-Dphe-Arg-Trp-Thr-Ile-Pro] 336892 N-(4-(2-aminoethyl)phenyl)-2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336896 N-[3-spiro(2,3-dihydro-1H-indene-1,4'-piperidine)-1-ylpropyl]-L-(-)-3-phenyllactoamide 336899 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-3,5-dimethylpyrimidine-2,4(1H,3H)-dione 336901 N-benzyl-2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336903 8-{5-[2-(4-acetyl-phenyl)-2-oxo-ethoxy]-2-methyl-2H-pyrazol-3-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 336909 N-(3-methoxybenzyl)-2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336910 N-benzyl-2-(4-(7-chloro-2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336914 N-(1H-benzo[d]imidazol-2-yl)-2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336924 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-5-ethyl-4-hydroxypyrimidin-2(1H)-one 336925 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-5-fluoro-4-hydroxypyrimidin-2(1H)-one 336929 N-(6-methoxypyridin-3-yl)-2-(4-(1-methyl-2,4-dioxo-3-propyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336931 N-(3-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}propyl)-2-phenylacetamide 336932 4-{2-[5-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-1-methyl-1H-pyrazol-3-yloxy]-acetyl}-benzoic acid ethyl ester 336939 1,3,5-triphenylimidazolidine-2,4-dione 336940 5-(4-chlorophenyl)-1,3-diphenylimidazolidine-2,4-dione 336948 1,3-bis(3-chlorophenyl)-5-(4-chlorophenyl)imidazolidine-2,4-dione 336949 5-(4-bromophenyl)-1,3-bis(4-chlorophenyl)imidazolidine-2,4-dione 336950 N-[3-spiro(2,3-dihydro-1H-indene-1,4'-piperidine)ylpropyl]-1,1'-biphenyl-2-carboxyamide 336954 N-(4-bromophenyl)-2-(3-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 336955 2-(4-(7-chloro-2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetic acid 336956 2-(4-(1-(3-methoxypropyl)-3-methyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetic acid 336957 (2E)-N-(3-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}propyl)-3-phenylprop-2-enamide 336958 N-(3-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}propyl)-2-phenylcyclopropane-1-carboxamide 336960 2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(furan-2-ylmethyl)acetamide 336963 2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-2-methoxyphenoxy)acetic acid 336964 ethyl 2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetate 336966 2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(1-phenylethyl)acetamide 336967 N-benzyl-2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-ethylacetamide 336982 8-{5-[2-(4-Iodo-phenyl)-2-oxo-ethoxy]-pyridin-2-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 336984 5-(4-bromophenyl)-1,3-diphenyl-2-thioxoimidazolidin-4-one 336986 (5-(2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetyl)-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)carbamic acid 336987 1,3-bis(3-iodophenyl)-5-phenyl-2-thioxoimidazolidin-4-one 336988 1,3-bis(4-methylphenyl)-5-phenyl-2-thioxoimidazolidin-4-one 336991 1,3-bis(4-chlorophenyl)-5-phenyl-2-thioxoimidazolidin-4-one 336992 2-(3-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-phenylacetamide 337008 2-(4-(1,3-bis(cyclopropylmethyl)-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-phenylacetamide 337012 5-benzo[1,3]dioxol-5-yl-2-oxo-1,2-dihydro-pyridine-3-carboxylic acid [4-(4-methyl-piperazin-1-yl)-phenyl]-amide 337013 1,3-bis(4-methoxyphenyl)-5-phenyl-2-thioxoimidazolidin-4-one 337015 N-biphenyl-4-yl-2-[4-(1-methyl-2,4-dioxo-3-propyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-phenoxy]-acetamide 337018 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-4-hydroxypyrimidin-2(1H)-one 337021 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-4-cyclohexylpyrimidin-2(1H)-one 337028 2-(4-(3-ethyl-1-(3-methoxypropyl)-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetic acid 337029 1,3-bis(4,3-dichlorophenyl)-5-phenyl-2-thioxoimidazolidin-4-one 337030 1,3-bis(4-bromophenyl)-5-phenyl-2-thioxoimidazolidin-4-one 337041 N-(4-chlorobenzyl)-2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 337042 N-(4-fluorobenzyl)-2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 337044 8-{4-[2-(4-iodo-phenyl)-2-oxo-ethoxy]-phenyl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 337048 2-(4-(7-bromo-2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetic acid 337049 N-(4-chlorobenzyl)-2-(4-(1-methyl-2,4-dioxo-3-propyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 337055 2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetic acid 337065 N-(4-cyanophenyl)-2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-2-methoxyphenoxy)acetamide 337066 1,3,5-tris(4-chlorophenyl)imidazolidine-2,4-dione 337087 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)pyrimidin-2(1H)-one 337089 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(pyridin-4-ylmethyl)acetamide 337090 6-(4-(2-(3-amino-1H-pyrazol-1-yl)-2-oxoethoxy)phenyl)-1,3-dipropyl-1H-pyrrolo[3,2-d]pyrimidine-2,4(3H,5H)-dione 337110 (S)-2-{3-[3-(4-Benzoylphenyl)ureido]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl}-N-(4-methoxyphenyl)-N-methylacetamide 337118 5-(4-bromophenyl)-1,3-diphenylimidazolidine-2,4-dione 337119 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetic acid 337125 2-(4-(1-methyl-2,4-dioxo-3-propyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetic acid 337126 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)propanoic acid 337143 2-(4-(3-methyl-2,4-dioxo-1-propyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetic acid 337144 ethyl 2-(4-(1-(3-methoxypropyl)-3-methyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetate 337148 (1S,7aS)-1-{[(4-amino-5-chloro-2-methoxybenzoyl)amino]methyl}-4-methylhexahydro-1H-pyrrolizinium, iodide 337150 5-benzo[1,3]dioxol-5-yl-2-oxo-1,2-dihydro-pyridine-3-carboxylic acid {4-[2-(4-methyl-piperazin-1-yl)-ethyl]-phenyl}-amide 337152 ethyl 2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-2-methoxyphenoxy)acetate 337160 4-amino-5-chloro-2-ethoxy-N-[(1S,7aS)-hexahydro-1H-pyrrolizin-1-ylmethyl]benzamide 337176 1,3-bis(4-chlorophenyl)-5-phenylimidazolidine-2,4-dione 337177 1,3-bis(3-chlorophenyl)-5-phenylimidazolidine-2,4-dione 337184 1,3-bis(4-bromophenyl)-5-phenylimidazolidine-2,4-dione 337185 1,3-bis(4-methoxyphenyl)-5-phenylimidazolidine-2,4-dione 337192 ethyl 2-(4-(3-ethyl-1-(3-methoxypropyl)-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetate 337199 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(3-hydroxypyridin-2-yl)acetamide 337201 2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-3-methoxyphenoxy)acetic acid 337202 ethyl 2-(4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-3-methoxyphenoxy)acetate 337207 (5-(2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamido)-1-methyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)carbamic acid 337214 2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)-N-(pyridin-2-yl)acetamide 337257 (R)-N-(3-(3H-spiro[isobenzofuran-1,4'-piperidine]-1'-yl)propyl)-1-benzylpyrrolidine-2-carboxamide 337275 2-Benzyloxy-N-[3-spiro(2,3-dihydro-1H-indene-1,4'-piperidine)-1-ylpropyl]benzamide 337276 1-benzyl-N-[3-spiro(2,3-dihydro-1H-indene-1,4'-piperidine)-1-ylpropyl]-L-prolineamide 337277 (1R,7aS)-hexahydro-1H-pyrrolizin-1-ylmethyl 4-amino-5-chloro-2-methoxybenzoate 337290 cis-N-[(hexahydro-1H-pyrrolizin-l-yl)methyl]-2,3-dihydro-3-(1-methylethyl)-2-oxo-lH-benzimidazole-l-carboxamide 337293 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-4-cyclopropylpyrimidin-2(1H)-one 337294 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-4-cyclobutylpyrimidin-2(1H)-one 337324 2-phenoxy-N-[3-spiro(2,3-dihydro-1H-indene-1,4'-piperidine)-1-ylpropyl]benzamide 337343 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-4-ethoxypyrimidin-2(1H)-one 337352 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-4-methylpyrimidin-2(1H)-one 337353 4-tert-butyl-1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)pyrimidin-2(1H)-one 337357 N-(3-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}propyl)-1-phenylcyclohexane-1-carboxamide 337375 2-(4-chlorophenoxy)-N-(3-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}propyl)-2-methylpropanamide 337392 (1S,7aR)-hexahydro-1H-pyrrolizin-1-ylmethyl 1-methyl-1Hindazole-3-carboxylate 337422 (4S,5S)-4-benzyl-N-(3-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}propyl)-2-oxo-1,3-oxazolidine-5-carboxamide 337428 N-(3-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}propyl)-3-(1H-indol-3-yl)propanamide 337466 N-(3-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}propyl)-2-(phenylsulfanyl)acetamide 337469 1-benzyl-N-[3-spiro(2,3-dihydro-1H-indene-1,4'-piperidine)-1-ylpropyl]-D-prolineamide 337488 (1R,7aS)-hexahydro-1H-pyrrolizin-1-ylmethyl 1-Methyl-1Hindole-3-carboxylate 337490 (1R,7aS)-hexahydro-1H-pyrrolizin-1-ylmethyl 5-Fluoro-1Hindole-3-carboxylate 337491 benzyl (4R)-4-[(3-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}propyl)carbamoyl]-1,3-oxazolidine-3-carboxylate 337492 N-(3-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}propyl)-2-(phenylamino)benzamide 337493 2-(1,3-benzothiazol-2-ylsulfanyl)-N-(3-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}propyl)acetamide 337499 (1S,7aR)-hexahydro-1H-pyrrolizin-1-ylmethyl 1H-indazole-3-carboxylate 337530 N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methyl-2-(phenylamino)acetamide 337543 N-(3-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}propyl)-2-(3-phenoxyphenyl)acetamide 337551 2-benzyl-N-(3-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}propyl)benzamide 337558 N-exo-((4S,7alphaS)-tetrahydro-1H-pyrrolizin-4(5H)-yl)-6-chloroimidazo[1,2-a]pyridine-8-carboxamide 337572 2-(pyridin-4-ylmethylamino)-N-(quinolin-3-yl)benzamide 337578 (2R)-1-benzyl-N-(3-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}propyl)-5-oxopyrrolidine-2-carboxamide 337586 (4R)-3-benzyl-N-(3-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}propyl)-2-oxo-1,3-oxazolidine-4-carboxamide 337594 N-(3-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}propyl)-2-(1H-indol-3-yl)-2-oxoacetamide 337629 N-(3-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}propyl)-2-phenoxypropanamide 337640 N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methyl-2-(4-(trifluoromethyl)phenylamino)acetamide 337663 2-(3,4-dichlorophenylamino)-N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methylacetamide 337670 N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methyl-2-(4-nitrophenylamino)acetamide 337760 N-(4-tert-butylphenyl)-4-(2-(pyridin-4-yl)ethyl)thiazole-5-carboxamide 337761 N-(2-fluoro-4-methylphenyl)-4-(2-(pyridin-4-yl)ethyl)thiazole-5-carboxamide 337762 N-(benzo[d][1,3]dioxol-5-yl)-4-(2-(pyridin-4-yl)ethyl)thiazole-5-carboxamide 337774 2-(4-cyanophenylamino)-N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methylacetamide 337775 5-methoxy-7,12-dioxo-7,12-dihydro-dinaphtho[1,2-b;2',3'-d]furan-6-carboxylic acid methyl ester 337777 5-(2-dimethylamino-ethoxy)-7,12-dioxo-7,12-dihydro-dinaphtho[1,2-b;2',3'-d]furan-6-carboxylic acid methylester 337789 N-(3-acetyl-6-(4-chlorophenyl)-7-(2,4-dichlorophenyl)-1-(2-hydroxyethyl)-2-oxo-1,2-dihydro-1,8-naphthyridin-4-yl)acetamide 337790 N-(3-acetyl-6-(4-chlorophenyl)-7-(2,4-dichlorophenyl)-2-oxo-1,2-dihydro-1,8-naphthyridin-4-yl)acetamide 337798 N-(3-acetyl-6-(4-chlorophenyl)-7-(2,4-dichlorophenyl)-1-methyl-2-oxo-1,2-dihydro-1,8-naphthyridin-4-yl)-2-methoxyacetamide 337804 N-(3,4-dichlorophenyl)-4-(2-(isoxazol-4-yl)ethyl)thiazole-5-carboxamide 337807 N-(6-(4-chlorophenyl)-7-(2,4-dichlorophenyl)-3-(dimethylamino)-1-methyl-2-oxo-1,2-dihydro-1,8-naphthyridin-4-yl)acetamide 337809 N-(4-tert-butylphenyl)-4-(2-(quinolin-4-yl)ethyl)thiazole-5-carboxamide 337811 N-(4-bromophenyl)-4-(2-(pyridin-4-yl)ethyl)thiazole-5-carboxamide 337814 2-(3-cyanophenylamino)-N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methylacetamide 337815 2-(2-cyanophenylamino)-N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methylacetamide 337817 N-(4-isopropylphenyl)-4-(2-(isoxazol-4-yl)ethyl)thiazole-5-carboxamide 337822 N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methyl-2-(methyl(phenyl)amino)acetamide 337831 N-(3,4-dichlorophenyl)-4-(2-(pyridin-4-yl)ethyl)thiazole-5-carboxamide 337832 N-(4-chloro-3-(trifluoromethyl)phenyl)-4-(2-(isoxazol-4-yl)ethyl)thiazole-5-carboxamide 337838 N-(3-acetyl-6-(4-chlorophenyl)-7-(2,4-dichlorophenyl)-1-(2-methoxyethyl)-2-oxo-1,2-dihydro-1,8-naphthyridin-4-yl)acetamide 337854 N-(6-(4-chlorophenyl)-7-(2,4-dichlorophenyl)-3-methoxy-1-methyl-2-oxo-1,2-dihydro-1,8-naphthyridin-4-yl)acetamide 337855 N-(6-(4-chlorophenyl)-7-(2,4-dichlorophenyl)-1,3-dimethyl-2-oxo-1,2-dihydro-1,8-naphthyridin-4-yl)acetamide 337862 N-(3-acetyl-6-(4-chlorophenyl)-7-(2,4-dichlorophenyl)-2-oxo-1-((tetrahydrofuran-2-yl)methyl)-1,2-dihydro-1,8-naphthyridin-4-yl)acetamide 337866 N-(4-isopropylphenyl)-4-(2-(pyridin-4-yl)ethyl)thiazole-5-carboxamide 337869 N-(3-acetyl-6-(4-chlorophenyl)-7-(2,4-dichlorophenyl)-1-methyl-2-oxo-1,2-dihydro-1,8-naphthyridin-4-yl)acetamide 337871 2-(Acetyl-phenyl-amino)-N-[(S)-2-((S)-3-hydroxy-pyrrolidin-1-yl)-1-phenyl-ethyl]-N-methyl-acetamide 337878 N-(6-(4-chlorophenyl)-7-(2,4-dichlorophenyl)-3-isopropyl-1-methyl-2-oxo-1,2-dihydro-1,8-naphthyridin-4-yl)acetamide 337880 N-(4-tert-butylphenyl)-4-(2-(isoxazol-4-yl)ethyl)thiazole-5-carboxamide 337881 N-(4-chloro-3-(trifluoromethyl)phenyl)-4-(2-(pyridin-4-yl)ethyl)thiazole-5-carboxamide 337882 N-(2-fluoro-4-methylphenyl)-4-(2-(isoxazol-4-yl)ethyl)thiazole-5-carboxamide 337905 N-(4-chlorophenyl)-4-(2-(quinolin-4-yl)ethyl)thiazole-5-carboxamide 337908 1-(3-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)propyl)-3,4-dihydroquinolin-2(1H)-one 337918 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-3,4-dihydroquinolin-2(1H)-one 337920 N-(3-acetyl-6-(4-chlorophenyl)-7-(2,4-dichlorophenyl)-1-isobutyl-2-oxo-1,2-dihydro-1,8-naphthyridin-4-yl)acetamide 337924 N-(4-morpholinophenyl)-4-(2-(pyridin-4-yl)ethyl)thiazole-5-carboxamide 337928 N-(3-acetyl-6-(4-chlorophenyl)-7-(2,4-dichlorophenyl)-1-methyl-2-oxo-1,2-dihydro-1,8-naphthyridin-4-yl)-2-hydroxyacetamide 337929 3-acetyl-6-(4-chlorophenyl)-7-(2,4-dichlorophenyl)-1,4-dimethyl-1,8-naphthyridin-2(1H)-one 337930 N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methyl-2-(4-(methylsulfonamido)phenylamino)acetamide 337931 N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methyl-2-(4-(propylsulfonamido)phenylamino)acetamide 337933 N-(4-phenoxyphenyl)-4-(2-(pyridin-4-yl)ethyl)thiazole-5-carboxamide 337936 5-(2-diethylamino-ethoxy)-7,12-dioxo-7,12-dihydro-dinaphtho[1,2-b;2',3'-d]furan-6-carboxylic acid methyl ester 337937 5-(3-dimethylamino-propoxy)-7,12-dioxo-7,12-dihydro-dinaphtho[1,2-b;2',3'-d]furan-6-carboxylic acid methyl ester 337945 7,12-dioxo-5-(2-pyrrolidin-1-yl-ethoxy)-7,12-dihydro-dinaphtho[1,2-b;2',3'-d]furan-6-carboxylic acid methyl ester 337948 N-(4-(chlorodifluoromethoxy)phenyl)-4-(2-(isoxazol-4-yl)ethyl)thiazole-5-carboxamide 337956 2-((4-cyanophenyl)(methyl)amino)-N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methylacetamide 337957 N-(4-(chlorodifluoromethoxy)phenyl)-4-(2-(pyridin-4-yl)ethyl)thiazole-5-carboxamide 337962 N-(3-acetyl-1-benzyl-6-(4-chlorophenyl)-7-(2,4-dichlorophenyl)-2-oxo-1,2-dihydro-1,8-naphthyridin-4-yl)acetamide 337976 2-((6S)-6-isopropyl-3-methylcyclohex-2-enyl)-5-(2-methyloctan-2-yl)benzene-1,3-diol 337983 2-((2S)-2-isopropyl-5-methylcyclohexyl)-5-pentylbenzene-1,3-diol 337985 3-acetyl-6-(4-chlorophenyl)-7-(2,4-dichlorophenyl)-4-(dimethylamino)-1-methyl-1,8-naphthyridin-2(1H)-one 337988 N-(4-chlorophenyl)-4-(2-(isoxazol-4-yl)ethyl)thiazole-5-carboxamide 337992 3-acetyl-4-amino-6-(4-chlorophenyl)-7-(2,4-dichlorophenyl)-1-methyl-1,8-naphthyridin-2(1H)-one 337993 N-(6-(4-chlorophenyl)-3-cyano-7-(2,4-dichlorophenyl)-1-methyl-2-oxo-1,2-dihydro-1,8-naphthyridin-4-yl)acetamide 337995 N-(4-chlorophenyl)-4-(2-(pyridin-4-yl)ethyl)thiazole-5-carboxamide 338001 N-(6-(4-chlorophenyl)-7-(2,4-dichlorophenyl)-1-methyl-2-oxo-1,2-dihydro-1,8-naphthyridin-4-yl)acetamide 338002 4-(2-(pyridin-4-yl)ethyl)-N-m-tolylthiazole-5-carboxamide 338009 N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methyl-2-(4-(methylsulfonamidomethyl)phenylamino)acetamide 338010 N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methyl-2-(3-(methylsulfonamidomethyl)phenylamino)acetamide 338011 4-(2-(isoxazol-4-yl)ethyl)-N-(4-morpholinophenyl)thiazole-5-carboxamide 338017 N-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N-methyl-2-(2-(methylsulfonamidomethyl)phenylamino)acetamide 338020 N-1,1'-biphenyl-4-yl-4-(2-pyridin-4-ylethyl)-1,3-thiazole-5-carboxamide 338031 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)-2-methylbut-2-enyl)-3,4-dihydroquinolin-2(1H)-one 338037 3-(2-alpha-ethyl-trans-4,5-dimethyl-1-phenethylpiperidin-4-yl)phenol 338038 (R)-1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)-2-methylbutyl)-3,4-dihydroquinolin-2(1H)-one 338044 3-(trans-4,5-dimethyl-1-phenethyl-2-alpha-propylpiperidin-4-yl)phenol 338054 3-(trans-4,5-dimethyl-1-phenethyl-2-alpha-phenylpiperidin-4-yl)phenol 338058 (S)-1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)pentyl)-3,4-dihydroquinolin-2(1H)-one 338059 4-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-2H-benzo[b][1,4]oxazin-3(4H)-one 338060 3-(2-alpha-benzyl-trans-4,5-dimethyl-1-phenethylpiperidin-4-yl)phenol 338061 3-(trans-4,5-dimethyl-1,2(alpha)-diphenethylpiperidin-4-yl)phenol 338077 3-(trans-4,5-dimethyl-1-(3-phenylpropyl)-2-alpha-propylpiperidin-4-yl)phenol 338078 3-(1-methyl-4,5-trans-dimethyl-2-alpha-propylpiperidin-4-yl)phenol 338079 3-(1-ethyl-trans-4,5-dimethyl-2-alpha-propylpiperidin-4-yl)phenol 338094 N-(3-fluorophenyl)-2-(2-(7-(3-(4-(hydroxymethyl)piperidin-1-yl)propoxy)-6-methoxyquinazolin-4-ylamino)thiazol-5-yl)acetamide 338103 3-(2(alpha),4,5(trans)-trimethyl-1-phenethylpiperidin-4-yl)phenol 338104 3-(trans-4,5-dimethyl-1-phenethyl-2-alpha-(3-phenylpropyl)piperidin-4-yl)phenol 338106 (S)-1-(1H-pyrrolo[3,2-h]quinolin-1-yl)propan-2-amine 338107 2-((2S)-2-isopropyl-5-methylcyclohexyl)-5-(2-methyloctan-2-yl)benzene-1,3-diol 338109 3-(trans-4,5-dimethyl-2-alpha-propylpiperidin-4-yl)phenol 338110 3-(1-benzyl-4,5-trans-dimethyl-2-alpha-propylpiperidin-4-yl)phenol 338129 1-(5-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)pentyl)-3,4-dihydroquinolin-2(1H)-one 338130 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)but-2-enyl)-3,4-dihydroquinolin-2(1H)-one 338133 3-(indole-3-yl)-4-(3,4-dimethoxyphenyl)-1H-pyrrole-2,5-dione 338134 2-(2-cyclopropoxy-5-(trifluoromethoxy)benzylamino)-1-(4-fluorophenyl)-8-aza-bicyclo[3.2.1]octane-6-carboxylic acid 338139 N-(3,5-bis(trifluoromethyl)benzyl)-1-phenyl-8-aza-bicyclo[3.2.1]octan-2-amine 338143 3-(2-alpha-isopropyl-trans-4,5-dimethyl-1-phenethylpiperidin-4-yl)phenol 338144 3-(2-alpha-butyl-trans-4,5-dimethyl-1-phenethylpiperidin-4-yl)phenol 338147 N-(2-methoxy-5-(trifluoromethoxy)benzyl)-1-phenyl-8-aza-bicyclo[3.2.1]octan-2-amine 338148 5,6,7-trimethoxy-1,2,3,8-tetrahydro-benzo[a]pyrrolo[3,4-c]-carbazol-1,3-dione 338149 (S)-N-(2-methoxybenzyl)-1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-amine 338151 3-(2-alpha-(2-aminoethyl)-trans-4,5-dimethyl-1-phenethylpiperidin-4-yl)phenol 338152 N-(2-(4-(3-hydroxyphenyl)-trans-4,5-dimethyl-1-phenethylpiperidin-2(alpha)-yl)ethyl)acetamide 338155 N-((2-(2-cyclopropoxy-5-(trifluoromethoxy)benzylamino)-1-(4-fluorophenyl)-8-aza-bicyclo[3.2.1]octan-6-yl)methyl)methanesulfonamide 338158 7,12-dioxo-5-(2-piperidin-1-yl-ethoxy)-7,12-dihydro-dinaphtho[1,2-b;2',3'-d]furan-6-carboxylic acid methyl ester 338162 (S)-N-(cyclohexylmethyl)-1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-amine 338169 (S)-N-(1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-yl)prop-2-en-1-amine 338175 (S)-1-(5-chloro-1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-amine 338188 2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-(2,2,2-trifluoroethyl)-2H-pyrazolo[3,4-d]pyridazin-7(6H)-one 338194 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-7,8-dimethoxy-3,4-dihydro-1H-benzo[b]azepine-2,5-dione 338195 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)azepane-2,5-dione 338199 N-(2-(4-(3-hydroxyphenyl)-trans-4,5-dimethyl-1-phenethylpiperidin-2(alpha)-yl)ethyl)benzamide 338202 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-3,4-dihydro-1H-benzo[b]azepine-2,5-dione 338227 3-(trans-4,5-dimethyl-1,2(alpha)-dipropylpiperidin-4-yl)phenol 338228 3-(1-butyl-trans-4,5-dimethyl-2-alpha-propylpiperidin-4-yl)phenol 338229 3-(trans-4,5-dimethyl-1-pentyl-2-alpha-propylpiperidin-4-yl)phenol 338235 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-6-hydroxy-4,5-dihydro-1H-benzo[b]azepin-2(3H)-one 338238 3-(1-hexyl-trans-4,5-dimethyl-2-alpha-propylpiperidin-4-yl)phenol 338247 3-(5-methoxyindole-3-yl)-4-(3,4,5-trimethoxyphenyl)-1H-pyrrole-2,5-dione 338253 2-(2-chlorophenyl)-3-(4-chlorophenyl)-5-isopropyl-6-(2,2,2-trifluoroethyl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one 338254 2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-(2,2,2-trifluoroethyl)-2H-pyrazolo[3,4-c]pyridin-7(6H)-one 338260 N-((2-(2-cyclopropoxy-5-(trifluoromethoxy)benzylamino)-1-(4-fluorophenyl)-8-aza-bicyclo[3.2.1]octan-6-yl)methyl)benzenesulfonamide 338311 3-{(1R,2R)-2-[(dimethylamino)methyl]-1-hydroxycyclohexyl}phenol 338326 SID29217699 338332 phosphoric acid mono-((R)-2-octanoylamino-2-octylcarbamoyl-ethyl) ester 338333 thiophosphoric acid (S)-2-octanoylamino-2-octylcarbamoyl-ethyl ester 338334 (1R,2R)-2-{[bis(²Hƒ)methylamino]methyl}-1-[3-(²Hƒ)methoxyphenyl]cyclohexan-1-ol 338338 (S)-O-2,3-bis(octyloxy)propyl O,O-dihydrogen phosphorothioate 338345 nonanoic acid (S)-2-nonanoyloxy-3-phosphonooxy-propyl ester 338346 phosphoric acid mono-((S)-2-octanoylamino-2-octylcarbamoyl-ethyl) ester 338347 octanoic acid (R)-2-octanoyloxy-3-thiophosphonooxy-propyl ester 338354 (S)-1-(1H-pyrrolo[3,2-h]isoquinolin-1-yl)propan-2-amine 338355 (S)-N-(naphthalen-2-ylmethyl)-1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-amine 338363 (S)-1-(1H-pyrrolo[2,3-f]isoquinolin-1-yl)propan-2-amine 338364 (S)-N-(benzo[d][1,3]dioxol-5-ylmethyl)-1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-amine 338368 8-(2-chlorophenyl)-9-(4-chlorophenyl)-1-(2,2,2-trifluoroethyl)-4,9-dihydro-1H-purin-6(5H)-one 338384 3-(1-heptyl-trans-4,5-dimethyl-2-alpha-propylpiperidin-4-yl)phenol 338404 5-(2-(2-cyclopropoxy-5-(trifluoromethoxy)benzylamino)-1-phenyl-8-aza-bicyclo[3.2.1]octan-6-yl)-2H-1,2,4-triazol-3(4H)-one 338410 2-(2-cyclopropoxy-5-(trifluoromethoxy)benzylamino)-1-(4-fluorophenyl)-N-(methylsulfonyl)-8-aza-bicyclo[3.2.1]octane-6-carboxamide 338412 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-6-methoxy-4,5-dihydro-1H-benzo[b]azepin-2(3H)-one 338413 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)quinolin-2(1H)-one 338415 N-(2-cyclopropoxy-5-(trifluoromethoxy)benzyl)-1-phenyl-8-aza-bicyclo[3.2.1]octan-2-amine 338416 3-(1-Methylindole-3-yl)-4-(3,4,5-trimethoxyphenyl)-1H-pyrrole-2,5-dione 338421 N-(2-cyclopropoxy-5-(trifluoromethoxy)benzyl)-1-phenyl-6-(1H-tetrazol-5-yl)-8-aza-bicyclo[3.2.1]octan-2-amine 338423 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)quinoline-2,4(1H,3H)-dione 338428 5,6,7-trimethoxy-8-methyl-1,2,3,8-tetrahydro-benzo[a]pyrrolo-[3,4-c]carbazol-1,3-dione 338430 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-4,5-dihydro-1H-benzo[b]azepin-2(3H)-one 338431 5-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-2,3-dihydrobenzo[b][1,4]thiazepin-4(5H)-one 338444 (2-methyl-benzyl)-((S)-1-methyl-2-pyrrolo[2,3-f]quinolin-1-yl-ethyl)-amine 338452 2-(2-chlorophenyl)-3-(4-chlorophenyl)-5-methyl-6-(2,2,2-trifluoroethyl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one 338453 2-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-1,2-dihydroisoquinolin-3(4H)-one 338459 2-(2-chlorophenyl)-3-(4-chlorophenyl)-5-ethyl-6-(2,2,2-trifluoroethyl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one 338472 3-(2-chlorophenyl)-2-(4-chlorophenyl)-6-cyclohexyl-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one 338473 3-(2-chlorophenyl)-2-(4-chlorophenyl)-6-(2,2,2-trifluoroethyl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one 338477 3-(1H-Indol-3-yl)-4-(3,4,5-trimethoxyphenyl)-1Hpyrrole-2,5-dione 338478 3-(1H-pyrrole-3-yl)-4-(3,4,5-trimethoxyphenyl)-1H-pyrrole-2,5-dione 338482 (S)-N-(2-chlorobenzyl)-1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-amine 338502 2-(2-cyclopropoxy-5-(trifluoromethoxy)benzylamino)-1-(4-fluorophenyl)-N-(phenylsulfonyl)-8-aza-bicyclo[3.2.1]octane-6-carboxamide 338504 (S)-N-benzyl-1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-amine 338517 N-(2-chloro-5-(trifluoromethoxy)benzyl)-1-phenyl-8-aza-bicyclo[3.2.1]octan-2-amine 338536 octanoic acid (S)-2-octanoyloxy-3-phosphonooxy-propyl ester 338537 octanoic acid (R)-2-octanoyloxy-3-phosphonooxy-propyl ester 338540 3-(2-chlorophenyl)-N-(2-((2-(dimethylamino)ethyl)(methyl)amino)-4-methylquinolin-6-yl)acrylamide 338552 thiophosphoric acid (R)-2-octanoylamino-2-octylcarbamoyl-ethyl ester 338603 N-[4-[(3-bromophenyl)amino]-6-quinazolinyl]-2-propynamide 338610 (S)-1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-amine 338644 (2-(2-cyclopropoxy-5-(trifluoromethoxy)benzylamino)-1-phenyl-8-aza-bicyclo[3.2.1]octan-6-yl)methanol 338652 (2S,3S,4R,5R)-5-[2-dimethylamino-6-(3-iodo-benzylamino)-purin-9-yl]-3,4-dihydroxy-tetrahydrofuran-2-carboxylic acid dimethylamide 338674 2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-(2,2-difluoroethyl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one 338675 5-(3-phenoxybenzylthio)-2-aminothiazolo[4,5-d]pyrimidin-7-ol 338683 5-(2,3-difluorobenzylthio)-2-aminothiazolo[4,5-d]pyrimidin-7-ol 338695 3-(7-((R)-((2S,5R)-4-benzyl-2,5-dimethylpiperazin-1-yl)(3-fluorophenyl)methyl)-3,4-dihydroisoquinolin-2(1H)-yl)-3-oxopropanoic acid 338703 [2-chloro-4-(3-methyl-pyrazol-1-yl)-phenyl]-(5,11-dihydro-benzo[b]pyrido[2,3-e][1,4]diazepin-6-yl)-methanone 338714 2-(5-((R)-((2S,5R)-4-benzyl-2,5-dimethylpiperazin-1-yl)(3-hydroxyphenyl)methyl)isoindolin-2-yl)acetic acid 338715 (2S,3S,4R,5R)-5-(6-(3-iodobenzylamino)-2-chloro-9H-purin-9-yl)-3,4-dihydroxy-N,N-dimethyl-tetrahydrofuran-2-carboxamide 338721 (S)-2-(2-amino-5-(benzylthio)thiazolo[4,5-d]pyrimidin-7-ylamino)butan-1-ol 338729 2-(7-((R)-((2S,5R)-4-benzyl-2,5-dimethylpiperazin-1-yl)(3-methoxyphenyl)methyl)-3,4-dihydroisoquinolin-2(1H)-yl)acetic acid 338733 2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-cyclohexyl-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one 338734 2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-(2-fluoroethyl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one 338737 5-(benzylthio)thiazolo[4,5-d]pyrimidine-2,7-diamine 338744 (R)-2-(2-amino-5-(benzylthio)thiazolo[4,5-d]pyrimidin-7-ylamino)butan-1-ol 338747 3-(7-((R)-((2S,5R)-4-benzyl-2,5-dimethylpiperazin-1-yl)(3-hydroxyphenyl)methyl)-3,4-dihydroisoquinolin-2(1H)-yl)-3-oxopropanoic acid 338755 N-[4-[(3-Chloro-4-fluorophenyl)amino]-6-quinazolinyl]-4-hydroxy-2-butynamide 338756 N-[4-[(3-chloro-4-fluorophenyl)amino]-6-quinazolinyl]-4-(diethylamino)-2-butynamide 338763 N-[4-[(3-chloro-4-fluorophenyl)amino]pyrido[3,4-d]pyrimidin-6-yl]-2-heptynamide 338764 N-[4-[(3-chloro-4-fluorophenyl)amino]pyrido[3,4-d]pyrimidin-6-yl]-4-(diethylamino)-2-butynamide 338778 (2S,3S,4R,5R)-5-(6-(3-iodobenzylamino)-2-chloro-9H-purin-9-yl)-3,4-dihydroxy-N,N-dimethyl-tetrahydrothiophene-2-carboxamide 338791 2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-isopropyl-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one 338841 (5,11-dihydro-benzo[b]pyrido[2,3-e][1,4]diazepin-6-yl)-[2-fluoro-4-(3-methyl-pyrazol-1-yl)-phenyl]-methanone 338855 N-(2-(1,4-diazepan-1-yl)-4-methylquinolin-6-yl)-2-(4-(trifluoromethoxy)phenoxy)acetamide 338867 2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-ethyl-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one 338909 2-amino-5-(pentylthio)thiazolo[4,5-d]pyrimidin-7-ol 338918 2-amino-5-(benzylthio)thiazolo[4,5-d]pyrimidin-7-ol 338919 5-(pentylthio)thiazolo[4,5-d]pyrimidin-7-ol 338926 (5,11-dihydro-benzo[b]pyrido[2,3-e][1,4]diazepin-6-yl)-[4-(3-methyl-pyrazol-1-yl)-2-trifluoromethyl-phenyl]-methanone 338958 2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-(piperidin-1-yl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one 338959 2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-(pentan-3-yl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one 338960 3-(7-((R)-((2S,5R)-4-benzyl-2,5-dimethylpiperazin-1-yl)(3-fluorophenyl)methyl)-3,4-dihydroisoquinolin-2(1H)-yl)propanoic acid 338961 N-(2-((2-(dimethylamino)ethyl)(methyl)amino)-4-methylquinolin-6-yl)-3-p-tolylacrylamide 338984 N-[4-[(3-chloro-4-fluorophenyl)amino]-6-quinazolinyl]-4-(dibutylamino)-2-butynamide 338985 N-[4-[(3-chloro-4-fluorophenyl)amino]-6-quinazolinyl]-4-(4-morpholinyl)-2-butynamide 338996 N-[4-[(3-chloro-4-fluorophenyl)amino]-6-quinazolinyl]-5-(4-diethylamino)-2-pentynamide 338997 N-[4-[(3-chloro-4-fluorophenyl)amino]pyrido[3,4-d]pyrimidin-6-yl]-4-(dibutylamino)-2-butynamide 339002 3-(5-((R)-((2S,5R)-4-benzyl-2,5-dimethylpiperazin-1-yl)(3-methoxyphenyl)methyl)isoindolin-2-yl)propanoic acid 339003 1-(3-(2,6-dibromo-4-(piperidin-1-ylmethyl)phenoxy)propyl)piperidine 339004 N-[4-[(3-chloro-4-fluorophenyl)amino]pyrido[3,4-d]pyrimidin-6-yl]-4-(4-morpholinyl)-2-butynamide 339007 2-(7-((R)-((2S,5R)-4-benzyl-2,5-dimethylpiperazin-1-yl)(3-hydroxyphenyl)methyl)-3,4-dihydroisoquinolin-2(1H)-yl)acetic acid 339008 (S)-2-(5-(3-phenoxybenzylthio)-2-aminothiazolo[4,5-d]pyrimidin-7-ylamino)butan-1-ol 339009 3-(5-((R)-((2S,5R)-4-benzyl-2,5-dimethylpiperazin-1-yl)(3-hydroxyphenyl)methyl)isoindolin-2-yl)propanoic acid 339015 3-(5-((R)-((2S,5R)-4-benzyl-2,5-dimethylpiperazin-1-yl)(3-fluorophenyl)methyl)isoindolin-2-yl)propanoic acid 339022 2-(2-amino-5-(pentylthio)thiazolo[4,5-d]pyrimidin-7-ylamino)ethanol 339023 3-(7-((R)-((2S,5R)-4-benzyl-2,5-dimethylpiperazin-1-yl)(3-methoxyphenyl)methyl)-3,4-dihydroisoquinolin-2(1H)-yl)propanoic acid 339030 N-(4-methyl-2-(4-methyl-1,4-diazepan-1-yl)quinolin-6-yl)-2-(4-(trifluoromethoxy)phenoxy)acetamide 339031 N-(2-(4-(2-hydroxyethyl)piperazin-1-yl)-4-methylquinolin-6-yl)-2-(4-(trifluoromethoxy)phenoxy)acetamide 339038 2-(4-chlorophenoxy)-N-(2-((2-(dimethylamino)ethyl)(methyl)amino)-4-methylquinolin-6-yl)acetamide 339066 N-[4-[(3-chloro-4-fluorophenyl)amino]-6-quinazolinyl]-4-(bis-(1-methylethyl)amino)-2-butynamide 339072 N-[4-[(3-chloro-4-fluorophenyl)amino]-6-quinazolinyl]-5-(4-morpholinyl)-2-pentynamide 339073 aplysamine 339074 3-(2,6-dibromo-4-((dimethylamino)methyl)phenoxy)-N,N-dimethylpropan-1-amine 339075 3-(4-((dimethylamino)methyl)phenoxy)-N,N-dimethylpropan-1-amine 339076 N-[4-[(3-chloro-4-fluorophenyl)amino]pyrido[3,4-d]pyrimidin-6-yl]-4-(bis(1-methylethyl)amino)-2-butynamide 339081 3-(5-((S)-((2S,5R)-4-benzyl-2,5-dimethylpiperazin-1-yl)(phenyl)methyl)isoindolin-2-yl)propanoic acid 339082 2-(5-((R)-((2S,5R)-4-benzyl-2,5-dimethylpiperazin-1-yl)(3-hydroxyphenyl)methyl)isoindoline-2-carbonyl)benzoic acid 339086 N,N-dimethyl-3-(4-(piperidin-1-ylmethyl)phenoxy)propan-1-amine 339090 3-(7-((R)-((2S,5R)-4-benzyl-2,5-dimethylpiperazin-1-yl)(3-hydroxyphenyl)methyl)-3,4-dihydroisoquinolin-2(1H)-yl)propanoic acid 339113 [2-chloro-4-(5-methyl-pyrazol-1-yl)-phenyl]-(5,11-dihydro-benzo[b]pyrido[2,3-e][1,4]diazepin-6-yl)-methanone 339120 (5,11-dihydro-benzo[b]pyrido[2,3-e][1,4]diazepin-6-yl)-[4-(5-methyl-pyrazol-1-yl)-2-trifluoromethyl-phenyl]-methanone 339150 2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-(2,2-difluoropropyl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one 339153 2-(5-(3-phenoxybenzylthio)-2-aminothiazolo[4,5-d]pyrimidin-7-ylamino)-2-methylpropan-1-ol 339154 (R)-2-(5-(2,3-difluorobenzylthio)-2-aminothiazolo[4,5-d]pyrimidin-7-ylamino)butan-1-ol 339157 2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-(3,3,3-trifluoropropyl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one 339158 2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-propyl-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one 339162 2-(5-(2,3-difluorobenzylthio)-2-aminothiazolo[4,5-d]pyrimidin-7-ylamino)-2-methylpropan-1-ol 339181 [2-bromo-4-(3-methyl-pyrazol-1-yl)-phenyl]-(5,11-dihydro-benzo[b]pyrido[2,3-e][1,4]diazepin-6-yl)-methanone 339202 (R)-2-(5-(3-phenoxybenzylthio)-2-aminothiazolo[4,5-d]pyrimidin-7-ylamino)butan-1-ol 339203 2-(7-((R)-((2S,5R)-4-benzyl-2,5-dimethylpiperazin-1-yl)(3-hydroxyphenyl)methyl)-3,4-dihydroisoquinolin-2(1H)-yl)-2-oxoacetic acid 339224 6-benzyl-2-(2-chlorophenyl)-3-(4-chlorophenyl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one 339225 2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-(2,2,2-trifluoroethyl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one 339236 des-bromoaplysamine-1 339243 N-[4-[(3-bromophenyl)amino]pyrido[3,4-d]pyrimidin-6-yl]-2-propynamide 339244 2-(4-(2-(dimethylamino)ethoxy)phenyl)-N,N-dimethylethanamine 339245 N-[4-[(3-chloro-4-fluorophenyl)amino]pyrido[3,4-d]pyrimidin-6-yl]-5-(4-morpholinyl)-2-pentynamide 339254 N-[4-[(3-bromo-4-fluorophenyl)amino]pyrido[3,4-d]pyrimidin-6-yl]-5-(4-morpholinyl)-2-pentynamide 339255 N-[4-[(3-chloro-4-fluorophenyl)amino]pyrido[3,4-d]pyrimidin-6-yl]-5-(1-piperidinyl)-2-pentynamide 339289 [2-chloro-4-(3-methyl-pyrazol-1-yl)-phenyl]-(11-methyl-5,11-dihydro-benzo[b]pyrido[2,3-e][1,4]diazepin-6-yl)-methanone 339290 N-(2-(3-(dimethylamino)-2,2-dimethylpropylamino)-4-methylquinolin-6-yl)-2-(4-(trifluoromethoxy)phenoxy)acetamide 339301 2-((5-((R)-((2S,5R)-4-benzyl-2,5-dimethylpiperazin-1-yl)(3-hydroxyphenyl)methyl)isoindolin-2-yl)methyl)benzoic acid 339310 2-(5-((R)-((2S,5R)-4-benzyl-2,5-dimethylpiperazin-1-yl)(3-methoxyphenyl)methyl)isoindolin-2-yl)acetic acid 339324 N-(2-(1-benzylpiperidin-4-ylamino)-4-methylquinolin-6-yl)-2-(4-(trifluoromethoxy)phenoxy)acetamide 339325 (R)-N-(4-methyl-2-(3-methylpiperazin-1-yl)quinolin-6-yl)-2-(4-(trifluoromethoxy)phenoxy)acetamide 339326 2-(4-((R)-((2S,5R)-4-benzyl-2,5-dimethylpiperazin-1-yl)(3-hydroxyphenyl)methyl)phenyl)acetic acid 339330 3-(4-((R)-((2S,5R)-4-benzyl-2,5-dimethylpiperazin-1-yl)(3-hydroxyphenyl)methyl)phenyl)propanoic acid 339344 N-(2-((2-(dimethylamino)ethyl)(methyl)amino)-4-methylquinolin-6-yl)-3-(4-(trifluoromethoxy)phenyl)propanamide 339346 4'-[(R)-((2S,5R)-4-benzyl-2,5-dimethyl-piperazin-1-yl)-(3-hydroxy-phenyl)-methyl]-biphenyl-2-carboxylic acid 339353 (S)-N-(4-methyl-2-(3-methylpiperazin-1-yl)quinolin-6-yl)-2-(4-(trifluoromethoxy)phenoxy)acetamide 339354 3-(5-((R)-((2S,5R)-4-benzyl-2,5-dimethylpiperazin-1-yl)(3-hydroxyphenyl)methyl)isoindoline-2-carbonyl)benzoic acid 339355 4-(5-((R)-((2S,5R)-4-benzyl-2,5-dimethylpiperazin-1-yl)(3-methoxyphenyl)methyl)isoindoline-2-carbonyl)benzoic acid 339411 (S)-4-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)methyl)-4-phenylimidazolidin-2-one 339414 4-((1H-imidazol-4-yl)methyl)-1-(3-(4-(cyclohexyloxy)phenoxy)propyl)piperidine 339415 4-((1H-imidazol-4-yl)methyl)-1-(3-(3-(cyclohexyloxy)phenoxy)propyl)piperidine 339419 (R)-4-(((S)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)methyl)-4-phenylimidazolidin-2-one 339422 1-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propoxy)phenyl)piperidine 339423 (4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propoxy)phenyl)(piperazin-1-yl)methanone 339429 (R)-(2-((1H-indol-3-yl)methyl)-4-(2-(2-morpholinoethoxyimino)-2-phenylethyl)piperazin-1-yl)(3,5-bis(trifluoromethyl)phenyl)methanone 339430 (R)-(2-((1H-indol-3-yl)methyl)-4-(2-(2-(4-methylpiperazin-1-yl)ethoxyimino)propyl)piperazin-1-yl)(3,5-bis(trifluoromethyl)phenyl)methanone 339431 (R)-(2-((1H-indol-3-yl)methyl)-4-(2-(2-thiomorpholinoethoxyimino)propyl)piperazin-1-yl)(3,5-bis(trifluoromethyl)phenyl)methanone 339434 (R)-3-((1H-indol-3-yl)methyl)-N-(2-(2-methoxybenzylamino)ethyl)-4-(3,5-bis(trifluoromethyl)benzoyl)piperazine-1-carboxamide 339435 (R)-(2-((1H-indol-3-yl)methyl)-4-(2-(3-morpholinopropoxyimino)-2-phenylethyl)piperazin-1-yl)(3,5-bis(trifluoromethyl)phenyl)methanone 339436 (R)-(2-((1H-indol-3-yl)methyl)-4-(3-(2-morpholinoethoxyimino)-3-phenylpropyl)piperazin-1-yl)(3,5-bis(trifluoromethyl)phenyl)methanone 339437 1-[(R)-4-(3,5-bis-trifluoromethyl-benzoyl)-3-(1H-indol-3-ylmethyl)-piperazin-1-yl]-propan-2-one O-[2-(1,1-dioxo-thiomorpholin-4-yl)-ethyl]-oxime 339444 1-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-3-(4-(piperidin-1-ylmethyl)phenoxy)propan-1-one 339445 1-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-3-(4-(piperidin-1-ylmethyl)phenyl)propan-1-one 339449 (R)-(2-((1H-indol-3-yl)methyl)-4-(2-(pyridin-2-ylmethoxyimino)propyl)piperazin-1-yl)(3,5-bis(trifluoromethyl)phenyl)methanone 339468 [2-chloro-4-(1-methyl-1H-pyrazol-3-yl)-phenyl]-(5,11-dihydro-benzo[b]pyrido[2,3-e][1,4]diazepin-6-yl)-methanone 339470 (R)-4-((3,5-bis(trifluoromethyl)benzyloxy)methyl)-4-phenylimidazolidin-2-one 339471 N-[4-[(3-chloro-4-fluorophenyl)amino]pyrido[3,4-d]pyrimidin-6-yl]-2-butynamide 339472 N,N-dimethyl-2-(4-(2-(piperidin-1-yl)ethoxy)phenyl)ethanamine 339473 N-[4-[(3-chloro-4-fluorophenyl)amino]pyrido[3,4-d]pyrimidin-6-yl]-2-hexynamide 339479 4-((3,5-bis(trifluoromethyl)benzyloxy)methyl)-4-(4-fluorophenyl)imidazolidin-2-one 339480 (S)-4-((3,5-bis(trifluoromethyl)benzyloxy)methyl)-4-(4-fluorophenyl)imidazolidin-2-one 339481 dimethyl-{2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-ethyl}-amine 339482 N-[4-[(3-chloro-4-fluorophenyl)amino]pyrido[3,4-d]pyrimidin-6-yl]-5-(4-methyl-1-piperazinyl)-2-pentynamide 339486 N-(2-((2-(dimethylamino)ethyl)(methyl)amino)-4-methylquinolin-6-yl)benzo[b]thiophene-2-carboxamide 339488 N-[4-[(3-bromo-4-fluorophenyl)amino]pyrido[3,4-d]pyrimidin-6-yl]-5-(4-methyl-1-piperazinyl)-2-pentynamide 339489 3-(4-((4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)methyl)phenoxy)-N,N-dimethylpropan-1-amine 339493 (R)-4-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)methyl)-1-methyl-4-phenylimidazolidin-2-one 339494 (R)-4-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)methyl)-1-ethyl-4-phenylimidazolidin-2-one 339498 4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propoxy)-N-cyclohexylbenzenamine 339499 N-(4-methyl-2-(2-morpholinoethylamino)quinolin-6-yl)-2-(4-(trifluoromethoxy)phenoxy)acetamide 339500 N-(4-methyl-2-(2-(piperidin-1-yl)ethylamino)quinolin-6-yl)-2-(4-(trifluoromethoxy)phenoxy)acetamide 339514 1-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-3-(4-(piperazine-1-carbonyl)phenoxy)propan-1-one 339517 N-(2-((2-(dimethylamino)ethyl)(methyl)amino)-4-methylquinolin-6-yl)-4-(trifluoromethoxy)benzamide 339518 2-(2,4-dichlorophenylamino)-N-(2-((2-(dimethylamino)ethyl)(methyl)amino)-4-methylquinolin-6-yl)acetamide 339521 5-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propoxy)-2-(piperidin-1-ylmethyl)pyridine 339522 (6-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propoxy)pyridin-3-yl)(piperidin-1-yl)methanone 339524 N-(2-((3S,5R)-3,5-dimethylpiperazin-1-yl)-4-methylquinolin-6-yl)-2-(4-(trifluoromethoxy)phenoxy)acetamide 339535 3-(7-((R)-((2S,5R)-4-benzyl-2,5-dimethylpiperazin-1-yl)(3-methoxyphenyl)methyl)-3,4-dihydroisoquinolin-2(1H)-yl)-3-oxopropanoic acid 339537 N-(2-((2-(dimethylamino)ethyl)(methyl)amino)-4-methylquinolin-6-yl)-6-phenoxynicotinamide 339538 4'-trifluoromethyl-biphenyl-4-carboxylic acid {2-[(2-dimethylamino-ethyl)-methyl-amino]-4-methyl-quinolin-6-yl}-amide 339544 [(R)-4-(3,5-bis-trifluoromethyl-benzoyl)-3-(1H-indol-3-ylmethyl)-piperazin-1-yl]-acetaldehyde O-(2-morpholin-4-yl-ethyl)-oxime 339545 ((R)-2-((1H-indol-3-yl)methyl)-4-((Z)-2-(2-morpholinopropoxyimino)propyl)piperazin-1-yl)(3,5-bis(trifluoromethyl)phenyl)methanone 339557 N-(2-((2-(dimethylamino)ethyl)(methyl)amino)-4-methylquinolin-6-yl)cinnamamide 339559 biphenyl-4-carboxylic acid {2-[(2-dimethylamino-ethyl)-methyl-amino]-4-methyl-quinolin-6-yl}-amide 339560 1-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propoxy)benzyl)-4,4-difluoropiperidine 339566 (E)-N-(2-((2-(dimethylamino)ethyl)(methyl)amino)-4-methylquinolin-6-yl)-2-methyl-3-phenylacrylamide 339570 [(R)-4-(3,5-bis-trifluoromethyl-benzoyl)-3-(1H-indol-3-ylmethyl)-piperazin-1-yl]-acetaldehyde O-(3-morpholin-4-yl-propyl)-oxime 339582 3-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propyl)phenoxy)-N,N-dimethylpropan-1-amine 339586 (S)-N-butyl-3-(2-(naphthalen-2-yl)propanamido)pyrrolo[3,4-c]pyrazole-5(1H,4H,6H)-carboxamide 339590 6-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propoxy)quinoline 339591 5-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propoxy)phenyl)pyrimidin-2-amine 339597 4-(4-chlorophenyl)-N-(2-((2-(dimethylamino)ethyl)(methyl)amino)-4-methylquinolin-6-yl)cyclohexanecarboxamide 339598 2-biphenyl-4-yl-N-{2-[(2-dimethylamino-ethyl)-methyl-amino]-4-methyl-quinolin-6-yl}-acetamide 339599 (4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propoxy)phenyl)(piperidin-1-yl)methanone 339607 N-(2-((2-(dimethylamino)ethyl)(methyl)amino)-4-methylquinolin-6-yl)-2-(5-methyl-2-phenyloxazol-4-yl)acetamide 339608 1-(3-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propoxy)benzyl)piperidine 339615 (R)-(2-((1H-indol-3-yl)methyl)-4-(3-(2-morpholinoethoxyimino)butyl)piperazin-1-yl)(3,5-bis(trifluoromethyl)phenyl)methanone 339616 (R)-(2-((1H-indol-3-yl)methyl)-4-(3-(3-morpholinopropoxyimino)butyl)piperazin-1-yl)(3,5-bis(trifluoromethyl)phenyl)methanone 339618 N-(2-(2-(diethylamino)ethylamino)-4-methylquinolin-6-yl)-2-(4-(trifluoromethoxy)phenoxy)acetamide 339619 N-(2-(2-(diisopropylamino)ethylamino)-4-methylquinolin-6-yl)-2-(4-(trifluoromethoxy)phenoxy)acetamide 339620 1-(4-(4-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)butoxy)benzyl)piperidine 339621 1-(4-(2-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)ethoxy)benzyl)piperidine 339624 (R)-(2-((1H-indol-3-yl)methyl)-4-(2-(methoxyimino)propyl)piperazin-1-yl)(3,5-bis(trifluoromethyl)phenyl)methanone 339625 1-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propoxy)benzyl)piperidine-4-carboxamide 339626 1-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propoxy)benzyl)-4-(piperidin-1-yl)piperidine 339627 1-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propoxy)phenethyl)piperidine 339628 1-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propoxy)phenyl)piperazine 339632 (R)-(2-((1H-indol-3-yl)methyl)-4-(2-(2-aminoethoxyimino)propyl)piperazin-1-yl)(3,5-bis(trifluoromethyl)phenyl)methanone 339633 4-((3,5-bis(trifluoromethyl)benzyloxy)methyl)-4-(4-fluorophenyl)-1-(piperidin-4-yl)imidazolidin-2-one 339634 4-((3,5-bis(trifluoromethyl)benzyloxy)methyl)-4-(4-fluorophenyl)-1-(1-methylpiperidin-4-yl)imidazolidin-2-one 339635 ((R)-2-((1H-indol-3-yl)methyl)-4-((5-(morpholinomethyl)-4,5-dihydroisoxazol-3-yl)methyl)piperazin-1-yl)(3,5-bis(trifluoromethyl)phenyl)methanone 339636 5-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propoxy)phenyl)pyrimidine 339637 2-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propoxy)phenyl)pyrimidine 339641 (R)-(2-((1H-indol-3-yl)methyl)-4-(2-(2-(methylamino)ethoxyimino)propyl)piperazin-1-yl)(3,5-bis(trifluoromethyl)phenyl)methanone 339642 (R)-(2-((1H-indol-3-yl)methyl)-4-(4-(2-morpholinoethoxyimino)pentyl)piperazin-1-yl)(3,5-bis(trifluoromethyl)phenyl)methanone 339643 (R)-(2-((1H-indol-3-yl)methyl)-4-(2-(2-(dimethylamino)ethoxyimino)propyl)piperazin-1-yl)(3,5-bis(trifluoromethyl)phenyl)methanone 339644 (R)-(2-((1H-indol-3-yl)methyl)-4-(2-(2-methyl-2-morpholinopropoxyimino)propyl)piperazin-1-yl)(3,5-bis(trifluoromethyl)phenyl)methanone 339647 (R)-(2-((1H-indol-3-yl)methyl)-4-((5-(morpholinomethyl)isoxazol-3-yl)methyl)piperazin-1-yl)(3,5-bis(trifluoromethyl)phenyl)methanone 339649 3-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propoxy)phenyl)pyridine 339650 4-((1H-imidazol-4-yl)methyl)-N-(thiazol-2-yl)piperidine-1-carboxamide 339658 (R)-4-((3,5-bis(trifluoromethyl)benzyloxy)methyl)-4-(4-fluorophenyl)imidazolidin-2-one 339659 3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(4-(piperidin-1-ylmethyl)phenyl)propanamide 339662 3-[2-(4-pyrrolidin-1-yl-phenyl)-acetylamino]-4,6-dihydro-1H-pyrrolo[3,4-c]pyrazole-5-carboxylic acid butylamide 339664 (R)-4-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)methyl)-4-phenylimidazolidin-2-one 339665 2-((R)-4-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)methyl)-4-(4-fluorophenyl)-2-oxoimidazolidin-1-yl)acetamide 339682 N-(2-((2-(dimethylamino)ethyl)(methyl)amino)-4-methylquinolin-6-yl)-4-phenoxybenzamide 339692 (R)-(2-((1H-indol-3-yl)methyl)-4-(2-(2-morpholinoethoxyimino)propyl)piperazin-1-yl)(3,5-bis(trifluoromethyl)phenyl)methanone 339693 (R)-(2-((1H-indol-3-yl)methyl)-4-(2-(3-morpholinopropoxyimino)propyl)piperazin-1-yl)(3,5-bis(trifluoromethyl)phenyl)methanone 339700 N-(2-((2-(dimethylamino)ethyl)(methyl)amino)-4-methylquinolin-6-yl)-3-(4,5-diphenyloxazol-2-yl)propanamide 339707 4-((3,5-bis(trifluoromethyl)benzyloxy)methyl)-4-(4-fluorophenyl)-1-(tetrahydro-2H-pyran-4-yl)imidazolidin-2-one 339708 1-(4-bromobenzyl)-3-(2-((2-(dimethylamino)ethyl)(methyl)amino)-4-methylquinolin-6-yl)urea 339709 (R)-4-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)methyl)-1-isopropyl-4-phenylimidazolidin-2-one 339715 4-((3,5-bis(trifluoromethyl)benzyloxy)methyl)-4-(4-fluorophenyl)-1-(2-(pyrrolidin-1-yl)ethyl)imidazolidin-2-one 339716 (R)-4-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)methyl)-4-(4-fluorophenyl)-1-methylimidazolidin-2-one 339717 (R)-4-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)methyl)-4-(4-fluorophenyl)imidazolidin-2-one 339718 1-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propoxy)benzyl)piperidine 339722 (R)-4-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)methyl)-1-ethyl-4-(4-fluorophenyl)imidazolidin-2-one 339723 N-(2-(2-(dimethylamino)ethylamino)-4-methylquinolin-6-yl)-2-(4-(trifluoromethoxy)phenoxy)acetamide 339724 rac-N-(2-(3-(dimethylamino)pyrrolidin-1-yl)-4-methylquinolin-6-yl)-2-(4-(trifluoromethoxy)phenoxy)acetamide 339725 4-((1H-imidazol-4-yl)methyl)-N-(pyrimidin-2-yl)piperidine-1-carboxamide 339733 N-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propoxy)benzyl)-N-ethylethanamine 339737 N-(2-((2-(dimethylamino)ethyl)(methyl)amino)-4-methylquinolin-6-yl)-2-(4-(trifluoromethoxy)phenoxy)acetamide 339738 1-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)propoxy)benzyl)piperidin-2-one 339749 3-(3,5-bis-trifluoromethyl-phenyl)-1-[4-(2-oxa-8-aza-spiro[4.5]dec-8-yl)-1-phenyl-cyclohexyl]-piperidin-2-one 339750 4-((1r,4r)-4-(3-(3,5-bis(trifluoromethyl)phenyl)-2-oxopyrrolidin-1-yl)-4-phenylcyclohexyl)-1-phenylpiperazin-2-one 339789 3-(3,5-bis(trifluoromethyl)phenyl)-1-((1r,4r)-4-(dimethylamino)-1-phenylcyclohexyl)pyrrolidin-2-one 339839 (R)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-[4-cyclohexyl-4-(5,5-dimethyl-1,1-dioxo-1lambda*6*-isothiazolidin-2-ylmethyl)-piperidin-1-yl]-2-oxo-ethyl}-amide 339840 (R)-N-((R)-3-(4-chlorophenyl)-1-(4-cyclohexyl-4-((N-isopropylmethan-2-ylsulfonamido)methyl)piperidin-1-yl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 339845 2-(3,5-bis-trifluoromethyl-phenyl)-N-[4-(2-oxa-8-aza-spiro[4.5]dec-8-yl)-1-phenyl-cyclohexyl]-propionamide 339846 2-(3,5-bis(trifluoromethyl)phenyl)-N-((1r,4r)-4-(3-oxo-4-phenylpiperazin-1-yl)-1-phenylcyclohexyl)propanamide 339859 5-[[(3-pyridyl)amino]carbonyl]amino-8-methyl-2-(2-furyl)-pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine 339860 5-[[(2-pyridyl)amino]carbonyl]amino-8-methyl-2-(2-furyl)-pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine 339870 5-[[(2-methyl-thiophen-3-yl)amino]carbonyl]amino-8-methyl-2-(2-furyl)-pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine 339871 4-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,4]triazolo-[1,5-c]pyrimidin-5-yl)-ureido]-N-methylpyridinium iodide 339873 3-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,4]triazolo-[1,5-c]pyrimidin-5-yl)-ureido]-N-methylpyridinium iodide 339874 2-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,4]triazolo-[1,5-c]pyrimidin-5-yl)-ureido]-N-methylpyridinium iodide 339875 (R)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-[4-cyclohexyl-4-(1,1-dioxo-1lambda*6*-isothiazolidin-2-ylmethyl)-piperidin-1-yl]-2-oxo-ethyl}-amide 339880 3-(3,5-bis-trifluoromethyl-phenyl)-1-[4-(2-oxa-8-aza-spiro[4.5]dec-8-yl)-1-phenyl-cyclohexyl]-pyrrolidin-2-one 339881 3-(3,5-bis-trifluoromethyl-phenyl)-3-methoxy-1-[4-(2-oxa-8-aza-spiro[4.5]dec-8-yl)-1-phenyl-cyclohexyl]-pyrrolidin-2-one 339885 5-[[(5-methyl-thiophen-2-yl)amino]carbonyl]amino-8-methyl-2-(2-furyl)-pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine 339890 4-(2,6-dimethylmorpholino)-6-(ethylthio)-1-styryl-1H-pyrazolo[3,4-d]pyrimidine 339894 1-(2-bromo-2-phenylethyl)-N-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 339897 N-cyclopropyl-1-styryl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 339901 1-(2-bromo-2-phenylethyl)-N-isopropyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 339902 1-(2-bromo-2-phenylethyl)-N-butyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 339909 (R)-N-((R)-3-(4-chlorophenyl)-1-(4-cyclohexyl-4-((3-methyl-2-oxoimidazolidin-1-yl)methyl)piperidin-1-yl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 339910 (R)-N-((R)-3-(4-chlorophenyl)-1-(4-cyclohexyl-4-((2-oxooxazolidin-3-yl)methyl)piperidin-1-yl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 339923 1-(2-bromo-2-phenylethyl)-N-(2-ethoxyethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 339924 1-(2-bromo-2-phenylethyl)-4-(pyrrolidin-1-yl)-1H-pyrazolo[3,4-d]pyrimidine 339925 1-(2-bromo-2-phenylethyl)-4-(piperidin-1-yl)-1H-pyrazolo[3,4-d]pyrimidine 339961 2-(6-(4-(3-morpholinopropyl)piperazin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile 339962 2-(6-(4-(2-(pyrrolidin-1-yl)ethyl)piperazin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile 340010 2-(6-(1,4-diazepan-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile 340011 2-(6-(4-(2-methoxyethyl)piperazin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile 340016 2-(6-(4-(2-morpholinoethyl)piperazin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile 340048 (R)-N-((R)-3-(4-chlorophenyl)-1-(4-cyclohexyl-4-((2-oxoimidazolidin-1-yl)methyl)piperidin-1-yl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 340049 ethyl (1-((R)-3-(4-chlorophenyl)-2-((R)-1,2,3,4-tetrahydroisoquinoline-3-carboxamido)propanoyl)-4-cyclohexylpiperidin-4-yl)methyl(isopropyl)carbamate 340061 5-[[(2-furyl)amino]carbonyl]amino-8-methyl-2-(2-furyl)-pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine 340062 5-[[(3-furyl)amino]carbonyl]amino-8-methyl-2-(2-furyl)-pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine 340067 5-[[(benzofuran-2-yl)amino]carbonyl]amino-8-methyl-2-(2-furyl)-pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine 340079 N-cyclohexyl-1-styryl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 340084 N-benzyl-1-(2-bromo-2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 340088 N-benzyl-1-styryl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 340094 (R)-N-((R)-3-(4-chlorophenyl)-1-(4-cyclohexyl-4-(((S)-4-methyl-2-oxooxazolidin-3-yl)methyl)piperidin-1-yl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 340095 (R)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-[4-cyclohexyl-4-(5-oxo-6-oxa-4-aza-spiro[2.4]hept-4-ylmethyl)-piperidin-1-yl]-2-oxo-ethyl}-amide 340122 (R)-N-((R)-3-(4-chlorophenyl)-1-(4-cyclohexyl-4-((4,4-dimethyl-2-oxooxazolidin-3-yl)methyl)piperidin-1-yl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 340123 (R)-N-((R)-3-(4-chlorophenyl)-1-(4-cyclohexyl-4-(((R)-4-methyl-2-oxooxazolidin-3-yl)methyl)piperidin-1-yl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 340135 4-((1r,4r)-4-(3-(3,5-bis(trifluoromethyl)phenyl)-3-methyl-2-oxopyrrolidin-1-yl)-4-phenylcyclohexyl)-1-phenylpiperazin-2-one 340136 4-((1r,4r)-4-(3-(3,5-bis(trifluoromethyl)phenyl)-3-methyl-2-oxopyrrolidin-1-yl)-4-phenylcyclohexyl)-1-(2-chlorophenyl)piperazin-2-one 340143 4-((1r,4r)-4-(3-(3,5-bis(trifluoromethyl)phenyl)-2-oxopiperidin-1-yl)-4-phenylcyclohexyl)-1-phenylpiperazin-2-one 340179 5-[[(quinolin-2-yl)amino]carbonyl]amino-8-methyl-2-(2-furyl)-pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine 340184 3-(3,5-bis-trifluoromethyl-phenyl)-3-hydroxy-1-[4-(2-oxa-8-aza-spiro[4.5]dec-8-yl)-1-phenyl-cyclohexyl]-pyrrolidin-2-one 340185 3-(3,5-bis-trifluoromethyl-phenyl)-3-methyl-1-[4-(2-oxa-8-aza-spiro[4.5]dec-8-yl)-1-phenyl-cyclohexyl]-pyrrolidin-2-one 340190 2-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,4]triazolo-[1,5-c]pyrimidin-5-yl)-ureido]pyridinium N-oxide 340195 4-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,4]triazolo-[1,5-c]pyrimidin-5-yl)-ureido]pyridinium N-oxide 340196 3-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,4]triazolo-[1,5-c]pyrimidin-5-yl)-ureido]pyridinium N-oxide 340202 (rac)-2-(6-(3-aminopyrrolidin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile 340207 1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-2-(hex-1-ynyl)-9H-purin-6-yl)-3-(4-methoxyphenyl)urea 340217 1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-2-(2-phenylethynyl)-9H-purin-6-yl)-3-(4-methoxyphenyl)urea 340266 (2S,3S,4R,5R)-N-ethyl-3,4-dihydroxy-5-(6-(4-methoxybenzamido)-9H-purin-9-yl)-tetrahydrofuran-2-carboxamide 340267 (2S,3S,4R,5R)-5-(6-(2-chlorobenzamido)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 340282 2-(4-(benzylamino)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)-1-phenylethanol 340284 2-(4-(phenethylamino)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)-1-phenylethanol 340286 1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-6-yl)-3-(furan-2-ylmethyl)urea 340287 (2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-{3-[4-(pyridin-2-ylsulfamoyl)-phenyl]-ureido}-purin-9-yl)-tetrahydro-furan-2-carboxylic acid ethylamide 340311 c[Nle-Nle-D-Nal(2')-Arg-Trp-Glu]-NH2 340318 2-(pyrimidin-4-ylamino)thiazole-5-carbonitrile 340319 2-(6-(4-aminoazepan-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile 340321 2-(2-aminopyrimidin-4-ylamino)thiazole-5-carbonitrile 340322 2-(6-aminopyrimidin-4-ylamino)thiazole-5-carbonitrile 340323 2-(2-(4-acetylpiperazin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile 340325 2-(6-(4-acetylpiperazin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile 340332 (R)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-[4-cyclohexyl-4-(6-oxo-7-oxa-5-aza-spiro[3.4]oct-5-ylmethyl)-piperidin-1-yl]-2-oxo-ethyl}-amide 340333 2-(6-(piperazin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile 340334 2-(6-(4-methylpiperazin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile 340335 2-(6-(4-aminopiperidin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile 340338 7-Methoxy-2-oxo-8-pentyloxy-1,2-dihydroquinoline-3-carboxylic Acid [2-(3,4-dihydroxyphenyl)ethyl]amide 340339 7-Methoxy-2-oxo-8-pentyloxy-1,2-dihydroquinoline-3-carboxylic Acid 3,4-dihydroxybenzylamide 340354 c[Nle-Glu-D-Phe-Arg-Trp-Glu]-NH2 340355 c[Nle-Asp-D-Nal(2')-Arg-Trp-Glu]-NH2 340358 1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-2-(3-hydroxy-3-phenylprop-1-ynyl)-9H-purin-6-yl)-3-(4-methoxyphenyl)urea 340375 c[Nle-Pro-D-Phe-Arg-Trp-Glu]-NH2 340376 c[Nle-His-D-Nal(2')-Arg-Trp-Glu]-NH2 340377 c[Nle-Glu-D-Nal(2')-Arg-Trp-Glu]-NH2 340380 H-Tyr-D-Ala-Gly-Phe-NH-NH-(NMe)Phe-Asp-Lys(Cpac)-Trp-Ac 340384 c[Nle-Gln-D-Phe-Arg-Trp-Glu]-NH2 340385 c[Nle-Pro-D-Nal(2')-Arg-Trp-Glu]-NH2 340392 [5-amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]-[3-(3-piperidin-1-ylprop-1-ynyl)phenyl]methanone 340394 H-Tyr-D-Ala-Gly-Phe-NH-NH-(NMe)Phe-Asp-Nle-Trp-Ac 340395 [5-amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]-{3-[3-(4-methyl-piperazin-1-yl)prop-1-ynyl]phenyl}methanon 340396 [5-amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]-{3-[2-(1-hydroxycyclopentyl)ethyl]phenyl}methanone 340406 5-amino-1-(4-fluorophenyl)-4-[3-(2-hydroxyethyl)benzoyl]-pyrazole 340407 5-Amino-4-[3-(2-aminosulfonylethyl) benzoyl]-1-(4-fluorophenyl) 340414 1-(4-acetylphenyl)-3-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-6-yl)urea 340417 [5-amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]-[3-(2-methanesulfonylethyl)phenyl]methanone 340418 (5-amino-1-(3-fluorophenyl)-1H-pyrazol-4-yl)(phenyl)methanone 340419 5-amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]-[3-(3-morpholin-4-ylprop-1-ynyl)phenyl]methanone 340420 (2S,3S,4R,5R)-5-(6-benzamido-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 340421 1-benzyl-3-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-6-yl)urea 340431 (2S,3S,4R,5R)-5-(6-{bis[(4-nitrophenyl)carbamoyl]amino}-9H-purin-9-yl)-N-ethyl-3,4-dihydroxyoxolane-2-carboxamide 340433 [5-amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]-[3-(3-hydroxy-3-methyl-butyl)phenyl]methanone 340434 [5-amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]-[3-(1,2-dihydroxy-ethyl)phenyl]methanone 340435 (2S,3S,4R,5R)-3,4-Dihydroxy-5-{6-[3-(4-sulfamoyl-phenyl)-ureido]-purin-9-yl}-tetrahydro-furan-2-carboxylic acid ethylamide 340443 (2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-{3-[4-(5-methyl-isoxazol-3-ylsulfamoyl)-phenyl]-ureido}-purin-9-yl)-tetrahydro-furan-2-carboxylic acid ethylamide 340447 [5-amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]-[4-(3-morpholin-4-ylprop-1-ynyl)phenyl]methanone 340449 5-benzoyloxymethyl-5-hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone 340452 5-hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]-5-(3-isobutyl-5-methyl-hexanoyloxymethyl)tetrahydro-2-furanone 340456 5-benzoyloxymethyl-5-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone 340457 5-[(E)-3-(tert-butoxy)-3-oxo-1-propenyl]-5-hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone 340458 5-[(E)-3-(tert-butoxy)-3-oxo-1-propenyl]-5-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone 340462 c[Nle-Arg-D-Phe-Arg-Trp-Glu]-NH2 340463 (5-amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl)(phenyl)methanone 340473 7-Methoxy-2-oxo-8-pentyloxy-1,2-dihydroquinoline-3-carboxylic Acid [2-(4-nitrophenyl)ethyl]amide 340479 7-Methoxy-2-oxo-8-pentyloxy-1,2-dihydroquinoline-3-carboxylic acid[2-(4-chlorophenyl)ethyl]amide 340480 7-Methoxy-2-oxo-8-pentyloxy-1,2-dihydroquinoline-3-carboxylic Acid [2-(4-hydroxyphenyl)-ethyl]amide 340482 7-Methoxy-2-oxo-8-pentyloxy-1,2-dihydroquinoline-3-carboxylic Acid [2-(4-aminophenyl)ethyl]amide 340487 7-Methoxy-2-oxo-8-pentyloxy-1,2-dihydroquinoline-3-carboxylic acid(3-phenylpropyl)amide 340505 (2S,3S,4R,5R)-5-(6-{bis[(5-chloropyridin-2-yl)carbamoyl]amino}-9H-purin-9-yl)-N-ethyl-3,4-dihydroxyoxolane-2-carboxamide 340516 1-(2-chloro-9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-6-yl)-3-(3-chlorophenyl)urea 340525 1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-2-(5-phenylpent-1-ynyl)-9H-purin-6-yl)-3-(4-methoxyphenyl)urea 340561 [5-amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]-[4-(3-morpholin-4-ylpropyl)phenyl]methanone 340587 (5-amino-1-(2-fluorophenyl)-1H-pyrazol-4-yl)(phenyl)methanone 340597 (5-amino-1-(4-methoxyphenyl)-1H-pyrazol-4-yl)(phenyl)methanone 340598 [5-amino-1-(2-methoxyphenyl)-1H-pyrazol-4-yl]phenylmethanone 340606 5-amino-1-(4-fluorophenyl)-4-[3-(2-morpholin-4-ylethoxy)-benzoyl]pyrazole 340607 [5-amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]-[3-(3-morpholin-4-ylpropyl)phenyl]methanone 340608 H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-Nle-D-Trp-2-Adoc 340609 H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-Nle-D-Trp-H 340630 5-amino-4-[3-(2-aminoethyl)benzoyl]-1-(4-fluorophenyl)pyrazole 340638 7-(4-(2-butoxyethoxy)phenyl)-1-isobutyl-N-(4-((1-propyl-1H-imidazol-5-yl)methylsulfinyl)phenyl)-2,3-dihydro-1H-benzo[b]azepine-4-carboxamide 340644 2-Benzo[1,3]dioxol-5-yl-N-(7-methoxy-2-oxo-8-pentyloxy-1,2-dihydroquinolin-3-yl)acetamide 340645 7-Methoxy-2-oxo-8-pentyloxy-1,2-dihydroquinoline-3-carboxylic Acid [2-(1H-indol-3-yl)ethyl]amide 340653 c[Nle-Gln-D-Nal(2')-Arg-Trp-Glu]-NH2 340664 c[Nle-His-D-Phe-Arg-Trp-Glu]-NH2 340668 c[Nle-Arg-D-Nal(2')-Arg-Trp-Glu]-NH2 340673 5-Amino-1-(4-fluorophenyl)-4-{3-[2(S),3-dihydro-xypropoxy]benzoyl}pyrazole 340676 [5-amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]-[3-(1,2-dihydroxy-1-hydroxymethylethyl)phenyl]methanone 340680 H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-Nle-Trp-Boc 340681 H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-Nle-Trp-Ac 340682 Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-NMeNle-D-Trp-Boc 340687 5-amino-1-(4-fluorophenyl)-4-[3-{2(R), 3-dihydroxypropoxy}benzoyl]pyrazole 340694 c[Nle-Val-D-Phe-Arg-Trp-Glu]-NH2 340695 c[Nle-Nle-D-Phe-Arg-Trp-Glu]-NH2 340696 c[Nle-Val-D-Nal(2')-Arg-Trp-Glu]-NH2 340697 [5-amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]-[3-(2-piperidin-1-yl-ethoxy)phenyl]methanone 340714 (2S,3S,4R,5R)-5-(6-(2-(2,4-dichlorophenyl)acetamido)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 340730 1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-6-yl)-3-((R)-1-phenylethyl)urea 340739 1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-6-yl)-3-((S)-1-phenylethyl)urea 340740 1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-6-yl)-3-(5-methylisoxazol-3-yl)urea 340741 (2S,3S,4R,5R)-5-{6-[(Biphenyl-4-carbonyl)-amino]-purin-9-yl}-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid 1-cyclohexylamide 2-[(3-imidazol-1-yl-propyl)-amide] ethylamide 340742 1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-6-yl)-3-(1,3,4-thiadiazol-2-yl)urea 340744 6-hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]-6-pivaloyloxymethyl-tetrahydro-2-pyranone 340746 1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-6-yl)-3-(4-propoxyphenyl)urea 340747 1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-6-yl)-3-phenethylurea 340748 6-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]-6-pivaloyloxymethyl-tetrahydro-2-pyranone 340749 6-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]-6-hexanoyloxymethyl-tetrahydro-2-pyranone 340758 5-(hydroxymethyl)-5-(pivaloyloxymethyl)-3,3-bis(3-methyl-2-butenyl)dihydro-2(3H)-furanone 340759 6-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]-6-octanoyloxymethyl-tetrahydro-2-pyranone 340760 (2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-{3-[4-(pyrimidin-2-ylsulfamoyl)-phenyl]-ureido}-purin-9-yl)-tetrahydro-furan-2-carboxylic acid ethylamide 340763 5-(hydroxymethyl)-5-(pivaloyloxymethyl)-3,3-bis(3-methylbutyl)dihydro-2(3H)-furanone 340779 7-Methoxy-2-oxo-8-pentyloxy-1,2-dihydroquinoline-3-carboxylic Acid (2-aminophenyl)amide 340792 Ac-Nle-c[Asp-His-DPhe-Arg-Trp-Lys]-NH2 340797 [5-amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]-[3-(3-(dimethylamino)prop-1-ynyl)phenyl]methanone 340798 [5-amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]-{3-[2-(4-methyl-piperazin-1-yl)ethyl]phenyl}methanone 340809 [5-amino-1-(2,4-difluorophenyl)-1H-pyrazol-4-yl]-(3-pyridin-3-ylphenyl)methanone 340810 [5-amino-1-(2,4-difluorophenyl)-1H-pyrazol-4-yl]-[3-(1-oxypyridin-3-yl)phenyl]methanone 340813 7-Methoxy-2-oxo-8-pentyloxy-1,2-dihydroquinoline-3-carboxylic Acid Benzylamide 340814 7-Methoxy-2-oxo-8-pentyloxy-1,2-dihydroquinoline-3-carboxylic acid(2-phenylethyl)amide 340823 (R,Z)-2-(2-(hydroxymethyl)-4-(3-isobutyl-5-methylhexylidene)-5-oxo-tetrahydrofuran-2-yl)ethyl pivalate 340828 5-hexanoyloxymethyl-5-hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone 340829 5-hexanoyloxymethyl-5-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone 340837 5-hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]-5-octanoyloxymethyltetrahydro-2-furanone 340838 1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-2-iodo-9H-purin-6-yl)-3-(4-methoxyphenyl)urea 340846 1-(3-chlorophenyl)-3-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-2-(hex-1-ynyl)-9H-purin-6-yl)urea 340854 1-(3-chlorophenyl)-3-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-2-(2-phenylethynyl)-9H-purin-6-yl)urea 340859 (5-amino-1-phenyl-1H-pyrazol-4-yl)phenylmethanone 340861 c[Nle-Asp-D-Phe-Arg-Trp-Glu]-NH2 340862 3-[5-amino-1-(4-fluorophenyl)-1H-pyrazole-4-carbonyl]-benzonitrile 340872 4-[5-amino-1-(4-fluorophenyl)-1H-pyrazole-4-carbonyl]benzonitrile 340873 5-amino-1-(4-fluorophenyl)-4-[3-(pyridin-3-yl)-benzoyl]pyrazole 340880 H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-Nle-D-Trp-Boc 340887 [5-amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]-(4-pyridin-3-ylphenyl)methanone 340888 [5-amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]-(3-pyridin-4-ylphenyl)methanone 340895 [5-amino-1-(2,4-difluorophenyl)-1H-pyrazol-4-yl]-(3-pyridin-4-ylphenyl)methanone 340899 5-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]-5-octanoyloxymethyltetrahydro-2-furanone 340908 1-(3-chlorophenyl)-3-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-2-(3-hydroxy-3-phenylprop-1-ynyl)-9H-purin-6-yl)urea 340919 5-[(Z)-3-(tert-butoxy)-3-oxo-1-propenyl]-5-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone 340920 1-(2-chloro-9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-6-yl)-3-(4-methoxyphenyl)urea 340928 1-(3-chlorophenyl)-3-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-2-iodo-9H-purin-6-yl)urea 340933 (5-amino-1-phenyl-1H-pyrazol-4-yl)phenylmethanone O-methyloxime 340934 (5-amino-1-O-tolyl-1H-pyrazol-4-yl)phenylmethanone 340942 [5-amino-1-(3-nitrophenyl)-1H-pyrazol-4-yl]phenylmethanone 340943 [5-amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]-[3-(3-hydroxyprop-1-ynyl)phenyl]methanone 340946 N5-(4-aminocyclohexyl)-N7-(4-(methylsulfonyl)phenyl)-[1,2,4]triazolo[1,5-a]pyrimidine-5,7-diamine 340953 1-methyl-5-[2-(6-methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1H-indole 340960 1-methyl-5-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-indole 340961 3-Chloro-2-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 340962 1-methyl-5-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-benzoimidazole 340970 5-[2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1-[3-(tetrahydro-pyran-2-yloxy)-propyl]-1H-benzoimidazole 340971 5-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1-[3-(tetrahydro-pyran-2-yloxy)-propyl]-1H-benzoimidazole 340972 (+/-)-(3R,3aS,4S,4aR,8aS,9aR)-4-(2-(6-fluoroquinolin-2-yl)vinyl)-3-methyl-decahydronaphtho[2,3-c]furan-1(3H)-one 340973 (+/-)-(3R,3aS,4S,4aR,8aS,9aR)-3-methyl-4-(2-(7-methylquinolin-2-yl)vinyl)-decahydronaphtho[2,3-c]furan-1(3H)-one 340992 biphenyl-2-carboxylic acid [1-(3,5-bis-trifluoromethyl-phenyl)-1-methyl-ethyl]-methyl-amide 340999 1-(3,4-dimethoxyphenethyl)-3-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-6-yl)urea 341000 N-(2-methoxyphenyl)-4-(2-(2-methoxyphenylamino)pyridin-4-yl)pyridin-2-amine 341001 biphenyl-2-ylmethyl-(3,5-bis-trifluoromethyl-benzyl)-amine 341011 2-(3,5-bis-trifluoromethyl-benzyloxymethyl)-biphenyl 341012 3-methoxy-N-(4-(2-(phenylamino)pyridin-4-yl)pyridin-2-yl)propanamide 341018 5-methyl-N-(4-(2-(phenylamino)pyridin-4-yl)pyridin-2-yl)pyrazine-2-carboxamide 341019 3-chloro-4-fluoro-N-5-6-methoxy-7-3-morpholinopropoxy-quinazolin-4-ylamino-pyrimidin-2-yl-benzamide 341020 (rac)-1-(4-methyl-4-(phenylsulfonyl)pentyl)-3-(oxazol-5-yl)piperidine 341023 H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-Nle-D-Trp-1-Adoc 341028 2-(3,5-bis(trifluoromethyl)phenyl)-N,2-dimethyl-N-(4-o-tolylpyridin-3-yl)propanamide 341038 N-(4-(2-(phenylamino)pyridin-4-yl)pyridin-2-yl)-tetrahydro-2H-pyran-4-carboxamide 341039 2-(3,5-bis(trifluoromethyl)phenyl)-N,2-dimethyl-N-(2-(4-methylpiperazin-1-yl)-4-o-tolylpyrimidin-5-yl)propanamide 341041 6-[2-(6-methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1Hbenzoimidazole 341042 1-methyl-6-[2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo-[1,2-b]pyrazol-3-yl]-1H-benzoimidazole 341089 5-(1-methyl-4-(pyridin-4-ylmethylamino)-1H-imidazol-5-yl)-N-(3-(trifluoromethoxy)phenyl)-1,3,4-oxadiazol-2-amine 341090 5-(1-methyl-4-(pyridin-4-ylmethylamino)-1H-imidazol-5-yl)-N-m-tolyl-1,3,4-oxadiazol-2-amine 341097 N-(3-methoxyphenyl)-5-(1-methyl-4-(pyridin-4-ylmethylamino)-1H-imidazol-5-yl)-1,3,4-oxadiazol-2-amine 341099 N-5-6-methoxy-7-3-morpholinopropoxy-quinazolin-4-ylamino-pyrimidin-2-yl-isonicotinamide 341101 1-acetyl-N-(4-(2-(phenylamino)pyridin-4-yl)pyridin-2-yl)piperidine-4-carboxamide 341103 N-(4-(2-(4-fluorophenylamino)pyridin-4-yl)pyridin-2-yl)-tetrahydro-2H-pyran-4-carboxamide 341105 3-[6-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-benzoimidazol-1-yl]-propan-1-ol 341109 N-(3,5-bis(trifluoromethyl)benzyl)-N-methyl-3-o-tolylisonicotinamide 341111 dimethyl-(3-{6-[2-(6-methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-benzoimidazol-1-yl}-propyl)-amine 341117 2-(3,5-bis(trifluoromethyl)phenyl)-N,2-dimethyl-N-(3-o-tolylpyridin-4-yl)propanamide 341128 2-(5-fluoro-1H-indol-3-yl)-N-((4-isopropyl-3,4-dihydro-2H-benzo[b][1,4]oxazin-2-yl)methyl)ethanamine 341129 N-((4-benzyl-3,4-dihydro-2H-benzo[b][1,4]oxazin-2-yl)methyl)-2-(5-fluoro-1H-indol-3-yl)ethanamine 341136 2-(1H-indol-3-yl)-N-((4-phenyl-3,4-dihydro-2H-benzo[b][1,4]oxazin-2-yl)methyl)ethanamine 341149 5-(3-bromophenyl)-N-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine 341150 5-(3-bromophenyl)-N-(pyridin-4-ylmethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine 341154 N-(3,4-dichlorophenyl)-5-(1-methyl-4-(pyridin-4-ylmethylamino)-1H-imidazol-5-yl)-1,3,4-oxadiazol-2-amine 341155 N-(3,4-dimethoxyphenyl)-5-(1-methyl-4-(pyridin-4-ylmethylamino)-1H-imidazol-5-yl)-1,3,4-oxadiazol-2-amine 341157 N-[1-(2',6'-dichloro-biphenyl-2-yl)-methylidene]-N'-(3,5-dichloro-pyridin-4-yl)-hydrazine 341158 4-ethyl-N-5-6-methoxy-7-3-morpholinopropoxy-quinazolin-4-ylamino-pyrimidin-2-yl-benzamide 341164 biphenyl-2-carboxylic acid (3,5-bis-trifluoromethyl-benzyl)-methyl-amide 341165 2'-methyl-biphenyl-2-carboxylic acid (3,5-bis-trifluoromethyl-benzyl)-methyl-amide 341168 2-(1H-indol-3-yl)-N-((4-propyl-3,4-dihydro-2H-benzo[b][1,4]oxazin-2-yl)methyl)ethanamine 341175 3-(1H-indol-3-yl)-N-((4-isopropyl-3,4-dihydro-2H-benzo[b][1,4]oxazin-2-yl)methyl)propan-1-amine 341176 3-(1H-indol-3-yl)-N-((4-phenyl-3,4-dihydro-2H-benzo[b][1,4]oxazin-2-yl)methyl)propan-1-amine 341182 (+/-)-(3R,3aS,4S,4aR,8aS,9aR)-4-(2-(8-methoxyquinolin-2-yl)vinyl)-3-methyl-decahydronaphtho[2,3-c]furan-1(3H)-one 341183 2-((4-(5-fluoro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)methyl)-8-methoxy-3,4-dihydro-2H-benzo[b][1,4]oxazine 341184 2-((4-(5-fluoro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)methyl)-8-methoxy-4-methyl-3,4-dihydro-2H-benzo[b][1,4]oxazine 341188 1-methyl-6-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1Hbenzoimidazole 341189 3-(6-(2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-benzo[d]imidazol-1-yl)propan-1-ol 341190 (+/-)-(3R,3aS,4S,4aR,8aS,9aR)-3-methyl-4-(2-(8-methylquinolin-2-yl)vinyl)-decahydronaphtho[2,3-c]furan-1(3H)-one 341194 [4-(4-chloro-phenylcarbamoyloxy)-but-2-ynyl]-trimethyl-ammonium chloride 341220 N-[1-(2'-chloro-biphenyl-2-yl)-methylidene]-N'-(3,5-dichloro-pyridin-4-yl)-hydrazine 341221 N-[1-(2'-bromo-biphenyl-2-yl)-methylidene]-N'-(3,5-dichloro-pyridin-4-yl)-hydrazine 341239 2'-chloro-biphenyl-2-carboxylic acid (3,5-bis-trifluoromethyl-benzyl)-methyl-amide 341240 N-(4-fluorophenyl)-4-(2-(4-fluorophenylamino)pyridin-4-yl)pyridin-2-amine 341251 1-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 341293 1-methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 341298 2-(3,5-bis(trifluoromethyl)phenyl)-N,2-dimethyl-N-(3-o-tolylpyridin-2-yl)propanamide 341317 2-(3,5-bis(trifluoromethyl)phenyl)-N,2-dimethyl-N-(6-morpholino-4-o-tolylpyridin-3-yl)propanamide 341318 3,11-Dihydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 341319 3,11-Dimethoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 341322 N-5-6-methoxy-7-3-morpholinopropoxy-quinazolin-4-ylamino-pyrimidin-2-yl-pentanamide 341325 2-(3,5-bis(trifluoromethyl)phenyl)-N-(6-(4-hydroxypiperidin-1-yl)-4-o-tolylpyridin-3-yl)-N,2-dimethylpropanamide 341332 N-(3,5-bis(trifluoromethyl)benzyl)-N-methyl-3-o-tolylpicolinamide 341380 2-(5-fluoro-1H-indol-3-yl)-N-((8-methoxy-3,4-dihydro-2H-benzo[b][1,4]oxazin-2-yl)methyl)ethanamine 341385 (rac)-1-(4-methyl-4-(phenylsulfonyl)pentyl)-3-phenylpiperidine 341388 2-(5-fluoro-1H-indol-3-yl)-N-((7-methoxy-3,4-dihydro-2H-benzo[b][1,4]oxazin-2-yl)methyl)ethanamine 341401 N-(2-ethoxyphenyl)-4-(2-(2-ethoxyphenylamino)pyridin-4-yl)pyridin-2-amine 341407 4-ethyl-2-((4-(5-fluoro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)methyl)-8-methoxy-3,4-dihydro-2H-benzo[b][1,4]oxazine 341411 2'-methyl-5-(4-methyl-piperazin-1-yl)-biphenyl-2-carboxylic acid (3,5-bis-trifluoromethyl-benzyl)-methyl-amide 341426 cis-N-(4-(2-(4-fluorophenylamino)pyridin-4-yl)pyridin-2-yl)-4-methoxycyclohexanecarboxamide 341427 trans-N-(4-(2-(4-fluorophenylamino)pyridin-4-yl)pyridin-2-yl)-4-methoxycyclohexanecarboxamide 341431 4-phenyl-1-(3-(1-(phenylsulfonyl)cyclobutyl)propyl)piperidine 341432 2-(3-(1-(phenylsulfonyl)cyclobutyl)propyl)-1,2,3,4-tetrahydroisoquinoline 341433 3-chloro-N-5-6-methoxy-7-3-piperidin-1-yl-propoxy-quinazolin-4-ylamino-pyrimidin-2-yl-benzamide 341438 4-(5-(cyclohexylmethoxy)-[1,2,4]triazolo[1,5-a]pyrimidin-7-ylamino)benzenesulfonamide 341439 4-(5-(cyclohexyloxy)-[1,2,4]triazolo[1,5-a]pyrimidin-7-ylamino)benzenesulfonamide 341441 (rac)-2-(4-(phenylsulfonyl)butyl)-decahydroisoquinoline 341442 S-N-5-7-2-hydroxy-3-piperidin-1-yl-propoxy-6-methoxyquinazolin-4-ylamino-pyrimidin-2-yl-benzamide 341446 (rac)-1-(4-(phenylsulfonyl)pentyl)-3-(trifluoromethyl)piperidine 341453 N,N-diethyl-3-(6-(2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-benzo[d]imidazol-1-yl)propan-1-amine 341460 4-(3-(6-(2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-benzo[d]imidazol-1-yl)propyl)morpholine 341462 4-(5-(cyclohexylamino)-[1,2,4]triazolo[1,5-a]pyrimidin-7-ylamino)benzenesulfonamide 341463 4-(5-(4-hydroxycyclohexylamino)-[1,2,4]triazolo[1,5-a]pyrimidin-7-ylamino)benzenesulfonamide 341469 (R)-ethyl 1-(4-methyl-4-(phenylsulfonyl)pentyl)piperidine-3-carboxylate 341477 (rac)-3-phenyl-1-(4-(1-(phenylsulfonyl)cyclobutyl)butyl)pyrrolidine 341489 (rac)-3-phenyl-1-(3-(1-(phenylsulfonyl)cyclobutyl)propyl)pyrrolidine 341491 N-biphenyl-2-yl-2-(3,5-bis-trifluoromethyl-phenyl)-N-methyl-acetamide 341495 3-methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 341497 4-chloro-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecin-3-ol 341498 (rac)-3-phenyl-1-(2-(1-(phenylsulfonyl)cyclobutyl)ethyl)pyrrolidine 341500 N-biphenyl-2-yl-2-(3,5-bis-trifluoromethyl-phenyl)-N-methyl-isobutyramide 341502 N-(4-(2-(phenylamino)pyridin-4-yl)pyridin-2-yl)nicotinamide 341507 1-acetyl-N-(4-(2-(phenylamino)pyridin-4-yl)pyridin-2-yl)piperidine-3-carboxamide 341508 1-acetyl-N-(4-(2-(phenylamino)pyridin-4-yl)pyridin-2-yl)piperidine-2-carboxamide 341509 N-(4-(2-(phenylamino)pyridin-4-yl)pyridin-2-yl)furan-2-carboxamide 341512 2-(3,5-bis-trifluoromethyl-phenyl)-N-[6-(1,1-dioxo-1lambda*6*-thiomorpholin-4-yl)-4-o-tolyl-pyridin-3-yl]-N-methyl-isobutyramide 341513 1-((3-(2,6-dichlorophenyl)-5-methylisoxazol-4-yl)methylene)-2-(3,5-dichloropyridin-4-yl)hydrazine 341518 (rac)-2-(4-methyl-4-(phenylsulfonyl)pentyl)-decahydroisoquinoline 341531 2-(3,5-bis(trifluoromethyl)phenyl)-N,2-dimethyl-N-(2-(4-methylpiperazin-1-yl)-5-o-tolylpyridin-4-yl)propanamide 341538 6-[2-(6-methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1-(3-pyrrolidin-1-yl-propyl)-1H-benzoimidazole 341541 N-(3,5-bis(trifluoromethyl)benzyl)-N-methyl-6-(4-methylpiperazin-1-yl)-3-o-tolylpicolinamide 341542 N-((4-benzyl-3,4-dihydro-2H-benzo[b][1,4]oxazin-2-yl)methyl)-3-(1H-indol-3-yl)propan-1-amine 341545 6-[2-(6-methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1-(3-piperidin-1-yl-propyl)-1H-benzoimidazole 341546 dimethyl-{3-[6-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-benzoimidazol-1-yl]-propyl}-amine 341547 N-(4-chlorophenyl)-5-(1-methyl-4-(quinolin-5-ylmethylamino)-1H-imidazol-5-yl)-1,3,4-oxadiazol-2-amine 341548 (3R,3aS,4S,4aR,8aS,9aR)-3-methyl-4-(2-(quinolin-2-yl)vinyl)-decahydronaphtho[2,3-c]furan-1(3H)-one 341549 2-(5-fluoro-1H-indol-3-yl)-N-((4-phenyl-3,4-dihydro-2H-benzo[b][1,4]oxazin-2-yl)methyl)ethanamine 341550 N-((7-chloro-4-methyl-3,4-dihydro-2H-benzo[b][1,4]oxazin-2-yl)methyl)-2-(5-fluoro-1H-indol-3-yl)ethanamine 341580 N-(4-tert-butylphenyl)-5-(1-methyl-4-(pyridin-4-ylmethylamino)-1H-imidazol-5-yl)-1,3,4-oxadiazol-2-amine 341583 N-biphenyl-2-yl-2-(3,5-bis-trifluoromethyl-phenyl)-isobutyramide 341589 N-(4-isopropylphenyl)-5-(1-methyl-4-(pyridin-4-ylmethylamino)-1H-imidazol-5-yl)-1,3,4-oxadiazol-2-amine 341590 N-(4-(chlorodifluoromethoxy)phenyl)-5-(1-methyl-4-(pyridin-4-ylmethylamino)-1H-imidazol-5-yl)-1,3,4-oxadiazol-2-amine 341594 N-(3,5-bis(trifluoromethyl)benzyl)-N-methyl-6-(4-methylpiperazin-1-yl)-4-o-tolylnicotinamide 341598 (3R,3aS,4S,4aR,8aS,9aR)-4-(2-(6-methoxyquinolin-2-yl)vinyl)-3-methyl-decahydronaphtho[2,3-c]furan-1(3H)-one 341599 (+/-)-(3R,3aS,4S,4aR,8aS,9aR)-4-(2-(6-chloroquinolin-2-yl)vinyl)-3-methyl-decahydronaphtho[2,3-c]furan-1(3H)-one 341603 2-(3,5-bis(trifluoromethyl)phenyl)-N,2-dimethyl-N-(6-(4-methylpiperazin-1-yl)-4-o-tolylpyridin-3-yl)propanamide 341608 N-(4-chloro-3-(trifluoromethyl)phenyl)-5-(1-methyl-4-(pyridin-4-ylmethylamino)-1H-imidazol-5-yl)-1,3,4-oxadiazol-2-amine 341612 2-(5-fluoro-1H-indol-3-yl)-N-((4-isobutyl-3,4-dihydro-2H-benzo[b][1,4]oxazin-2-yl)methyl)ethanamine 341613 2-(1H-indol-3-yl)-N-((4-methyl-3,4-dihydro-2H-benzo[b][1,4]oxazin-2-yl)methyl)ethanamine 341615 6-(2-(pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1-(3-(pyrrolidin-1-yl)propyl)-1H-benzo[d]imidazole 341619 2-(5-fluoro-1H-indol-3-yl)-N-((4-methyl-3,4-dihydro-2H-benzo[b][1,4]oxazin-2-yl)methyl)ethanamine 341621 N-((3,4-dihydro-2H-benzo[b][1,4]oxazin-2-yl)methyl)-2-(1H-indol-3-yl)ethanamine 341622 5-(2-(pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-benzo[d]imidazole 341629 2-((4-(1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)methyl)-3,4-dihydro-2H-benzo[b][1,4]oxazine 341630 2-((4-(5-fluoro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)methyl)-8-methoxy-4-propyl-3,4-dihydro-2H-benzo[b][1,4]oxazine 341636 4-(5-(diethylamino)-[1,2,4]triazolo[1,5-a]pyrimidin-7-ylamino)benzenesulfonamide 341648 4-(5-(4-aminocyclohexylamino)-[1,2,4]triazolo[1,5-a]pyrimidin-7-ylamino)benzenesulfonamide 341649 4-(5-(4-aminocyclohexylamino)-[1,2,4]triazolo[1,5-a]pyrimidin-7-ylamino)-N,N-dimethylbenzenesulfonamide 341657 (3R)-1-acetyl-N-(4-(2-(4-fluorophenylamino)pyridin-4-yl)pyridin-2-yl)piperidine-3-carboxamide 341658 (3S)-1-acetyl-N-(4-(2-(4-fluorophenylamino)pyridin-4-yl)pyridin-2-yl)piperidine-3-carboxamide 341659 N-[1-biphenyl-2-yl-methylidene]-N'-(3,5-dichloro-pyridin-4-yl)-hydrazine 341660 N-(3,5-dichloro-pyridin-4-yl)-N'-[1-(2'-methyl-biphenyl-2-yl)-methylidene]-hydrazine 341667 N-(2'-(phenylamino)-4,4'-bipyridin-2-yl)tetrahydrofuran-3-carboxamide 341671 5-(1-methyl-4-(pyridin-4-ylmethylamino)-1H-imidazol-5-yl)-N-(4-(trifluoromethoxy)phenyl)-1,3,4-oxadiazol-2-amine 341672 5-(1-methyl-4-(pyridin-4-ylmethylamino)-1H-imidazol-5-yl)-N-(4-(trifluoromethyl)phenyl)-1,3,4-oxadiazol-2-amine 341686 N-(2-fluoro-4-methylphenyl)-5-(1-methyl-4-(pyridin-4-ylmethylamino)-1H-imidazol-5-yl)-1,3,4-oxadiazol-2-amine 341687 N-(benzo[d][1,3]dioxol-5-ylmethyl)-5-(1-methyl-4-(pyridin-4-ylmethylamino)-1H-imidazol-5-yl)-1,3,4-oxadiazol-2-amine 341695 N-(4-bromophenyl)-5-(1-methyl-4-(pyridin-4-ylmethylamino)-1H-imidazol-5-yl)-1,3,4-oxadiazol-2-amine 341696 biphenyl-4-yl-(5-{3-methyl-5-[(pyridin-4-ylmethyl)-amino]-3H-imidazol-4-yl}-[1,3,4]oxadiazol-2-yl)-amine 341698 4-(4'-Benzamidoanilino)-6,7-dimethoxyquinazoline 341705 1-acetyl-N-(4-(2-(4-fluorophenylamino)pyridin-4-yl)pyridin-2-yl)piperidine-3-carboxamide 341712 N-((4-ethyl-3,4-dihydro-2H-benzo[b][1,4]oxazin-2-yl)methyl)-2-(5-fluoro-1H-indol-3-yl)ethanamine 341716 (-)-N-(4-(2-(4-fluorophenylamino)pyridin-4-yl)pyridin-2-yl)-tetrahydrofuran-3-carboxamide 341719 N-((3,4-dihydro-2H-benzo[b][1,4]oxazin-2-yl)methyl)-2-(5-fluoro-1H-indol-3-yl)ethanamine 341794 2-Amino-3-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 341800 2-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 341801 2-methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 341802 1,3-Dichloro-2-methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 341803 N5-(4-aminocyclohexyl)-N7-(4-(phenylsulfonyl)phenyl)-[1,2,4]triazolo[1,5-a]pyrimidine-5,7-diamine 341811 1-Chloro-2-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 341814 4-methyl-1-(3-(1-(phenylsulfonyl)cyclobutyl)propyl)piperidine 341815 1-methyl-4-(3-(1-(phenylsulfonyl)cyclobutyl)propyl)piperazine 341822 1-phenyl-4-(3-(1-(phenylsulfonyl)cyclobutyl)propyl)piperazine 341823 (rac)-2-(3-(1-(phenylsulfonyl)cyclobutyl)propyl)-decahydroisoquinoline 341828 N-(2-fluorophenyl)-4-(2-(2-fluorophenylamino)pyridin-4-yl)pyridin-2-amine 341833 N1-(4-(2-(2-aminophenylamino)pyridin-4-yl)pyridin-2-yl)benzene-1,2-diamine 341837 2,4-dichloro-3-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 341841 4-(2-(o-toluidino)pyridin-4-yl)-N-o-tolylpyridin-2-amine 341844 (S)-ethyl 1-(4-methyl-4-(phenylsulfonyl)pentyl)piperidine-3-carboxylate 341848 1-(3-(1-(phenylsulfonyl)cyclobutyl)propyl)piperidine 341851 4-methoxy-N-(4-(2-(phenylamino)pyridin-4-yl)pyridin-2-yl)cyclohexanecarboxamide 341856 biphenyl-2-ylmethyl-(3,5-bis-trifluoromethyl-benzyl)-methyl-amine 341857 N-(5-(6-methoxy-7-(3-morpholinopropoxy)quinazolin-4-ylamino)pyrimidin-2-yl)benzamide 341865 N-2-6-methoxy-7-3-morpholinopropoxy-quinazolin-4-ylamino-pyrimidin-5-yl-benzamide 341868 2'-bromo-biphenyl-2-carboxylic acid (3,5-bis-trifluoromethyl-benzyl)-methyl-amide 341880 N-(3,5-bis(trifluoromethyl)benzyl)-N-methyl-2-(4-methylpiperazin-1-yl)-5-o-tolylpyrimidine-4-carboxamide 341884 N-(3,5-bis(trifluoromethyl)benzyl)-N-methyl-4-o-tolylnicotinamide 341889 2-(3,5-bis(trifluoromethyl)phenyl)-N,2-dimethyl-N-(2-(4-methylpiperazin-1-yl)-5-o-tolylpyrimidin-4-yl)propanamide 341892 SID29215551 341899 N-(3,5-bis(trifluoromethyl)benzyl)-N-methyl-2-(4-methylpiperazin-1-yl)-4-o-tolylpyrimidine-5-carboxamide 341915 2-(3,5-bis(trifluoromethyl)phenyl)-N,2-dimethyl-N-(6-(4-methylpiperazin-1-yl)-3-o-tolylpyridin-2-yl)propanamide 341929 (+)-(3R,3aS,4S,4aR,8aS,9aR)-3-methyl-4-(2-(6-(2-morpholino-2-oxoethoxy)quinolin-2-yl)vinyl)-decahydronaphtho[2,3-c]furan-1(3H)-one 341932 (4R,9aR)-6-chloro-4-methyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene 341933 (4R,9aS)-6-chloro-4-methyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene 341935 (+)-(3R,3aS,4S,4aR,8aS,9aR)-3-methyl-4-(2-(6-(3-(trifluoromethyl)phenyl)quinolin-2-yl)vinyl)-decahydronaphtho[2,3-c]furan-1(3H)-one 341936 (+)-N-(2-(2-((3R,3aS,4S,4aR,8aS,9aR)-3-methyl-1-oxo-dodecahydronaphtho[2,3-c]furan-4-yl)vinyl)quinolin-6-yl)butyramide 341944 N*1*-(3-Bromo-phenyl)-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cycloheptene-1,8-diamine 341945 (+)-N-(2-(2-((3R,3aS,4S,4aR,8aS,9aR)-3-methyl-1-oxo-dodecahydronaphtho[2,3-c]furan-4-yl)vinyl)quinolin-6-yl)pivalamide 341951 N*1*-(3-Chloro-4-fluoro-phenyl)-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cycloheptene-1,8-diamine 341968 (+)-2-methyl-2-(2-(2-((3R,3aS,4S,4aR,8aS,9aR)-3-methyl-1-oxo-dodecahydronaphtho[2,3-c]furan-4-yl)vinyl)quinolin-6-yloxy)propanamide 341969 2-((1H-pyrrolo[3,2-c]pyridin-1-yl)methyl)-N-(4-morpholinophenyl)benzamide 341970 2-((5H-imidazo[4,5-c]pyridin-5-yl)methyl)-N-(4-morpholinophenyl)benzamide 341973 (3-Bromo-phenyl)-(8-chloro-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 341974 N-[1-(3-Bromo-phenylamino)-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-8-yl]-methanesulfonamide 341975 (+)-2-(2-(2-((3R,3aS,4S,4aR,8aS,9aR)-3-methyl-1-oxo-dodecahydronaphtho[2,3-c]furan-4-yl)vinyl)quinolin-6-yloxy)-N-phenylacetamide 341976 2-((1H-pyrrolo[3,2-c]pyridin-1-yl)methyl)-N-(3,4-dichlorophenyl)benzamide 341981 (+)-2-methyl-2-(2-(2-((3R,3aS,4S,4aR,8aS,9aR)-3-methyl-1-oxo-dodecahydronaphtho[2,3-c]furan-4-yl)vinyl)quinolin-6-yloxy)-N-phenylpropanamide 342006 N-(4-chlorophenyl)-2-((5,6-dimethoxy-1H-benzo[d]imidazol-1-yl))benzamide 342012 (+)-(3R,3aS,4S,4aR,8aS,9aR)-3-methyl-4-(2-(6-(thiophen-3-yl)quinolin-2-yl)vinyl)-decahydronaphtho[2,3-c]furan-1(3H)-one 342017 (8-Bromo-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-(3-bromo-phenyl)-amine 342020 (+)-(3R,3aS,4S,4aR,8aS,9aR)-3-methyl-4-(2-(6-(thiophen-2-yl)quinolin-2-yl)vinyl)-decahydronaphtho[2,3-c]furan-1(3H)-one 342021 (+)-N-(2-(2-((3R,3aS,4S,4aR,8aS,9aR)-3-methyl-1-oxo-dodecahydronaphtho[2,3-c]furan-4-yl)vinyl)quinolin-6-yl)benzamide 342030 (+/-)-(3R,3aS,4S,4aR,8aS,9aR)-4-(2-(6-ethoxyquinolin-2-yl)vinyl)-3-methyl-decahydronaphtho[2,3-c]furan-1(3H)-one 342031 (+)-(3R,3aS,4S,4aR,8aS,9aR)-4-(2-(6-(benzyloxy)quinolin-2-yl)vinyl)-3-methyl-decahydronaphtho[2,3-c]furan-1(3H)-one 342033 (R)-4-(6-chloro-5-(2-(pyridin-4-yl)vinyl)pyridin-3-yl)-1-(1H-indol-3-yl)butan-2-amine 342034 (S)-N1-(6-chloro-5-(2-(pyridin-4-yl)vinyl)pyridin-3-yl)-3-(1H-indol-3-yl)propane-1,2-diamine 342042 N-((S)-2-amino-3-(indolin-3-yl)propyl)-6-chloro-5-(2-(pyridin-4-yl)vinyl)pyridin-3-amine 342043 (S)-N-(2-amino-3-(1H-indol-3-yl)propyl)-5-(2-(pyridin-4-yl)vinyl)pyridin-3-amine 342046 2-((1H-pyrrolo[3,2-c]pyridin-1-yl)methyl)-N-m-tolylbenzamide 342051 2-phenyl-2-(5-(2-(pyridin-4-yl)vinyl)pyridin-3-yl)ethanamine 342055 2-((5H-imidazo[4,5-c]pyridin-5-yl)methyl)-N-m-tolylbenzamide 342057 (S)-4-(2-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)vinyl)-N-benzylpyridin-2-amine 342058 (S)-1-(5-(2-(2-(1H-indol-1-yl)pyridin-4-yl)vinyl)pyridin-3-yloxy)-3-(1H-indol-3-yl)propan-2-amine 342061 (+)-2-(2-(2-((3R,3aS,4S,4aR,8aS,9aR)-3-methyl-1-oxo-dodecahydronaphtho[2,3-c]furan-4-yl)vinyl)quinolin-6-yloxy)acetic acid 342068 (4R,9aR)-6-methoxy-4-methyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene 342069 (4R,9aR)-4,6-dimethyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene 342070 (4R,9aR)-4-methyl-6-trifluoromethyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene 342071 ((4R,9aR)-4-methyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluoren-6-yl)-methanol 342077 (4R,9aR)-6-methoxymethyl-4-methyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene 342081 (R)-2-acetylamino-N-{(R)-1-benzyl-2-[(2S,4R)-4-benzyloxy-2-(3-guanidino-propyl)-pyrrolidin-1-yl]-2-oxo-ethyl}-3-(4-hydroxy-phenyl)-propionamide 342082 (S)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-benzyl-2-[(2S,4R)-4-benzyloxy-2-(3-guanidino-propyl)-pyrrolidin-1-yl]-2-oxo-ethyl}-amide 342084 (2-Fluoro-4-methylphenyl)-(4-isoquinolin-5-ylphthalazin-1-yl)amine 342089 2-((1H-pyrrolo[3,2-c]pyridin-1-yl)methyl)-N-(4-chlorophenyl)benzamide 342090 2-((5H-imidazo[4,5-c]pyridin-5-yl)methyl)-N-(4-chlorophenyl)benzamide 342092 (3-Bromo-phenyl)-(8-fluoro-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 342093 (3-Bromo-phenyl)-(7-methoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 342097 (4-Isoquinolin-5-yl-phthalazin-1-yl)-(2-methyl-1Hindol-5-yl)amine 342104 (3-Bromo-phenyl)-(8-methoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 342105 (8-Bromo-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-(3-chloro-4-fluoro-phenyl)-amine 342110 (S)-2-amino-3-(1H-indol-3-yl)-N-(5-(2-(pyridin-4-yl)vinyl)pyridin-3-yl)propanamide 342111 (3-Bromo-phenyl)-(10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 342112 (3-Chloro-4-fluoro-phenyl)-(10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 342114 1-(4-(4-(3-chloro-4-fluorophenylamino)-7-methoxyquinazolin-5-yloxy)piperidin-1-yl)ethanone 342119 (1R,3S)-1-(4-chlorophenoxy)-3-(4-methylpiperidin-1-yl)-9-(piperidin-4-ylmethyl)-2,3-dihydro-1H-carbazol-4(9H)-one 342120 1-[3,5-dihydroxy-4-((1R,6R)-6-isopropenyl-3-methyl-cyclohex-2-enyl)-phenyl]-cyclohexanecarbonitrile 342130 (4R,9aR)-4-methyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene-6-carbonitrile 342155 (3,4-Dichloro-phenyl)-(4-isoquinolin-5-yl-phthalazin-1-yl)-amine 342159 N-(3-chloro-4-fluorophenyl)-7-methoxy-5-(1-methylpiperidin-4-yloxy)quinazolin-4-amine 342167 (S)-2-((R)-2-benzyl-4-(R)-1,2,3,4-tetrahydro-isoquinolin-3-yl-butyrylamino)-5-guanidino-pentanoic acid ((S)-1-methylcarbamoyl-2-naphthalen-2-yl-ethyl)-amide 342168 (4-Chloro-3-trifluoromethylphenyl)-(4-isoquinolin-5-yl-phthalazin-1-yl)amine 342169 N-(4-chlorophenyl)-2-((4-(pyridin-4-yl)-1H-pyrazol-1-yl)methyl)benzamide 342172 N-(3-chloro-4-fluorophenyl)-6-methoxy-5-(1-methylpiperidin-4-yloxy)quinazolin-4-amine 342173 2-((1R,6R)-6-isopropenyl-3-methyl-cyclohex-2-enyl)-5-naphthalen-1-yl-benzene-1,3-diol 342174 1-[3,5-dihydroxy-4-((1R,6R)-6-isopropenyl-3-methyl-cyclohex-2-enyl)-phenyl]-cyclopentanecarbonitrile 342178 (8-Chloro-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-(3-chloro-4-fluoro-phenyl)-amine 342179 N-(3-chloro-4-fluorophenyl)-7-methoxy-5-(1-(methylsulfonyl)piperidin-4-yloxy)quinazolin-4-amine 342180 N-(3-chloro-4-fluorophenyl)-7-(2-methoxyethoxy)-5-(tetrahydro-2H-pyran-4-yloxy)quinazolin-4-amine 342185 (3-Chloro-4-fluoro-phenyl)-(8-fluoro-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 342186 2-((1H-pyrrolo[3,2-c]pyridin-1-yl)methyl)-N-(4-bromophenyl)benzamide 342188 N-[1-(3-Bromo-phenylamino)-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-8-yl]-acrylamide 342193 2-((5H-imidazo[4,5-c]pyridin-5-yl)methyl)-N-(4-bromophenyl)benzamide 342194 (1R,3R)-1-(4-chlorophenoxy)-3-(4-methylpiperidin-1-yl)-9-(piperidin-4-ylmethyl)-2,3-dihydro-1H-carbazol-4(9H)-one 342195 N-[1-(3-Chloro-4-fluoro-phenylamino)-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-8-yl]-acrylamide 342202 (1R)-1-(4-chlorophenoxy)-3-(4-fluoro-4-methylpiperidin-1-yl)-9-(piperidin-4-ylmethyl)-2,3-dihydro-1H-carbazol-4(9H)-one 342203 (S)-1-phenyl-3-(5-(2-(pyridin-4-yl)vinyl)pyridin-2-yloxy)propan-2-amine 342204 (S)-1-(1H-indol-3-yl)-3-(5-(2-(2-methoxypyridin-4-yl)vinyl)pyridin-3-yloxy)propan-2-amine 342209 (1R)-1-(4-chlorophenoxy)-3-(4,4-difluoropiperidin-1-yl)-9-(piperidin-4-ylmethyl)-2,3-dihydro-1H-carbazol-4(9H)-one 342218 (S)-3-(2-amino-3-(5-(2-(pyridin-4-yl)vinyl)pyridin-3-yloxy)propyl)phenol 342220 (6aR,10aR)-3-(4-ethylphenyl)-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol 342224 (3-bromo-phenyl)-(7,8-dimethoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 342225 (3-chloro-4-fluoro-phenyl)-(7,8-dimethoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 342226 N-bphenyl-4-yl-2-imidazo[4,5-c]pyridin-5-ylmethyl-benzamide 342227 2-((5H-imidazo[4,5-c]pyridin-5-yl)methyl)-N-(4-phenoxyphenyl)benzamide 342228 (S)-3-methyl-1-(5-(2-(pyridin-4-yl)vinyl)pyridin-3-yloxy)butan-2-amine 342236 2-((5H-imidazo[4,5-c]pyridin-5-yl)methyl)-N-(4-benzylphenyl)benzamide 342237 (1R)-1-(4-chlorophenoxy)-3-(4-methyl-3-oxopiperazin-1-yl)-9-(piperidin-4-ylmethyl)-2,3-dihydro-1H-carbazol-4(9H)-one 342239 (S)-1-phenyl-3-(5-(2-(pyridin-4-yl)vinyl)pyridin-3-yloxy)propan-2-amine 342240 5-(4-(3,4-difluorobenzylamino)-1-methyl-1H-imidazol-5-yl)-N-(4-chlorophenyl)-1,3,4-oxadiazol-2-amine 342241 5-(4-((1H-indazol-5-yl)methylamino)-1-methyl-1H-imidazol-5-yl)-N-(4-chlorophenyl)-1,3,4-oxadiazol-2-amine 342242 (S)-1-(1H-indol-3-yl)-3-(5-(2-(2-phenoxypyridin-4-yl)vinyl)pyridin-3-yloxy)propan-2-amine 342243 (1R)-1-(4-chlorophenoxy)-3-(4-methylpiperazin-1-yl)-9-((1-methylpiperidin-4-yl)methyl)-2,3-dihydro-1H-carbazol-4(9H)-one 342244 (S)-4-phenyl-1-(5-(2-(pyridin-4-yl)vinyl)pyridin-3-yloxy)butan-2-amine 342256 (S)-3-(2-amino-3-(5-(2-(pyridin-4-yl)vinyl)pyridin-3-yloxy)propyl)benzonitrile 342263 (S)-1-(naphthalen-1-yl)-3-(5-(2-(pyridin-4-yl)vinyl)pyridin-3-yloxy)propan-2-amine 342273 (R)-1-(1H-indol-3-yl)-3-(5-(2-(pyridin-4-yl)vinyl)pyridin-3-yloxy)propan-2-amine 342278 (4-tert-Butylphenyl)-(4-quinolin-5-yl-phthalazin-1-yl)amine 342290 (1R)-1-(4-chlorophenoxy)-9-methyl-3-(4-methylpiperazin-1-yl)-2,3-dihydro-1H-carbazol-4(9H)-one 342293 2-((1H-pyrrolo[3,2-c]pyridin-1-yl)methyl)-N-(4-tert-butylphenyl)benzamide 342296 2-(1-methyl-1H-indol-3-yl)-2-(5-(2-(pyridin-4-yl)vinyl)pyridin-3-yl)ethanamine 342309 (S)-1-(naphthalen-2-yl)-3-(5-(2-(pyridin-4-yl)vinyl)pyridin-3-yloxy)propan-2-amine 342319 2-(5-(2-(pyridin-4-yl)vinyl)pyridin-3-yloxy)ethanamine 342321 3-(5-(2-(pyridin-4-yl)vinyl)pyridin-3-yloxy)propan-1-amine 342323 N-(4-chlorophenyl)-5-(1-methyl-4-(pyridin-4-ylmethylamino)-1H-imidazol-5-yl)-1,3,4-oxadiazol-2-amine 342327 (S)-1-(6-chloro-5-(2-(pyridin-4-yl)vinyl)pyridin-3-yloxy)-3-(1H-indol-3-yl)propan-2-amine 342334 (1R)-1-(4-chlorophenoxy)-3-(4-methylpiperazin-1-yl)-9-(3-(piperidin-1-yl)propyl)-2,3-dihydro-1H-carbazol-4(9H)-one 342335 (S)-1,1-diphenyl-3-(5-(2-(pyridin-4-yl)vinyl)pyridin-3-yloxy)propan-2-amine 342339 N-{3-[(2S,4R)-4-benzyloxy-1-((R)-2-benzyl-4-(S)-1,2,3,4-tetrahydro-isoquinolin-3-yl-butyryl)-pyrrolidin-2-yl]-propyl}-guanidine 342340 5-(4-(2-(benzo[d][1,3]dioxol-5-yl)ethylamino)-1-methyl-1H-imidazol-5-yl)-N-(4-chlorophenyl)-1,3,4-oxadiazol-2-amine 342345 N-(3-chloro-4-fluorophenyl)-5-(1-methylpiperidin-4-yloxy)quinazolin-4-amine 342350 (R)-1-(4-chlorophenoxy)-9-(3-(piperidin-1-yl)propyl)-2,3-dihydro-1H-carbazol-4(9H)-one 342351 (1R)-1-(4-chlorophenoxy)-3-morpholino-9-(3-(piperidin-1-yl)propyl)-2,3-dihydro-1H-carbazol-4(9H)-one 342355 N-(3-chloro-4-fluorophenyl)-7-(3-(4-methylpiperazin-1-yl)propoxy)-5-(tetrahydro-2H-pyran-4-yloxy)quinazolin-4-amine 342370 (S)-2-amino-3-phenyl-N-(5-(2-(pyridin-4-yl)vinyl)pyridin-3-yl)propanamide 342373 Benzyl-(8-bromo-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 342374 Benzyl-(8-fluoro-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 342379 2-((5H-imidazo[4,5-c]pyridin-5-yl)methyl)-N-(4-(chlorodifluoromethoxy)phenyl)benzamide 342381 Biphenyl-3-yl-(8-fluoro-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 342382 Biphenyl-3-yl-(8-methoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 342386 (+/-)-tert-butyl 2-(2-(2-((3R,3aS,4S,4aR,8aS,9aR)-3-methyl-1-oxo-dodecahydronaphtho[2,3-c]furan-4-yl)vinyl)quinolin-6-yloxy)ethylcarbamate 342395 (+)-(3R,3aS,4S,4aR,8aS,9aR)-4-(2-(6-aminoquinolin-2-yl)vinyl)-3-methyl-decahydronaphtho[2,3-c]furan-1(3H)-one 342397 (1R)-1-(4-chlorophenoxy)-9-(((3R,4R)-3-fluoro-1-methylpiperidin-4-yl)methyl)-3-(4-methylpiperazin-1-yl)-2,3-dihydro-1H-carbazol-4(9H)-one 342399 (1R)-1-(4-chlorophenoxy)-3-(piperidin-1-yl)-9-(3-(piperidin-1-yl)propyl)-2,3-dihydro-1H-carbazol-4(9H)-one 342401 (S)-1-(2-chloro-5-(2-(pyridin-4-yl)vinyl)pyridin-3-yloxy)-3-(1H-indol-3-yl)propan-2-amine 342402 (S)-1-(1-methyl-1H-indol-3-yl)-3-(5-(2-(pyridin-4-yl)vinyl)pyridin-3-yloxy)propan-2-amine 342403 (1R)-1-(4-chlorophenoxy)-9-(((3R,4S)-3-fluoropiperidin-4-yl)methyl)-3-(4-methylpiperazin-1-yl)-2,3-dihydro-1H-carbazol-4(9H)-one 342406 (3-Bromo-phenyl)-(7,9-dimethoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 342407 Ac-Tyr-D-Phe-Arg-2-Nal-NHCH3 342409 (S)-2-amino-3-(naphthalen-1-yl)-N-(5-(2-(pyridin-4-yl)vinyl)pyridin-3-yl)propanamide 342412 (1R)-1-(4-chlorophenoxy)-9-(((3R,4S)-3-fluoro-1-methylpiperidin-4-yl)methyl)-3-(4-methylpiperazin-1-yl)-2,3-dihydro-1H-carbazol-4(9H)-one 342414 (S)-1-(1H-indol-3-yl)-3-(5-(2-(2-(phenylthio)pyridin-4-yl)vinyl)pyridin-3-yloxy)propan-2-amine 342415 (S)-1-(5-(2-(2-(benzylthio)pyridin-4-yl)vinyl)pyridin-3-yloxy)-3-(1H-indol-3-yl)propan-2-amine 342424 (S)-4-(2-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)vinyl)pyridin-2-amine 342425 (4-Chlorophenyl)-(4-isoquinolin-5-yl-phthalazin-1-yl)amine 342428 (+)-(3R,3aS,4S,4aR,8aS,9aR)-4-(2-(5,6-dimethoxyquinolin-2-yl)vinyl)-3-methyl-decahydronaphtho[2,3-c]furan-1(3H)-one 342435 (+)-N-(2-(2-((3R,3aS,4S,4aR,8aS,9aR)-3-methyl-1-oxo-dodecahydronaphtho[2,3-c]furan-4-yl)vinyl)quinolin-6-yl)acetamide 342448 Tic-D-Phe-Arg-2-Nal-NHCH3 342452 (+)-N-(2-(2-((3R,3aS,4S,4aR,8aS,9aR)-3-methyl-1-oxo-dodecahydronaphtho[2,3-c]furan-4-yl)vinyl)quinolin-6-yl)propionamide 342455 2-((5H-imidazo[4,5-c]pyridin-5-yl)methyl)-N-(4-tert-butylphenyl)benzamide 342456 (3-Chloro-4-fluoro-phenyl)-(7-methoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 342457 (3-Chloro-4-fluoro-phenyl)-(8-methoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 342459 (+)2-(2-(2-((3R,3aS,4S,4aR,8aS,9aR)-3-methyl-1-oxo-dodecahydronaphtho[2,3-c]furan-4-yl)vinyl)quinolin-6-yloxy)acetamide 342461 2-((1H-pyrrolo[3,2-c]pyridin-1-yl)methyl)-N-(4-isopropylphenyl)benzamide 342462 2-((5H-imidazo[4,5-c]pyridin-5-yl)methyl)-N-(4-isopropylphenyl)benzamide 342463 (1R)-1-(4-chlorophenoxy)-9-(((3R,4R)-3-fluoropiperidin-4-yl)methyl)-3-(4-methylpiperazin-1-yl)-2,3-dihydro-1H-carbazol-4(9H)-one 342464 (S)-4-(2-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)vinyl)-N-methylpyridin-2-amine 342473 2-((1H-pyrrolo[3,2-c]pyridin-1-yl)methyl)-N-(4-(chlorodifluoromethoxy)phenyl)benzamide 342488 (+)-N-cyclopropyl-2-(2-(2-((3R,3aS,4S,4aR,8aS,9aR)-3-methyl-1-oxo-dodecahydronaphtho[2,3-c]furan-4-yl)vinyl)quinolin-6-yloxy)acetamide 342503 (+)-(3R,3aS,4S,4aR,8aS,9aR)-4-(2-(6-hydroxyquinolin-2-yl)vinyl)-3-methyl-decahydronaphtho[2,3-c]furan-1(3H)-one 342508 (4-Chloro-phenyl)-(8-methoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 342509 2-((5H-imidazo[4,5-c]pyridin-5-yl)methyl)-N-(3,4-dichlorophenyl)benzamide 342513 (+/-)-(3R,3aS,4S,4aR,8aS,9aR)-4-(2-(5-chloro-6-methoxyquinolin-2-yl)vinyl)-3-methyl-decahydronaphtho[2,3-c]furan-1(3H)-one 342514 (4R,9aR)-6-Cyclopropylmethoxymethyl-4-methyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene 342515 1-((4R,9aR)-4-methyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluoren-6-yl)-ethanol 342523 2-((1H-pyrrolo[3,2-c]pyridin-1-yl)methyl)-N-(4-chloro-3-(trifluoromethyl)phenyl)benzamide 342525 1-((6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-3-yl)cyclohexanecarbonitrile 342526 4-((1R,6R)-6-isopropenyl-3-methyl-cyclohex-2-enyl)-4'-methyl-biphenyl-3,5-diol 342531 2-(2-((1H-pyrrolo[3,2-c]pyridin-1-yl)methyl)phenyl)-5-chloro-1H-benzo[d]imidazole 342538 (1R)-1-(4-chlorophenoxy)-3-(4-methylpiperidin-1-yl)-9-(3-(piperidin-1-yl)propyl)-2,3-dihydro-1H-carbazol-4(9H)-one 342539 (S)-3-(2-(pyridin-4-yl)vinyl)-5-(pyrrolidin-2-ylmethoxy)pyridine 342555 (S)-1-(1H-indol-3-yl)-3-(6-(2-(pyridin-4-yl)vinyl)pyridin-2-yloxy)propan-2-amine 342563 (4R,9aR)-6-bromo-4-methyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene 342564 (4R,9aS)-6-bromo-4-methyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene 342567 (S)-1-(benzo[b]thiophen-3-yl)-3-(5-(2-(pyridin-4-yl)vinyl)pyridin-3-yloxy)propan-2-amine 342568 2-((5H-imidazo[4,5-c]pyridin-5-yl)methyl)-N-(4-chloro-3-(trifluoromethyl)phenyl)benzamide 342575 2-((1H-pyrrolo[3,2-c]pyridin-1-yl)methyl)-N-(2-fluoro-4-methylphenyl)benzamide 342576 2-((5H-imidazo[4,5-c]pyridin-5-yl)methyl)-N-(2-fluoro-4-methylphenyl)benzamide 342580 (4R,9aR)-6-[1-((S)-ethoxy)-ethyl]-4-methyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene 342582 2-((1H-pyrrolo[3,2-c]pyridin-1-yl)methyl)-N-(benzo[d][1,3]dioxol-5-yl)benzamide 342583 (1R)-1-(4-chlorophenoxy)-3-(piperazin-1-yl)-9-(3-(piperidin-1-yl)propyl)-2,3-dihydro-1H-carbazol-4(9H)-one 342586 (4R,9aR)-6-[1-((R)-ethoxy)-ethyl]-4-methyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene 342589 (4-tert-Butylphenyl)-(4-isoquinolin-5-yl-phthalazin-1-yl)amine 342597 (2R,5R)-5-acetylamino-2-benzyl-6-(4-hydroxy-phenyl)-hexanoic acid [(S)-4-guanidino-1-((S)-1-methylcarbamoyl-2-naphthalen-2-yl-ethylcarbamoyl)-butyl]-amide 342603 (2R,5R)-5-acetylamino-2-(4-fluoro-benzyl)-6-(4-hydroxy-phenyl)-hexanoic acid [(S)-4-guanidino-1-((S)-1-methylcarbamoyl-2-naphthalen-2-yl-ethylcarbamoyl)-butyl]-amide 342604 (2R,5R)-5-acetylamino-2-(4-fluoro-benzyl)-6-phenyl-hexanoic acid [(S)-4-guanidino-1-((S)-1-methylcarbamoyl-2-naphthalen-2-yl-ethylcarbamoyl)-butyl]-amide 342607 (1R)-1-(4-chlorophenoxy)-9-((4-(methylamino)cyclohexyl)methyl)-3-(4-methylpiperazin-1-yl)-2,3-dihydro-1H-carbazol-4(9H)-one 342608 Benzyl-(8-methoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 342609 (8-Bromo-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-phenyl-amine 342610 (8-Fluoro-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-phenyl-amine 342625 (1R,3S)-1-(4-chlorophenoxy)-3-(4-methylpiperazin-1-yl)-9-(piperidin-4-ylmethyl)-2,3-dihydro-1H-carbazol-4(9H)-one 342626 (8-Methoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-phenyl-amine 342627 1-(3-Bromo-phenylamino)-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cycloheptene-8-carboxylic acid 342628 N-(3-chloro-4-fluorophenyl)-7-methoxy-5-(piperidin-4-yloxy)quinazolin-4-amine 342629 (6aR,10aR)-6,6,9-trimethyl-3-p-tolyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol 342634 1-(3-Chloro-4-fluoro-phenylamino)-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cycloheptene-8-carboxylic acid 342637 (6aR,10aR)-6,6,9-trimethyl-3-(naphthalen-1-yl)-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol 342641 (S)-1-(1H-indol-3-yl)-N,N-dimethyl-3-(5-(2-(pyridin-4-yl)vinyl)pyridin-3-yloxy)propan-2-amine 342646 1-((6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-3-yl)cyclopentanecarbonitrile 342650 1-(1H-indol-3-yl)-3-(5-(2-(pyridin-4-yl)vinyl)pyridin-3-yloxy)propan-2-ol 342659 3-(4-bromophenyl)-N-(2-(5-((E)-2-(pyridin-4-yl)vinyl)pyridin-3-yloxy)ethyl)prop-2-en-1-amine 342669 (1R,3R)-1-(4-chlorophenoxy)-3-(4-methylpiperazin-1-yl)-9-(piperidin-4-ylmethyl)-2,3-dihydro-1H-carbazol-4(9H)-one 342675 (1R)-1-(4-chlorophenoxy)-3-(4-(2-hydroxyethyl)piperazin-1-yl)-9-(piperidin-4-ylmethyl)-2,3-dihydro-1H-carbazol-4(9H)-one 342676 (S)-4-(2-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)vinyl)-N-ethylpyridin-2-amine 342682 (S)-4-(2-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)vinyl)-N-cyclopropylpyridin-2-amine 342685 6-chloro-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene 342691 (4-Isoquinolin-5-yl-phthalazin-1-yl)-(4-morpholin-4-ylphenyl)-amine 342697 (2R,5R)-5-acetylamino-6-(4-chloro-phenyl)-2-(4-fluoro-benzyl)-hexanoic acid [(S)-4-guanidino-1-((S)-1-methylcarbamoyl-2-naphthalen-2-yl-ethylcarbamoyl)-butyl]-amide 342714 N-(3-chloro-4-fluorophenyl)-7-methoxy-5-(tetrahydro-2H-pyran-4-yloxy)quinazolin-4-amine 342734 (6aR,10aR)-6,6,9-trimethyl-3-(4-propylphenyl)-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol 342763 (S)-3-(azetidin-2-ylmethoxy)-5-(2-(pyridin-4-yl)vinyl)pyridine 342770 (S)-1-(benzyloxy)-3-(5-(2-(pyridin-4-yl)vinyl)pyridin-3-yloxy)propan-2-amine 342771 N-(3-chloro-4-fluorophenyl)-7-methoxy-5-(tetrahydrofuran-3-yloxy)quinazolin-4-amine 342772 N-(3-chloro-4-fluorophenyl)-5-isopropoxy-7-methoxyquinazolin-4-amine 342789 (S)-1-(1H-indol-3-yl)-3-(5-(2-(pyridin-4-yl)vinyl)pyridin-3-yloxy)propan-2-amine 342790 2-((5H-imidazo[4,5-c]pyridin-5-yl)methyl)-N-(benzo[d][1,3]dioxol-5-yl)benzamide 342794 (4-Isopropylphenyl)-(4-isoquinolin-5-yl-phthalazin-1-yl)amine 342795 [4-(Chloro-difluoro-methoxy)-phenyl]-(4-isoquinolin-5-yl-phthalazin-1-yl)amine 342802 (4-Isoquinolin-5-yl-phthalazin-1-yl)-m-tolylamine 342830 2-morpholin-1-yl-N-{4-[4-(3-pyridin-2-yl-1H-pyrazol-4-yl)-pyridin-2-yl]phenyl}acetamide 342831 N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-6,7-dichloro-4-oxo-4H-chromene-2-carboxamide 342833 H-[Trp-Arg-Nva-Arg-Tyr]2-NH2 342834 H-[Trp-Arg-Nva-Arg-Tyr]3-NH2 342838 N-{2-[2-(3-(S)-hydroxypyrrolidin-1-yl)ethyl]-2H-indazol-5-yl}-N'-(4-phenoxyphenyl)urea 342839 6-ethyl-5-[4-(4-trifluoromethanesulfonyl-benzylamino)-phenyl]-pyrimidine-2,4-diamine 342845 5-{4-[(2-chloro-pyridin-4-ylmethyl)-amino]-phenyl}-6-ethylpyrimidine-2,4-diamine 342846 5-{4-[(5-chloro-thiophen-3-ylmethyl)-amino]-phenyl}-6-ethyl-pyrimidine-2,4-diamine 342848 2-(3-methoxyphenyl)-4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridine 342851 6-benzyloxymethyl-5-[4-(4-trifluoromethyl-benzylamino)-phenyl]-pyrimidine-2,4-diamine 342852 6-benzyloxymethyl-5-{4-[(5-chloro-thiophen-3-ylmethyl)-amino]-phenyl}-pyrimidine-2,4-diamine 342853 2-[4-methylphenyl]-4-3-pyridin-2-yl-1H-pyrazol-4-yl pyridine 342854 4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)-2-(4-(trifluoromethyl)phenyl)pyridine 342857 6-[(benzyloxy)methyl]-5-{4-[(4-methoxybenzyl)amino]phenyl}-pyrimidine-2,4-diamine 342858 6-benzyloxymethyl-5-{4-[(4-chloro-phenylamino)-methyl]-phenyl}-pyrimidine-2,4-diamine 342863 5-[3-chloro-4-(4-methanesulfonyl-benzylamino)-phenyl]-6-ethyl-pyrimidine-2,4-diamine 342864 5-[3-bromo-4-(4-methanesulfonyl-benzylamino)-phenyl]-6-ethyl-pyrimidine-2,4-diamine 342868 6-ethyl-5-(4-{methyl[4-(methylsulfonyl)benzyl]amino}phenyl)-pyrimidine-2,4-diamine 342882 2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(3-hydroxymethyl-phenyl)-acetamide 342893 (1-(2-cyclopropyl-6-(cyclopropylamino)-5-methylpyrimidin-4-yl)piperidin-4-yl)methanol 342894 N,2-dicyclopropyl-5-methyl-6-(4-(trifluoromethyl)piperidin-1-yl)pyrimidin-4-amine 342895 N,2-dicyclopropyl-6-(4,4-difluoropiperidin-1-yl)-5-methylpyrimidin-4-amine 342896 4-({[4-(2,4-diamino-6-ethylpyrimidin-5-yl)phenyl]amino}-methyl)benzonitrile 342900 (1-benzo{1,3}dioxol-5-ylmethylpiperidin-4-yl)(6-methoxyquinolin-4-yl)amine 342901 N-(4-phenoxyphenyl)-N'-[2-(2-pyrrolidin-1-ylethyl)-2H-indazol-5-yl]urea 342905 2-[4-methoxyphenyl]-4-(3-pyridin-2-yl-1H-pyrazol-4-yl)pyridine 342906 tert-butyl-[5-(1H-imidazol-4-yl)-pentyl]-amine 342907 cyclopentyl-[5-(1H-imidazol-4-yl)-pentyl]-amine 342909 2-((R)-5-cyclohexyl-2,3-dihydro-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1H-benzo[e][1,4]diazepin-3-yl)-N-(3-(methylamino)phenyl)-acetamide 342910 4-{[(4-{2,4-diamino-6-[(benzyloxy)methyl]pyrimidin-5-yl}-phenyl)amino]methyl}benzonitrile 342912 4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)-2-(3-(trifluoromethyl)phenyl)pyridine 342913 2-(4-fluorophenyl)-4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridine 342918 2-[4-isopropylphenyl]-4-[3-(pyridin-2-yl)-1H-pyrazol-4-yl]pyridine 342922 6-ethyl-5-[4-({[4-(methylsulfonyl)phenyl]amino}methyl)phenyl]-pyrimidine-2,4-diamine 342930 N-[3-(3-cyanophenyl)-2-cyclopenten-1-yl]-N'-(3,5-dichlorophenyl)-N-[2-(1-pyrrolidinyl)ethyl]urea 342943 2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(3-hydroxy-phenyl)-acetamide 342963 2-(4-chlorophenyl)-4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridine 342969 4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methyl-6-(2-(1-methylpiperidin-4-yl)ethoxy)pyrrolo[1,2-f][1,2,4]triazine 342970 4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrrolo[2,1-f][1,2,4]triazine 342971 4-(4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridin-2-yl)-N-(tetrahydro-2H-pyran-4-yl)benzamide 342972 N-methyl-4-(4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridin-2-yl)-N-(tetrahydro-2H-pyran-4-yl)benzamide 342976 N'-(3-chloro-4-fluorophenyl)-N-[trans-3-(3-cyanophenyl)cyclopentyl]-N-[3-(4-methyl-1-piperazinyl)propyl]urea 342977 N'-(3-chloro-4-fluorophenyl)-N-[cis-3-(3-cyanophenyl)cyclopentyl]-N-[3-(4-methyl-1-piperazinyl)propyl]urea 342978 N-(4-(4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridin-2-yl)phenyl)tetrahydro-2H-pyran-4-carboxamide 342982 N-[5-(3-cyanophenyl)bicyclo[3.1.0]hex-2-yl]-N'-(3,5-dichlorophenyl)-N-[2-(1-pyrrolidinyl)ethyl]urea 342995 1-[5-(1H-imidazol-4-yl)-pentyl]-piperidine 342996 1-[5-(1H-imidazol-4-yl)-pentyl]-azepane 343016 6-[(benzyloxy)methyl]-5-{4-[(pyridin-4-ylmethyl)amino]-phenyl}pyrimidine-2,4-diamine 343017 6-benzyloxymethyl-5-{4-[(5-chloro-thiophen-2-ylmethyl)-amino]-phenyl}-pyrimidine-2,4-diamine 343024 5-[4-(benzylamino)phenyl]-6-[(benzyloxy)methyl]pyrimidine-2,4-diamine 343030 4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methyl-6-(3-(methylsulfonyl)propoxy)pyrrolo[2,1-f][1,2,4]triazine 343034 (R)-1-(2-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy)ethyl)pyrrolidin-3-ol 343039 cyclohexyl-[5-(1H-imidazol-4-yl)-pentyl]-amine 343040 cycloheptyl-[5-(1H-imidazol-4-yl)-pentyl]-amine 343041 (R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[1,2-f][1,2,4]triazin-6-yloxy)propan-2-ol 343042 (S)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy)propan-2-ol 343045 4-chloro-benzyl-[5-(1H-imidazol-4-yl)-pentyl]-amine 343046 [5-(1H-imidazol-4-yl)-pentyl]-dimethyl-amine 343047 [5-(1H-imidazol-4-yl)-pentyl]-diethyl-amine 343048 [5-(1H-imidazol-4-yl)-pentyl]-isobutyl-amine 343049 (R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy)-3-methoxypropan-2-ol 343050 N'-(3-chloro-4-fluorophenyl)-N-[trans-5-(3-cyanophenyl)-bicyclo[3.1.0]hex-2-yl]-N-[2-(1-pyrrolidinyl)ethyl]urea 343055 4-(5-pyrrolidin-1-yl-pentyl)-1H-imidazole 343058 (-)-N'-(3-chloro-4-fluorophenyl)-N-[trans-5-(3-cyanophenyl)bicyclo[3.1.0]hex-2-yl]-N-[2-[3(R)-hydroxy-1-pyrrolidinyl]ethyl]urea 343064 Loxiglumide 343068 N-arachidonoyl-N-(2-hydroxyethyl)hydroxylamine 343078 ethyl[4-(1H-imidazol-4-yl)butyl]amine 343079 [4-(1H-Imidazol-4-yl)butyl]propylamine 343080 [4-(1H-imidazol-4-yl)-butyl]-iso-propyl-amine 343087 1-((1S,2R,5S)-5-(3-acetamidophenyl)bicyclo[3.1.0]hexan-2-yl)-3-(3-chloro-4-fluorophenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)urea 343095 N-[3-[trans-4-[[[(3-chloro-4-fluorophenyl)amino]carbonyl][3-(4-methyl-1-piperazinyl)propyl]amino]bicyclo[3.1.0]hex-1-yl]-phenyl]methanesulfonamide 343096 (Z)-3-(2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,2-dihydrobenzo[e][1,2,4]triazepin-3-yl)acetamido)benzoic acid 343101 N'-(3-chloro-4-fluorophenyl)-N-[3-(4-methyl-1-piperazinyl)-propyl]-N-[trans-5-[4-(methylsulfonyl)phenyl]bicyclo[3.1.0]hex-2-yl]urea 343106 N-[trans-5-(4-fluorophenyl)bicyclo[3.1.0]hex-2-yl]-N'-[4-fluoro-3-(trifluoromethyl)phenyl)-N-[3-(4-methyl-1-piperazinyl)propyl]-urea 343107 N'-(3-chloro-4-fluorophenyl)-N-[trans-5-(3-methylphenyl)-bicyclo[3.1.0]hex-2-yl]-N-[3-(4-methyl-1-piperazinyl)propyl]-urea 343112 N'-(3-chloro-4-fluorophenyl)-N-[3-(4-methyl-1-piperazinyl)-propyl]-N-[trans-5-(3-thienyl)bicyclo[3.1.0]hex-2-yl]urea 343113 N-[trans-5-(4-cyanophenyl)bicyclo[3.1.0]hex-2-yl]-N'-[4-fluoro-3-(trifluoromethyl)phenyl)-N-[3-(1-piperazinyl)propyl]urea 343119 (+/-)-2-(2-(1H-indole-2-carboxamido)benzamido)-3-phenylpropanoic acid 343120 2-(R,S)-{2-[(1H-Indole-2-carbonyl)-amino]-benzoylamino}-propionic acid 343121 O-arachidonoyl-N-(2-hydroxyethyl)hydroxylamine 343122 4-[4-(3-pyridin-2-yl-1H-pyrazol-4-yl)pyridin-2-yl]benzoic acid methyl ester 343129 4-(4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridin-2-yl)benzonitrile 343130 2-(4-(2-cyclohexylethoxy)phenyl)-4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridine 343144 3-(3-chloro-4-fluorophenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)-1-((1S,2R,5S)-5-phenylbicyclo[3.1.0]hexan-2-yl)urea 343153 N'-(3-chloro-4-fluorophenyl)-N-[3-(4-methyl-1-piperazinyl)-propyl]-N-[trans-5-[3-(trifluoromethoxy)phenyl]bicyclo[3.1.0]-hex-2-yl]urea 343157 6-(3-cyano-phenyl)-bicyclo[4.1.0]hept-3-yl]-3-(4-fluoro-3-trifluoromethyl-phenyl)-1-[2-((S)-3-hydroxy-pyrrolidin-1-yl)-ethyl]-urea 343158 3-(3-chloro-4-fluorophenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)-1-((1S,2R,5S)-5-(pyridin-3-yl)bicyclo[3.1.0]hexan-2-yl)urea 343159 N'-[4-fluoro-3-(trifluoromethyl)phenyl)-N-[trans-5-(3-methoxyphenyl)bicyclo[3.1.0]hex-2-yl]-N-[3-(4-methyl-1-piperazinyl)propyl]urea 343162 N'-[4-fluoro-3-(trifluoromethyl)phenyl)-N-[trans-5-(4-methoxyphenyl)bicyclo[3.1.0]hex-2-yl]-N-[3-(4-methyl-1-piperazinyl)propyl]urea 343172 2(R,S)-{2-[(2-acetylaminocinnamoyl)amino]benzoylamino}-3-phenylpropionic acid 343173 (+/-)-2-(2-cinnamamidobenzamido)-3-phenylpropanoic acid 343176 N-arachidonoyl-O-(2-hydroxyethyl)hydroxylamine 343178 5-(4-(4-chlorobenzylamino)phenyl)-6-(benzyloxymethyl)pyrimidine-2,4-diamine 343183 2-{4-[(2-chloroethyl)oxy]phenyl}-4-[3-(pyridin-2-yl)-1H-pyrazol-4-yl]pyridine 343187 6-[(benzyloxy)methyl]-5-[4-(neopentylamino)phenyl]pyrimidine-2,4-diamine 343190 1-(4-(4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridin-2-yl)phenoxy)propan-2-one 343191 dimethyl-{2-[(4-{4-[3-(pyridin-2-yl)-1H-pyrazol-4-yl]-2-pyridinyl}phenyl)oxy]ethyl}amine 343195 N-oleoyl-O-(2-hydroxyethyl)hydroxylamine 343197 4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)-2-(4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)pyridine 343198 N-[trans-5-(3-cyanophenyl)bicyclo[3.1.0]hex-2-yl]-N'-[4-fluoro-3-(trifluoromethyl)phenyl]-N-[2-(3(R)-hydroxy-1-pyrrolidinyl]ethyl]urea 343205 N'-(3-chloro-4-fluorophenyl)-N-[trans-5-(3-cyanophenyl)-bicyclo[3.1.0]hex-2-yl]-N-[2-(1-piperidinyl)ethyl]urea 343206 N-[trans-5-(3-cyanophenyl)bicyclo[3.1.0]hex-2-yl]-N'-[4-fluoro-3-(trifluoromethyl)phenyl]-N-[2-(4-methyl-1-piperazinyl)-ethyl]urea 343207 2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(3-(methyl-(2-methylaminoethyl)-amino)-phenyl)-acetamide 343213 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-ethylpyrimidine-2,4-diamine 343226 5-(4-{[3,5-difluoro-4-(methylsulfonyl)benzyl]amino}phenyl)-6-ethylpyrimidine-2,4-diamine 343227 6-[(benzyloxy)methyl]-5-[4-({4-[(trifluoromethyl)sulfonyl]-benzyl}amino)phenyl]pyrimidine-2,4-diamine 343244 6-ethyl-5-{4-[(4-nitrobenzyl)amino]phenyl}pyrimidine-2,4-diamine 343250 6-benzyloxymethyl-5-{4-[(quinolin-3-ylmethyl)-amino]-phenyl}-pyrimidine-2,4-diamine 343251 5-[4-(4-chloro-benzylamino)-phenyl]-6-phenethyl-pyrimidine-2,4-diamine 343256 N-(3-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy)propyl)methanesulfonamide 343260 butyl-[4-(1H-imidazol-4-yl)-butyl]-amine 343261 [4-(1H-imidazol-4-yl)-butyl]-isobutyl-amine 343262 tert-Butyl-[4-(1H-imidazol-4-yl)-butyl]-amine 343263 cyclopentyl-[4-(1H-imidazol-4-yl)-butyl]-amine 343267 6-[(benzyloxy)methyl]-5-{4-[(4-nitrobenzyl)amino]phenyl}-pyrimidine-2,4-diamine 343268 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-(benzyloxymethyl)pyrimidine-2,4-diamine 343274 cyclohexyl-[4-(1H-imidazol-4-yl)-butyl]-amine tartaric acid 343280 N-[trans-5-(3-cyanophenyl)bicyclo[3.1.0]hex-2-yl]-N'-[4-fluoro-3-(trifluoromethyl)phenyl]-N-[2-[4-(2-methylpropyl)-1-piperazinyl]ethyl]urea 343283 6-[(benzyloxy)methyl]-5-(4-{[4-(methylsulfonyl)benzyl]oxy}-phenyl)pyrimidine-2,4-diamine 343287 N-[trans-5-(3-cyanophenyl)bicyclo[3.1.0]hex-2-yl]-N'-[4-fluoro-3-(trifluoromethyl)phenyl)-N-[4-(4-morpholinyl)butyl]urea 343302 5-(4-(4-chlorobenzylamino)phenyl)-6-ethylpyrimidine-2,4-diamine 343313 2-(4-(2-(1H-imidazol-1-yl)ethoxy)phenyl)-4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridine 343339 2-[2-(trifluoromethyl)phenyl]-4-(3-pyridin-2-yl-1H-pyrazol-4-yl)pyridine 343346 [(4-{4-[3-(pyridin-2-yl)-1H-pyrazol-4-yl]-pyridin-2-yl}phenyl)-methyl]tetrahydro-2H-pyran-4-ylamine 343351 1-(2-cyclopropyl-6-(cyclopropylamino)-5-methylpyrimidin-4-yl)piperidin-4-ol 343358 1-(2-cyclopropyl-6-(cyclopropylamino)-5-methylpyrimidin-4-yl)piperidin-4-one 343359 N,2-dicyclopropyl-5-methyl-6-(piperidin-1-yl)pyrimidin-4-amine 343360 2-(4-Methoxyphenyl)-N-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-6-yl]acetamide 343363 2-[3-methylphenyl]-4-(3-pyridin-2-yl-1H-pyrazol-4-yl)pyridine 343364 methyl 4-(1H-indol-5-yloxy)pyrrolo[2,1-f][1,2,4]triazine-6-carboxylate 343376 N-oleoyl-N-(2-hydroxyethyl)hydroxylamine 343379 cycloheptyl-[4-(1H-imidazol-4-yl)-butyl]-amine 343385 O-oleoyl-N-(2-hydroxyethyl)hydroxylamine 343390 ethyl 4-(1H-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazine-6-carboxylate 343391 4-[3-(pyridin-2-yl)-1H-pyrazol-4-yl]-2-[4-(1-pyrrolidinylmethyl)phenyl]pyridine 343405 2-(4-phenoxyphenyl)-N-[1-(2-pyrrolidin-1-ylethyl)-1H-indazol-5-yl]acetamide 343408 1-(4-{[4-(2,4-diamino-6-ethyl-pyrimidin-5-yl)-phenylamino]-methyl}-phenyl)-ethanone 343414 1-(4-{[4-(2,4-diamino-6-ethyl-pyrimidin-5-yl)-phenylamino]-methyl}-phenyl)-ethanol 343418 2-phenyl-4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridine 343422 cyclopropyl-(2-cyclopropyl-5-methyl-6-thiomorpholin-4-yl-pyrimidin-4-yl)-amine 343424 1-(4-{[4-(2,4-diamino-6-benzyloxymethyl-pyrimidin-5-yl)-phenylamino]-methyl}-phenyl)-ethanone 343425 6-[(benzyloxy)methyl]-5-(4-{[(2-chloropyridin-4-yl)methyl]-amino}phenyl)pyrimidine-2,4-diamine 343426 2-(2-fluorophenyl)-4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridine 343429 2-((S)-5-cyclohexyl-2,3-dihydro-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1H-benzo[e][1,4]diazepin-3-yl)-N-(3-(methylamino)phenyl)-acetamide 343431 4-[4-(2,4-diamino-6-benzyloxymethyl-pyrimidin-5-yl)-phenoxymethyl]-benzonitrile 343432 2-(2-methylphenyl)-4-[3-(pyridin-2-yl)-1H-pyrazol-4-yl]pyridine 343436 6-[(benzyloxy)methyl]-5-(4-{[(4-nitro-phenyl)amino]methyl}-phenyl)pyrimidine-2,4-diamine 343437 6-ethyl-5-(4-{[(4-nitro-phenyl)amino]methyl}phenyl)-pyrimidine-2,4-diamine 343438 4-{2-[(4-{4-[3-(pyridin-2-yl)-1H-pyrazol-4-yl]-pyridin-2-yl}-phenyl)oxy]ethyl}morpholine 343441 N'-(3-chloro-4-fluorophenyl)-N-[3-(4-methyl-1-piperazinyl)-propyl]-N-[trans-5-[4-(trifluoromethoxy)phenyl]bicyclo[3.1.0]-hex-2-yl]urea 343445 N-(4-phenoxyphenyl)-N'-[1-(2-piperidin-1-ylethyl)-1H-indazol-5-yl]urea 343446 N-(4-phenoxyphenyl)-N'-[1-(2-azepan-1-yl-ethyl)-1H-indazol-5-yl]urea 343447 N'-(3-chloro-4-fluorophenyl)-N-[trans-5-(3, 5-difluorophenyl)-bicyclo[3.1.0]hex-2-yl]-N-[3-(4-methyl-1-piperazinyl)propyl]-urea 343448 N'-(3-chloro-4-fluorophenyl)-N-[trans-5-(3, 4-difluorophenyl)-bicyclo[3.1.0]hex-2-yl]-N-[3-(4-methyl-1-piperazinyl)propyl]-urea 343449 4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-ol 343455 1-((1S,2R,5S)-5-(4-cyanophenyl)bicyclo[3.1.0]hexan-2-yl)-3-(4-fluoro-3-(trifluoromethyl)phenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)urea 343457 4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methyl-6-(3-(piperidin-1-yl)propoxy)pyrrolo[2,1-f][1,2,4]triazine 343460 N,2-dicyclopropyl-5-methyl-6-(4-methylpiperidin-1-yl)pyrimidin-4-amine 343468 ethyl-[5-(1H-imidazol-4-yl)-pentyl]-amine 343469 [5-(1H-imidazol-4-yl)-pentyl]-propyl-amine 343470 [5-(1H-imidazol-4-yl)-pentyl]-iso-propyl-amine 343472 N-[trans-5-(3-cyanophenyl)bicyclo[3.1.0]hex-2-yl]-N'-[4-fluoro-3-(trifluoromethyl)phenyl)-N-[4-(4-methyl-1-piperazinyl)butyl]-urea 343479 butyl-[5-(1H-imidazol-4-yl)-pentyl]-amine 343483 N-[trans-5-(3-cyanophenyl)bicyclo[3.1.0]hex-2-yl]-N'-[4-fluoro-3-(trifluoromethyl)phenyl)-N-[4-(1-piperidinyl)butyl]urea 343487 N'-(3-chloro-4-fluorophenyl)-N-[trans-5-(3-chlorophenyl)-bicyclo[3.1.0]hex-2-yl]-N-[3-(4-methyl-1-piperazinyl)propyl]urea 343493 N'-(3-chloro-4-fluorophenyl)-N-[trans-5-(3-fluorophenyl)-bicyclo[3.1.0]hex-2-yl]-N-[3-(4-methyl-1-piperazinyl)propyl]-urea 343494 N-[trans-5-(3-fluorophenyl)bicyclo[3.1.0]hex-2-yl]-N'-[4-fluoro-3-(trifluoromethyl)phenyl)-N-[3-(4-methyl-1-piperazinyl)propyl]-urea 343501 N-[trans-5-(3-cyano-4-fluorophenyl)bicyclo[3.1.0]hex-2-yl]-N'-[4-fluoro-3-(trifluoromethyl)phenyl)-N-[3-(4-methyl-1-piperazinyl)propyl]urea 343507 N-[trans-5-(4-cyano-3-fluorophenyl)bicyclo[3.1.0]hex-2-yl]-N'-[4-fluoro-3-(trifluoromethyl)phenyl)-N-[3-(4-methyl-1-piperazinyl)propyl]urea 343511 ethyl 4-(1H-indol-5-yloxy)-5-ethylpyrrolo[2,1-f][1,2,4]triazine-6-carboxylate 343512 ethyl 4-(1H-indol-5-yloxy)-5-isopropylpyrrolo[2,1-f][1,2,4]triazine-6-carboxylate 343521 methyl 5-methyl-4-(2-methyl-1H-indol-5-yloxy)pyrrolo[2,1-f][1,2,4]triazine-6-carboxylate 343522 methyl 4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazine-6- 343530 4-chloro-benzyl-[4-(1H-imidazol-4-yl)-butyl]-amine 343531 [4-(1H-imidazol-4-yl)-butyl]-dimethyl-amine 343532 [4-(1H-imidazol-4-yl)-butyl]-diethyl-amine 343533 4-(4-pyrrolidin-1-yl-butyl)-1H-imidazole 343534 N-(2-methoxyethyl)-4-(4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridin-2-yl)benzamide 343535 2-pyrrolidin-1-yl-N-{4-[4-(3-pyridin-2-yl-1H-pyrazol-4-yl)-pyridin-2-yl]phenyl}acetamide 343539 1-[4-(1H-imidazol-4-yl)-butyl]-piperidine 343540 1-[4-(1H-imidazol-4-yl)-butyl]-azepane 343550 N'-(3-chloro-4-fluorophenyl)-N-[3-(4-methyl-1-piperazinyl)-propyl]-N-[trans-5-[3-(methylsulfonyl)phenyl]bicyclo[3.1.0]hex-2-yl]urea 343551 1-((1S,2R,5S)-5-(3-aminophenyl)bicyclo[3.1.0]hexan-2-yl)-3-(3-chloro-4-fluorophenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)urea 343559 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-4-(trifluoromethyl)pyridin-2(1H)-one 343572 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-(bicyclo[2.2.1]heptan-2-yl)pyrimidine-2,4-diamine 343574 1-benzyl-3-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)urea 343586 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-((3-methylbut-2-enyloxy)methyl)pyrimidine-2,4-diamine 343588 2-(4-(4-chlorophenoxy)phenyl)-1H-benzo[d]imidazole-5-carboxylic acid 343595 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-((methyl(phenyl)amino)methyl)pyrimidine-2,4-diamine 343637 N,2-dicyclopropyl-6-(4-ethylpiperidin-1-yl)-5-methylpyrimidin-4-amine 343642 N,2-dicyclopropyl-6-(5,6-dihydropyridin-1(2H)-yl)-5-methylpyrimidin-4-amine 343643 N,2-dicyclopropyl-6-(4,4-dimethylpiperidin-1-yl)-5-methylpyrimidin-4-amine 343644 [6-(8-aza-spiro[4.5]dec-8-yl)-2-cyclopropyl-5-methyl-pyrimidin-4-yl]-cyclopropyl-amine 343652 6-(4-benzylpiperidin-1-yl)-N,2-dicyclopropyl-5-methylpyrimidin-4-amine 343653 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-cyclobutylpyrimidine-2,4-diamine 343660 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-cyclopentylpyrimidine-2,4-diamine 343661 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-cyclohexylpyrimidine-2,4-diamine 343668 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-((furan-2-ylmethoxy)methyl)pyrimidine-2,4-diamine 343669 5-[4-(4-methanesulfonyl-benzylamino)-phenyl]-6-(5-methyl-furan-2-ylmethoxymethyl)-pyrimidine-2,4-diamine 343676 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-((pyridin-3-ylmethoxy)methyl)pyrimidine-2,4-diamine 343677 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-((cyclopentylamino)methyl)pyrimidine-2,4-diamine 343682 N'-(3-chloro-4-fluorophenyl)-N-[trans-5-[4(methylsulfonyl)-phenyl]bicyclo[3.1.0]hex-2-yl]-N-[3-(2-oxo-1-pyrrolidinyl)propyl]-urea 343683 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-((cyclopentylmethylamino)methyl)pyrimidine-2,4-diamine 343684 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-((phenylamino)methyl)pyrimidine-2,4-diamine 343686 3-(4-(3-phenoxybenzylamino)phenyl)propanoic acid 343690 4-[[[[(3-chloro-4-fluorophenyl)amino]carbonyl][(trans-5-[4-(methylsulfonyl)phenyl]bicyclo[3.1.0]hex-2-yl]amino]methyl]-1-(methylsulfonyl)piperidine 343699 5-(3-((S)-2-(4-(4-ethylphenyl)-3-hydroxybutyl)-5-oxopyrrolidin-1-yl)propyl)thiophene-2-carboxylic acid 343720 7-((S)-2-(3-hydroxy-4-phenylbutyl)-5-oxopyrrolidin-1-yl)heptanoic acid 343721 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-3-(trifluoromethyl)pyridin-2(1H)-one 343727 4-(3-(2-(3-hydroxy-4-phenylbutyl)-5-oxopyrrolidin-1-yl)propyl)benzoic acid 343729 1-benzyl-3-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-1-ethylurea 343733 N-benzyl-6-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)hexanamide 343750 7-[(S)-2-((R)-4-biphenyl-3-yl-3-hydroxy-butyl)-5-oxo-pyrrolidin-1-yl]-heptanoic acid 343759 4-{3-[2-(4-biphenyl-3-yl-3-hydroxy-butyl)-5-oxo-pyrrolidin-1-yl]-propyl}-benzoic acid 343760 7-((S)-2-((R)-3-hydroxy-4-(3-(trifluoromethoxy)phenyl)butyl)-5-oxopyrrolidin-1-yl)heptanoic acid 343765 7-((S)-2-(3-hydroxy-4-(3-phenoxyphenyl)butyl)-5-oxopyrrolidin-1-yl)heptanoic acid 343766 4-(3-(2-(3-hydroxy-4-(3-phenoxyphenyl)butyl)-5-oxopyrrolidin-1-yl)propyl)benzoic acid 343770 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-4-phenylpyridin-2(1H)-one 343771 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-3-methoxypyridin-2(1H)-one 343777 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-3-methylpyridin-2(1H)-one 343778 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-3-phenethylurea 343783 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-3-(cyclohexylmethyl)urea 343784 3-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-1,1-diethylurea 343793 5-(3-((S)-2-(3-hydroxy-4-phenylbutyl)-5-oxopyrrolidin-1-yl)propyl)thiophene-2-carboxylic acid 343796 4-(3-(2-(4-(3-chlorophenyl)-3-hydroxybutyl)-5-oxopyrrolidin-1-yl)propyl)benzoic acid 343801 5-(3-((S)-2-(3-hydroxy-4-(naphthalen-2-yl)butyl)-5-oxopyrrolidin-1-yl)propyl)thiophene-2-carboxylic acid 343803 5-(3-((S)-2-((R)-4-(3-chlorophenyl)-3-hydroxybutyl)-5-oxopyrrolidin-1-yl)propyl)thiophene-2-carboxylic acid 343804 5-{3-[(S)-2-(4-biphenyl-2-yl-3-hydroxy-butyl)-5-oxo-pyrrolidin-1-yl]-propyl}-thiophene-2-carboxylic acid 343811 7-((S)-2-((R)-3-hydroxy-4-(3-(methoxymethyl)phenyl)butyl)-5-oxopyrrolidin-1-yl)heptanoic acid 343812 7-((S)-2-((R)-3-hydroxy-4-(3-(2-methoxyethyl)phenyl)butyl)-5-oxopyrrolidin-1-yl)heptanoic acid 343813 N4-benzyl-N6,2-dicyclopropyl-N4,5-dimethylpyrimidine-4,6-diamine 343814 6-(azepan-1-yl)-N,2-dicyclopropylpyrimidin-4-amine 343815 6-(azepan-1-yl)-N,2-dicyclopropyl-5-fluoropyrimidin-4-amine 343822 6-(azepan-1-yl)-5-bromo-N,2-dicyclopropylpyrimidin-4-amine 343832 6-(azepan-1-yl)-N-cyclobutyl-2-cyclopropyl-5-methylpyrimidin-4-amine 343842 (S)-N-(3-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)phenyl)pyrimidin-2-amine 343844 N,2-dicyclopropyl-5-methyl-6-(4-methylenepiperidin-1-yl)pyrimidin-4-amine 343845 N,2-dicyclopropyl-5-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-amine 343847 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-((4-fluorophenylamino)methyl)pyrimidine-2,4-diamine 343848 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-(((4-fluorophenyl)(methyl)amino)methyl)pyrimidine-2,4-diamine 343849 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-isopropylpyrimidine-2,4-diamine 343850 3-(azepan-1-yl)-N,5-dicyclopropyl-2-methylbenzenamine 343851 6-(azocan-1-yl)-N,2-dicyclopropyl-5-methylpyrimidin-4-amine 343852 N4-cyclohexyl-N6,2-dicyclopropyl-5-methylpyrimidine-4,6-diamine 343854 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-ethyl-N4-isobutylpyrimidine-2,4-diamine 343855 2-(5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-2-amino-6-ethylpyrimidin-4-ylamino)ethanol 343856 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-(2,3-dihydrobenzofuran-2-yl)pyrimidine-2,4-diamine 343857 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-((benzylamino)methyl)pyrimidine-2,4-diamine 343860 (-)-6-(azepan-1-yl)-N-cyclopropyl-5-methyl-2-(2-methylcyclopropyl)pyrimidin-4-amine 343863 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-N4-cyclopropyl-6-ethylpyrimidine-2,4-diamine 343866 (+)-6-(azepan-1-yl)-N-cyclopropyl-2-(2-methylcyclopropyl)pyrimidin-4-amine 343869 exo-5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-((2S)-bicyclo[2.2.1]hept-5-en-2-yl)pyrimidine-2,4-diamine 343870 endo-5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-(bicyclo[2.2.1]hept-5-en-2-yl)pyrimidine-2,4-diamine 343871 N,2-dicyclopropyl-5-ethyl-6-thiomorpholinopyrimidin-4-amine 343877 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-butylpyrimidine-2,4-diamine 343878 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-isobutylpyrimidine-2,4-diamine 343880 4-(3-(2-(4-(4-fluorophenyl)-3-hydroxybutyl)-5-oxopyrrolidin-1-yl)propyl)benzoic acid 343892 (S)-5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-(tetrahydrofuran-2-yl)pyrimidine-2,4-diamine 343893 (R)-5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-(tetrahydrofuran-2-yl)pyrimidine-2,4-diamine 343900 6-(azepan-1-yl)-N,2-dicyclopropyl-5-nitropyrimidin-4-amine 343937 N4-cycloheptyl-N6,2-dicyclopropyl-5-methylpyrimidine-4,6-diamine 343938 6-(3-aza-bicyclo[3.2.1]octan-3-yl)-N,2-dicyclopropyl-5-methylpyrimidin-4-amine 343939 N4-benzyl-N6,2-dicyclopropyl-5-methylpyrimidine-4,6-diamine 343947 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-tert-butylpyrimidine-2,4-diamine 343948 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-pentylpyrimidine-2,4-diamine 343959 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-hexylpyrimidine-2,4-diamine 343960 ethyl 3-(5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-2,6-diaminopyrimidin-4-yl)propanoate 343965 N-(3,5-dimethylbenzyl)-3-(5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-2,6-diaminopyrimidin-4-yl)propanamide 343973 N-(3-chlorobenzyl)-3-(5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-2,6-diaminopyrimidin-4-yl)propanamide 343984 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-(2,3-dihydrobenzo[b][1,4]dioxin-2-yl)pyrimidine-2,4-diamine 343985 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-(aminomethyl)pyrimidine-2,4-diamine 343993 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-((methylamino)methyl)pyrimidine-2,4-diamine 343994 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-(indolin-1-ylmethyl)pyrimidine-2,4-diamine 344024 (S)-1-(1H-indol-3-yl)-3-(6-(pyridin-4-yl)quinolin-3-yloxy)propan-2-amine 344025 (2S)-1-(1H-indol-3-yl)-3-(6-(pyridin-3-yl)quinolin-3-yloxy)propan-2-amine 344030 3-methyl-2-(4-phenoxyphenyl)-3H-benzo[d]imidazole-5-carboxamide 344038 (S)-2-(3-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)phenyl)acetamide 344039 (S)-N-(4-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)phenyl)acetamide 344042 N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-7-methoxy-4-oxo-4H-chromene-2-carboxamide 344044 N-(3-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)phenyl)acetamide 344045 N-(3-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)phenyl)thiazol-2-amine 344050 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-((benzyl(methyl)amino)methyl)pyrimidine-2,4-diamine 344051 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-(isoindolin-2-ylmethyl)pyrimidine-2,4-diamine 344052 (S)-(2-amino-5-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)phenyl)(3-chlorophenyl)methanone 344053 (S)-5-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)-1-naphthamide 344056 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-N4-cyclopropyl-6-ethylpyrimidine-2,4-diamine 344057 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-N4-benzyl-6-ethylpyrimidine-2,4-diamine 344060 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-((dimethylamino)methyl)pyrimidine-2,4-diamine 344062 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-4-ethyl-6-morpholinopyrimidin-2-amine 344075 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-4-hydroxypyridin-2(1H)-one 344081 2-(4-(4-chlorophenoxy)phenyl)-1H-indole-6-carboxylic acid 344082 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-4-(trifluoromethyl)pyrimidin-2(1H)-one 344083 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-6-methylpyridin-2(1H)-one 344088 1-tert-butyl-3-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)urea 344089 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-3-neopentylurea 344096 2-(4-(4-chlorophenoxy)phenyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide 344097 2-(4-(4-chlorophenoxy)phenyl)-1H-imidazo[4,5-b]pyridine-5-carboxamide 344109 7-(2-(4-(3-chlorophenyl)-3-hydroxybutyl)-5-oxopyrrolidin-1-yl)heptanoic acid 344114 7-((S)-2-((R)-3-hydroxy-4-(3-hydroxyphenyl)butyl)-5-oxopyrrolidin-1-yl)heptanoic acid 344130 5-(3-((S)-2-((R)-4-(4-fluorophenyl)-3-hydroxybutyl)-5-oxopyrrolidin-1-yl)propyl)thiophene-2-carboxylic acid 344134 N-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-3-phenylpropanamide 344135 2-(3-(piperidin-1-yl)propyl)-2H-isoindole-1-carbonitrile 344137 5-{3-[(S)-2-(4-biphenyl-3-yl-3-hydroxy-butyl)-5-oxo-pyrrolidin-1-yl]-propyl}-thiophene-2-carboxylic acid 344141 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-3-phenylurea 344146 4-(3-(2-(4-(3-fluorophenyl)-3-hydroxybutyl)-5-oxopyrrolidin-1-yl)propyl)benzoic acid 344147 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-5-(trifluoromethyl)pyridin-2(1H)-one 344151 5-(3-((S)-2-(4-(3-fluorophenyl)-3-hydroxybutyl)-5-oxopyrrolidin-1-yl)propyl)thiophene-2-carboxylic acid 344152 5-(3-((S)-2-(4-(4-chlorophenyl)-3-hydroxybutyl)-5-oxopyrrolidin-1-yl)propyl)thiophene-2-carboxylic acid 344157 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-4-methylpyridin-2(1H)-one 344160 4-(3-((S)-2-((R)-3-hydroxy-4-(3-(trifluoromethyl)phenyl)butyl)-5-oxopyrrolidin-1-yl)propyl)benzoic acid 344161 5-(3-((S)-2-((R)-3-hydroxy-4-(3-(trifluoromethyl)phenyl)butyl)-5-oxopyrrolidin-1-yl)propyl)thiophene-2-carboxylic acid 344168 7-((S)-2-((R)-4-(3-cyanophenyl)-3-hydroxybutyl)-5-oxopyrrolidin-1-yl)heptanoic acid 344172 1-(4-(4-(2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl)piperazin-1-yl)butyl)-5-chloropyridin-2(1H)-one 344189 6-(azepan-1-yl)-N4,2-dicyclopropylpyrimidine-4,5-diamine 344201 6-(azepan-1-yl)-2-cyclopropyl-5-methyl-N-(1-methylcyclopropyl)pyrimidin-4-amine 344202 (+,)-6-(azepan-1-yl)-2-cyclopropyl-5-methyl-N-(2-methylcyclopropyl)pyrimidin-4-amine 344216 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-((3,4-dihydroisoquinolin-2(1H)-yl)methyl)pyrimidine-2,4-diamine 344230 2-(4-(piperidin-1-yl)butyl)-2H-isoindole-1-carbonitrile 344231 2-(5-(piperidin-1-yl)pentyl)-2H-isoindole-1-carbonitrile 344232 2-(6-(piperidin-1-yl)hexyl)-2H-isoindole-1-carbonitrile 344234 6-(azepan-1-yl)-N-cyclopropyl-2-isopropyl-5-methylpyrimidin-4-amine 344239 7-nitro-N-(4-(piperidin-1-yl)butyl)benzo[c][1,2,5]oxadiazol-4-amine 344240 7-nitro-N-(5-(piperidin-1-yl)pentyl)benzo[c][1,2,5]oxadiazol-4-amine 344241 6-(azepan-1-yl)-N-cyclopropyl-2-(cyclopropylmethyl)-5-methylpyrimidin-4-amine 344242 N,2-dicyclopropyl-6-(3,4-dihydroisoquinolin-2(1H)-yl)-5-methylpyrimidin-4-amine 344243 6-(azepan-1-yl)-2-benzyl-N-cyclopropyl-5-methylpyrimidin-4-amine 344251 N,2-dicyclopropyl-5-methoxy-6-thiomorpholinopyrimidin-4-amine 344259 4-(azepan-1-yl)-2-cyclopropyl-5,6,7,8-tetrahydropyrido[2,3-d]pyrimidine 344260 (S)-N-(4-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)phenyl)methanesulfonamide 344261 (S)-1-(5-(4-(2H-tetrazol-5-yl)phenyl)pyridin-3-yloxy)-3-(1H-indol-3-yl)propan-2-amine 344268 4-(azepan-1-yl)-2-cyclopropyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b]azepine 344284 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-ethyl-N4-methylpyrimidine-2,4-diamine 344287 N4-(2,6-difluorobenzyl)-N6,2-dicyclopropyl-5-methylpyrimidine-4,6-diamine 344288 N4,2-dicyclopropyl-5-methyl-N6-(thiophen-2-ylmethyl)pyrimidine-4,6-diamine 344289 N4,2-dicyclopropyl-5-methyl-N6-(2-(thiophen-2-yl)ethyl)pyrimidine-4,6-diamine 344291 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-ethyl-N4,N4-dimethylpyrimidine-2,4-diamine 344292 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-N4,6-diethylpyrimidine-2,4-diamine 344295 6-(azepan-1-yl)-2-cyclobutyl-N-cyclopropyl-5-methylpyrimidin-4-amine 344296 6-(azepan-1-yl)-2-cyclopentyl-N-cyclopropyl-5-methylpyrimidin-4-amine 344308 7-(pyridin-2-yl)-N-m-tolyl-7H-pyrrolo[2,3-d]pyrimidin-2-amine 344314 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-heptylpyrimidine-2,4-diamine 344315 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-octylpyrimidine-2,4-diamine 344322 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-cyclopropylpyrimidine-2,4-diamine 344330 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-(isopentyloxymethyl)pyrimidine-2,4-diamine 344331 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-(methoxymethyl)pyrimidine-2,4-diamine 344342 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-((isopentylamino)methyl)pyrimidine-2,4-diamine 344346 3-(1H-benzo[d]imidazol-2-yl)-4-hydroxyquinolin-2(1H)-one 344348 5-bromo-N4-(pyridin-2-yl)-N2-(3,4,5-trimethoxyphenyl)pyrimidine-2,4-diamine 344350 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-((cyclopropylamino)methyl)pyrimidine-2,4-diamine 344351 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-N4,N4,6-triethylpyrimidine-2,4-diamine 344352 1-(5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)pyridin-2-yl)-3-phenylurea 344353 (S)-N4-(4-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)phenyl)pyrimidine-2,4-diamine 344354 4-amino-3-(1H-benzo[d]imidazol-2-yl)quinolin-2(1H)-one 344360 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-6-ethyl-N4-propylpyrimidine-2,4-diamine 344361 5-(4-(4-(methylsulfonyl)benzylamino)phenyl)-N4-butyl-6-ethylpyrimidine-2,4-diamine 344362 (S)-N-(4-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)phenyl)pyrimidin-2-amine 344363 (S)-1-(1H-indol-3-yl)-3-(5-(isoquinolin-6-yl)pyridin-3-yloxy)propan-2-amine 344368 (2R)-1-(1H-indol-3-yl)-3-(5-(isoquinolin-6-yl)pyridin-3-yloxy)propan-2-amine 344371 2-(4-(4-(3-methoxyphenyl)piperazin-1-yl)butyl)-4-methyl-1,2,4-triazine-3,5(2H,4H)-dione 344408 1-(4-amino-5-chloro-2-methoxyphenyl)-3-(5-cyanopyrazin-2-yl)urea 344409 1-(5-chloro-4-(2-(dimethylamino)acetamido)-2-methoxyphenyl)-3-(5-cyanopyrazin-2-yl)urea 344411 (S)-3-(1H-indol-3-yl)-N1-(5-(isoquinolin-5-yloxy)pyridin-3-yl)propane-1,2-diamine 344417 (S)-N3-(2-amino-3-(1H-indol-3-yl)propyl)-N5-(isoquinolin-5-yl)pyridine-3,5-diamine 344418 (S)-1-(1H-indol-3-yl)-3-(2-(pyridin-4-yl)-1,7-naphthyridin-5-yloxy)propan-2-amine 344425 N-{2-[2-(5-bromo-2-methoxy-phenyl)-ethyl]-3-fluoro-benzoyl}-N'-(4-piperidin-1-yl-butyl)-guanidine 344426 N-{2-[2-(5-bromo-2-methoxy-phenyl)-ethyl]-3-fluoro-benzoyl}-N'-[4-(octahydro-isoquinolin-2-yl)-butyl]-guanidine 344432 N-(2-chlorophenyl)-7-(pyridin-2-yl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 344433 N-{2-[2-(5-bromo-2-methoxy-phenyl)-ethyl]-3-fluoro-benzoyl}-N'-[4-(3,4-dihydro-1H-isoquinolin-2-yl)-butyl]-guanidine 344440 N-(2-bromophenyl)-7-(pyridin-2-yl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 344441 7-(pyridin-2-yl)-N-(2-(trifluoromethyl)phenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 344509 4-((5-methyl-5H-[1,3]dioxolo[4,5-f]indol-7-yl)methylene)-3-(pyrazin-2-yl)-1H-pyrazol-5(4H)-one 344530 (2S)-1-phenyl-3-(5-(4-(pyridin-4-yl)thiazol-2-yl)pyridin-3-yloxy)propan-2-amine 344531 (2S)-1-phenyl-3-(5-(4-(pyridin-3-yl)thiazol-2-yl)pyridin-3-yloxy)propan-2-amine 344577 4-((1-methyl-1H-indol-3-yl)methylene)-3-(thiazol-2-yl)-1H-pyrazol-5(4H)-one 344578 4-((5-fluoro-1-methyl-1H-indol-3-yl)methylene)-3-(thiazol-2-yl)-1H-pyrazol-5(4H)-one 344586 4-((5-chloro-1-methyl-1H-indol-3-yl)methylene)-3-(thiazol-2-yl)-1H-pyrazol-5(4H)-one 344587 4-((4-bromo-1-methyl-1H-indol-3-yl)methylene)-3-(thiazol-2-yl)-1H-pyrazol-5(4H)-one 344589 7-(pyridin-3-ylmethyl)-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 344600 (S)-1-(3,4'-bipyridin-5-yloxy)-3-(1H-indol-3-yl)propan-2-amine 344606 ethyl 2-(4-(pyridin-2-ylamino)-2-(3,4,5-trimethoxyphenylamino)pyrimidin-5-yl)acetate 344607 4-amino-3-(3H-imidazo[4,5-b]pyridin-2-yl)-1,7-naphthyridin-2(1H)-one 344627 7-(4-methoxypyridin-3-yl)-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 344628 (S)-1-(1H-indol-3-yl)-3-(5-(2-(pyridin-4-yl)ethynyl)pyridin-3-yloxy)propan-2-amine 344630 (S)-5-(2-amino-3-(1H-indol-3-yl)propoxy)-N-(pyridin-4-yl)pyridin-3-amine 344637 7-(2-chloropyrimidin-4-yl)-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 344638 (S)-5-(2-amino-3-(1H-indol-3-yl)propoxy)-N-(pyridin-3-yl)pyridin-3-amine 344639 (S)-5-(2-amino-3-phenylpropoxy)-N-(pyridin-4-yl)pyridin-3-amine 344640 1-(5-chloro-2-methoxy-4-(2-(2-methoxyethoxy)acetamido)phenyl)-3-(5-cyanopyrazin-2-yl)urea 344643 7-(2-chloropyridin-4-yl)-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 344645 (S)-5-(2-amino-3-phenylpropoxy)-N-(pyridin-3-yl)pyridin-3-amine 344647 2-(2-chloro-4-(3-(5-cyanopyrazin-2-yl)ureido)-5-methoxyphenylamino)-2-oxoethyl acetate 344656 methyl 4-(2-chloro-4-(3-(5-cyanopyrazin-2-yl)ureido)-5-methoxyphenylamino)-4-oxobutanoate 344657 1-(5-chloro-2-methoxy-4-(3-phenylpropanamido)phenyl)-3-(5-cyanopyrazin-2-yl)urea 344665 1-(5-chloro-2-methoxy-4-(4-phenylbutanamido)phenyl)-3-(5-cyanopyrazin-2-yl)urea 344666 1-(5-chloro-2-methoxy-4-(3-methyl-2-phenylpentanamido)phenyl)-3-(5-cyanopyrazin-2-yl)urea 344667 N-(3-methoxyphenyl)-7-(pyridin-2-yl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 344673 2-(3,5-bis(trifluoromethyl)benzyloxy)-1-phenyl-8-aza-bicyclo[3.2.1]octane 344674 2-(3,5-bis(trifluoromethyl)benzyloxy)-1-phenyl-6-(phenylsulfonyl)-8-aza-bicyclo[3.2.1]octane 344675 7-(2-(pyridin-4-yl)ethyl)-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 344677 4-((5-methyl-5H-[1,3]dioxolo[4,5-f]indol-7-yl)methylene)-3-(thiazol-2-yl)-1H-pyrazol-5(4H)-one 344684 2-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-1-phenyl-8-aza-bicyclo[3.2.1]octane 344689 1-(5-chloro-4-(3-ethoxypropanamido)-2-methoxyphenyl)-3-(5-cyanopyrazin-2-yl)urea 344703 1-(5-chloro-2-methoxy-4-(2-(thiophen-3-yl)acetamido)phenyl)-3-(5-cyanopyrazin-2-yl)urea 344704 1-(5-chloro-2-methoxy-4-(4-(thiophen-2-yl)butanamido)phenyl)-3-(5-cyanopyrazin-2-yl)urea 344712 N-(2-methyl-5-(quinoxalin-2-yl)phenyl)-7-(pyridin-2-yl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 344715 (S)-1-(1H-indol-3-yl)-3-(5-(2-(pyridin-3-yl)ethynyl)pyridin-3-yloxy)propan-2-amine 344722 N-{2-[2-(5-bromo-2-methoxy-phenyl)-ethyl]-3-fluoro-benzoyl}-N'-piperidin-4-ylmethyl-guanidine 344723 N-{2-[2-(5-bromo-2-methoxy-phenyl)-ethyl]-3-fluoro-benzoyl}-N'-(1-ethyl-piperidin-4-ylmethyl)-guanidine 344731 N-{2-[2-(5-bromo-2-methoxy-phenyl)-ethyl]-3-chloro-benzoyl}-N'-(4-diethylamino-1-methyl-butyl)-guanidine 344738 N-{2-[2-(5-bromo-2-methoxy-phenyl)-ethyl]-3-fluoro-benzoyl}-N'-isobutyl-guanidine 344739 N-{2-[2-(5-bromo-2-methoxy-phenyl)-ethyl]-3-fluoro-benzoyl}-N'-(2-cyclohexyl-ethyl)-guanidine 344743 N-(3-(methylthio)phenyl)-7-(pyridin-2-yl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 344746 N-{2-[2-(5-bromo-2-methoxy-phenyl)-ethyl]-3-fluoro-benzoyl}-N'-(2-pyrrolidin-1-yl-ethyl)-guanidine 344747 N-{2-[2-(5-bromo-2-methoxy-phenyl)-ethyl]-thiophene-3-carbonyl}-N'-(4-diethylamino-1-methyl-butyl)-guanidine 344756 methyl 8-(2-chloro-4-(3-(5-cyanopyrazin-2-yl)ureido)-5-methoxyphenylamino)-8-oxooctanoate 344763 7-(pyridin-2-yl)-N-o-tolyl-7H-pyrrolo[2,3-d]pyrimidin-2-amine 344766 1-(5-chloro-2-methoxy-4-(3-(4-methoxyphenyl)propanamido)phenyl)-3-(5-cyanopyrazin-2-yl)urea 344767 4-methyl-3-(7-(pyridin-2-yl)-7H-pyrrolo[2,3-d]pyrimidin-2-ylamino)benzamide 344768 N-(2-ethylphenyl)-7-(pyridin-2-yl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 344771 N-[4-(benzyl-methyl-amino)-butyl]-N'-{2-[2-(5-bromo-2-methoxy-phenyl)-ethyl]-3-fluoro-benzoyl}-guanidine 344777 N-{2-[2-(5-bromo-2-methoxy-phenyl)-ethyl]-3-fluoro-benzoyl}-N'-[4-(methyl-naphthalen-1-ylmethyl-amino)-butyl]-guanidine 344783 2-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-1-phenyl-6-(phenylsulfonyl)-8-aza-bicyclo[3.2.1]octane 344791 2-(3,5-bis(trifluoromethyl)benzyloxy)-6-(2-methyl-2H-tetrazol-5-yl)-1-phenyl-8-aza-bicyclo[3.2.1]octane 344792 2-(3,5-bis(trifluoromethyl)benzyloxy)-6-(1-methyl-1H-tetrazol-5-yl)-1-phenyl-8-aza-bicyclo[3.2.1]octane 344794 3-(1H-benzo[d]imidazol-2-yl)-4-hydroxy-1,8-naphthyridin-2(1H)-one 344803 4-amino-5-(1H-benzo[d]imidazol-2-yl)-1-methyl-1H-pyrazolo[3,4-b]pyridin-6(7H)-one 344811 SID4259879 344814 3-(1H-benzo[d]imidazol-2-yl)-4-hydroxy-1,7-naphthyridin-2(1H)-one 344816 N-(2-methoxyphenyl)-7-(pyridin-2-yl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 344817 N-(2-(methylthio)phenyl)-7-(pyridin-2-yl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 344824 4-Amino-3-(6-morpholin-4-ylbenzimidazol-2-yl)hydroquinolin-2-one 344825 4-Amino-3-[6-(4-methylpiperazinyl)benzimidazol-2-yl]hydroquinolin-2-one 344829 4-((5-fluoro-1-methyl-1H-indol-3-yl)methylene)-3-(pyrazin-2-yl)-1H-pyrazol-5(4H)-one 344831 4-amino-3-(5-morpholino-3H-imidazo[4,5-b]pyridin-2-yl)quinolin-2(1H)-one 344832 4-amino-3-(5-(4-methylpiperazin-1-yl)-3H-imidazo[4,5-b]pyridin-2-yl)quinolin-2(1H)-one 344838 4-amino-5-(1H-benzo[d]imidazol-2-yl)thieno[2,3-b]pyridin-6(7H)-one 344839 7-amino-6-(1H-benzo[d]imidazol-2-yl)-3H-imidazo[4,5-b]pyridin-5(4H)-one 344840 4-amino-5-(1H-benzo[d]imidazol-2-yl)-1H-pyrazolo[3,4-b]pyridin-6(7H)-one 344843 N-{2-[2-(5-bromo-2-methoxy-phenyl)-ethyl]-3-chloro-benzoyl}-guanidine 344844 N-{2-[2-(5-bromo-2-methoxy-phenyl)-ethyl]-3-fluoro-benzoyl}-N'-butyl-guanidine 344882 7-(pyridin-2-yl)-N-(3,4,5-trimethoxyphenyl)-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidin-2-amine 344902 N-{2-[2-(5-bromo-2-methoxy-phenyl)-ethyl]-3-fluoro-benzoyl}-N'-(3-piperidin-1-yl-propyl)-guanidine 344930 1-(5-chloro-2-methoxy-4-(3-(3-methoxyphenyl)propanamido)phenyl)-3-(5-cyanopyrazin-2-yl)urea 344949 4-((3,5-dimethyl-1H-pyrrol-2-yl)methylene)-3-(thiazol-2-yl)-1H-pyrazol-5(4H)-one 344950 4-((3,5-dimethyl-1H-pyrrol-2-yl)methylene)-3-(pyrazin-2-yl)-1H-pyrazol-5(4H)-one 344985 4-((3,5-dimethyl-1H-pyrrol-2-yl)methylene)-3-phenyl-1H-pyrazol-5(4H)-one 344994 4-((3,5-dimethyl-1H-pyrrol-2-yl)methylene)-3-(furan-3-yl)-1H-pyrazol-5(4H)-one 344996 (S)-1-(5-(4-fluorophenyl)pyridin-3-yloxy)-3-(1H-indol-3-yl)propan-2-amine 345004 (S)-4-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)benzenamine 345006 4-((5-chloro-1-methyl-1H-indol-3-yl)methylene)-3-(pyrazin-2-yl)-1H-pyrazol-5(4H)-one 345007 4-((5-methoxy-1-methyl-1H-indol-3-yl)methylene)-3-(pyrazin-2-yl)-1H-pyrazol-5(4H)-one 345008 (S)-5-(2-amino-3-(1H-indol-3-yl)propoxy)-N-(pyridin-4-yl)nicotinamide 345015 4-((4-fluoro-1-methyl-1H-indol-3-yl)methylene)-3-(pyrazin-2-yl)-1H-pyrazol-5(4H)-one 345016 4-((4-chloro-1-methyl-1H-indol-3-yl)methylene)-3-(pyrazin-2-yl)-1H-pyrazol-5(4H)-one 345018 (S)-5-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)-1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonitrile 345022 1-(5-chloro-2-methoxy-4-(nicotinamido)phenyl)-3-(5-cyanopyrazin-2-yl)urea 345025 1-(5-chloro-2,4-dimethoxyphenyl)-3-(5-cyanopyrazin-2-yl)urea 345027 1-(5-chloro-4-(isonicotinamido)-2-methoxyphenyl)-3-(5-cyanopyrazin-2-yl)urea 345028 1-(5-chloro-4-formyl-2-methoxyphenyl)-3-(5-cyanopyrazin-2-yl)urea 345035 1-(5-chloro-2-methoxy-4-(piperidin-1-ylmethyl)phenyl)-3-(5-cyanopyrazin-2-yl)urea 345036 1-(5-chloro-4-(2-(dimethylamino)ethoxy)-2-(pyrrolidin-1-yl)phenyl)-3-(5-cyanopyrazin-2-yl)urea 345044 N-[2-(5-bromo-2-methoxy-benzyloxy)-3-fluoro-benzoyl]-N'-(4-diethylamino-1-methyl-butyl)-guanidine 345045 2-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-6-(2-methyl-2H-tetrazol-5-yl)-1-phenyl-8-aza-bicyclo[3.2.1]octane 345049 1-(5-chloro-2-methoxy-4-(2-(4-methoxyphenyl)acetamido)phenyl)-3-(5-cyanopyrazin-2-yl)urea 345050 1-(5-chloro-2-methoxy-4-(2-(4-(methylsulfonyl)phenyl)acetamido)phenyl)-3-(5-cyanopyrazin-2-yl)urea 345054 2-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-6-(1-methyl-1H-tetrazol-5-yl)-1-phenyl-8-aza-bicyclo[3.2.1]octane 345055 1-(5-chloro-2-methoxy-4-(4-phenoxybutanamido)phenyl)-3-(5-cyanopyrazin-2-yl)urea 345057 N-(5-methoxy-2-methylphenyl)-7-(pyridin-2-yl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 345060 2-(3,5-bis(trifluoromethyl)benzyloxy)-6-fluoro-6-(2-methyl-2H-tetrazol-5-yl)-1-phenyl-8-aza-bicyclo[3.2.1]octane 345079 7-(thiazol-2-yl)-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 345088 7-(4-fluoropyridin-3-yl)-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 345089 7-(4-chloropyridin-3-yl)-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 345093 7-(pyridin-2-yl)-N-(2,4,6-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 345094 (S)-N-(5-(2-amino-3-phenylpropoxy)pyridin-3-yl)isonicotinamide 345100 7-(pyridin-3-yl)-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 345101 7-(pyridin-4-yl)-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 345110 8-(pyridin-2-yl)-2-(3,4,5-trimethoxyphenylamino)-5,6,7,8-tetrahydropyrido[2,3-d]pyrimidin-7-ol 345111 8-(pyridin-2-yl)-N-(3,4,5-trimethoxyphenyl)-5,6,7,8-tetrahydropyrido[2,3-d]pyrimidin-2-amine 345113 (S)-4-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)benzonitrile 345125 1-(5-chloro-4-(furan-2-carboxamido)-2-methoxyphenyl)-3-(5-cyanopyrazin-2-yl)urea 345126 1-(5-chloro-2-methoxy-4-(thiophene-2-carboxamido)phenyl)-3-(5-cyanopyrazin-2-yl)urea 345133 N-{2-[2-(5-bromo-2-methoxy-phenyl)-ethyl]-3-fluoro-benzoyl}-N'-(4-diethylamino-1-methyl-butyl)-N''-isopropyl-guanidine 345139 N-{2-[2-(5-bromo-2-methoxy-phenyl)-ethyl]-3-fluoro-benzoyl}-N'-(4-diethylamino-1-methyl-butyl)-N''-phenyl-guanidine 345140 4-amino-3-(6-morpholino-1H-benzo[d]imidazol-2-yl)-1,6-naphthyridin-2(1H)-one 345141 4-amino-3-(6-(4-methylpiperazin-1-yl)-1H-benzo[d]imidazol-2-yl)-1,5-naphthyridin-2(1H)-one 345146 N-{2-[2-(5-bromo-2-methoxy-phenyl)-ethyl]-3-fluoro-benzoyl}-N'-(4-diethylamino-1-methyl-butyl)-N''-methyl-guanidine 345147 2-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-6-fluoro-6-(2-methyl-2H-tetrazol-5-yl)-1-phenyl-8-aza-bicyclo[3.2.1]octane 345149 4-amino-3-(3H-imidazo[4,5-b]pyridin-2-yl)quinolin-2(1H)-one 345156 2-((S)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-1-phenyl-8-aza-bicyclo[3.2.1]octane 345162 N-(4-iodo-2-methylphenyl)-7-(pyridin-2-yl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 345170 7-(pyridin-2-yl)-N-(5,6,7,8-tetrahydronaphthalen-1-yl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 345183 4-amino-3-(1H-benzo[d]imidazol-2-yl)-1,7-naphthyridin-2(1H)-one 345187 1-(5-chloro-2-methoxy-4-nitrophenyl)-3-(5-cyanopyrazin-2-yl)urea 345192 4-amino-3-(6-morpholino-1H-benzo[d]imidazol-2-yl)-1,7-naphthyridin-2(1H)-one 345193 4-amino-3-(6-(4-methylpiperazin-1-yl)-1H-benzo[d]imidazol-2-yl)-1,7-naphthyridin-2(1H)-one 345196 N-{2-[2-(5-bromo-2-methoxy-phenyl)-ethyl]-3-fluoro-benzoyl}-N'-[3-(4-methyl-piperazin-1-yl)-propyl]-guanidine 345197 N-{2-[2-(5-bromo-2-methoxy-phenyl)-ethyl]-3-fluoro-benzoyl}-N'-(3-cyclohexylamino-propyl)-guanidine 345204 N-{2-[2-(5-bromo-2-methoxy-phenyl)-ethyl]-3-fluoro-benzoyl}-N'-(4-diethylamino-1-methyl-butyl)-guanidine 345216 (S)-4-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)benzoic acid 345219 N-(2-fluorophenyl)-7-(pyridin-2-yl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 345222 (S)-4-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)benzamide 345224 4-((4-bromo-1-methyl-1H-indol-3-yl)methylene)-3-(pyrazin-2-yl)-1H-pyrazol-5(4H)-one 345225 4-((4-methoxy-1-methyl-1H-indol-3-yl)methylene)-3-(pyrazin-2-yl)-1H-pyrazol-5(4H)-one 345227 N-(5-iodo-2-methylphenyl)-7-(pyridin-2-yl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 345233 1-(5-chloro-2-methoxy-4-(2-(pyridin-3-yl)acetamido)phenyl)-3-(5-cyanopyrazin-2-yl)urea 345247 1-(5-chloro-4-(2-(2-(dimethylamino)ethoxy)ethoxy)-2-(pyrrolidin-1-yl)phenyl)-3-(5-cyanopyrazin-2-yl)urea 345248 1-(5-chloro-4-(2-((2-(2-(dimethylamino)ethoxy)ethyl)(methyl)amino)ethoxy)-2-(pyrrolidin-1-yl)phenyl)-3-(5-cyanopyrazin-2-yl)urea 345250 N-(4-(chlorodifluoromethoxy)phenyl)-5-(2-(2-(pyridin-4-yl)ethyl)pyridin-3-yl)-1,3,4-oxadiazol-2-amine 345252 N-(4-methyl-3-(trifluoromethyl)phenyl)-5-(2-(2-(pyridin-4-yl)ethyl)pyridin-3-yl)-1,3,4-oxadiazol-2-amine 345257 5-(2-(2-(pyridin-4-yl)ethyl)pyridin-3-yl)-N-(4-(trifluoromethoxy)phenyl)-1,3,4-oxadiazol-2-amine 345258 5-(2-(2-(pyridin-4-yl)ethyl)pyridin-3-yl)-N-m-tolyl-1,3,4-oxadiazol-2-amine 345263 1-(5-cyanopyrazin-2-yl)-3-(4-(((2-(dimethylamino)ethyl)(methyl)amino)methyl)-2-methoxyphenyl)urea 345265 N-(3-methoxyphenyl)-5-(2-(2-(pyridin-4-yl)ethyl)pyridin-3-yl)-1,3,4-oxadiazol-2-amine 345275 N-{2-[2-(2-chloro-phenyl)-ethyl]-3-fluoro-benzoyl}-N'-(4-diethylamino-1-methyl-butyl)-guanidine 345284 5-(2-(2-(pyridin-4-yl)ethyl)pyridin-3-yl)-N-(3-(trifluoromethyl)phenyl)-1,3,4-oxadiazol-2-amine 345293 5-(2-(2-(1H-indazol-5-yl)ethyl)pyridin-3-yl)-N-(3-(trifluoromethyl)phenyl)-1,3,4-oxadiazol-2-amine 345299 1-(5-chloro-4-(pyridin-3-ylmethoxy)-2-(pyrrolidin-1-yl)phenyl)-3-(5-cyanopyrazin-2-yl)urea 345301 5-(2-(2-(pyridin-4-yl)ethyl)pyridin-3-yl)-N-(4-(trifluoromethyl)phenyl)-1,3,4-oxadiazol-2-amine 345306 1-(5-chloro-2-(pyrrolidin-1-yl)-4-((tetrahydrofuran-2-yl)methoxy)phenyl)-3-(5-cyanopyrazin-2-yl)urea 345307 1-(5-chloro-4-(4-methylpiperazin-1-yl)-2-(tetrahydrofuran-3-yloxy)phenyl)-3-(5-cyanopyrazin-2-yl)urea 345308 N-(4-(chlorodifluoromethoxy)phenyl)-5-(3-(2-(pyridin-4-yl)ethyl)pyridin-4-yl)-1,3,4-oxadiazol-2-amine 345309 5-(3-(2-(pyridin-4-yl)ethyl)pyridin-4-yl)-N-(4-(trifluoromethoxy)phenyl)-1,3,4-oxadiazol-2-amine 345313 1-(5-chloro-2-(2-(dimethylamino)ethoxy)-4-(4-methylpiperazin-1-yl)phenyl)-3-(5-cyanopyrazin-2-yl)urea 345325 N-(3,4-dichlorophenyl)-5-(2-(2-(pyridin-4-yl)ethyl)pyridin-3-yl)-1,3,4-oxadiazol-2-amine 345326 N-(3,4-dimethoxyphenyl)-5-(2-(2-(pyridin-4-yl)ethyl)pyridin-3-yl)-1,3,4-oxadiazol-2-amine 345341 N-(4-tert-butylphenyl)-5-(4-(2-(pyridin-4-yl)ethyl)pyridin-3-yl)-1,3,4-oxadiazol-2-amine 345346 1-(5-chloro-4-(4-methylpiperazin-1-yl)-2-(pyridin-3-ylmethoxy)phenyl)-3-(5-cyanopyrazin-2-yl)urea 345355 N-{2-[2-(5-bromo-2-chloro-phenyl)-ethyl]-3-fluoro-benzoyl}-N'-(4-diethylamino-1-methyl-butyl)-guanidine 345356 N-(4-diethylamino-1-methyl-butyl)-N'-{2-[2-(3,5-dimethoxy-phenyl)-ethyl]-3-fluoro-benzoyl}-guanidine 345357 N-(4-diethylamino-1-methyl-butyl)-N'-[3-fluoro-2-(2-naphthalen-1-yl-ethyl)-benzoyl]-guanidine 345364 5-(2-(2-(quinolin-5-yl)ethyl)pyridin-3-yl)-N-(3-(trifluoromethyl)phenyl)-1,3,4-oxadiazol-2-amine 345375 5-(3-(2-(pyridin-4-yl)ethyl)pyridin-4-yl)-N-(3-(trifluoromethyl)phenyl)-1,3,4-oxadiazol-2-amine 345380 5-(3-(2-(pyridin-4-yl)ethyl)pyridin-4-yl)-N-(4-(trifluoromethyl)phenyl)-1,3,4-oxadiazol-2-amine 345381 1-(5-cyanopyrazin-2-yl)-3-(2-methoxy-4-((4-methylpiperazin-1-yl)methyl)phenyl)urea 345384 1-(5-cyanopyrazin-2-yl)-3-(2-methoxy-4-(pyrrolidin-1-ylmethyl)phenyl)urea 345385 N-(4-diethylamino-1-methyl-butyl)-N'-[3-fluoro-2-(2-naphthalen-2-yl-ethyl)-benzoyl]-guanidine 345388 5-(4-(2-(pyridin-4-yl)ethyl)pyridin-3-yl)-N-(3-(trifluoromethyl)phenyl)-1,3,4-oxadiazol-2-amine 345392 N-(5-(2-(2-(pyridin-4-yl)ethyl)pyridin-3-yl)-1,3,4-oxadiazol-2-yl)quinolin-3-amine 345396 N-(4-tert-butylphenyl)-5-(2-(2-(pyridin-4-yl)ethyl)pyridin-3-yl)-1,3,4-oxadiazol-2-amine 345397 N-(4-(chlorodifluoromethoxy)phenyl)-5-(4-(2-(pyridin-4-yl)ethyl)pyridin-3-yl)-1,3,4-oxadiazol-2-amine 345399 5-(4-(2-(pyridin-4-yl)ethyl)pyridin-3-yl)-N-(4-(trifluoromethoxy)phenyl)-1,3,4-oxadiazol-2-amine 345400 5-(4-(2-(pyridin-4-yl)ethyl)pyridin-3-yl)-N-(4-(trifluoromethyl)phenyl)-1,3,4-oxadiazol-2-amine 345401 N-(benzo[d][1,3]dioxol-5-ylmethyl)-5-(2-(2-(pyridin-4-yl)ethyl)pyridin-3-yl)-1,3,4-oxadiazol-2-amine 345402 biphenyl-4-yl-{5-[2-(2-pyridin-4-yl-ethyl)-pyridin-3-yl]-[1,3,4]oxadiazol-2-yl}-amine 345406 N-(4-isopropylphenyl)-5-(2-(2-(pyridin-4-yl)ethyl)pyridin-3-yl)-1,3,4-oxadiazol-2-amine 345407 N-(4-tert-butylphenyl)-5-(3-(2-(pyridin-4-yl)ethyl)pyridin-4-yl)-1,3,4-oxadiazol-2-amine 345410 N-(4-isopropylphenyl)-5-(3-(2-(pyridin-4-yl)ethyl)pyridin-4-yl)-1,3,4-oxadiazol-2-amine 345411 5-(2-(2-(pyridin-4-yl)ethyl)pyridin-3-yl)-N-(3-(trifluoromethoxy)phenyl)-1,3,4-oxadiazol-2-amine 345417 5-(3-(2-(pyridin-4-yl)ethyl)pyridin-4-yl)-N-(3-(trifluoromethoxy)phenyl)-1,3,4-oxadiazol-2-amine 345418 5-(4-(2-(pyridin-4-yl)ethyl)pyridin-3-yl)-N-(3-(trifluoromethoxy)phenyl)-1,3,4-oxadiazol-2-amine 345419 1-(5-chloro-4-(2-(dimethylamino)ethoxy)-2-((3-methyloxetan-3-yl)methoxy)phenyl)-3-(5-cyanopyrazin-2-yl)urea 345420 1-(5-cyanopyrazin-2-yl)-3-(4-formyl-2-methoxyphenyl)urea 345423 1-(5-cyanopyrazin-2-yl)-3-(2-methoxy-4-(piperidin-1-ylmethyl)phenyl)urea 345424 1-(5-cyanopyrazin-2-yl)-3-(2-methoxy-4-(morpholinomethyl)phenyl)urea 345431 (2S,3S,4R,5R)-5-(2-(2-cyclohexenylethynyl)-6-(ethylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345434 (2S,3S,4R,5R)-N-ethyl-5-(6-(ethylamino)-2-(2-(1-hydroxycyclopentyl)ethynyl)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345435 (2S,3S,4R,5R)-N-ethyl-5-(6-(ethylamino)-2-(2-(1-hydroxycyclohexyl)ethynyl)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345438 (2S,3S,4R,5R)-5-(2-((R,S)-3-cyclohexyl-3-hydroxyprop-1-ynyl)-6-(ethylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345439 (2S,3S,4R,5R)-N-ethyl-5-(6-(ethylamino)-2-((R,S)-3-hydroxy-3-phenylprop-1-ynyl)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345442 (2S,3S,4R,5R)-N-ethyl-5-(6-(ethylamino)-2-((R,S)-3-hydroxy-3-(2-methoxyphenyl)prop-1-ynyl)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345444 (2S,3S,4R,5R)-5-(2-(2-(1-aminocyclohexyl)ethynyl)-6-(ethylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345445 N-(4-(3-fluorobenzyloxy)-3-chlorophenyl)pyrimidin-4-amine 345446 (2S,3S,4R,5R)-N-ethyl-5-(6-(ethylamino)-2-(oct-1-ynyl)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345448 N-(4-(3-fluorobenzyloxy)-3-chlorophenyl)-5-ethynylpyrimidin-4-amine 345449 N-(4-(3-fluorobenzyloxy)-3-chlorophenyl)-5-(2-(pyridin-3-yl)ethynyl)pyrimidin-4-amine 345451 (E)-N-(5-(3-(1-acetylpiperazine-4-carbonyl)styryl)thiazol-2-yl)-4-(dimethylamino)benzamide 345452 N-(5-(3-acetamido-5-(1-acetylpiperazine-4-carbonyl)benzylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345453 (E)-N-(5-(4-(4-acetylpiperazin-1-yl)-4-oxobut-2-enylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345454 N-(5-((4-(1-acetylpiperazine-4-carbonyl)oxazol-2-yl)methylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345455 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-4-aminobenzylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345456 N-(5-(3-(1-(2-hydroxyethyl)piperazine-4-carbonyl)benzylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345457 N-(5-(3-(1-acetyl-1,4-diazepane-4-carbonyl)benzylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345462 N-(5-(4-acetamido-3-(1-acetylpiperazine-4-carbonyl)benzylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345463 (2S)-2-[(3'S,6'R)-6'-[(2S)-2-[(2S)-2-(2-{[(2S)-1-{[(2S)-1-[(2S)-2-[(2R)-2-amino-5-[(diaminomethylidene)amino]pentanamido]-5-[(diaminomethylidene)amino]pentanoyl]pyrrolidin-2-yl]carbonyl}-4-hydroxypyrrolidin-2-yl]formamido}acetamido)-3-(thiophen-2-yl)propanamido]-3-hydroxypropanamido]-6'-benzyl-5'-oxo-octahydrospiro[cyclopentane-1,1'-pyrrolo[1,2-a]azepine]-3'-ylformamido]-5-[(diaminomethylidene)amino]pentanoic acid 345468 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-4-nitrobenzylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345471 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-4-chlorobenzylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345499 N-(5-(3-(morpholine-4-carbonyl)benzylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345500 N-(5-(3-(1-(pyrimidin-2-yl)piperazine-4-carbonyl)benzylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345502 (S)-2-amino-3-(4-chlorophenyl)-1-((S)-3-(4-phenyl-1H-imidazol-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)propan-1-one 345503 N-(5-(3-(1-acetylpiperazine-4-carbonyl)benzylthio)-4-phenylthiazol-2-yl)-4-(dimethylamino)benzamide 345508 (S)-2-amino-1-((S)-3-(5-methyl-4-phenyl-1H-imidazol-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)-3-phenylpropan-1-one 345509 (S)-2-amino-3-phenyl-1-((S)-2-(4-phenyl-1H-imidazol-2-yl)piperidin-1-yl)propan-1-one 345510 (S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-1-((S)-3-(4-phenyl-1H-imidazol-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)propan-1-one 345511 4-(dimethylamino)-N-[5-({[3-(dimethylcarbamoyl)phenyl]methyl}sulfanyl)-1,3-thiazol-2-yl]benzamide 345519 4-((S)-2-amino-3-((S)-3-(5-methyl-4-phenyl-1H-imidazol-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)-3-oxopropyl)benzonitrile 345520 N-(4-((S)-2-amino-3-oxo-3-((S)-3-(4-phenyl-1H-imidazol-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)propyl)phenyl)methanesulfonamide 345527 1-((6-(2-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamino)pyrimidin-5-yl)ethynyl)pyridin-2-yl)methyl)-3-(2-(methylsulfonyl)ethyl)urea 345531 (S)-2-amino-3-(4-(hydroxymethyl)phenyl)-1-((S)-3-(4-phenyl-1H-imidazol-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)propan-1-one 345532 (6-(2-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamino)pyrimidin-5-yl)ethynyl)pyridin-2-yl)methanol 345536 N-(4-(3-fluorobenzyloxy)-3-chlorophenyl)-5-(2-(6-(aminomethyl)pyridin-2-yl)ethynyl)pyrimidin-4-amine 345537 1-((6-(2-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamino)pyrimidin-5-yl)ethynyl)pyridin-2-yl)methyl)-3-methylurea 345539 4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)imidazo[1,2-a]pyridin-3-yl)pyrimidin-2-amine 345543 (S)-3-(4-acetylphenyl)-2-amino-1-((S)-3-(4-phenyl-1H-imidazol-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)propan-1-one 345546 (2S,3S,4R,5R)-5-(6-(5-chloro-2-methoxybenzylamino)-9H-purin-9-yl)-3-(aminomethyl)-4-hydroxy-N-methyl-tetrahydrofuran-2-carboxamide 345547 N6-(3-iodobenzyl)-9-(3-deoxy-3-ureido-B-D-ribofuranosyl)adenine 345550 4-((S)-2-amino-3-oxo-3-((S)-3-(4-phenyl-1H-imidazol-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)propyl)benzenesulfonamide 345579 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-4,5-dimethylbenzylthio)thiazol-2-yl)-4-((3,3-dimethylbutan-2-ylamino)methyl)benzamide 345585 4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-imidazo[1,2-a]pyridin-3-yl)-N-methylpyrimidin-2-amine 345586 4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-imidazo[1,2-a]pyridin-3-yl)-N,N-dimethylpyrimidin-2-amine 345591 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-5-aminobenzylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345608 N-(5-(3-(1-acetylpiperazine-4-carbonyl)benzylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345614 N-(5-((4-(1-acetylpiperazine-4-carbonyl)thiazol-2-yl)methylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345615 (S)-2-amino-3-(4-hydroxyphenyl)-1-((S)-2-(4-phenyl-1H-imidazol-2-yl)piperidin-1-yl)propan-1-one 345621 N-(5-((5-(1-acetylpiperazine-4-carbonyl)furan-2-yl)methylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345623 (S)-2-amino-3-phenyl-1-((S)-3-(4-phenyl-1H-imidazol-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)propan-1-one 345634 (2S)-2-[(3'S,6'S)-6'-[(2S)-2-[(2S)-2-(2-{[(2S)-1-{[(2S)-1-[(2S)-2-[(2R)-2-amino-5-[(diaminomethylidene)amino]pentanamido]-5-[(diaminomethylidene)amino]pentanoyl]pyrrolidin-2-yl]carbonyl}-4-hydroxypyrrolidin-2-yl]formamido}acetamido)-3-(thiophen-2-yl)propanamido]-3-hydroxypropanamido]-6'-benzyl-5'-oxo-octahydrospiro[cyclopentane-1,1'-pyrrolo[1,2-a]azepine]-3'-ylformamido]-5-[(diaminomethylidene)amino]pentanoic acid 345659 2-(4-{1-[3-(2-chloro-phenoxy)-benzyl]-piperidin-4-ylcarbamoyl}-4-phenyl-piperidin-1-yl)-2-methyl-propionic acid 345660 2-(3-((1-(3-(2-chlorophenoxy)benzyl)piperidin-4-yl)carbamoyl)-3-phenylpyrrolidin-1-yl)-2-methylpropanoic acid 345663 (2S,3S,4R,5R)-N-ethyl-5-(6-(ethylamino)-2-(6-hydroxyhex-1-ynyl)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345664 (2S,3S,4R,5R)-N-ethyl-5-(6-(ethylamino)-2-(4-hydroxybut-1-ynyl)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345668 (2S,3S,4R,5R)-N-ethyl-5-(6-(ethylamino)-2-((R,S)-4-hydroxypent-1-ynyl)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345669 (2S,3S,4R,5R)-N-ethyl-5-(6-(ethylamino)-2-((R,S)-3-hydroxy-3-(2-nitrophenyl)prop-1-ynyl)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345670 (2S,3S,4R,5R)-N-ethyl-5-(6-(ethylamino)-2-(2-(4-methoxyphenyl)ethynyl)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345671 (2S,3S,4R,5R)-N-ethyl-5-(6-(ethylamino)-2-((R)-3-hydroxybut-1-ynyl)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345675 (2S,3S,4R,5R)-N-ethyl-5-(6-(ethylamino)-2-((R,S)-3-hydroxy-3-(3-nitrophenyl)prop-1-ynyl)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345676 (2S,3S,4R,5R)-N-ethyl-5-(6-(ethylamino)-2-(3-phenylprop-1-ynyl)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345677 (2S,3S,4R,5R)-N-ethyl-5-(6-(ethylamino)-2-((S)-3-hydroxybut-1-ynyl)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345684 (R,S)-3-(3-(6-(ethylamino)-9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-2-yl)-1-hydroxyprop-2-ynyl)benzoic acid 345685 N-(4-(3-fluorobenzyloxy)-3-chlorophenyl)-5-(2-(2-aminophenyl)ethynyl)pyrimidin-4-amine 345686 (R,S)-methyl 3-(3-(6-(ethylamino)-9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-2-yl)-1-hydroxyprop-2-ynyl)benzoate 345688 (3-(2-aminopyrimidin-4-yl)-2-(4-fluorophenyl)H-imidazo[1,2-a]pyridin-7-yl)methanol 345691 N-(4-(3-fluorobenzyloxy)-3-chlorophenyl)-5-(2-(3-aminophenyl)ethynyl)pyrimidin-4-amine 345692 N-(4-(3-fluorobenzyloxy)-3-chlorophenyl)-5-(2-(4-aminophenyl)ethynyl)pyrimidin-4-amine 345693 (2S,3S,4R,5R)-N-ethyl-5-(6-(ethylamino)-2-((R,S)-3-hydroxy-3-(3-methoxyphenyl)prop-1-ynyl)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345694 N-(5-((5-(1-acetylpiperazine-4-carbonyl)thiophen-2-yl)methylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345702 N-(3-(2-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamino)pyrimidin-5-yl)ethynyl)phenyl)acetamide 345703 N-(4-(2-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamino)pyrimidin-5-yl)ethynyl)phenyl)acetamide 345708 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-2-methylbenzylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345709 (+/-) 3-phenyl-pyrrolidine-3-carboxylic acid {1-[3-(2-chloro-phenoxy)-benzyl]-piperidin-4-yl}-amide 345712 {4-[7-dimethylaminomethyl-2-(4-fluorophenyl)imidazo[1,2-a]pyridin-3-yl]pyrimidin-2-yl}propylamine 345713 {5-[2-chloro-6-(3-iodo-benzylamino)-purin-9-yl]-4-hydroxy-2-hydroxymethyl-tetrahydro-furan-3-yl}urea 345714 (2S,3S,4R,5R)-5-(6-(3,5-dichlorobenzylamino)-9H-purin-9-yl)-3-amino-4-hydroxy-N-methyl-tetrahydrofuran-2-carboxamide 345715 (2S,3S,4R,5R)-5-(6-(2,5-dimethoxybenzylamino)-9H-purin-9-yl)-3-amino-4-hydroxy-N-methyl-tetrahydrofuran-2-carboxamide 345723 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-4,5-dimethylbenzylthio)thiazol-2-yl)-1H-pyrrole-2-carboxamide 345724 (2S,3S,4R,5R)-N-ethyl-5-(6-(ethylamino)-2-(5-phenylpent-1-ynyl)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345730 (2R,3R,4S,5S)-2-(6-(5-chloro-2-methoxybenzylamino)-9H-purin-9-yl)-4-(aminomethyl)-5-(hydroxymethyl)-tetrahydrofuran-3-ol 345736 (2S,3S,4R,5R)-5-(6-(5-chloro-2-methoxybenzylamino)-9H-purin-9-yl)-3-amino-4-hydroxy-N-methyl-tetrahydrofuran-2-carboxamide 345737 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-4,5-dimethylbenzylthio)thiazol-2-yl)-5-((3,3-dimethylbutan-2-ylamino)methyl)-1H-pyrrole-2-carboxamide 345742 (2S,3S,4R,5R)-N-ethyl-5-(6-(ethylamino)-2-((R,S)-3-hydroxy-3-(4-methoxyphenyl)prop-1-ynyl)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345744 4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-imidazo[1,2-a]pyridin-3-yl)-N-neopentylpyrimidin-2-amine 345745 (2S,3S,4R,5R)-5-(6-(2-(benzyloxy)-5-chlorobenzylamino)-9H-purin-9-yl)-3-amino-4-hydroxy-N-methyl-tetrahydrofuran-2-carboxamide 345751 N-(4-(3-fluorobenzyloxy)-3-chlorophenyl)-5-(2-phenylethynyl)pyrimidin-4-amine 345754 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-4,5-dimethylbenzylthio)thiazol-2-yl)-4-((1-hydroxy-3-methylbutan-2-ylamino)methyl)benzamide 345757 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-4-methylbenzylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345770 3'-{2-[(R)-2-(3-chloro-phenyl)-2-hydroxy-ethylamino]-ethylamino}-biphenyl-3-carboxylic acid 345782 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-5-nitrobenzylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345787 N-(4-((S)-2-amino-3-((S)-3-(5-methyl-4-phenyl-1H-imidazol-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)-3-oxopropyl)phenyl)acetamide 345788 N-(5-(3-(1-(2H-tetrazol-5-yl)piperazine-4-carbonyl)benzylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345796 (S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-1-((S)-3-(5-methyl-4-phenyl-1H-imidazol-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)propan-1-one 345797 (S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-1-((S)-2-(4-phenyl-1H-imidazol-2-yl)piperidin-1-yl)propan-1-one 345803 3-ureido-5-(6-(3-iodobenzylamino)purin-9-yl)-4-hydroxy-tetrahydro-furan-2-carboxylic acid methyl amide 345804 (S)-2-amino-3-(4-fluorophenyl)-1-((S)-3-(5-methyl-4-phenyl-1H-imidazol-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)propan-1-one 345805 4-((S)-2-amino-3-oxo-3-((S)-3-(4-phenyl-1H-imidazol-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)propyl)benzoic acid 345810 4-((S)-2-amino-3-oxo-3-((S)-3-(4-phenyl-1H-imidazol-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)propyl)-3,5-dimethylbenzamide 345812 4-((S)-2-amino-3-oxo-3-((S)-3-(4-phenyl-1H-imidazol-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)propyl)benzamide 345813 4-((S)-2-amino-3-oxo-3-((S)-2-(4-phenyl-1H-imidazol-2-yl)piperidin-1-yl)propyl)benzamide 345815 4-((S)-2-amino-3-oxo-3-((S)-2-(4-phenyl-1H-imidazol-2-yl)piperidin-1-yl)propyl)-3,5-dimethylbenzamide 345816 N-(4-(3-fluorobenzyloxy)-3-chlorophenyl)-5-(2-(pyrimidin-2-yl)ethynyl)pyrimidin-4-amine 345832 N-(4-(3-fluorobenzyloxy)-3-chlorophenyl)-5-(2-(pyridin-2-yl)ethynyl)pyrimidin-4-amine 345835 (S)-2-amino-3-(4-methoxyphenyl)-1-((S)-3-(5-methyl-4-phenyl-1H-imidazol-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)propan-1-one 345836 (S)-2-amino-3-(4-aminophenyl)-1-((S)-3-(5-methyl-4-phenyl-1H-imidazol-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)propan-1-one 345837 5-(2-(1H-pyrazol-3-yl)ethynyl)-N-(4-(3-fluorobenzyloxy)-3-chlorophenyl)pyrimidin-4-amine 345838 N-(4-(3-fluorobenzyloxy)-3-chlorophenyl)-5-(2-(2-aminopyrimidin-4-yl)ethynyl)pyrimidin-4-amine 345842 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-5-methylbenzylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345847 (2S,3S,4R,5R)-N-ethyl-5-(6-(ethylamino)-2-(hex-1-ynyl)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345849 N-(5-(5-(1-acetylpiperazine-4-carbonyl)-2-methylbenzylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345856 1-[3-(2-methoxy-phenoxy)-benzyl]-4-[(4-phenyl-piperidine-4-carbonyl)-amino]-piperidine-4-carboxylic acid 345861 1-[3-(2-chlorophenoxy)benzyl]-4-{[(1-ethyl-4-phenylpiperidin-4-yl)carbonyl]amino} piperidine-4-carboxylic acid 345862 4-(7-(aminomethyl)-2-(4-fluorophenyl)H-imidazo[1,2-a]pyridin-3-yl)pyrimidin-2-amine 345863 4-(2-(4-fluorophenyl)-7-((methylamino)methyl)H-imidazo[1,2-a]pyridin-3-yl)pyrimidin-2-amine 345867 N-(5-(3-(4-methylpiperidine-1-carbonyl)benzylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345873 (2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carbohydrazide 345874 N-(6-(2-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamino)pyrimidin-5-yl)ethynyl)pyridin-2-yl)acetamide 345875 (4-(2-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamino)pyrimidin-5-yl)ethynyl)thiazol-2-yl)methanol 345876 (2S,3S,4R,5R)-5-(6-(5-chloro-2-(2-morpholino-2-oxoethoxy)benzylamino)-9H-purin-9-yl)-3-amino-4-hydroxy-N-methyl-tetrahydrofuran-2-carboxamide 345879 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-4,5-dimethylbenzylthio)thiazol-2-yl)-4-(hydroxymethyl)benzamide 345880 (5-(2-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamino)pyrimidin-5-yl)ethynyl)furan-2-yl)methanol 345888 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-4-methoxybenzylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345892 (2S,3S,4R,5R)-5-(2-(dec-1-ynyl)-6-(ethylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345895 Tyr-D-Ala-Gly-Trp-NMeNle-Asp-Phe-NH2 345903 (2S,3S,4R,5R)-N-ethyl-5-(6-(ethylamino)-2-((R)-3-hydroxyoct-1-ynyl)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345904 (2S,3S,4R,5R)-N-ethyl-5-(6-(ethylamino)-2-((S)-3-hydroxyoct-1-ynyl)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345912 (2S,3S,4R,5R)-5-(2-((R,S)-3-cyclopentyl-3-hydroxyprop-1-ynyl)-6-(ethylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345913 (2-(4-fluorophenyl)-3-(pyrimidin-4-yl)H-imidazo[1,2-a]pyridin-7-yl)-N,N-dimethylmethanamine 345914 3-(2-aminopyrimidin-4-yl)-2-(4-fluorophenyl)H-imidazo[1,2-a]pyridine-7-carbonitrile 345915 N-(3-(2-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamino)pyrimidin-5-yl)ethynyl)phenyl)methanesulfonamide 345921 (2S,3S,4R,5R)-N-ethyl-5-(6-(ethylamino)-2-iodo-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 345922 3-(2-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamino)pyrimidin-5-yl)ethynyl)-N-methylbenzamide 345927 N-(3-(2-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamino)pyrimidin-5-yl)ethynyl)benzyl)acetamide 345937 Tyr-D-Ala-Gly-D-Trp-NMeNle-Asp-Phe-NH2 345938 N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1-(2-fluorophenyl)ethyl)piperazin-1-yl)-1-oxopropan-2-yl)-2-(isoindolin-1-yl)acetamide 345940 Tyr-D-Ala-Gly-D-Trp-Nle-Asp-Phe-NH2 345941 (2-(4-fluorophenyl)-3-(2-methoxypyrimidin-4-yl)H-imidazo[1,2-a]pyridin-7-yl)-N,N-dimethylmethanamine 345942 4-[2-(4-Fluorophenyl)-7-piperidin-4-ylimidazo-[1,2-a]pyridin-3-yl]piperidin-2-ylamine 345943 N-(3-(2-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamino)pyrimidin-5-yl)ethynyl)phenyl)-3-(methylsulfonyl)propanamide 345948 4-(2-(4-fluorophenyl)-7-(1-methylpiperidin-4-yl)imidazo[1,2-a]pyridin-3-yl)pyrimidin-2-amine 345949 4-(7-chloro-2-(4-fluorophenyl)H-imidazo[1,2-a]pyridin-3-yl)pyrimidin-2-amine 345951 methyl 5-(3-(2-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamino)pyrimidin-5-yl)ethynyl)phenylamino)-5-oxopentanoate 345952 (R)-1-((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)piperidine-2-carboxamide 345955 4-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-ylamino)-6-chloroquinolin-2(1H)-one 345956 (E)-6-chloro-4-(1-cinnamylpiperidin-4-ylamino)-1-methylquinolin-2(1H)-one 345962 4-((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)morpholine-3-carboxamide 345963 (S)-2-(((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)(methyl)amino)-3-methoxypropanamide 345964 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-4,5-dimethylbenzylthio)thiazol-2-yl)-4-(piperazin-1-yl)benzamide 345969 (R)-2-(((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)(methyl)amino)-N,N-dimethylpropanamide 345977 (2S,3S,4R,5R)-5-(6-(5-chloro-2-(2-oxo-2-(piperazin-1-yl)ethoxy)benzylamino)-9H-purin-9-yl)-3-amino-4-hydroxy-N-methyl-tetrahydrofuran-2-carboxamide 345985 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-5-methoxybenzylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345987 (2S,3S,4R,5R)-5-(6-(2,5-dimethoxybenzylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyl-tetrahydrofuran-2-carboxamide 345988 (2S,4R,5R)-4-hydroxy-N-methyl-5-(6-(methylamino)-9H-purin-9-yl)-tetrahydrofuran-2-carboxamide 345989 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-5-chlorobenzylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 345992 (2S,3S,4R,5R)-5-(6-(3,5-dichlorobenzylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyl-tetrahydrofuran-2-carboxamide 345994 (2S,3S,5R)-3-hydroxy-N-methyl-5-(6-(methylamino)-9H-purin-9-yl)-tetrahydrofuran-2-carboxamide 345996 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-4,5-dimethylbenzylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 346001 N-benzyl-4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-imidazo[1,2-a]pyridin-3-yl)pyrimidin-2-amine 346002 2-(2-((9-((2R,3R,4S,5S)-4-amino-3-hydroxy-5-(methylcarbamoyl)-tetrahydrofuran-2-yl)-9H-purin-6-ylamino)methyl)-4-chlorophenoxy)acetic acid 346003 (2S,3S,4R,5R)-5-(6-(2-(2-amino-2-oxoethoxy)-5-chlorobenzylamino)-9H-purin-9-yl)-3-amino-4-hydroxy-N-methyl-tetrahydrofuran-2-carboxamide 346010 (2S,3S,4R,5R)-5-(6-(5-chloro-2-(2-oxo-2-(piperidin-1-yl)ethoxy)benzylamino)-9H-purin-9-yl)-3-amino-4-hydroxy-N-methyl-tetrahydrofuran-2-carboxamide 346023 3-azido-5-(6-(3-iodobenzylamino)purin-9-yl)-4-hydroxy-tetrahydro-furan-2-carboxylic acid methyl amide 346026 4-(4-cyano-phenoxymethyl)-6-methyl-thieno[2,3-b]pyridine-2-carboxylic acid amide 346027 4-(4-methoxy-phenoxymethyl)-6-methyl-thieno[2,3-b]pyridine-2-carboxylic acid amide 346031 N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1-(2-fluorophenyl)ethyl)piperazin-1-yl)-1-oxopropan-2-yl)isoquinoline-3-carboxamide 346032 N-((R)-3-(4-chlorophenyl)-1-(4-(1-(2-chlorophenyl)-2-(diethylamino)ethyl)piperazin-1-yl)-1-oxopropan-2-yl)-2-(1,2,3,4-tetrahydroisoquinolin-1-yl)acetamide 346040 3-amino-6-isobutyl-4-methyl-thieno[2,3-b]pyridine-2-carboxylic acid amide 346041 3-amino-6-butyl-4-methyl-thieno[2,3-b]pyridine-2-carboxylic acid amide 346042 3-amino-6-tert-butyl-2-carbamoyl-thieno[2,3-b]pyridine-4-carboxylic acid ethyl ester 346063 5-amino-2-(4-tert-butyl-phenyl)-oxazole-4-carboxylic acid amide 346064 5-amino-2-(4-tert-butyl-phenyl)-oxazole-4-carboxylic acid amide 346065 5-amino-2-(2-chloro-phenyl)-oxazole-4-carboxylic acid amide 346066 5-amino-2-(2-methoxy-phenyl)-oxazole-4-carboxylic acid amide 346076 amino-4-(4-carbamoyl-phenoxymethyl)-6-methyl-thieno[2,3-b]pyridine-2-carboxylic acid amide 346079 3-(4-(2-(benzyloxy)-5-chlorophenyl)-2-oxo-2,5-dihydrofuran-3-yl)benzoic acid 346084 3-(2-(2-(benzyloxy)-5-chlorophenyl)cyclopent-1-enyl)benzoic acid 346108 6-chloro-9-hydroxy-3-(2-methoxyethyl)-1-methyl-1H-pyrazolo[3,4-b]quinolin-4(9H)-one 346117 4-(6-chloro-9-hydroxy-1-methyl-4-oxo-4,9-dihydro-1H-pyrazolo[3,4-b]quinolin-3-yl)butanoic acid 346130 5-amino-2-p-tolyl-oxazole-4-carboxylic acid amide 346131 5-amino-2-(4-trifluoromethyl-phenyl)-oxazole-4-carboxylic acid amide 346152 N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1-(2-fluorophenyl)ethyl)piperazin-1-yl)-1-oxopropan-2-yl)-2-(2-methylisoindolin-1-yl)acetamide 346153 N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1-(2-fluorophenyl)ethyl)piperazin-1-yl)-1-oxopropan-2-yl)-2-(1,2,3,4-tetrahydroisoquinolin-1-yl)acetamide 346169 6-chloro-1-methyl-4-(1-(naphthalen-2-ylmethyl)piperidin-4-ylamino)quinolin-2(1H)-one 346187 (2S)-2-(2-(4-(4-aminophenyl)-1H-imidazol-1-yl)-6-butylpyrimidin-4-ylamino)-N-(3-ethoxypropyl)-4-methylpentanamide 346191 (2S,3S,4R,5R)-5-(6-(5-chloro-2-(2-(4-(dimethylamino)piperidin-1-yl)-2-oxoethoxy)benzylamino)-9H-purin-9-yl)-3-amino-4-hydroxy-N-methyl-tetrahydrofuran-2-carboxamide 346193 N-{3-[4-(3-carbamoylbenzyl)piperidin-1-yl]propyl}-N-(3,4-dichlorophenyl)-1-(methylsulfonyl)piperidine-4-carboxamide 346198 5-(4-fluoro-phenyl)-3-methylamino-thiophene-2-carboxylic acid amide 346201 N-{3-[4-(4-cyanobenzyl)piperidin-1-yl]propyl}-N-(3,4-dichlorophenyl)-1-(methylsulfonyl)piperidine-4-carboxamide 346202 TAK-220 346204 3-amino-5-(4-chlorophenyl)thiophene-2-carboxamide 346205 3-(3-methyl-ureido)-5-phenyl-thiophene-2-carboxylic acid amide 346206 4-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-ylamino)-6-chloro-1-methylquinazolin-2(1H)-one 346207 6-chloro-1-methyl-4-(1-(quinolin-6-ylmethyl)piperidin-4-ylamino)quinazolin-2(1H)-one 346208 methyl 4-({1-[3-((3,4-Dichlorophenyl){[1-(methylsulfonyl)-piperidin-4-yl]carbonyl}amino)propyl]piperidin-4-yl}methyl)-benzoate 346210 8-octyl-benzolactam-V9 346215 6-chloro-4-(1-(naphthalen-2-ylmethyl)piperidin-4-ylamino)-1-(2,2,2-trifluoroethyl)quinazolin-2(1H)-one 346221 SID47199001 346225 (2S)-N-(3-ethoxypropyl)-4-methyl-2-(6-propyl-2-(4-(4-(trifluoromethoxy)phenyl)-1H-imidazol-1-yl)pyrimidin-4-ylamino)pentanamide 346227 1-(3-phenoxy-benzyl)-piperidine-4-carboxylic acid ethylamide 346228 N-[1-(3-phenoxy-benzyl)-piperidin-4-yl]-propionamide 346239 (2S)-2-(6-butyl-2-(pyridin-3-yl)pyrimidin-4-ylamino)-N-(3-ethoxypropyl)-4-methylpentanamide 346242 N-(3-(4-(4-(methylsulfonyl)benzyl)piperidin-1-yl)propyl)-N-(3,4-dichlorophenyl)-1-(methylsulfonyl)piperidine-4-carboxamide 346243 (2S)-N-(3-ethoxypropyl)-2-(6-ethyl-2-(4-(4-(trifluoromethoxy)phenyl)-1H-imidazol-1-yl)pyrimidin-4-ylamino)-4-methylpentanamide 346244 1-((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)azetidine-3-carboxamide 346252 Tyr-D-Nle-Gly-Trp-Nle-Asp-Phe-NH2 346253 N-(3-(4-(4-fluorobenzyl)piperidin-1-yl)propyl)-N-(3,4-dichlorophenyl)-1-(methylsulfonyl)piperidine-4-carboxamide 346257 Tyr-D-Phe-Gly-D-Trp-Nle-Asp-Phe-NH2 346259 4-({1-[3-((3,4-dichlorophenyl){[1-(methylsulfonyl)piperidin-4-yl]carbonyl}amino)propyl]piperidin-4-yl}methyl)benzoic acid 346262 (R)-2-((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methylamino)propanamide 346263 N-(3-(4-(4-fluorobenzyl)piperidin-1-yl)propyl)-1-acetyl-N-(3,4-dichlorophenyl)piperidine-4-carboxamide 346265 N-{3-[4-(4-carbamoylbenzyl)piperidin-1-yl]propyl}-N-(3,4-dichlorophenyl)-1-(methylsulfonyl)piperidine-4-carboxamide 346266 1-acetyl-N-(3-(4-benzylpiperidin-1-yl)propyl)-N-phenylpiperidine-4-carboxamide 346267 1-acetyl-N-(3,4-dichlorophenyl)-N-(3-{4-[(4-fluorophenyl)sulfanyl]piperidin-1-yl}propyl)piperidine-4-carboxamide 346270 5-phenyl-3-propionylamino-thiophene-2-carboxylic acid amide 346271 2-Benzyloxy-5-chloro-[1,1';2',1'']terphenyl-3''-carboxylic acid 346272 3-(3-(2-(benzyloxy)-5-chlorophenyl)pyridin-2-yl)benzoic acid 346291 6-chloro-9-methoxy-1,3-dimethyl-1H-pyrazolo[3,4-b]quinolin-4(9H)-one 346292 6-chloro-9-ethoxy-1,3-dimethyl-1H-pyrazolo[3,4-b]quinolin-4(9H)-one 346294 3-amino-5-(4-fluoro-phenyl)-thiophene-2-carboxylic acid amide 346297 6-chloro-1,3-dimethyl-9-propoxy-1H-pyrazolo[3,4-b]quinolin-4(9H)-one 346298 6,7-dichloro-9-hydroxy-1-methyl-3-(trifluoromethyl)-1H-pyrazolo[3,4-b]quinolin-4(9H)-one 346299 3-(2-aminoethyl)-6-chloro-9-hydroxy-1-methyl-1H-pyrazolo[3,4-b]quinolin-4(9H)-one 346300 4-(6-chloro-9-hydroxy-1-methyl-4-oxo-4,9-dihydro-1H-pyrazolo[3,4-b]quinolin-3-yl)-N-methylbutanamide 346301 3-amino-5-phenyl-thiophene-2-carboxylic acid amide 346302 5-amino-2-(2-methyl-phenyl)-oxazole-4-carboxylic acid amide 346303 5-amino-2-(3-chloro-phenyl)-oxazole-4-carboxylic acid amide 346304 5-amino-2-(3-methoxy-phenyl)-oxazole-4-carboxylic acid amide 346306 (2S)-2-(6-butyl-2-(4-tert-butyl-1H-imidazol-1-yl)pyrimidin-4-ylamino)-N-(3-ethoxypropyl)-4-methylpentanamide 346307 (2S)-2-(6-butyl-2-(4-phenyl-1H-imidazol-1-yl)pyrimidin-4-ylamino)-N-(3-ethoxypropyl)-4-methylpentanamide 346308 N-(2-(6-chloro-9-hydroxy-1-methyl-4-oxo-4,9-dihydro-1H-pyrazolo[3,4-b]quinolin-3-yl)ethyl)acetamide 346309 (2S)-2-(6-butyl-2-(4-(4-cyanophenyl)-1H-imidazol-1-yl)pyrimidin-4-ylamino)-N-(3-ethoxypropyl)-4-methylpentanamide 346312 6-chloro-1-methyl-4-(1-(naphthalen-2-ylmethyl)piperidin-4-ylamino)quinazolin-2(1H)-one 346313 (2S)-2-(6-butyl-2-(4-(4-nitrophenyl)-1H-imidazol-1-yl)pyrimidin-4-ylamino)-N-(3-ethoxypropyl)-4-methylpentanamide 346317 8-cyclohexyl-2,6-diphenyl-9H-purine 346318 8-cyclohexyl-6-(4-chlorophenyl)-2-phenyl-9H-purine 346322 8-cyclohexyl-6-(4-tolyl)-2-phenyl-9H-purine 346327 Tyr-D-Pro-Gly-Trp-NMeNle-Asp-Phe-NH2 346328 N-((R)-3-(4-chlorophenyl)-1-(4-(1-(2-chlorophenyl)-2-(diethylamino)ethyl)piperazin-1-yl)-1-oxopropan-2-yl)-2-(isoindolin-1-yl)acetamide 346329 Tyr-D-Nle-Gly-D-Trp-NMeNle-Asp-Phe-NH2 346330 N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1-(2-fluorophenyl)ethyl)piperazin-1-yl)-1-oxopropan-2-yl)-1,1-dimethyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 346331 (2S)-2-(6-butyl-2-(4-p-tolyl-1H-imidazol-1-yl)pyrimidin-4-ylamino)-N-(3-ethoxypropyl)-4-methylpentanamide 346337 N-(3-chloro-2-fluorophenyl)-7-methoxy-6-(pyrrolidin-1-ylmethyl)quinazolin-4-amine 346338 2-(((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)(methyl)amino)acetamide 346339 5-amino-2-pyridin-3-yl-oxazole-4-carboxylic acid amide 346348 (R)-2-(((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)(methyl)amino)propanamide 346349 (S)-2-(((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)(methyl)amino)propanamide 346350 (2S,3S,4R,5R)-5-(6-(3-iodobenzylamino)-9H-purin-9-yl)-3-(aminomethyl)-4-hydroxy-N-methyl-tetrahydrofuran-2-carboxamide 346351 N-(((2S,3S,4R,5R)-5-(6-(3-iodobenzylamino)-9H-purin-9-yl)-4-hydroxy-2-(hydroxymethyl)-tetrahydrofuran-3-yl)methyl)acetamide 346354 (R)-1-((4-(3-chloro-4-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)pyrrolidine-2-carboxamide 346355 (S)-1-((4-(3-chloro-4-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)pyrrolidine-2-carboxamide 346356 6-chloro-4-(1-(naphthalen-2-ylmethyl)piperidin-4-ylamino)-1-(pyridin-2-ylmethyl)quinolin-2(1H)-one 346357 (R)-2-(((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)(methyl)amino)-N-methylpropanamide 346361 (S)-1-((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)pyrrolidine-2-carboxamide 346362 1-((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)azetidine-2-carboxamide 346375 Tyr-Pro-Gly-Trp-NMeNle-Asp-Phe-NH2 346385 1-(3-(6-chloro-9-hydroxy-1-methyl-4-oxo-4,9-dihydro-1H-pyrazolo[3,4-b]quinolin-3-yl)propyl)-3-ethylurea 346394 ethyl 2-(6-chloro-9-hydroxy-1-methyl-4-oxo-4,9-dihydro-1H-pyrazolo[3,4-b]quinolin-3-yl)ethylcarbamate 346395 2-(6-chloro-9-hydroxy-3-methyl-4-oxo-4H-pyrazolo[3,4-b]quinolin-1(9H)-yl)acetic acid 346405 (R)-1-((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)pyrrolidine-2-carboxamide 346406 (2R,4R)-1-((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)-4-methoxypyrrolidine-2-carboxamide 346411 (R)-N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1-(2-fluorophenyl)ethyl)piperazin-1-yl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 346412 3-(2-(2-(benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 346413 3-(2-(2-(benzyloxy)-5-chlorophenyl)-1H-pyrrol-1-yl)benzoic acid 346417 4-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-ylamino)-6-methoxy-1-methylquinolin-2(1H)-one 346418 4-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-ylamino)-6-(difluoromethoxy)-1-methylquinolin-2(1H)-one 346419 8-cyclohexyl-6-(3,4-dichlorophenyl)-2-phenyl-9H-purine 346422 8-cyclohexyl-6-(4-methoxyphenyl)-2-phenyl-9H-purine 346423 8-isopropyl-2,6-diphenyl-9H-purine 346424 4-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-ylamino)-6-chloro-1-(2,2,2-trifluoroethyl)quinazolin-2(1H)-one 346425 4-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-ylamino)-6-chloro-1-pentylquinazolin-2(1H)-one 346430 Tyr-D-Nle-Gly-Trp-NMeNle-Asp-Phe-NH2 346432 Tyr-D-Ala-Gly-Trp-Nle-Asp-Phe-NH2 346448 4-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-ylamino)-1-methyl-6-(trifluoromethoxy)quinolin-2(1H)-one 346449 4-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-ylamino)-1-benzyl-6-chloroquinolin-2(1H)-one 346454 4-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-ylamino)-6-chloro-1-(pyridin-4-ylmethyl)quinolin-2(1H)-one 346460 8-cyclopentyl-2,6-diphenyl-9H-purine 346466 3-(4-(2-(benzyloxy)-5-chlorophenyl)pyridin-3-yl)benzoic acid 346484 3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 346485 ethyl 2-(6-chloro-9-hydroxy-3-methyl-4-oxo-4H-pyrazolo[3,4-b]quinolin-1(9H)-yl)acetate 346486 2-(6-chloro-9-hydroxy-3-methyl-4-oxo-4H-pyrazolo[3,4-b]quinolin-1(9H)-yl)-N-methylacetamide 346487 6-chloro-9-hydroxy-1-(2-hydroxyethyl)-3-methyl-1H-pyrazolo[3,4-b]quinolin-4(9H)-one 346488 6-chloro-9-hydroxy-1,3-dimethyl-1H-pyrazolo[3,4-b]quinolin-4(9H)-one 346489 6-chloro-9-hydroxy-1-methyl-3-(trifluoromethyl)-1H-pyrazolo[3,4-b]quinolin-4(9H)-one 346490 6-bromo-9-hydroxy-1,3-dimethyl-1H-pyrazolo[3,4-b]quinolin-4(9H)-one 346493 7-chloro-11-methyl-10-oxy-3,4-dihydro-2H,11H-2,10,11,11a-tetraaza-benzo[b]fluorene-1,5-dione 346494 6-chloro-3-ethyl-9-hydroxy-1-methyl-1H-pyrazolo[3,4-b]quinolin-4(9H)-one 346495 6-chloro-9-hydroxy-1-methyl-3-propyl-1H-pyrazolo[3,4-b]quinolin-4(9H)-one 346496 3-butyl-6-chloro-9-hydroxy-1-methyl-1H-pyrazolo[3,4-b]quinolin-4(9H)-one 346497 Tyr-D-Phe-Gly-Trp-Nle-Asp-Phe-NH2 346508 (2S)-N-(3-ethoxypropyl)-4-methyl-2-(6-methyl-2-(4-(4-(trifluoromethoxy)phenyl)-1H-imidazol-1-yl)pyrimidin-4-ylamino)pentanamide 346511 3-amino-benzo[b]thiophene-2-carboxylic acid amide 346512 4-amino-biphenyl-3-carboxylic acid amide 346513 5-amino-2-thiophen-3-yl-oxazole-4-carboxylic acid amide 346514 5-amino-2-phenyl-oxazole-4-carboxylic acid amide 346516 (2S)-N-(3-ethoxypropyl)-4-methyl-2-(2-(4-(4-(trifluoromethoxy)phenyl)-1H-imidazol-1-yl)pyrimidin-4-ylamino)pentanamide 346519 3-(3-(2-(benzyloxy)-5-chlorophenyl)pyrazin-2-yl)benzoic acid 346521 (2S)-2-(2-(1H-imidazol-1-yl)-6-(octylthio)pyrimidin-4-ylamino)-N-(3-ethoxypropyl)-4-methylpentanamide 346522 (2S)-2-(2-(1H-imidazol-1-yl)-6-octylpyrimidin-4-ylamino)-N-(3-ethoxypropyl)-4-methylpentanamide 346526 N-[1-(3-phenoxy-benzyl)-piperidin-4-yl]-2-phenyl-acetamide 346528 (2S)-N-(3-ethoxypropyl)-2-(6-hexyl-2-(1H-imidazol-1-yl)pyrimidin-4-ylamino)-4-methylpentanamide 346529 6-chloro-9-hydroxy-3-isopropyl-1-methyl-1H-pyrazolo[3,4-b]quinolin-4(9H)-one 346530 5-amino-2-(4-chloro-phenyl)-oxazole-4-carboxylic acid amide 346531 5-amino-2-(4-methoxy-phenyl)-oxazole-4-carboxylic acid amide 346532 4-(8-(benzo[d][1,3]dioxol-5-ylmethyl)-8-aza-bicyclo[3.2.1]octan-3-ylamino)-6-chloro-1-(2,2,2-trifluoroethyl)quinazolin-2(1H)-one 346536 (2S)-2-(6-butyl-2-(4-(4-methoxyphenyl)-1H-imidazol-1-yl)pyrimidin-4-ylamino)-N-(3-ethoxypropyl)-4-methylpentanamide 346537 4-(8-(benzo[d][1,3]dioxol-5-ylmethyl)-8-aza-bicyclo[3.2.1]octan-3-ylamino)-6-chloro-1-methylquinazolin-2(1H)-one 346547 (2S)-2-(6-butyl-2-(4-(4-hydroxyphenyl)-1H-imidazol-1-yl)pyrimidin-4-ylamino)-N-(3-ethoxypropyl)-4-methylpentanamide 346549 N-{3-[4-(2-carbamoylbenzyl)piperidin-1-yl]propyl}-N-(3,4-dichlorophenyl)-1-(methylsulfonyl)piperidine-4-carboxamide 346552 N-(3-{4-[4-(tert-butylcarbamoyl)benzyl]piperidin-1-yl}propyl)-N-(3,4-dichlorophenyl)-1-(methylsulfonyl)piperidine-4-carboxamide 346554 (2S)-N-(3-ethoxypropyl)-4-methyl-2-(6-propyl-2-(4-(3-(trifluoromethoxy)phenyl)-1H-imidazol-1-yl)pyrimidin-4-ylamino)pentanamide 346559 (2S)-N-(3-ethoxypropyl)-4-methyl-2-(6-propyl-2-(4-(2-(trifluoromethoxy)phenyl)-1H-imidazol-1-yl)pyrimidin-4-ylamino)pentanamide 346560 2-(2-(4-phenylpiperazin-1-yl)ethyl)-4-p-tolylphthalazin-1(2H)-one 346564 N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1-(2-fluorophenyl)ethyl)piperazin-1-yl)-1-oxopropan-2-yl)-2-(1-methylisoindolin-1-yl)acetamide 346573 6-chloro-1-ethyl-9-hydroxy-3-methyl-1H-pyrazolo[3,4-b]quinolin-4(9H)-one 346574 6-chloro-9-hydroxy-3-methyl-1-phenyl-1H-pyrazolo[3,4-b]quinolin-4(9H)-one 346595 3-amino-5-(4-methoxyphenyl)thiophene-2-carboxamide 346598 3-(1-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-2-yl)benzoic acid 346599 3-(5-(2-(benzyloxy)-5-chlorophenyl)-1H-pyrazol-1-yl)benzoic acid 346605 2-amino-5-phenylthiophene-3-carboxamide 346606 2-amino-quinoline-3-carboxylic acid amide 346607 5-amino-2-benzthiophene-2-yl-oxazole-4-carboxylic acid amide 346608 3-amino-4-(hydroxymethyl)-6-methylthieno[2,3-b]pyridine-2-carboxamide 346609 3-amino-thieno[2,3-b]pyridine-2-carboxylic acid amide 346610 3-amino-5-methyl-thieno[2,3-b]pyridine-2-carboxylic acid amide 346611 3-amino-4,6-dimethylthieno[2,3-b]pyridine-2-carboxamide 346614 3-(5-(2-(benzyloxy)-5-chlorophenyl)-1H-imidazol-1-yl)benzoic acid 346618 3-amino-6-methyl-4-phenoxymethyl-thieno[2,3-b]pyridine-2-carboxylic acid amide 346620 3-amino-2-carbamoyl-6-methyl-thieno[2,3-b]pyridine-4-carboxylic acid ethyl ester 346623 3-(2-(2-(benzyloxy)-5-chlorophenyl)pyridin-3-yl)benzoic acid 346624 3-(3-(2-(benzyloxy)-5-chlorophenyl)pyridin-4-yl)benzoic acid 346634 N-(3,4-dichlorophenyl)-N-(3-{4-[4-(methylcarbamoyl)benzyl]-piperidin-1-yl}propyl)-1-(methylsulfonyl)piperidine-4-carboxamide 346635 N-{1-[3-(2-methoxy-phenoxy)-benzyl]-piperidin-4-yl}-2-phenyl-acetamide 346638 4-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-ylamino)-6-chloro-1-methyl-2-oxo-1,2-dihydroquinoline-3-carbonitrile 346643 Tyr-D-Phe-Gly-Trp-NMeNle-Asp-Phe-NH2 346646 Tyr-D-Phe-Gly-D-Trp-NMeNle-Asp-Phe-NH2 346648 Tyr-D-Nle-Gly-D-Trp-Nle-Asp-Phe-NH2 346649 1-(4-chloro-phenyl)-cyclohexanecarboxylic acid {1-[3-(2-methoxy-phenoxy)-benzyl]-piperidin-4-yl}-amide 346653 methyl 4-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-ylamino)-6-chloro-1-methyl-2-oxo-1,2-dihydroquinoline-3-carboxylate 346654 4-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-ylamino)-6-chloro-1-methyl-3-(pyrrolidine-1-carbonyl)quinolin-2(1H)-one 346656 4-phenyl-piperidine-4-carboxylic acid {1-[3-(2-methoxy-phenoxy)-benzyl]-piperidin-4-yl}-amide 346666 (2S)-2-(6-butyl-2-(1H-imidazol-1-yl)pyrimidin-4-ylamino)-N-(3-ethoxypropyl)-4-methylpentanamide 346669 (2S)-2-(6-tert-butyl-2-(1H-imidazol-1-yl)pyrimidin-4-ylamino)-N-(3-ethoxypropyl)-4-methylpentanamide 346673 4-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-ylamino)-6-chloro-1-(pyridin-2-ylmethyl)quinolin-2(1H)-one 346674 4-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-ylamino)-6-chloro-2-oxo-1,2-dihydroquinoline-3-carbonitrile 346675 (2S)-2-(6-butyl-2-(4-(4-(trifluoromethoxy)phenyl)-1H-imidazol-1-yl)pyrimidin-4-ylamino)-N-(3-ethoxypropyl)-4-methylpentanamide 346679 (2S)-2-(6-butyl-2-(4-methyl-1H-imidazol-1-yl)pyrimidin-4-ylamino)-N-(3-ethoxypropyl)-4-methylpentanamide 346680 6-chloro-1-methyl-4-(1-(naphthalen-2-ylmethyl)piperidin-4-ylamino)-2-oxo-1,2-dihydroquinoline-3-carbonitrile 346681 (2S)-2-(6-butyl-2-(4-(4-chlorophenyl)-1H-imidazol-1-yl)pyrimidin-4-ylamino)-N-(3-ethoxypropyl)-4-methylpentanamide 346682 (2S)-2-(6-butyl-2-(4-(4-fluorophenyl)-1H-imidazol-1-yl)pyrimidin-4-ylamino)-N-(3-ethoxypropyl)-4-methylpentanamide 346690 2-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-4-p-tolylphthalazin-1(2H)-one 346691 3-(((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)(methyl)amino)pyrrolidin-2-one 346692 2-(4-methoxyphenyl)-6-phenyl-9H-purine 346693 2,6,8-triphenyl-9H-purine 346697 (S)-2-(((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)(isopropyl)amino)propanamide 346703 (2S)-2-(6-butyl-2-(4-(4-(trifluoromethyl)phenyl)-1H-imidazol-1-yl)pyrimidin-4-ylamino)-N-(3-ethoxypropyl)-4-methylpentanamide 346704 (R)-1-((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)-N-methylpyrrolidine-2-carboxamide 346705 (S)-2-(((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)(2-(dimethylamino)ethyl)amino)propanamide 346706 (S)-2-(((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)(methyl)amino)-3-hydroxypropanamide 346707 N-(3,4-dichlorophenyl)-N-[3-(4-{[(4-fluorophenyl)sulfonyl]-amino}piperidin-1-yl)propyl]-1-(methylsulfonyl)piperidine-4-carboxamide 346709 (R)-1-((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)-N,N-dimethylpyrrolidine-2-carboxamide 346710 (S)-2-(((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)(2-methoxyethyl)amino)propanamide 346717 N-(3,4-dichlorophenyl)-N-(3-{4-[(4-fluorobenzoyl)amino]-piperidin-1-yl}propyl)-1-(methylsulfonyl)piperidine-4-carboxamide 346718 8-propyl-2,6-diphenyl-9H-purine 346727 1-acetyl-N-{3-[4-(4-carbamoylbenzyl)piperidin-1-yl]propyl}-N-(3,4-dichlorophenyl)piperidine-4-carboxamide 346734 1-ethyl-4-phenyl-piperidine-4-carboxylic acid {1-[3-(2-methoxy-phenoxy)-benzyl]-piperidin-4-yl}-amide 346737 2,6-bis(4-chlorophenyl)-9H-purine 346738 1-acetyl-N-(3,4-dichlorophenyl)-N-(3-{4-[(4-fluorophenyl)-sulfinyl]piperidin-1-yl}propyl)piperidine-4-carboxamide 346739 1-ethyl-4-phenyl-piperidine-4-carboxylic acid {1-[3-(2-chloro-phenoxy)-benzyl]-piperidin-4-yl}-amide 346740 2,6-bis(4-tolyl)-9H-purine 346741 2,6-bis(4-methoxyphenyl)-9H-purine 346742 2-(4-chlorophenyl)-6-phenyl-9H-purine 346743 1-acetyl-N-(3,4-dichlorophenyl)-N-(3-{4-[(4-fluorophenyl)sulfonyl]piperidin-1-yl}propyl)piperidine-4-carboxamide 346744 2,6-diphenyl-9H-purine 346748 2-tolyl-6-phenyl-9H-purine 346751 1-acetyl-N-(3,4-dichlorophenyl)-N-{3-[4-(4-fluoroanilino)piperidin-1-yl]propyl}piperidine-4-carboxamide 346756 N-(3,4-dichlorophenyl)-N-(3-{4-[4-(dimethylcarbamoyl)benzyl]piperidin-1-yl}propyl)-1-(methylsulfonyl)piperidine-4-carboxamide 346758 (S)-2-(1-((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)pyrrolidin-2-yl)acetamide 346759 1-((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)-4-methylpiperazine-2-carboxamide 346768 4-((ethylamino)methyl)-N-(naphthalen-1-yl)thiazol-2-amine 346769 4-((diethylamino)methyl)-N-(naphthalen-1-yl)thiazol-2-amine 346770 4-isopropyl-N-(naphthalen-1-yl)thiazol-2-amine 346776 methyl 2-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzoate 346777 3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzoic acid 346783 N-(2-(pyrrolidin-1-yl)ethyl)-3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzamide 346784 2-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)phenyl)acetic acid 346785 3-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)phenyl)propanoic acid 346791 N-(2-acetamidoethyl)-3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzamide 346794 N-methyl-2-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzamide 346798 N-(3-(dimethylamino)propyl)-3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzamide 346802 2-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzoic acid 346807 N-(4-(dimethylamino)butyl)-3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzamide 346808 N-(2-hydroxyethyl)-3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzamide 346809 7-m-tolyl-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 346810 N-methyl-3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzenesulfonamide 346811 methyl 2-(2-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)phenyl)acetamido)acetate 346815 N-(3-hydroxypropyl)-3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzamide 346816 N-methyl-3-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)phenyl)propanamide 346822 N-ethyl-3-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)phenyl)propanamide 346823 N-isobutyl-3-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)phenyl)propanamide 346829 2-(2-(5-(4-fluorophenyl)-4-(pyridin-4-yl)-1H-pyrrol-2-yl)pyrrolidin-1-yl)ethanol 346830 (2S)-1-(2-(5-(4-fluorophenyl)-4-(pyridin-4-yl)-1H-pyrrol-2-yl)pyrrolidin-1-yl)propan-2-ol 346831 N-(3-aminopropyl)-6-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)picolinamide 346832 N-(cyanomethyl)-6-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)picolinamide 346837 (2R)-1-(2-(5-(4-fluorophenyl)-4-(pyridin-4-yl)-1H-pyrrol-2-yl)pyrrolidin-1-yl)propan-2-ol 346838 2-(5-(4-fluorophenyl)-4-(pyridin-4-yl)-1H-pyrrol-2-yl)-N-methylpyrrolidine-1-carboxamide 346839 N-(2-cyanoethyl)-6-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)picolinamide 346844 2-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzonitrile 346855 4-tert-butyl-N-(naphthalen-1-yl)thiazol-2-amine 346859 N-(naphthalen-1-yl)-4-neopentylthiazol-2-amine 346860 N-(naphthalen-1-yl)-4-phenylthiazol-2-amine 346861 4-(4-tert-butylphenyl)-N-(naphthalen-1-yl)thiazol-2-amine 346870 N-(4-tert-butylthiazol-2-yl)-1-methyl-1H-indol-4-amine 346871 N-(4-tert-butylthiazol-2-yl)-1-ethyl-1H-indol-4-amine 346873 7-o-tolyl-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 346877 4-tert-butyl-N-(naphthalen-1-yl)oxazol-2-amine 346878 3-(((2-(trifluoromethyl)benzyl)(cyclohexylmethyl)amino)methyl)-N-(2,3-dimethylphenyl)isoxazol-5-amine 346881 (1-((5-(4-fluorophenyl)-4-(pyridin-4-yl)-1H-pyrrol-2-yl)methyl)piperidin-4-yl)methanol 346887 4-(2-(4-fluorophenyl)-5-(pyrrolidin-2-yl)-1H-pyrrol-3-yl)pyridine 346893 (S)-1-((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)pyrrolidine-3-carboxamide 346909 2-(4-(4-phenylpiperazin-1-yl)butyl)-4-p-tolylphthalazin-1(2H)-one 346910 2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-4-p-tolylphthalazin-1(2H)-one 346912 7-p-tolyl-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 346917 2-(4-(4-(2-ethoxyphenyl)piperazin-1-yl)butyl)-4-p-tolylphthalazin-1(2H)-one 346921 2-(7-(4-(3-chlorophenyl)piperazin-1-yl)heptyl)-4-p-tolylphthalazin-1(2H)-one 346927 4-p-tolyl-2-(7-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)heptyl)phthalazin-1(2H)-one 346959 4-(2-(4-fluorophenyl)-5-(1-(4-fluorophenylsulfonyl)pyrrolidin-2-yl)-1H-pyrrol-3-yl)pyridine 346986 N-(2-(dimethylamino)ethyl)-3-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)phenyl)propanamide 346987 2-(2-(4-(2-ethoxyphenyl)piperazin-1-yl)ethyl)-4-p-tolylphthalazin-1(2H)-one 346988 2-(2-(4-(2-isopropoxyphenyl)piperazin-1-yl)ethyl)-4-p-tolylphthalazin-1(2H)-one 346989 4-(2-(4-fluorophenyl)-5-(piperidin-1-ylmethyl)-1H-pyrrol-3-yl)pyridine 346990 4-((5-(4-fluorophenyl)-4-(pyridin-4-yl)-1H-pyrrol-2-yl)methyl)morpholine 346994 methyl 2-(2-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)picolinamido)acetate 347001 3-(6-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)pyridin-2-yl)propanoic acid 347007 N-methyl-3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzamide 347021 benzyl 2-(5-(4-fluorophenyl)-4-(pyridin-4-yl)-1H-pyrrol-2-yl)pyrrolidine-1-carboxylate 347032 2-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)butyl)-4-p-tolylphthalazin-1(2H)-one 347039 (S)-2-(((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)(methyl)amino)-4-methoxybutanamide 347040 (S)-2-(((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)(methyl)amino)-3-(dimethylamino)propanamide 347054 4-(((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)(methyl)amino)-1-methylpiperidine-4-carboxamide 347061 4-(((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)(methyl)amino)-1-isopropylpiperidine-4-carboxamide 347062 3-(((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)(methyl)amino)-1-methylazetidine-3-carboxamide 347064 4-((bis(cyclohexylmethyl)amino)methyl)-N-(naphthalen-1-yl)thiazol-2-amine 347072 3-(((2-(trifluoromethyl)benzyl)(cyclohexylmethyl)amino)methyl)-N-(2,3-dimethylphenyl)-1-methyl-1H-pyrazol-5-amine 347073 6-(((2-(trifluoromethyl)benzyl)(cyclohexylmethyl)amino)methyl)-N-(2,3-dimethylphenyl)pyridin-2-amine 347154 4-tert-butyl-N-(2-isopropylphenyl)thiazol-2-amine 347155 4-tert-butyl-N-(2,3-dimethylphenyl)thiazol-2-amine 347163 4-methyl-N-(naphthalen-1-yl)thiazol-2-amine 347165 4-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzoic acid 347166 4-tert-butyl-N-(5,6,7,8-tetrahydronaphthalen-1-yl)thiazol-2-amine 347167 N-ethyl-3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzamide 347168 7-(4-ethylphenyl)-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 347171 7-(3-(2H-tetrazol-5-yl)phenyl)-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 347172 N-cyclopropyl-3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzamide 347173 N-ethyl-2-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)phenyl)acetamide 347174 N-cyclopropyl-2-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)phenyl)acetamide 347178 N-isobutyl-3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzamide 347179 N-cyclopentyl-3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzamide 347180 N-cyclopentyl-2-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)phenyl)acetamide 347184 N-(2-aminoethyl)-2-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)phenyl)acetamide 347185 N-(3-aminopropyl)-2-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)phenyl)acetamide 347186 methyl 2-(3-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)phenyl)propanamido)acetate 347187 N-methyl-6-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)picolinamide 347192 N-propyl-2-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzenesulfonamide 347197 N-(2-aminoethyl)-6-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)picolinamide 347212 7-(2-nitrophenyl)-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 347213 (2-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)phenyl)methanol 347221 7-(3-(trifluoromethyl)phenyl)-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 347222 3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzonitrile 347239 4-(((2-(trifluoromethyl)benzyl)(cyclohexylmethyl)amino)methyl)-N-(naphthalen-1-yl)thiazol-2-amine 347240 4-tert-butyl-N-phenylthiazol-2-amine 347241 4-tert-butyl-N-o-tolylthiazol-2-amine 347245 3-(((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)(methyl)amino)-1-isopropylazetidine-3-carboxamide 347247 4-tert-butyl-N-m-tolylthiazol-2-amine 347248 4-((diisobutylamino)methyl)-N-(naphthalen-1-yl)thiazol-2-amine 347262 N-methyl-2-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)phenyl)acetamide 347304 (5-(4-fluorophenyl)-4-(pyridin-4-yl)-1H-pyrrol-2-yl)-N,N-dimethylmethanamine 347312 2-(4-(4-((2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)piperazin-1-yl)butyl)-4-p-tolylphthalazin-1(2H)-one 347316 7-(4-(trifluoromethyl)phenyl)-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 347325 2-(4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)-4-p-tolylphthalazin-1(2H)-one 347326 4-p-tolyl-2-(4-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)butyl)phthalazin-1(2H)-one 347327 7-(4-nitrophenyl)-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 347328 methyl 4-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzoate 347346 2-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)phenyl)acetonitrile 347347 3-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)phenyl)propanenitrile 347352 methyl 3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzoate 347353 7-(4-butylphenyl)-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 347358 2-(5-(4-fluorophenyl)-4-(pyridin-4-yl)-1H-pyrrol-2-yl)-N,N-dimethylacetamide 347359 7-(3-((2H-tetrazol-5-yl)methyl)phenyl)-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 347361 7-(4-tert-butylphenyl)-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 347362 7-(4-(methylthio)phenyl)-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 347365 7-(3-(2-(2H-tetrazol-5-yl)ethyl)phenyl)-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 347366 N-(2-aminoethyl)-3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzamide 347374 N-(2-(dimethylamino)ethyl)-3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)benzamide 347380 N-(2-(dimethylamino)ethyl)-6-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)picolinamide 347404 2-(5-(4-fluorophenyl)-4-(pyridin-4-yl)-1H-pyrrol-2-yl)-N,N-dimethylethanamine 347411 ethyl 5-(4-fluorophenyl)-4-(pyridin-4-yl)-1H-pyrrole-2-carboxylate 347412 N-ethyl-3-(5-(4-fluorophenyl)-4-(pyridin-4-yl)-1H-pyrrol-2-yl)-N-methylpropan-1-amine 347420 3-(((4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)(methyl)amino)-1-(2-methoxyethyl)azetidine-3-carboxamide 347421 N-(4-tert-butylthiazol-2-yl)-1H-indol-4-amine 347449 1-(5-(4-fluorophenyl)-4-(pyridin-4-yl)-1H-pyrrol-2-yl)-N,N,2-trimethylpropan-1-amine 347450 4-(2-(4-fluorophenyl)-5-(1-methylpyrrolidin-2-yl)-1H-pyrrol-3-yl)pyridine 347457 4-(5-(azetidin-1-ylmethyl)-2-(4-fluorophenyl)-1H-pyrrol-3-yl)pyridine 347458 4-(2-(4-fluorophenyl)-5-(1-methylpiperidin-2-yl)-1H-pyrrol-3-yl)pyridine 347460 N-(4-tert-butylthiazol-2-yl)quinolin-5-amine 347461 N-(4-tert-butylthiazol-2-yl)isoquinolin-5-amine 347464 2-(4-(4-(pyrimidin-2-yl)piperazin-1-yl)butyl)-4-p-tolylphthalazin-1(2H)-one 347465 2-(7-(4-(2-methoxyphenyl)piperazin-1-yl)heptyl)-4-p-tolylphthalazin-1(2H)-one 347470 2-(7-(4-(2-ethoxyphenyl)piperazin-1-yl)heptyl)-4-p-tolylphthalazin-1(2H)-one 347510 [4-(4-chloro-benzyl)-7-dimethylsulfamoyl-1,2,3,4-tetrahydro-cyclopenta[b]indol-3-yl]-acetic acid 347519 [5-bromo-4-(4-chloro-benzyl)-7-dimethylsulfamoyl-1,2,3,4-tetrahydro-cyclopenta[b]indol-3-yl]-acetic acid 347522 2-(5-bromo-4-((7-chloroquinolin-2-yl)methyl)-7-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid 347538 2-(9-(4-chlorobenzyl)-6,8-difluoro-2,3,4,9-tetrahydro-1H-carbazol-1-yl)acetic acid 347539 2-(9-(4-chlorobenzyl)-2,3,4,9-tetrahydro-1H-carbazol-1-yl)acetic acid 347548 2-(9-(4-chlorobenzyl)-8-(phenylcarbamoyl)-2,3,4,9-tetrahydro-1H-carbazol-1-yl)acetic acid 347581 2-(4-(4-chlorobenzyl)-5-bromo-7-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid 347590 2-(4-(4-chlorobenzyl)-7-(methylsulfonyl)-5-vinyl-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid 347612 N-{4-[4-(3-methanesulfonylamino-phenyl)-piperazin-1-yl]-butyl}-4-methyl-benzenesulfonamide 347613 (S)-(2-((diethylamino)methyl)pyrrolidin-1-yl)(5-(trifluoromethyl)benzofuran-2-yl)methanone 347615 2-(4-(4-chlorobenzyl)-5-cyclohexyl-7-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid 347616 2-(4-(4-chlorobenzyl)-5-cyano-7-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid 347618 N-{4-[4-(3-ethanesulfonylamino-phenyl)-piperazin-1-yl]-butyl}-4-methyl-benzenesulfonamide 347619 4-methyl-N-(4-{4-[3-(propane-2-sulfonylamino)-phenyl]-piperazin-1-yl}-butyl)-benzenesulfonamide 347620 (S)-(2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl)(5-(trifluoromethoxy)benzofuran-2-yl)methanone 347621 (S)-2-(2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl)benzofuran-5-carbonitrile 347626 (2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 9-acetoxy-6a,10b-dimethyl-2-(1-(methylsulfonyl)-1H-pyrrol-3-yl)-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 347637 (S)-(2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl)(6-(trifluoromethyl)benzofuran-2-yl)methanone 347643 (S)-(2-(piperidin-1-ylmethyl)pyrrolidin-1-yl)(6-(trifluoromethyl)benzofuran-2-yl)methanone 347644 (S)-(2-((diethylamino)methyl)pyrrolidin-1-yl)(6-(trifluoromethyl)benzofuran-2-yl)methanone 347653 (S)-(7-ethoxybenzofuran-2-yl)(2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl)methanone 347657 2-(4-(4-(methylsulfonyl)benzyl)-5-bromo-7-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid 347659 N-(2-fluorophenyl)-2-(1-(3-(2-(pyridin-2-yl)ethynyl)benzoyl)piperidin-4-yl)acetamide 347663 N-(3-{4-[4-(toluene-4-sulfonylamino)-butyl]-piperazin-1-yl}-phenyl)-propionamide 347664 4-methyl-N-(4-(4-phenylpiperazin-1-yl)butyl)benzenesulfonamide 347686 N-(3-{4-[4-(toluene-4-sulfonylamino)-butyl]-piperazin-1-yl}-phenyl)-butyramide 347692 N-{2-[4-((S)-2-amino-5-(dimethylamino)pentanoyl)piperazin-1-yl]-1,1-dimethyl-2-oxoethyl}-2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonamide 347693 (S)-N-(1-(4-(2-amino-5-(dimethylamino)pentanoyl)piperazin-1-yl)-2-methyl-1-oxopropan-2-yl)-2,4-dichloro-3-((2,4-dimethylquinolin-8-yloxy)methyl)benzenesulfonamide 347699 (2S)-1-(1H-indol-3-yl)-3-(5-(1-methoxyisoquinolin-6-yl)pyridin-3-yloxy)propan-2-amine 347700 (S)-6-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)isoquinolin-3-amine 347707 (S)-6-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)isoquinolin-5-amine 347708 (2S)-1-(1H-indol-3-yl)-3-(5-(8-methylisoquinolin-6-yl)pyridin-3-yloxy)propan-2-amine 347709 (S)-6-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)isoquinolin-1-amine 347710 (S)-1-(5-(3-fluoroisoquinolin-6-yl)pyridin-3-yloxy)-3-(1H-indol-3-yl)propan-2-amine 347717 8-(2-(4-(2,4-difluorophenethyl)piperidin-1-ylsulfonyl)phenyl)quinoline 347718 (4-(2,4-difluorophenethyl)piperidin-1-yl)(2-fluorophenyl)methanone 347719 (2S)-1-(5-(3-chloroisoquinolin-6-yl)pyridin-3-yloxy)-3-(1H-indol-3-yl)propan-2-amine 347722 [(R)-5-Acetyl-4-(4-chloro-benzyl)-7-methanesulfonyl-1,2,3,4-tetrahydro-cyclopenta[b]indol-3-yl]-acetic acid 347723 (4-(2,4-difluorophenethyl)piperidin-1-yl)(quinolin-8-yl)methanone 347726 7-(1-(2,4-difluorophenethyl)piperazine-4-carbonyl)-1H-indole-3-carbonitrile 347727 1-(2,4-difluorophenethyl)-4-(4-fluorophenylsulfonyl)piperazine 347732 [(3R)-4-(4-chlorobenzyl)-5-(1-hydroxyethyl)-7-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl]acetic acid 347733 2-(9-(4-chlorobenzyl)-8-isopropyl-2,3,4,9-tetrahydro-1H-carbazol-1-yl)acetic acid 347738 4-(2,4-difluorophenethyl)-1-(4-fluorophenylsulfonyl)piperidin-4-ol 347741 6-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)isoquinoline-3-carbonitrile 347743 2-(9-(4-chlorobenzyl)-8-(methylthio)-2,3,4,9-tetrahydro-1H-carbazol-1-yl)acetic acid 347747 N-{2-[4-((S)-2-amino-6-(dimethylamino)hexanoyl)piperazin-1-yl]-1,1-dimethyl-2-oxoethyl}-2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonamide 347750 (2S)-1-(5-(3-ethylisoquinolin-6-yl)pyridin-3-yloxy)-3-(1H-indol-3-yl)propan-2-amine 347751 2-(9-(4-chlorobenzyl)-8-(methylsulfinyl)-2,3,4,9-tetrahydro-1H-carbazol-1-yl)acetic acid 347755 (S)-N-(1-(4-(2-amino-6-(dimethylamino)hexanoyl)piperazin-1-yl)-2-methyl-1-oxopropan-2-yl)-2,4-dichloro-3-((2,4-dimethylquinolin-8-yloxy)methyl)benzenesulfonamide 347770 Bis-(5-hydroxy-1H-indol-2-yl)-methanone 347771 2-(9-(4-chlorobenzyl)-8-bromo-2,3,4,9-tetrahydro-1H-carbazol-1-yl)acetic acid 347778 2-((R)-9-(4-chlorobenzyl)-8-((S)-methylsulfinyl)-2,3,4,9-tetrahydro-1H-carbazol-1-yl)acetic acid 347779 2-(9-(4-chlorobenzyl)-8-(methylsulfonyl)-2,3,4,9-tetrahydro-1H-carbazol-1-yl)acetic acid 347814 N-(3-(4-(4-(4-methylphenylsulfonamido)butyl)piperazin-1-yl)phenyl)acetamide 347867 (R)-3-(1H-benzo[d]imidazol-2-yl)-6-chloro-4-(pyrrolidin-3-ylamino)quinolin-2(1H)-one 347868 N-(3-{4-[4-(4-fluoro-benzenesulfonylamino)-butyl]-piperazin-1-yl}-phenyl)-acetamide 347869 N-(3-(4-(4-(cyclohexylsulfonylamino)butyl)piperazin-1-yl)-phenyl)acetamide 347872 N-(4-fluorophenyl)-2-(1-(3-(2-(pyridin-2-yl)ethynyl)benzoyl)piperidin-4-yl)acetamide 347876 N-(3-{4-[4-(propane-2-sulfonylamino)-butyl]-piperazin-1-yl}-phenyl)-acetamide 347877 N-(3-(4-(4-(cyclohexylmethylsulfonamido)butyl)piperazin-1-yl)phenyl)acetamide 347913 SID24715130 347924 (2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 9-acetoxy-6a,10b-dimethyl-4,10-dioxo-2-(1-(phenylsulfonyl)-1H-pyrrol-3-yl)-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 347925 (S)-3-(1H-benzo[d]imidazol-2-yl)-6-chloro-4-(quinuclidin-3-ylamino)quinolin-2(1H)-one 347931 cyclopropanecarboxylic acid (3-{4-[4-(toluene-4-sulfonylamino)-butyl]-piperazin-1-yl}-phenyl)-amide 347932 N-(3-(4-(4-(tosylamino)butyl)piperazin-1-yl)phenyl)pivalamide 347933 SID24715131 347935 3-(1H-benzo[d]imidazol-2-yl)-6-chloro-4-(piperidin-3-ylamino)quinolin-2(1H)-one 347936 3-(1H-benzo[d]imidazol-2-yl)-6-chloro-4-(piperidin-4-ylamino)quinolin-2(1H)-one 347943 2-(4-(4-chlorobenzyl)-7-(methylsulfonyl)-5-(thiophen-2-yl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid 347983 methyl 2-((2S,4aR,6aR,7R,9S,10aS,10bR)-9-acetoxy-7-(methoxycarbonyl)-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-benzo[f]isochromen-2-yl)oxazole-4-carboxylate 347986 2-(9-(4-chlorobenzyl)-8-formyl-2,3,4,9-tetrahydro-1H-carbazol-1-yl)acetic acid 347990 (2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 9-acetoxy-6a,10b-dimethyl-2-(3-methyl-1,2,4-oxadiazol-5-yl)-4,10-dioxododecahydro-1H-benzo[f]isochromene-7-carboxylate 347991 (S)-3-(1H-benzo[d]imidazol-2-yl)-5,6-dichloro-4-(quinuclidin-3-ylamino)quinolin-2(1H)-one 347994 2-(9-(4-chlorobenzyl)-8-(ethylsulfinyl)-2,3,4,9-tetrahydro-1H-carbazol-1-yl)acetic acid 347995 2-(9-(4-chlorobenzyl)-8-(isopropylsulfinyl)-2,3,4,9-tetrahydro-1H-carbazol-1-yl)acetic acid 347996 2-(5-bromo-4-((2,3-dichlorothieno[3,2-b]pyridin-5-yl)methyl)-7-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid 347998 (S)-3-(1H-benzo[d]imidazol-2-yl)-8-methyl-4-(quinuclidin-3-ylamino)quinolin-2(1H)-one 348005 2-(9-(4-chlorobenzyl)-8-(hydroxymethyl)-2,3,4,9-tetrahydro-1H-carbazol-1-yl)acetic acid 348007 2-(4-(4-chlorobenzyl)-5-acetyl-7-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid 348012 2-(9-(4-chlorobenzyl)-8-(phenylsulfinyl)-2,3,4,9-tetrahydro-1H-carbazol-1-yl)acetic acid 348013 2-((R)-9-(4-chlorobenzyl)-8-((R)-methylsulfinyl)-2,3,4,9-tetrahydro-1H-carbazol-1-yl)acetic acid 348014 2-(4-(4-chlorobenzyl)-5-(1-hydroxyethyl)-7-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid 348015 2-(4-(3-chlorobenzyl)-5-bromo-7-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid 348036 cyclopropanecarboxylic acid {3-[4-(4-cyclohexylmethanesulfonylamino-butyl)-piperazin-1-yl]-phenyl}-amide 348041 N-(3-{4-[4-(2-methyl-propane-1-sulfonylamino)-butyl]-piperazin-1-yl}-phenyl)-acetamide 348046 N-(3-{4-[4-(cyclohexylmethanesulfonyl-methyl-amino)-butyl]-piperazin-1-yl}-phenyl)-acetamide 348049 N-[3-(4-{4-[methyl-(2-methyl-propane-1-sulfonyl)-amino]-butyl}-piperazin-1-yl)-phenyl]-acetamide 348051 N-{2-[4-((S)-3-amino-7-guanidinoheptanoyl)piperazin-1-yl]-1,1-dimethyl-2-oxoethyl}-2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonamide 348059 (S)-N-(1-(4-(3-amino-6-(dimethylamino)hexanoyl)piperazin-1-yl)-2-methyl-1-oxopropan-2-yl)-2,4-dichloro-3-((2,4-dimethylquinolin-8-yloxy)methyl)benzenesulfonamide 348065 N-(3-{4-[4-(toluene-4-sulfonylamino)-butyl]-piperazin-1-yl}-phenyl)-isobutyramide 348081 4-(2,4-difluorophenethyl)-4-fluoro-1-(4-fluorophenylsulfonyl)piperidine 348082 N-{2-[4-((S)-3-amino-7-(dimethylamino)heptanoyl)piperazin-1-yl]-1,1-dimethyl-2-oxoethyl}-2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonamide 348083 N-{2-[4-((S)-3-amino-7-(dimethylamino)heptanoyl)piperazin-1-yl]-1,1-dimethyl-2-oxoethyl}-2,4-dichloro-3-(2,4-dimethylquinolin-8-yloxymethyl)benzenesulfonamide 348084 N-[(S)-1-(4-{2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-2-methylpropionyl}piperazine-1-carbonyl)-5-(dimethylamino)pentyl]acetamide 348092 2-(4-(3-(trifluoromethoxy)benzyl)-5-bromo-7-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid 348103 (2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 9-acetoxy-2-(1-(4-methoxyphenylsulfonyl)-1H-pyrrol-3-yl)-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 348111 N-{3-[4-(1-Cyclohexylmethanesulfonyl-piperidin-4-ylmethyl)-piperizine-1-yl]-phenyl}-acetamide 348112 4-(2,4-difluorophenethyl)-1-(2-fluorophenylsulfonyl)piperidine 348118 N-(3-{4-[1-(propane-2-sulfonyl)-piperidin-4-ylmethyl]-piperizine-1-yl}-phenyl)-acetamide 348170 2-(9-(4-chlorobenzyl)-8-(dimethylcarbamoyl)-2,3,4,9-tetrahydro-1H-carbazol-1-yl)acetic acid 348171 2-(9-(4-chlorobenzyl)-8-(benzylsulfinyl)-2,3,4,9-tetrahydro-1H-carbazol-1-yl)acetic acid 348179 2-(9-(4-chlorobenzyl)-6-(methylsulfonyl)-2,3,4,9-tetrahydro-1H-carbazol-1-yl)acetic acid 348180 2-(4-(4-chlorobenzyl)-7-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid 348188 (S)-benzo[b]thiophen-2-yl(2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl)methanone 348204 4-[3-(4-Chlorophenyl)-3-hydroxy-8-azabicyclo[3.2.1]oct-8-yl]-1-(4-fluorophenyl)butan-1-one 348217 (S)-(3-chlorobenzo[b]thiophen-2-yl)(2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl)methanone 348218 (S)-(5-chlorobenzofuran-2-yl)(2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl)methanone 348225 (S)-(2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl)(5-(trifluoromethyl)benzofuran-2-yl)methanone 348226 (S)-(2-(piperidin-1-ylmethyl)pyrrolidin-1-yl)(5-(trifluoromethyl)benzofuran-2-yl)methanone 348227 (S)-1-(1H-indol-3-yl)-3-(5-(3-vinylisoquinolin-6-yl)pyridin-3-yloxy)propan-2-amine 348228 (2S)-1-(5-(3-(furan-2-yl)isoquinolin-6-yl)pyridin-3-yloxy)-3-(1H-indol-3-yl)propan-2-amine 348229 (S)-1-(1H-indol-3-yl)-3-(5-(3-(pyridin-4-yl)isoquinolin-6-yl)pyridin-3-yloxy)propan-2-amine 348230 (2S)-1-(1H-indol-3-yl)-3-(5-(3-(prop-1-ynyl)isoquinolin-6-yl)pyridin-3-yloxy)propan-2-amine 348234 (S)-1-(1H-indol-3-yl)-3-(5-(3-phenylisoquinolin-6-yl)pyridin-3-yloxy)propan-2-amine 348235 4-(2,4-difluorophenethyl)-1-(4-fluorophenylsulfonyl)-1,2,3,6-tetrahydropyridine 348236 (2S)-1-(1H-indol-3-yl)-3-(5-(3-(2-phenylethynyl)isoquinolin-6-yl)pyridin-3-yloxy)propan-2-amine 348237 4-(2,4-difluorophenethyl)-1-(2-chlorophenylsulfonyl)piperidine 348244 4-(2,4-difluorophenethyl)-1-(4-fluorophenylsulfonyl)piperidine 348245 4-(2,4-difluorophenethyl)-1-(3-fluorophenylsulfonyl)piperidine 348246 2-(4-(2,4-difluorophenethyl)piperidin-1-ylsulfonyl)benzonitrile 348247 4-(2,4-difluorophenethyl)-1-(2-(naphthalen-1-yl)phenylsulfonyl)piperidine 348252 (S)-3-(1H-benzo[d]imidazol-2-yl)-4-(quinuclidin-3-ylamino)quinolin-2(1H)-one 348259 3-(1-hydroxy-3,3-dimethyl-3,4,10,11-tetrahydro-2H-dibenzo[b,e][1,4]diazepin-11-yl)-benzene-1,2-diol 348260 (R)-3-(1H-benzo[d]imidazol-2-yl)-4-(quinuclidin-3-ylamino)quinolin-2(1H)-one 348261 (S)-3-(1H-benzo[d]imidazol-2-yl)-6-methyl-4-(quinuclidin-3-ylamino)quinolin-2(1H)-one 348268 3-(1H-benzo[d]imidazol-2-yl)-6-methyl-4-(piperidin-3-ylamino)quinolin-2(1H)-one 348290 N-(5-((1H-indol-3-yl)methyl)-1,3,4-thiadiazol-2-yl)-4-methoxybenzamide 348298 4-(3-(benzyloxy)benzylidene)-1-(3,4-dichlorophenyl)pyrazolidine-3,5-dione 348299 4-((5-(3-chloro-4-methylphenyl)furan-2-yl)methylene)-1-(3,4-dimethylphenyl)pyrazolidine-3,5-dione 348317 1-(5-benzyl-1,3,4-thiadiazol-2-yl)-3-phenylurea 348327 (Z)-{2-(hydroxymethyl)-4-[4-methyl-3-(methylethyl)pentylidene]-5-oxo-2,3-dihydrofur-2-yl}methyl 4-hydroxybenzoate 348328 (E)-{2-(hydroxymethyl)-4-[(4-methoxyphenyl)methylene]-5-oxo-2,3-dihydrofur-2-yl}methyl 4-methyl-3-(methylethyl)pentanoate 348332 3-(1H-benzo[d]imidazol-2-yl)-6-methyl-4-(piperidin-4-ylamino)quinolin-2(1H)-one 348336 N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-4-methylbenzenesulfonamide 348337 N-(3-(4-((1-(4-fluorophenylsulfonyl)piperidin-4-yl)methyl)piperazin-1-yl)phenyl)acetamide 348339 (S)-3-(1H-benzo[d]imidazol-2-yl)-6-chloro-4-(pyrrolidin-3-ylamino)quinolin-2(1H)-one 348342 4-((6-bromobenzo[d][1,3]dioxol-5-yl)methylene)-1-(4-iodophenyl)pyrazolidine-3,5-dione 348372 2-(4-(4-tert-butylbenzyl)-5-bromo-7-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid 348393 des-Ac-[D-4Aph(CO-NH-(C2H4O)2-C2H5)6]-C2H5-(C2H4O)2-NHCO- 348394 [4Aph(CO-NH-OCH3)5,D-4Aph(CO-NH-OCH3)6]degarelix 348395 [N-alpha-Me-4Aph(CO-NH-OCH3)5,D-4Aph(CO-NH-OCH3)6]degarelix 348396 3-(4-chlorophenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 348398 (2S)-1-(6-ethynyl-5-(isoquinolin-6-yl)pyridin-3-yloxy)-3-(1H-indol-3-yl)propan-2-amine 348399 (2S)-1-(1H-indol-3-yl)-3-(5-(isoquinolin-6-yl)-6-(2-phenylethynyl)pyridin-3-yloxy)propan-2-amine 348402 N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]-2,2-trimethyleneethyl)cyclobutanecarboxamide 348403 N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]-2,2-tetramethyleneethyl)acetamide 348435 Ac-Cys-Ile-cyclo[Phe-Lys]-Tyr-Tyr 348436 des-Ac-[4Aph(CO-NH-OCH3)5]-CH3-(CH2)2-CO-degarelix 348437 des-Ac-[4Aph(CO-NH-OCH3)5]-CH3-(CH2)6-CO-degarelix 348447 N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]propyl)butanamide 348459 N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]-2,2-tetramethyleneethyl)propanamide 348460 N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]-2,2-tetramethyleneethyl)butanamide 348461 N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]-2,2-tetramethyleneethyl)cyclopropanecarboxamide 348462 beta,beta-dimethylmelatonin 348463 (R)-1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonyl]-pyrrolidine-2-carboxylic acid [3-(4-carbamimidoyl-benzoylamino)-propyl]-amide 348464 Ac-Cys-Ile-cyclo[Phe-Lys]-Tyr-Tyr 348465 [D-Dab(CO-NH-OCH3)3]degarelix 348466 [D-Dap(CO-NH-OCH3)3]degarelix 348469 (S)-1-(6-chloro-5-(isoquinolin-6-yl)pyridin-3-yloxy)-3-(1H-indol-3-yl)propan-2-amine 348470 (S)-5-(2-amino-3-(1H-indol-3-yl)propoxy)-3-(isoquinolin-6-yl)picolinonitrile 348471 N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]-2,2-tetramethyleneethyl)cyclobutanecarboxamide 348472 N-(2-[5-methoxy-1H-indol-3-yl]-2,2-trimethyleneethyl)acetamide 348478 (S)-1-(1H-indol-3-yl)-3-(5-(isoquinolin-6-yl)-6-vinylpyridin-3-yloxy)propan-2-amine 348479 N-(4-chloro-phenyl)-2-cyclopentyl-1H-imidazo[4,5-c]quinolin-4-amine 348488 N-(2-[5-methoxy-1H-indol-3-yl]-2,2-trimethyleneethyl)propanamide 348495 N-(2-[5-methoxy-1H-indol-3-yl]-2,2-trimethyleneethyl)butanamide 348501 (S)-1-(3,4-dimethoxyphenethylamino)-3-(4-(2-ethoxyethoxy)phenoxy)propan-2-ol 348506 4-(2-(benzyloxy)benzylidene)-1-phenylpyrazolidine-3,5-dione 348518 N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]propyl)propanamide 348520 4-benzylidene-1-(4-iodophenyl)pyrazolidine-3,5-dione 348522 (S)-1-(6-(furan-2-yl)-5-(isoquinolin-6-yl)pyridin-3-yloxy)-3-(1H-indol-3-yl)propan-2-amine 348534 N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]propyl)acetamide 348575 [D-4Aph(CO-NH-(C2H4O)2-C2H5)6]degarelix 348576 des-Ac-[D-4Aph(CO-NH-OCH3)6]-CH3-(CH2)2-CO-degarelix 348630 Cyclo[Ac-Cys-Ile-Tyr-Lys-Tyr-Tyr] 348635 [4Aph(CO-NH-OCH3)5,D-4Aph(CO-NH-OCH3)6,Orn(IGly)8]-degarelix 348636 [D-Dab(CO-NH-OCH3)3, 4Aph(CO-NH-OCH3)5,D-4Aph(CO-NHOCH3)6]-degarelix 348661 N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]-2-methylpropyl)acetamide 348663 SID47203119 348668 N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]-2-methylpropyl)-propanamide 348670 4-iodo-N-(5-phenethyl-1,3,4-thiadiazol-2-yl)benzamide 348671 2-iodo-N-(5-phenethyl-1,3,4-thiadiazol-2-yl)benzamide 348672 (E)-[4-decylidene-2-(hydroxymethyl)-5-oxo-2,3-dihydrofur-2-yl]methyl benzoate 348675 N-(2-[5-methoxy-1H-indol-3-yl]-2,2-trimethyleneethyl)cyclopropanecarboxamide 348676 [4Aph(CO-NH-OCH3)5]degarelix 348677 [4Aph(CO-NH-OH)5]degarelix 348678 (Z)-[{2-(hydroxymethyl)-4-[4-methyl-3-(methylethyl)pentylidene]-5-oxo-2,3-dihydrofur-2-yl}methyl 3-methoxybenzoate 348680 (E)-[4-decylidene-2-(hydroxymethyl)-5-oxo-2,3-dihydrofur-2-yl]methyl cyclohexanecarboxylate 348685 N-(2-[1-methyl-1H-indol-3-yl]-2,2-trimethylene-ethyl)cyclopropanecarboxamide 348687 4-(4-iodobenzylidene)-1-(4-iodophenyl)pyrazolidine-3,5-dione 348695 (E)-{2-(hydroxymethyl)-4-[4-methyl-3-(methylethyl)pentylidene]-5-oxo-2,3-dihydrofur-2-yl}methyl 4-hydroxybenzoate 348697 (E)-[2-(hydroxymethyl)-4-[4-methyl-3-(methylethyl)pentylidene]- 348701 (Z)-[4-decylidene-2-(hydroxymethyl)-5-oxo-2,3-dihydrofur-2-yl]methyl cyclohexanecarboxylate 348706 (Z)-{2-(hydroxymethyl)-4-[4-methyl-3-(methylethyl)pentylidene]-5-oxo-2,3-dihydrofur-2-yl}methyl 2-hydroxybenzoate 348708 (E)-{2-(hydroxymethyl)-4-[4-methyl-3-(methylethyl)pentylidene]-5-oxo-2,3-dihydrofur-2-yl}methyl benzoate 348709 (Z)-{2-(hydroxymethyl)-4-[4-methyl-3-(methylethyl)pentylidene]-5-oxo-2,3-dihydrofur-2-yl}methyl benzoate 348727 (Z)-[{2-(hydroxymethyl)-4-[4-methyl-3-(methylethyl)pentylidene]-5-oxo-2,3-dihydrofur-2-yl}methyl 2-methoxybenzoate 348734 (E)-[{2-(hydroxymethyl)-4-[4-methyl-3-(methylethyl)pentylidene]-5-oxo-2,3-dihydrofur-2-yl}methyl 3-methoxybenzoate 348749 N-(2-[5-methoxy-1H-indol-3-yl]-2,2-trimethyleneethyl)cyclobutanecarboxamide 348750 N-(2-[1-methyl-1H-indol-3-yl]-2,2-trimethylene-ethyl)acetamide 348751 N-(2-[1-methyl-1H-indol-3-yl]-2,2-trimethylene-ethyl)propaneamide 348752 (E)-{2-(hydroxymethyl)-4-[4-methyl-3-(methylethyl)pentylidene]-5-oxo-2,3-dihydrofur-2-yl}methyl 3-hydroxybenzoate 348753 (Z)-{2-(hydroxymethyl)-4-[4-methyl-3-(methylethyl)pentylidene]-5-oxo-2,3-dihydrofur-2-yl}methyl 3-hydroxybenzoate 348756 N-(2-[1-methyl-1H-indol-3-yl]-2,2-trimethylene-ethyl)butanamide 348759 (E)-{2-(hydroxymethyl)-4-[(2-hydroxyphenyl)methylene]-5-oxo-2,3-dihydrofur-2-yl}methyl 4-methyl-3-(methylethyl)pentanoate 348761 (S)-1-(2-chloro-5-(isoquinolin-6-yl)pyridin-3-yloxy)-3-(1H-indol-3-yl)propan-2-amine 348766 (E)-{2-(hydroxymethyl)-4-[(3-hydroxyphenyl)methylene]-5-oxo-2,3-dihydrofur-2-yl}methyl 4-methyl-3-(methylethyl)pentanoate 348767 (E)-{2-(hydroxymethyl)-4-[(4-hydroxyphenyl)methylene]-5-oxo-2,3-dihydrofur-2-yl}methyl 4-methyl-3-(methylethyl)pentanoate 348783 1-(2-(3-(2-cyano-4-(2-(cyclopropylmethoxy)ethoxy)phenoxy)-2-hydroxypropylamino)ethyl)-3-(4-hydroxyphenyl)urea 348812 cyanopindolol 348824 des-Ac-[4Aph(CO-NH-OCH3)5]-C2H5-(C2H4O)2-NH-CO-degarelix 348825 des-Ac-[4Aph(CO-NH-(C2H4O)2-C2H5)5]-C2H5-(C2H4O)2-NHCO-degarelix 348840 2,4-dichloro-N-(5-phenethyl-1,3,4-thiadiazol-2-yl)benzamide 348841 2-methoxy-4-(methylthio)-N-(5-phenethyl-1,3,4-thiadiazol-2-yl)benzamide 348860 4-(4-(diethylamino)-2-hydroxybenzylidene)-1-(4-iodophenyl)pyrazolidine-3,5-dione 348874 (S)-6-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)isoquinolin-1-ol 348885 (2S)-1-(5-(1-chloroisoquinolin-6-yl)pyridin-3-yloxy)-3-(1H-indol-3-yl)propan-2-amine 348890 N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]-2-methylpropyl)butanamide 348891 N-(2-(5-methoxy-1-methyl-1H-indol-3-yl)-2-methylpropyl)cyN-(2-(5-Methoxy-1-methyl-1H-indol-3-yl)-2-methylpropyl)cyclobutanecarboxamide 348903 N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]-2,2-dimethyleneethyl)acetamide 348904 N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]-2,2-dimethyleneethyl)propanamide 348905 N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]-2,2-dimethyleneethyl)butanamide 348923 beta-methylmelatonin 348936 1-(2-chloroethyl)-3-{[4-(3-methylphenyl)amino]quinazolin-6-yl}urea 348942 N-(4-methyl-phenyl)-2-cyclopentyl-1H-imidazo[4,5-c]quinolin-4-amine 348943 [4Aph(CO-NH-(C2H4O)2-C2H5)5,D-4Aph(CO-NH-(C2H4O)2-C2H5)6]-degarelix 348944 [4Aph(CO-NH-OCH3)5,D-4Aph(CO-(C2H4O)6-C2H4-NH-CONH-OCH3)6]degarelix 348945 des-Ac-[4Aph(CO-NH-OCH3)5,D-4Aph(CO-NH-OCH3)6]-CH3-(CH2)2-CO-degarelix 348954 des-Ac-[D-4Aph(CO-NH-OCH3)6]-CH3-(CH2)6-CO-degarelix 348955 des-Ac-[D-4Aph(CO-NH-OCH3)6]-C2H5-(C2H4O)2-NH-COdegarelix 348970 N-(4-methoxy-phenyl)-2-cyclopentyl-1H-imidazo[4,5-c]quinolin-4-amine 348971 2-cyclopentyl-N-(3,4-dichlorophenyl)-1H-imidazo[4,5-c]quinolin-4-amine 348986 Ac-Cys-Ile-cyclo[Phe-Lys-Tyr-Tyr] 348988 4-[(3-methylphenyl)amino]-6-(methylamino)quinazoline 348991 (2S)-1-(1H-indol-3-yl)-3-(5-(isoquinolin-6-yl)-4-methylpyridin-3-yloxy)propan-2-amine 348995 4-(4-morpholinobenzylidene)-1-(4-iodophenyl)pyrazolidine-3,5-dione 349000 4-[(3-chlorophenyl)amino]-6-(methylamino)quinazoline 349001 N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]-2,2-trimethyleneethyl)acetamide 349002 N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]-2,2-trimethyleneethyl)propanamide 349003 [D-Dab(CO-NH-OH)3]degarelix 349004 [D-Dap(CO-NH-OH)3]degarelix 349007 [4Aph(CO-NH-(C2H4O)2-C2H5)5]degarelix 349008 [4Aph(CO-(C2H4O)3-C2H4-NH-CO-NH-OCH3)5]degarelix 349009 (E)-3-(3-((S)-2-amino-3-(1H-indol-3-yl)propoxy)-5-(isoquinolin-6-yl)pyridin-4-yl)acrylonitrile 349010 (2S)-1-(5-(1-fluoroisoquinolin-6-yl)pyridin-3-yloxy)-3-(1H-indol-3-yl)propan-2-amine 349022 N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]-2,2-trimethyleneethyl)butanamide 349023 N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]-2,2-trimethyleneethyl)cyclopropanecarboxamide 349024 N-(2-[1-methyl-1H-indol-3-yl]-2,2-trimethylene-ethyl)cyclobutanecarboxamide 349057 N-(5-methoxy-1H-benzo[d]imidazol-2-yl)-3-nitrobenzamide 349061 (H-Dmt-Tic-Glu-NH-(CH(2))(5)-CO-Dap(6DMN)-NH(2) 349064 (4R,5S)-5-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-4-(4-fluorophenyl)-1-methylazepan-2-one 349066 8-(1-(2-chloro-5-fluorobenzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349067 8-(1-(2-chloro-5-(trifluoromethyl)benzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349068 8-(1-(4-methylbenzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349081 N-n-pentyl-N'-[2-(3, 5-dimethylphenylamino)-5-nitrobenzenesulfonyl]urea 349084 2-(cis-5-(4-(5-(4-((R)-3,3-difluorocyclopentyl)phenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-2-yl)acetic acid 349089 methyl 2-(3-nitrobenzamido)-1H-benzo[d]imidazole-5-carboxylate 349090 3-nitro-N-(5-(propylsulfonyl)-1H-benzo[d]imidazol-2-yl)benzamide 349093 N-{4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl}tricyclo[8.2.2.2^{4,7}]hexadeca-1(12),4,6,10,13,15-hexaene-5-carboxamide 349095 N-[3-(4-carbamimidoylphenylamino)propyl]-2-[2,4-dichloro-3-(2,4-dimethylquinolin-8-yloxymethyl)benzenesulfonylamino]-2-methylpropionamide 349096 N-[3-(4-carbamimidoylphenylamino)propyl]-2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-2-methylpropionamide 349100 8-(1-(3-chloro-2-fluoro-5-(trifluoromethyl)benzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349102 8-(1-(2-methoxybenzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349103 8-(1-(3-methoxybenzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349104 8-(1-(3-fluorobenzyl)-1H-pyrazol-4-yl)-1,3-diethyl-1H-purine-2,6(3H,7H)-dione 349105 8-(1-(3-(trifluoromethyl)benzyl)-1H-pyrazol-4-yl)-1,3-diethyl-1H-purine-2,6(3H,7H)-dione 349111 (E)-[2-(hydroxymethyl)-4-octylidene-5-oxo-2,3-dihydrofur-2-yl]methyl 3-phenylpropanoate 349112 (Z)-[2-(hydroxymethyl)-4-octylidene-5-oxo-2,3-dihydrofur-2-yl]methyl 3-phenylpropanoate 349115 N-n-pentyl-N'-[2-(3-methyl-4-bromophenylamino)-5-nitrobenzenesulfonyl]urea 349125 1-(2-chloroethyl)-3-{[4-(3-chlorophenyl)amino]quinazolin-6-yl}urea 349126 (6S,7S)-7-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-6-(4-fluorophenyl)-6,7,8,9-tetrahydro-5H-imidazo[1,2-a]azepine 349127 ethyl 3-(2-(3-nitrobenzamido)-1H-benzo[d]imidazol-1-yl)propanoate 349130 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-o-tolylacetamide 349132 2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-N-(3-(dimethylamino)propyl)-2-methylpropionamide 349133 2,4-dichloro-N-(2-guanidino-1,1-dimethyl-2-oxoethyl)-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonamide 349136 8-(1-(4-(trifluoromethyl)benzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349137 8-(1-(2,3-difluorobenzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1Hpurine-2,6(3H,7H)-dione 349138 8-(1-benzyl-1H-pyrazol-4-yl)-1,3-dibutyl-1H-purine-2,6(3H,7H)-dione 349143 (E)-[2-(hydroxymethyl)-4-nonylidene-5-oxo-2,3-dihydrofur-2-yl]methyl 2-phenylacetate 349153 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-(4-bromo-2,5-dimethoxyphenyl)acetamide 349154 1-(2-chloroethyl)-3-{[4-(3-bromophenyl)amino]quinazolin-6-yl}urea 349155 3-(2-chloroethyl)-1-methyl-1-{[4-(3-methylphenyl)amino]quinazolin-6-yl}urea 349156 3-nitro-N-(1-(2-oxo-tetrahydrofuran-3-yl)-1H-benzo[d]imidazol-2-yl)benzamide 349157 N-(2-aminoethyl)-2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-2-methylpropionamide 349160 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-m-tolylacetamide 349161 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-(2,5-dimethylphenyl)acetamide 349166 8-(1-(2,4-difluorobenzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1Hpurine-2,6(3H,7H)-dione 349168 N-n-pentyl-N'-[2-(2, 6-dimethylphenylamino)-5-nitrobenzenesulfonyl]urea 349186 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-[(2-hydroxyethyl)propylamino]acetamide 349187 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-piperidin-1-ylacetamide 349188 3-(2-chloroethyl)-1-methyl-1-{[4-(3-chlorophenyl)amino]quinazolin-6-yl}urea 349189 8-(1-ethyl-3-methyl-1H-pyrazol-5-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349190 1-(2-methoxyphenyl)-4-((1-phenyl-1H-pyrazol-4-yl)methyl)piperazine 349191 1-((3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl)-4-phenylpiperazine 349194 N-n-pentyl-N'-[2-(4-methylphenoxy)-5-nitrobenzenesulfonyl]urea 349195 N-n-hexyl-N'-[2-(4-methylphenoxy)-5-nitrobenzenesulfonyl]urea 349199 8-(1-(2,4,6-trifluorobenzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349202 pentanoic acid (4-amino-5-cyano-6-ethoxypyridin-2-yl)amide 349203 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)acetamide 349208 (E)-{2-(hydroxymethyl)-4-[4-methyl-3-(methylethyl)pentylidene]-5-oxo-2,3-dihydrofur-2-yl}methylcyclohexanecarboxylate 349209 (Z)-{2-(hydroxymethyl)-4-[4-methyl-3-(methylethyl)pentylidene]-5-oxo-2,3-dihydrofur-2-yl}methylcyclohexanecarboxylate 349212 8-(1-(3-phenylpropyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349217 N-(4-amino-5-cyano-6-phenylpyridin-2-yl)acetamide 349219 N-(4-amino-5-cyanopyridin-2-yl)-2-(2,5-dimethoxyphenyl)acetamide 349220 8-(1-phenyl-1H-pyrazol-5-yl)-1,3-dipropyl-1H-purine-2,6-(3H,7H)-dione 349221 8-(1-phenyl-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6-(3H,7H)-dione 349222 2-(4-((1-phenyl-1H-pyrazol-4-yl)methyl)piperazin-1-yl)pyrimidine 349223 1-((5-methyl-1-phenyl-1H-pyrazol-4-yl)methyl)-4-phenylpiperazine 349235 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)isobutyramide 349240 (E)-{2-(hydroxymethyl)-4-[4-methyl-3-(methylethyl)pentylidene]-5-oxo-2,3-dihydrofur-2-yl}methyl 2-hydroxybenzoate 349243 8-(1-(2-methylbenzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349250 N-(1-allyl-1H-benzo[d]imidazol-2-yl)-3-nitrobenzamide 349252 N-(6-ethoxypyridin-2-yl)acetamide 349262 H-Tyr-Pro-Dap(6DMN)-Phe-NH2 349264 (5S,6S)-5-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-6-(4-fluorophenyl)azepan-2-one 349274 N-(6-aminohexyl)-4-{2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-2-methylpropionyl}-piperazine-1-carboxamidine 349287 8-(1-(4-fluorobenzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349288 8-(1-(2-(trifluoromethyl)benzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349291 3-nitro-N-(1-pentyl-1H-benzo[d]imidazol-2-yl)benzamide 349292 (+/-)-cis-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidine-2-carboxylic acid 349302 (4R,5S)-5-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-4-(4-fluorophenyl)azepan-2-one 349303 (5S,6S)-5-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-6-(4-fluorophenyl)-1-methylazepan-2-one 349324 (E)-[2-(hydroxymethyl)-5-oxo-4-(2-phenylethylidene)-2,3-dihydrofur-2-yl]methyl 4-methyl-3-(methylethyl)pentanoate 349325 (E)-[2-(hydroxymethyl)-5-oxo-4-(3-phenylpropylidene)-2,3-dihydrofur-2-yl]methyl 4-methyl-3-(methylethyl)pentanoate 349327 8-(1-(4-chlorobenzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349332 (+/-)-trans-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidine-2-carboxylic acid 349333 (+/-)-2-(cis-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-2-yl)acetic acid 349336 SID24784096 349337 H-Tyr-Pro-Phe-Phe-NH-(CH2)5-(C=O)-Dap(6DMN)-NH2 349339 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-(2,5-dimethoxy-4-nitrophenyl)acetamide 349342 (7S,8R)-7-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-8-(4-fluorophenyl)-6,7,8,9-tetrahydro-5H-imidazo[1,2-a]azepine 349343 (6S,7S)-7-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-6-(4-fluorophenyl)-6,7,8,9-tetrahydro-2H-[1,2,4]triazolo[4,3-a]azepin-3(5H)-one 349345 N-[4-(4-(2,3-dichlorophenyl)piperazin-1-yl]butyl][2.2]-paracyclophane-4-carboxamide 349353 (E)-[4-heptylidene-2-(hydroxymethyl)-5-oxo-2,3-dihydrofur-2-yl]methyl 4-phenylbutanoate 349356 (E)-{2-(hydroxymethyl)-4-[(2-methoxyphenyl)methylene]-5-oxo-2,3-dihydrofur-2-yl}methyl 4-methyl-3-(methylethyl)pentanoate 349357 (E)-{2-(hydroxymethyl)-4-[(3-methoxyphenyl)methylene]-5-oxo-2,3-dihydrofur-2-yl}methyl 4-methyl-3-(methylethyl)pentanoate 349358 8-(1-(2-fluorobenzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349367 N-(3H-imidazo[4,5-c]pyridin-2-yl)-3-nitrobenzamide 349369 N-(5-chloro-1H-benzo[d]imidazol-2-yl)-3-nitrobenzamide 349372 3-(2-chloroethyl)-1-methyl-1-{[4-(3-bromophenyl)amino]quinazolin-6-yl}urea 349373 1-(2-Chloroethyl)-1-nitroso-3-{[4-(3-methylphenyl)amino]quinazolin-6-yl}urea 349374 (7S,8R)-7-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-8-(4-fluorophenyl)-6,7,8,9-tetrahydro-2H-[1,2,4]triazolo[4,3-a]azepin-3(5H)-one 349375 N-(3-aminopropyl)-2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-2-methylpropionamide 349376 5-(3,3,6-trimethyl-indan-5-yloxy)-furan-2-carboxylic Acid [4,6-dimethoxy-2-(3-morpholin-4-yl-propylamino)-pyrimidine-5-yl]-amide 349377 N-4-[4-(3-chloro-2-methoxyphenyl)piperazin-1-yl]butyl][2.2]-paracyclophane-4-carboxamide 349378 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-p-tolylacetamide 349379 8-(1-benzyl-1H-pyrazol-4-yl)-1,3-dimethyl-1H-purine-2,6-(3H,7H)-dione 349382 8-(1-(4-methoxybenzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349384 (Z)-[4-heptylidene-2-(hydroxymethyl)-5-oxo-2,3-dihydrofur-2-yl]methyl 4-phenylbutanoate 349391 8-(1-(4-fluoro-3-(trifluoromethyl)benzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349392 8-(1-(4-chloro-3-(trifluoromethyl)benzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349399 N-n-pentyl-N'-[2-(3-methylphenylamino)-5-nitrobenzenesulfonyl]urea 349400 N-(5-fluoro-1H-benzo[d]imidazol-2-yl)-3-nitrobenzamide 349401 N-(5-methyl-1H-benzo[d]imidazol-2-yl)-3-nitrobenzamide 349402 N-(1-(2-cyclobutylethyl)-1H-benzo[d]imidazol-2-yl)-3-nitrobenzamide 349404 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-morpholin-4-ylacetamide 349405 1-(2-Chloroethyl)-1-nitroso-3-{[4-(3-chlorophenyl)amino]quinazolin-6-yl}urea 349406 1-(2-chloroethyl)-1-nitroso-3-{[4-(3-bromophenyl)amino]quinazolin-6-yl}urea 349407 N-(3-aminopropyl)-2-[2,4-dichloro-3-(2,4-dimethylquinolin-8-yloxymethyl)benzenesulfonylamino]-2-methylpropionamide 349408 N-(4-aminobutyl)-2-[2,4-dichloro-3-(2,4-dimethylquinolin-8-yloxymethyl)benzenesulfonylamino]-2-methylpropionamide 349409 8-(1-(3-(trifluoromethyl)-4-methoxybenzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349410 8-(1-(2,5-dichlorobenzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1Hpurine-2,6(3H,7H)-dione 349418 N-2-[4-(6-aminohexyl)piperazin-1-yl]-1,1-dimethyl-2-oxoethyl-2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonamide 349422 8-(1-(3-(trifluoromethyl)benzyl)-1H-pyrazol-4-yl)-1,3-dimethyl-1H-purine-2,6(3H,7H)-dione 349423 8-(1-benzyl-1H-pyrazol-4-yl)-1,3-diethyl-1H-purine-2,6(3H,7H)-dione 349437 8-(1-(3,5-bis(trifluoromethyl)benzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349445 N-(1-(2-methoxyethyl)-1H-benzo[d]imidazol-2-yl)-3-nitrobenzamide 349446 N-(1-(2-ethoxyethyl)-1H-benzo[d]imidazol-2-yl)-3-nitrobenzamide 349447 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-(4-hydroxypiperidin-1-yl)acetamide 349448 1-[(4-amino-5-cyano-6-ethoxypyridin-2-ylcarbamoyl)methyl]-piperidine-4-carboxylic acid butylamide 349451 1-Phenyl-4-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperazine 349452 1-(2-methoxyphenyl)-4-((1-phenyl-1H-1,2,3-triazol-4-yl)methyl)piperazine 349465 8-(1-(2,6-difluorobenzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1Hpurine-2,6(3H,7H)-dione 349467 (E)-[{2-(hydroxymethyl)-4-[4-methyl-3-(methylethyl)pentylidene]-5-oxo-2,3-dihydrofuryl}methyl 4-methoxybenzoate 349468 (Z)-[{2-(hydroxymethyl)-4-[4-methyl-3-(methylethyl)pentylidene]-5-oxo-2,3-dihydrofuryl}methyl 4-methoxybenzoate 349481 2,4-dichloro-N-{2-[4-(6-guanidinohexyl)piperazin-1-yl]-1,1-dimethyl-2-oxoethyl}-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonamide 349482 2,4-dichloro-N-{1,1-dimethyl-2-oxo-2-[4-(2-piperazin-1-ylacetyl)piperazin-1-yl]ethyl}-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonamide 349483 N-{2-[4-((S)-3-amino-6-(dimethylamino)hexanoyl)piperazin-1-yl]-1,1-dimethyl-2-oxoethyl}-2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonamide 349492 ethyl 2-(2-(3-nitrobenzamido)-1H-benzo[d]imidazol-1-yl)acetate 349493 (+/-)-2-(trans-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-2-yl)acetic acid 349494 1-[(4-amino-5-cyano-6-ethoxypyridin-2ylcarbamoyl)methyl]-piperidine-4-carboxylic acid isopropyl amide 349503 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-(4-methoxyphenyl)acetamide 349510 8-(1-(3-methylbenzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349512 H-Dmt-Tic-Glu-Dap(6DMN)-NH(2) 349524 des-Ac-[4Aph(CO-NH-(C2H4O)2-C2H5)5,D-4Aph(CO-NH-(C2H4O)2-C2H5)6]-C2H5-(C2H4O)2-NH-CO-degarelix 349525 [D-Gln3, 4Aph(CO-NH-OCH3)5,D-4Aph(CO-NH-OCH3)6]-degarelix 349526 des-Ac-[4Aph(CO-NH-OCH3)5,D-4Aph(CO-NH-OCH3)6]-CH3-(CH2)6-CO-degarelix 349534 (+/-)-3-(cis-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-2-yl)propanoic acid 349535 1-(4-Fluorophenyl)-4-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperazine 349538 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-(2,5-dimethoxyphenyl)acetamide 349539 N-tert-butyl-N'-[2-(4-methylphenoxy)-5-nitrobenzenesulfonyl]urea 349557 [D-4Aph(CO-NH-OH)6]degarelix 349558 [D-4Aph(CO-NH-OCH3)6]degarelix 349566 N-(4-amino-6-butylsulfanyl-5-cyanopyridin-2-yl)acetamide 349567 N-(4-amino-5-cyano-6-(ethylamino)pyridin-2-yl)acetamide 349570 1-(2-fluorophenyl)-4-((1-phenyl-1H-pyrazol-4-yl)methyl)piperazine 349574 N-tert-butyl-N'-[2-(4-methylphenylthio)-5-nitrobenzenesulfonyl]urea 349589 (E)-[2-(hydroxymethyl)-5-oxo-4-(phenylmethylene)-2,3-dihydrofur-2-yl]methyl 4-methyl-3-(methylethyl)pentanoate 349602 N-(4-amino-5-cyano-6-isopropylaminopyridin-2-yl)acetamide 349606 8-(1,3-dimethyl-1H-pyrazol-5-yl)-1,3-dipropyl-1H-purine-2,6-(3H,7H)-dione 349613 N-(4-amino-6-bromo-5-cyanopyridin-2-yl)-2-(2,5-dimethoxyphenyl)acetamide 349614 N-(4-amino-5-cyano-6-isopropoxypyridin-2-yl)acetamide 349622 1,3-Dipropyl-8-(1H-pyrazol-4-yl)-1H-purine-2,6(3H,7H)-dione 349624 N-(5,6-difluoro-1H-benzo[d]imidazol-2-yl)-3-nitrobenzamide 349625 N-(1-(2-hydroxyethyl)-1H-benzo[d]imidazol-2-yl)-3-nitrobenzamide 349627 3-(6-acetylamino-4-amino-3-cyanopyridin-2-yloxy)propionic acid 349628 N-[4-amino-5-cyano-6-(tetrahydrofuran-3-yloxy)pyridin-2-yl]-acetamide 349631 N-(1-isopropyl-1H-benzo[d]imidazol-2-yl)-3-nitrobenzamide 349633 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-dibutylaminoacetamide 349634 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-butylaminoacetamide 349645 2,4-dichloro-N-{2-[4-(2-guanidinoethyl)piperazin-1-yl]-1,1-dimethyl-2-oxoethyl}-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonamide 349658 N-(1-(3-hydroxypropyl)-1H-benzo[d]imidazol-2-yl)-3-nitrobenzamide 349660 N-(4-amino-6-butoxy-5-cyanopyridin-2-yl)acetamide 349665 1-(2-chloroethyl)-1-nitroso-3-methyl-3-{[4-(3-methylphenyl)amino]quinazolin-6-yl}urea 349666 1-(2-chloroethyl)-1-nitroso-3-methyl-3-{[4-(3-chloro-phenyl)amino]quinazolin-6-yl}urea 349667 2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-2-methyl-N-phenylpropionamide 349668 2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-N-(2-guanidinoethyl)-2-methylpropionamide 349687 3-(2-(3-nitrobenzamido)-1H-benzo[d]imidazol-1-yl)propanoic acid 349688 (+/-)-2-(cis-5-(4-(5-(4-cyclopentyl-3-fluorophenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-2-yl)acetic acid 349691 1-(2-chloroethyl)-1-nitroso-3-methyl-3-{[4-(3-bromophenyl)amino]quinazolin-6-yl}urea 349692 2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-N-(3-guanidinopropyl)-2-methylpropionamide 349698 8-(1-(2-chlorobenzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349699 8-(1-(3-chlorobenzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349713 (+/-)-2-(cis-5-(4-(5-(4-((S)-3,3-difluorocyclopentyl)phenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-2-yl)acetic acid 349718 2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-2-methyl-N-piperidin-4-ylpropionamide 349726 8-(1-(3,4-difluorobenzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1Hpurine-2,6(3H,7H)-dione 349727 8-(1-(3-chloro-2-fluorobenzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349729 8-(1-(3-fluorobenzyl)-1H-pyrazol-4-yl)-1,3-diisobutyl-1H-purine-2,6(3H,7H)-dione 349730 2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-2-methyl-N-(2-morpholin-4-ylethyl)propionamide 349734 N-(2-azepan-1-yl-1,1-dimethyl-2-oxoethyl)-2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonamide 349741 1-(2-(p-toluidino)-5-nitrophenylsulfonyl)-3-tert-butylurea 349744 2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-2-methyl-N-piperidin-4-ylmethyl-ropionamide 349749 (3R,5S,6S)-5-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-6-(4-fluorophenyl)-1,3-dimethylazepan-2-one 349750 (5S,6S,7S)-5-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-6-(4-fluorophenyl)-1,7-dimethylazepan-2-one 349751 8-(1-(2-fluoro-3-methylbenzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 349753 8-(1-(3-(trifluoromethyl)benzyl)-1H-pyrazol-4-yl)-1,3-diisobutyl-1H-purine-2,6(3H,7H)-dione 349759 2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-2-methyl-N-{3-[(pyridin-2-ylmethyl)amino]-propyl}propionamide 349761 2,4-dichloro-N-(2-[1,4]diazepan-1-yl-1,1-dimethyl-2-oxoethyl)-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonamide 349768 N-n-heptyl-N'-[2-(cyclohexylamino)-5-nitrobenzenesulfonyl]urea 349775 2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-2-methyl-N-(2-piperidin-1-yl-ethyl)propionamide 349778 N-[4-[4-(2,3-difluorophenyl)piperazin-1-yl]butyl][2.2]-paracyclophane-4-carboxamide 349779 N-tert-butyl-N'-[2-(2,6-dimethylphenylamino)-5-nitrobenzenesulfonyl]urea 349780 2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-N-(2-methoxyethyl)-2-methylpropionamide 349781 2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-N-(3-methoxypropyl)-2-methylpropionamide 349798 N-(1H-benzo[d]imidazol-2-yl)-4-fluoro-3-nitrobenzamide 349799 N-(1H-benzo[d]imidazol-2-yl)-4-methyl-3-nitrobenzamide 349800 N-(1-butyl-1H-benzo[d]imidazol-2-yl)-3-nitrobenzamide 349827 N-(1-butyl-1H-benzo[d]imidazol-2-yl)-3-chlorobenzamide 349831 N-[2-(4-methylphenylamino)-5-nitrobenzenesulfonyl]-piperidine-1-carboxamide 349837 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-(3-methoxyphenyl)acetamide 349838 2-(4-acetylamino-2,5-dimethoxyphenyl)-N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)acetamide 349840 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-(3-chlorophenyl)acetamide 349844 2,4-dichloro-N-[1,1-dimethyl-2-(4-methylpiperazin-1-yl)-2-oxoethyl]-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonamide 349847 (+/-)-3-(trans-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-2-yl)propanoic acid 349848 (+/-)-2-(cis-5-(4-(5-(4-cyclohexylphenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-2-yl)acetic acid 349856 N-(5,6-dimethyl-1H-benzo[d]imidazol-2-yl)-3-nitrobenzamide 349857 N-(1-ethyl-1H-benzo[d]imidazol-2-yl)-3-nitrobenzamide 349858 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-diethylaminoacetamide 349859 N-(4-amino-5-cyano-6-methoxypyridin-2-yl)acetamide 349860 N-[4-amino-5-cyano-6-(2-hydroxyethoxy)pyridin-2-yl]-2-(2,5-dimethoxyphenyl)acetamide 349865 1-(5-nitro-2-(o-tolyloxy)phenylsulfonyl)-3-pentylurea 349866 N-(4-amino-5-cyano-6-isopropoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamide 349869 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-(4-chlorophenyl)acetamide 349871 2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-2-methyl-N-(3-morpholin-4-yl-propyl)propionamide 349872 4-{2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-2-methylpropionyl}piperazine-1-carboxamidine 349874 (+/-)-2-(cis-5-(4-(5-(4-cyclopentyl-2-fluorophenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-2-yl)acetic acid 349875 N-n-pentyl-N'-[2-(4-methylphenylamino)-5-nitrobenzenesulfonyl]urea 349881 N-(1-(3-(dimethylamino)propyl)-1H-benzo[d]imidazol-2-yl)-3-nitrobenzamide 349882 N-(1-(2-(diethylamino)ethyl)-1H-benzo[d]imidazol-2-yl)-3-nitrobenzamide 349883 N-[4-amino-5-cyano-6-(2-methoxyethoxy)pyridin-2-yl]-2-(2,5-dimethoxyphenyl)acetamide 349884 N-[4-amino-5-cyano-6-(2-methanesulfonylethoxy)-2-pyridinyl]-2-(2,5-dimethoxyphenyl)acetamide 349896 2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-2-methyl-N-[3-(4-methylpiperazin-1-yl)propyl]-propionamide 349897 2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-N-[3-(4-(dimethylamino)benzylamino)propyl]-2-methylpropionamide 349902 N-n-hexyl-N'-[2-(cyclohexylamino)-5-nitrobenzenesulfonyl]urea 349906 8-(1-phenethyl-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6-(3H,7H)-dione 349907 N-(1-(2-morpholinoethyl)-1H-benzo[d]imidazol-2-yl)-3-nitrobenzamide 349908 3-nitro-N-(1-((tetrahydrofuran-2-yl)methyl)-1H-benzo[d]imidazol-2-yl)benzamide 349915 (3R,5S,6S)-5-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-6-(4-fluorophenyl)-3-methylazepan-2-one 349916 (5S,6S,7S)-5-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-6-(4-fluorophenyl)-7-methylazepan-2-one 349929 N-benzyl-N'-[2-(4-methylphenylamino)-5-nitrobenzenesulfonyl]urea 349935 4-phenyl-1-((1-phenyl-1H-pyrazol-4-yl)methyl)-1,2,3,6-tetrahydropyridine 349936 1-(4-(1H-pyrazol-1-yl)benzyl)-4-phenylpiperazine 349943 H-Tyr-Pro-Phe-Phe-NH-(CH2)5-NH-(C=S)-NH-fluorescein 349944 (4R,5S,7R)-5-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-4-(4-fluorophenyl)-1,7-dimethylazepan-2-one 349948 8-(1-benzyl-1H-pyrazol-4-yl)-1,3-diisobutyl-1H-purine-2,6-(3H,7H)-dione 349953 N-(3-benzylaminopropyl)-2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-2-methylpropionamide 349954 2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-N-[3-(4-fluorobenzylamino)propyl]-2-methylpropionamide 349955 4-[(3-{2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)-benzenesulfonylamino]-2-methylpropionylamino}propylamino)-methyl]benzamide 349966 4-phenyl-1-((1-phenyl-1H-1,2,3-triazol-4-yl)methyl)-1,2,3,6-tetrahydropyridine 349977 N-4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl-1(4,7)-benzofurano-4-(1,4)-benzolhexaphanyl-12-carboxamide 349981 2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-N-{3-[(furan-3-ylmethyl)amino]propyl}-2-methylpropionamide 349982 N-(3-aminopropyl)-4-{2-[2,4-dichloro-3-(2,4-dimethylquinolin-8-yloxymethyl)benzenesulfonylamino]-2-methylpropionyl}-piperazine-1-carboxamidine 349988 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-3-methylbutyramide 349994 N-(4-amino-5-chloro-6-ethoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamide 349997 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-(2-methoxyphenyl)acetamide 349999 1-phenyl-4-((1-(pyridin-2-yl)-1H-pyrazol-4-yl)methyl)piperazine 350002 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-phenylacetamide 350019 N-(1H-benzo[d]imidazol-2-yl)-3-cyanobenzamide 350024 N-(1-butyl-1H-benzo[d]imidazol-2-yl)-3,4-dichlorobenzamide 350026 N-cyclohexyl-N'-[2-(4-methylphenoxy)-5-nitrobenzenesulfonyl]urea 350027 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-(2,5-dibromophenyl)acetamide 350028 1-(2-methoxyphenyl)-4-((1-(pyridin-2-yl)-1H-pyrazol-4-yl)methyl)piperazine 350029 1-Phenyl-4-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperazine 350035 N-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-(2-chlorophenyl)acetamide 350051 N-(4-amino-5-cyano-6-isopropoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamide 350053 N-(1-butyl-1H-benzo[d]imidazol-2-yl)-4-methoxybenzamide 350054 (4R,5S,7R)-5-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-4-(4-fluorophenyl)-7-methylazepan-2-one 350055 N-n-butyl-N'-[2-(4-methylphenoxy)-5-nitrobenzenesulfonyl]urea 350056 1-(5-nitro-2-(m-tolyloxy)phenylsulfonyl)-3-pentylurea 350057 1-(4-Chlorophenyl)-4-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperazine 350067 2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-N-{3-[(1H-imidazol-4-ylmethyl)amino]propyl}-2-methylpropionamide 350077 2N-[3-(4-chlorobenzylamino)propyl]-2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-2-methylpropionamide 350078 2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-N-[3-(4-methoxybenzylamino)propyl]-2-methylpropionamide 350079 2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-N-[3-(4-hydroxybenzylamino)propyl]-2-methylpropionamide 350080 2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-2-methyl-N-[3-(4-methylbenzylamino)propyl]-propionamide 350081 N-(3-aminopropyl)-4-{2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-2-methylpropionyl}-piperazine-1-carboxamidine 350083 2-[2,4-dichloro-3-(2-methylquinolin-8-yloxymethyl)benzenesulfonylamino]-N-[3-(4-methanesulfonylbenzylamino)propyl]-2-methylpropionamide 350101 N-((R)-3-(4-chlorophenyl)-1-(4-(1-(cyclobutylamino)-3-cyclohexylpropan-2-yl)piperazin-1-yl)-1-oxopropan-2-yl)-2-(indolin-2-yl)acetamide 350102 N-((R)-3-(4-chlorophenyl)-1-(4-(3-cyclohexyl-1-morpholinopropan-2-yl)piperazin-1-yl)-1-oxopropan-2-yl)-2-(indolin-2-yl)acetamide 350103 2-{4-[(R)-3-(4-chloro-phenyl)-2-(2-2,3-dihydro-1H-indol-2-yl-acetylamino)-propionyl]-piperazin-1-yl}-2-cyclohexyl-N,N-diethyl-acetamide 350104 N-((R)-3-(4-chlorophenyl)-1-(4-(1-cyclohexyl-2-(methylsulfonamido)ethyl)piperazin-1-yl)-1-oxopropan-2-yl)-2-(indolin-2-yl)acetamide 350105 N-((R)-3-(4-chlorophenyl)-1-(4-(1-cyclohexyl-2-(N-ethylmethan-4-ylsulfonamido)ethyl)piperazin-1-yl)-1-oxopropan-2-yl)-2-(indolin-2-yl)acetamide 350156 N-(3-chloro-4-fluoro-phenyl)-2-[1-cyclopentyl-4-(3'-fluoro-biphenyl-4-yl)-piperidin-4-ylamino]-acetamide 350157 N-(4-(5-amino-1-(2,6-difluorobenzoyl)-1H-1,2,4-triazol-3-ylamino)phenylsulfonyl)-3-(4-methylpiperazin-1-yl)propanamide 350158 2-amino-N-(4-(5-amino-1-(2,6-difluorobenzoyl)-1H-1,2,4-triazol-3-ylamino)phenylsulfonyl)acetamide 350159 N-(5-(5-(1-acetylpiperazine-4-carbonyl)-2-methylphenylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 350160 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-4-chlorophenylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 350161 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-4,5-dimethylphenylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 350195 (2S)-1-(5-(3-methyl-1H-indazol-5-yl)pyridin-3-yloxy)-3-(2-methyl-1H-indol-3-yl)propan-2-amine 350196 3-(2-chloro-6-methylphenyl)-1-(6-(4-(diethylamino)phenylamino)pyrimidin-4-yl)-1-(3-(dimethylamino)propyl)urea 350197 3-(2,6-dichlorophenyl)-1-(3-(dimethylamino)propyl)-1-(6-(methylamino)pyrimidin-4-yl)urea 350199 N-(3-chloro-4-fluoro-phenyl)-2-[1-cyclopentyl-4-(3'-formyl-biphenyl-4-yl)-piperidin-4-ylamino]-acetamide 350200 N-(4-(5-amino-1-(2,6-difluorobenzoyl)-1H-1,2,4-triazol-3-ylamino)phenylsulfonyl)-2-(2-methoxyethoxy)acetamide 350201 N-(5-(3-(1-acetylpiperazine-4-carbonyl)benzyl)thiazol-2-yl)-4-(dimethylamino)benzamide 350202 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-4-aminophenylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 350203 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-4-hydroxyphenylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 350204 N-(5-(5-(1-acetylpiperazine-4-carbonyl)-2,3-dimethylphenylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 350217 6-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroquinoline 350218 1-ethyl-6-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroquinoline 350222 (R)-N-((R)-3-(4-chlorophenyl)-1-(4-(1-(diethylamino)propan-2-yl)piperazin-1-yl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 350223 (R)-N-((R)-3-(4-chlorophenyl)-1-(4-(1-cyclopentyl-2-(diethylamino)ethyl)piperazin-1-yl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 350224 (R)-N-((R)-3-(4-chlorophenyl)-1-(4-(1-cyclohexyl-2-(diethylamino)ethyl)piperazin-1-yl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 350227 (2S)-1-(benzo[b]thiophen-3-yl)-3-(5-(3-methyl-1H-indazol-5-yl)pyridin-3-yloxy)propan-2-amine 350228 (2S)-1-(5-(isoquinolin-6-yl)pyridin-3-yloxy)-3-(pyridin-4-yl)propan-2-amine 350229 3-(2,6-dichlorophenyl)-1-(6-(4-(2-(diethylamino)ethoxy)phenylamino)pyrimidin-4-yl)-1-(3-(dimethylamino)propyl)urea 350230 1-benzyl-3-(2-chloro-6-methylphenyl)-1-(6-(4-fluorophenylamino)pyrimidin-4-yl)urea 350231 3-(2,6-dichlorophenyl)-1-(6-(3-(dimethylamino)propylamino)pyrimidin-4-yl)-1-methylurea 350232 N-(3-chloro-4-fluoro-phenyl)-2-[1-cyclopentyl-4-(4'-fluoro-biphenyl-4-yl)-piperidin-4-ylamino]-acetamide 350233 2-[4-(2'-chloro-biphenyl-4-yl)-1-cyclopentyl-piperidin-4-ylamino]-N-(3-chloro-4-fluoro-phenyl)-acetamide 350235 N-(5-(5-(4-acetylpiperazine-1-carbonyl)-4-methoxy-2-methylphenylthio)thiazol-2-yl)-4-((3,3-dimethylbutan-2-ylamino)methyl)benzamide 350236 1-(6-(4-(2-(diethylamino)ethoxy)phenylamino)pyrimidin-4-yl)-1-methyl-3-(2-methyl-5-((3-(trifluoromethyl)phenyl)carbamoyl)phenyl)urea 350237 1-(6-(4-(2-(diethylamino)ethoxy)phenylamino)pyrimidin-4-yl)-1-methyl-3-(2-methyl-5-(1-methyl-1H-indole-2-carboxamido)phenyl)urea 350238 3-(5-(benzo[b]thiophene-2-carboxamido)-2-methylphenyl)-1-(6-(4-(2-(diethylamino)ethoxy)phenylamino)pyrimidin-4-yl)-1-methylurea 350239 1-(6-(4-(2-(diethylamino)ethoxy)phenylamino)pyrimidin-4-yl)-1-methyl-3-(2-methyl-5-(3-(trifluoromethyl)benzamido)phenyl)urea 350240 N-(5-((3-(1-acetylpiperazine-4-carbonyl)benzyloxy)methyl)thiazol-2-yl)-4-tert-butylbenzamide 350241 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-4-methoxyphenylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 350246 N-((R)-3-(4-chlorophenyl)-1-(4-(1,3-dicyclohexylpropan-2-yl)piperazin-1-yl)-1-oxopropan-2-yl)-2-(indolin-2-yl)acetamide 350248 N-((R)-3-(4-chlorophenyl)-1-(4-(1-cyclohexyl-2-(diethylamino)ethyl)piperazin-1-yl)-1-oxopropan-2-yl)-2-(indolin-2-yl)acetamide 350253 1-(cyclohexylmethyl)-6-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroquinoline 350254 1-(phenylsulfonyl)-6-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroquinoline 350259 3-(2-chlorophenyl)-1-methyl-1-(6-(4-(4-methylpiperazin-1-yl)phenylamino)pyrimidin-4-yl)urea 350260 3-(2,6-dichlorophenyl)-1-(6-(4-(2-(diethylamino)ethoxy)phenylamino)pyrimidin-4-yl)-1-methylurea 350261 2-{[4-(3'-cyano-biphenyl-4-yl)-1-cyclopentyl-piperidin-4-yl]-methyl-amino}-N-(3,5-dichloro-phenyl)-acetamide 350262 N-(4-chloro-3-trifluoromethyl-phenyl)-2-[4-(3'-cyano-biphenyl-4-yl)-1-cyclopentyl-piperidin-4-yloxy]-acetamide 350263 N-(3-chloro-4-fluoro-phenyl)-2-[1-cyclopentyl-4-(3'-trifluoromethyl-biphenyl-4-yl)-piperidin-4-ylamino]-acetamide 350264 N-(3-chloro-4-fluoro-phenyl)-2-[1-cyclopentyl-4-(2'-fluoro-biphenyl-4-yl)-piperidin-4-ylamino]-acetamide 350266 N-(5-(((3-(1-acetylpiperazine-4-carbonyl)benzyl)(methyl)amino)methyl)thiazol-2-yl)-4-tert-butylbenzamide 350281 7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroquinoline 350282 1-ethyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroquinoline 350289 3-(2-chloro-6-methylphenyl)-1-(6-(4-(2-(diethylamino)ethoxy)phenylamino)pyrimidin-4-yl)-1-methylurea 350290 3-(2-chloro-6-(trifluoromethyl)phenyl)-1-(6-(4-(2-(diethylamino)ethoxy)phenylamino)pyrimidin-4-yl)-1-methylurea 350291 2-(4-biphenyl-4-yl-1-cyclopentyl-piperidin-4-ylamino)-N-(3-chloro-4-fluoro-phenyl)-acetamide 350292 2-[4-(3'-chloro-biphenyl-4-yl)-1-cyclopentyl-piperidin-4-ylamino]-N-(3-chloro-4-fluoro-phenyl)-acetamide 350295 N-(5-((3-(1-acetylpiperazine-4-carbonyl)benzylamino)methyl)thiazol-2-yl)-4-tert-butylbenzamide 350296 N-(5-(3-(1-acetylpiperazine-4-carbonyl)phenylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 350308 7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 350309 2-ethyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 350310 2-(cyclohexylmethyl)-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 350323 1-(6-(4-(2-(diethylamino)ethoxy)phenylamino)pyrimidin-4-yl)-3-(2,6-difluorophenyl)-1-methylurea 350325 N-(3-chloro-4-fluoro-phenyl)-2-[4-(4'-cyano-biphenyl-4-yl)-1-cyclopentyl-piperidin-4-ylamino]-acetamide 350326 N-(3-chloro-4-fluoro-phenyl)-2-[1-cyclopentyl-4-(3'-trifluoromethoxy-biphenyl-4-yl)-piperidin-4-ylamino]-acetamide 350341 N-[(R)-2-{4-[2-(acetyl-ethyl-amino)-1-cyclohexyl-ethyl]-piperazin-1-yl}-1-(4-chloro-benzyl)-2-oxo-ethyl]-2-(2,3-dihydro-1H-indol-2-yl)-acetamide 350342 N-((R)-3-(4-chlorophenyl)-1-(4-(1-cyclohexyl-2-(2,5-dioxopyrrolidin-1-yl)ethyl)piperazin-1-yl)-1-oxopropan-2-yl)-2-(indolin-2-yl)acetamide 350348 2-(phenylsulfonyl)-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 350349 2-(phenylsulfonyl)-6-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 350352 3-isopropyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-tetrahydro-1H-benzo[d]azepine 350357 2-{[4-(3'-cyano-biphenyl-4-yl)-1-cyclopentyl-piperidin-4-yl]-methyl-amino}-N-(3,5-dichloro-phenyl)-acetamide 350358 N-(3-chloro-4-fluoro-phenyl)-2-[1-cyclopentyl-4-(4'-trifluoromethyl-biphenyl-4-yl)-piperidin-4-ylamino]-acetamide 350359 N-(3-chloro-4-fluoro-phenyl)-2-[1-cyclopentyl-4-(3'-methoxy-biphenyl-4-yl)-piperidin-4-ylamino]-acetamide 350366 4-(3'-cyano-biphenyl-4-yl)-4-[2-(3,4-difluoro-phenylcarbamoyl)-ethyl]-piperidine-1-carboxylic acid benzylester 350367 3-[4-(3'-cyano-biphenyl-4-yl)-1-cyclopropylmethyl-piperidin-4-yl]-N-(3,4-difluoro-phenyl)-propionamide 350375 3,4-Dihydro-1H-isoquinoline-2-carboxylic acid ((R)-1-(4-chloro-benzyl)-2-{4-[2-diethylamino-1-(2-fluoro-phenyl)-ethyl]-piperazin-1-yl}-2-oxo-ethyl)-amide 350384 (6-(3-(piperidin-1-yl)propoxy)-3,4-dihydroisoquinolin-2(1H)-yl)(thiophen-2-yl)methanone 350385 (7-(3-(piperidin-1-yl)propoxy)-3,4-dihydroisoquinolin-2(1H)-yl)(thiophen-2-yl)methanone 350387 N-isopropyl-7-(3-(piperidin-1-yl)propoxy)-1,2,4,5-tetrahydrobenzo[d]azepine-3-carboxamide 350388 3-(methylsulfonyl)-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-tetrahydro-1H-benzo[d]azepine 350392 (R)-N-((R)-3-(4-chlorophenyl)-1-(4-(1-cycloheptyl-2-(diethylamino)ethyl)piperazin-1-yl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 350393 (R)-N-((R)-3-(4-chlorophenyl)-1-(4-(3-cyclohexyl-1-(diethylamino)propan-2-yl)piperazin-1-yl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 350394 N-((R)-3-(4-chlorophenyl)-1-(4-(3-cyclohexyl-1-(diethylamino)propan-2-yl)piperazin-1-yl)-1-oxopropan-2-yl)-2-(indolin-2-yl)acetamide 350397 2-{[4-(3'-cyano-biphenyl-4-yl)-1-cyclopentyl-piperidin-4-yl]-methyl-amino}-N-(4-fluoro-3-trifluoromethyl-phenyl)-acetamide 350398 N-(3-chloro-4-fluoro-phenyl)-2-{[4-(3'-cyano-biphenyl-4-yl)-1-cyclopentyl-piperidin-4-yl]-methyl-amino}-acetamide 350399 2-[4-(4'-chloro-biphenyl-4-yl)-1-cyclopentyl-piperidin-4-ylamino]-N-(3-chloro-4-fluoro-phenyl)-acetamide 350403 (R)-1-benzyl-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 350407 3-[4-(3'-cyano-biphenyl-4-yl)-1-cyclobutyl-piperidin-4-yl]-N-(3,4-difluoro-phenyl)-propionamide 350408 N-((R)-3-(4-chlorophenyl)-1-(4-(2,6-dimethylheptan-4-yl)piperazin-1-yl)-1-oxopropan-2-yl)-2-(indolin-2-yl)acetamide 350409 N-((R)-3-(4-chlorophenyl)-1-(4-(dicyclohexylmethyl)piperazin-1-yl)-1-oxopropan-2-yl)-2-(indolin-2-yl)acetamide 350415 8-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 350418 1-(cyclohexylmethyl)-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroquinoline 350419 1-(7-(3-(piperidin-1-yl)propoxy)-1,2,4,5-tetrahydrobenzo[d]azepin-3-yl)ethanone 350420 2-isopropyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 350429 2-[4-(3'-cyano-biphenyl-4-yl)-1-cyclopentyl-piperidin-4-yloxy]-N-(3,5-dichloro-phenyl)-acetamide 350438 3-[4-(3'-cyano-biphenyl-4-yl)-1-cyclopentyl-piperidin-4-yl]-N-(3,4-difluoro-phenyl)-propionamide 350439 N-((R)-3-(4-chlorophenyl)-1-(4-(1-cyclohexyl-3-methylbutyl)piperazin-1-yl)-1-oxopropan-2-yl)-2-(indolin-2-yl)acetamide 350448 1-(phenylsulfonyl)-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroquinoline 350449 (7-(3-(piperidin-1-yl)propoxy)-3,4-dihydroquinolin-1(2H)-yl)(thiophen-2-yl)methanone 350450 N-isopropyl-7-(3-(piperidin-1-yl)propoxy)-3,4-dihydroisoquinoline-2(1H)-carboxamide 350451 2-(methylsulfonyl)-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 350456 2-(2-(3-(2-(bicyclo[2.2.1]heptan-2-yl)ethyl)-1,2,4-oxadiazol-5-yl)-1H-indol-4-yl)-N,N-dimethylethanamine 350463 N-(3-chloro-4-fluoro-phenyl)-2-[1-cyclopentyl-4-(2',6'-dichloro-biphenyl-4-yl)-piperidin-4-ylamino]-acetamide 350465 (R)-N-((2-(4-(2-(3-aminopropanamido)-3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)pyridin-3-yl)methyl)benzamide 350466 (R)-N-((2-(4-(2-(3-aminopropanamido)-3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)pyridin-3-yl)methyl)-4-methoxybenzamide 350467 (R)-3-amino-N-(3-(2,4-dichlorophenyl)-1-(4-(3-((2-(2-fluorophenyl)acetamido)methyl)pyridin-2-yl)piperazin-1-yl)-1-oxopropan-2-yl)propanamide 350468 (R)-3-amino-N-(3-(2,4-dichlorophenyl)-1-(4-(3-((2-(2-methoxyphenyl)acetamido)methyl)pyridin-2-yl)piperazin-1-yl)-1-oxopropan-2-yl)propanamide 350469 (R)-3-amino-N-(3-(2,4-dichlorophenyl)-1-(4-(3-((2-(4-fluorophenyl)acetamido)methyl)pyridin-2-yl)piperazin-1-yl)-1-oxopropan-2-yl)propanamide 350470 (R)-3-amino-N-(3-(2,4-dichlorophenyl)-1-(4-(3-((2-(4-methoxyphenyl)acetamido)methyl)pyridin-2-yl)piperazin-1-yl)-1-oxopropan-2-yl)propanamide 350471 4'-[1-(1-benzyl-piperidin-4-yl)-3-(4-chloro-5-fluoro-1H-benzoimidazol-2-yl)-propyl]-biphenyl-3-carbonitrile 350472 4'-[1-(1-benzyl-piperidin-4-yl)-3-(4,6-dichloro-1H-benzoimidazol-2-yl)-propyl]-biphenyl-3-carbonitrile 350473 4'-[1-(1-benzyl-piperidin-4-yl)-3-(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-propyl]-biphenyl-3-carbonitrile 350474 (R)-2-methoxyphenyl (2-(4-(2-(3-aminopropanamido)-3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)pyridin-3-yl)methylcarbamate 350475 (R)-benzyl (2-(4-(2-(3-aminopropanamido)-3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)pyridin-3-yl)methylcarbamate 350476 4-[[(6-chloro-5-fluoro-1H-benzoimidazol-2-ylmethyl)-amino]-(3'-cyano-biphenyl-4-yl)-methyl]-piperidine-1-carboxylic acid benzyl ester 350477 (R)-1-((2-(4-(2-(3-aminopropanamido)-3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)pyridin-3-yl)methyl)-3-(2-fluorophenyl)urea 350478 (R)-1-((2-(4-(2-(3-aminopropanamido)-3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)pyridin-3-yl)methyl)-3-(2-methoxyphenyl)urea 350480 (R)-1-(2-fluorobenzyl)-3-((2-(4-(2-(3-aminopropanamido)-3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)pyridin-3-yl)methyl)urea 350481 (R)-1-(2-methoxybenzyl)-3-((2-(4-(2-(3-aminopropanamido)-3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)pyridin-3-yl)methyl)urea 350492 2-ethyl-8-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 350506 1-(7-(3-(piperidin-1-yl)propoxy)-3,4-dihydroisoquinolin-2(1H)-yl)ethanone 350511 2-(2-(3-(3-cyclohexylpropyl)-1,2,4-oxadiazol-5-yl)-1H-indol-4-yl)-N,N-dimethylethanamine 350520 3-[4-(3'-cyano-biphenyl-4-yl)-piperidin-4-yl]-N-(3,4-difluoro-phenyl)-propionamide 350521 (R)-N-((2-(4-(2-(3-aminopropanamido)-3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)pyridin-3-yl)methyl)-4-fluorobenzamide 350530 2-(cyclohexylmethyl)-8-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 350541 (2S)-1-(5-(3-methyl-1H-indazol-5-yl)pyridin-3-yloxy)-3-(naphthalen-2-yl)propan-2-amine 350547 3-(5-((5-tert-butylisoxazol-3-yl)carbamoyl)-2-methylphenyl)-1-(6-(4-(2-(diethylamino)ethoxy)phenylamino)pyrimidin-4-yl)-1-methylurea 350548 N-(3-chloro-4-fluoro-phenyl)-2-[1-cyclopentyl-4-(3',4'-dichloro-biphenyl-4-yl)-piperidin-4-ylamino]-acetamide 350550 (R)-N-((2-(4-(2-(3-aminopropanamido)-3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)pyridin-3-yl)methyl)furan-2-carboxamide 350574 2-(2-(3-(2-cyclopentylethyl)-1,2,4-oxadiazol-5-yl)-1H-indol-4-yl)-N,N-dimethylethanamine 350575 (2S)-1-(5-(3-methyl-1H-indazol-5-yl)pyridin-3-yloxy)-3-(naphthalen-1-yl)propan-2-amine 350576 (2S)-1-(2-methoxynaphthalen-1-yl)-3-(5-(3-methyl-1H-indazol-5-yl)pyridin-3-yloxy)propan-2-amine 350577 (2S)-1-cyclohexyl-3-(5-(3-methyl-1H-indazol-5-yl)pyridin-3-yloxy)propan-2-amine 350578 (1S)-2-(5-(3-methyl-1H-indazol-5-yl)pyridin-3-yloxy)-1-phenylethanamine 350581 N-(3-chloro-4-fluoro-phenyl)-2-[1-cyclopentyl-4-(3',5'-dichloro-biphenyl-4-yl)-piperidin-4-ylamino]-acetamide 350582 ethyl 4-(4-(5-amino-1-(2,6-difluorobenzoyl)-1H-1,2,4-triazol-3-ylamino)phenylsulfonamido)-4-oxobutanoate 350583 (R)-2-amino-N-(4-(5-amino-1-(2,6-difluorobenzoyl)-1H-1,2,4-triazol-3-ylamino)phenylsulfonyl)-3-hydroxypropanamide 350584 (R)-N-((2-(4-(2-(3-aminopropanamido)-3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)pyridin-3-yl)methyl)thiophene-2-carboxamide 350593 2-ethyl-5-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 350594 1-(cyclohexylmethyl)-5-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroquinoline 350596 2-ethyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-tetrahydro-1H-benzo[c]azepine 350597 2-benzyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-tetrahydro-1H-benzo[c]azepine 350602 (R)-N-((R)-3-(4-chlorophenyl)-1-(4-(1-((diethylamino)methyl)cyclopentyl)piperazin-1-yl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 350603 2-(2-(3-(cyclohexylmethyl)-1,2,4-oxadiazol-5-yl)-1H-indol-4-yl)-N,N-dimethylethanamine 350606 (2S)-1-(5-(3-methyl-1H-indazol-5-yl)pyridin-3-yloxy)-3-(quinolin-3-yl)propan-2-amine 350607 (2S)-4-(5-(3-methyl-1H-indazol-5-yl)pyridin-3-yloxy)-1-phenylbutan-2-amine 350608 (2R)-5-(5-(3-methyl-1H-indazol-5-yl)pyridin-3-yloxy)-1-phenylpentan-2-amine 350609 (2S)-1-(1H-indol-3-yl)-3-(5-(3-methyl-1H-indazol-5-yl)pyridin-3-ylthio)propan-2-amine 350611 N-(3-chloro-4-fluoro-phenyl)-2-[1-cyclopentyl-4-(3',5'-difluoro-biphenyl-4-yl)-piperidin-4-ylamino]-acetamide 350613 1-(4-((5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)methoxy)benzyl)azetidine-3-carboxylic acid 350614 N-(5-(4-acetamido-3-(1-acetylpiperazine-4-carbonyl)phenylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 350620 N-((R)-3-(4-chlorophenyl)-1-(4-(1-cyclohexyl-2-(N-ethylmethan-4-ylsulfonamido)ethyl)piperazin-1-yl)-1-oxopropan-2-yl)-2H-isoindole-2-carboxamide 350625 2-(cyclohexylmethyl)-5-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 350628 2-isopropyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-tetrahydro-1H-benzo[c]azepine 350629 N-isopropyl-7-(3-(piperidin-1-yl)propoxy)-4,5-dihydro-1H-benzo[c]azepine-2(3H)-carboxamide 350633 2-(2-(3-(2-cyclohexylethyl)-1,2,4-oxadiazol-5-yl)-1H-indol-4-yl)-N,N-dimethylethanamine 350635 (S)-1-(5-(3-methyl-1H-indazol-5-yl)pyridin-3-yloxy)-3-phenylpropan-2-amine 350636 (2S)-1-(5-(3-methyl-1H-indazol-5-yl)pyridin-3-yloxy)-3-(pyridin-4-yl)propan-2-amine 350637 (2S)-1-(5-(3-methyl-1H-indazol-5-yl)pyridin-3-yloxy)-5-phenylpentan-2-amine 350641 1-(6-(4-(2-(diethylamino)ethoxy)phenylamino)pyrimidin-4-yl)-3-(5-methoxy-2-methylphenyl)-1-methylurea 350642 N-(3-chloro-4-fluoro-phenyl)-2-[1-cyclopentyl-4-(2',5'-dichloro-biphenyl-4-yl)-piperidin-4-ylamino]-acetamide 350643 (R)-N-(1-(4-(3-(acetamidomethyl)pyridin-2-yl)piperazin-1-yl)-3-(2,4-dichlorophenyl)-1-oxopropan-2-yl)-3-aminopropanamide 350644 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-5-aminophenylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 350655 6-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 350663 2-(methylsulfonyl)-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-tetrahydro-1H-benzo[c]azepine 350665 3-ethyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-tetrahydro-1H-benzo[d]azepine 350670 (1S)-2-(5-(isoquinolin-6-yl)pyridin-3-yloxy)-1-phenylethanamine 350672 N-((S)-2-amino-3-phenylpropyl)-5-(3-methyl-1H-indazol-5-yl)pyridin-3-amine 350673 3-(2,6-dichlorophenyl)-1-(3-(dimethylamino)propyl)-1-(6-(4-morpholinophenylamino)pyrimidin-4-yl)urea 350674 1-(6-(4-(2-(diethylamino)ethoxy)phenylamino)pyrimidin-4-yl)-3-(5-hydroxy-2-methylphenyl)-1-methylurea 350675 3-(5-hydroxy-2-methylphenyl)-1-methyl-1-(6-(4-morpholinophenylamino)pyrimidin-4-yl)urea 350676 N-(4-(5-amino-1-(2,6-difluorobenzoyl)-1H-1,2,4-triazol-3-ylamino)phenylsulfonyl)-3-morpholinopropanamide 350677 4-(4-(5-amino-1-(2,6-difluorobenzoyl)-1H-1,2,4-triazol-3-ylamino)phenylsulfonamido)-4-oxobutanoic acid 350678 (R)-3-amino-N-(3-(2,4-dichlorophenyl)-1-(4-(3-((2-methoxyacetamido)methyl)pyridin-2-yl)piperazin-1-yl)-1-oxopropan-2-yl)propanamide 350679 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-4-methylphenylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 350680 N-(5-(3-(1-acetylpiperazine-4-carbonyl)-5-(trifluoromethyl)phenylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 350689 2-ethyl-6-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 350690 2-(cyclohexylmethyl)-6-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 350692 3-(cyclohexylmethyl)-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-tetrahydro-1H-benzo[d]azepine 350697 (2S)-1-cyclohexyl-3-(5-(isoquinolin-6-yl)pyridin-3-yloxy)propan-2-amine 350698 (S)-1-(1H-indol-3-yl)-3-(5-(3-methyl-1H-indazol-5-yl)pyridin-3-yloxy)propan-2-amine 350700 3-(2-chlorophenyl)-1-(6-(4-(diethylamino)phenylamino)pyrimidin-4-yl)-1-(3-(dimethylamino)propyl)urea 350701 3-(2,6-dichlorophenyl)-1-(4-methylpiperazin-1-yl)-1-(6-(4-morpholinophenylamino)pyrimidin-4-yl)urea 350706 N-((S)-3-(1H-indol-3-yl)-1-(5-(thieno[2,3-c]pyridin-2-yl)pyridin-3-yloxy)propan-2-yl)thieno[2,3-c]pyridin-2-amine 350707 (S)-3-(2-chlorophenyl)-1-(4-fluorophenyl)-1-(2-(3-hydroxy-3-methylbutan-2-ylamino)pyrimidin-4-yl)urea 350708 (S)-1-(4-fluorophenyl)-1-(2-(3-hydroxy-3-methylbutan-2-ylamino)pyrimidin-4-yl)-3-o-tolylurea 350712 (S)-N-(1-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-2,5-dioxopyrrolidin-3-yl)cyclohexanecarboxamide 350713 (S)-N-(1-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-2,5-dioxopyrrolidin-3-yl)benzamide 350714 6-chloro-2-[4-(4-chlorophenyl)piperazin-1-ylmethyl]imidazo[1,2-b]pyridazine 350716 8-bromo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]-6-methylimidazo[1,2-a]pyridine 350721 (S)-1-(2-(1-methoxypropan-2-ylamino)pyrimidin-4-yl)-1-phenyl-3-o-tolylurea 350723 (E)-1-allyl-3-(3,4-dichlorophenylimino)indolin-2-one 350724 1-(ethylpropyl)-3-{[3-(trifluoromethyl)phenyl]azamethylene}benzo[d]azolidin-2-one 350725 1-(2-propynyl)-3-{[3-(trifluoromethyl)phenyl]azamethylene}benzo[d]azolidin-2-one 350734 N-((S)-3-(1H-indol-3-yl)-1-(5-(thieno[3,2-c]pyridin-2-yl)pyridin-3-yloxy)propan-2-yl)thieno[3,2-c]pyridin-2-amine 350737 ethyl 4-(4-(3-(2-chlorophenyl)-1-(4-fluorophenyl)ureido)pyrimidin-2-ylamino)piperidine-1-carboxylate 350738 3-(2-chlorophenyl)-1-(4-fluorophenyl)-1-(2-(1-(propylsulfonyl)piperidin-4-ylamino)pyrimidin-4-yl)urea 350741 Adamantane-1-carboxylic acid ((S)-1-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]-propyl}-2,5-dioxo-pyrrolidin-3-yl)-amide 350742 (S)-N-(1-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2,5-dioxopyrrolidin-3-yl)acetamide 350743 2-[4-(4-fluorophenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyrazine 350744 2-[4-(4-fluorophenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyrimidine 350745 8-iodo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]-6-methylimidazo[1,2-a]pyridine 350749 3-(2-chlorophenyl)-1-(6-(4-fluorophenylamino)pyrimidin-4-yl)-1-methylurea 350751 (S)-3-(2-chlorophenyl)-1-(3-fluorophenyl)-1-(2-(1-phenylethylamino)pyrimidin-4-yl)urea 350752 1,3-dihydro-1-phenyl-3-[[3-(trilfluoromethyl)phenyl]imino]-2H-indol-2-one 350754 3-(1-(1H-imidazol-2-yl)-2-methylpropan-2-yl)-5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)indolin-2-one 350757 (R)-N-(1-(3-(3-chloro-5-fluorophenyl)-3-(4-(methylsulfonyl)phenyl)propyl)piperidin-4-yl)-N-ethyl-2-(4-(methylsulfonyl)phenyl)acetamide 350758 (R)-N-(1-(3-(3-tert-butylphenyl)-3-(4-(methylsulfonyl)phenyl)propyl)piperidin-4-yl)-N-ethyl-2-(4-(methylsulfonyl)phenyl)acetamide 350759 (R)-N-ethyl-N-(1-(3-(3-isopropylphenyl)-3-(4-(methylsulfonyl)phenyl)propyl)piperidin-4-yl)-2-(4-(methylsulfonyl)phenyl)acetamide 350766 N-((S)-1-(5-(benzo[c][1,2,5]oxadiazol-5-yl)pyridin-3-yloxy)-3-(1H-indol-3-yl)propan-2-yl)benzo[c][1,2,5]oxadiazol-5-amine 350768 N-(5-(5-(1-acetylpiperazine-4-carbonyl)-2,4-dimethylphenylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 350771 4-(3'-cyano-biphenyl-4-yl)-N-(3,4-difluoro-phenyl)-4-(1-methanesulfonyl-piperidin-4-yl)-butyramide 350773 N-((S)-1-{4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl}pyrrolidin-2,5-dion-3-yl)cyclopentanecarboxamide 350775 2-[4-(3,4-dichlorophenyl)piperazin-1-ylmethyl]-6-(piperidin-1-yl)imidazo[1,2-b]pyridazine 350780 3-(2-chlorophenyl)-1-(6-(4-(diethylamino)phenylamino)pyrimidin-4-yl)-1-methylurea 350781 3-(2,6-dichlorophenyl)-1-methyl-1-(6-(4-morpholinophenylamino)pyrimidin-4-yl)urea 350785 5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)-3-(2-methyl-1-(thiophen-2-yl)propan-2-yl)indolin-2-one 350786 ethyl 3-((benzyl(methyl)amino)methyl)-2-(4-methoxyphenyl)-7-methyl-4-oxo-4,7-dihydrothieno[2,3-b]pyridine-5-carboxylate 350787 ethyl 7-(2-methoxybenzyl)-3-((dimethylamino)methyl)-2-(4-methoxyphenyl)-4-oxo-4,7-dihydrothieno[2,3-b]pyridine-5-carboxylate 350788 (R)-N-(1-(3-(3-cyanophenyl)-3-(4-(methylsulfonyl)phenyl)propyl)piperidin-4-yl)-N-ethyl-2-(4-(methylsulfonyl)phenyl)acetamide 350789 ethyl 7-(3-methoxybenzyl)-3-((benzyl(methyl)amino)methyl)-2-(4-methoxyphenyl)-4-oxo-4,7-dihydrothieno[2,3-b]pyridine-5-carboxylate 350790 ethyl 7-(4-methoxybenzyl)-3-((benzyl(methyl)amino)methyl)-2-(4-methoxyphenyl)-4-oxo-4,7-dihydrothieno[2,3-b]pyridine-5-carboxylate 350793 ethyl 7-(4-fluorobenzyl)-3-((benzyl(methyl)amino)methyl)-2-(4-methoxyphenyl)-4-oxo-4,7-dihydrothieno[2,3-b]pyridine-5-carboxylate 350796 6-{5-[(2S)-3-(1H-indol-3-yl)-2-[(2-oxo-2,3-dihydro-1H-indol-6-yl)amino]propoxy]pyridin-3-yl}-2,3-dihydro-1H-indol-2-one 350800 4a-(3'-cyano-biphenyl-4-yl)-N-(3,4-difluoro-phenyl)-4-piperidin-4-yl-butyramide 350801 2-[4-(4-fluorophenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine 350802 2-[4-(3,4-dichlorophenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine 350803 2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine 350809 (R)-N-(1-(4-(3-((2-methoxyphenethylamino)methyl)pyridin-2-yl)piperazin-1-yl)-3-(2,4-dichlorophenyl)-1-oxopropan-2-yl)acetamide 350810 3-(2-chloro-6-methylphenyl)-1-methyl-1-(6-(4-morpholinophenylamino)pyrimidin-4-yl)urea 350811 3-(2-chlorophenyl)-1-methyl-1-(6-(4-morpholinophenylamino)pyrimidin-4-yl)urea 350814 5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)-3-(1-(furan-2-yl)-2-methylpropan-2-yl)indolin-2-one 350815 N-methoxy-3-((2-(pyridin-2-ylamino)thiazol-5-ylthio)methyl)benzamide 350817 ethyl 7-(2-methoxybenzyl)-3-((benzyl(methyl)amino)methyl)-4-oxo-2-phenyl-4,7-dihydrothieno[2,3-b]pyridine-5-carboxylate 350821 N-(((1R,3S)-3-(N-benzylpivalamido)cyclohexyl)methyl)-4-fluoro-N-(3-(2-(pyrrolidin-1-yl)ethoxy)phenyl)benzamide 350823 5-{5-[(2S)-3-(1H-indol-3-yl)-2-[(2-oxo-2,3-dihydro-1H-indol-5-yl)amino]propoxy]pyridin-3-yl}-2,3-dihydro-1H-indol-2-one 350829 (R)-phenyl (2-(4-(2-(3-aminopropanamido)-3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)pyridin-3-yl)methylcarbamate 350831 2-[4-(4-chlorophenyl)piperazin-1-yl)methyl]imidazo[1,2-a]pyridine 350836 (R)-N-(3-(2,4-dichlorophenyl)-1-oxo-1-(4-(3-((2-(thiophen-2-yl)ethylamino)methyl)pyridin-2-yl)piperazin-1-yl)propan-2-yl)acetamide 350837 3-(2,6-dichlorophenyl)-1-methyl-1-(6-(4-(4-methylpiperazin-1-yl)phenylamino)pyrimidin-4-yl)urea 350838 3-(2-chloro-6-methylphenyl)-1-methyl-1-(6-(4-(4-methylpiperazin-1-yl)phenylamino)pyrimidin-4-yl)urea 350841 5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)-3-(2-methyl-1-(5-methylfuran-2-yl)propan-2-yl)indolin-2-one 350843 N-methyl-3-((2-(pyridin-2-ylamino)thiazol-5-ylthio)methyl)benzamide 350845 ethyl 7-benzyl-3-((benzyl(methyl)amino)methyl)-2-(2-methoxyphenyl)-4-oxo-4,7-dihydrothieno[2,3-b]pyridine-5-carboxylate 350849 ethyl 3-(N-benzyl-N-methylaminomethyl)-7-(2,6-difluorobenzyl)-4,7-dihydro-4-oxo-2-(4-propionylamidophenyl)thieno[2,3-b]pyridine-5-carboxylate 350852 rac-N-((3-(N-(3-chlorobenzyl)-2,2,2-trichloroacetamido)cyclohexyl)methyl)-4-fluoro-N-(3-(2-(pyrrolidin-1-yl)ethoxy)phenyl)benzamide 350853 rac-N-((3-(N-(3-chlorobenzyl)-2,2,2-trichloroacetamido)cyclohexyl)methyl)-4-fluoro-N-(3-(2-(piperidin-1-yl)ethoxy)phenyl)benzamide 350860 (R)-1-((2-(4-(2-(3-aminopropanamido)-3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)pyridin-3-yl)methyl)-3-isopropylurea 350862 6-chloro-2-[4-(4-fluorophenyl)piperazin-1-ylmethyl]imidazo[1,2-b]pyridazine 350866 (R)-N-(1-(4-(3-((2-fluorobenzylamino)methyl)pyridin-2-yl)piperazin-1-yl)-3-(2,4-dichlorophenyl)-1-oxopropan-2-yl)-3-aminopropanamide 350867 2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]-6-methyl-8-phenylimidazo[1,2-a]pyridine 350868 2-[4-(3'-cyano-biphenyl-4-yl)-1-cyclopentyl-piperidin-4-ylamino]-N-(4-fluoro-3-trifluoromethyl-phenyl)-acetamide 350874 N-methyl-3-((2-(pyridin-2-ylamino)thiazol-5-ylmethyl)amino)benzamide 350877 ethyl 7-benzyl-3-((benzyl(methyl)amino)methyl)-2-(4-isobutyramidophenyl)-4-oxo-4,7-dihydrothieno[2,3-b]pyridine-5-carboxylate 350883 N-((3-(N-(3-nitrobenzyl)-2,2,2-trichloroacetamido)cyclohexyl)methyl)-4-fluoro-N-(3-(2-(pyrrolidin-1-yl)ethoxy)phenyl)benzamide 350888 3-[1-acetyl-4-(3'-cyano-biphenyl-4-yl)-piperidin-4-yl]-N-(3,4-difluoro-phenyl)-propionamide 350889 3-[4-(3'-cyano-biphenyl-4-yl)-1-methanesulfonyl-piperidin-4-yl]-N-(3,4-difluoro-phenyl)-propionamide 350892 6-chloro-2-[4-(3,4-dichlorophenyl)piperazin-1-ylmethyl]imidazo[1,2-b]pyridazine 350893 2-{[4-(3'-cyano-biphenyl-4-yl)-1-cyclopentyl-piperidin-4-yl]-methyl-amino}-N-(3,5-difluoro-phenyl)-acetamide 350895 3-amino-N-((R)-3-(2,4-dichlorophenyl)-1-(4-(3-((1-methoxypropan-2-ylamino)methyl)pyridin-2-yl)piperazin-1-yl)-1-oxopropan-2-yl)propanamide 350896 (R)-N-(1-(4-(3-((2-fluorophenethylamino)methyl)pyridin-2-yl)piperazin-1-yl)-3-(2,4-dichlorophenyl)-1-oxopropan-2-yl)-3-aminopropanamide 350897 (R)-N-(1-(4-(3-((2-methoxyphenethylamino)methyl)pyridin-2-yl)piperazin-1-yl)-3-(2,4-dichlorophenyl)-1-oxopropan-2-yl)-3-aminopropanamide 350898 3-amino-N-((R)-3-(2,4-dichlorophenyl)-1-(4-(2-((1-methoxypropan-2-ylamino)methyl)phenyl)piperazin-1-yl)-1-oxopropan-2-yl)propanamide 350899 N-(3-chloro-4-fluoro-phenyl)-2-[4-(3'-cyano-biphenyl-4-yl)-1-cyclopentyl-piperidin-4-ylamino]-acetamide 350907 N-cyclopropyl-4-fluoro-3-(2-(2-(pyridin-2-ylamino)thiazol-5-yl)ethyl)benzamide 350919 6-{5-[(2S)-2-[(2-hydroxy-1,3-benzoxazol-6-yl)amino]-3-(1H-indol-3-yl)propoxy]pyridin-3-yl}-1,3-benzoxazol-2-ol 350920 4-(3'-cyano-biphenyl-4-yl)-4-[2-(3,4-difluoro-phenylcarbamoyl)-ethyl]-piperidine-1-carboxylic acid ethyl ester 350921 2-(bicyclo[2.2.1]heptan-2-yl)-N-((S)-1-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-2,5-dioxopyrrolidin-3-yl)acetamide 350922 (S)-N-(1-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-2,5-dioxopyrrolidin-3-yl)acetamide 350924 3-amino-N-((R)-3-(2,4-dichlorophenyl)-1-(4-(3-((1-hydroxypropan-2-ylamino)methyl)pyridin-2-yl)piperazin-1-yl)-1-oxopropan-2-yl)propanamide 350925 (R)-3-amino-N-(3-(2,4-dichlorophenyl)-1-(4-(3-((1-hydroxy-2-methylpropan-2-ylamino)methyl)pyridin-2-yl)piperazin-1-yl)-1-oxopropan-2-yl)propanamide 350926 (R)-3-amino-N-(3-(2,4-dichlorophenyl)-1-oxo-1-(4-(3-((2-(thiophen-2-yl)ethylamino)methyl)pyridin-2-yl)piperazin-1-yl)propan-2-yl)propanamide 350927 N-((R)-3-(2,4-dichlorophenyl)-1-(4-(3-((1-methoxypropan-2-ylamino)methyl)pyridin-2-yl)piperazin-1-yl)-1-oxopropan-2-yl)acetamide 350928 (2R)-1-[(adamantan-1-yl)carbonyl]-N-{4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl}pyrrolidine-2-carboxamide 350929 2-[4-(3'-cyano-biphenyl-4-yl)-1-cyclopentyl-piperidin-4-ylamino]-N-(3,5-difluoro-phenyl)-acetamide 350931 5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)-3-(2-methyl-1-(1H-pyrrol-2-yl)propan-2-yl)indolin-2-one 350937 (R)-N-ethyl-N-(1-(3-(3-methoxyphenyl)-3-(4-(methylsulfonyl)phenyl)propyl)piperidin-4-yl)-2-(4-(methylsulfonyl)phenyl)acetamide 350940 N-cyclopentyl-4-fluoro-3-((2-(pyridin-2-ylamino)thiazol-5-ylmethyl)amino)benzamide 350953 6-{5-[(2S)-2-[(2-hydroxy-1,3-benzothiazol-6-yl)amino]-3-(1H-indol-3-yl)propoxy]pyridin-3-yl}-1,3-benzothiazol-2-ol 350955 4-(3'-cyano-biphenyl-4-yl)-4-[2-(3,4-difluoro-phenylcarbamoyl)-ethyl]-piperidine-1-carboxylic acid diethylamide 350956 (S)-N-(1-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-2,5-dioxopyrrolidin-3-yl)cyclopentanecarboxamide 350958 3-amino-N-((R)-3-(2,4-dichlorophenyl)-1-(4-(3-((1-methoxybutan-2-ylamino)methyl)pyridin-2-yl)piperazin-1-yl)-1-oxopropan-2-yl)propanamide 350959 (R)-3-amino-N-(3-(2,4-dichlorophenyl)-1-(4-(3-((1,3-dihydroxypropan-2-ylamino)methyl)pyridin-2-yl)piperazin-1-yl)-1-oxopropan-2-yl)propanamide 350960 (S)-1-(cyclohexanecarbonyl)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-5-oxopyrrolidine-2-carboxamide 350961 (R)-N-(1-(4-(2-((2-methoxyphenethylamino)methyl)phenyl)piperazin-1-yl)-3-(2,4-dichlorophenyl)-1-oxopropan-2-yl)-3-aminopropanamide 350962 (S)-N-(4-amino-1-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butylamino)-1,4-dioxobutan-2-yl)cyclohexanecarboxamide 350963 (2S)-2-(2-(bicyclo[2.2.1]heptan-2-yl)acetamido)-N1-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)succinamide 350966 5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)-3-(2-methyl-1-(pyrrolidin-2-yl)propan-2-yl)indolin-2-one 350971 ethyl 7-(2-nitrobenzyl)-3-((benzyl(methyl)amino)methyl)-2-(4-methoxyphenyl)-4-oxo-4,7-dihydrothieno[2,3-b]pyridine-5-carboxylate 350976 N-benzyl-4-fluoro-3-((2-(pyridin-2-ylamino)thiazol-5-ylmethyl)amino)benzamide 350977 ethyl 2-(4-benzamidophenyl)-7-benzyl-3-((benzyl(methyl)amino)methyl)-4-oxo-4,7-dihydrothieno[2,3-b]pyridine-5-carboxylate 350978 ethyl 3-(N-benzyl-N-methylaminomethyl)-4,7-dihydro-7-(2-fluorobenzyl)-2-(4-(3-methyluriedo)phenyl)-4-oxo-thieno[2,3-b]pyridine-5-carboxylate 350979 ethyl 7-benzyl-3-((benzyl(methyl)amino)methyl)-4-oxo-2-(4-(3-phenylureido)phenyl)-4,7-dihydrothieno[2,3-b]pyridine-5-carboxylate 350980 ethyl 3-(N-benzyl-N-methylaminomethyl)-4,7-dihydro-2-[4-(1,3-dimethyluriedo)phenyl]-7-(2-fluorobenzyl)-4-oxo-thieno[2,3-b]pyridine-5-carboxylate 350998 3-[4-(3'-cyano-biphenyl-4-yl)-1-diethylsulfamoyl-piperidin-4-yl]-N-(3,4-difluoro-phenyl)-propionamide 351002 3-amino-N-((R)-3-(2,4-dichlorophenyl)-1-(4-(3-((1-hydroxybutan-2-ylamino)methyl)pyridin-2-yl)piperazin-1-yl)-1-oxopropan-2-yl)propanamide 351003 (R)-3-amino-N-(3-(2,4-dichlorophenyl)-1-(4-(3-((2-hydroxyethylamino)methyl)pyridin-2-yl)piperazin-1-yl)-1-oxopropan-2-yl)propanamide 351004 (2S)-1-(2-(bicyclo[2.2.1]heptan-2-yl)acetyl)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-5-oxopyrrolidine-2-carboxamide 351005 (S)-1-(cyclohexanecarbonyl)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)pyrrolidine-2-carboxamide 351006 5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)-3-(1-(2,4-dichlorophenyl)-2-methylpropan-2-yl)indolin-2-one 351008 2-(bicyclo[2.2.1]heptan-2-yl)-N-((R)-1-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2,5-dioxopyrrolidin-3-yl)acetamide 351011 5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)-3-(1-cyclopropyl-2-methylpropan-2-yl)indolin-2-one 351012 5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)-3-(2-methyl-1-(1-methyl-1H-pyrrol-2-yl)propan-2-yl)indolin-2-one 351013 ethyl 4,7-dihydro-7-(2-methoxybenzyl)-2-(4-methoxyphenyl)-3-methyl-4-oxothieno[2,3-b]pyridine-5-carboxylate 351014 (R)-N-(1-(3-(3,5-difluorophenyl)-3-(4-(methylsulfonyl)phenyl)propyl)piperidin-4-yl)-N-ethyl-2-(4-(methylsulfonyl)phenyl)acetamide 351015 (R)-N-ethyl-2-(4-(methylsulfonyl)phenyl)-N-(1-(3-(4-(methylsulfonyl)phenyl)-3-(3-(trifluoromethyl)phenyl)propyl)piperidin-4-yl)acetamide 351016 (R)-N-ethyl-2-(4-(methylsulfonyl)phenyl)-N-(1-(3-(4-(methylsulfonyl)phenyl)-3-(3,4,5-trifluorophenyl)propyl)piperidin-4-yl)acetamide 351017 (R)-N-(1-(3-(2,3-difluorophenyl)-3-(4-(methylsulfonyl)phenyl)propyl)piperidin-4-yl)-N-ethyl-2-(4-(methylsulfonyl)phenyl)acetamide 351018 (R)-N-(1-(3-(2,6-difluorophenyl)-3-(4-(methylsulfonyl)phenyl)propyl)piperidin-4-yl)-N-ethyl-2-(4-(methylsulfonyl)phenyl)acetamide 351020 ethyl 7-(2-methoxybenzyl)-3-((benzyl(ethyl)amino)methyl)-2-(4-methoxyphenyl)-4-oxo-4,7-dihydrothieno[2,3-b]pyridine-5-carboxylate 351025 ethyl 3-(N-benzyl-N-methylaminomethyl)-4,7-dihydro-7-(2-methoxybenzyl)-2-(3-methoxyphenyl)-4-oxothieno[2,3-b]pyridine-5-carboxylate 351031 rac-N-((3-(N-benzylpivalamido)cyclohexyl)methyl)-4-fluoro-N-(3-(2-(pyrrolidin-1-yl)ethoxy)phenyl)benzamide 351033 N-(((1S,3R)-3-(N-benzylpivalamido)cyclohexyl)methyl)-4-fluoro-N-(3-(2-(pyrrolidin-1-yl)ethoxy)phenyl)benzamide 351037 ethyl 3-(N-benzyl-N-methylaminomethyl)-7-(2,6-difluorobenzyl)-4,7-dihydro-2-[4-(3-methyluriedo)phenyl]-4-oxothieno[2,3-b]pyridine-5-carboxylate 351038 3-(N-benzyl-N-methylaminomethyl)-7-(2,6-difluorobenzyl)-4,7-dihydro-N-isopropyl-4-oxo-2-(4-propionylamidophenyl)-thieno[2,3-b]pyridine-5-carboxamide 351039 (S)-N-(1-(3-(3,5-difluorophenyl)-3-(4-(methylsulfonyl)phenyl)propyl)piperidin-4-yl)-N-ethyl-2-(4-(methylsulfonyl)phenyl)acetamide 351040 5-{5-[(2S)-2-[(2,3-dioxo-2,3-dihydro-1H-indol-5-yl)amino]-3-(1H-indol-3-yl)propoxy]pyridin-3-yl}-2,3-dihydro-1H-indole-2,3-dione 351041 5-{5-[(2S)-2-[(2-hydroxy-3-nitroso-1H-indol-5-yl)amino]-3-(1H-indol-3-yl)propoxy]pyridin-3-yl}-3-nitroso-1H-indol-2-ol 351042 {6-[(S)-2-[5-(3-Cyanomethyl-2-oxo-2,3-dihydro-1H-benzoimidazol-5-yl)-pyridin-3-yloxy]-1-(1H-indol-3-ylmethyl)-ethylamino]-2-oxo-2,3-dihydro-benzoimidazol-1-yl}-acetonitrile 351043 3-(N-benzyl-N-methylaminomethyl)-7-(2,6-difluorobenzyl)-4,7-dihydro-2-(4-isobutyrylamidophenyl)-4-oxo-5-propionyl-thieno[2,3-b]pyridine 351044 N-(4-(7-(2,6-difluorobenzyl)-3-((benzyl(methyl)amino)methyl)-5-isobutyryl-4-oxo-4,7-dihydrothieno[2,3-b]pyridin-2-yl)phenyl)isobutyramide 351046 (S)-3-(2-chlorophenyl)-1-(4-fluorophenyl)-1-(2-(1-methoxypropan-2-ylamino)pyrimidin-4-yl)urea 351047 (S)-1-(4-fluorophenyl)-1-(2-(1-methoxypropan-2-ylamino)pyrimidin-4-yl)-3-o-tolylurea 351048 4-(1-benzyl-piperidin-4-yl)-4-(3'-cyano-biphenyl-4-yl)-N-(3,4-difluoro-phenyl)-butyramide 351051 (R)-1-((2-(4-(2-(3-aminopropanamido)-3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)pyridin-3-yl)methyl)-3-(thiophen-2-ylmethyl)urea 351054 (2S)-1-(2-(bicyclo[2.2.1]heptan-2-yl)acetyl)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)pyrrolidine-2-carboxamide 351055 3-(2,6-dichlorophenyl)-1-(6-(4-fluorophenylamino)pyrimidin-4-yl)-1-methylurea 351056 3-[4-(3'-cyano-biphenyl-4-yl)-1-cyclopentyl-piperidin-4-yl]-N-(3,5-difluoro-phenyl)-propionamide 351059 5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)-3-(2-methyl-1-phenylpropan-2-yl)indolin-2-one 351060 5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)-3-(2-methyl-1-(1H-pyrrol-3-yl)propan-2-yl)indolin-2-one 351061 3-(1-(1H-indol-3-yl)-2-methylpropan-2-yl)-5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)indolin-2-one 351062 ethyl 7-(2-methoxybenzyl)-3-((benzylamino)methyl)-2-(4-methoxyphenyl)-4-oxo-4,7-dihydrothieno[2,3-b]pyridine-5-carboxylate 351063 ethyl 7-(2-fluorobenzyl)-3-((benzyl(methyl)amino)methyl)-2-(4-methoxyphenyl)-4-oxo-4,7-dihydrothieno[2,3-b]pyridine-5-carboxylate 351070 (S)-3-(2-fluorophenyl)-1-(4-fluorophenyl)-1-(2-(1-methoxypropan-2-ylamino)pyrimidin-4-yl)urea 351072 (R)-3-amino-N-(3-(2,4-dichlorophenyl)-1-oxo-1-(4-(3-((2-(thiophen-2-yl)acetamido)methyl)pyridin-2-yl)piperazin-1-yl)propan-2-yl)propanamide 351073 3-(2-(2-(2-chloro-6-fluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351076 (R)-3-amino-N-(3-(2,4-dichlorophenyl)-1-oxo-1-(4-(3-((2,2,2-trifluoroethylamino)methyl)pyridin-2-yl)piperazin-1-yl)propan-2-yl)propanamide 351078 (R)-N-(1-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2,5-dioxopyrrolidin-3-yl)cyclohexanecarboxamide 351080 (S)-1-(Adamantane-1-carbonyl)-pyrrolidine-2-carboxylic acid {4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-amide 351082 2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]-6-methyl-8-(pyrazol-1-yl)imidazo[1,2-a]pyridine 351085 5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)-3-(2-methyl-1-(pyridin-3-yl)propan-2-yl)indolin-2-one 351087 ethyl 3-(N-acetyl-N-benzylaminomethyl)-4,7-dihydro-7-(2-methoxybenzyl)-2-(4-methoxyphenyl)-4-oxothieno[2,3-b]pyridine-5-carboxylate 351088 (R)-N-(1-(3-(2,5-difluorophenyl)-3-(4-(methylsulfonyl)phenyl)propyl)piperidin-4-yl)-N-ethyl-2-(4-(methylsulfonyl)phenyl)acetamide 351089 ethyl 7-(3-fluorobenzyl)-3-((benzyl(methyl)amino)methyl)-2-(4-methoxyphenyl)-4-oxo-4,7-dihydrothieno[2,3-b]pyridine-5-carboxylate 351090 ethyl 2-(4-aminophenyl)-3-(N-benzyl-N-methylaminomethyl)-4,7-dihydro-7-(2-fluorobenzyl)-4-oxothieno[2,3-b]pyridine-5-carboxylate 351095 6-{5-[(2S)-3-(1H-indol-3-yl)-2-({2-oxo-1H,2H,3H-pyrrolo[2,3-b]pyridin-6-yl}amino)propoxy]pyridin-3-yl}-1H,2H,3H-pyrrolo[2,3-b]pyridin-2-one 351096 (S)-3-(2-chlorophenyl)-1-(4-fluorophenyl)-1-(2-(1-phenylethylamino)pyrimidin-4-yl)urea 351097 3-(2-(2-(2-fluoro-4-(trifluoromethyl)benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351098 3-(2-(2-(2-fluoro-6-(trifluoromethyl)benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351100 4'-{[(6-chloro-5-fluoro-1H-benzoimidazol-2-ylmethyl)-amino]-piperidin-4-yl-methyl}-biphenyl-3-carbonitrile 351101 (S)-N-(1-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2,5-dioxopyrrolidin-3-yl)cyclohexanecarboxamide 351102 (S)-N-(1-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2,5-dioxopyrrolidin-3-yl)benzamide 351103 (2R)-1-(2-(bicyclo[2.2.1]heptan-2-yl)acetyl)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)pyrrolidine-2-carboxamide 351104 2-[4-(3'-cyano-biphenyl-4-yl)-1-cyclopentyl-piperidin-4-ylamino]-N-(3,5-dichloro-phenyl)-acetamide 351105 2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]-5-(pyrazol-1-yl)imidazo[1,2-a]pyridine 351106 (2S)-1-(5-(isoquinolin-6-yl)pyridin-3-yloxy)-3-(1-methyl-1H-indol-3-yl)propan-2-amine 351107 5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)-3-(2-methyl-1-(pyridin-2-yl)propan-2-yl)indolin-2-one 351110 ethyl 7-benzyl-3-((benzyl(methyl)amino)methyl)-2-(4-methoxyphenyl)-4-oxo-4,7-dihydrothieno[2,3-b]pyridine-5-carboxylate 351121 5-{5-[(2S)-2-[(2-hydroxy-1H-1,3-benzodiazol-5-yl)amino]-3-(1H-indol-3-yl)propoxy]pyridin-3-yl}-1H-1,3-benzodiazol-2-ol 351123 3-(2-chlorophenyl)-1-(4-fluorophenyl)-1-(2-(tetrahydro-2H-pyran-4-ylamino)pyrimidin-4-yl)urea 351126 4'-[[(6-chloro-5-fluoro-1H-benzoimidazol-2-ylmethyl)-amino]-(1-cyclopentyl-piperidin-4-yl)-methyl]-biphenyl-3-carbonitrile 351128 2-(bicyclo[2.2.1]heptan-2-yl)-N-((S)-1-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2,5-dioxopyrrolidin-3-yl)acetamide 351129 N-[(3R)-1-{4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl}-2,5-dioxopyrrolidin-3-yl]adamantane-1-carboxamide 351131 3-[4-(3'-cyano-biphenyl-4-yl)-1-cyclopentyl-piperidin-4-yl]-N-(3,5-dichloro-phenyl)-propionamide 351132 6-bromo-2-[4-(3,4-dichlorophenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine 351133 N-(4-chloro-3-trifluoromethyl-phenyl)-2-[4-(3'-cyano-biphenyl-4-yl)-1-cyclopentyl-piperidin-4-ylamino]-acetamide 351135 (2S)-1-(1H-indazol-3-yl)-3-(5-(isoquinolin-6-yl)pyridin-3-yloxy)propan-2-amine 351136 (2S)-1-(benzo[b]thiophen-3-yl)-3-(5-(isoquinolin-6-yl)pyridin-3-yloxy)propan-2-amine 351139 (S)-N-ethyl-2-(4-(methylsulfonyl)phenyl)-N-(1-(3-(4-(methylsulfonyl)phenyl)-3-phenylpropyl)piperidin-4-yl)acetamide 351140 (S)-1-((S)-2-((S)-2-(2-((S)-2-((S)-2-((S)-2-((S)-3-(1H-imidazol-5-yl)-2-((S)-2-oxopyrrolidine-5-carboxamido)propanamido)-3-(1H-indol-2-yl)propanamido)-3-hydroxypropanamido)-3-(4-hydroxyphenyl)propanamido)acetamido)-4-methylpentanamido)-5-(diaminomethylene 351141 N-(5-((5-tert-butyloxazol-2-yl)methylthio)thiazol-2-yl)-3,4-dimethoxybenzamide 351143 4-fluoro-N-methyl-3-((2-(pyridin-2-ylamino)thiazol-5-ylmethyl)amino)benzamide 351150 N-(4-(7-(2,6-difluorobenzyl)-5-benzoyl-3-((benzyl(methyl)amino)methyl)-4-oxo-4,7-dihydrothieno[2,3-b]pyridin-2-yl)phenyl)isobutyramide 351153 {5-[(S)-2-[5-(1-cyanomethyl-2-oxo-2,3-dihydro-1H-benzoimidazol-5-yl)-pyridin-3-yloxy]-1-(1H-indol-3-ylmethyl)-ethylamino]-2-oxo-2,3-dihydro-benzoimidazol-1-yl}-acetonitrile 351154 (2,2-dioxo-2,3-dihydro-1H-2lambda*6*-benzo[1,2,5]thiadiazol-5-yl)-[(S)-2-[5-(2,2-dioxo-2,3-dihydro-1H-2lambda*6*-benzo[1,2,5]thiadiazol-5-yl)-pyridin-3-yloxy]-1-(1H-indol-3-ylmethyl)-ethyl]-amine 351155 5-{5-[(2S)-2-[(3,3-dimethyl-2-oxo-2,3-dihydro-1H-indol-5-yl)amino]-3-(1H-indol-3-yl)propoxy]pyridin-3-yl}-3,3-dimethyl-2,3-dihydro-1H-indol-2-one 351156 3-(N-benzyl-N-methylaminomethyl)-7-(2,6-difluorobenzyl)-4,7-dihydro-5-(1-hydroxy-2-methylpropyl)-2-(4-isobutyrylamidophenyl)-4-oxothieno[2,3-b]pyridine 351157 3-(N-benzyl-N-methylaminomethyl)-7-(2,6-difluorobenzyl)-4,7-dihydro-5-isobutyryl-2-[4-(3-methyluriedo)phenyl]-4-oxothieno[2,3-b]pyridine 351160 4'-[[(6-chloro-5-fluoro-1H-benzoimidazol-2-ylmethyl)-amino]-(1-cyclopropylmethyl-piperidin-4-yl)-methyl]-biphenyl-3-carbonitrile 351161 Adamantane-1-carboxylic acid ((S)-1-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-2,5-dioxo-pyrrolidin-3-yl)-amide 351164 2-[4-(3,4-dichlorophenyl)piperazin-1-ylmethyl]-6-(4-methylpiperazin-1-yl)imidazo[1,2-b]pyridazine 351165 2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]-6-methylimidazo[1,2-a]pyridine-8-carbonitrile 351166 N-(4-chloro-3-trifluoromethyl-phenyl)-3-[4-(3'-cyano-biphenyl-4-yl)-1-cyclopentyl-piperidin-4-yl]-propionamide 351169 (2S)-1-(5-(isoquinolin-6-yl)pyridin-3-yloxy)-3-(naphthalen-2-yl)propan-2-amine 351170 (2S)-1-(5-(isoquinolin-6-yl)pyridin-3-yloxy)-3-(quinolin-3-yl)propan-2-amine 351172 (E)-3-(2,3-dichlorophenylimino)indolin-2-one 351180 5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)-3-(1-(4-ethyl-3,5-dimethyl-1H-pyrrol-2-yl)-2-methylpropan-2-yl)indolin-2-one 351181 (R)-N-ethyl-N-(1-(3-(3-fluorophenyl)-3-(4-(methylsulfonyl)phenyl)propyl)piperidin-4-yl)-2-(4-(methylsulfonyl)phenyl)acetamide 351182 (S)-N-ethyl-N-(1-(3-(4-fluorophenyl)-3-(4-(methylsulfonyl)phenyl)propyl)piperidin-4-yl)-2-(4-(methylsulfonyl)phenyl)acetamide 351183 (R)-N-(1-(3-(3-chlorophenyl)-3-(4-(methylsulfonyl)phenyl)propyl)piperidin-4-yl)-N-ethyl-2-(4-(methylsulfonyl)phenyl)acetamide 351184 (R)-N-(1-(3-(3,4-difluorophenyl)-3-(4-(methylsulfonyl)phenyl)propyl)piperidin-4-yl)-N-ethyl-2-(4-(methylsulfonyl)phenyl)acetamide 351185 (S)-N-ethyl-N-(1-(3-(4-methoxyphenyl)-3-(4-(methylsulfonyl)phenyl)propyl)piperidin-4-yl)-2-(4-(methylsulfonyl)phenyl)acetamide 351189 N-cyclopropyl-4-fluoro-3-((2-(pyridin-2-ylamino)thiazol-5-ylmethyl)amino)benzamide 351199 2-[4-(2-aminoacetamido)phenyl]-3-(N-benzyl-N-methylaminomethyl)-7-(2,6-difluorobenzyl)-4,7-dihydro-5-isobutyryl-4-oxothieno[2,3-b]pyridine 351201 5-{5-[(2S)-3-(1H-indol-3-yl)-2-[(3-methyl-2-oxo-2,3-dihydro-1H-indol-5-yl)amino]propoxy]pyridin-3-yl}-3-methyl-2,3-dihydro-1H-indol-2-one 351202 3-ethyl-5-{5-[(2S)-2-[(3-ethyl-2-oxo-2,3-dihydro-1H-indol-5-yl)amino]-3-(1H-indol-3-yl)propoxy]pyridin-3-yl}-2,3-dihydro-1H-indol-2-one 351203 3-benzyl-5-{5-[(2S)-2-[(3-benzyl-2-oxo-2,3-dihydro-1H-indol-5-yl)amino]-3-(1H-indol-3-yl)propoxy]pyridin-3-yl}-2,3-dihydro-1H-indol-2-one 351204 5-{5-[(2S)-3-(1H-indol-3-yl)-2-{[2-oxo-3-(propan-2-ylidene)-2,3-dihydro-1H-indol-5-yl]amino}propoxy]pyridin-3-yl}-3-(propan-2-ylidene)-2,3-dihydro-1H-indol-2-one 351205 5-{5-[(2S)-2-[(3,3-difluoro-2-oxo-2,3-dihydro-1H-indol-5-yl)amino]-3-(1H-indol-3-yl)propoxy]pyridin-3-yl}-3,3-difluoro-2,3-dihydro-1H-indol-2-one 351206 3-(N-benzyl-N-methylaminomethyl)-7-(2,6-difluorobenzyl)-4,7-dihydro-2-(4-(2-hydroxy-2-methylpropionylamido)phenyl)-5-isobutyryl-4-oxothieno[2,3-b]pyridine 351207 3-(N-benzyl-N-methylaminomethyl)-7-(2,6-difluorobenzyl)-4,7-dihydro-2-[4-(1-hydroxy-1-cyclopropanecarboxamido)-phenyl]-5-isobutyryl-4-oxothieno[2,3-b]pyridine 351208 ethyl 7-(2-cyanobenzyl)-3-((benzyl(methyl)amino)methyl)-2-(4-methoxyphenyl)-4-oxo-4,7-dihydrothieno[2,3-b]pyridine-5-carboxylate 351209 3-(N-benzyl-N-methylaminomethyl)-7-(2,6-difluorobenzyl)-4,7-dihydro-2-[4-(2-hydroxyacetamido)phenyl]-5-isobutyryl-4-oxothieno[2,3-b]pyridine 351213 (R)-1-((2-(4-(2-(3-aminopropanamido)-3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)pyridin-3-yl)methyl)-3-phenylurea 351216 6-chloro-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo[1,2-b]pyridazine 351217 6-bromo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine 351218 6-iodo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine 351219 2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]-6-methyl-8-morpholinoimidazo[1,2-a]pyridine 351220 N-(4-chloro-3-trifluoromethyl-phenyl)-3-[4-(3'-cyano-biphenyl-4-yl)-1-cyclopentyl-piperidin-4-yl]-propionamide 351223 (2S)-1-(5-(isoquinolin-6-yl)pyridin-3-yloxy)-3-phenylpropan-2-amine 351224 (S)-3-(2-chlorophenyl)-1-(2-(3-hydroxy-3-methylbutan-2-ylamino)pyrimidin-4-yl)-1-phenylurea 351225 (E)-3-(4-chlorophenylimino)indolin-2-one 351227 3-{[3-(trifluoromethyl)phenyl]azamethylene}benzo[d]azolidin-2-one 351234 5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)-3-(1-(4,5-dimethylfuran-2-yl)-2-methylpropan-2-yl)indolin-2-one 351239 ethyl 2-(4-acetamidophenyl)-7-benzyl-3-((benzyl(methyl)amino)methyl)-4-oxo-4,7-dihydrothieno[2,3-b]pyridine-5-carboxylate 351240 ethyl 3-(N-benzyl-N-methylaminomethyl)-4,7-dihydro-7-(2-fluorobenzyl)-4-oxo-2-(4-propionylamidophenyl)thieno[2,3-b]pyridine-5-carboxylate 351251 Tyr-Pro-Phe-Phg-NH2 351253 (S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-((3-(dimethylamino)propyl)(methyl)amino)-2-phenylacetamide 351254 (S)-2-[acetyl-(2-dimethylamino-ethyl)-amino]-N-(3,5-bis-trifluoromethyl-benzyl)-2-phenyl-acetamide 351257 3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-chloro-1H-pyrrol-1-yl)benzoic acid 351258 3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-ethyl-1H-pyrrol-1-yl)benzoic acid 351263 N-(1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl)-2,2-diphenylacetamide 351269 N-(1-(4-fluorobenzyl)piperidin-4-yl)-4-(1,3-diethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)benzenesulfonamide 351273 diethyl 2,4-diethyl-6-phenylpyridine-3,5-dicarboxylate 351274 3-ethyl 5-propyl 2,4-diethyl-6-phenylpyridine-3,5-dicarboxylate 351276 Tyr-Pro-Hfe-Pro-NH2 351277 1-(4-(3-(2-(pyrimidin-2-ylamino)thiazol-5-ylthio)benzoyl)piperazin-1-yl)ethanone 351278 1-(4-(3-(2-(pyrazin-2-ylamino)thiazol-5-ylthio)benzoyl)piperazin-1-yl)ethanone 351279 (S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(3-(dimethylamino)propylideneamino)-2-phenylacetamide 351280 (S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-(dimethylamino)ethoxy)-2-phenylacetamide 351282 3-(2-(2-(benzyloxy)-5-bromophenyl)-5-ethyl-1H-pyrrol-1-yl)benzoic acid 351283 3-(2-(2-(4-fluorobenzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351286 4-benzamido-2-(4-methoxyphenyl)-1,2-dihydro-1,2,4-triazolo[4,3-a]quinoxalin-1-one 351287 N-(6-nitro-1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl)-2,2-diphenylacetamide 351292 2-(2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-1H-indol-4-yl)-N-ethyl-N-methylethanamine 351293 2-(2-(2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-1H-indol-4-yl)ethoxy)-N,N-dimethylethanamine 351296 4-(1,3-diethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-N-(2-(pyridin-2-yl)ethyl)benzenesulfonamide 351297 N-(1-benzylpiperidin-4-yl)-4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)benzenesulfonamide 351302 3-ethyl 5-propyl 2-ethyl-6-phenyl-4-propylpyridine-3,5-dicarboxylate 351303 dipropyl 2-(3-chlorophenyl)-4,6-diethylpyridine-3,5-dicarboxylate 351305 N-(2-((1-(4-chlorobenzyl)piperidin-4-yl)methylamino)-2-oxoethyl)-2-amino-5-(trifluoromethyl)benzamide 351306 1-(4-(3-(2-(thiazol-2-ylamino)thiazol-5-ylthio)benzoyl)piperazin-1-yl)ethanone 351307 1-(4-(2-hydroxy-5-(2-(pyridin-2-ylamino)thiazol-5-ylthio)benzoyl)piperazin-1-yl)ethanone 351310 3-(2-(2-(benzyloxy)-5-(trifluoromethyl)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351311 3-(2-(2-(benzyloxy)-5-(methylsulfonyl)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351316 4-benzamido-1,2-dihydro-2-(4-nitrophenyl)-1,2,4-triazolo[4,3-a]quinoxalin-1-one 351317 N-(6-nitro-1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl)benzamide 351323 3-(2-(2-(2,3-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351324 2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-4-(2-(pyrrolidin-1-yl)ethyl)-1H-indole 351328 4-((4-(4-(1-methyl-2,4-dioxo-3-propyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenylsulfonyl)piperazin-1-yl)methyl)benzonitrile 351329 4-(1-methyl-2,4-dioxo-3-propyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-N-(2-(pyridin-2-yl)ethyl)benzenesulfonamide 351337 ethyl 5-(ethylthiocarbonyl)-4,6-dimethyl-2-phenylnicotinate 351338 1-(3,4-dichlorobenzyl)-5-hydroxy-1H-indole-2-carboxylic acid 351339 1-(4-(5-(2-(6-bromopyridin-2-ylamino)thiazol-5-ylthio)-2-hydroxybenzoyl)piperazin-1-yl)ethanone 351340 1-(4-(5-(2-(4,6-dimethylpyridin-2-ylamino)thiazol-5-ylthio)-2-hydroxybenzoyl)piperazin-1-yl)ethanone 351341 (S)-3-(2-chlorophenyl)-1-(2-(3-hydroxy-3-methylbutan-2-ylamino)pyrimidin-4-yl)-1-(4-methoxyphenyl)urea 351342 (S)-1-(2-(3-hydroxy-3-methylbutan-2-ylamino)pyrimidin-4-yl)-1-(4-methoxyphenyl)-3-o-tolylurea 351343 3-(2-(2-(benzyloxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351344 3-[2-(4-Benzyloxy-biphenyl-3-yl)-5-methyl-pyrrol-1-yl]-benzoic acid 351349 N-(2-(4-methoxyphenyl)-6-nitro-1-oxo-1,2-dihydro-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl)benzamide 351350 6-amino-4-benzamido-1,2-dihydro-2-phenyl-1,2,4-triazolo[4,3-a]quinoxalin-1-one 351354 N-benzoyl-N-(2-(4-methoxyphenyl)-6-nitro-1-oxo-1,2-dihydro-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl)benzamide 351355 3-(2-(2-(2,6-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351356 3-(2-(2-(2,4,6-trifluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351359 6-(4-(4-(3-fluorobenzyl)piperazin-1-ylsulfonyl)phenyl)-1,3-dimethyl-1H-pyrrolo[3,2-d]pyrimidine-2,4(3H,5H)-dione 351360 6-(4-(4-(4-fluorobenzyl)piperazin-1-ylsulfonyl)phenyl)-1,3-dimethyl-1H-pyrrolo[3,2-d]pyrimidine-2,4(3H,5H)-dione 351361 6-(4-(4-(3-fluorobenzyl)piperazin-1-ylsulfonyl)phenyl)-1,3-diethyl-1H-pyrrolo[3,2-d]pyrimidine-2,4(3H,5H)-dione 351372 Tyr-Pro-Phe-D-Phg-NH2 351374 (2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-1H-indol-4-yl)-N,N-dimethylmethanamine 351375 3-(2-(2-(benzyloxy)-5-(thiophen-3-yl)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351379 N-(6-amino-2-(4-methoxyphenyl)-1-oxo-1,2-dihydro-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl)acetamide 351383 3-(2-(2-(3-(difluoromethoxy)benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351384 3-(2-(2-(2-chlorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351385 3-(2-(2-(3-chlorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351388 6-(4-(4-(2,4-difluorobenzyl)piperazin-1-ylsulfonyl)phenyl)-1,3-dimethyl-1H-pyrrolo[3,2-d]pyrimidine-2,4(3H,5H)-dione 351389 6-(4-{[4-(4-bromobenzyl)piperazin-1-yl]sulfonyl}phenyl)-1,3-dimethyl-1H-pyrrolo[3,2-d]pyrimidine-2,4(3H,5H)-dione 351408 4-acetamido-2-(4-methoxyphenyl)-1,2-dihydro-1,2,4-triazolo[4,3-a]quinoxalin-1-one 351409 N-(6-nitro-1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl)acetamide 351415 3-(2-(2-(4-(trifluoromethoxy)benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351416 3-(2-(2-(2-fluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351417 3-(2-(2-(4-chlorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351418 3-(2-(2-(2,4-dichlorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351420 4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-N-(2-(pyridin-2-yl)ethyl)benzenesulfonamide 351421 6-(4-(4-((5-chlorothiophen-2-yl)methyl)piperazin-1-ylsulfonyl)phenyl)-1,3-dimethyl-1H-pyrrolo[3,2-d]pyrimidine-2,4(3H,5H)-dione 351422 1,3-dimethyl-6-(4-(4-(pyridin-4-ylmethyl)piperazin-1-ylsulfonyl)phenyl)-1H-pyrrolo[3,2-d]pyrimidine-2,4(3H,5H)-dione 351430 3,5-bis-ethoxycarbonyl-4-ethyl-1,2-dimethyl-6-phenyl-pyridinium 351431 3-ethoxycarbonyl-4,6-diethyl-5-ethylsulfanylcarbonyl-1-methyl-2-phenyl-pyridinium 351432 N-(5-(5-(1-acetylpiperazine-4-carbonyl)-4-methoxy-2-methylphenylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 351434 1-(4-(5-(2-(4,6-dimethylpyridin-2-ylamino)thiazol-5-ylthio)-2-methoxy-4-methylbenzoyl)piperazin-1-yl)ethanone 351442 N-(6-amino-1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl)acetamide 351447 3-(2-(2-(4-fluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351448 3-(2-(2-(3,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351451 4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-N-(2-(pyridin-2-yloxy)ethyl)benzenesulfonamide 351452 N-(1-benzylpiperidin-4-yl)-4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)benzenesulfonamide 351465 1-[8-(2-benzyloxy-ethyl)-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl]-3-pyridin-4-yl-urea 351466 N-(5-(5-(1-acetylpiperazine-4-carbonyl)-4-methoxy-2-methylphenylthio)thiazol-2-yl)-4-(methoxymethyl)benzamide 351467 (S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-(dimethylamino)ethylamino)-2-(thiophen-2-yl)acetamide 351468 Tyr-Pro-Hfe-Phe-NH2 351469 Tyr-Pro-Phe-Hfe-NH2 351470 2-[(1-cyclopropylmethyl-piperidin-4-ylidene)-(3'-methanesulfonyl-biphenyl-4-yl)-methyl]-5-fluoro-6-trifluoromethyl-1H-benzoimidazole 351471 N-(5-(5-(1-ethylpiperazine-4-carbonyl)-4-methoxy-2-methylphenylthio)thiazol-2-yl)cyclopropanecarboxamide 351472 N-(5-(5-(1-(2-(dimethylamino)acetyl)piperazine-4-carbonyl)-4-methoxy-2-methylphenylthio)thiazol-2-yl)cyclopropanecarboxamide 351478 H-Dmt-Aba-Gly-NH-Ph 351480 3-{2-[5-Bromo-2-(2-methyl-benzyloxy)-phenyl]-5-methyl-pyrrol-1-yl}-benzoic acid 351481 3-(2-(2-(2,5-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351485 N-(1-benzylpiperidin-4-yl)-4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-N-methylbenzenesulfonamide 351486 6-(4-(4-benzylpiperazin-1-ylsulfonyl)phenyl)-1,3-dimethyl-1H-pyrrolo[3,2-d]pyrimidine-2,4(3H,5H)-dione 351499 5-[[(4-pyridyl)amino]carbonyl]amino-[8-(3-benzyloxypropyl)-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine 351500 (S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-(dimethylamino)ethylamino)-2-(4-fluorophenyl)acetamide 351502 Tyr-Pro-Phg-Pro-NH2 351503 (S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-(dimethylamino)ethylamino)-2-(thiophen-3-yl)acetamide 351504 2-((5-(5-(1-acetylpiperazine-4-carbonyl)-4-methoxy-2-methylphenylthio)thiazol-2-yl)carbamoyl)cyclopropanecarboxylic acid 351505 N-(5-(4-methoxy-2-methyl-5-(morpholine-4-carbonyl)phenylthio)thiazol-2-yl)-5-((methylamino)methyl)-1H-pyrrole-2-carboxamide 351514 H-Dmt-Aba-Gly-NH-CH2-Bid 351517 3-{2-[5-Bromo-2-(4-methyl-benzyloxy)-phenyl]-5-methyl-pyrrol-1-yl}-benzoic acid 351518 3-(2-(2-(3-(trifluoromethyl)benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351519 N-(2-(4-methoxyphenyl)-6-nitro-1-oxo-1,2-dihydro-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl)-2,2-diphenylacetamide 351524 1,3-dimethyl-6-(4-(4-phenylpiperazin-1-ylsulfonyl)phenyl)-1H-pyrrolo[3,2-d]pyrimidine-2,4(3H,5H)-dione 351541 N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-(dimethylamino)ethylamino)-2-(furan-2-yl)acetamide 351542 1-(5-(2-(6-bromopyridin-2-ylamino)thiazol-5-ylthio)-2-hydroxybenzoyl)piperidine-3-carboxylic acid 351555 3-(2-(2-(4-(trifluoromethyl)benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351556 3-(2-(2-(3-methoxybenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351559 N-(6-amino-1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl)-N-benzoyl-benzamide 351571 (S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-(dimethylamino)ethylamino)-2-phenylacetamide 351574 N-(5-(5-(1-acetylpiperazine-4-carbonyl)-4-methoxy-2-methylphenylthio)thiazol-2-yl)-4-isopropoxybenzamide 351583 3-(2-(5-chloro-2-(cyclopentylmethoxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351584 3-(2-(2-(4-methoxybenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351585 3-(2-(5-bromo-2-((5-methylisoxazol-3-yl)methoxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351587 6-amino-1,2-dihydro-2-phenyl-4-diphenylacetamido-1,2,4-triazolo[4,3-a]quinoxalin-1-one 351588 4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-N-(pyridin-2-yl)benzenesulfonamide 351601 N-(5-(5-(1-acetylpiperazine-4-carbonyl)-4-methoxy-2-methylphenylthio)thiazol-2-yl)-4-((ethylamino)methyl)benzamide 351602 N-(5-(5-(1-acetylpiperazine-4-carbonyl)-4-methoxy-2-methylphenylthio)thiazol-2-yl)-1H-pyrrole-2-carboxamide 351610 (S)-2-amino-N-((S)-2-(2-(benzylamino)-2-oxoethyl)-3-oxo-2,3,4,5-tetrahydro-1H-benzo[c]azepin-4-yl)-3-(4-hydroxy-2,6-dimethylphenyl)propanamide 351611 3-(2-(5-bromo-2-(cyclopentylmethoxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351612 3-(2-(5-chloro-2-((tetrahydrofuran-2-yl)methoxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351615 6-amino-1,2-dihydro-2-(methoxyphenyl)-4-diphenylacetamido-1,2,4-triazolo[4,3-a]quinoxalin-1-one 351616 4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-N-(6-methoxypyridin-3-yl)benzenesulfonamide 351617 4-(1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)-N-((5-methoxypyridin-2-yl)methyl)benzenesulfonamide 351631 1-[8-(2-benzyloxy-ethyl)-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl]-3-pyridin-3-yl-urea 351632 1-[2-furan-2-yl-8-(2-hydroxy-ethyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl]-3-pyridin-4-yl-urea 351633 N-(5-(5-(1-acetylpiperazine-4-carbonyl)-4-methoxy-2-methylphenylthio)thiazol-2-yl)cyclopropanecarboxamide 351634 1-(4-(3-(2-(phenylamino)thiazol-5-ylthio)benzoyl)piperazin-1-yl)ethanone 351636 1-(5-(2-(6-bromopyridin-2-ylamino)thiazol-5-ylthio)-2-hydroxybenzoyl)piperidine-4-carboxylic acid 351643 3-(2-(2-(2,4-difluorobenzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351645 3-(2-(5-chloro-2-isobutoxyphenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351646 3-(2-(5-bromo-2-isobutoxyphenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351649 N-benzoyl-N-(1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl)-benzamide 351653 2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-4-(4-methylpiperazin-1-yl)-1H-indole 351657 N-((5-methoxypyridin-2-yl)methyl)-4-(1-methyl-2,4-dioxo-3-propyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)benzenesulfonamide 351658 6-(4-(4-(3-fluorobenzyl)piperazin-1-ylsulfonyl)phenyl)-3-methyl-1-propyl-1H-pyrrolo[3,2-d]pyrimidine-2,4(3H,5H)-dione 351670 1-[2-furan-2-yl-8-(3-hydroxy-propyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl]-3-pyridin-4-yl-urea 351671 1-[2-furan-2-yl-8-(2-hydroxy-ethyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl]-3-pyridin-3-yl-urea 351672 1-(4-(3-(2-(pyridin-2-ylamino)thiazol-5-ylthio)benzoyl)piperazin-1-yl)ethanone 351674 2-(5-(2-(6-bromopyridin-2-ylamino)thiazol-5-ylthio)-2-hydroxy-N-methylbenzamido)acetic acid 351675 1-(5-(2-(6-bromopyridin-2-ylamino)thiazol-5-ylthio)-2-hydroxybenzoyl)-N-(methylsulfonyl)piperidine-3-carboxamide 351682 3-(5-(2-(benzyloxy)-5-chlorophenyl)-3-bromo-2-methyl-1H-pyrrol-1-yl)benzoic acid 351684 3-(2-(5-bromo-2-((3,5-dimethylisoxazol-4-yl)methoxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351685 3-(2-(5-chloro-2-((tetrahydro-2H-pyran-4-yl)methoxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351688 N-benzoyl-N-[2-(4-methoxy-phenyl)-1-oxo-1,2-dihydro-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl]-benzamide 351690 2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-4-(4-methylpiperazin-1-yl)-1H-pyrrolo[3,2-c]pyridine 351696 6-(4-(4-(benzo[d][1,3]dioxol-5-ylmethyl)piperazin-1-ylsulfonyl)phenyl)-3-methyl-1-propyl-1H-pyrrolo[3,2-d]pyrimidine-2,4(3H,5H)-dione 351702 4-(5,6-dichloro-1H-benzo[d]imidazol-2-yl)-N-methyl-N-(2-(piperidin-1-yl)ethyl)benzenamine 351703 Tyr-Pro-Phg-Phe-NH2 351704 4'-[(1-cyclopropylmethyl-piperidin-4-ylidene)-(5,6-dichloro-1H-benzoimidazol-2-yl)-methyl]-biphenyl-3-carbonitrile 351705 4'-[(1-cyclopropylmethyl-piperidin-4-ylidene)-(5,6-difluoro-1H-benzoimidazol-2-yl)-methyl]-biphenyl-3-carbonitrile 351710 3-(2-(5-chloro-2-(cyclohexylmethoxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351711 3-(2-(5-bromo-2-(cyclohexylmethoxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351714 6-amino-4-benzamido-1,2-dihydro-2-(4-methoxyphenyl)-1,2,4-triazolo[4,3-a]quinoxalin-1-one 351715 N-(2-(4-methoxyphenyl)-1-oxo-1,2-dihydro-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl)-2,2-diphenylacetamide 351720 2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-4-(1-methylpiperidin-4-yl)-1H-indole 351731 1-(3'-cyano-biphenyl-4-yl)-1-(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-6-aza-spiro[2.5]octane-6-carboxylic acid dimethylamide 351732 4'-[1-(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-6-(pyrrolidine-1-carbonyl)-6-aza-spiro[2.5]oct-1-yl]-biphenyl-3-carbonitrile 351733 4'-[1-(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-6-(propane-2-sulfonyl)-6-aza-spiro[2.5]oct-1-yl]-biphenyl-3-carbonitrile 351734 1-(3'-cyano-biphenyl-4-yl)-1-(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-6-aza-spiro[2.5]octane-6-carboxylic acid diethylamide 351735 1'-{2-[2-(4-fluorophenyl)-1,3-oxazol-4-yl]ethyl}-6-methyl-1,2-dihydrospiro[3,1-benzoxazine-4,4'-piperidine]-2-one 351737 Tyr-Pro-D-Phg-Phe-NH2 351738 4'-[(1-cyclopropylmethyl-piperidin-4-ylidene)-(4,6-dichloro-1H-benzoimidazol-2-yl)-methyl]-biphenyl-3-carbonitrile 351742 3-(2-(2-(4-fluorobenzyloxy)-5-chlorophenyl)-5-(trifluoromethyl)-1H-pyrrol-1-yl)benzoic acid 351743 3-(2-(2-(2,4-difluorobenzyloxy)-5-chlorophenyl)-5-(trifluoromethyl)-1H-pyrrol-1-yl)benzoic acid 351744 3-(2-(2-(cyclohexylmethoxy)-5-(trifluoromethyl)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 351751 3-(2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-1H-indol-4-yl)-N,N-dimethylpropan-1-amine 351753 2-(2-(5-(4-chlorophenethyl)-1,2,4-oxadiazol-3-yl)-1H-indol-4-yl)-N,N-dimethylethanamine 351769 N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-(dimethylamino)ethylamino)-2-phenylacetamide 351770 1-{3-[4-(tert-butyl) phenyl]-5-N,N-dimethylamino-(1,2,4-triazol-4-yl)}-3-phenol 351772 3-(1-(1,2-dihydroacenaphthylen-1-yl)piperidin-4-yl)-5-fluoro-1H-indole 351773 (R)-1-(3-(1-(cyclooctylmethyl)piperidin-4-yl)-5-fluoro-1H-indol-1-yl)-3-(dimethylamino)propan-2-ol 351774 2-(1H-indazol-3-yl)-5-(4-(piperidin-1-yl)piperidin-1-yl)-1H-benzo[d]imidazole 351775 2-(1H-indazol-3-yl)-N-methyl-N-(1-methylpiperidin-4-yl)-1H-benzo[d]imidazol-5-amine 351785 (R)-6-(6-(3-(methylamino)pyrrolidin-1-yl)pyridin-3-yl)-2-(4-(trifluoromethyl)phenyl)thieno[2,3-d]pyridazin-7(6H)-one 351799 3-(3-(3-tert-butylphenyl)-5-((dimethylamino)methyl)-4H-1,2,4-triazol-4-yl)phenol 351800 3-(3-(4-tert-butylphenyl)-5-((dimethylamino)methyl)-4H-1,2,4-triazol-4-yl)phenol 351825 (S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-(dimethylamino)ethylthio)-2-phenylacetamide 351826 (S)-N-(3,5-bis(trifluoromethyl)benzyl)-5-(dimethylamino)-2-phenylpentanamide 351827 2-[(1-cyclopropylmethyl-piperidin-4-ylidene)-(4-pyrimidin-5-yl-phenyl)-methyl]-5-fluoro-6-trifluoromethyl-1H-benzoimidazole 351828 1-[3-(4-biphenyl)-(1,2,4-triazol-4-yl)]-3-phenol 351829 1-{3-[4-(tert-butyl)phenyl]-5-[2-(N,N-dimethylamino)ethyl]-(1,2,4-triazol-4-yl)}-3-phenol 351836 2-(2-(3-(4-fluorophenethyl)-1,2,4-oxadiazol-5-yl)-1H-indol-4-yl)-N,N-dimethylethanamine 351854 4'-[(1-cyclopropylmethyl-piperidin-4-ylidene)-(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-methyl]-biphenyl-3-carbonitrile 351855 1-[(3-naphthalen-2-yl)-(1,2,4-triazol-4-yl)]-3-phenol 351856 4'-[(1-cyclopropylmethyl-piperidin-4-ylidene)-(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-methyl]-biphenyl-3-carboxylic acid amide 351857 (S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-(piperidin-1-yl)ethylamino)-2-(thiophen-3-yl)acetamide 351858 4'-[1-(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-6-aza-spiro[2.5]oct-1-yl]-biphenyl-3-carbonitrile 351861 5-(4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)phenyl)pyrrolidine-3-carboxylic acid 351864 dimethyl-(2-{2-[3-(2-p-tolyl-ethyl)-[1,2,4]oxadiazol-5-yl]-1H-indol-4-yl}-ethyl)-amine 351869 4-fluoro-N-(2-morpholinoethyl)-3-((2-(pyridin-2-ylamino)thiazol-5-ylmethyl)amino)benzamide 351878 (2R)-2-(1-benzofuran-5-yl)-2-[(3R,6R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(2-methylpropyl)-2,5-dioxo-1-piperazinyl]-N-(1-methylethyl)ethanamide 351887 4'-[(1-cyclopropylmethyl-piperidin-4-ylidene)-(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-methyl]-6-fluoro-biphenyl-3-carbonitrile 351889 (S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-phenyl-2-(2-(piperidin-1-yl)ethylamino)acetamide 351890 (S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(4-fluorophenyl)-2-(2-(piperidin-1-yl)ethylamino)acetamide 351891 4'-[6-cyclopropylmethyl-1-(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-6-aza-spiro[2.5]oct-1-yl]-biphenyl-3-carbonitrile 351895 3-(1-(cyclooctylmethyl)piperidin-4-yl)-1H-pyrrolo[2,3-b]pyridine 351897 2-(5-phenoxy-1H-indazol-3-yl)-5-(4-(piperidin-1-yl)piperidin-1-yl)-1H-benzo[d]imidazole 351898 2-(2-(3-(4-methoxyphenethyl)-1,2,4-oxadiazol-5-yl)-1H-indol-4-yl)-N,N-dimethylethanamine 351903 2,4-difluoro-N-methyl-5-((2-(pyridin-2-ylamino)thiazol-5-ylmethyl)amino)benzamide 351916 5-{4-[(1-cyclopropylmethyl-piperidin-4-ylidene)-(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-methyl]-phenyl}-nicotinonitrile 351918 4'-[(1-acetyl-piperidin-4-ylidene)-(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-methyl]-biphenyl-3-carbonitrile 351919 [1-(3'-cyano-biphenyl-4-yl)-1-(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-6-aza-spiro[2.5]oct-6-yl]-acetic acid 351922 3-(1-(1,2-dihydroacenaphthylen-1-yl)piperidin-4-yl)-1H-pyrrolo[2,3-b]pyridine 351923 3-(1-(1,2-dihydroacenaphthylen-1-yl)piperidin-4-yl)-1-methyl-1H-pyrrolo[2,3-b]pyridine 351924 N-(cyclohexylmethyl)-3-(5-(4-(piperidin-1-yl)piperidin-1-yl)-1H-benzo[d]imidazol-2-yl)-1H-indazol-5-amine 351926 2-(2-(3-(4-(trifluoromethyl)phenethyl)-1,2,4-oxadiazol-5-yl)-1H-indol-4-yl)-N,N-dimethylethanamine 351942 {4'-[(1-cyclopropylmethyl-piperidin-4-ylidene)-(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-methyl]-biphenyl-3-yl}-acetonitrile 351943 N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-(diethylamino)ethylamino)-2-phenylacetamide 351944 N-(3,5-bis(trifluoromethyl)benzyl)-2-phenyl-2-(2-(pyrrolidin-1-yl)ethylamino)acetamide 351945 4'-[(1-cyclopropanecarbonyl-piperidin-4-ylidene)-(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-methyl]-biphenyl-3-carbonitrile 351946 1-(2-(3-methylpyridin-2-yl)quinazolin-4-yl)-3-phenylurea 351949 2-(3-(1-(1,2-dihydroacenaphthylen-1-yl)piperidin-4-yl)-1H-pyrrolo[2,3-b]pyridin-1-yl)ethanol 351951 1-tert-butyl-3-(3-(5-(4-(piperidin-1-yl)piperidin-1-yl)-1H-benzo[d]imidazol-2-yl)-1H-indazol-5-yl)urea 351952 methyl 3-(5-(4-(piperidin-1-yl)piperidin-1-yl)-1H-benzo[d]imidazol-2-yl)-1H-indazole-5-carboxylate 351969 2-[(3'-cyano-biphenyl-4-yl)-(1-cyclopropylmethyl-piperidin-4-ylidene)-methyl]-1H-benzoimidazole-5-carbonitrile 351971 N-(3,5-bis(trifluoromethyl)benzyl)-2-phenyl-2-(2-(piperidin-1-yl)ethylamino)acetamide 351972 (S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-(azepan-1-yl)ethylamino)-2-phenylacetamide 351976 1-(1,2-dihydroacenaphthylen-1-yl)-4-(1-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)piperidin-3-ol 351977 2-(6-fluoro-1H-indazol-3-yl)-5-(4-(piperidin-1-yl)piperidin-1-yl)-1H-benzo[d]imidazole 351978 2-(6-(benzyloxy)-1H-indazol-3-yl)-5-(4-(piperidin-1-yl)piperidin-1-yl)-1H-benzo[d]imidazole 351998 N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-morpholinoethylamino)-2-phenylacetamide 351999 4'-[(1-cyclopropylmethyl-piperidin-4-ylidene)-(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-methyl]-biphenyl-2-carbonitrile 352003 5-(1H-imidazol-1-yl)-2-(1H-indazol-3-yl)-1H-benzo[d]imidazole 352005 2-(trans-5-(4-(5-(4-((R)-3,3-difluorocyclopentyl)phenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-3-yl)acetic acid 352021 2-(5-methoxy-1H-indazol-3-yl)-5-(4-(piperidin-1-yl)piperidin-1-yl)-1H-benzo[d]imidazole 352022 1-(8-ethyl-2-furan-2-yl-8,9b-dihydro-3H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-p-tolyl-urea 352023 4'-[(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-piperidin-4-ylidene-methyl]-biphenyl-3-carbonitrile 352024 1-3-[3-(tert-butyl) phenyl]-5-N,N-dimethylamino-(1,2,4-triazol-4-yl)]-3-phenol 352025 3-(2-(2-(3,4-dichlorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 352026 3-(1-(1,2-dihydroacenaphthylen-1-yl)piperidin-4-yl)-6-fluoro-1H-indole 352027 (2R)-1-(3-(1-(1,2-dihydroacenaphthylen-1-yl)piperidin-4-yl)-6-fluoro-1H-indol-1-yl)-3-(dimethylamino)propan-2-ol 352028 2-(1H-indazol-3-yl)-5-(3-(pyrrolidin-1-yl)propoxy)-1H-benzo[d]imidazole 352029 2-(1H-indazol-3-yl)-5-((4-methylpiperazin-1-yl)methyl)-1H-benzo[d]imidazole 352030 2-(trans-5-(4-(5-(4-(4,4-difluorocyclohexyl)phenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-3-yl)acetic acid 352053 3-(1-benzyl-1,2,3,6-tetrahydropyridin-4-yl)-5-chloro-1H-indole 352057 1-(8-ethyl-2-furan-2-yl-8,9b-dihydro-3H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-fluoro-phenyl)-urea 352058 1-(8-ethyl-2-furan-2-yl-8,9b-dihydro-3H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(2-methoxy-phenyl)-urea 352059 4'-{(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-[1-(2-hydroxy-ethyl)-piperidin-4-ylidene]-methyl}-biphenyl-3-carbonitrile 352060 1-[3-(3-biphenyl)-5-N,N-dimethylamino-(1,2,4-triazol-4-yl)]-3-phenol 352061 3-(2-(2-(2-chloro-4-fluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 352063 7-chloro-3-(1-(cyclooctylmethyl)piperidin-4-yl)-1H-indole 352064 7-chloro-3-(1-(1,2-dihydroacenaphthylen-1-yl)piperidin-4-yl)-1H-indole 352065 2-(4-(benzyloxy)-1H-indazol-3-yl)-5-(4-(piperidin-1-yl)piperidin-1-yl)-1H-benzo[d]imidazole 352067 2-(2-(3-(4-chlorobenzyl)-1,2,4-oxadiazol-5-yl)-1H-indol-4-yl)-N,N-dimethylethanamine 352071 4-fluoro-3-((2-(pyridin-2-ylamino)thiazol-5-ylmethyl)amino)-N-(pyridin-2-ylmethyl)benzamide 352080 1-((R)-3-amino-2-hydroxypropyl)-3-(1-(1,2-dihydroacenaphthylen-1-yl)-1,2,3,6-tetrahydropyridin-4-yl)-1H-indole-5-carbonitrile 352084 2-(5-(benzyloxy)-1H-indazol-3-yl)-5-(4-(piperidin-1-yl)piperidin-1-yl)-1H-benzo[d]imidazole 352086 5-{4-[(1-cyclopropylmethyl-piperidin-4-ylidene)-(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-methyl]-phenyl}-6-hydroxy-nicotinonitrile 352088 1-[3-(4-biphenyl)-5-N,N-dimethylamino-(1,2,4-triazol-4-yl)]-3-phenol 352089 (2S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-(2-methylpiperidin-1-yl)ethylamino)-2-phenylacetamide 352090 N-(5-(5-(1-acetylpiperazine-4-carbonyl)-4-hydroxy-2-methylphenylthio)thiazol-2-yl)-4-(dimethylamino)benzamide 352093 3-(1-(cyclohexylmethyl)piperidin-4-yl)-1H-pyrrolo[2,3-b]pyridine 352095 1-tert-butyl-3-(3-(5-(4-(piperidin-1-yl)piperidin-1-yl)-1H-benzo[d]imidazol-2-yl)-1H-indazol-4-yl)urea 352096 2-(2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-1H-indol-4-yl)-N,N-dimethylethanamine 352103 N-cyclopropyl-2,4-difluoro-5-((2-(pyridin-2-ylamino)thiazol-5-yl)methylamino)benzamide 352110 3-(1-(1,2-dihydroacenaphthylen-1-yl)-1,2,3,6-tetrahydropyridin-4-yl)-6-fluoro-1H-indole 352111 3-(1-benzylpiperidin-4-yl)-5-chloro-1H-indole 352117 1-{3-[3-(tert-butyl) phenyl]-(1,2,4-triazol-4-yl)]-3-phenol 352119 (S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-(4-methylpiperidin-1-yl)ethylamino)-2-phenylacetamide 352120 4-[(3'-cyano-biphenyl-4-yl)-(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-methylene]-piperidine-1-carboxylic acid dimethylamide 352123 3-(1-(4-phenoxybenzyl)piperidin-4-yl)-1H-pyrrolo[2,3-b]pyridine 352124 3-(1-(naphthalen-1-ylmethyl)piperidin-4-yl)-1H-pyrrolo[2,3-b]pyridine 352125 2-(5-(4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)phenyl)pyrrolidin-3-yl)acetic acid 352128 2-(2-(3-((4-chlorophenoxy)methyl)-1,2,4-oxadiazol-5-yl)-1H-indol-4-yl)-N,N-dimethylethanamine 352138 5-chloro-2-methyl-3-(1-(naphthalen-1-ylmethyl)piperidin-4-yl)-1H-indole 352147 5-{4-[(1-cyclopropylmethyl-piperidin-4-ylidene)-(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-methyl]-phenyl}-pyridin-2-ol 352148 1-3-[4-(tert-butyl) phenyl]-(1,2,4-triazol-4-yl)]-3-phenol 352149 (S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-phenyl-2-(2-(4-phenylpiperidin-1-yl)ethylamino)acetamide 352150 4'-[(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-(1-methanesulfonyl-piperidin-4-ylidene)-methyl]-biphenyl-3-carbonitrile 352153 2-(trans-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-3-yl)acetic acid 352154 2-(cis-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-3-yl)acetic acid 352166 (3Z,6Z,9Z,12Z)-17-((R)-1-hydroxypropan-2-ylamino)-17-oxoheptadeca-3,6,9,12-tetraenyl 2-azido-5-iodobenzoate 352171 1-[3-(3-biphenyl)-(1,2,4-triazol-4-yl)]-3-phenol 352173 4'-{(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-[1-(propane-2-sulfonyl)-piperidin-4-ylidene]-methyl}-biphenyl-3-carbonitrile 352174 5-chloro-3-(1-(cyclooctylmethyl)piperidin-4-yl)-2-methyl-1H-indole 352175 5-chloro-3-(1-(1,2-dihydroacenaphthylen-1-yl)piperidin-4-yl)-2-methyl-1H-indole 352176 2-(1H-indazol-3-yl)-1H-benzo[d]imidazole 352177 2-(1H-indazol-3-yl)-4-morpholino-1H-benzo[d]imidazole 352181 2-(trans-5-(4-(5-(4-cyclopentylphenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-3-yl)acetic acid 352182 2-(trans-5-(4-(5-(4-cyclohexylphenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-3-yl)acetic acid 352210 2-{4-[(3'-cyano-biphenyl-4-yl)-(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-methylene]-piperidin-1-yl}-acetamide 352211 1-[(3-naphthalen-2-yl)-5-N,N-dimethylamino-(1,2,4-triazol-4-yl)]-3-phenol 352212 4'-[(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-(1-thiazol-2-ylmethyl-piperidin-4-ylidene)-methyl]-biphenyl-3-carbonitrile 352213 4'-{(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-[1-(thiophene-2-carbonyl)-piperidin-4-ylidene]-methyl}-biphenyl-3-carbonitrile 352214 4'-{(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-[1-(1-methyl-1H-pyrrole-2-carbonyl)-piperidin-4-ylidene]-methyl}-biphenyl-3-carbonitrile 352215 4-[(3'-cyano-biphenyl-4-yl)-(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-methylene]-piperidine-1-carboxylic acid diethylamide 352216 4'-[6-benzyl-1-(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-6-aza-spiro[2.5]oct-1-yl]-biphenyl-3-carbonitrile 352217 4'-[6-(2-diethylamino-ethyl)-1-(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-6-aza-spiro[2.5]oct-1-yl]-biphenyl-3-carbonitrile 352222 4-[(3'-cyano-biphenyl-4-yl)-(5-fluoro-6-trifluoromethyl-1H-benzoimidazol-2-yl)-methylene]-piperidine-1-sulfonic acid dimethylamide 352223 5-fluoro-3-(1-(naphthalen-1-ylmethyl)piperidin-4-yl)-1H-indole 352224 3-(1-(cyclooctylmethyl)piperidin-4-yl)-5-fluoro-1H-indole 352225 2-(1H-indazol-3-yl)-5-morpholino-1H-benzo[d]imidazole 352226 2-(1H-indazol-3-yl)-5-(4-methylpiperazin-1-yl)-1H-benzo[d]imidazole 352227 2-(trans-5-(4-(5-(4-(3,3,3-trifluoropropyl)phenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-3-yl)acetic acid 352229 5-(4-(piperidin-1-yl)piperidin-1-yl)-2-(6-(trifluoromethyl)-1H-indazol-3-yl)-1H-benzo[d]imidazole 352230 2-(7-fluoro-1H-indazol-3-yl)-5-(4-(piperidin-1-yl)piperidin-1-yl)-1H-benzo[d]imidazole 352241 (R)-(+)-(4,5,6-trimethoxyindan-1-yl)methanamine 352242 (S)-(-)-(4,5,6-trimethoxyindan-1-yl)methanamine 352267 SID24274407 352268 trans-N-{3-[(R)-1-(3,5-bis-trifluoromethyl-phenyl)-ethoxymethyl]-3-phenyl-cyclobutyl}-acetamide 352269 cis-N-{3-[(R)-1-(3,5-bis-trifluoromethyl-phenyl)-ethoxymethyl]-3-phenyl-cyclobutyl}-acetamide 352284 N-(5-(2-(cyclohexyloxy)pyrimidin-4-yl)thiazol-2-yl)pyridin-2-amine 352295 trans-1-{3-[(R)-1-(3,5-bis-trifluoromethyl-phenyl)-ethoxymethyl]-3-phenyl-cyclobutyl}-pyrrolidin-2-one 352296 cis-1-{3-[(R)-1-(3,5-bis-trifluoromethyl-phenyl)-ethoxymethyl]-3-phenyl-cyclobutyl}-pyrrolidin-2-one 352297 trans-3-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)methyl)-1-amino-3-phenylcyclobutyl)(piperidin-1-yl)methanone 352317 2-(5,6-bis(benzyloxy)-1H-indazol-3-yl)-5-(4-(piperidin-1-yl)piperidin-1-yl)-1H-benzo[d]imidazole 352324 N-(5-(2-(cyclohexyloxy)-5-methylpyrimidin-4-yl)thiazol-2-yl)pyridin-2-amine 352325 N-(5-(2-(cyclohexyloxy)-6-methylpyrimidin-4-yl)thiazol-2-yl)pyridin-2-amine 352329 (2R)-2-(2,4-difluorophenyl)-2-[(3R,6R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(2-methylpropyl)-2,5-dioxo-1-piperazinyl]ethanamide 352351 3-(5-(4-(piperidin-1-yl)piperidin-1-yl)-1H-benzo[d]imidazol-2-yl)-N-(thiazol-2-ylmethyl)-1H-indazol-5-amine 352356 N-(5-(2-(cyclohexyloxy)-6-methylpyrimidin-4-yl)thiazol-2-yl)-5-((4-methylpiperazin-1-yl)methyl)pyrazin-2-amine 352358 c(his-D-phe-arg-trp-Aoc) 352359 c(his-D-phe-arg-trp-Ahp) 352367 c(his-D-phe-arg-trp-Ahx) 352368 (2R)-2-(2,4-difluorophenyl)-2-[(3R,6R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(2-methylpropyl)-2,5-dioxo-1-piperazinyl]-N-methylethanamide 352369 (2R)-2-(2,4-difluorophenyl)-2-[(3R,6R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(2-methylpropyl)-2,5-dioxo-1-piperazinyl]-N,N-dimethylethanamide 352397 (2R)-2-(1,3-benzodioxol-5-yl)-2-[(3R,6R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(2-methylpropyl)-2,5-dioxo-1-piperazinyl]-N-(1,1-dimethylethyl)ethanamide 352423 8-(4-(4-benzylpiperazin-1-ylsulfonyl)phenyl)-1-propyl-1H-purine-2,6(3H,7H)-dione 352424 8-[4-(isopropylamidosulfonyl)phenyl]-1,3-dimethylxanthine 352427 N-benzyl-3-(5-(4-(piperidin-1-yl)piperidin-1-yl)-1H-benzo[d]imidazol-2-yl)-1H-indazol-5-amine 352428 N-(1-benzylpiperidin-4-yl)-3-(5-(4-(piperidin-1-yl)piperidin-1-yl)-1H-benzo[d]imidazol-2-yl)-1H-indazol-5-amine 352442 (2R)-2-(2,3-dihydro-1-benzofuran-5-yl)-2-[(3R,6R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(2-methylpropyl)-2,5-dioxo-1-piperazinyl]-N-(1,1-dimethylethyl)ethanamide 352451 1-(3-methoxyphenyl)-3-(5-(pyridin-4-yl)-1,3,4-thiadiazol-2-yl)urea 352455 8-[4-(phenylethylamidosulfonyl)phenyl]-1,3-dimethylxanthine 352456 2-(5-(benzyloxy)-6-methoxy-1H-indazol-3-yl)-5-(4-(piperidin-1-yl)piperidin-1-yl)-1H-benzo[d]imidazole 352467 (2R)-2-{(3R,6R)-3-(2,3-dihydro-1H-inden-2-yl)-6-[(1R)-1-methylpropyl]-2,5-dioxo-1-piperazinyl}-2-[2-fluoro-4-(4-morpholinyl)phenyl]-N-(1-methylethyl)ethanamide 352470 c(his-D-phe-arg-trp-Abu) 352486 1-(3,4-dichlorophenyl)-4-(4-hydroxy-3-methoxybenzylidene)pyrazolidine-3,5-dione 352487 8-[4-(2-Hydroxyethylamidosulfonyl)phenyl]-1-propylxanthine 352488 8-[4-(butylamidosulfonyl)phenyl]-1,3-dimethylxanthine 352489 N-(3-(5-(4-(piperidin-1-yl)piperidin-1-yl)-1H-benzo[d]imidazol-2-yl)-1H-indazol-5-yl)furan-2-carboxamide 352500 (3R,6R)-1-[(1R)-2-(1-azetidinyl)-1-(2,4-difluorophenyl)-2-oxoethyl]-3-(2,3-dihydro-1H-inden-2-yl)-6-(2-methylpropyl)-2,5-piperazinedione 352505 (R)-3-((1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)methyl)-3-phenylcyclobutanone 352506 (R)-3-((1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)methyl)-3-phenylcyclobutanamine 352507 2-(5-(2-chlorophenyl)-1H-pyrazol-3-yl)-4-methoxyphenol 352509 4-(1-propylxanthin-8-yl)phenylsulfonamidoacetic acid 352510 8-[4-(2-hydroxyethylamidosulfonyl)phenyl]-1,3-dimethylxanthine 352511 2-(5-(2-methoxyphenoxy)-1H-indazol-3-yl)-5-(4-(piperidin-1-yl)piperidin-1-yl)-1H-benzo[d]imidazole 352512 N-(furan-2-ylmethyl)-3-(5-(4-(piperidin-1-yl)piperidin-1-yl)-1H-benzo[d]imidazol-2-yl)-1H-indazol-5-amine 352524 (3R,6R)-1-[(1R)-1-(2,4-difluorophenyl)-2-(4-morpholinyl)-2-oxoethyl]-3-(2,3-dihydro-1H-inden-2-yl)-6-(2-methylpropyl)-2,5-piperazinedione 352528 (+/-)-(2,3-dihydro-4,5,6-trimethoxy-1H-inden-1-yl)aminomethane 352529 8-[4-(dipropylamidosulfonyl)phenyl]-1-propylxanthine 352530 2-(5-(3-methoxyphenoxy)-1H-indazol-3-yl)-5-(4-(piperidin-1-yl)piperidin-1-yl)-1H-benzo[d]imidazole 352543 c(his-L-phe-arg-trp-Aoc) 352545 (2R)-2-(2,4-difluorophenyl)-2-[(3R,6R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(2-methylpropyl)-2,5-dioxo-1-piperazinyl]-N-(2-hydroxyethyl)-N-methylethanamide 352549 trans-3-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)methyl)-1-amino-3-phenylcyclobutanecarboxamide 352550 cis-3-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)methyl)-1-amino-3-phenylcyclobutanecarboxamide 352555 N-{(R)-1-(4-chloro-benzyl)-2-[4-(1-methyl-4-phenyl-piperidin-4-yl)-piperazin-1-yl]-2-oxo-ethyl}-2-(2,3-dihydro-1H-isoindol-1-yl)-acetamide trifluoroacetic acid 352556 N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-hexyl-1-methyl-piperidin-4-yl)-piperazin-1-yl]-2-oxo-ethyl}-2-(2,3-dihydro-1H-isoindol-1-yl)-acetamide trifluoroacetic acid 352557 N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-ethyl-1-methyl-piperidin-4-yl)-piperazin-1-yl]-2-oxo-ethyl}-2-(2,3-dihydro-1H-isoindol-1-yl)-acetamide trifluoroacetic acid 352558 N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-isopropyl-1-methyl-piperidin-4-yl)-piperazin-1-yl]-2-oxo-ethyl}-2-(2,3-dihydro-1H-isoindol-1-yl)-acetamide trifluoroacetic acid 352564 8-[4-(phenylamidosulfonyl)phenyl]-1-propylxanthine 352567 2-(5-(4-methoxyphenoxy)-1H-indazol-3-yl)-5-(4-(piperidin-1-yl)piperidin-1-yl)-1H-benzo[d]imidazole 352587 (3R,6R)-1-[(1R)-1-(2,4-difluorophenyl)-2-(3-hydroxy-1-azetidinyl)-2-oxoethyl]-3-(2,3-dihydro-1H-inden-2-yl)-6-(2-methylpropyl)-2,5-piperazinedione 352588 TCMDC-138777 352591 trans-3-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)methyl)-1-amino-N-methyl-3-phenylcyclobutanecarboxamide 352592 cis-3-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)methyl)-1-amino-N-methyl-3-phenylcyclobutanecarboxamide 352616 (3R,6R)-1-[(1R)-1-(2,4-difluorophenyl)-2-hydroxyethyl]-3-(2,3-dihydro-1H-inden-2-yl)-6-(2-methylpropyl)-2,5-piperazinedione 352621 diethyl 4-(4-acetamidophenylamino)quinoline-3,6-dicarboxylate 352622 trans-3-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)methyl)-1-amino-N,N-dimethyl-3-phenylcyclobutanecarboxamide 352623 trans-3-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)methyl)-1-amino-3-phenylcyclobutyl)(pyrrolidin-1-yl)methanone 352649 (Z)-3-(2-(4-fluorophenylamino)-4-oxothiazol-5(4H)-ylidene)-1-methylindolin-2-one 352676 5-(5-(2-(allyloxy)-5-bromobenzylidene)-4-oxo-4,5-dihydrothiazol-2-ylamino)-2-chlorobenzoic acid 352677 GNF-Pf-2722 352681 N-benzyl-4-(2,6-dioxo-1-propyl-2,3,6,7-tetrahydro-1H-purin-8-yl)benzenesulfonamide 352706 (2R)-2-[(3R,6R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(2-methylpropyl)-2,5-dioxo-1-piperazinyl]-N-(1,1-dimethylethyl)-2-[4-(4-hydroxy-1-piperidinyl)phenyl]ethanamide 352715 8-[4-(phenylethylamidosulfonyl)phenyl]-1-propylxanthine 352735 3-ethyl 6-methyl 4-(3-acetylphenylamino)quinoline-3,6-dicarboxylate 352736 (R)-3-((1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)methyl)-N-benzyl-3-phenylcyclobutanamine 352737 (R)-5-((3-((1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)methyl)-3-phenylcyclobutylamino)methyl)-2H-1,2,4-triazol-3(4H)-one 352742 N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-cyclohexylmethyl-1-methyl-piperidin-4-yl)-piperazin-1-yl]-2-oxo-ethyl}-2-(2,3-dihydro-1H-isoindol-1-yl)-acetamide trifluoroacetic acid 352743 N-[(R)-2-[4-(4-benzyl-1-methyl-piperidin-4-yl)-piperazin-1-yl]-1-(4-chloro-benzyl)-2-oxo-ethyl]-2-(2,3-dihydro-1H-isoindol-1-yl)-acetamide trifluoroacetic acid 352780 N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-isobutyl-tetrahydro-thiopyran-4-yl)-piperazin-1-yl]-2-oxo-ethyl}-2-(2,3-dihydro-1H-isoindol-1-yl)-acetamide trifluoroacetic acid 352781 N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-isobutyl-1,1-dioxo-hexahydrothiopyran-4-yl)-piperazin-1-yl]-2-oxo-ethyl}-2-(2,3-dihydro-1H-isoindol-1-yl)-acetamide trifluoroacetic acid 352782 N-((R)-3-(4-chlorophenyl)-1-(4-(1-cyclohexyl-3-(diethylamino)propan-2-yl)piperazin-1-yl)-1-oxopropan-2-yl)-2-(isoindolin-1-yl)acetamide 352817 N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-isobutyl-1-isobutyryl-piperidin-4-yl)-piperazin-1-yl]-2-oxo-ethyl}-2-(2,3-dihydro-1H-isoindol-1-yl)-acetamide trifluoroacetic acid 352818 N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-isobutyl-1-methanesulfonyl-piperidin-4-yl)-piperazin-1-yl]-2-oxo-ethyl}-2-(2,3-dihydro-1H-isoindol-1-yl)-acetamide trifluoroacetic acid 352819 N-{(R)-1-(4-chloro-benzyl)-2-[4-(1-isobutyl-cyclohexyl)-piperazin-1-yl]-2-oxo-ethyl}-2-(2,3-dihydro-1H-isoindol-1-yl)-acetamide trifluoroacetic acid 352820 N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-isobutyl-tetrahydro-pyran-4-yl)-piperazin-1-yl]-2-oxo-ethyl}-2-(2,3-dihydro-1H-isoindol-1-yl)-acetamide trifluoroacetic acid 352832 2-(4-(1,3-dimethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)phenylsulfonamido)acetic acid 352896 8-chloro-2-fluoro-11-(4-methylpiperazin-1-yl)-dibenzo[b,f][1,4]oxazepine 352911 N-(tert-Butyl)-N'-(4-{2,4-diamino-6-[(benzyloxy)methyl]pyrimidin-5-yl}phenyl)urea 352943 7-chloro-3-fluoro-11-(4-methylpiperazin-1-yl)-dibenzo[b,f][1,4]oxazepine 352953 N-(4-{2,4-diamino-6-[(benzyloxy)methyl]pyrimidin-5-yl}-phenyl)-N'-phenyl-urea 352954 N-benzyl-N'-(4-{2,4-diamino-6-[(benzyloxy)methyl]pyrimidin-5-yl}phenyl-urea 352980 N-(4-{2,4-diamino-6-[(benzyloxy)methyl]pyrimidin-5-yl}phenyl)-thiophene-3-carboxamide 352981 N-(4-{2,4-diamino-6-[(benzyloxy)methyl]pyrimidin-5-yl}-phenyl)-N'-(1-phenylethyl)urea 352982 N-(4-{2,4-diamino-6-[(benzyloxy)methyl]pyrimidin-5-yl}-phenyl)-N'-(2-phenylethyl)urea 352993 8-chloro-11-(4-isopropylpiperazin-1-yl)-dibenzo[b,f][1,4]oxazepine 353009 N-(4-{2,4-diamino-6-[(benzyloxy)methyl]pyrimidin-5-yl}-phenyl)-2-thien-3-ylacetamide 353010 2-(2-bromothien-3-yl)-N-(4-{2,4-diamino-6-[(benzyloxy)methyl]pyrimidin-5-yl}phenyl)-acetamide 353014 N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-isobutyl-1-methyl-piperidin-4-yl)-piperazin-1-yl]-2-oxo-ethyl}-2-(2,3-dihydro-1H-isoindol-1-yl)-acetamide trifluoroacetic id 353015 N-{(R)-1-(4-chloro-benzyl)-2-[4-(1-ethyl-4-isobutyl-piperidin-4-yl)-piperazin-1-yl]-2-oxo-ethyl}-2-(2,3-dihydro-1H-isoindol-1-yl)-acetamide trifluoroacetic acid 353016 N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-isobutyl-1-isopropyl-piperidin-4-yl)-piperazin-1-yl]-2-oxo-ethyl}-2-(2,3-dihydro-1H-isoindol-1-yl)-acetamide trifluoroacetic acid 353017 N-[(R)-2-[4-(1-acetyl-4-isobutyl-piperidin-4-yl)-piperazin-1-yl]-1-(4-chloro-benzyl)-2-oxo-ethyl]-2-(2,3-dihydro-1H-isoindol-1-yl)-acetamide trifluoroacetic acid 353046 N-[4-(2,4-diamino-6-benzyloxymethyl-pyrimidin-5-yl)-phenyl]-propionamide 353047 N-[4-(2,4-diamino-6-benzyloxymethyl-pyrimidin-5-yl)-phenyl]-3-methyl-butyramide 353048 N-(4-{2,4-diamino-6-[(benzyloxy)methyl]pyrimidin-5-yl}-phenyl)-2-phenylacetamide 353049 N-(4-{2,4-diamino-6-[(benzyloxy)methyl]pyrimidin-5-yl}-phenyl)-3-phenylpropanamide 353058 2-[4-(8-chloro-5H-dibenzo[b,e][1,4]diazepin-11-yl)-piperazin-1-yl]-ethanol 353068 3,8-dichloro-11-(4-methylpiperazin-1-yl)-dibenzo[b,f][1,4]oxazepine 353069 8-chloro-4-Fluoro-11-(4-methylpiperazin-1-yl)-dibenzo[b,f][1,4]oxazepine 353070 7-chloro-11-(4-methylpiperazin-1-yl)dibenzo[b,f][1,4]oxazepine 353077 cyclopropanecarboxylic acid [4-(2,4-diamino-6-benzyloxymethyl-pyrimidin-5-yl)-phenyl]-amide 353078 cyclopentanecarboxylic acid [4-(2,4-diamino-6-benzyloxymethyl-pyrimidin-5-yl)-phenyl]-amide 353079 1-[4-(2,4-diamino-6-benzyloxymethyl-pyrimidin-5-yl)-phenyl]-3-isopropyl-urea 353103 7-methyl-11-(4-methyl-piperazin-1-yl)-dibenzo[b,f][1,4]oxazepine 353110 cyclopentanecarboxylic acid [4-(2,4-diamino-6-benzyloxymethyl-pyrimidin-5-yl)-phenyl]-methyl-amide 353111 tetrahydro-furan-2-carboxylic acid [4-(2,4-diamino-6-benzyloxymethyl-pyrimidin-5-yl)-phenyl]-amide 353128 4,7-dichloro-11-(4-methylpiperazin-1-yl)-dibenzo[b,f][1,4]oxazepine 353133 N-[4-(2,4-diamino-6-benzyloxymethyl-pyrimidin-5-yl)-phenyl]-isonicotinamide 353156 7-chloro-4-fluoro-11-(4-methylpiperazin-1-yl)-dibenzo[b,f][1,4]oxazepine 353161 6-ethyl-5-[1-(4-methanesulfonyl-benzyl)-1H-benzoimidazol-5-yl]-pyrimidine-2,4-diamine 353162 5-[2-cyclopentyl-1-(4-methanesulfonyl-benzyl)-1H-benzoimidazol-5-yl]-6-ethyl-pyrimidine-2,4-diamine 353192 6-ethyl-5-[1-(4-methanesulfonyl-benzyl)-2-phenyl-1H-benzoimidazol-5-yl]-pyrimidine-2,4-diamine 353193 N-[4-(2,4-diamino-6-benzyloxymethyl-pyrimidin-5-yl)-phenyl]-acetamide 353273 rac-8-fluoro-3-[[2-(5-fluoro-1H-indol-3-yl)ethyl](propyl)amino] chromane-5-carboxamide 353282 4-amino-5-cyano-6-ethoxy-pyridine-2-carboxylic acid 2,5-dimethoxy-benzylamide 353289 (S)-2-Acetamido-N-((R)-1-((2S,4S)-2-(3-guanidinopropyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)-3-(1H-imidazol-4-yl)propanamide 353290 (S)-N-((R)-1-((2S,4S)-2-(3-guanidinopropyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 353291 (S)-N-((R)-1-((2S,4S)-2-(3-guanidinopropyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)piperidine-2-carboxamide 353292 (S)-2-acetamido-N1-((R)-1-((2S,4S)-2-(3-guanidinopropyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)pentanediamide 353293 (S)-2-acetamido-N-((R)-1-((2R,4S)-2-(3-guanidinopropyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)-3-(4-hydroxyphenyl)propanamide 353294 (S)-2-acetamido-N-((R)-1-((2R,4S)-2-(3-guanidinopropyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)-3-(1H-imidazol-4-)propanamide 353295 (S)-N-((R)-1-((2R,4S)-2-(3-guanidinopropyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 353296 (S)-N-((R)-1-((2R,4S)-2-(3-guanidinopropyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)piperidine-2-carboxamide 353308 rac-8-fluoro-3-[[4-(5-fluoro-1H-indol-3-yl)butyl](propyl)amino] chromane-5-carboxamide 353309 rac-3-{(cyclopropylmethyl)[2-(5-fluoro-1H-indol-3-yl)ethyl]amino}-8-fluorochromane-5-carboxamide 353344 (S)-2-acetamido-N1-((R)-1-((2R,4S)-2-(3-guanidinopropyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)pentanediamide 353352 Demotensin 3 353353 Demotensin 4 353362 rac-3-{(cyclopropylmethyl)[4-(5-fluoro-1H-indol-3-yl)butyl]amino}-8-fluorochromane-5-carboxamide 353363 rac-3-{cyclobutyl[4-(5-fluoro-1H-indol-3-yl)butyl]amino}-8-fluorochromane-5-carboxamide 353366 H2N-CO-DPhe-c[Cys-Aph(CONH2)-DTrp-Lys-Thr-Cys]-Thr-NH2 353371 H2N-CO-Phe-c[Cys-Aph(CONH2)-DTrp-Lys-Thr-Cys]-Thr-NH2 353372 H2N-CO-DPhe-c[Cys-Aph(CONHOCH3)-DTrp-Lys-Thr-Cys]-Thr-NH2 353373 H-c[Cys-Phe-DTrp-Lys-Thr-Cys]-OH 353406 4-amino-5-cyano-6-ethoxy-pyridine-2-carboxylic acid methylamide 353425 Ac-His-D-Phe-Arg-2-Nal-NHCH3 353428 (2R,4R)-1-((R)-2-((S)-2-acetamido-3-(1H-imidazol-4-yl)propanamido)-3-phenylpropanoyl)-N-(2-guanidinoethyl)-4-(naphthalen-2-ylmethoxy)pyrrolidine-2-carboxamide 353429 (2R,4R)-1-((R)-2-((S)-2-amino-3-(1H-imidazol-4-yl)propanamido)-3-phenylpropanoyl)-N-(2-guanidinoethyl)-4-(naphthalen-2-ylmethoxy)pyrrolidine-2-carboxamide 353430 (2R,4R)-1-((R)-2-((S)-2-acetamido-3-(4-hydroxyphenyl)propanamido)-3-phenylpropanoyl)-N-(2-guanidinoethyl)-4-(naphthalen-2-ylmethoxy)pyrrolidine-2-carboxamide 353431 (S)-N-((R)-1-((2R,4R)-2-(2-guanidinoethylcarbamoyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 353433 (3R)-8-fluoro-3-[[3-(5-fluoro-1H-indol-3-yl)propyl](methyl)amino]chromane-5-carboxamide 353451 4-amino-5-cyano-6-ethoxy-pyridine-2-carboxylic acid benzylamide 353469 (R)-3-(ethyl(3-(5-fluoro-1H-indol-3-yl)propyl)amino)-8-fluoro-3,4-dihydro-2H-chromene-5-carboxamide 353470 (S)-3-(ethyl(3-(5-fluoro-1H-indol-3-yl)propyl)amino)-8-fluoro-3,4-dihydro-2H-chromene-5-carboxamide 353484 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-ethoxypicolinamide 353497 8-Fluoro-3-{[3-(5-fluoro-1H-indol-3-yl)propyl](propyl)amino}-chromane-5-carboxamide 353498 (3R)-(-)-8-Fluoro-3-{[3-(5-fluoro-1H-indol-3-yl)propyl](propyl)amino}chromane-5-carboxamide 353504 (4R,7S,10S,13R,16S,19R)-13-((1H-indol-3-yl)methyl)-N-((2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl)-19-((R)-2-amino-3-phenylpropanamido)-10-(4-aminobutyl)-16-benzyl-7-((R)-1-hydroxyethyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentaazacycloicosane-4-carboxamide 353511 4-amino-5-cyano-6-ethoxy-pyridine-2-carboxylic acid 2-sulfamoyl-benzylamide 353512 4-amino-5-cyano-6-ethoxy-pyridine-2-carboxylic acid (pyridin-3-ylmethyl)-amide 353517 H-D-Phe-c[Cys-Ala-D-Trp-Lys-Thr-Cys]-Thr-NH2 353529 (3S)-(+)-8-Fluoro-3-{[3-(5-fluoro-1H-indol-3-yl)propyl](propyl)amino}-chromane-5-carboxamide 353530 rac-3-{(cyclopropylmethyl)[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide 353531 N-((R)-1-((2S,4R)-2-(3-guanidinopropyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)acetamide 353532 1-(3-((2S,4R)-1-((R)-2-amino-3-phenylpropanoyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-2-yl)propyl)guanidine 353538 4-(5-{[(4-amino-5-cyano-6-ethoxy-pyridine-2-carbonyl)-amino]-methyl}-pyridin-2-yl)-benzoic acid 353568 (S)-N-((R)-1-((2R,4R)-2-(2-guanidinoethylcarbamoyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)piperidine-2-carboxamide 353569 N-((R)-1-((2R,4R)-2-(2-guanidinoethylcarbamoyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)piperidine-4-carboxamide 353570 (S)-2-acetamido-N1-((R)-1-((2R,4R)-2-(2-guanidinoethylcarbamoyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)pentanediamide 353571 (S)-2-acetamido-N-((R)-1-((2S,4R)-2-(3-guanidinopropyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)-3-(1H-imidazol-4-yl)propanamide 353585 4-amino-5-cyano-6-ethoxy-pyridine-2-carboxylic acid (4-methanesulfonyl-benzyl)-methylamide 353604 (S)-2-acetamido-N-((R)-1-((2S,4R)-2-(3-guanidinopropyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)-3-(4-hydroxyphenyl)propanamide 353605 (S)-2-acetamido-N1-((R)-1-((2S,4R)-2-(3-guanidinopropyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)pentanediamide 353606 (S)-N-((R)-1-((2S,4R)-2-(3-guanidinopropyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 353607 (S)-N-((R)-1-((2S,4R)-2-(3-guanidinopropyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)piperidine-2-carboxamide 353608 (S)-N-((R)-1-((2S,4R)-2-(3-guanidinopropyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)pyrrolidine-2-carboxamide 353615 (S)-2-acetamido-N-((R)-1-((2S,4R)-2-(3-guanidinopropyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)-3-phenylpropanamide 353616 N-((R)-1-((2S,4R)-2-(3-guanidinopropyl)-4-(naphthalen-2-yl-methoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)-3-phenylpropanamide 353617 (S)-2-acetamido-N-((R)-1-((2R,4R)-2-(3-guanidinopropyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)-3-(4-hydroxyphenyl)propanamide 353635 N-(4-(methylsulfonyl)benzyl)-4-amino-5-chloro-6-ethoxypicolinamide 353636 4-amino-5-chloro-6-isopropoxy-pyridine-2-carboxylic acid 4-methanesulfonyl-benzylamide 353649 (3R)-3-{(cyclopropylmethyl)[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide 353658 4-amino-6-chloro-5-cyano-pyridine-2-carboxylic acid 4-methanesulfonyl-benzylamide 353659 5-cyano-6-ethoxy-pyridine-2-carboxylic acid 4-methanesulfonyl-benzylamide 353671 (3S)-3-{(cyclopropylmethyl)[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide 353672 3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide 353695 5-cyano-N-(2,5-dimethoxybenzyl)-6-ethoxypyridine-2-carboxamide 353716 rac-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxy-N-methylchroman-3-amine 353717 (3R)-(-)-3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide 353718 (3S)-(+)-3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide 353736 rac-N-ethyl-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxychroman-3-amine 353737 N-[3-(5-Fluoro-1H-indol-3-yl)propyl]-5-methoxy-N-propylchroman-3-amine 353738 rac-3-{ethyl[2-(5-fluoro-1H-indol-3-yl)ethyl]amino}-8-fluorochromane-5-carboxamide 353739 rac-3-{ethyl[4-(5-fluoro-1H-indol-3-yl)butyl]amino}-8-fluorochromane-5-carboxamide 353765 rac-N-(cyclopropylmethyl)-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-N-(5-methoxy-3,4-dihydro-2H-chromen-3-yl)amine 353766 N-Cyclobutyl-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxychroman-3-amine 353788 (3R)-(-)-N-Cyclobutyl-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxychroman-3-amine 353789 (3R)-8-fluoro-3-{[3-(5-fluoro-1H-indol-3-yl)propyl]amino}chromane-5-carboxamide 353801 (S)-2-acetamido-N-((R)-1-((2R,4R)-2-(3-guanidinopropyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)-3-(1H-imidazol-4-yl)propanamide 353802 (S)-N-((R)-1-((2R,4R)-2-(3-guanidinopropyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 353803 (S)-N-((R)-1-((2R,4R)-2-(3-guanidinopropyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)piperidine-2-carboxamide 353804 (S)-2-acetamido-N1-((R)-1-((2R,4R)-2-(3-guanidinopropyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)pentanediamide 353805 (S)-2-acetamido-N-((R)-1-((2S,4S)-2-(3-guanidinopropyl)-4-(naphthalen-2-ylmethoxy)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)-3-(4-hydroxyphenyl)propanamide 353825 5-(p-toluidino)-N-(cyclohexylmethyl)-3-hydroxyisothiazole-4-carboxamidine 353834 5-(4-chloro-3-(trifluoromethyl)phenylamino)-3-hydroxyisothiazole-4-carbonitrile 353842 5-(2,4-dichlorophenylamino)-3-hydroxyisothiazole-4-carbonitrile 353857 5-(3,5-dichlorophenylamino)-3-hydroxyisothiazole-4-carbonitrile 353861 SID26731526 353864 5-(2,5-dichlorophenylamino)-3-hydroxyisothiazole-4-carbonitrile 353875 5-(4-chloro-3-nitrophenylamino)-N-(cyclohexylmethyl)-3-hydroxyisothiazole-4-carboxamidine 353880 N-(cyclohexylmethyl)-3-hydroxy-5-(2-methoxyphenylamino)isothiazole-4-carboxamidine 353881 5-(4-chlorophenylamino)-N-(cyclohexylmethyl)-3-hydroxyisothiazole-4-carboxamidine 353884 5-(3-chlorophenylamino)-N-(cyclohexylmethyl)-3-hydroxyisothiazole-4-carboxamidine 353885 5-(3-bromophenylamino)-N-(cyclohexylmethyl)-3-hydroxyisothiazole-4-carboxamidine 353886 5-(4-bromophenylamino)-N-(cyclohexylmethyl)-3-hydroxyisothiazole-4-carboxamidine 353890 N-(cyclohexylmethyl)-3-hydroxy-5-(pyridin-3-ylamino)isothiazole-4-carboxamidine 353891 methyl 4-(4-(N-(cyclohexylmethyl)carbamimidoyl)-3-hydroxyisothiazol-5-ylamino)benzoate 353898 N-(cyclohexylmethyl)-5-(2-fluorophenylamino)-3-hydroxyisothiazole-4-carboxamidine 353911 N-(cyclohexylmethyl)-3-hydroxy-5-(2-methoxy-4-nitrophenylamino)isothiazole-4-carboxamidine 353919 N-(cyclohexylmethyl)-5-(2,4-dimethylphenylamino)-3-hydroxyisothiazole-4-carboxamidine 353920 N-(cyclohexylmethyl)-5-(3,5-dichlorophenylamino)-3-hydroxyisothiazole-4-carboxamidine 353924 5-(3-bromophenylamino)-3-hydroxyisothiazole-4-carbonitrile 353925 SID26731729 353926 N-(cyclohexylmethyl)-5-(2,4-dichlorophenylamino)-3-hydroxyisothiazole-4-carboxamidine 353947 1-(3-fluoro-4-methoxyphenyl)-3-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-1H-pyrrol-2(5H)-one 353948 4-(3,4-dioxo-2-(phenylamino)cyclobut-1-enylamino)-3-hydroxybenzoic acid 353949 3-(3,4-dioxo-2-(phenylamino)cyclobut-1-enylamino)-2-hydroxybenzoic acid 353950 (3aS,8R,8aS)-6,7-dichloro-8-methyl-1,2,3,3a,8,8a-hexahydro-indeno[1,2-c]pyrrole 353957 1-(3-(2-(diethylamino)ethoxy)phenyl)-3-(3-(trifluoromethyl)phenylimino)indolin-2-one 353958 N-(4-(3-(3,4-dichlorophenyl)-2-oxo-2H-pyrrol-1(5H)-yl)-2-(2-(piperidin-1-yl)ethoxy)phenyl)acetamide 353959 1-(3-(3-(pyrrolidin-1-yl)propoxy)phenyl)-3-(3-(trifluoromethyl)phenylimino)indolin-2-one 353960 7-(2-(6-((dimethylamino)methyl)pyridin-2-yl)ethynyl)-4-(3,4,5-trimethoxyphenylamino)quinoline-3-carbonitrile 353979 1-(3-fluorophenyl)-3-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-1H-pyrrol-2(5H)-one 353980 1-(4-chlorophenyl)-3-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-4-methyl-1H-pyrrol-2(5H)-one 353981 methyl 3-(3,4-dioxo-2-(phenylamino)cyclobut-1-enylamino)-2-hydroxybenzoate 353982 3-(3,4-dioxo-2-(phenylamino)cyclobut-1-enylamino)-2-hydroxybenzamide 353989 1,3-dihydro-1-[3-(2-pyrrolidinylethoxy)phenyl]-3-[[3-(trifluoromethyl)phenyl]imino]-2H-indol-2-one 353990 1-(3-(2-(piperidin-1-yl)ethoxy)phenyl)-3-(3-(trifluoromethyl)phenylimino)indolin-2-one 353991 3-(3,4-dichlorophenyl)-1-(4-methyl-3-(2-(piperidin-1-yl)ethoxy)phenyl)-1H-pyrrol-2(5H)-one 353992 1-(3-(4-(diethylamino)butoxy)phenyl)-3-(3-(trifluoromethyl)phenylimino)indolin-2-one 354002 3-(3,4-dichlorophenyl)-1-(4-methoxy-3-(2-morpholinoethoxy)phenyl)-1H-pyrrol-2(5H)-one 354015 1-(3,4-dichlorophenyl)-3-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-4-methyl-1H-pyrrol-2(5H)-one 354016 3-(2-hydroxy-4-nitrophenylamino)-4-(phenylamino)cyclobut-3-ene-1,2-dione 354017 3-(3,4-dioxo-2-(phenylamino)cyclobut-1-enylamino)-2-hydroxy-N-methylbenzamide 354025 1-(3-(3-(dimethylamino)propoxy)phenyl)-3-(3-(trifluoromethyl)phenylimino)indolin-2-one 354026 3-(3,4-dichlorophenyl)-1-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-1H-pyrrol-2(5H)-one 354027 4-(2,4-dichloro-5-methoxyphenylamino)-7-(2-(5-((dimethylamino)methyl)thiophen-2-yl)ethynyl)-6-methoxyquinoline-3-carbonitrile 354028 4-(2,4-dichloro-5-methoxyphenylamino)-7-(2-(3-((dimethylamino)methyl)phenyl)ethynyl)-6-methoxyquinoline-3-carbonitrile 354035 3-(3,4-dichlorophenyl)-1-(4-methoxy-3-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-1H-pyrrol-2(5H)-one 354036 3-(3,4-dichlorophenyl)-1-(3-(2-(4,4-difluoropiperidin-1-yl)ethoxy)-4-methoxyphenyl)-1H-pyrrol-2(5H)-one 354054 1-(3-fluoro-4-methoxyphenyl)-3-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)pyrrolidin-2-one 354055 1-(3,4-dichlorophenyl)-3-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)pyrrolidin-2-one 354056 3-((2-hydroxyphenyl)(methyl)amino)-4-(phenylamino)cyclobut-3-ene-1,2-dione 354057 3-(4-nitrophenylamino)-4-(phenylamino)cyclobut-3-ene-1,2-dione 354058 3-(2-hydroxyphenylamino)-4-(phenylamino)cyclobut-3-ene-1,2-dione 354061 (3aS,8R,8aS)-6-chloro-5-methoxy-8-methyl-1,2,3,3a,8,8a-hexahydro-indeno[1,2-c]pyrrole 354067 1-(4-chloro-3-(2-(piperidin-1-yl)ethoxy)phenyl)-3-(3,4-dichlorophenyl)-1H-pyrrol-2(5H)-one 354068 4-(2,4-dichloro-5-methoxyphenylamino)-6-methoxy-7-(2-(5-((4-methylpiperazin-1-yl)methyl)pyridin-2-yl)ethynyl)quinoline-3-carbonitrile 354069 4-(2,4-dichloro-5-methoxyphenylamino)-7-(2-(4-((dimethylamino)methyl)phenyl)ethynyl)-6-methoxyquinoline-3-carbonitrile 354077 3-(3,4-dichlorophenyl)-1-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)-1H-pyrrol-2(5H)-one 354078 3-(3,4-dichlorophenyl)-1-(3-(2-(4,4-dimethylpiperidin-1-yl)ethoxy)-4-methoxyphenyl)-1H-pyrrol-2(5H)-one 354088 1-(3,4-dichlorophenyl)-3-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-3-methylpyrrolidin-2-one 354089 1-(3-fluorophenyl)-3-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)pyrrolidin-2-one 354093 (3aS,8R,8aS)-6-bromo-5-methoxy-8-methyl-1,2,3,3a,8,8a-hexahydro-indeno[1,2-c]pyrrole 354094 (3aS,8R,8aS)-6-chloro-5-ethoxy-8-methyl-1,2,3,3a,8,8a-hexahydro-indeno[1,2-c]pyrrole 354095 (3aS,8R,8aS)-6-chloro-8-methyl-1,2,3,3a,8,8a-hexahydro-indeno[1,2-c]pyrrol-5-ol 354096 (3aS,8R,8aS)-6-chloro-5,8-dimethyl-1,2,3,3a,8,8a-hexahydro-indeno[1,2-c]pyrrole 354103 1-(2-(2-(diethylamino)ethoxy)phenyl)-3-(3-(trifluoromethyl)phenylimino)indolin-2-one 354104 4-(2,4-dichloro-5-methoxyphenylamino)-6-methoxy-7-(2-(6-(2-(4-methylpiperazin-1-yl)ethyl)pyridin-2-yl)ethynyl)quinoline-3-carbonitrile 354105 4-(2,4-dichloro-5-methoxyphenylamino)-6-methoxy-7-(2-(6-((4-methylpiperazin-1-yl)methyl)pyridin-2-yl)ethynyl)quinoline-3-carbonitrile 354106 4-(2,4-dichloro-5-methoxyphenylamino)-7-(2-(6-((dimethylamino)methyl)pyridin-2-yl)ethynyl)-6-ethoxyquinoline-3-carbonitrile 354107 4-(2,4-dichloro-5-methoxyphenylamino)-7-(2-(6-((dimethylamino)methyl)pyridin-2-yl)ethynyl)quinoline-3-carbonitrile 354113 3-(3,4-dichlorophenyl)-1-(3-(2-(4-isopropylpiperidin-1-yl)ethoxy)-4-methoxyphenyl)-1H-pyrrol-2(5H)-one 354114 3-(3,4-dichlorophenyl)-1-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)pyrrolidin-2-one 354121 3-(3,4-dichlorophenyl)-1-(3-(2-(4,4-dimethylpiperidin-1-yl)ethoxy)-4-methoxyphenyl)pyrrolidin-2-one 354122 3-(3,4-dichlorophenyl)-1-(3-(2-(4-isopropylpiperidin-1-yl)ethoxy)-4-methoxyphenyl)pyrrolidin-2-one 354123 1-(3,4-dichlorophenyl)-3-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-1H-pyrrol-2(5H)-one 354124 3-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-1-(4-methoxyphenyl)-1H-pyrrol-2(5H)-one 354127 (3aS,8R,8aS)-5-chloro-6,8-dimethyl-1,2,3,3a,8,8a-hexahydro-indeno[1,2-c]pyrrole 354135 1-(2-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-3-(3-(trifluoromethyl)phenylimino)indolin-2-one 354136 1-(3-(2-(dimethylamino)ethoxy)phenyl)-3-(3-(trifluoromethyl)phenylimino)indolin-2-one 354137 4-(2,4-dichloro-5-methoxyphenylamino)-7-(2-(3-((dimethylamino)methyl)pyridin-2-yl)ethynyl)-6-methoxyquinoline-3-carbonitrile 354144 1-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)-3-(4-(trifluoromethyl)phenyl)-1H-pyrrol-2(5H)-one 354145 3-(4-bromophenyl)-1-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)-1H-pyrrol-2(5H)-one 354152 3-(3-fluorophenyl)-1-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)pyrrolidin-2-one 354153 3-(3,4-dichlorophenyl)-1-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-3-methylpyrrolidin-2-one 354154 1-(3-chloro-4-methoxyphenyl)-3-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-1H-pyrrol-2(5H)-one 354155 (+/-)-(3aS,8aS)-5-bromo-6,8-dimethyl-1,2,3,3a,8,8a-hexahydro-indeno[1,2-c]pyrrole 354158 (+/-)-(3aS,8aS)-5,6-dichloro-8-methyl-1,2,3,3a,8,8a-hexahydro-indeno[1,2-c]pyrrole 354166 4-(2,4-dichloro-5-methoxyphenylamino)-7-(2-(4-((dimethylamino)methyl)pyridin-2-yl)ethynyl)-6-methoxyquinoline-3-carbonitrile 354168 4-(2,4-dichloro-5-methoxyphenylamino)-7-(2-(5-((dimethylamino)methyl)pyridin-3-yl)ethynyl)-6-methoxyquinoline-3-carbonitrile 354174 3-(3-chlorophenyl)-1-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-1H-pyrrol-2(5H)-one 354175 3-(4-chlorophenyl)-1-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-1H-pyrrol-2(5H)-one 354182 3-(3,4-dichlorophenyl)-1-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)-3-methylpyrrolidin-2-one 354183 3-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-1-(4-methoxyphenyl)pyrrolidin-2-one 354185 (+/-)-(3aS,8aS)-6-bromo-5,8-dimethyl-1,2,3,3a,8,8a-hexahydro-indeno[1,2-c]pyrrole 354197 4-(2,4-dichloro-5-methoxyphenylamino)-7-(2-(6-(2-(dimethylamino)ethyl)pyridin-2-yl)ethynyl)-6-methoxyquinoline-3-carbonitrile 354202 1-(4-(2-(dimethylamino)ethoxy)phenyl)-3-(3-(trifluoromethyl)phenylimino)indolin-2-one 354203 3-(4-chlorophenyl)-1-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)-1H-pyrrol-2(5H)-one 354204 1-(4-(3-(diethylamino)propoxy)phenyl)-3-(3-(trifluoromethyl)phenylimino)indolin-2-one 354205 1-(4-(4-(diethylamino)butoxy)phenyl)-3-(3-(trifluoromethyl)phenylimino)indolin-2-one 354213 1-(3-chloro-4-methoxyphenyl)-3-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)pyrrolidin-2-one 354214 (3aS,8R,8aS)-6-chloro-8-methyl-1,2,3,3a,8,8a-hexahydro-indeno[1,2-c]pyrrole 354227 4-(2,4-dichloro-5-methoxyphenylamino)-7-(2-(5-((dimethylamino)methyl)pyridin-2-yl)ethynyl)-6-methoxyquinoline-3-carbonitrile 354233 3-(4-chloro-3-fluorophenyl)-1-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)-1H-pyrrol-2(5H)-one 354234 1-(4-(2-(diethylamino)ethoxy)phenyl)-3-(3-(trifluoromethyl)phenylimino)indolin-2-one 354243 1-(4-chloro-3-(2-(piperidin-1-yl)ethoxy)phenyl)-3-(3,4-dichlorophenyl)pyrrolidin-2-one 354244 (+/-)-(3aS,8aS)-5-fluoro-8-methyl-1,2,3,3a,8,8a-hexahydro-indeno[1,2-c]pyrrole 354245 (+/-)-(3aS,8aS)-4,8-dimethyl-1,2,3,3a,8,8a-hexahydro-indeno[1,2-c]pyrrole 354246 (+/-)-(3aS,8aS)-5,8-dimethyl-1,2,3,3a,8,8a-hexahydro-indeno[1,2-c]pyrrole 354247 (+/-)-(3aS,8aS)-6,8-dimethyl-1,2,3,3a,8,8a-hexahydro-indeno[1,2-c]pyrrole 354258 4-(2,4-dichloro-5-methoxyphenylamino)-7-(2-(6-((dimethylamino)methyl)pyridin-2-yl)ethynyl)-6-methoxyquinoline-3-carbonitrile 354265 3-(4-fluorophenyl)-1-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)-1H-pyrrol-2(5H)-one 354266 1-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)-3-p-tolyl-1H-pyrrol-2(5H)-one 354274 3-(3,4-dichlorophenyl)-1-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)pyrrolidin-2-one 354275 3-(3,4-dichlorophenyl)-1-(3-(2-(piperidin-1-yl)ethoxy)-4-(trifluoromethoxy)phenyl)pyrrolidin-2-one 354276 (+/-)-(3aS,8aS)-7,8-dimethyl-1,2,3,3a,8,8a-hexahydro-indeno[1,2-c]pyrrole 354277 (+/-)-(3aS,8aS)-6-chloro-5-methoxy-8-methyl-1,2,3,3a,8,8a-hexahydro-indeno[1,2-c]pyrrole 354278 (+/-)-(3aS,8aS)-5-chloro-6,8-dimethyl-1,2,3,3a,8,8a-hexahydro-indeno[1,2-c]pyrrole 354279 (+/-)-(3aS,8aS)-6-chloro-5,8-dimethyl-1,2,3,3a,8,8a-hexahydro-indeno[1,2-c]pyrrole 354286 (R)-3-(2-(2,3-dihydro-1H-inden-1-ylamino)-3,4-dioxocyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide 354287 3-(3,4-dioxo-2-(pentan-3-ylamino)cyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide 354294 (R)-1-(3-(3-(diethylamino)-2-hydroxypropoxy)phenyl)-3-(3-(trifluoromethyl)phenylimino)indolin-2-one 354304 N-(4-(3-(3,4-dichlorophenyl)-2-oxopyrrolidin-1-yl)-2-(2-(piperidin-1-yl)ethoxy)phenyl)acetamide 354305 3-(3-chlorophenyl)-1-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)pyrrolidin-2-one 354312 (E)-5-(4-Hydroxybenzylidene)-1-phenethylhydantoin 354314 3-(3,4-dioxo-2-(phenylamino)cyclobut-1-enylamino)-N-ethyl-2-hydroxybenzamide 354315 2-hydroxy-3-(2-(isopropylamino)-3,4-dioxocyclobut-1-enylamino)-N,N-dimethylbenzamide 354316 3-(2-(tert-butylamino)-3,4-dioxocyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide 354322 3-(3,4-dichlorophenyl)-1-(3-(2-(piperidin-1-yl)ethoxy)-4-(pyrrolidin-1-yl)phenyl)-1H-pyrrol-2(5H)-one 354323 (S)-1-(3-(3-(diethylamino)-2-hydroxypropoxy)phenyl)-3-(3-(trifluoromethyl)phenylimino)indolin-2-one 354324 1-(3-((diethylamino)methoxy)phenyl)-3-(3-(trifluoromethyl)phenylimino)indolin-2-one 354334 3-(4-fluorophenyl)-1-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)pyrrolidin-2-one 354335 3-(3,4-dichlorophenyl)-1-(4-methyl-3-(2-(piperidin-1-yl)ethoxy)phenyl)pyrrolidin-2-one 354342 N-benzyl-3-(3,4-dioxo-2-(phenylamino)cyclobut-1-enylamino)-2-hydroxybenzamide 354343 3-(3,4-dioxo-2-(phenylamino)cyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide 354344 3-(2-(furan-2-ylmethylamino)-3,4-dioxocyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide 354345 3-(3,4-dioxo-2-(phenethylamino)cyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide 354351 3-(3-fluorophenyl)-1-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-1H-pyrrol-2(5H)-one 354352 1-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-3-(3-(trifluoromethyl)phenyl)-1H-pyrrol-2(5H)-one 354353 1-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-3-p-tolyl-1H-pyrrol-2(5H)-one 354354 3-(4-bromophenyl)-1-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-1H-pyrrol-2(5H)-one 354370 5-chloro-3-(3,4-dioxo-2-(phenylamino)cyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide 354371 2-hydroxy-N,N-dimethyl-3-(2-(methyl(phenyl)amino)-3,4-dioxocyclobut-1-enylamino)benzamide 354380 3-(4-fluorophenyl)-1-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-1H-pyrrol-2(5H)-one 354381 1-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-3-(4-(trifluoromethyl)phenyl)-1H-pyrrol-2(5H)-one 354382 3-(3-chlorophenyl)-1-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)-1H-pyrrol-2(5H)-one 354399 3-(2-(cyclohexylamino)-3,4-dioxocyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide 354400 3-(2-(cyclopentylamino)-3,4-dioxocyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide 354409 1-(3-(3-(diethylamino)-2-hydroxypropoxy)phenyl)-3-(3-(trifluoromethyl)phenylimino)indolin-2-one 354438 3-(2-hydroxy-5-nitrophenylamino)-4-(phenylamino)cyclobut-3-ene-1,2-dione 354439 3-(3,4-dioxo-2-(phenylamino)cyclobut-1-enylamino)-4-hydroxybenzonitrile 354440 4-(3,4-dioxo-2-(phenylamino)cyclobut-1-enylamino)-3-hydroxybenzonitrile 354441 3-(3,4-dioxo-2-(tetrahydro-2H-pyran-4-ylamino)cyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide 354442 (3aS,8R,8aS)-5,6-dichloro-8-methyl-1,2,3,3a,8,8a-hexahydro-indeno[1,2-c]pyrrole 354443 (3aS,8S,8aS)-5,6-dichloro-8-methyl-1,2,3,3a,8,8a-hexahydro-indeno[1,2-c]pyrrole 354450 1-(3-(3-(diethylamino)propoxy)phenyl)-3-(3-(trifluoromethyl)phenylimino)indolin-2-one 354452 7-(2-(6-((dimethylamino)methyl)pyridin-2-yl)ethynyl)-6-methoxy-4-(3,4,5-trimethoxyphenylamino)quinoline-3-carbonitrile 354466 4-[4-(2,6-dichloro-phenyl)-3-oxo-2,3-dihydro-1H-3a,7,9,9b-tetraaza-cyclopenta[a]naphthalen-8-ylamino]-benzoic acid methyl ester 354467 4-(2,6-dichloro-phenyl)-8-(4-dimethylamino-phenylamino)-1,2-dihydro-3a,7,9,9b-tetraaza-cyclopenta[a]naphthalen-3-one 354468 N-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-2-m-tolylacetamide 354473 7-(4-bromophenyl)-3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-4H-chromen-4-one 354474 3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-7-(4-ethylphenyl)-4H-chromen-4-one 354486 3-(3,4-dichlorophenyl)-1-methyl-1-((5-(7-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)urea 354487 4-(5-((2,4-dichlorophenethylamino)methyl)thiophen-2-yl)-N-methylpyrimidin-2-amine 354488 1-((1S,2R,5S)-5-(4-aminophenyl)bicyclo[3.1.0]hexan-2-yl)-3-(3-chloro-4-fluorophenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)urea 354489 3-(4-fluoro-3-(trifluoromethyl)phenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)-1-((1S,2R,5S)-5-(thiophen-3-yl)bicyclo[3.1.0]hexan-2-yl)urea 354491 N-(2-(2,4-dichlorophenyl)propyl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide 354492 4-(2,6-dichloro-phenyl)-8-(4-diethylamino-phenylamino)-1,2-dihydro-3a,7,9,9b-tetraaza-cyclopenta[a]naphthalen-3-one 354493 7-((1H-imidazol-1-yl)methyl)-3-(thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole 354494 3-(5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)-N-m-tolylpropanamide 354501 3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-7-(4-(trifluoromethyl)phenyl)-4H-chromen-4-one 354502 3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-7-(4-methoxyphenyl)-4H-chromen-4-one 354516 7-(4-chlorophenyl)-3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-1-methylquinolin-4(1H)-one 354518 1-(4'-piperidin-1-ylmethyl-biphenyl-4-ylmethyl)piperidin-2-one 354524 (S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(4-fluorophenyl)-5-(piperidin-1-yl)pentanamide 354529 7-((4-methylpiperazin-1-yl)methyl)-3-(thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole 354530 1-((5-(7-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-m-tolylurea 354539 3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-7-(4-(trifluoromethoxy)phenyl)-4H-chromen-4-one 354540 7-(2,4-dichlorophenyl)-3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-4H-chromen-4-one 354551 4,4'-[Biphenyl-4,4'-diylbis(methylene)]bis-(piperazin-1yl-ethan-2-one) 354552 3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-1-methyl-7-(4-(trifluoromethyl)phenyl)quinolin-4(1H)-one 354553 1-[4-(4'-Piperidin-1-ylmethyl-biphenyl-4-ylmethyl)-piperazin-1yl]ethanone 354554 Cyclohexyl-(4'-piperidin-1-ylmethyl-biphenyl-4-ylmethyl)amine 354555 3-(2-chlorophenyl)-1-methyl-1-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)urea 354559 3-hydroxy-5-4-iodo-2-methylphenylamino-N-isopropylisothiazole-4-carboximidamide 354560 3-hydroxy-N-(1-hydroxypropan-2-yl)-5-(4-iodo-2-methylphenylamino)isothiazole-4-carboxamidine 354561 5-2-chloro-4-iodophenylamino-3-hydroxy-N-isopropylisothiazole-4-carboximidamide 354562 1-((1S,2R,5S)-5-(4-acetamidophenyl)bicyclo[3.1.0]hexan-2-yl)-3-(3-chloro-4-fluorophenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)urea 354566 1-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-m-tolylurea 354578 3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-7-phenoxy-4H-chromen-4-one 354579 3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-7-(4-fluorophenoxy)-4H-chromen-4-one 354580 1,1'-[Biphenyl-4,4'-diylbis(ethylene)]bis-piperidine 354581 1-ethyl-1-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-m-tolylurea 354584 1-(2-methoxyethyl)-1-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-m-tolylurea 354591 5-(2-chloro-4-iodophenylamino)-3-hydroxy-N-(1-hydroxypropan-2-yl)isothiazole-4-carboxamidine 354592 5-(2-chloro-4-(trifluoromethyl)phenylamino)-3-hydroxy-N-isopropylisothiazole-4-carboxamidine 354593 5-(2-chloro-4-(trifluoromethyl)phenylamino)-3-hydroxy-N-(1-hydroxypropan-2-yl)isothiazole-4-carboxamidine 354594 3-(3-chloro-4-fluorophenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)-1-((1S,2R,5S)-5-(3-propionamidophenyl)bicyclo[3.1.0]hexan-2-yl)urea 354595 (S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(4-fluorophenyl)-4-(4-(thiophen-3-yl)piperidin-1-yl)butanamide 354598 1-((4-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-m-tolylurea 354606 N,N'-[biphenyl-4,4'diylbis(methylene)]bis-dimethylamine 354617 N,N'-[biphenyl-4,4'diylbis(methylene)]bis-cyclohexylamine 354621 1-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-1-propyl-3-m-tolylurea 354625 5-(2,3-dichlorophenylamino)-3-hydroxy-N-isopropylisothiazole-4-carboxamidine 354626 5-2,3-dichlorophenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 354629 N-(4-bromophenethyl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide 354631 3-(2,6-dichlorophenyl)-N-(4-fluorophenyl)-1,2-dimethyl-1,2-dihydropyrimido[4,5-c]pyridazin-7-amine 354632 1-((4-(7-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-m-tolylurea 354633 N-((R)-1-amino-3-(2,4-dichlorophenyl)propan-2-yl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide 354644 3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-7-phenyl-4H-chromen-4-one 354645 N,N'-[biphenyl-4,4'diylbis(methylene)]bis-pentylamine 354659 1-((1S,2R,5S)-5-(3-(azetidin-1-yl)phenyl)bicyclo[3.1.0]hexan-2-yl)-3-(3-chloro-4-fluorophenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)urea 354664 4-(2,6-dichloro-phenyl)-8-(4-fluoro-phenylamino)-1,2-dihydro-3a,7,9,9b-tetraaza-cyclopenta[a]naphthalen-3-one 354665 N-((S)-1-amino-3-(2,4-dichlorophenyl)propan-2-yl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide 354666 N-((S)-1-(2,4-dichlorophenyl)-3-(dimethylamino)propan-2-yl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide 354673 3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-7-(4-fluorophenyl)-4H-chromen-4-one 354674 1,1'-[Biphenyl-4,4'-diylbis(methylene)]bis-piperidine 354678 3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-7-(4-methoxypyridin-3-yl)-4H-chromen-4-one 354684 1-((5-(7-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-phenylurea 354687 3-(3-chloro-4-fluorophenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)-1-((1S,2R,5S)-5-(3-(pyrrolidin-1-yl)phenyl)bicyclo[3.1.0]hexan-2-yl)urea 354692 3-(3-chloro-4-fluorophenyl)-1-((1S,2R,5S)-5-(3-isobutyramidophenyl)bicyclo[3.1.0]hexan-2-yl)-1-(3-(4-methylpiperazin-1-yl)propyl)urea 354694 3-(3-chloro-4-fluorophenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)-1-((1S,2R,5S)-5-(3-pivalamidophenyl)bicyclo[3.1.0]hexan-2-yl)urea 354695 1-(3-chloro-4-fluorophenyl)-3-[(1S,2R,5S)-5-{3-[(ethylcarbamoyl)amino]phenyl}bicyclo[3.1.0]hexan-2-yl]-3-[3-(4-methylpiperazin-1-yl)propyl]urea 354698 5-(2-methylamino-pyrimidin-4-yl)-thiophene-2-carboxylic acid [2-(4-sulfamoyl-phenyl)-ethyl]-amide 354700 4-(2,6-dichloro-phenyl)-8-phenylamino-1,2-dihydro-3a,7,9,9b-tetraaza-cyclopenta[a]naphthalen-3-one 354701 4-(2,6-dichloro-phenyl)-8-methylamino-1,2-dihydro-3a,7,9,9b-tetraaza-cyclopenta[a]naphthalen-3-one 354702 N-((S)-4-amino-1-(2,4-dichlorophenyl)butan-2-yl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide 354703 N-(2-aminoethyl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide 354704 N-(2-(dimethylamino)ethyl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide 354710 7-(4-chlorophenyl)-3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-4H-chromen-4-one 354714 1,1'-[Biphenyl-4,4'-diylbis(methylene)]bis-4-methylpiperidine 354715 3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-7-(4-(trifluoromethyl)pyridin-3-yl)-4H-chromen-4-one 354718 7-(4-chlorophenoxy)-3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-4H-chromen-4-one 354724 1-((5-(7-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-o-tolylurea 354728 N-(2,4-dichlorophenethyl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide 354729 N-(2,4-dichlorophenethyl)-5-(2-aminopyrimidin-4-yl)thiophene-2-carboxamide 354730 4-(2,6-dichloro-phenyl)-8-(4-methoxy-phenylamino)-1,2-dihydro-3a,7,9,9b-tetraaza-cyclopenta[a]naphthalen-3-one 354731 trans-(S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(4-fluorophenyl)-4-(3-methyl-4-phenylpiperidin-1-yl)butan-1-amine 354740 1,1'-[Biphenyl-4,4'-diylbis(methylene)]bis(3,5-dimethylpiperidine) 354743 N,N'-[biphenyl-4,4'diylbis(methylene)]bis-(N-methyl-N-cyclohexylamine) 354744 3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-7-(p-tolyloxy)-4H-chromen-4-one 354755 (S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(4-fluorophenyl)-4-(piperidin-1-yl)butanamide 354759 N-(2,4-dichlorophenethyl)-5-(2-(ethylamino)pyrimidin-4-yl)thiophene-2-carboxamide 354760 3-(4-fluoro-3-(trifluoromethyl)phenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)-1-((1S,2R,5S)-5-(thiazol-2-yl)bicyclo[3.1.0]hexan-2-yl)urea 354761 N-(2-(2,4-dichlorophenyl)butyl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide 354774 7-(4-chloro-3-methylphenyl)-3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-4H-chromen-4-one 354775 4,4'-[Biphenyl-4,4'-diylbis(methylene)]bis-morpholine 354776 (S)-7-(4-chlorophenyl)-3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-4H-chromen-4-one 354778 3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-7-(4-methoxyphenoxy)-4H-chromen-4-one 354785 3-(4-bromophenyl)-1-methyl-1-((5-(7-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)urea 354786 (2S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(4-fluorophenyl)-4-(4-phenylpiperidin-1-yl)butanamide 354788 3-(4-fluoro-3-(trifluoromethyl)phenyl)-1-((1S,2R,5S)-5-(6-methoxypyridin-3-yl)bicyclo[3.1.0]hexan-2-yl)-1-(3-(4-methylpiperazin-1-yl)propyl)urea 354789 N-((S)-2-amino-2-(2,4-dichlorophenyl)ethyl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide 354790 N-((R)-1-(2,4-dichlorophenyl)propan-2-yl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide 354800 7-(4-chloro-2-methylphenyl)-3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-4H-chromen-4-one 354801 3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-7-(4-methoxy-2-methylphenyl)-4H-chromen-4-one 354803 7-(2,3-dihydrobenzofuran-5-yloxy)-3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-4H-chromen-4-one 354809 1-isobutyl-1-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-m-tolylurea 354814 3-(4-chlorophenyl)-1-methyl-1-((5-(7-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)urea 354815 3-hydroxy-5-4-iodophenylamino-N-isopropylisothiazole-4-carboximidamide 354817 (S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(4-fluorophenyl)-5-(4-phenylpiperidin-1-yl)pentanamide 354819 3-(4-fluoro-3-(trifluoromethyl)phenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)-1-((1S,2R,5S)-5-(6-oxo-1,6-dihydropyridin-3-yl)bicyclo[3.1.0]hexan-2-yl)urea 354820 (2S)-methyl 3-(2,4-dichlorophenyl)-2-(2-(2-(methylamino)pyrimidin-4-yl)thiophene-5-carboxamido)propanoate 354821 N-((S)-3-(2,4-dichlorophenyl)-1-hydroxypropan-2-yl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide 354840 7-(2,4-dimethoxyphenyl)-3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-4H-chromen-4-one 354841 7-(benzo[d][1,3]dioxol-5-yl)-3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-4H-chromen-4-one 354853 3-hydroxy-N-(1-hydroxypropan-2-yl)-5-(4-iodophenylamino)isothiazole-4-carboxamidine 354854 methyl 4-((1R,4S,5R)-4-(3-(4-fluoro-3-(trifluoromethyl)phenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)ureido)bicyclo[3.1.0]hexan-1-yl)benzoate 354855 (2S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(4-fluorophenyl)-4-(3-methyl-4-phenylpiperazin-1-yl)butanamide 354857 (R)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(4-fluorophenyl)-2-methyl-4-(4-phenylpiperidin-1-yl)butan-1-amine 354858 N-(1-amino-3-(2,4-dichlorophenyl)propan-2-yl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide 354861 4-(2,6-dichloro-phenyl)-8-[4-(2-dimethylamino-ethyl)-phenylamino]-1,2-dihydro-3a,7,9,9b-tetraaza-cyclopenta[a]naphthalen-3-one 354862 4-(2,6-dichloro-phenyl)-8-(4-morpholin-4-yl-phenylamino)-1,2-dihydro-3a,7,9,9b-tetraaza-cyclopenta[a]naphthalen-3-one 354872 3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-7-(2,3,4a,5,8,8a-hexahydrobenzo[b][1,4]dioxin-6-yl)-4H-chromen-4-one 354880 1-isopropyl-1-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-m-tolylurea 354881 1-isopentyl-1-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-m-tolylurea 354886 1-methyl-1-((5-(7-((4-methylpiperazin-1-yl)methyl)-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-(3-(trifluoromethyl)phenyl)urea 354887 1-methyl-1-((5-(7-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-(4-(trifluoromethoxy)phenyl)urea 354892 3-(3-chloro-4-fluorophenyl)-1-((1S,2R,5S)-5-(4-fluorophenyl)bicyclo[3.1.0]hexan-2-yl)-1-(3-(4-methylpiperazin-1-yl)propyl)urea 354894 (R)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(4-fluorophenyl)-4-(4-phenylpiperidin-1-yl)butanamide 354896 (2S)-N-[3,5-bis(trifluoromethyl)benzyl]-2-(4-fluorophenyl)-4-(1'H-spiro[indene-1,4'-piperidin]-1'yl)butanamide 354897 (2S)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-4-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-2-(4-fluorophenyl)butanamide 354898 1-((1S,2R,5S)-5-(3-aminobenzo[d]isoxazol-6-yl)bicyclo[3.1.0]hexan-2-yl)-3-(4-fluoro-3-(trifluoromethyl)phenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)urea 354899 1-((1S,2R,5S)-5-(3-aminobenzo[d]isoxazol-5-yl)bicyclo[3.1.0]hexan-2-yl)-3-(4-fluoro-3-(trifluoromethyl)phenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)urea 354906 3-(4-fluoro-3-(trifluoromethyl)phenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)-1-((1S,2R,5S)-5-(2-oxoindolin-5-yl)bicyclo[3.1.0]hexan-2-yl)urea 354908 (2S)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-2-(4-fluorophenyl)-4-{5'-methylspiro[indene-1,4'-piperidine]-1'-yl}butanamide 354909 (2S)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-4-{5'-ethylspiro[indene-1,4'-piperidine]-1'-yl}-2-(4-fluorophenyl)butanamide 354910 (2S)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-2-(4-fluorophenyl)-4-[(1S,5'S)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]butanamide 354911 (2S)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-2-(4-fluorophenyl)-4-[(1R,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]butanamide 354912 N-(4-fluorobenzyl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide 354918 4-(2,6-dichloro-phenyl)-8-[4-(2-diethylamino-ethoxy)-phenylamino]-1,2-dihydro-3a,7,9,9b-tetraaza-cyclopenta[a]naphthalen-3-one 354919 4-(2-chloro-5-methoxy-phenyl)-8-(4-fluoro-phenylamino)-1,2-dihydro-3a,7,9,9b-tetraaza-cyclopenta[a]naphthalen-3-one 354934 1-cyclopropyl-1-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-m-tolylurea 354937 3-(3-chloro-4-fluorophenyl)-1-((1S,2R,5S)-5-(3-methoxyphenyl)bicyclo[3.1.0]hexan-2-yl)-1-(3-(4-methylpiperazin-1-yl)propyl)urea 354941 N-(3-(4-fluorophenyl)propyl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide 354942 5-(2-(methylamino)pyrimidin-4-yl)-N-phenethylthiophene-2-carboxamide 354943 (2S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(4-fluorophenyl)-4-(4-phenylpiperidin-1-yl)pentan-1-amine 354946 4-(2-chloro-5-methoxy-phenyl)-8-(4-dimethylamino-phenylamino)-1,2-dihydro-3a,7,9,9b-tetraaza-cyclopenta[a]naphthalen-3-one 354947 4-(2-chloro-5-hydroxy-phenyl)-8-(4-dimethylamino-phenylamino)-1,2-dihydro-3a,7,9,9b-tetraaza-cyclopenta[a]naphthalen-3-one 354961 1-methoxy-1-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-m-tolylurea 354963 3-(3-chlorophenyl)-1-methyl-1-((5-(7-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)urea 354969 N-(4-fluorophenethyl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide 354970 3-(4-fluorophenyl)-N-(5-(2-(methylamino)pyrimidin-4-yl)thiophen-2-yl)propanamide 354971 N-(3-chlorophenethyl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide 354972 N-(2-chlorophenethyl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide 354973 cis-(S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(4-fluorophenyl)-4-(3-methyl-4-phenylpiperidin-1-yl)butan-1-amine 354976 4-(2,6-dichloro-phenyl)-8-(3-methoxy-phenylamino)-1,2-dihydro-3a,7,9,9b-tetraaza-cyclopenta[a]naphthalen-3-one 354977 3-methyl-N-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)benzamide 354992 3-(3-fluoro-5-(trifluoromethyl)phenyl)-1-methyl-1-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)urea 354993 1-methyl-1-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-(3-(trifluoromethoxy)phenyl)urea 354998 3-(4-fluorophenyl)-1-methyl-1-((5-(7-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)urea 355001 3-(4-fluoro-3-(trifluoromethyl)phenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)-1-((1S,2R,5S)-5-(4-(methylsulfonyl)phenyl)bicyclo[3.1.0]hexan-2-yl)urea 355002 3-(4-fluoro-3-(trifluoromethyl)phenyl)-1-((1S,2R,5S)-5-(4-(methylcarbamoyl)phenyl)bicyclo[3.1.0]hexan-2-yl)-1-(3-(4-methylpiperazin-1-yl)propyl)urea 355003 benzyl 4-((1S,4R,5S)-4-(3-(3-chloro-4-fluorophenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)ureido)bicyclo[3.1.0]hexan-1-yl)phenylcarbamate 355004 1-(2,4-dichlorobenzyl)-3-(5-(2-(methylamino)pyrimidin-4-yl)thiophen-2-yl)urea 355005 4-fluorobenzyl 5-(2-(methylamino)pyrimidin-4-yl)thiophen-2-ylcarbamate 355006 N-(4-chlorophenethyl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide 355007 3-(3-chloro-4-fluorophenyl)-1-((1S,2R,5S)-5-(3-(cyclopropanecarboxamido)phenyl)bicyclo[3.1.0]hexan-2-yl)-1-(3-(4-methylpiperazin-1-yl)propyl)urea 355010 4-(2,6-dichloro-phenyl)-8-(2-methoxy-phenylamino)-1,2-dihydro-3a,7,9,9b-tetraaza-cyclopenta[a]naphthalen-3-one 355011 4-(2,6-dichloro-phenyl)-8-(4-ethoxy-phenylamino)-1,2-dihydro-3a,7,9,9b-tetraaza-cyclopenta[a]naphthalen-3-one 355012 9-hydroxy-5-methyl-4-phenylpyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355013 5-ethyl-9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355017 1-(2-chlorophenyl)-3-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)urea 355031 2-(2,5-dimethyl-3-(8-methylquinolin-4-yl)-1H-indol-1-yl)acetic acid 355032 2-(3-(8-chloroquinolin-4-yl)-2,5-dimethyl-1H-indol-1-yl)acetic acid 355033 1-(4-(4-aminoisoxazolo[5,4-d]pyrimidin-3-yl)phenyl)-3-m-tolylurea 355042 9-hydroxy-4-methyl-5-phenylpyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355043 9-hydroxy-4,5-diphenylpyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355046 2-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)-N-m-tolyl-4,5-dihydrothieno[2,3-c]pyridine-6(7H)-carboxamide 355047 1-(3,5-dimethylphenyl)-3-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)urea 355054 4-(4-fluoro-phenyl)-8-[1-(4-fluoro-phenyl)-cyclohexyl]-2,8-diaza-spiro[4.5]decan-1-one 355064 2-(3-(8-fluoroquinolin-4-yl)-2,5-dimethyl-1H-indol-1-yl)acetic acid 355065 2-(3-(8-methoxyquinolin-4-yl)-2,5-dimethyl-1H-indol-1-yl)acetic acid 355066 1-(4-(4-aminoisothiazolo[5,4-d]pyrimidin-3-yl)phenyl)-3-(3-(trifluoromethyl)phenyl)urea 355067 1-(4-(4-aminoisoxazolo[5,4-d]pyrimidin-3-yl)phenyl)-3-(3-(trifluoromethyl)phenyl)urea 355069 M3S 355074 9-hydroxy-5-phenylpyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355076 N-((4-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)benzenesulfonamide 355077 1-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-o-tolylurea 355088 rac-4-(4-fluoro-phenyl)-8-(1-o-tolyl-cyclohexyl)-2,8-diaza-spiro[4.5]decan-1-one 355089 2-(2,5-dimethyl-3-(8-(methylsulfonyl)quinolin-4-yl)-1H-indol-1-yl)acetic acid 355090 2-(3-(8-cyanoquinolin-4-yl)-2,5-dimethyl-1H-indol-1-yl)acetic acid 355091 1-(4-((4-aminoisothiazolo[5,4-d]pyrimidin-3-yl)methyl)phenyl)-3-m-tolylurea 355092 1-(4-((4-aminoisothiazolo[5,4-d]pyrimidin-3-yl)methyl)phenyl)-3-(3-(trifluoromethyl)phenyl)urea 355093 8-[2-(4-fluoro-phenyl)-2-hydroxy-cyclohexyl]-4-phenyl-2,8-diaza-spiro[4.5]decan-1-one 355102 1-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-p-tolylurea 355113 4-(4-fluoro-phenyl)-8-(1-m-tolyl-cyclohexyl)-2,8-diaza-spiro[4.5]decan-1-one 355117 1-(5-(4-aminoisoxazolo[5,4-d]pyrimidin-3-yl)furan-2-yl)-3-m-tolylurea 355118 1-(5-(4-aminoisoxazolo[5,4-d]pyrimidin-3-yl)furan-2-yl)-3-(3-(trifluoromethyl)phenyl)urea 355122 9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355126 phenyl (5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methylcarbamate 355145 8-(1-phenyl-cyclohexyl)-4-propyl-2,8-diaza-spiro[4.5]decan-1-one 355146 4-phenyl-8-(2-phenyl-cyclohexyl)-2,8-diaza-spiro[4.5]decan-1-one 355148 1-(4-(4-aminoisoxazolo[5,4-d]pyrimidin-3-yl)phenyl)-3-(3-ethylphenyl)urea 355150 9-hydroxy-4-iodopyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355151 8-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355163 DC6S 355165 8-[1-(3-fluoro-phenyl)-cyclohexyl]-4-phenyl-2,8-diaza-spiro[4.5]decan-1-one 355170 2-(1-(7-chloroquinolin-4-yl)-5-methoxy-2-methyl-1H-indol-3-yl)acetic acid 355171 2-(3-(7-chloroquinolin-4-yl)-5-methoxy-2-methyl-1H-indol-1-yl)acetic acid 355176 1-(4-(4-aminoisoxazolo[5,4-d]pyrimidin-3-yl)phenyl)-3-(2-fluoro-5-(trifluoromethyl)phenyl)urea 355178 1-phenyl-8-(1-phenyl-cyclohexyl)-1,3,8-triaza-spiro[4.5]decan-4-one 355179 9-hydroxy-4-phenyl-1H-benzofuro[3,2-e]isoindole-1,3(2H)-dione 355180 4-(2-chlorophenyl)-9-hydroxy-6-pentylpyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355181 5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)-7-(neopentylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one 355182 5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)-7-(6,7-dihydro-1H-pyrazolo[4,3-c]pyridin-5(4H)-yl)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one 355202 2-(3-(7-chloroquinolin-4-yl)-2,6-dimethyl-1H-indol-1-yl)acetic acid 355203 2-(3-(7-chloroquinolin-4-yl)-2,5-dimethyl-1H-indol-1-yl)acetic acid 355205 3-(4-aminophenyl)isothiazolo[5,4-d]pyrimidin-4-amine 355206 1-(4-(4-aminoisothiazolo[5,4-d]pyrimidin-3-yl)phenyl)-3-m-tolylurea 355211 (R)-4-phenyl-8-((1R,2R)-2-phenyl-cyclohexyl)-2,8-diaza-spiro[4.5]decan-1-one 355212 (R)-4-phenyl-8-((1S,2S)-2-phenyl-cyclohexyl)-2,8-diaza-spiro[4.5]decan-1-one 355217 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355221 5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)-7-hydroxy-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one 355222 5-(2,4-dichlorophenyl)-1-(2,6-dichlorophenyl)-7-(2-methoxyethylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one 355240 2-(2,5-dimethyl-3-(quinolin-4-yl)-1H-indol-1-yl)acetic acid 355241 2-(2,5-dimethyl-3-(2-methylquinolin-4-yl)-1H-indol-1-yl)acetic acid 355242 3-(4-(5,7-dimethylbenzo[d]oxazol-2-ylamino)phenyl)isothiazolo[5,4-d]pyrimidin-4-amine 355253 5-(2,4-dichlorophenyl)-1-(2,6-dichlorophenyl)-7-(2-(dimethylamino)ethylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one 355254 5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)-7-(2-(dimethylamino)ethoxy)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one 355274 2-(2,5-dimethyl-3-(6-(trifluoromethyl)quinolin-4-yl)-1H-indol-1-yl)acetic acid 355278 1-(4-(4-aminoisothiazolo[5,4-d]pyrimidin-3-yl)phenyl)-3-(2-fluoro-5-(trifluoromethyl)phenyl)urea 355282 DM6S 355283 DM3A6S 355309 2-(2-methyl-1-(pyrimidin-4-yl)-1H-indol-3-yl)acetic acid 355312 1-(4-(4-aminoisothiazolo[5,4-d]pyrimidin-3-yl)phenyl)-3-(2-fluoro-5-methylphenyl)urea 355316 DM3B6S 355317 MM3A6S 355318 5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)-7-(methylthio)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one 355319 5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)-7-(methylsulfonyl)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one 355327 4-(2-chloro-5-hydroxy-phenyl)-8-[4-(4-methyl-piperazin-1-yl)-phenylamino]-1,2-dihydro-3a,7,9,9b-tetraaza-cyclopenta[a]naphthalen-3-one 355336 8-[1-(4-chloro-phenyl)-cyclohexyl]-4-phenyl-2,8-diaza-spiro[4.5]decan-1-one 355339 rac-4-(4-fluoro-phenyl)-8-[1-(3-fluoro-phenyl)-cyclohexyl]-2,8-diaza-spiro[4.5]decan-1-one 355343 1-phenyl-8-(2-phenyl-cyclohexyl)-1,3,8-triaza-spiro[4.5]decan-4-one 355344 8-(2-hydroxy-2-phenyl-cyclohexyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 355348 MM3B6S 355349 C6S 355350 7-amino-5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one 355351 5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one 355360 1-(3,5-dichlorophenyl)-3-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)urea 355363 4-phenyl-8-(1-p-tolyl-cyclohexyl)-2,8-diaza-spiro[4.5]decan-1-one 355383 1-(4-(4-aminoisothiazolo[5,4-d]pyrimidin-3-yl)phenyl)-3-(3-ethylphenyl)urea 355386 M6S 355388 (S)-4-(4-fluoro-phenyl)-8-[(1S,2S)-2-(4-fluoro-phenyl)-cyclohexyl]-2,8-diaza-spiro[4.5]decan-1-one 355389 5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)-7-(dimethylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one 355390 5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)-7-(isopropylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one 355391 9-hydroxy-1-methoxy-4-phenyl-1,2-dihydropyrrolo[3,4-c]carbazol-3(6H)-one 355392 9-hydroxy-4-phenyl-1,2-dihydropyrrolo[3,4-c]carbazol-3(6H)-one 355411 1-(4-(4-aminoisothiazolo[5,4-d]pyrimidin-3-yl)phenyl)-3-(3-chlorophenyl)urea 355414 M3A6S 355415 M3Pr6S 355417 (R)-4-(4-fluoro-phenyl)-8-[(1R,2R)-2-(4-fluoro-phenyl)-cyclohexyl]-2,8-diaza-spiro[4.5]decan-1-one 355421 3,9-dihydroxy-4-phenyl-2,3-dihydropyrrolo[3,4-c]carbazol-1(6H)-one 355426 1-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-(2-(trifluoromethyl)phenyl)urea 355427 1-methyl-3-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-1-m-tolylurea 355429 4-phenyl-8-(1-phenyl-cyclohexyl)-2,8-diaza-spiro[4.5]decan-1-one 355435 3-phenyl-1,4-dihydroindeno[1,2-c]pyrazole 355436 5-((4-methylpiperazin-1-yl)methyl)-3-phenyl-1,4-dihydroindeno[1,2-c]pyrazole 355446 M3IBu6S 355447 M3P6S 355448 (S)-4-(4-fluoro-phenyl)-8-[(1R,2R)-2-(4-fluoro-phenyl)-cyclohexyl]-2,8-diaza-spiro[4.5]decan-1-one 355452 9-hydroxy-4-phenyl-1H-furo[3,4-c]carbazole-1,3-(6H)-dione 355453 2-amino-9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355454 (5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl m-tolylcarbamate 355455 1-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-(3-(trifluoromethyl)phenyl)urea 355456 1,3-dimethyl-1-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-m-tolylurea 355461 6-((4-methylpiperazin-1-yl)methyl)-3-phenyl-1,4-dihydroindeno[1,2-c]pyrazole 355462 7-((4-methylpiperazin-1-yl)methyl)-3-phenyl-1,4-dihydroindeno[1,2-c]pyrazole 355466 rac-8-[1-(4-fluoro-phenyl)-cyclohexyl]-4-propyl-2,8-diaza-spiro[4.5]decan-1-one 355468 M3B6S 355473 4-(2-chlorophenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355474 4-(2-chlorophenyl)-9-methoxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355476 1-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-(4-(trifluoromethyl)phenyl)urea 355477 1-methyl-1-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-o-tolylurea 355494 2-(2,5-dimethyl-3-(7-(trifluoromethyl)quinolin-4-yl)-1H-indol-1-yl)acetic acid 355495 2-(2,5-dimethyl-3-(8-(trifluoromethyl)quinolin-4-yl)-1H-indol-1-yl)acetic acid 355499 NalBzOH 355504 9-Hydroxy-4-phenyl-6-thia-2-aza-cyclopenta[c]fluorene-1,3-dione 355505 9-hydroxy-6-methyl-4-phenylpyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355507 (Z)-1-(4-chlorophenyl)-2-hydroxy-3-(4-pyridin-2-ylpiperazin-1-yl)propanon-1-one O-methyloxime 355512 5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)-7-hydroxy-3,4-dihydroquinazolin-2(1H)-one 355513 6-(4-(2,4-difluorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 355518 9-hydroxy-4-m-tolylpyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355520 4-(4-chlorophenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355524 6-(4-(2,4-difluorophenyl)oxazol-5-yl)-3-(1-methylcyclopropyl)-[1,2,4]triazolo[4,3-a]pyridine 355525 3-cyclobutyl-6-(4-(2,4-difluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355526 9-hydroxy-4-(thiophen-2-yl)pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355527 9-hydroxy-4-(thiophen-3-yl)pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355531 (Z)-1-(3,5-difluorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)-propan-1-one O-methyloxime 355543 1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-(1-isopropylpiperidin-4-yl)-3,4-dihydroquinazolin-2(1H)-one 355550 9-hydroxy-4-(3-(hydroxymethyl)phenyl)pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355551 4-(3-(aminomethyl)phenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355556 6-(4-(2,4-difluorophenyl)oxazol-5-yl)-3-(1-methylcyclobutyl)-[1,2,4]triazolo[4,3-a]pyridine 355557 3-tert-butyl-6-(4-(2,4-difluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355558 9-hydroxy-4-(1H-pyrrol-2-yl)pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355559 9-hydroxy-4-(1H-pyrrol-3-yl)pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355566 (Z)-1-(4-Fluorophenyl)-2-(4-pyridin-2-yl)ethanone O-Methyloxime 355572 5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)-7-(quinuclidin-3-ylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one 355573 5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)-7-(8-methyl-8-aza-bicyclo[3.2.1]octan-3-ylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one 355574 3-isopropyl-6-(4-phenyloxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355575 3-isopropyl-6-(4-m-tolyloxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355580 4-(2-ethoxyphenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355581 9-hydroxy-4-(2-(methylthio)phenyl)pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355582 3-(9-hydroxy-1,3-dioxo-1,2,3,6-tetrahydropyrrolo[3,4-c]carbazol-4-yl)benzonitrile 355588 6-(4-(4-fluorophenyl)oxazol-5-yl)-3-phenyl-[1,2,4]triazolo[4,3-a]pyridine 355589 2-(6-(4-(2,5-difluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl)propan-2-ol 355590 3-cyclopropyl-6-(4-(2,5-difluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355591 9-hydroxy-4-(pyrrolidin-3-yl)pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355592 9-hydroxy-4-(pyridin-4-yl)pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355603 5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)-7-(4-(2-(dimethylamino)ethyl)piperazin-1-yl)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one 355604 5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)-7-(1-isopropylpiperidin-4-ylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one 355605 5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)-7-(2,2,6,6-tetramethylpiperidin-4-ylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one 355611 9-hydroxy-4-(2-(methylsulfinyl)phenyl)pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355612 9-hydroxy-4-(2-nitrophenyl)pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355617 3-cyclobutyl-6-(4-(4-fluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355618 3-cyclopropyl-6-(4-(4-fluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355619 6-(4-(4-fluorophenyl)oxazol-5-yl)-3-(2-methoxyphenyl)-[1,2,4]triazolo[4,3-a]pyridine 355620 3-(2-ethoxyphenyl)-6-(4-(4-fluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355621 6-(4-(2,5-difluorophenyl)oxazol-5-yl)-3-(1-methylcyclopropyl)-[1,2,4]triazolo[4,3-a]pyridine 355622 3-cyclobutyl-6-(4-(2,5-difluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355624 9-hydroxy-4-(pyridin-3-yl)pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355626 (E)-1-(3-chloro-4-fluorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime 355632 4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S)-1-{[(2S)-1-amino-3-(4-hydroxyphenyl)propan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}methyl)pyrrolidin-1-yl]-3-phenylpropan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 355637 3-hydroxyl-4-palmitoyloxylbutane 1,3-cyclic phosphonothioate 355638 1-fluoro-(3S)-hydroxyl-4-oleoyloxylbutane 1,3-cyclic phosphonate 355639 5-(2,4-dichlorophenyl)-1-(2,6-dichlorophenyl)-7-(4-(2-(dimethylamino)ethyl)piperazin-1-yl)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one 355640 7-amino-5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)-3,4-dihydroquinazolin-2(1H)-one 355650 3-(difluoromethyl)-6-(4-phenyloxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355651 6-(4-phenyloxazol-5-yl)-3-(2,2,2-trifluoroethyl)-[1,2,4]triazolo[4,3-a]pyridine 355652 6-(4-(4-fluorophenyl)oxazol-5-yl)-3-isobutyl-[1,2,4]triazolo[4,3-a]pyridine 355653 6-(4-(4-fluorophenyl)oxazol-5-yl)-N-isopropyl-[1,2,4]triazolo[4,3-a]pyridin-3-amine 355654 3-tert-butyl-6-(4-(4-fluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355655 6-(4-(4-fluorophenyl)oxazol-5-yl)-3-morpholino-[1,2,4]triazolo[4,3-a]pyridine 355664 (E)-1-(3,4-dichlorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)-propan-1-one O-methyloxime 355672 5-(2,4-dichlorophenyl)-1-(2,6-dichlorophenyl)-7-(4-isopropylpiperazin-1-yl)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one 355673 5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)-7-(morpholinoamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one 355680 9-hydroxy-4-(2-hydroxyphenyl)pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355686 3-(isoxazol-5-yl)-6-(4-phenyloxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355687 6-(4-(4-fluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355688 3-ethyl-6-(4-(4-fluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355689 6-(4-(4-fluorophenyl)oxazol-5-yl)-N-propyl-[1,2,4]triazolo[4,3-a]pyridin-3-amine 355690 N-ethyl-6-(4-(4-fluorophenyl)oxazol-5-yl)-N-methyl-[1,2,4]triazolo[4,3-a]pyridin-3-amine 355691 3-benzyl-6-(4-(4-fluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355692 3-cyclopropyl-6-(4-(2,4-difluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355693 3-(thiophen-2-yl)-1,4-dihydroindeno[1,2-c]pyrazole 355705 (Z)-4-[1-methoxyimino-3-(4-pyridin-2-ylpiperazin-1-yl)propyl]benzonitrile 355725 (E)-1-(4-chlorophenyl)-3-(3',4',5',6'-tetrahydro-2'H-[2,4']bipyridinyl-1'-yl)propan-1-one O-methyloxime 355730 5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)-7-morpholino-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one 355731 5-(2,4-dichlorophenyl)-1-(2,6-dichlorophenyl)-7-((2S,6R)-2,6-dimethylmorpholino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one 355738 9-hydroxy-4-(2-methoxyphenyl)pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355741 6-(4-(4-chloro-2,5-difluorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 355742 6-(4-(2-chloro-4,5-difluorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 355743 6-(4-(4-fluorophenyl)oxazol-5-yl)-N,N-dimethyl-[1,2,4]triazolo[4,3-a]pyridin-3-amine 355744 N-ethyl-6-(4-(4-fluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-amine 355745 6-(4-(4-fluorophenyl)oxazol-5-yl)-3-isopropoxy-[1,2,4]triazolo[4,3-a]pyridine 355746 6-(4-(4-fluorophenyl)oxazol-5-yl)-3-(1-methylcyclobutyl)-[1,2,4]triazolo[4,3-a]pyridine 355755 (E)-1-(4-fluorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime 355756 (Z)-1-(4-fluorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime 355759 (Z)-1-(4-chlorophenyl)-3-(3',4',5',6'-tetrahydro-2'H-[2,4']bipyridinyl-1'-yl)propan-1-one O-methyloxime 355771 2-(9-hydroxy-1,3-dioxo-1,2,3,6-tetrahydropyrrolo[3,4-c]carbazol-4-yl)benzamide 355774 3-isopropyl-6-(4-(3,4,5-trifluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355775 3-isopropyl-6-(4-(2,4,5-trifluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355776 6-(4-(3-bromo-4-fluorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 355777 3-ethyl-6-(4-phenyloxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355778 3-cyclopropyl-6-(4-phenyloxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355779 3-ethoxy-6-(4-(4-fluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355780 6-((4-methylpiperazin-1-yl)methyl)-3-(thiazol-5-yl)-1,4-dihydroindeno[1,2-c]pyrazole 355781 7-(2-(4-methylpiperazin-1-yl)ethyl)-3-(thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole 355782 N-ethyl-N-((3-(thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazol-7-yl)methyl)ethanamine 355787 4-(2,5-dimethylphenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355788 4-(2,6-dimethylphenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355789 6-(4-(4-fluorophenyl)oxazol-5-yl)-3-(pyrrolidin-1-yl)-[1,2,4]triazolo[4,3-a]pyridine 355790 6-(3-(2,5-difluorophenyl)-1H-pyrazol-4-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 355791 (E)-1-(4-chlorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime 355799 1-(4-chlorophenyl)-2-methyl-3-(4-pyridin-2-ylpiperazin-1-yl)-propanon-1-one O-methyloxime 355804 9-hydroxy-4-(2-(hydroxymethyl)phenyl)pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355809 3-isopropyl-6-(4-(2,4,6-trifluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355810 3-isopropyl-6-(4-(2,3,5-trifluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355811 3-cyclobutyl-6-(4-phenyloxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355812 N-ethyl-6-(4-phenyloxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-amine 355813 N-ethyl-N-methyl-6-(4-phenyloxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-amine 355814 6-((4-methylpiperazin-1-yl)methyl)-3-(thiazol-4-yl)-1,4-dihydroindeno[1,2-c]pyrazole 355815 6-((4-methylpiperazin-1-yl)methyl)-3-(thiazol-2-yl)-1,4-dihydroindeno[1,2-c]pyrazole 355816 7-((4-isopropylpiperazin-1-yl)methyl)-3-(thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole 355817 (4-methylpiperazin-1-yl)(3-(thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazol-7-yl)methanone 355820 4-(2-chloro-5-hydroxyphenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355821 4-(4-amino-2-methoxyphenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355822 4-(5-amino-2-methoxyphenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355823 6-(5-(2,5-difluorophenyl)isoxazol-4-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 355824 6-(4-(2,5-difluorophenyl)-1H-imidazol-5-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 355836 2-(9-hydroxy-1,3-dioxo-1,2,3,6-tetrahydropyrrolo[3,4-c]carbazol-4-yl)benzonitrile 355837 4-(biphenyl-2-yl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355839 6-(4-(2,5-difluorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 355840 6-(4-(2,6-difluorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 355841 3-isopropyl-6-(4-(2,3,4-trifluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355842 6-(4-(3,4-dichlorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 355845 6-((4-methylpiperazin-1-yl)methyl)-3-(5-methylthiophen-2-yl)-1,4-dihydroindeno[1,2-c]pyrazole 355846 6-((4-methylpiperazin-1-yl)methyl)-3-(4-methylthiophen-2-yl)-1,4-dihydroindeno[1,2-c]pyrazole 355847 4-((3-(thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazol-7-yl)methyl)piperazine-1-carbaldehyde 355848 7-((1H-1,2,3-triazol-1-yl)methyl)-3-(thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole 355849 4-(5-amino-2-chlorophenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355850 4-(2,6-dichlorophenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355851 4-(2,6-dimethoxyphenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355852 4-(2-fluoro-6-methoxyphenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355857 (E)-1-(3,5-difluorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)-propan-1-one O-methyloxime 355868 4-(2-chlorophenyl)-9-hydroxy-6-methylpyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355873 6-(4-(3,4-difluorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 355874 6-(4-(3-chloro-4-fluorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 355875 6-(4-(2,4-dichlorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 355876 6-(4-(2,3-dichlorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 355878 6-((4-methylpiperazin-1-yl)methyl)-3-(thiophen-2-yl)-1,4-dihydroindeno[1,2-c]pyrazole 355881 7-((1H-1,2,4-triazol-1-yl)methyl)-3-(thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole 355882 4-(2-chloro-6-hydroxyphenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355883 4-(2-chloro-6-methoxyphenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355884 4-(2,6-dichloro-3-hydroxyphenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355899 4-(2-chlorophenyl)-9-hydroxy-1H-benzofuro[3,2-e]isoindole-1,3(2H)-dione 355900 4-(2-fluorophenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355901 4-(2-acetylphenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355905 6-(4-(4-chloro-2-fluorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 355906 6-(4-(5-chloro-2-fluorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 355907 3-(3-((4-methylpiperazin-1-yl)methyl)phenyl)-1,4-dihydroindeno[1,2-c]pyrazole 355908 3-(4-((4-methylpiperazin-1-yl)methyl)phenyl)-1,4-dihydroindeno[1,2-c]pyrazole 355910 6-((4-methylpiperazin-1-yl)methyl)-3-(thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole 355911 6-(4-methylpiperazin-1-yl)-3-(thiophen-2-yl)-1,4-dihydroindeno[1,2-c]pyrazole 355912 9-hydroxy-4-p-tolylpyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355913 9-hydroxy-4-[4-(methanesulfonyl)phenyl]pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355914 4-(4-aminophenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355915 4-(4-amino-2-bromophenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355916 4-(2,6-dibromophenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355919 9-hydroxy-4-(piperidin-3-yl)pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355920 4-(2-chlorophenyl)-6-ethyl-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355932 4-(2-bromophenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355933 9-hydroxy-4-(2-iodophenyl)pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355937 6-(4-(2-chloro-4-fluorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 355938 6-(4-(4-chloro-3-fluorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 355939 4-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenol 355940 6-((4-methylpiperazin-1-yl)methyl)-3-(pyridin-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole 355941 4-(3-acetylphenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355943 9-hydroxy-4-(4-(hydroxymethyl)phenyl)pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355944 4-(2,3-dichlorophenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355945 4-(2-chloro-3-hydroxyphenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355946 4-(2,3-dimethylphenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355948 6-(4-(2,5-difluorophenyl)oxazol-5-yl)-3-(1-methylcyclobutyl)-[1,2,4]triazolo[4,3-a]pyridine 355949 3-tert-butyl-6-(4-(2,5-difluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355950 4-(2-chlorophenyl)-9-hydroxy-6-propylpyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355951 4-(2-chlorophenyl)-9-hydroxy-6-isopropylpyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355954 (Z)-1-(4-chloro-3-methylphenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime 355961 9-hydroxy-4-o-tolylpyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355962 4-(2-ethylphenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355965 6-(4-(3-fluorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 355966 6-(4-(4-fluoro-3-methylphenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 355971 4-(biphenyl-3-yl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355972 9-hydroxy-4-(3-hydroxyphenyl)pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355973 4-(9-hydroxy-1,3-dioxo-1,2,3,6-tetrahydropyrrolo[3,4-c]carbazol-4-yl)benzonitrile 355974 4-(4-acetylphenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355975 4-(3-amino-2-chlorophenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355976 4-(2-chloro-4-hydroxyphenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355978 3-cyclopropyl-6-(4-(2,4,5-trifluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355979 3-(1-methylcyclopropyl)-6-(4-(2,4,5-trifluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 355980 6-butyl-4-(2-chlorophenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355981 4-(2-chlorophenyl)-9-hydroxy-6-isopentylpyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355984 (E)-1-(3,4-dimethylphenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)-propan-1-one O-methyloxime 355992 9-hydroxy-4-(2-(trifluoromethyl)phenyl)pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 355996 6-(4-(2-fluoro-5-methylphenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 355997 6-(4-(4-chlorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 356002 4-(2-aminophenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 356003 9-hydroxy-4-(3-methoxyphenyl)pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 356004 9-hydroxy-4-(3-nitrophenyl)pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 356005 9-hydroxy-4-(4-hydroxyphenyl)pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 356006 9-hydroxy-4-(4-methoxyphenyl)pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 356007 4-(4-amino-2-chlorophenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 356008 4-(2,5-dichlorophenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 356009 3-cyclobutyl-6-(4-(2,4,5-trifluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 356010 3-(1-methylcyclobutyl)-6-(4-(2,4,5-trifluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 356021 1-pyridin-3-yl-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime 356022 (E)-1-(4-chlorophenyl)-3-(2-methyl-4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime 356028 4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S,3R)-1-{[(2S)-1-amino-4-(methylsulfanyl)butan-2-yl]amino}-3-hydroxybutan-2-yl]amino}methyl)pyrrolidin-1-yl]-3-phenylpropan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356029 4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S,3R)-1-[(2S)-2-(aminomethyl)pyrrolidin-1-yl]-3-hydroxybutan-2-yl]amino}methyl)pyrrolidin-1-yl]-3-phenylpropan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356030 4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S)-1-[(2S)-2-(aminomethyl)pyrrolidin-1-yl]-3-(4-hydroxyphenyl)propan-2-yl]amino}methyl)pyrrolidin-1-yl]-3-phenylpropan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356031 4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S)-1-{[(2R)-1-amino-3-hydroxypropan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}methyl)pyrrolidin-1-yl]-3-phenylpropan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356037 4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S,3R)-1-{[(2S)-1-amino-3-hydroxypropan-2-yl]amino}-3-hydroxybutan-2-yl]amino}methyl)pyrrolidin-1-yl]-3-phenylpropan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356038 4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S,3R)-1-{[(2S)-1-amino-3-(4-hydroxyphenyl)propan-2-yl]amino}-3-hydroxybutan-2-yl]amino}methyl)pyrrolidin-1-yl]-3-phenylpropan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356039 3-hydroxyl-4-oleoyloxylbutane 1,3-cyclic phosphonothioate 356040 (E)-1-(4-chlorophenyl)-2-hydroxy-3-(4-pyridin-2-ylpiperazin-1-yl)propanon-1-one O-methyloxime 356041 1-(4-chlorophenyl)-2-(methoxyaminomethyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propanon-1-one O-methyloxime 356045 6-(4-(3-chlorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 356046 6-(4-(2-chlorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]triazolo[4,3-a]pyridine 356050 4-(3-fluorophenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 356051 4-(3-chlorophenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 356052 4-(3-aminophenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 356053 4-(4-fluorophenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 356054 9-hydroxy-4-(4-(methylthio)phenyl)pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 356057 3-tert-butyl-6-(4-(2,4,5-trifluorophenyl)oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine 356062 4-(2,6-dichloro-4-hydroxyphenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione 356077 [1-phenyl-3-(4-pyridin-2-ylpiperazin-1-yl)propylideneaminooxy]-acetonitrile 356099 4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S)-1-{[(2S)-1-amino-3-(4-hydroxyphenyl)propan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}methyl)pyrrolidin-1-yl]-3-(4-hydroxyphenyl)propan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356101 4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S)-1-{[(2R)-1-amino-3-hydroxypropan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}methyl)pyrrolidin-1-yl]-3-(4-hydroxyphenyl)propan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356114 (E)-1-phenyl-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime 356131 4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S)-1-{[(2S)-1-amino-3-phenylpropan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}methyl)pyrrolidin-1-yl]-3-phenylpropan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356132 4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S,3R)-1-{[(2S)-1-amino-3-hydroxypropan-2-yl]amino}-3-hydroxybutan-2-yl]amino}methyl)pyrrolidin-1-yl]-3-(4-hydroxyphenyl)propan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356133 4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S)-1-{[(2S)-1-amino-4-(methylsulfanyl)butan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}methyl)pyrrolidin-1-yl]-3-phenylpropan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356134 4-[(2S)-2-amino-3-{ethyl[(2S)-1-{ethyl[(2S)-1-[(2S)-2-[(ethylamino)methyl]pyrrolidin-1-yl]-3-phenylpropan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}propyl]phenol 356135 4-[(2S)-2-amino-3-{benzyl[(2S)-1-{benzyl[(2S)-1-[(2S)-2-[(benzylamino)methyl]pyrrolidin-1-yl]-3-phenylpropan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}propyl]phenol 356144 4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S,3R)-1-{[(2S)-1-amino-3-phenylpropan-2-yl]amino}-3-hydroxybutan-2-yl]amino}methyl)pyrrolidin-1-yl]-3-phenylpropan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356153 (E)-1-phenyl-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-ethyloxime 356161 (E)-1-(3-fluorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime 356171 4-[(2S)-3-{[(2S)-1-{[(2S)-1-{[(2S)-1-amino-3-(4-hydroxyphenyl)propan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356172 4-[(2S)-3-{[(2S)-1-{[(2S)-1-amino-3-phenylpropan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356173 4-[(2S,5S,8S,11S,14S)-1-amino-14-(ethylamino)-2,5,8,11-tetrakis[(4-hydroxyphenyl)methyl]-3,6,9,12-tetraazapentadecan-15-yl]phenol 356174 4-[(2S)-2-amino-3-{[(2S)-1-(4-hydroxyphenyl)-3-{methyl[(2S)-1-[(2S)-2-[(methylamino)methyl]pyrrolidin-1-yl]-3-phenylpropan-2-yl]amino}propan-2-yl](methyl)amino}propyl]phenol 356176 4-[(2S)-2-amino-3-{[(2S)-1-(4-hydroxyphenyl)-3-[(naphthalen-2-ylmethyl)[(2S)-1-[(2S)-2-{[(naphthalen-2-ylmethyl)amino]methyl}pyrrolidin-1-yl]-3-phenylpropan-2-yl]amino]propan-2-yl](naphthalen-2-ylmethyl)amino}propyl]phenol 356179 4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S,3R)-1-[(2S)-2-(aminomethyl)pyrrolidin-1-yl]-3-hydroxybutan-2-yl]amino}methyl)pyrrolidin-1-yl]-3-(4-hydroxyphenyl)propan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356180 4-[(2S,5S,8S,11S,14S)-2-{[(2S)-2-(aminomethyl)pyrrolidin-1-yl]methyl}-5,8-dibenzyl-14-(ethylamino)-1-(4-hydroxyphenyl)-11-[(4-hydroxyphenyl)methyl]-3,6,9,12-tetraazapentadecan-15-yl]phenol 356181 4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S,3R)-1-{[(2S)-1-amino-3-(4-hydroxyphenyl)propan-2-yl]amino}-3-hydroxybutan-2-yl]amino}methyl)pyrrolidin-1-yl]-3-(4-hydroxyphenyl)propan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356182 4-[(2S)-2-(dimethylamino)-3-{[(2S)-1-(4-hydroxyphenyl)-3-{methyl[(2S)-1-(methylamino)-3-phenylpropan-2-yl]amino}propan-2-yl](methyl)amino}propyl]phenol 356183 4-[(2R)-2-(dimethylamino)-3-{[(2S)-1-(4-hydroxyphenyl)-3-{methyl[(2S)-1-(methylamino)-3-phenylpropan-2-yl]amino}propan-2-yl](methyl)amino}propyl]phenol 356207 (Z)-1-(3-fluorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime 356208 (E)-1-(3-chlorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime 356209 2,6-dimethylphenyl 2-((3,5-bis(methyloxy)-4-((2-(4-methyl-1-piperazinyl)ethyl)oxy)phenyl)amino)-4-pyrimidinyl(2,4-bis(methyloxy)phenyl)carbamate 356210 2,6-dimethylphenyl 2-((3,5-bis(methyloxy)-4-((2-(4-morpholinyl)ethyl)oxy)phenyl)amino)-4-pyrimidinyl(2,4-bis(methyloxy)-phenyl)carbamate 356211 2,6-dimethylphenyl-2,4-bis(methyloxy)phenyl(2-((4-((3-(1-piperidinyl)propyl)oxy)phenyl)amino)-4-pyrimidinyl)carbamate 356217 (4S,7S,10S,13S,16S,17R)-16-{[(2S)-2-(aminomethyl)pyrrolidin-1-yl]methyl}-13-benzyl-4,7,10-tris[(4-hydroxyphenyl)methyl]-3,6,9,12,15-pentaazaoctadecan-17-ol 356218 (2S,5S,8S,11S,14S,17S)-2-(aminomethyl)-8-benzyl-5-[(1R)-1-hydroxyethyl]-11,14,17-tris[(4-hydroxyphenyl)methyl]-3,6,9,12,15,18-hexaazaicosan-1-ol 356219 4-[(2S,5S,8S,11S,14S,17S)-1-amino-2,8,11-tribenzyl-17-(ethylamino)-5,14-bis[(4-hydroxyphenyl)methyl]-3,6,9,12,15-pentaazaoctadecan-18-yl]phenol 356222 4-[(2S)-2-amino-3-{[(2S)-1-{[(2S)-1-[(2S)-2-(aminomethyl)pyrrolidin-1-yl]-3-phenylpropan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}propyl]phenol 356250 (E)-3-(4-pyridin-2-ylpiperazin-1-yl)-1-(m-tolyl)propan-1-one O-methyloxime 356251 2,6-dimethylphenyl 2,4-bis(methyloxy)phenyl(2-((3-(methyloxy)-4-((3-(4-methyl-1-piperazinyl)propyl)oxy)phenyl)amino)-4-pyrimidinyl)-carbamate 356252 2,6-dimethylphenyl 2,4-bis(methyloxy)phenyl(2-((3,5-bis(methyloxy)-4-((3-(4-methyl-1-piperazinyl)propyl)-oxy)phenyl)amino)-4-pyrimidinyl(2,4-bis-(methyloxy)phenyl)carbamate 356253 2,6-dimethylphenyl 2,4-bis(methyloxy)phenyl(2-((3-fluoro-4-((3-(4-methyl-1-piperazinyl)propyl)-oxy)phenyl)amino)-4-pyrimidinyl)carbamate 356254 2,6-dimethylphenyl 2,4-bis(methyloxy)phenyl(2-((3-fluoro-4-((3-(1-piperidinyl)propyl)-oxy)phenyl)amino)-4-pyrimidinyl)carbamate 356258 4-[(2S)-3-{[(2S)-1-(benzylamino)-3-(4-hydroxyphenyl)propan-2-yl](methyl)amino}-2-(dimethylamino)propyl]phenol 356259 4-[(2S)-2-amino-3-{benzyl[(2S)-1-(4-hydroxyphenyl)-3-(methylamino)propan-2-yl]amino}propyl]phenol 356276 (Z)-3-(4-pyridin-2-ylpiperazin-1-yl)-1-(m-tolyl)propan-1-one O-methyloxime 356284 4-[(2S)-3-{benzyl[(2S)-1-(4-hydroxyphenyl)-3-(methylamino)propan-2-yl]amino}-2-(methylamino)propyl]phenol 356285 4-[(2S)-3-{benzyl[(2S)-1-(4-hydroxyphenyl)-3-(methylamino)propan-2-yl]amino}-2-(dimethylamino)propyl]phenol 356316 4-[(2S,5S,8S,11S,14S,17S)-1-amino-8,11-dibenzyl-17-(ethylamino)-2,5,14-tris[(4-hydroxyphenyl)methyl]-3,6,9,12,15-pentaazaoctadecan-18-yl]phenol 356317 (4S,7S,10S,13S,16S,17R)-16-({[(2S)-1-amino-3-phenylpropan-2-yl]amino}methyl)-10,13-dibenzyl-4,7-bis[(4-hydroxyphenyl)methyl]-3,6,9,12,15-pentaazaoctadecan-17-ol 356320 2,6-dimethylphenyl (2,5-bis(methyloxy)phenyl)methyl(2-((4-(4-methyl-1-piperazinyl)phenyl)amino)-4-pyrimidinyl)carbamate 356321 2,6-dimethylphenyl 2-((4-(4-methyl-1-piperazinyl)phenyl)-amino)-4-pyrimidinyl(2-naphthalenyl)carbamate 356322 2,6-dimethylphenyl-1,1'-biphenyl-4-yl(2-((4-(4-methyl-1-piperazinyl)phenyl)amino)-4-pyrimidinyl)carbamate 356330 (E)-1-phenyl-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one oxime 356352 4-[(2S)-2-amino-3-{[(2S)-1-amino-3-(4-hydroxyphenyl)propan-2-yl]amino}propyl]phenol 356382 (4S,7S,10S,13S,16S,17R)-16-({[(2S)-1-amino-4-(methylsulfanyl)butan-2-yl]amino}methyl)-13-benzyl-4,7,10-tris[(4-hydroxyphenyl)methyl]-3,6,9,12,15-pentaazaoctadecan-17-ol 356383 (4S,7S,10S,13S,16S,17R)-16-({[(2S)-1-amino-3-(4-hydroxyphenyl)propan-2-yl]amino}methyl)-13-benzyl-4,7,10-tris[(4-hydroxyphenyl)methyl]-3,6,9,12,15-pentaazaoctadecan-17-ol 356384 4-[(2S,5S,8S,11S,14S,17S)-1-amino-2,8-dibenzyl-17-(ethylamino)-5,11,14-tris[(4-hydroxyphenyl)methyl]-3,6,9,12,15-pentaazaoctadecan-18-yl]phenol 356389 4-[(2S)-2-amino-3-{[(2S)-1-(4-hydroxyphenyl)-3-{methyl[(2R)-1-(methylamino)-3-phenylpropan-2-yl]amino}propan-2-yl](methyl)amino}propyl]phenol 356390 4-[(2S)-3-{[(2S)-1-amino-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(methylamino)propyl]phenol 356391 4-[(2S)-3-{[(2S)-1-amino-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(dimethylamino)propyl]phenol 356392 2,6-dimethylphenyl-2-((4-(4-methyl-1-piperazinyl)phenyl)amino)-4-pyrimidinyl(phenyl)carbamate 356424 4-[(2S)-2-amino-3-{[(2R)-1-(4-hydroxyphenyl)-3-{methyl[(2S)-1-(methylamino)-3-phenylpropan-2-yl]amino}propan-2-yl](methyl)amino}propyl]phenol 356426 2,6-dimethylphenyl 2-(methyloxy)phenyl(2-((4-(4-methyl-1-piperazinyl)phenyl)amino)-4-pyrimidinyl)carbamate 356450 (E)-1-phenyl-3-(4-thiazol-2-ylpiperazin-1-yl)propanon-1-one O-ethyloxime 356454 4-[(5S,8S,11S,14S,17S,20S)-5-(aminomethyl)-11-benzyl-20-(ethylamino)-8,14,17-tris[(4-hydroxyphenyl)methyl]-2-thia-6,9,12,15,18-pentaazahenicosan-21-yl]phenol 356455 4-[(2S,5S,8S,11S,14S,17S)-1-amino-8-benzyl-17-(ethylamino)-2,5,11,14-tetrakis[(4-hydroxyphenyl)methyl]-3,6,9,12,15-pentaazaoctadecan-18-yl]phenol 356466 4-[(2S)-3-{[(2S)-1-(benzylamino)-3-(4-hydroxyphenyl)propan-2-yl](methyl)amino}-2-(methylamino)propyl]phenol 356468 2,6-dimethylphenyl 4-(methyloxy)phenyl(2-((4-(4-methyl-1-piperazinyl)phenyl)amino)-4-pyrimidinyl)carbamate 356490 4-[(2S)-3-{[(2S)-1-(4-hydroxyphenyl)-3-{methyl[(2S)-1-[(2S)-2-[(methylamino)methyl]pyrrolidin-1-yl]-3-phenylpropan-2-yl]amino}propan-2-yl](methyl)amino}-2-(methylamino)propyl]phenol 356492 4-[(2S)-2-(dimethylamino)-3-{[(2S)-1-(4-hydroxyphenyl)-3-{methyl[(2S)-1-[(2S)-2-[(methylamino)methyl]pyrrolidin-1-yl]-3-phenylpropan-2-yl]amino}propan-2-yl](methyl)amino}propyl]phenol 356514 (E)-3-(4-pyridin-2-ylpiperazin-1-yl)-1-(o-tolyl)propan-1-one O-methyloxime 356518 (4S,7S,10S,13S,16S,17R)-16-({[(2S)-1-amino-4-(methylsulfanyl)butan-2-yl]amino}methyl)-10,13-dibenzyl-4,7-bis[(4-hydroxyphenyl)methyl]-3,6,9,12,15-pentaazaoctadecan-17-ol 356521 2,6-dimethylphenyl 2,4-bis(methyloxy)phenyl(2-((3-fluoro-4-(4-methyl-1-piperazinyl)phenyl)amino)-4-pyrimidinyl)carbamate 356522 4-[(2S)-3-{[(2S)-1-amino-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356523 4-[(2S)-3-{[(2S)-1-{[(2S)-1-amino-3-(4-hydroxyphenyl)propan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356533 Dcp-c[D-Cys-Gly-Phe(pNO2)-D-Cys]NH2 356534 4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S,3R)-1-{[(2S)-1-amino-4-(methylsulfanyl)butan-2-yl]amino}-3-hydroxybutan-2-yl]amino}methyl)pyrrolidin-1-yl]-3-(4-hydroxyphenyl)propan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356537 4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S)-1-{[(2S)-1-amino-4-(methylsulfanyl)butan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}methyl)pyrrolidin-1-yl]-3-(4-hydroxyphenyl)propan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356558 (2S,5S,8S,11S,14S,17S)-2-(aminomethyl)-8-benzyl-5,11,14,17-tetrakis[(4-hydroxyphenyl)methyl]-3,6,9,12,15,18-hexaazaicosan-1-ol 356560 4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S)-1-amino-3-(4-hydroxyphenyl)propan-2-yl]amino}methyl)pyrrolidin-1-yl]-3-phenylpropan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356561 4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-(aminomethyl)pyrrolidin-1-yl]-3-(4-hydroxyphenyl)propan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356574 (2S,5S,8S,11S,14S,17S)-2-(aminomethyl)-8,11-dibenzyl-5-[(1R)-1-hydroxyethyl]-14,17-bis[(4-hydroxyphenyl)methyl]-3,6,9,12,15,18-hexaazaicosan-1-ol 356575 2,6-dimethylphenyl 4-fluoro-2-((1-methylethyl)oxy)phenyl-(2-((4-(4-methyl-1-piperazinyl)phenyl)amino)-4-pyrimidinyl)carbamate 356576 2,6-dimethylphenyl-2,4-bis(methyloxy)phenyl(2-((4-(4-methyl-1-piperazinyl)phenyl)amino)-4-pyrimidinyl)carbamate 356579 2,6-dimethylphenyl 1,1'-biphenyl-3-yl(2-((4-(4-methyl-1-piperazinyl)phenyl)amino)-4-pyrimidinyl)carbamate 356580 2,6-dimethylphenyl 2,4-bis(methyloxy)phenyl(2-((3-(methyloxy)-4-(4-methyl-1-piperazinyl)phenyl)amino)-4-pyrimidinyl)-carbamate 356581 2,6-dimethylphenyl 2-((3,5-bis(methyloxy)-4-(4-methyl-1-piperazinyl)phenyl)amino)-4-pyrimidinyl(2,4-bis(methyloxy)phenyl)-carbamate 356582 Dhp-c[D-Cys-Gly-Phe(pNO2)-D-Cys]NH2 356583 [Dcp1]Dyn A(1-11)-NH2 356599 2,6-dimethylphenyl-2,4-bis(methyloxy)phenyl(2-((4-((2-(dimethylamino)ethyl)-oxy)phenyl)amino)-4-pyrimidinyl)carbamate 356600 2,6-dimethylphenyl 2,4-bis(methyloxy)phenyl(2-((4-((3-(dimethylamino)propyl)oxy)phenyl)amino)-4-pyrimidinyl)carbamate 356601 2,6-dimethylphenyl-2,4-bis(methyloxy)phenyl(2-((3-fluoro-4-((2-(4-methyl-1-piperazinyl)ethyl)oxy)phenyl)amino)-4-pyrimidinyl)carbamate 356611 (2S,5S,8S,11S,14S,17S)-2-(aminomethyl)-8,11-dibenzyl-5,14,17-tris[(4-hydroxyphenyl)methyl]-3,6,9,12,15,18-hexaazaicosan-1-ol 356612 (4S,7S,10S,13S,16S,17R)-16-({[(2S)-1-amino-3-(4-hydroxyphenyl)propan-2-yl]amino}methyl)-10,13-dibenzyl-4,7-bis[(4-hydroxyphenyl)methyl]-3,6,9,12,15-pentaazaoctadecan-17-ol 356613 4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S)-1-[(2S)-2-(aminomethyl)pyrrolidin-1-yl]-3-(4-hydroxyphenyl)propan-2-yl]amino}methyl)pyrrolidin-1-yl]-3-(4-hydroxyphenyl)propan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356614 4-[(2R)-2-(dimethylamino)-3-{[(2R)-1-(4-hydroxyphenyl)-3-{methyl[(2R)-1-(methylamino)-3-phenylpropan-2-yl]amino}propan-2-yl](methyl)amino}propyl]phenol 356615 4-[(2S)-2-(dimethylamino)-3-{[(2R)-1-(4-hydroxyphenyl)-3-{methyl[(2R)-1-(methylamino)-3-phenylpropan-2-yl]amino}propan-2-yl](methyl)amino}propyl]phenol 356616 4-[(2R)-2-(dimethylamino)-3-{[(2S)-1-(4-hydroxyphenyl)-3-{methyl[(2R)-1-(methylamino)-3-phenylpropan-2-yl]amino}propan-2-yl](methyl)amino}propyl]phenol 356619 4-[(2S)-2-amino-3-{[(2S)-1-(benzylamino)-3-(4-hydroxyphenyl)propan-2-yl](methyl)amino}propyl]phenol 356639 4-[(5S,8S,11S,14S,17S,20S)-5-(aminomethyl)-11,14-dibenzyl-20-(ethylamino)-8,17-bis[(4-hydroxyphenyl)methyl]-2-thia-6,9,12,15,18-pentaazahenicosan-21-yl]phenol 356640 4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S,3R)-1-{[(2S)-1-amino-3-phenylpropan-2-yl]amino}-3-hydroxybutan-2-yl]amino}methyl)pyrrolidin-1-yl]-3-(4-hydroxyphenyl)propan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356641 4-[(2S,5S,8S,11S,14S)-2-{[(2S)-2-(aminomethyl)pyrrolidin-1-yl]methyl}-5-benzyl-14-(ethylamino)-1-(4-hydroxyphenyl)-8,11-bis[(4-hydroxyphenyl)methyl]-3,6,9,12-tetraazapentadecan-15-yl]phenol 356647 4-[(2R)-2-(dimethylamino)-3-{[(2R)-1-(4-hydroxyphenyl)-3-{methyl[(2S)-1-(methylamino)-3-phenylpropan-2-yl]amino}propan-2-yl](methyl)amino}propyl]phenol 356648 (4S,7S,10S,13S,16S,17R)-16-{[(2S)-2-(aminomethyl)pyrrolidin-1-yl]methyl}-10,13-dibenzyl-4,7-bis[(4-hydroxyphenyl)methyl]-3,6,9,12,15-pentaazaoctadecan-17-ol 356650 4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S)-1-{[(2S)-1-amino-3-phenylpropan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}methyl)pyrrolidin-1-yl]-3-(4-hydroxyphenyl)propan-2-yl]amino}-3-(4-hydroxyphenyl)propan-2-yl]amino}-2-(ethylamino)propyl]phenol 356686 3-(2,4-dichlorophenyl)-1-(4-(2-((1S)-2-methyl-1-(phenethylamino)butyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)propan-1-one 356687 1-phenyl-5-trifluoromethyl-1H-pyrazole-4-carboxylic acid [8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-amide 356694 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-4-methoxy-benzamide 356695 1-(4-(2-((1S)-1-amino-2-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(4-chlorophenyl)propan-1-one 356696 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(3-methoxyphenyl)propan-1-one 356728 (+/-)-trans-5-((((3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentyl)methyl)(methyl)amino)methyl)-2H-1,2,4-triazol-3(4H)-one 356729 1-(4-(2-((1S)-1-amino-2-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(2-chloro-4-methoxyphenyl)propan-1-one 356730 1-(4-(2-((1S)-1-amino-2-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(2-chloro-3,4-dimethoxyphenyl)propan-1-one 356731 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(4-methoxyphenyl)propan-1-one 356752 4'-trifluoromethyl-biphenyl-4-carboxylic acid {(S)-1-[(R)-3-(cyclobutylmethyl-amino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-methyl-amide 356758 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-butyramide 356759 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-3-cyclopentyl-propionamide 356760 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(2-fluorophenyl)propan-1-one 356761 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(2-chlorophenyl)propan-1-one 356776 3-amino-N-(1-(2-(4-(3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)-5-fluorophenyl)-2-ethoxyethyl)propanamide 356777 4'-trifluoromethyl-biphenyl-4-carboxylic acid methyl-{(S)-1-[(R)-3-(3-phenyl-propylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-amide 356778 4'-trifluoromethyl-biphenyl-4-carboxylic acid ((S)-1-{(R)-3-[2-(4-fluoro-phenoxy)-ethylamino]-pyrrolidine-1-carbonyl}-pyrrolidin-3-yl)-methyl-amide 356780 4'-trifluoromethyl-biphenyl-4-carboxylic acid {(S)-1-[(R)-3-(cyclohexylmethyl-amino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-methyl-amide 356784 biphenyl-4,4'-dicarboxylic acid 4-amide 4'-(methyl-{(S)-1-[(S)-3-(3-phenyl-propylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-amide) 356785 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-3-phenyl-propionamide 356786 3-(3-chloro-4-methoxy-phenyl)-N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-propionamide 356787 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(2-hydroxyphenyl)propan-1-one 356788 N-methyl-N-{(S)-1-[(S)-3-(3-phenyl-propylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-4-pyrimidin-5-yl-benzamide 356804 1-(4-(2-(1-(2-aminoethylamino)-2-(benzyloxy)ethyl)-4-fluorophenyl)piperazin-1-yl)-3-(2,4-dichlorophenyl)propan-1-one 356805 4'-trifluoromethyl-biphenyl-4-carboxylic acid methyl-{(S)-1-[(R)-3-(4-methyl-cyclohexylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-amide 356809 (+/-)-trans-4-(((3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentyl)(methyl)amino)methyl)-1H-imidazol-2(3H)-one 356810 trans-(S)-5-((3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentylamino)methyl)pyrrolidin-2-one 356811 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-3-phenyl-acrylamide 356812 cyclobutanecarboxylic acid [8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-amide 356813 N-methyl-N-{(S)-1-[(S)-3-(3-phenyl-propylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-4-pyridin-3-yl-benzamide 356828 3-amino-N-(2-(benzyloxy)-1-(2-(4-(3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)-5-fluorophenyl)ethyl)propanamide 356829 (+/-)-trans-4-((3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentyl)methyl)morpholine 356830 (+/-)-trans-methyl-3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentylcarbamate 356831 4'-trifluoromethyl-biphenyl-4-carboxylic acid methyl-{(S)-1-[(R)-3-(2-pyrrol-1-yl-ethylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-amide 356832 4'-trifluoromethyl-biphenyl-4-carboxylic acid {(S)-1-[(R)-3-(cyclohexylmethyl-methyl-amino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-methyl-amide 356833 trans-(S)-5-((3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentylamino)methyl)pyrrolidin-2-one 356834 trans-(S)-5-(((3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentyl)(methyl)amino)methyl)pyrrolidin-2-one 356835 1-(4-(2-((2S)-1-amino-2-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(2,4-dichlorophenyl)propan-1-one 356836 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(2,4-dichlorophenyl)propan-1-one 356837 N-methyl-N-{(S)-1-[(S)-3-(3-phenyl-propylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-4-pyridin-4-yl-benzamide 356852 4'-trifluoromethyl-biphenyl-4-carboxylic acid [(S)-1-((R)-3-amino-pyrrolidine-1-carbonyl)-pyrrolidin-3-yl]-methyl-amide 356853 4'-trifluoromethyl-biphenyl-4-carboxylic acid methyl-[(S)-1-((R)-3-methylamino-pyrrolidine-1-carbonyl)-pyrrolidin-3-yl]-amide 356854 (+/-)-trans-methyl-3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentyl(methyl)carbamate 356855 (+/-)-cis-methyl-3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentylcarbamate 356856 4'-trifluoromethyl-biphenyl-4-carboxylic acid methyl-{(S)-1-[(R)-3-(4,4,4-trifluoro-butylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-amide 356857 4'-trifluoromethyl-biphenyl-4-carboxylic acid {(S)-1-[(R)-3-(cyclobutylmethyl-methyl-amino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-methyl-amide 356858 (+/-)-trans-3-(3,5-bis(trifluoromethyl)benzyloxy)-N-((4H-1,2,4-triazol-3-yl)methyl)-N-methyl-2-phenylcyclopentanamine 356859 (+/-)-trans-5-(((2-(3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentyl)ethyl)(methyl)amino)methyl)-2H-1,2,4-triazol-3(4H)-one 356860 (S)-1-(4-(2-(1-amino-3-methylbutyl)-6-fluorophenyl)piperazin-1-yl)-3-(2,4-dichlorophenyl)propan-1-one 356861 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-fluorophenyl)piperazin-1-yl)-3-(2,4-dichlorophenyl)propan-1-one 356862 4-(5-methoxy-pyridin-3-yl)-N-methyl-N-{(S)-1-[(S)-3-(3-phenyl-propylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-benzamide 356877 (+/-)-trans-3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentanecarboxylic acid 356878 (+/-)-trans-benzyl-3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentylcarbamate 356879 4'-trifluoromethyl-biphenyl-4-carboxylic acid [(S)-1-((R)-3-dimethylamino-pyrrolidine-1-carbonyl)-pyrrolidin-3-yl]-methyl-amide 356880 4'-trifluoromethyl-biphenyl-4-carboxylic acid {(S)-1-[(R)-3-(ethyl-methyl-amino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-methyl-amide 356881 4'-trifluoromethyl-biphenyl-4-carboxylic acid methyl-((S)-1-{(R)-3-[methyl-(tetrahydro-pyran-4-yl)-amino]-pyrrolidine-1-carbonyl}-pyrrolidin-3-yl)-amide 356884 1-(4-(2-(1-amino-2-ethoxyethyl)-4-fluorophenyl)piperazin-1-yl)-3-(2,4-dichlorophenyl)propan-1-one 356885 1-(4-(2-(1-amino-2-(benzyloxy)ethyl)-4-fluorophenyl)piperazin-1-yl)-3-(2,4-dichlorophenyl)propan-1-one 356886 4-(6-methoxy-pyridin-3-yl)-N-methyl-N-{(S)-1-[(S)-3-(3-phenyl-propylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-benzamide 356889 1-(4-(2-(1-amino-2-methylpropyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(2,4-dichlorophenyl)propan-1-one 356909 (S)-3-(2,4-dichlorophenyl)-1-(4-(2-(1-(ethylamino)-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)propan-1-one 356910 (+/-)-trans-3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentanecarboxamide 356911 (+-)-trans-(3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentyl)methanamine 356912 (+/-)-cis-benzyl-3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentylcarbamate 356914 4'-trifluoromethyl-biphenyl-4-carboxylic acid {(S)-1-[(R)-3-(isobutyl-methyl-amino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-methyl-amide 356915 4'-trifluoromethyl-biphenyl-4-carboxylic acid methyl-((S)-1-{(R)-3-[methyl-(4-methyl-cyclohexyl)-amino]-pyrrolidine-1-carbonyl}-pyrrolidin-3-yl)-amide 356916 8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-ylamine 356917 4'-chloro-biphenyl-4-carboxylic acid methyl-{(S)-1-[(S)-3-(3-phenyl-propylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-amide 356936 (S)-3-(2,4-dichlorophenyl)-1-(4-(2-(1-(2-methoxyethylamino)-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)propan-1-one 356937 (+-)-trans-(3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentyl)-N-methylmethanamine 356938 (+/-)-trans-(3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentyl)methanol 356941 4'-trifluoromethyl-biphenyl-4-carboxylic acid {(S)-1-[(R)-3-(cyclopropylmethyl-methyl-amino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-methyl-amide 356942 (+/-)-cis-3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentanamine 356943 (+/-)-trans-2-((3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentyl)(methyl)amino)acetamide 356944 (+/-)-cis-2-(3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentylamino)acetamide 356945 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-acetamide 356946 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-2,2-dimethyl-propionamide 356947 4'-methoxy-biphenyl-4-carboxylic acid methyl-{(S)-1-[(S)-3-(3-phenyl-propylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-amide 356949 1-(4-(2-(1-amino-2-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(2,4-dichlorophenyl)propan-1-one 356963 ((2-chloro-5-methylphenyl)(6-(4-(3-(dimethylamino)-2-hydroxypropoxy)phenylamino)pyrimidin-4-yl)amino)acetonitrile 356964 N-(1S-[2-{4-[3-(4-chlorophenyl)propionyl]-1-piperazinyl}-5-(trifluoromethyl)phenyl]-3-methylbutyl)-2-aminoacetamide 356965 (+/-)-trans-1-((3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentyl)methyl)piperidine 356970 4'-trifluoromethyl-biphenyl-4-carboxylic acid ((S)-1-{(R)-3-[(1-acetyl-piperidin-4-yl)-methyl-amino]-pyrrolidine-1-carbonyl}-pyrrolidin-3-yl)-methyl-amide 356972 4'-trifluoromethyl-biphenyl-4-carboxylic acid ((S)-1-{(R)-3-[(3-cyclohexyl-propyl)-methyl-amino]-pyrrolidine-1-carbonyl}-pyrrolidin-3-yl)-methyl-amide 356973 4'-trifluoromethyl-biphenyl-4-carboxylic acid [(S)-1-((R)-3-{[3-(4-chloro-phenyl)-3-methyl-butyl]-methyl-amino}-pyrrolidine-1-carbonyl)-pyrrolidin-3-yl]-methyl-amide 356974 4'-trifluoromethyl-biphenyl-4-carboxylic acid [(S)-1-((R)-3-{[3-(4-chloro-phenyl)-3-methyl-butyl]-ethyl-amino}-pyrrolidine-1-carbonyl)-pyrrolidin-3-yl]-methyl-amide 356975 4'-trifluoromethyl-biphenyl-4-carboxylic acid [(S)-1-((R)-3-{acetyl-[3-(4-chloro-phenyl)-3-methyl-butyl]-amino}-pyrrolidine-1-carbonyl)-pyrrolidin-3-yl]-methyl-amide 356978 4'-acetylamino-biphenyl-4-carboxylic acid methyl-{(S)-1-[(S)-3-(3-phenyl-propylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-amide 356979 4'-(methyl-{(S)-1-[(S)-3-(3-phenyl-propylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-carbamoyl)-biphenyl-4-carboxylic acid methyl ester 356980 4'-trifluoromethoxy-biphenyl-4-carboxylic acid methyl-{(S)-1-[(S)-3-(3-phenyl-propylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-amide 356983 (+/-)-cis-3-(3,5-bis(trifluoromethyl)benzyloxy)-N-methyl-2-phenylcyclopentanamine 356984 trans-3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentanamine 356985 (+/-)-cis-2-((3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentyl)(methyl)amino)acetamide 356986 trans-2-(3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentylamino)acetamide 356987 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-2,2,2-trifluoro-acetamide 356989 4'-methylsulfanyl-biphenyl-4-carboxylic acid methyl-{(S)-1-[(S)-3-(3-phenyl-propylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-amide 357005 (S)-3-amino-N-(1-(2-(4-(3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)-5-(trifluoromethyl)phenyl)-3-methylbutyl)propanamide 357008 4'-trifluoromethyl-biphenyl-4-carboxylic acid methyl-{(S)-1-[(S)-3-(3-phenyl-propylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-amide 357010 4'-trifluoromethyl-biphenyl-4-carboxylic acid methyl-[(S)-1-((R)-3-phenethylamino-pyrrolidine-1-carbonyl)-pyrrolidin-3-yl]-amide 357011 trans-3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentanamine 357012 (+/-)-trans-2-((3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentyl)methylamino)acetamide 357013 trans-2-(3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentylamino)acetamide 357014 (+/-)-trans-4-((3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentylamino)methyl)-1H-imidazol-2(3H)-one 357020 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-4-trifluoromethyl-benzamide 357021 4'-trifluoromethyl-biphenyl-4-carboxylic acid ((S)-1-{(S)-3-[3-(4-chloro-phenyl)-3-methyl-butylamino]-pyrrolidine-1-carbonyl}-pyrrolidin-3-yl)-methyl-amide 357045 4'-trifluoromethyl-biphenyl-4-carboxylic acid methyl-((S)-1-{(R)-3-[(5-methyl-furan-2-ylmethyl)-amino]-pyrrolidine-1-carbonyl}-pyrrolidin-3-yl)-amide 357046 (+/-)-trans-2-(((3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentyl)methyl)(methyl)amino)acetamide 357053 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-3-methyl-benzamide 357054 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-3-methoxy-benzamide 357072 4'-trifluoromethyl-biphenyl-4-carboxylic acid methyl-((S)-1-{(R)-3-[(pyridin-2-ylmethyl)-amino]-pyrrolidine-1-carbonyl}-pyrrolidin-3-yl)-amide 357073 (+/-)-trans-1-(3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentyl)urea 357077 4'-cyano-biphenyl-4-carboxylic acid methyl-{(S)-1-[(S)-3-(3-phenyl-propylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-amide 357078 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-3-fluoro-benzamide 357079 3-chloro-N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-benzamide 357088 1-(4-(2-(1-aminoethyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(2,4-dichlorophenyl)propan-1-one 357089 1-(4-(2-(1-aminopentyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(2,4-dichlorophenyl)propan-1-one 357097 4'-trifluoromethyl-biphenyl-4-carboxylic acid ((S)-1-{(R)-3-[3-(4-chloro-phenyl)-3-methyl-butylamino]-pyrrolidine-1-carbonyl}-pyrrolidin-3-yl)-methyl-amide 357098 4'-trifluoromethyl-biphenyl-4-carboxylic acid {(S)-1-[(R)-3-(1-acetyl-piperidin-4-ylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-methyl-amide 357099 4'-trifluoromethyl-biphenyl-4-carboxylic acid {(S)-1-[(R)-3-(3-cyclohexyl-propylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-methyl-amide 357107 (+/-)-cis-1-(3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentyl)urea 357108 (+/-)-trans-1-(3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentyl)-3-methylurea 357112 4'-fluoro-biphenyl-4-carboxylic acid methyl-{(S)-1-[(S)-3-(3-phenyl-propylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-amide 357114 cyclohexanecarboxylic acid [8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-amide 357115 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-3-iodo-benzamide 357116 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(2-methoxyphenyl)propan-1-one 357135 (+/-)-trans-3-(3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentyl)-1,1-dimethylurea 357136 (+/-)-trans-1-(3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentyl)-1,3,3-trimethylurea 357140 (+/-)-cis-5-((((3-(3,5-bis(trifluoromethyl)benzyloxy)-2-phenylcyclopentyl)methyl)(methyl)amino)methyl)-2H-1,2,4-triazol-3(4H)-one 357142 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-benzamide 357143 4-bromo-N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-benzamide 357144 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-m-tolylpropan-1-one 357145 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(3-(trifluoromethyl)phenyl)propan-1-one 357166 (+/-)-trans-3-(3,5-bis(trifluoromethyl)benzyloxy)-N-methyl-2-phenylcyclopentanamine 357170 4-chloro-N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-benzamide 357171 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-4-methyl-benzamide 357174 (1R,2S,3S)-N-((1H-imidazol-2-yl)methyl)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)cyclopentanamine 357181 quinoline-2-carboxylic acid [8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-amide 357182 quinoline-3-carboxylic acid [8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-amide 357183 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-2-phenoxy-benzamide 357191 (-)-H-Dmt-Tic-beta-Ala-O-3-hydroxy-N-cyclobutylmethylmorphinan 357192 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-3-cyano-benzamide 357193 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-3-trifluoromethyl-benzamide 357194 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-2,6-dimethoxy-benzamide 357195 (1R,2R)-cis-2-[2-(4-chlorobenzylamino)ethyl]-1-(1H-imidazol-4-yl)cyclopropane 357198 (+)-N-[(1S,4R,5R,7S)-5-(3-hydroxyphenyl)-4-methyl-2-(3-phenylpropyl)-2-azabicyclo[3.3.1]non-7-yl]-2-methyl-2-phenylpropanamide 357199 (+)-N-{(1S,4R,5R,7S)-5-(3-hydroxyphenyl)-4-methyl-2-[3-(2-methylphenyl)prop-2-en-1-yl]-2-azabicyclo[3.3.1]non-7-yl}-2-methyl-2-phenylpropanamide 357209 isoxazole-3-carboxylic acid [8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-amide 357210 2-chloro-N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-nicotinamide 357211 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-2-cyclohexylamino-benzamide 357216 [8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-o-tolyl-methanone 357218 2-bromo-N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-benzamide 357219 2-chloro-N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-benzamide 357221 (1R,2R)-trans-2-(4-chlorobenzylamino)methyl-1-(1H-imidazol-4-yl)cyclopropane 357222 (1R,2R)-trans-2-(cyclohexylmethylamino)methyl-1-(1H-imidazol-4yl)cyclopropane 357227 (+)-2-ethyl-N-[(1S,4R,5R,7S)-5-(3-hydroxyphenyl)-4-methyl-2-(3-phenylpropyl)-2-azabicyclo[3.3.1]non-7-yl]-2-phenylbutanamide 357242 naphthalene-1-carboxylic acid [8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-amide 357243 naphthalene-2-carboxylic acid [8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-amide 357244 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-2-piperidin-1-yl-benzamide 357249 8-chloro-11-(4-methyl-piperazin-1-yl)-5-(toluene-4-sulfonyl)-5H-dibenzo[b,e][1,4]diazepine 357250 8-chloro-11-(4-methyl-piperazin-1-yl)-5-(toluene-2-sulfonyl)-5H-dibenzo[b,e][1,4]diazepine 357251 [8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-(2-methoxy-benzyl)-amine 357252 H-Dmt-Tic-beta-Ala-OH 357253 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-2,3-difluoro-benzamide 357255 (1R,2S)-trans-2-[2-(4-chlorobenzylamino)ethyl]-1-(1H-imidazol-4-yl)cyclopropane 357256 (1R,2S)-trans-2-[2-(cyclohexylmethylamino)ethyl]-1-(1H-imidazol-4-yl)cyclopropane 357257 (1S,2S)-trans-2-(4-chlorobenzylamino)methyl-1-(1H-imidazol-4-yl)cyclopropane 357266 N-[2-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-3-cyano-benzamide 357267 N-[2-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-3-methoxy-benzamide 357269 (2R)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-fluorophenyl)propanoyl]pyrrolidine-2-yl)-carbonyl-N-(1-methyl-4-piperidinylmethyl)pyrrolidine-2-carboxamide 357270 (2R)-N-(1-ethyl-4-piperidinylmethyl)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-fluorophenyl)propanoyl]pyrrolidine-2-yl)carbonylpyrrolidine-2-carboxamide 357271 (2R)-N-(1-cyclopropylmethyl-4-piperidinylmethyl)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-fluorophenyl)propanoyl]pyrrolidine-2-yl)carbonylpyrrolidine-2-carboxamide 357277 furan-2-carboxylic acid [8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-amide 357278 2-ethoxy-naphthalene-1-carboxylic acid [8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-amide 357279 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-2-(4-methyl-piperazin-1-yl)-benzamide 357286 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-2-methoxy-benzamide 357289 (1S,2S)-trans-2-(cyclohexylmethylamino)methyl-1-(1H-imidazol-4-yl)cyclopropane 357290 (1S,2R)-trans-2-[2-(4-chlorobenzylamino)ethyl]-1-(1H-imidazol-4-yl)cyclopropane 357291 (1S,2R)-trans-2-[2-(cyclohexylmethylamino)ethyl]-1-(1H-imidazol-4-yl)cyclopropane 357295 (+)-5-(3-hydroxyphenyl)-4-methyl-2-(3-phenylpropyl)-2-azabicyclo-[3.3.1]non-7-yl-(1-phenyl-1-cyclopentane)carboxamide 357296 8-chloro-11-[4-(2,3-dihydro-benzo[1,4]dioxin-6-ylmethyl)-piperazin-1-yl]-5H-dibenzo[b,e][1,4]diazepine 357297 (+/-)-3-(cyclopropylmethyl)-1,2,3,4,5,6-hexahydro-cis-6,11-dimethyl-N-[1,1'-biphenyl]-4-yl-2,6-methano-3-benzazocine-8-carboxamide 357298 2-chloro-N-{8-chloro-11-[4-(2,4-difluoro-benzyl)-piperazin-1-yl]-dibenzo[b,e][1,4]diazepin-5-yl}-benzamide 357299 N-[11-(4-benzo[1,3]dioxol-4-ylmethyl-piperazin-1-yl)-8-chloro-dibenzo[b,e][1,4]diazepin-5-yl]-2-chloro-benzamide 357300 (+)-N-[(1S,4R,5R,7S)-5-(3-hydroxyphenyl)-4-methyl-2-(3-phenylpropyl)-2-azabicyclo[3.3.1]non-7-yl]-1-(4-methoxyphenyl)-1-cyclopentanecarboxamide 357301 (+)-1-(4-fluorophenyl)-N-[(1S,4R,5R,7S)-5-(3-hydroxyphenyl)-4-methyl-2-(3-phenylpropyl)-2-azabicyclo[3.3.1]non-7-yl]-1-cyclopentanecarboxamide 357302 (+)-N-[(1S,4R,5R,7S)-5-(3-hydroxyphenyl)-4-methyl-2-(3-phenylpropyl)-2-azabicyclo[3.3.1]non-7-yl]-1-(1-naphthyl)cyclopentanecarboxamide 357303 (-)-N-(1S,4R,5R,7S)-{5-(3-hydroxy)phenyl-4-methyl-2-(3-phenylpropyl)-2-azabicyclo[3.3.1]non-7-yl}-1-(naphthalen-2-yl)-cyclopentanecarboxamide 357306 N-[2-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-5-fluoro-2-trifluoromethyl-benzamide 357307 N-[2-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-2,3,4,5-tetrafluoro-benzamide 357314 thiophene-2-carboxylic acid [8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-amide 357315 thiophene-3-carboxylic acid [8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-amide 357316 1-(4-(2-((1S)-1-(2-aminoethylamino)-2-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(2,4-dichlorophenyl)propan-1-one 357317 N-((1S)-1-(2-(4-(3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)-5-(trifluoromethyl)phenyl)-2-methylbutyl)methanesulfonamide 357320 N-[2,8-dichloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-2,6-dimethoxy-benzamide 357330 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-4-cyano-benzamide 357331 (1S,2R)-cis-2-(4-chlorobenzylamino)methyl-1-(1H-imidazol-4-yl)cyclopropane 357333 (1S,2S)-cis-2-[2-(4-chlorobenzylamino)ethyl]-1-(1H-imidazol-4-yl)cyclopropane 357338 (+)-N-[(1S,4R,5R,7S)-5-(3-hydroxyphenyl)-2,4-dimethyl-2-azabicyclo[3.3.1]non-7-yl]-1-phenylcyclopentanecarboxamide 357340 8-chloro-11-[4-(2,2-difluoro-benzo[1,3]dioxol-4-ylmethyl)-piperazin-1-yl]-5H-dibenzo[b,e][1,4]diazepine 357341 8-chloro-11-[4-(3-trifluoromethoxy-benzyl)-piperazin-1-yl]-5H-dibenzo[b,e][1,4]diazepine 357344 2-chloro-N-{8-chloro-11-[4-(2,4-dimethyl-benzyl)-piperazin-1-yl]-dibenzo[b,e][1,4]diazepin-5-yl}-benzamide 357345 2-chloro-N-{8-chloro-11-[4-(2,3-dihydro-benzo[1,4]dioxin-6-ylmethyl)-piperazin-1-yl]-dibenzo[b,e][1,4]diazepin-5-yl}-benzamide 357346 2-chloro-N-{8-chloro-11-[4-(2,2-difluoro-benzo[1,3]dioxol-4-ylmethyl)-piperazin-1-yl]-dibenzo[b,e][1,4]diazepin-5-yl}-benzamide 357347 2-chloro-N-{8-chloro-11-[4-(3-trifluoromethoxy-benzyl)-piperazin-1-yl]-dibenzo[b,e][1,4]diazepin-5-yl}-benzamide 357348 benzo[1,3]dioxole-5-carboxylic acid [2-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-amide 357349 N-[2-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-3,4,5-trimethoxy-benzamide 357359 4-ethoxy-thiophene-2-carboxylic acid [8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-amide 357360 3-phenyl-thiophene-2-carboxylic acid [8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-amide 357361 1-(4-(2-((1S)-1-((S)-2-aminopropylamino)-2-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(2,4-dichlorophenyl)propan-1-one 357362 methyl (1S)-1-(2-(4-(3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)-5-(trifluoromethyl)phenyl)-2-methylbutylcarbamate 357363 cis-rac-3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid (2-biphenyl-4-yl-ethyl)-amide 357364 (-)-3-(cyclopropylmethyl)-1,2,3,4,5,6-hexahydro-cis-6,11-dimethyl-N-(2-[1,1'-biphenyl]-4-ylethyl)-2,6-methano-3-benzazocine-8-carboxamide 357371 (1S,2S)-cis-2-[2-(cyclohexylmethylamino)ethyl]-1-(1H-imidazol-4-yl)cyclopropane 357387 N-[2,8-dichloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-5-fluoro-2-trifluoromethyl-benzamide 357390 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-2-fluoro-6-trifluoromethyl-benzamide 357391 3-ethoxy-benzo[b]thiophene-2-carboxylic acid [8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-amide 357392 3-(2,4-dichlorophenyl)-1-(4-(2-((1S)-2-methyl-1-((R)-pyrrolidin-2-ylmethylamino)butyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)propan-1-one 357393 N-((1S)-1-(2-(4-(3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)-5-(trifluoromethyl)phenyl)-2-methylbutyl)acetamide 357394 (+)-3-(cyclopropylmethyl)-1,2,3,4,5,6-hexahydro-cis-6,11-dimethyl-N-(2-[1,1'-biphenyl]-4-ylethyl)-2,6-methano-3-benzazocine-8-carboxamide 357414 N-[2,8-dichloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-2,3,4,5-tetrafluoro-benzamide 357415 benzo[1,3]dioxole-5-carboxylic acid [2,8-dichloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-amide 357417 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-2-fluoro-benzamide 357418 2-amino-6-chloro-N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-benzamide 357419 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-2,6-dimethyl-benzamide 357420 3-(2,4-dichlorophenyl)-1-(4-(2-((1S)-2-methyl-1-(2-methylbutylamino)butyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)propan-1-one 357421 3-(2,4-dichlorophenyl)-1-(4-(2-((1S)-2-methyl-1-((S)-pyrrolidin-2-ylmethylamino)butyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)propan-1-one 357422 2-amino-N-((1S)-1-(2-(4-(3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)-5-(trifluoromethyl)phenyl)-2-methylbutyl)acetamide 357423 (+/-)-3-(cyclopropylmethyl)-1,2,3,4,5,6-hexahydro-cis-6,11-dimethyl-N-(3-[1,1'-biphenyl]-4-ylpropyl)-2,6-methano-3-benzazocine-8-carboxamide 357437 (+)-N-[(1S,4R,5R,7S)-5-(3-hydroxyphenyl)-4-methyl-2-(3-phenylpropyl)-2-azabicyclo[3.3.1]non-7-yl]-1-phenyl-1-cyclohexanecarboxamide 357438 (+)-N-[(1S,4R,5R,7S)-5-(3-hydroxyphenyl)-4-methyl-2-(3-phenylpropyl)-2-azabicyclo[3.3.1]non-7-yl]-1-phenyl-1-cycloheptanecarboxamide 357444 N-[2,8-dichloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-3,4,5-trimethoxy-benzamide 357445 N-[2,8-dichloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-2-methyl-benzamide 357446 3,4-dichloro-N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-benzamide 357447 2-amino-N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-6-methyl-benzamide 357448 2-amino-N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-6-trifluoromethyl-benzamide 357449 3-(2,4-dichlorophenyl)-1-(4-(2-((1S)-2-methyl-1-((tetrahydrofuran-2-yl)methylamino)butyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)propan-1-one 357450 1-(4-(2-((1S)-1-(3-aminopropylamino)-2-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(2,4-dichlorophenyl)propan-1-one 357452 3-amino-N-((1S)-1-(2-(4-(3-(2,4-dichlorophenyl)propanoyl)piperazin-1-yl)-5-(trifluoromethyl)phenyl)-2-methylbutyl)propanamide 357453 (S)-3-(2,4-dichlorophenyl)-1-(4-(2-(3-methyl-1-(methylamino)butyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)propan-1-one 357454 (+/-)-3-(cyclopropylmethyl)-1,2,3,4,5,6-hexahydro-cis-6,11-dimethyl-N-(2-[1,1'-biphenyl]-4-ylethyl)-N-methyl-2,6-methano-3-benzazocine-8-carboxamide 357470 cis-rac-3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid benzylamide 357471 (+/-)-3-(cyclopropylmethyl)-1,2,3,4,5,6-hexahydro-cis-6,11-dimethyl-N-(2-phenylethyl)-2,6-methano-3-benzazocine-8-carboxamide 357473 (+)-(2R)-N-[(1S,4R,5R,7S)-5-(3-hydroxyphenyl)-4-methyl-2-(3-phenylpropyl)-2-azabicyclo[3.3.1]non-7-yl]-2-phenylpropanamide 357474 (+)-N-{(1S,4R,5R,7S)-5-(3-hydroxyphenyl)-4-methyl-2-[3-phenylprop-2-en-1-yl]-2-azabicyclo[3.3.1]non-7-yl}-2-methyl-2-phenylpropanamide 357475 N-[2,8-dichloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-2-iodo-benzamide 357477 2,6-dichloro-N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-benzamide 357478 2,4,6-trichloro-N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-benzamide 357479 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(thiophen-2-yl)propan-1-one 357480 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(benzo[b]thiophen-3-yl)propan-1-one 357481 1-(4-(2-((1S)-1-(benzylamino)-2-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(2,4-dichlorophenyl)propan-1-one 357496 8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepine-5-carboxylic acid (3,5-dichloro-phenyl)-amide 357500 (S)-N-(3-(4-(5-benzyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl)-1-phenylpropyl)cyclobutanecarboxamide 357503 (+/-)-3-(cyclopropylmethyl)-1,2,3,4,5,6-hexahydro-cis-6,11-dimethyl-N-(3-phenylpropyl)-2,6-methano-3-benzazocine-8-carboxamide 357504 8-chloro-11-[4-(2,4-difluoro-benzyl)-piperazin-1-yl]-5H-dibenzo[b,e][1,4]diazepine 357505 N-[2-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-4-cyano-benzamide 357510 (2S,4aR,6aR,7R,9R,10aS,10bR)-9-(Acetyloxy)-2-(3-furanyl)-dodecahydro-6a,10b-dimethyl-4,10-dioxo-2H-naphtho[2,1-c]pyran-7-carboxylic acid methyl ester 357511 3,5-dichloro-N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-benzamide 357512 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(4-(methylsulfonyl)phenyl)propan-1-one 357513 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(1H-indol-3-yl)propan-1-one 357514 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(1-methyl-1H-indol-3-yl)propan-1-one 357529 (S)-N-(3-(4-(2-(4-fluorophenyl)acetamido)piperidin-1-yl)-1-phenylpropyl)cyclobutanecarboxamide 357530 (S)-N-(3-(4-(3-benzyl-5-methyl-4H-1,2,4-triazol-4-yl)piperidin-1-yl)-1-phenylpropyl)cyclobutanecarboxamide 357532 2-chloro-N-[8-chloro-11-(4-isobutyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-benzamide 357533 2-chloro-N-{8-chloro-11-[4-(2,2-dimethyl-propyl)-piperazin-1-yl]-dibenzo[b,e][1,4]diazepin-5-yl}-benzamide 357534 11-(4-benzo[1,3]dioxol-4-ylmethyl-piperazin-1-yl)-8-chloro-5H-dibenzo[b,e][1,4]diazepine 357538 (+)-N-{(1S,4R,5R,7S)-5-(3-hydroxyphenyl)-4-methyl-2-[3-(2-methylphenyl)prop-2-en-1-yl]-2-azabicyclo[3.3.1]non-7-yl}-1-phenylcyclopentanecarboxamide 357545 (2S,4aR,6aR,7R,9R,10aS,10bR)-methyl 2-(furan-3-yl)-6a,10b-dimethyl-4,10-dioxo-9-(propionyloxy)-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 357546 (2S,4aR,6aR,7R,9R,10aS,10bR)-methyl 9-(butyryloxy)-2-(furan-3-yl)-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 357547 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(2,6-dichlorophenyl)propan-1-one 357548 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(benzo[d][1,3]dioxol-5-yl)propan-1-one 357549 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(2-methyl-1H-indol-3-yl)propan-1-one 357550 3-(2,4-dichlorophenyl)-1-(4-(2-((1S)-1-(ethylamino)-2-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)propan-1-one 357568 (S)-N-(3-(4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl)-1-phenylpropyl)cyclobutanecarboxamide 357569 (S)-N-(3-(4-(3,5-dimethyl-4H-1,2,4-triazol-4-yl)piperidin-1-yl)-1-phenylpropyl)cyclobutanecarboxamide 357571 2-chloro-N-{8-chloro-11-[4-(2-ethyl-butyl)-piperazin-1-yl]-dibenzo[b,e][1,4]diazepin-5-yl}-benzamide 357572 8-chloro-11-[4-(2,4-dimethyl-benzyl)-piperazin-1-yl]-5H-dibenzo[b,e][1,4]diazepine 357579 2-(((1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)cyclopentyl)(methyl)amino)-N-(2-hydroxyethyl)-N-methylacetamide 357580 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(3,4-dimethoxyphenyl)propan-1-one 357581 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(2,5-dimethoxyphenyl)propan-1-one 357595 N-((S)-3-(3-(2-methyl-1H-benzo[d]imidazol-1-yl)-8-aza-bicyclo[3.2.1]octan-8-yl)-1-phenylpropyl)cyclobutanecarboxamide 357597 benzo[1,3]dioxole-5-carboxylic acid [8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-amide 357599 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-nicotinamide 357600 2-chloro-N-[8-chloro-11-(4-cyclohexylmethyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-benzamide 357606 N-[2-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-2-methyl-benzamide 357607 2-(((1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)cyclopentyl)(methyl)amino)-1-(pyrrolidin-1-yl)ethanone 357608 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(2,4,5-trimethoxyphenyl)propan-1-one 357624 N-[(1S)-3-[2'-(2-methyl-1H-1,3-benzodiazol-1-yl)-7-azaspiro[bicyclo[2.2.1]heptane-2,1'-cyclopropane]-7-yl]-1-phenylpropyl]cyclobutanecarboxamide 357625 N-((S)-3-(7-(2-methyl-1H-benzo[d]imidazol-1-yl)-3-oxa-9-aza-bicyclo[3.3.1]nonan-9-yl)-1-phenylpropyl)cyclobutanecarboxamide 357626 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-4-fluoro-2-trifluoromethyl-benzamide 357627 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-isonicotinamide 357628 2-chloro-N-[8-chloro-11-(4-ethyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-benzamide 357629 2-chloro-N-{8-chloro-11-[4-(2-fluoro-benzyl)-piperazin-1-yl]-dibenzo[b,e][1,4]diazepin-5-yl}-benzamide 357633 (+)-N-[(1S,4R,5R,7S)-5-(3-hydroxyphenyl)-4-methyl-2-(3-phenylpropyl)-2-azabicyclo[3.3.1]non-7-yl]-1-(2-thienyl)cyclopentanecarboxamide 357634 N-[2-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-2-iodo-benzamide 357635 N-[2-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-2,6-dimethoxy-benzamide 357636 2-(((1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)cyclopentyl)(methyl)amino)-1-morpholinoethanone 357646 (+/-)-3-(cyclopropylmethyl)-6-ethyl-1,2,3,4,5,6-hexaahydro-cis-11-methyl-N-(2-[1,1'-biphenyl]-4-ylethyl)-1-oxo-2,6-methano-3-benzazocine-8-carboxamide 357653 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-3,4,5-trimethoxy-benzamide 357654 2-chloro-N-[8-chloro-11-(4-propyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-benzamide 357655 2-chloro-N-[8-chloro-11-(4-isopropyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-benzamide 357660 (+)-N-[(1S,4R,5R,7S)-5-(3-hydroxyphenyl)-4-methyl-2-(3-phenylpropyl)-2-azabicyclo[3.3.1]non-7-yl]-1-(3-thienyl)cyclopentanecarboxamide 357661 4-cyano-N-[2,8-dichloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-benzamide 357662 3-cyano-N-[2,8-dichloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-benzamide 357663 2-(((1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)cyclopentyl)(methyl)amino)-1-(4-methylpiperazin-1-yl)ethanone 357668 isoquinoline-1-carboxylic acid [8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-amide 357669 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-2-imidazol-1-yl-benzamide 357675 (S)-N-(3-(4-(3-benzyl-1H-1,2,4-triazol-1-yl)piperidin-1-yl)-1-phenylpropyl)cyclobutanecarboxamide 357676 N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-2,3,4,5-tetrafluoro-benzamide 357679 (+)-N-[(1S,4R,5R,7S)-5-(3-hydroxyphenyl)-4-methyl-2-(3-phenylpropyl)-2-azabicyclo[3.3.1]non-7-yl]-1-phenyl-1-cyclobutanecarboxamide 357680 (+)-N-[(1S,4R,5R,7S)-5-(3-hydroxyphenyl)-4-methyl-2-(2-phenoxyethyl)-2-azabicyclo[3.3.1]non-7-yl]-2-methyl-2-phenylpropanamide 357681 N-[2,8-dichloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-3-methoxy-benzamide 357683 1-(2-(benzyloxy)-5-bromobenzyl)-4-(hydroxymethyl)-1H-pyrazole-3-carboxylic acid 357687 (2S,4aR,6aR,7R,9R,10aS,10bR)-methyl 2-(furan-3-yl)-6a,10b-dimethyl-9-(N-methylpropionamido)-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 357688 (2S,4aR,6aR,7R,9R,10aS,10bR)-methyl 9-(N-ethylacetamido)-2-(furan-3-yl)-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 357693 deoxy salvinorin A 357705 N-(4-chloro-3-(trifluoromethyl)phenyl)-4-methyl-3-(2-(methylamino)quinazolin-6-yl)benzamide 357706 N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-3-hydroxy-2-{2-[(1R,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]ethyl}butanamide 357707 4-methyl-3-(2-(methylamino)quinazolin-6-yl)-N-(2-(piperidin-1-yl)-5-(trifluoromethyl)phenyl)benzamide 357709 2-[6-(3-cyano-phenyl)-1'-ethyl-3,4-dihydro-spiro[isoquinoline-1,4'-piperidin]-2-yl]-N-(3,5-dichloro-phenyl)-acetamide 357710 2-[6-(3-cyano-phenyl)-1'-cyclobutyl-3,4-dihydro-spiro[isoquinoline-1,4'-piperidin]-2-yl]-N-(3,5-dichloro-phenyl)-acetamide 357711 3-(2-(methylamino)quinazolin-6-yl)-N-(3-(trifluoromethyl)-phenyl)benzamide 357716 (R)-5-((((1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)cyclopentyl)(methyl)amino)methyl)pyrrolidin-2-one 357721 (2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 2-(furan-3-yl)-6a,10b-dimethyl-9-(methylamino)-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 357722 (2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 9-(ethylamino)-2-(furan-3-yl)-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 357726 (1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-N-ethyl-2-(4-fluorophenyl)cyclopentanamine 357727 (2S,4aR,6aS,7R,9S,10aS)-2-(furan-3-yl)-7-(hydroxymethyl)-6a,10b-dimethyl-5,10-dioxo-dodecahydro-1H-benzo[f]isochromen-9-yl acetate 357731 (2S)-N-[3,5-bis(trifluoromethyl)benzyl]-2-cyclopropyl-4-[(1R,3R')-3'methyl-1'H-spiro[indene-1,4'-piperidin]-1'yl]butanamide 357735 4-methyl-N-(2-(3-methyl-2-oxoimidazolidin-1-yl)-5-(trifluoromethyl)phenyl)-3-(2-(methylamino)quinazolin-6-yl)benzamide 357737 3-(2-aminoquinazolin-6-yl)-N-(3-(trifluoromethyl)phenyl)-benzamide 357741 (S)-5-((((1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)cyclopentyl)(methyl)amino)methyl)-1-methylpyrrolidin-2-one 357743 (2R)-N-(1-cyclobutylmethyl-4-piperidinylmethyl)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-fluorophenyl)propanoyl]pyrrolidine-2-yl)carbonylpyrrolidine-2-carboxamide 357744 (2R)-N-(1-cyclopentylmethyl-4-piperidinylmethyl)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-fluorophenyl)propanoyl]pyrrolidine-2-yl)carbonylpyrrolidine-2-carboxamide 357745 (2R)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-fluorophenyl)propanoyl]pyrrolidine-2-yl)carbonyl-N-[1-(2-propyl)-4-piperidinylmethyl]pyrrolidine-2-carboxamide 357747 (2R)-N-(1-cyclopentyl-4-piperidinylmethyl)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-fluorophenyl)-propanoyl]pyrrolidine-2-yl)carbonylpyrrolidine-2-carboxamide 357751 (2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 2-(furan-3-yl)-9-(isopropylamino)-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 357752 (2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 9-(dimethylamino)-2-(furan-3-yl)-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 357760 1-((S)-2-((R)-2-(4-(aminomethyl)piperidine-1-carbonyl)pyrrolidine-1-carbonyl)pyrrolidin-1-yl)-3,3,3-triphenylpropan-1-one trifluoroacetic acid 357761 (R)-N-(piperidin-4-ylmethyl)-1-((S)-1-(3,3,3-triphenylpropanoyl)pyrrolidine-2-carbonyl)pyrrolidine-2-carboxamide trifluoroacetic acid 357763 (R)-N-((R)-piperidin-3-ylmethyl)-1-((S)-1-(3,3,3-triphenylpropanoyl)pyrrolidine-2-carbonyl)pyrrolidine-2-carboxamide trifluoroacetic acid 357771 (1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)-N-(2-methoxyethyl)cyclopentanamine 357772 (1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)-N-(2-methoxyethyl)-N-methylcyclopentanamine 357777 N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-2-cyclopropyl-4-{spiro[indene-1,4'-piperidine]-1'-yl}butanamide 357778 (2R)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-2-cyclopropyl-4-[(1R,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]butanamide 357780 N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-2-methanesulfonamido-4-{spiro[indene-1,4'-piperidine]-1'-yl}butanamide 357783 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-4-(4-chlorophenyl)butane-1,4-dione 357784 (S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-cyclopropyl-4-(4-phenylpiperidin-1-yl)butanamide 357785 (R)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-(4-phenylpiperidin-1-yl)ethyl)pentanamide 357786 N-(2-(3,3-dimethyl-2-oxoazetidin-1-yl)-5-(trifluoromethyl)phenyl)-4-methyl-3-(2-(methylamino)quinazolin-6-yl)benzamide 357790 (2S,4aR,6aR,7R,9R,10aS,10bR)-methyl 9-amino-2-(furan-3-yl)-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 357791 4-((((1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)cyclopentyl)(methyl)amino)methyl)-1H-imidazol-2(3H)-one 357794 1-(2-(benzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid 357799 (R)-N-(2-(piperidin-4-yl)ethyl)-1-((S)-1-(3,3,3-triphenylpropanoyl)pyrrolidine-2-carbonyl)pyrrolidine-2-carboxamide trifluoroacetic acid 357801 (R)-N-(3-aminocyclohexyl)-1-((S)-1-(3,3,3-triphenylpropanoyl)pyrrolidine-2-carbonyl)pyrrolidine-2-carboxamide trifluoroacetic acid 357802 (S)-2-((S)-4-((R)-2-amino-3-(4-fluorophenyl)propanoyl)-3-(3-guanidinopropyl)-2-oxopiperazin-1-yl)-N-methyl-3-(naphthalen-2-yl)propanamide 357803 (S)-2-[(S)-4-{(R)-2-[(S)-2-acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-3-phenyl-propionyl}-3-(3-guanidino-propyl)-2-oxo-piperazin-1-yl]-N-methyl-3-naphthalen-2-yl-propionamide 357804 (S)-2-[(S)-4-{(R)-2-[(S)-2-acetylamino-3-(4-hydroxy-phenyl)-propionylamino]-3-phenyl-propionyl}-3-(3-guanidino-propyl)-2-oxo-piperazin-1-yl]-N-methyl-3-naphthalen-2-yl-propionamide 357809 (R)-N-((1S,2S)-2-aminocyclohexyl)-1-((S)-1-(3,3,3-triphenylpropanoyl)pyrrolidine-2-carbonyl)pyrrolidine-2-carboxamide trifluoroacetic acid 357812 (S)-2-[(S)-4-[(R)-2-[(S)-2-acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-3-(4-fluoro-phenyl)-propionyl]-3-(3-guanidino-propyl)-2-oxo-piperazin-1-yl]-N-methyl-3-naphthalen-2-yl-propionamide 357813 (S)-2-[(S)-4-[(R)-2-[(S)-2-acetylamino-3-(4-hydroxy-phenyl)-propionylamino]-3-(4-fluoro-phenyl)-propionyl]-3-(3-guanidino-propyl)-2-oxo-piperazin-1-yl]-N-methyl-3-naphthalen-2-yl-propionamide 357814 (S)-2-((S)-4-((R)-3-(4-fluorophenyl)-2-(piperazin-1-yl)propanoyl)-3-(3-guanidinopropyl)-2-oxopiperazin-1-yl)-N-methyl-3-(naphthalen-2-yl)propanamide 357815 2-((1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)cyclopentylamino)acetamide 357816 2-(((1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)cyclopentyl)(methyl)amino)acetamide 357819 (2S)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-2-cyclopropyl-4-{spiro[indene-1,4'-piperidine]-1'-yl}butanamide 357824 4-(4-(2-((S)-1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-1-(4-chlorophenyl)-2-methylbutane-1,4-dione 357825 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-cyclohexylpropan-1-one 357826 (R)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-(4-phenylpiperidin-1-yl)ethyl)pent-4-enamide 357831 (2S,4aR,6aR,7R,9R,10aS,10bR)-methyl 9-(ethylamino)-2-(furan-3-yl)-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 357832 (1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-N-((4H-1,2,4-triazol-3-yl)methyl)-2-(4-fluorophenyl)-N-methylcyclopentanamine 357839 1-(2-(benzyloxy)-5-bromobenzyl)-1H-pyrazole-3-carboxylic acid 357841 (S)-2-((S)-4-((R)-2-amino-3-phenylpropanoyl)-3-(3-guanidinopropyl)-2-oxopiperazin-1-yl)-N-methyl-3-(naphthalen-2-yl)propanamide 357844 2-(((1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)cyclopentyl)(ethyl)amino)acetamide 357847 (2R)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-2-methyl-4-{spiro[indene-1,4'-piperidine]-1'-yl}butanamide 357848 4-methyl-3-(2-(methylamino)quinazolin-6-yl)-N-(4-(1-methylpiperidin-4-yloxy)phenyl)benzamide 357855 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-4-cyclohexylbutan-1-one 357856 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-2-(2,4-dichlorophenoxy)ethanone 357857 N-(2-(2-(diethylamino)acetamido)-5-(trifluoromethyl)phenyl)-4-methyl-3-(2-(methylamino)quinazolin-6-yl)benzamide 357859 N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-(4-(4-fluorophenyl)piperidin-1-yl)ethyl)-3-hydroxybutanamide 357864 (2S)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-4-[(1R,3'R)-3'-ethylspiro[indene-1,4'-piperidine]-1'-yl]-2-(4-fluorophenyl)butanamide 357865 (2S,4aR,6aR,7R,9R,10aS,10bR)-methyl 2-(furan-3-yl)-9-(isopropylamino)-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 357866 (1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)-N-(pyridin-3-ylmethyl)cyclopentanamine 357872 (2S,4aS,6aS,7R,9S,10aS)-2-(furan-3-yl)-7-(methoxymethyl)-6a,10b-dimethyl-5,10-dioxo-dodecahydro-1H-benzo[f]isochromen-9-yl acetate 357875 2-propyl-pentanoic acid [8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b,e][1,4]diazepin-5-yl]-amide 357881 D-Phe-Arg-2-Nal-NHCH3 357882 N-(2,3-dihydro-1H-inden-4-yl)-4-methyl-3-(2-(methylamino)quinazolin-6-yl)benzamide 357883 (2S)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-2-methyl-4-{spiro[indene-1,4'-piperidine]-1'-yl}butanamide 357884 N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-2-cyclohexyl-4-{spiro[indene-1,4'-piperidine]-1'-yl}butanamide 357897 1-(4-(2-((S)-1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(4-chlorophenyl)-2-methylpropan-1-one 357898 (R)-1-(4-(2-((S)-1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(4-chlorophenyl)-2-methylpropan-1-one 357899 (1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)-N-(pyridin-4-ylmethyl)cyclopentanamine 357903 1-(2-(benzyloxy)-5-bromobenzyl)-5-butyl-1H-pyrazole-3-carboxylic acid 357908 (S)-2-((R)-2-amino-3-(4-fluorophenyl)propanamido)-5-guanidino-N-((S)-1-(methylamino)-3-(naphthalen-2-yl)-1-oxopropan-2-yl)pentanamide 357909 (2R)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-2-(2-{spiro[indene-1,4'-piperidine]-1'-yl}ethyl)pent-4-enamide 357926 1-(4-(2-((S)-1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(4-methoxyphenyl)-2-methylpropan-1-one 357927 1-(4-(2-((S)-1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(3-chlorophenyl)-2-methylpropan-1-one 357928 N-((1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)cyclopentyl)-N-methylpyrazin-2-amine 357934 (R)-N-((S)-piperidin-3-ylmethyl)-1-((S)-1-(3,3,3-triphenylpropanoyl)pyrrolidine-2-carbonyl)pyrrolidine-2-carboxamide 357945 (S)-2-((S)-4-((R)-2-amino-3-(4-fluorophenyl)propanoyl)-3-(2-aminoethyl)-2-oxopiperazin-1-yl)-N-methyl-3-(naphthalen-2-yl)propanamide 357946 (2S)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-3-methyl-2-(2-{spiro[indene-1,4'-piperidine]-1'-yl}ethyl)butanamide 357949 2-(1-acetylpiperidin-3-yl)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-4-{spiro[indene-1,4'-piperidine]-1'-yl}butanamide 357950 2-benzyl-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-4-{spiro[indene-1,4'-piperidine]-1'-yl}butanamide 357963 1-(4-(2-((S)-1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(3-methoxyphenyl)-2-methylpropan-1-one 357964 1-(4-(2-((S)-1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(3-ethoxyphenyl)-2-methylpropan-1-one 357965 N-((1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)cyclopentyl)-2-(1H-imidazol-4-yl)-N-methylacetamide 357966 (2S,4aR,6aR,7R,9R,10aS,10bR)-methyl 9-(N-ethylpropionamido)-2-(furan-3-yl)-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 357971 (2S,4aR,6aR,7R,9S,10aS,10bR)-9-(Acetylamino)-2-(3-furanyl)-dodecahydro-6a,10b-dimethyl-4,10-dioxo-2H-naphtho[2,1-c]pyran-7-carboxylic acid methyl ester 357972 (2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 2-(furan-3-yl)-6a,10b-dimethyl-4,10-dioxo-9-propionamido-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 357975 1-(2-((S)-1-((R)-2-amino-3-(4-fluorophenyl)propanoyl)-4-((S)-1-(methylamino)-3-(naphthalen-2-yl)-1-oxopropan-2-yl)-3-oxopiperazin-2-yl)ethyl)urea 357977 (2R)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-3-methyl-2-(2-{spiro[indene-1,4'-piperidine]-1'-yl}ethyl)butanamide 357983 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-2-(2,4-dichlorophenyl)ethanone 357987 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-2-(2-chlorophenoxy)ethanone 357988 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-2-(2,4-dimethylphenoxy)ethanone 357991 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-2-(2,4-dichlorophenylthio)ethanone 357993 1-(2-(benzyloxy)-5-bromobenzyl)-4-(trifluoromethyl)-1H-pyrazole-3-carboxylic acid 357994 (S)-5-(((1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)cyclopentylamino)methyl)pyrrolidin-2-one 357999 (2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 2-(furan-3-yl)-6a,10b-dimethyl-9-(N-methylacetamido)-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 358000 (2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 2-(furan-3-yl)-6a,10b-dimethyl-9-(N-methylpropionamido)-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 358019 (S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-cyclopropyl-4-(4-(4-fluorophenyl)piperidin-1-yl)butanamide 358021 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-2-(3,4-dichlorophenoxy)ethanone 358022 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-2-(2,3-dichlorophenoxy)ethanone 358023 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-2-(phenylamino)ethanone 358024 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-2-(1H-benzo[d]imidazol-1-yl)ethanone 358027 (S)-5-((((1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)cyclopentyl)(methyl)amino)methyl)pyrrolidin-2-one 358034 (2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 9-(N-ethylacetamido)-2-(furan-3-yl)-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 358035 (2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 9-(N-ethylpropionamido)-2-(furan-3-yl)-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 358040 (S)-2-acetamido-N1-((R)-3-(4-fluorophenyl)-1-((S)-2-(3-guanidinopropyl)-4-((S)-1-(methylamino)-3-(naphthalen-2-yl)-1-oxopropan-2-yl)-3-oxopiperazin-1-yl)-1-oxopropan-2-yl)pentanediamide 358046 (2R)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-chlorophenyl)propanoyl]pyrrolidine-2-yl)carbonyl-N-((3R)-3-piperidinylmethyl)-pyrrolidine-2-carboxamide 358047 (2R)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-fluorophenyl)propanoyl]pyrrolidine-2-yl)carbonyl-N-(4-piperidinylmethyl)pyrrolidine-2-carboxamide 358048 (2R)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-fluorophenyl)propanoyl]pyrrolidine-2-yl)carbonyl-N-(4-piperidinylethyl)pyrrolidine-2-carboxamide 358049 (2R)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-fluorophenyl)propanoyl]pyrrolidine-2-yl)carbonyl-N-[(3R)-3-piperidinylmethyl]-pyrrolidine-2-carboxamide 358050 N-((R)-3-(4-fluorophenyl)-1-((S)-2-(3-guanidinopropyl)-4-((S)-1-(methylamino)-3-(naphthalen-2-yl)-1-oxopropan-2-yl)-3-oxopiperazin-1-yl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 358059 N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-4-{spiro[indene-1,4'-piperidine]-1'-yl}-2-(trifluoromethane)sulfonamidobutanamide 358065 N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-2-[(2-oxoimidazolidin-4-yl)formamido]-4-{spiro[indene-1,4'-piperidine]-1'-yl}butanamide 358071 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-2-(4-chlorophenoxy)ethanone 358073 1-(2-(4-methyl-3-(2-(methylamino)quinazolin-6-yl)benzamido)-4-(trifluoromethyl)phenyl)-3-(2-morpholinoethyl)urea 358074 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-2-(naphthalen-1-yloxy)ethanone 358075 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-2-(naphthalen-2-yloxy)ethanone 358076 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(cyclohexylamino)propan-1-one 358083 (1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-N-((4H-1,2,4-triazol-3-yl)methyl)-N-ethyl-2-(4-fluorophenyl)cyclopentanamine 358092 2-(((1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)cyclopentyl)(2-methoxyethyl)amino)acetamide 358103 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-2-(p-tolyloxy)ethanone 358104 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-2-(4-methoxyphenoxy)ethanone 358105 2-[6-(3-cyano-phenyl)-1'-isopropyl-3,4-dihydro-spiro[isoquinoline-1,4'-piperidin]-2-yl]-N-(3,5-dichloro-phenyl)-acetamide 358111 5-((((1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)cyclopentyl)(methyl)amino)methyl)-2H-1,2,4-triazol-3(4H)-one 358115 (2S,4aS,6aR,7R,9S,10aS,10bR)-9-(Butyryloxy)-2-(3-furanyl)-dodecahydro-6a,10b-dimethyl-4,10-dioxo-2H-naphtho[2,1-c]pyran-7-carboxylic Acid Methyl Ester 358116 salvinorin B 358126 (2R)-1-[(2S,4R)-4-hydroxy-1-(3,3,3-triphenylpropanoyl)pyrrolidine-2-yl]carbonyl-N-(4-piperidinylmethyl)pyrrolidine-2-carboxamide 358127 (S)-2-((S)-4-((R)-2-acetamido-3-(4-fluorophenyl)propanoyl)-3-(3-guanidinopropyl)-2-oxopiperazin-1-yl)-N-methyl-3-(naphthalen-2-yl)propanamide 358128 2-(((1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)cyclopentyl)(methyl)amino)-N-methylacetamide 358129 2-(((1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)cyclopentyl)(methyl)amino)-N,N-dimethylacetamide 358131 1-(2-(benzyloxy)-5-bromobenzyl)-5-(thiophen-2-yl)-1H-pyrazole-3-carboxylic acid 358136 4-methyl-3-(2-(methylamino)quinazolin-6-yl)-N-(2-(1-methylpiperidin-4-yloxy)-5-(trifluoromethyl)phenyl)benzamide 358137 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-2-(4-hydroxyphenoxy)ethanone 358138 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-2-(4-nitrophenoxy)ethanone 358139 2-[6-(3-cyano-phenyl)-1'-cyclopropylmethyl-3,4-dihydro-spiro[isoquinoline-1,4'-piperidin]-2-yl]-N-(3,5-dichloro-phenyl)-acetamide 358140 1-(2-(benzyloxy)-5-bromobenzyl)-4-fluoro-1H-pyrazole-3-carboxylic acid 358142 5-(2-aminoquinazolin-6-yl)-2-fluoro-N-(3-(trifluoromethyl)phenyl)benzamide 358149 (2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 2-(furan-3-yl)-9-methoxy-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 358153 (1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)cyclopentanamine 358156 (2R)-1-[(2S,4R)-4-hydroxy-1-(3,3,3-triphenylpropanoyl)pyrrolidine-2-yl]carbonyl-N-(4-piperidinylethyl)pyrrolidine-2-carboxamide 358157 (2R)-1-[(2S,4R)-4-hydroxy-1-(3,3,3-triphenylpropanoyl)pyrrolidine-2-yl]carbonyl-N-((3R)-3-piperidinylmethyl)pyrrolidine-2-carboxamide 358158 (2R)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-chlorophenyl)propanoyl]pyrrolidine-2-yl)carbonyl-N-(4-piperidinylmethyl)pyrrolidine-2-carboxamide 358159 (2R)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-chlorophenyl)propanoyl]pyrrolidine-2-yl)carbonyl-N-(4-piperidinylethyl)pyrrolidine-2-carboxamide 358160 1-(3-((S)-1-((R)-2-amino-3-(4-fluorophenyl)propanoyl)-4-((S)-1-(methylamino)-3-(naphthalen-2-yl)-1-oxopropan-2-yl)-3-oxopiperazin-2-yl)propyl)urea 358161 2-(((1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)cyclopentyl)(methyl)amino)-N-(2-methoxyethyl)acetamide 358165 N-(4-chloro-2-methyl-3-(trifluoromethyl)phenyl)-4-methyl-3-(2-(methylamino)quinazolin-6-yl)benzamide 358166 methyl N-[1-({[3,5-bis(trifluoromethyl)phenyl]methyl}carbamoyl)-3-{spiro[indene-1,4'-piperidine]-1'-yl}propyl]carbamate 358167 (S)-1-(4-(2-(1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-2-(3-chlorophenoxy)ethanone 358168 2-[6-(3-cyano-phenyl)-1'-cyclopentyl-3,4-dihydro-spiro[isoquinoline-1,4'-piperidin]-2-yl]-N-(3,5-dichloro-phenyl)-acetamide 358169 1-(2-(benzyloxy)-5-bromobenzyl)-4-methyl-1H-pyrazole-3-carboxylic acid 358170 3-(2-aminoquinazolin-6-yl)-4-chloro-N-(3-(trifluoromethyl)-phenyl)benzamide 358171 (2S,4aR,6aR,7R,9R,10aS,10bR)-methyl 9-(dimethylamino)-2-(furan-3-yl)-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 358172 (2S,4aR,6aR,7R,9R,10aS,10bR)-methyl 9-acetamido-2-(furan-3-yl)-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 358189 (1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)-N-methylcyclopentanamine 358190 (S)-2-[(S)-4-[(R)-2-Amino-3-(4-fluoro-phenyl)-propionyl]-3-(2-guanidino-ethyl)-2-oxo-piperazin-1-yl]-N-methyl-3-naphthalen-2-yl-propionamide 358191 2-(((1R,2S,3S)-3-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-2-(4-fluorophenyl)cyclopentyl)(methyl)amino)-N-(2-methoxyethyl)-N-methylacetamide 358197 (2S)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-2-cyclobutyl-4-[(1R,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]butanamide 358199 2-[6-(3-cyano-phenyl)-3,4-dihydro-spiro[isoquinoline-1,4'-piperidin]-2-yl]-N-(3,5-dichloro-phenyl)-acetamide 358200 2-[6-(3-cyano-phenyl)-1'-methyl-3,4-dihydro-spiro[isoquinoline-1,4'-piperidin]-2-yl]-N-(3,5-dichloro-phenyl)-acetamide 358201 2-[6-(3-cyano-phenyl)-1'-(1-hydroxy-ethyl)-3,4-dihydro-spiro[isoquinoline-1,4'-piperidin]-2-yl]-N-(3,5-dichloro-phenyl)-acetamide 358202 1-(2-(benzyloxy)-5-bromobenzyl)-4-bromo-1H-pyrazole-3-carboxylic acid 358203 2-fluoro-4-methyl-5-(2-(methylamino)quinazolin-6-yl)-N-(3-(trifluoromethyl)phenyl)benzamide 358206 (2S,4aR,6aR,7R,9R,10aS,10bR)-methyl 2-(furan-3-yl)-6a,10b-dimethyl-4,10-dioxo-9-propionamido-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 358207 (2S,4aR,6aR,7R,9R,10aS,10bR)-methyl 2-(furan-3-yl)-6a,10b-dimethyl-9-(N-methylacetamido)-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 358222 (S)-2-((S)-4-(3-(4-fluorophenyl)propanoyl)-3-(3-guanidinopropyl)-2-oxopiperazin-1-yl)-N-methyl-3-(naphthalen-2-yl)propanamide 358225 (2S,4aR,6aR,7R,9S,10aS,10bR)-2-(furan-3-yl)-6a,10b-dimethyl-7-(methylcarbamoyl)-4,10-dioxo-dodecahydro-1H-benzo[f]isochromen-9-yl acetate 358229 N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-2-(1-methanesulfonylpiperidin-3-yl)-4-{spiro[indene-1,4'-piperidine]-1'-yl}butanamide 358232 (2S)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-2-(cyclopropylmethyl)-4-[(1R,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]butanamide 358236 Ac-RYYRIK-K-(NH2)-YAFGYPS 358237 Ac-RYYRIK-GGG-K-(NH2)-YAFGYPS-GG 358240 1-(4-(2-((S)-1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(4-chloro-2-fluorophenyl)-2-methylpropan-1-one 358241 1-(4-(2-((S)-1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(4-chloro-2-methylphenyl)-2-methylpropan-1-one 358242 1-(4-(2-((S)-1-amino-3-methylbutyl)-4-chlorophenyl)piperazin-1-yl)-3-(4-chlorophenyl)-2-methylpropan-1-one 358243 1-(4-(2-((S)-1-amino-3-methylbutyl)-4-chlorophenyl)piperazin-1-yl)-3-(4-methoxyphenyl)-2-methylpropan-1-one 358244 1-(2-(2,4-difluorobenzyloxy)-5-fluorobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid 358245 4-methyl-N-(2-methyl-3-(trifluoromethyl)phenyl)-3-(2-(3-morpholinopropylamino)quinazolin-6-yl)benzamide 358252 12'-bromo-4'-(furan-2-yl)-1-methyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358253 12'-bromo-1-methyl-4'-(thiophen-2-yl)-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358258 12'-bromo-4'-(4-bromophenyl)-1-propyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358259 12'-bromo-4'-(4-methoxyphenyl)-1-propyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358268 2-(1-(1-cyclopentylpiperidin-4-yl)-6-(3-formylphenyl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358269 2-(1-(1-cyclopentylpiperidin-4-yl)-6-(2,5-dichlorophenyl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358270 2-(1-(1-cyclopentylpiperidin-4-yl)-6-(quinolin-8-yl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358274 2-(6-(3-(1H-imidazol-2-yl)phenyl)-1-(1-cyclopentylpiperidin-4-yl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358277 (+/-)-(4-bromo-3,6-dimethoxybenzocyclobuten-1-yl)methylamine 358280 2-(1-(1-benzylpiperidin-4-yl)-6-(3-cyanophenyl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358281 2-(6-(3-cyanophenyl)-1-(1-(5-hydroxypentyl)piperidin-4-yl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358282 2-(6-(3-cyanophenyl)-1-(1-cycloheptylpiperidin-4-yl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358283 2-(6-(3-cyanophenyl)-1-(1-(tetrahydro-2H-pyran-4-yl)piperidin-4-yl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358284 2-(6-(3-cyanophenyl)-1-(1-(tetrahydrothiophen-3-yl)piperidin-4-yl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358289 1-(4-(2-((S)-1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(4-chloro-2-hydroxyphenyl)-2-methylpropan-1-one 358290 (1S)-[2-{4-[2-methyl-3-(2-methoxy-4-chlorophenyl)propionyl]-1-piperazinyl}-5-(trifluoromethyl)phenyl]-3-methylbutylamine 358291 1-[5-bromo-2-(3-methyl-benzyloxy)-benzyl]-5-methyl-1H-pyrazole-3-carboxylic acid 358292 1-(2-(3-nitrobenzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid 358293 (R)-1-(4-(2-((S)-1-amino-3-methylbutyl)-4-methylphenyl)piperazin-1-yl)-3-(2,4-dichlorophenyl)-2-methylpropan-1-one 358294 (R)-1-(4-(2-((S)-1-amino-3-methylbutyl)phenyl)piperazin-1-yl)-3-(4-chlorophenyl)-2-methylpropan-1-one 358295 1-methyl-4'-(pyridin-4-yl)-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358296 12'-bromo-4'-(4-fluorophenyl)-1-methyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358300 N-(4-(3-fluorobenzyloxy)-3-chlorophenyl)-6-(5-((2-(phenylsulfonyl)ethoxy)methyl)furan-2-yl)quinazolin-4-amine 358301 N-(4-(benzyloxy)-3-chlorophenyl)-6-(5-((4-(phenylsulfonyl)butylamino)methyl)furan-2-yl)quinazolin-4-amine 358302 N-(4-(3-fluorobenzyloxy)-3-chlorophenyl)-6-(5-(((2-(methylsulfonyl)ethyl)(propyl)amino)methyl)furan-2-yl)quinazolin-4-amine 358303 2-(((5-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamino)quinazolin-6-yl)furan-2-yl)methyl)(2-(methylsulfonyl)ethyl)amino)acetonitrile 358305 12'-bromo-1-methyl-4'-(naphthalen-2-yl)-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358311 1-propyl-4'-(pyridin-4-yl)-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358316 N-(4-chloro-3-trifluoromethyl-phenyl)-2-[6-(3-cyano-phenyl)-1'-cyclopropylmethyl-3,4-dihydro-spiro[isoquinoline-1,4'-piperidin]-2-yl]-acetamide 358331 1-(4-(2-((S)-1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(4-chloro-3-methylphenyl)-2-methylpropan-1-one 358333 (R)-1-(4-(2-((S)-1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(4-chloro-2-methoxyphenyl)-2-methylpropan-1-one 358334 1-(2-(3-(trifluoromethyl)benzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid 358335 1-(2-(3,5-dichlorobenzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid 358338 (R)-1-(4-(2-((S)-1-amino-3-methylbutyl)phenyl)piperazin-1-yl)-3-(4-chloro-2-fluorophenyl)-2-methylpropan-1-one 358339 (R)-1-(4-(2-((S)-1-amino-3-methylbutyl)phenyl)piperazin-1-yl)-3-(2,4-dichlorophenyl)-2-methylpropan-1-one 358341 N-(4-(benzyloxy)-3-(trifluoromethyl)phenyl)-6-(5-((2-(methylsulfonyl)ethylamino)methyl)furan-2-yl)quinazolin-4-amine 358342 N-(4-(3-fluorobenzyloxy)-3-(trifluoromethyl)phenyl)-6-(5-((2-(methylsulfonyl)ethylamino)methyl)furan-2-yl)quinazolin-4-amine 358343 N-(4-(3-fluorobenzyloxy)-3-chlorophenyl)-6-(5-((2-(propylsulfonyl)ethylamino)methyl)furan-2-yl)quinazolin-4-amine 358344 N-(4-(3-fluorobenzyloxy)-3-chlorophenyl)-6-(5-((2-(isopropylsulfonyl)ethylamino)methyl)furan-2-yl)quinazolin-4-amine 358350 4'-(4-fluorophenyl)-10'-methoxy-1-methyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358356 2-(4-fluorophenyl)-1,10b-dihydro-benzo[e]pyrazolo[1,5-c][1,3]oxazine-5-spiro-4'-(1'-propylpiperidine) 358361 2-[6-(3-cyano-phenyl)-1'-cycloheptyl-3,4-dihydro-spiro[isoquinoline-1,4'-piperidin]-2-yl]-N-(3,5-dichloro-phenyl)-acetamide 358362 2-[6-(3-cyano-phenyl)-1'-(tetrahydro-pyran-4-yl)-3,4-dihydro-spiro[isoquinoline-1,4'-piperidin]-2-yl]-N-(3,5-dichloro-phenyl)-acetamide 358363 2-[6-(3-cyano-phenyl)-1'-furan-3-ylmethyl-3,4-dihydro-spiro[isoquinoline-1,4'-piperidin]-2-yl]-N-(3,5-dichloro-phenyl)-acetamide 358374 1-(4-(2-((S)-1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(3,4-dimethylphenyl)-2-methylpropan-1-one 358375 1-(4-(2-((S)-1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(3-fluoro-4-methoxyphenyl)-2-methylpropan-1-one 358376 1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid 358377 1-(2-(4-fluorobenzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid 358378 1-(2-(4-chloro-3-(trifluoromethyl)benzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid 358379 1-(2-(4-tert-butylbenzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid 358381 6-(3-iodophenyl)-3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)thieno[3,2-d]pyrimidin-4(3H)-one 358382 (R)-1-(4-(2-((S)-1-amino-3-methylbutyl)phenyl)piperazin-1-yl)-3-(4-chloro-2-methylphenyl)-2-methylpropan-1-one 358383 (R)-1-(4-(2-((R)-1-amino-3-methylbutyl)phenyl)piperazin-1-yl)-3-(4-chloro-2-methylphenyl)-2-methylpropan-1-one 358388 [3-chloro-4-(3-fluoro-benzyloxy)-phenyl]-{6-[5-(1-oxo-1lambda*4*-thiomorpholin-4-ylmethyl)-furan-2-yl]-quinazolin-4-yl}-amine 358396 2-[6-(3-cyano-phenyl)-1'-(tetrahydro-thiophen-3-yl)-3,4-dihydro-spiro[isoquinoline-1,4'-piperidin]-2-yl]-N-(3,5-dichloro-phenyl)-acetamide 358401 2-(1-(1-cyclopentylpiperidin-4-yl)-6-(3-methoxyphenyl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358402 2-(1-(1-cyclopentylpiperidin-4-yl)-6-(3-(trifluoromethyl)phenyl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358403 2-(1-(1-cyclopentylpiperidin-4-yl)-6-(3-(trifluoromethoxy)phenyl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358405 N-(4-(benzyloxy)phenyl)-6-(5-((2-(methylsulfonyl)ethylamino)methyl)furan-2-yl)quinazolin-4-amine 358408 1-(4-(2-((S)-1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(4-chloro-3-methoxyphenyl)-2-methylpropan-1-one 358409 1-(4-(2-((S)-1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(3,4-dichlorophenyl)-2-methylpropan-1-one 358410 1-(2-(2-chlorobenzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid 358411 1-(2-(2-methoxybenzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid 358412 1-(2-(3,5-bis(trifluoromethyl)benzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid 358415 6-(2-chlorophenyl)-3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)thieno[3,2-d]pyrimidin-4(3H)-one 358416 3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-6-(pyridin-4-yl)thieno[3,2-d]pyrimidin-4(3H)-one 358430 (4-benzyloxy-3-fluoro-phenyl)-{6-[5-(1-oxo-1lambda*4*-thiomorpholin-4-ylmethyl)-furan-2-yl]-quinazolin-4-yl}-amine 358435 2-[1'-acetyl-6-(3-cyano-phenyl)-3,4-dihydro-spiro[isoquinoline-1,4'-piperidin]-2-yl]-N-(3,5-dichloro-phenyl)-acetamide 358437 4'-(4-fluorophenyl)-12'-methyl-1-propyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358448 N-(4-(3-fluorobenzyloxy)phenyl)-6-(5-((2-(methylsulfonyl)ethylamino)methyl)furan-2-yl)quinazolin-4-amine 358451 1-(4-(2-((S)-1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(2,4-dimethylphenyl)-2-methylpropan-1-one 358453 1-(2-(4-(trifluoromethyl)benzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid 358454 1-(2-(2,6-difluorobenzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid 358455 3-(2-aminoquinazolin-6-yl)-4-methyl-N-(2-methyl-3-(trifluoromethyl)phenyl)benzamide 358458 3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-6-(pyridin-3-yl)thieno[3,2-d]pyrimidin-4(3H)-one 358459 4-Methyl-3-(2-(methylamino)quinazolin-6-yl)-N-(3-(trifluoromethyl)phenyl)benzamide 358460 4-methyl-N-(2-methyl-3-4-methyl-N-(2-methyl-3-(2-(methylamino)quinazolin-6-yl)benzamide 358462 2-(6-(3-cyanophenyl)-1-(1-cyclohexylpiperidin-4-yl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358463 12'-bromo-4'-(2-chlorophenyl)-1-methyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358464 12'-bromo-4'-(2-methoxyphenyl)-1-methyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358465 (4-benzyloxy-3-chloro-phenyl)-{6-[5-(1-oxo-1lambda*4*-thiomorpholin-4-ylmethyl)-furan-2-yl]-quinazolin-4-yl}-amine 358472 12'-fluoro-4'-(4-fluorophenyl)-1-propyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358473 12'-chloro-4'-(4-fluorophenyl)-1-propyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358474 N-(3-chloro-4-fluoro-phenyl)-2-[6-(3-cyano-phenyl)-1'-cyclopropylmethyl-3,4-dihydro-spiro[isoquinoline-1,4'-piperidin]-2-yl]-acetamide 358477 2-(1-(1-cyclopentylpiperidin-4-yl)-6-(pyridin-4-yl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358478 sodium 2-(3-(((1S,2S)-2-(4,5-diphenyloxazol-2-yl)cyclohexyl)methyl)phenoxy)acetate 358479 sodium 2-(3-(((1S,2R)-2-(4,5-diphenyloxazol-2-yl)cyclohexyl)methyl)phenoxy)acetate 358481 YRFB 358484 1-(2-(3-bromobenzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid 358485 1-(2-(3-chlorobenzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid 358486 4-methyl-3-(2-(2-morpholinoethylamino)quinazolin-6-yl)-N-(3-(trifluoromethyl)phenyl)benzamide 358489 3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-6-(thiophen-3-yl)thieno[3,2-d]pyrimidin-4(3H)-one 358490 N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-4-{spiro[indene-1,4'-piperidine]-1'-yl}butanamide 358491 N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-4-[(1R,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]butanamide 358492 2-(1-(1-acetylpiperidin-4-yl)-6-(3-cyanophenyl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358493 12'-bromo-4'-(4-methoxyphenyl)-1-methyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358494 12'-bromo-4'-[2-(difluoromethoxy)phenyl]-1-methyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358500 12'-bromo-4'-(4-fluorophenyl)-1-propyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358501 4'-(2-chlorophenyl)-1-propyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358502 N-(4-chloro-phenyl)-2-[6-(3-cyano-phenyl)-1'-cyclopropylmethyl-3,4-dihydro-spiro[isoquinoline-1,4'-piperidin]-2-yl]-acetamide 358505 2-(1-(1-cyclopentylpiperidin-4-yl)-6-(pyridin-3-yl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358506 sodium 2-(3-(((1S,2S)-2-(4,5-diphenyloxazol-2-yl)cyclopentyl)methyl)phenoxy)acetate 358507 sodium 2-(3-(((1S,2R)-2-(4,5-diphenyloxazol-2-yl)cyclopentyl)methyl)phenoxy)acetate 358513 4-methyl-N-(2-methyl-3-(trifluoromethyl)phenyl)-3-(2-(2-morpholinoethylamino)quinazolin-6-yl)benzamide 358514 (1S)-(2-{4-[(2R)-methyl-3-(4-chlorophenyl)propionyl]-1-piperazinyl}-5-methylphenyl)-3-methylbutylamine 358515 (R)-1-(4-(2-((S)-1-amino-3-methylbutyl)-4-methylphenyl)piperazin-1-yl)-3-(4-chloro-2-methylphenyl)-2-methylpropan-1-one 358517 4-methyl-N-(2-methyl-3-(trifluoromethyl)phenyl)-3-(2-(phenylamino)quinazolin-6-yl)benzamide 358518 2-(6-(3-cyanophenyl)-1-(1-(methylsulfonyl)piperidin-4-yl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358520 N-(4-(3-fluorobenzyloxy)-3-(trifluoromethyl)phenyl)-6-(5-((2-(pyridin-2-ylsulfonyl)ethylamino)methyl)furan-2-yl)quinazolin-4-amine 358521 N-(4-(3-fluorobenzyloxy)-3-(trifluoromethyl)phenyl)-6-(5-((2-(1-methyl-1H-imidazol-2-ylsulfonyl)ethylamino)methyl)furan-2-yl)quinazolin-4-amine 358522 12'-bromo-4'-[4-(difluoromethoxy)phenyl]-1-methyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358523 12'-bromo-4'-(3,4-dichlorophenyl)-1-methyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358529 1-benzyl-4'-(4-chlorophenyl)-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358530 1-(2-phenylethyl)-4'-(pyridin-4-yl)-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358532 N-(3-chloro-phenyl)-2-[6-(3-cyano-phenyl)-1'-cyclopropylmethyl-3,4-dihydro-spiro[isoquinoline-1,4'-piperidin]-2-yl]-acetamide 358535 sodium (R)-2-(3-((2-(4,5-diphenyloxazol-2-yl)pyrrolidin-1-yl)methyl)phenoxy)acetate 358536 sodium (S)-2-(3-((2-(4,5-diphenyloxazol-2-yl)pyrrolidin-1-yl)methyl)phenoxy)acetate 358539 1-(2-(2,4-dichlorobenzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid 358540 1-(2-(2,4-difluorobenzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid 358541 1-(4-methyl-3-(2-(methylamino)quinazolin-6-yl)phenyl)-3-(3-(trifluoromethyl)phenyl)urea 358542 4-(3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-4-oxo-3,4-dihydrothieno[3,2-d]pyrimidin-6-yl)benzonitrile 358543 3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-6-(4-(methylsulfonyl)phenyl)thieno[3,2-d]pyrimidin-4(3H)-one 358544 (R)-1-(4-(2-((S)-1-amino-3-methylbutyl)-4-methylphenyl)piperazin-1-yl)-3-(4-chloro-2-fluorophenyl)-2-methylpropan-1-one 358545 (R)-1-(4-(2-((S)-1-amino-3-methylbutyl)-4-methylphenyl)piperazin-1-yl)-3-(4-chloro-2-methoxyphenyl)-2-methylpropan-1-one 358550 12'-bromo-4'-(3,4-dimethoxyphenyl)-1-methyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358551 TCMDC-138529 358558 1-ethyl-4'-(pyridin-4-yl)-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358561 2-[6-(3-cyano-phenyl)-1'-cyclopropylmethyl-3,4-dihydro-spiro[isoquinoline-1,4'-piperidin]-2-yl]-N-(3,4-difluoro-phenyl)-acetamide 358567 ((R)-4-bromo-3,6-dimethoxybenzocyclobuten-1-yl)methylamine 358569 ((S)-4-bromo-3,6-dimethoxybenzocyclobuten-1-yl)methylamine 358571 5-(2-aminoquinazolin-6-yl)-2-fluoro-4-methyl-N-(3-(trifluoromethyl)phenyl)benzamide 358572 N-methyl-6-(2-methyl-5-(5-(trifluoromethyl)-1Hbenzo[d]imidazol-2-ylamino)phenyl)quinazolin-2-amine 358573 6-o-tolylquinazolin-2-amine 358574 3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-6-(4-nitrophenyl)thieno[3,2-d]pyrimidin-4(3H)-one 358575 N-(4-(3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-4-oxo-3,4-dihydrothieno[3,2-d]pyrimidin-6-yl)phenyl)acetamide 358578 4-methyl-3-(2-(methyl(3-morpholinopropyl)amino)quinazolin-6-yl)-N-(2-methyl-3-(trifluoromethyl)phenyl)benzamide 358580 1-methyl-4'-phenyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358581 12'-bromo-1-methyl-4'-phenyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358589 1-(2-methylpropyl)-4'-(pyridin-4-yl)-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358590 12'-bromo-4'-phenyl-1-(propan-2-yl)-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358597 2-[6-(3-cyano-phenyl)-1'-cyclopropylmethyl-3,4-dihydro-spiro[isoquinoline-1,4'-piperidin]-2-yl]-N-(4-fluoro-3-trifluoromethyl-phenyl)-acetamide 358598 2-[6-(3-cyano-phenyl)-1'-cyclopropylmethyl-3,4-dihydro-spiro[isoquinoline-1,4'-piperidin]-2-yl]-N-(3-fluoro-5-trifluoromethyl-phenyl)-acetamide 358599 2-(6-(3-cyanophenyl)-1-(1-cyclopentylpiperidin-4-yl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358600 2-(6-(4-cyanophenyl)-1-(1-cyclopentylpiperidin-4-yl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358602 2-(1-(1-cyclopentylpiperidin-4-yl)-6-(3-fluorophenyl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358617 3-(2-aminoquinazolin-6-yl)-2-methyl-N-(3-(trifluoromethyl)phenyl)benzamide 358618 3-(2-aminoquinazolin-6-yl)-4-methyl-N-(3-(trifluoromethyl)phenyl)benzamide 358619 6-(4-fluorophenyl)-3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)thieno[3,2-d]pyrimidin-4(3H)-one 358620 6-(3-chlorophenyl)-3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)thieno[3,2-d]pyrimidin-4(3H)-one 358621 6-(3,4-dichlorophenyl)-3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)thieno[3,2-d]pyrimidin-4(3H)-one 358622 4-methyl-N-(2-methyl-3-(trifluoromethyl)phenyl)-3-(2-(2-(piperidin-1-yl)ethylamino)quinazolin-6-yl)benzamide 358625 4'-(4-chlorophenyl)-1-methyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358630 4'-(4-chlorophenyl)-1-(propan-2-yl)-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358636 2-(6-(3-chlorophenyl)-1-(1-cyclopentylpiperidin-4-yl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358640 C-(5-bromo-4,7-dimethoxyindan-1-yl)methylamine 358641 C-(3-bromo-5-methoxy-1,6,7,8,9,9a-hexahydro-2-oxabenzo-[cd]azulen-6-yl)methylamine 358643 N-(4-(3-(trifluoromethyl)benzyloxy)phenyl)-6-(5-((2-(methylsulfonyl)ethylamino)methyl)furan-2-yl)quinazolin-4-amine 358648 6-(4-chlorophenyl)-3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)thieno[3,2-d]pyrimidin-4(3H)-one 358650 1-(4-(2-((S)-1-amino-3-methylbutyl)-4-chlorophenyl)piperazin-1-yl)-3-(4-chloro-2-methoxyphenyl)-2-methylpropan-1-one 358651 4-methyl-N-(2-methyl-3-(trifluoromethyl)phenyl)-3-(2-(2-(pyrrolidin-1-yl)ethylamino)quinazolin-6-yl)benzamide 358652 2-(6-(3-cyanophenyl)-1-(1-(furan-3-ylmethyl)piperidin-4-yl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358653 4'-(4-bromophenyl)-1-methyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358670 sodium 2-(3-(2-(4,5-diphenyloxazol-2-yl)benzyl)phenoxy)acetate 358671 N-(4-(3-bromobenzyloxy)phenyl)-6-(5-((2-(methylsulfonyl)ethylamino)methyl)furan-2-yl)quinazolin-4-amine 358672 (3-chloro-2-fluoro-phenyl)-(7,8-dimethoxy-10,11-dihydro-5-thia-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 358673 (7,8-dimethoxy-10,11-dihydro-5-thia-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-(1H-indazol-6-yl)-amine 358674 N-(4-methyl-3-(2-(methylamino)quinazolin-6-yl)phenyl)-3-(trifluoromethyl)benzamide 358677 3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-6-(4-methoxyphenyl)thieno[3,2-d]pyrimidin-4(3H)-one 358678 3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-6-(4-(trifluoromethyl)phenyl)thieno[3,2-d]pyrimidin-4(3H)-one 358680 1-(4-(2-((S)-1-amino-3-methylbutyl)-4-fluorophenyl)piperazin-1-yl)-3-(4-chlorophenyl)-2-methylpropan-1-one 358681 4-methyl-N-(2-methyl-3-(trifluoromethyl)phenyl)-3-(2-(1-methylpiperidin-4-ylamino)quinazolin-6-yl)benzamide 358682 2-(1-(1-(2-methoxybenzyl)piperidin-4-yl)-6-(3-cyanophenyl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358683 2-(6-(3-cyanophenyl)-1-(1-(cyclopropylmethyl)piperidin-4-yl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358684 12'-bromo-4'-(4-chlorophenyl)-1-methyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358685 4'-(2-chlorophenyl)-1-methyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358689 4'-(4-chlorophenyl)-10'-methoxy-1-methyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358701 2-(1-(1-cyclopentylpiperidin-4-yl)-6-(1H-pyrrol-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358702 N-(4-(benzyloxy)-3-chlorophenyl)-6-(5-((2-(methylsulfonyl)ethylamino)methyl)furan-2-yl)quinazolin-4-amine 358708 6-(4-aminophenyl)-3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)thieno[3,2-d]pyrimidin-4(3H)-one 358709 (S)-1-(4-(2-((S)-1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(4-chloro-2-methoxyphenyl)-2-methylpropan-1-one 358710 1-(2-(2,4-dichlorobenzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid 358712 4-methyl-N-(2-methyl-3-(trifluoromethyl)phenyl)-3-(2-(phenylamino)quinazolin-6-yl)benzamide 358713 3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-6-(thiophen-2-yl)thieno[3,2-d]pyrimidin-4(3H)-one 358714 2-(6-(3-cyanophenyl)-1-(1-cyclobutylpiperidin-4-yl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358718 4'-(4-bromophenyl)-10'-methoxy-1-methyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358719 4,4-dimethyl-2-pyridin-4-yl-1,9b-dihydro-5-oxa-3,3a-diaza-cyclopenta[a]naphthalene 358726 2-[6-(3-cyano-phenyl)-1'-cyclopropylmethyl-3,4-dihydro-spiro[isoquinoline-1,4'-piperidin]-2-yl]-N-(3,5-difluoro-phenyl)-acetamide 358730 2-(1-(1-cyclopentylpiperidin-4-yl)-6-(thiophen-3-yl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358731 N-(4-(benzyloxy)-3-bromophenyl)-6-(5-((2-(methylsulfonyl)ethylamino)methyl)furan-2-yl)quinazolin-4-amine 358732 (3-chloro-phenyl)-(7,8-dimethoxy-10,11-dihydro-5-thia-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-methyl-amine 358733 (3-bromo-phenyl)-(7,8-dimethoxy-3-methyl-10,11-dihydro-5-thia-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 358738 (R)-1-(4-(2-((S)-1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(2,4-dichlorophenyl)-2-methylpropan-1-one 358739 1-(2-(2,4-difluorobenzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid 358741 3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)thieno[3,2-d]pyrimidin-4(3H)-one 358742 6-(4-chlorophenyl)-3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)furo[3,2-d]pyrimidin-4(3H)-one 358743 2-(6-(3-cyanophenyl)-1-(1-isopropylpiperidin-4-yl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358744 C-(3-bromo-5-methoxy-1,6,7,8,9,9a-hexahydro-2-oxabenzo-[cd]azulen-6-yl)methylamine 358757 2-[6-(3-cyano-phenyl)-1'-cyclopropylmethyl-3,4-dihydro-spiro[isoquinoline-1,4'-piperidin]-2-yl]-N-(3,4-dichloro-phenyl)-acetamide 358763 2-(6-(3-cyanophenyl)-1-(piperidin-4-yl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358764 2-(6-(3-cyanophenyl)-1-(1-methylpiperidin-4-yl)-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358765 N-(4-(3-fluorobenzyloxy)-3-methoxyphenyl)-6-(5-((2-(methylsulfonyl)ethylamino)methyl)furan-2-yl)quinazolin-4-amine 358769 3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-6-phenylthieno[3,2-d]pyrimidin-4(3H)-one 358771 (S)-1-(4-(2-((S)-1-amino-3-methylbutyl)-4-(trifluoromethyl)phenyl)piperazin-1-yl)-3-(2,4-dichlorophenyl)-2-methylpropan-1-one 358772 1-(2-(2,4-dichlorobenzyloxy)benzyl)-5-methyl-1H-pyrazole-3-carboxylic acid 358773 1-(2-(2,4-dichlorobenzyloxy)-5-fluorobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid 358774 7-(4-chlorophenyl)-3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)quinazolin-4(3H)-one 358775 2-(4-chlorophenyl)-6-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)thiazolo[4,5-d]pyrimidin-7(6H)-one 358783 N-(4-(3-fluorobenzyloxy)-3-chlorophenyl)-6-(5-((benzyl(2-(methylsulfonyl)ethyl)amino)methyl)furan-2-yl)quinazolin-4-amine 358784 [4-(3-fluoro-benzyloxy)-3-trifluoromethyl-phenyl]-{6-[5-(1-oxo-1lambda*4*-thiomorpholin-4-ylmethyl)-furan-2-yl]-quinazolin-4-yl}-amine 358789 12'-bromo-4'-(4-methylphenyl)-1-propyl-8'-oxa-5',6'-diazaspiro[piperidine-4,7'-tricyclo[7.4.0.0^{2,6}]tridecane]-1'(13'),4',9',11'-tetraene 358793 2-(1-(1-cyclopentylpiperidin-4-yl)-6-phenyl-3,4-dihydroisoquinolin-2(1H)-yl)-N-(3,5-dichlorophenyl)acetamide 358807 4-cyclohexyl-N-(4-(2-(diisopropylamino)ethoxy)-3-methoxyphenyl)benzamide 358808 2-methyl-biphenyl-4-carboxylic acid [4-(2-diisopropylamino-ethoxy)-3-methoxy-phenyl]-amide 358809 4'-methoxy-2'-methyl-biphenyl-4-carboxylic acid {(S)-1-[(R)-3-(3-cyclohexyl-propylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-methyl-amide 358810 N-(3-dimethylaminomethyl-quinolin-8-ylmethyl)-6-(4-fluoro-phenyl)-nicotinamide 358814 biphenyl-4-carboxylic acid [3-methoxy-4-(2-pyrrolidin-1-yl-ethoxy)-phenyl]-methyl-amide 358815 4-cyclohexyl-N-(4-(2-(diisopropylamino)ethoxy)-3-methoxyphenyl)-N-methylbenzamide 358822 3-amino-N-(1-phenethylpiperidin-4-yl)-N-phenylpropanamide 358823 3-(1,3-dioxoisoindolin-2-yl)-N-(1-phenethylpiperidin-4-yl)-N-phenylpropanamide 358835 N-(4-(2-(diisopropylamino)ethoxy)phenyl)-N-methyl-9H-fluorene-2-carboxamide 358838 (7,8-dimethoxy-3-methyl-10,11-dihydro-5-thia-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-(3H-indazol-5-yl)-amine 358839 1-(3-bromo-phenoxy)-7,8-dimethoxy-10,11-dihydro-5-thia-2,4,11-triaza-dibenzo[a,d]cycloheptene 358840 4'-ethyl-biphenyl-4-carboxylic acid {(S)-1-[(R)-3-(3-cyclohexyl-propylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-methyl-amide 358845 4-benzyl-N-(4-(2-(diisopropylamino)ethoxy)-3-methoxyphenyl)-N-methylbenzamide 358846 N-(4-(2-(diisopropylamino)ethoxy)-3-methoxyphenyl)-N-methyl-3-phenoxybenzamide 358847 N-(5-chloro-2-fluorophenyl)-7-methoxy-6-(3-morpholinopropoxy)quinazolin-4-amine 358848 N-(3-chloro-2-fluorophenyl)-7-methoxy-6-((1-methylpiperidin-4-yl)methoxy)quinazolin-4-amine 358854 3-acetamido-N-(1-phenethylpiperidin-4-yl)-N-phenylpropanamide 358855 N-(1-phenethyl-piperidin-4-yl)-N-phenyl-3-propionylamino-propionamide 358880 biphenyl-4-carboxylic acid [4-(2-diethylamino-ethoxy)-3-methoxy-phenyl]-ethyl-amide 358881 (7,8-dimethoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-m-tolyl-amine 358882 N-(3-chloro-2-fluorophenyl)-7-methoxy-6-(1-methylpiperidin-4-yloxy)quinazolin-4-amine 358888 7-(3-bromophenoxy)-13,14-dimethoxy-9-methyl-2-oxa-4,6,9-triazatricyclo[9.4.0.0^{3,8}]pentadeca-1(11),3,5,7,12,14-hexaene 358889 1-(3-chloro-2-fluoro-phenoxy)-7,8-dimethoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cycloheptene 358894 22-hydroxy-15-oxa-8-thia-9,12,21,23-tetraazapentacyclo[14.6.2.1^{6,9}.0^{2,7}.0^{20,24}]pentacosa-1(23),2(7),3,5,16(24),17,19,21-octaen-25-one 358901 Ac-RYYRIK-K-(NH2)-YRFB 358902 Ac-RYYRIK-GGG-K-(NH2)-YRFB-GGGGG 358925 N-(3-chloro-4-fluorophenyl)-7-methoxy-6-((1-methylpiperidin-4-yl)methoxy)quinazolin-4-amine 358926 N-(3-chloro-4-fluorophenyl)-7-methoxy-6-(1-methylpiperidin-4-yloxy)quinazolin-4-amine 358931 2-(2-((3R,3aS,4S,4aR,8aS,9aR)-3-methyl-dodecahydronaphtho[2,3-c]furan-4-yl)vinyl)-5-(3-(trifluoromethyl)phenyl)pyridine 358933 1-(3-chloro-4-fluoro-phenoxy)-7,8-dimethoxy-11-methyl-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cycloheptene 358934 1-(3-bromo-phenylsulfanyl)-7,8-dimethoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cycloheptene 358946 3'-trifluoromethyl-biphenyl-4-carboxylic acid [4-(2-diisopropylamino-ethoxy)-3-methoxy-phenyl]-amide 358947 benzothiazol-6-yl-(7,8-dimethoxy-3-methyl-10,11-dihydro-5-thia-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 358948 4'-fluoro-biphenyl-4-carboxylic acid (3-diethylaminomethyl-quinolin-8-ylmethyl)-amide 358949 4'-fluoro-biphenyl-4-carboxylic acid (3-morpholin-4-ylmethyl-quinolin-8-ylmethyl)-amide 358954 biphenyl-4-carboxylic acid [3-acetyl-4-(2-diethylamino-ethoxy)-phenyl]-amide 358955 biphenyl-4-carboxylic acid [4-(2-diethylamino-ethoxy)-3-(1-hydroxy-ethyl)-phenyl]-amide 358963 2-(2-((1S,4aS,8aR)-decahydronaphthalen-1-yl)vinyl)-6-methoxyquinoline 358964 1-(3-chloro-phenylsulfanyl)-7,8-dimethoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cycloheptene 358965 (3-bromo-phenyl)-(7,8-dimethoxy-10,11-dihydro-5-thia-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 358977 (R)-4-cyclohexyl-N-(3-methoxy-4-((1-methylpyrrolidin-2-yl)methoxy)phenyl)benzamide 358982 2'-methyl-biphenyl-4-carboxylic acid [4-(2-diisopropylamino-ethoxy)-3-methoxy-phenyl]-amide 358983 (7,8-dimethoxy-3-methyl-10,11-dihydro-5-thia-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-(1H-indazol-6-yl)-amine 358990 biphenyl-4-carboxylic acid {4-[2-(benzyl-methyl-amino)-ethoxy]-3-methoxy-phenyl}-amide 358991 biphenyl-4-carboxylic acid [3-methoxy-4-(2-pyrrolidin-1-yl-ethoxy)-phenyl]-amide 358992 biphenyl-4-carboxylic acid [4-(2-diethylamino-ethoxy)-3-ethyl-phenyl]-amide 359002 (2-chloro-4-fluoro-phenyl)-(7,8-dimethoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 359003 (3-chloro-4-fluoro-phenyl)-(7,8-dimethoxy-10,11-dihydro-5-thia-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 359021 (S)-4-cyclohexyl-N-(3-methoxy-4-((1-methylpyrrolidin-2-yl)methoxy)phenyl)benzamide 359022 4-cyclohexyl-N-(4-((1S,2S)-2-(dimethylamino)cyclohexyloxy)-3-methoxyphenyl)benzamide 359027 Ac-Phe-[Orn-Pro-cha-Trp-Cha] 359028 Ac-Phe-[Orn-Pro-cha-Trp-Hch] 359029 Ac-Phe-[Orn-Pro-cha-Trp-Ocg] 359035 Ac-Phe-[Orn-Pro-cha-Trp-nle] 359044 biphenyl-4-carboxylic acid [3-methoxy-4-(2-piperidin-1-yl-ethoxy)-phenyl]-amide 359045 biphenyl-4-carboxylic acid [4-(2-diisopropylamino-ethoxy)-phenyl]-amide 359047 biphenyl-4-carboxylic acid [4-(2-diisopropylamino-ethoxy)-3-methoxy-phenyl]-methyl-amide 359048 (3R,3aS,4S,4aS,9aR)-3-ethyl-4-(2-(quinolin-2-yl)vinyl)-3,3a,4,4a,5,6,7,8-octahydronaphtho[2,3-c]furan-1(9aH)-one 359049 (3aS,4S,4aS,9aR)-4-(2-(quinolin-2-yl)vinyl)-3,3a,4,4a,5,6,7,8-octahydronaphtho[2,3-c]furan-1(9aH)-one 359056 (7,8-dimethoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-(1H-indazol-6-yl)-amine 359057 (7,8-dimethoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-naphthalen-2-yl-amine 359068 N-(4-(1-aza-bicyclo[3.2.1]octan-5-yloxy)-3-methoxyphenyl)-4-cyclohexylbenzamide 359069 4-cyclohexyl-N-(4-(4-ethylpiperazin-1-yloxy)-3-methoxyphenyl)benzamide 359079 3-methyl-biphenyl-4-carboxylic acid [4-(2-diisopropylamino-ethoxy)-3-methoxy-phenyl]-amide 359080 (7,8-dimethoxy-10,11-dihydro-5H-2,4,5,11-tetraaza-dibenzo[a,d]cyclohepten-1-yl)-((R)-1-phenyl-ethyl)-amine 359081 biphenyl-4-carboxylic acid [4-(2-diisopropylamino-ethoxy)-3-methyl-phenyl]-amide 359082 biphenyl-4-carboxylic acid [4-(2-diisopropylamino-ethoxy)-3-fluoro-phenyl]-amide 359083 biphenyl-4-carboxylic acid [4-(2-diethylamino-ethoxy)-3-methoxy-phenyl]-methyl-amide 359086 (3aS,4S,4aS,9aR)-3,3-dimethyl-4-(2-(quinolin-2-yl)vinyl)-3,3a,4,4a,5,6,7,8-octahydronaphtho[2,3-c]furan-1(9aH)-one 359087 (1R,3R,3aS,4S,4aR,8aS,9aR)-4-(2-(6-ethylpyridin-2-yl)vinyl)-3-methyl-dodecahydronaphtho[2,3-c]furan-1-ol 359092 6-methoxy-2-(2-((3R,3aS,4S,4aR,8aS,9aR)-3-methyl-dodecahydronaphtho[2,3-c]furan-4-yl)vinyl)quinoline 359093 benzothiazol-6-yl-(7,8-dimethoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 359099 21-hydroxy-14-oxa-8-thia-9,20,22-triazapentacyclo[13.6.2.1^{6,9}.0^{2,7}.0^{19,23}]tetracosa-1(22),2,4,6,15(23),16,18,20-octaen-24-one 359107 N-(4-(2-(diisopropylamino)ethoxy)phenyl)-9-oxo-9H-fluorene-2-carboxamide 359108 N-(4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-9H-fluorene-2-carboxamide 359109 (3-chloro-4-fluoro-phenyl)-(7,8-dimethoxy-3-methyl-10,11-dihydro-5-thia-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 359115 4'-trifluoromethyl-biphenyl-4-carboxylic acid [4-(2-diisopropylamino-ethoxy)-3-methoxy-phenyl]-amide 359116 3-benzyl-N-(4-(2-(diisopropylamino)ethoxy)-3-methoxyphenyl)benzamide 359117 biphenyl-4-carboxylic acid [4-(2-diisopropylamino-ethoxy)-2-methyl-phenyl]-amide 359118 6-(4-fluoro-phenyl)-N-[3-((S)-3-hydroxy-pyrrolidin-1-ylmethyl)-quinolin-8-ylmethyl]-nicotinamide 359122 (1R,3R,3aS,4S,4aR,8aS,9aR)-3-methyl-4-(2-(quinolin-2-yl)vinyl)-dodecahydronaphtho[2,3-c]furan-1-ol 359136 N-(3-chloro-2-fluorophenyl)-7-methoxy-6-(1-(methylsulfonyl)piperidin-4-yloxy)quinazolin-4-amine 359137 N-(5-chloro-2-fluorophenyl)-7-methoxy-6-(1-(2-methoxyethyl)piperidin-4-yloxy)quinazolin-4-amine 359139 1-(3-bromo-phenoxy)-7,8-dimethoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cycloheptene 359144 22-hydroxy-15-oxa-8-thia-9,21,23-triazapentacyclo[14.6.2.1^{6,9}.0^{2,7}.0^{20,24}]pentacosa-1(23),2(7),3,5,16(24),17,19,21-octaen-25-one 359154 (7,8-dimethoxy-3-methyl-10,11-dihydro-5-thia-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-naphthalen-2-yl-amine 359158 biphenyl-4-carboxylic acid [4-(2-diisopropylamino-ethoxy)-3-methoxy-phenyl]-amide 359159 biphenyl-4-carboxylic acid [4-(2-dimethylamino-ethoxy)-3-methoxy-phenyl]-amide 359160 N-((S)-1-((R)-3-(3-cyclohexylpropylamino)pyrrolidine-1-carbonyl)pyrrolidin-3-yl)-N-methyl-5-(4-(trifluoromethyl)phenyl)thiophene-2-carboxamide 359165 N-(3-chloro-2-fluorophenyl)-7-methoxy-6-(3-morpholinopropoxy)quinazolin-4-amine 359166 (R)-1-((1S,2S,3R,4aS,8aR)-3-(hydroxymethyl)-1-(2-(5-(3-(trifluoromethyl)phenyl)pyridin-2-yl)vinyl)-decahydronaphthalen-2-yl)ethanol 359168 2-(4-(4-(5-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yloxy)piperidin-1-yl)acetamide 359169 N-(5-chloro-2-fluorophenyl)-7-methoxy-6-(1-(methylsulfonyl)piperidin-4-yloxy)quinazolin-4-amine 359175 23-hydroxy-16-oxa-8-thia-9,22,24-triazapentacyclo[15.6.2.1^{6,9}.0^{2,7}.0^{21,25}]hexacosa-1(24),2(7),3,5,17(25),18,20,22-octaen-26-one 359177 (15S)-16-oxa-8,9,12,22,24-pentaazahexacyclo[15.6.2.1^{6,9}.1^{12,15}.0^{2,7}.0^{21,25}]heptacosa-1(24),2,4,6(27),7,17(25),18,20,22-nonaene-23,27-diol 359178 (13R,15S)-13-methyl-16-oxa-8,9,12,22,24-pentaazahexacyclo[15.6.2.1^{6,9}.1^{12,15}.0^{2,7}.0^{21,25}]heptacosa-1(24),2,4,6(27),7,17(25),18,20,22-nonaene-23,27-diol 359184 biphenyl-3-carboxylic acid [4-(2-diisopropylamino-ethoxy)-3-methoxy-phenyl]-amide 359190 biphenyl-4-carboxylic acid [4-(2-diethylamino-ethoxy)-3-methoxy-phenyl]-amide 359191 N-(3-diethylaminomethyl-quinolin-8-ylmethyl)-6-(4-fluoro-phenyl)-nicotinamide 359192 6-(4-fluoro-phenyl)-N-[3-(4-methyl-piperazin-1-ylmethyl)-quinolin-8-ylmethyl]-nicotinamide 359193 4'-fluoro-biphenyl-4-carboxylic acid methyl-(3-piperidin-1-ylmethyl-quinolin-8-ylmethyl)-amide 359195 6-(2,6-Dichlorophenyl)-8-methyl-2-(3-(methylthio)phenylamino)pyrido[2,3-d]pyrimidin-7(8H)-one 359199 2-(2-((1R,3R,3aS,4S,4aR,8aS,9aR)-1-methoxy-3-methyl-dodecahydronaphtho[2,3-c]furan-4-yl)vinyl)quinoline 359201 (3-chloro-2-fluoro-phenyl)-(7,8-dimethoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 359207 Ac-RYYRIK-NH2 359220 (1H-benzoimidazol-5-yl)-(7,8-dimethoxy-3-methyl-10,11-dihydro-5-thia-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 359224 1-(3-chloro-2-fluoro-phenoxy)-7,8-dimethoxy-10,11-dihydro-5-thia-2,4,11-triaza-dibenzo[a,d]cycloheptene 359225 1-(3-bromo-phenylsulfanyl)-7,8-dimethoxy-10,11-dihydro-5-thia-2,4,11-triaza-dibenzo[a,d]cycloheptene 359226 6-(4-fluoro-phenyl)-N-(3-morpholin-4-ylmethyl-quinolin-8-ylmethyl)-nicotinamide 359227 N-((S)-1-((R)-3-(4,4-dimethylcyclohexylamino)pyrrolidine-1-carbonyl)pyrrolidin-3-yl)-5-(4-ethylphenyl)-N-methylthiophene-2-carboxamide 359232 6-methoxy-2-(2-((1R,3R,3aS,4S,4aR,8aS,9aR)-1-methoxy-3-methyl-dodecahydronaphtho[2,3-c]furan-4-yl)vinyl)quinoline 359234 (5-chloro-2-fluoro-phenyl)-(7,8-dimethoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 359239 N-(1-phenethylpiperidin-4-yl)-N-phenyl-3-(2,2,2-trifluoroacetamido)propanamide 359240 1-ethyl-3-(3-oxo-3-((1-phenethylpiperidin-4-yl)(phenyl)amino)propyl)urea 359241 (S)-2-amino-3-(4-hydroxy-phenyl)-N-((R)-1-{[((S)-1-{2-[(1-phenethyl-piperidin-4-yl)-phenyl-carbamoyl]-ethylcarbamoyl}-2-phenyl-ethylcarbamoyl)-methyl]-carbamoyl}-ethyl)-propionamide 359249 4-cyclohexyl-N-(3-methoxy-4-(1-methylpyrrolidin-3-yloxy)phenyl)benzamide 359258 1-(3-chloro-phenylsulfanyl)-7,8-dimethoxy-10,11-dihydro-5-thia-2,4,11-triaza-dibenzo[a,d]cycloheptene 359259 (3-bromo-phenyl)-(7,8-dimethoxy-10,11-dihydro-5H-2,4,5,11-tetraaza-dibenzo[a,d]cyclohepten-1-yl)-amine 359260 N-((S)-1-((R)-3-(3-cyclohexylpropylamino)pyrrolidine-1-carbonyl)pyrrolidin-3-yl)-5-(4-methoxy-2-methylphenyl)-N-methylthiophene-2-carboxamide 359261 N-((S)-1-((R)-3-(4,4-dimethylcyclohexylamino)pyrrolidine-1-carbonyl)pyrrolidin-3-yl)-5-(4-methoxyphenyl)-N-methylthiophene-2-carboxamide 359266 2-(2-((3R,3aS,4S,4aR,8aS,9aR)-3-methyl-dodecahydronaphtho[2,3-c]furan-4-yl)vinyl)quinoline 359267 N-(5-chloro-2-fluorophenyl)-7-methoxy-6-((1-methylpiperidin-4-yl)methoxy)quinazolin-4-amine 359273 2-acetylamino-N-{2-[(1-phenethyl-piperidin-4-yl)-phenyl-carbamoyl]-ethyl}-3-phenyl-propionamide 359274 N-(1-phenethyl-piperidin-4-yl)-N-phenyl-succinamic acid 359290 (3-chloro-4-fluoro-benzyl)-(7,8-dimethoxy-10,11-dihydro-5H-2,4,5,11-tetraaza-dibenzo[a,d]cyclohepten-1-yl)-amine 359291 (7,8-dimethoxy-10,11-dihydro-5H-2,4,5,11-tetraaza-dibenzo[a,d]cyclohepten-1-yl)-(3-methoxy-benzyl)-amine 359292 6-(4-fluoro-phenyl)-N-[3-(4-hydroxy-piperidin-1-ylmethyl)-quinolin-8-ylmethyl]-nicotinamide 359295 (3R,3aS,4S,4aS,9aR,E)-3-methyl-4-(2-(quinolin-2-yl)vinyl)-3,3a,4,4a,5,6,7,8-octahydronaphtho[2,3-c]furan-1(9aH)-one 359296 (1R,3R,3aS,4S,4aR,8aS,9aR)-4-(2-(6-methoxyquinolin-2-yl)vinyl)-3-methyl-dodecahydronaphtho[2,3-c]furan-1-ol 359298 (7,8-dimethoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-(3-ethynyl-phenyl)-amine 359299 (4-bromo-phenyl)-(7,8-dimethoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-amine 359324 N-(4-(2-(diisopropylamino)ethoxy)-3-methoxyphenyl)-4-phenoxybenzamide 359325 benzyl-(7,8-dimethoxy-10,11-dihydro-5H-2,4,5,11-tetraaza-dibenzo[a,d]cyclohepten-1-yl)-amine 359326 4'-fluoro-biphenyl-4-carboxylic acid [3-(4-hydroxy-piperidin-1-ylmethyl)-quinolin-8-ylmethyl]-amide 359327 N-((S)-1-((R)-3-(3-cyclohexylpropylamino)pyrrolidine-1-carbonyl)pyrrolidin-3-yl)-5-(4-ethylphenyl)-N-methylthiophene-2-carboxamide 359334 (R)-1-((1S,2S,3R,4aS,8aR)-1-(2-(6-ethylpyridin-2-yl)vinyl)-3-(hydroxymethyl)-decahydronaphthalen-2-yl)ethanol 359339 N-(5-chloro-2-fluorophenyl)-7-methoxy-6-(1-methylpiperidin-4-yloxy)quinazolin-4-amine 359340 N-(3-chloro-2-fluorophenyl)-7-methoxy-6-(1-(2-methoxyethyl)piperidin-4-yloxy)quinazolin-4-amine 359347 (1R,3R,3aS,4R,5aS,9aR,9bS)-3-methyl-1-(quinolin-2-ylmethyl)-dodecahydronaphtho[2,1-c]furan-4-carboxylic acid 359358 4-(3,4-dimethylphenoxy)-3-(3-phenylpropanamido)-N-(2-(pyrrolidin-1-yl)ethyl)benzamide 359360 Ac-Ala-[Orn-Pro-cha-Trp-Eag] 359361 Ac-Phe-[Orn-Pro-cha-Trp-Phe] 359364 N-(4-(2-(diisopropylamino)ethoxy)-3-methoxyphenyl)-3-phenoxybenzamide 359366 4'-fluoro-biphenyl-4-carboxylic acid [3-((S)-3-hydroxy-pyrrolidin-1-ylmethyl)-quinolin-8-ylmethyl]-amide 359367 4'-fluoro-biphenyl-4-carboxylic acid [3-(4-methanesulfonyl-piperidin-1-ylmethyl)-quinolin-8-ylmethyl]-amide 359372 (R)-1-((1S,2S,3R,4aS,8aR)-3-(hydroxymethyl)-1-(2-(6-methoxyquinolin-2-yl)vinyl)-decahydronaphthalen-2-yl)ethanol 359373 2-(4-(4-(3-chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yloxy)piperidin-1-yl)acetamide 359374 (7,8-dimethoxy-10,11-dihydro-5-oxa-2,4,11-triaza-dibenzo[a,d]cyclohepten-1-yl)-(4-fluoro-phenyl)-amine 359393 6-(4-chlorophenyl)-3-(2-(4-methylpiperazin-1-yl)-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359395 3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-7-phenylquinazolin-4(3H)-one 359397 N-((S)-1-((R)-3-(4,4-dimethylcyclohexylamino)pyrrolidine-1-carbonyl)pyrrolidin-3-yl)-N-methyl-5-phenylthiophene-2-carboxamide 359401 4'-ethyl-biphenyl-4-carboxylic acid {(S)-1-[(R)-3-((S)-1,2-dimethyl-propylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-methyl-amide 359404 9-(3-oxo-3,4-dihydro-quinoxalin-2-yl)-1,2,3,9b-tetrahydro-pyrrolo[2,1-a]isoindol-5-one 359434 1-(2-(3,4-dimethylphenoxy)-5-((2-(pyrrolidin-1-yl)ethyl)carbamoyl)phenyl)-3-(3-fluorophenyl)urea 359435 6-(4-chlorophenyl)-3-(1-(4-(dimethylamino)phenyl)-2-methyl-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359442 N-((S)-1-((R)-3-(4,4-dimethylcyclohexylamino)pyrrolidine-1-carbonyl)pyrrolidin-3-yl)-N-methyl-5-(4-(trifluoromethyl)phenyl)furan-2-carboxamide 359443 4'-ethyl-biphenyl-4-carboxylic acid [(S)-1-((R)-3-amino-pyrrolidine-1-carbonyl)-pyrrolidin-3-yl]-methyl-amide 359448 4'-ethyl-biphenyl-4-carboxylic acid {(S)-1-[(R)-3-((S)-2-methoxy-1-methyl-ethylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-methyl-amide 359450 3-(2-cyclopentyl-1-oxo-2,3-dihydro-1H-isoindol-4-yl)-1H-quinoxalin-2-one 359460 3-(3-biphenyl-4-yl-ureido)-4-(3,4-dimethyl-phenoxy)-N-(2-pyrrolidin-1-yl-ethyl)-benzamide 359461 1-(2-(3,4-dimethylphenoxy)-5-((2-(pyrrolidin-1-yl)ethyl)carbamoyl)phenyl)-3-(4-phenoxyphenyl)urea 359470 N-(4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-9,10-dihydrophenanthrene-2-carboxamide 359471 N-(4-(2-(diisopropylamino)ethoxy)phenyl)-N-methyl-9,10-dihydrophenanthrene-2-carboxamide 359474 N-((S)-1-((R)-3-(cyclopentylamino)pyrrolidine-1-carbonyl)pyrrolidin-3-yl)-5-(4-ethylphenyl)-N-methylthiophene-2-carboxamide 359475 4'-ethyl-biphenyl-4-carboxylic acid methyl-{(S)-1-[(R)-3-(tetrahydro-pyran-4-ylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-amide 359481 3-(2-cyclopentyl-3-oxo-2,3-dihydro-benzo[d]isothiazol-7-yl)-1H-quinoxalin-2-one 359496 6-(4-chlorophenyl)-3-(1-cyclohexyl-2-methyl-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359497 6-(4-chlorophenyl)-3-(2-methyl-1-(2-morpholinoethyl)-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359498 dibenzofuran-2-carboxylic acid [4-(2-pyrrolidin-1-yl-ethoxy)-phenyl]-amide 359499 dibenzofuran-2-carboxylic acid [4-(2-diisopropylamino-ethoxy)-phenyl]-amide 359512 6-(4-chlorophenyl)-3-(1-methyl-2-(pyrrolidin-1-yl)-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359520 3-(1-(1-(cyclopropylmethyl)piperidin-4-yl)-2-((5,6-dichloro-1H-benzo[d]imidazol-2-yl)methyl)-1,2,3,4-tetrahydroisoquinolin-6-yl)benzonitrile 359522 1-(2-chlorophenyl)-3-(2-(3,4-dimethylphenoxy)-5-((2-(pyrrolidin-1-yl)ethyl)carbamoyl)phenyl)urea 359525 6-(4-chlorophenyl)-3-(2-methyl-1-(2-(pyrrolidin-1-yl)ethyl)-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359526 6-(4-chlorophenyl)-3-(1-(3-methoxypropyl)-2-methyl-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359527 2-(4-(2-(diisopropylamino)ethoxy)-3-methoxyphenyl)-6-phenylisoindolin-1-one 359529 2-(((8-((6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)methyl)quinolin-3-yl)methyl)(methyl)amino)-N,N-dimethylacetamide 359530 6-(4-chlorophenyl)-3-((3-((4-methylpiperazin-1-yl)methyl)quinolin-8-yl)methyl)thieno[3,2-d]pyrimidin-4(3H)-one 359531 3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-6-phenylthieno[2,3-d]pyrimidin-4(3H)-one 359539 6-(4-chlorophenyl)-3-(3-methyl-2-(pyrrolidin-1-yl)-3H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359550 1-(4-bromophenyl)-3-(2-(3,4-dimethylphenoxy)-5-((2-(pyrrolidin-1-yl)ethyl)carbamoyl)phenyl)urea 359551 6-(4-chlorophenyl)-3-(2-methyl-1-phenyl-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359557 6-(4-chlorophenyl)-3-(1-(3-hydroxypropyl)-2-methyl-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359558 3-(2-amino-1H-benzo[d]imidazol-5-yl)-6-(4-chlorophenyl)thieno[3,2-d]pyrimidin-4(3H)-one 359561 5-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-N-((S)-1-((R)-3-(4,4-dimethylcyclohexylamino)pyrrolidine-1-carbonyl)pyrrolidin-3-yl)-N-methylthiophene-2-carboxamide 359564 5-(4-ethylphenyl)-N-methyl-N-((S)-1-((R)-3-(methylamino)pyrrolidine-1-carbonyl)pyrrolidin-3-yl)thiophene-2-carboxamide 359584 6-(4-chlorophenyl)-3-(2-methyl-1-p-tolyl-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359585 6-(4-chlorophenyl)-3-(1-(4-methoxyphenyl)-2-methyl-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359589 6-(4-chlorophenyl)-3-(2-(methylamino)-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359593 N-((S)-1-((R)-3-(4,4-dimethylcyclohexylamino)pyrrolidine-1-carbonyl)pyrrolidin-3-yl)-5-(4-methoxy-2-methylphenyl)-N-methylthiophene-2-carboxamide 359596 5-(4-ethylphenyl)-N-methyl-N-((S)-1-((R)-3-(methyl(2,2,2-trifluoroethyl)amino)pyrrolidine-1-carbonyl)pyrrolidin-3-yl)thiophene-2-carboxamide 359597 5-(4-ethylphenyl)-N-methyl-N-((S)-1-((R)-3-(tetrahydro-2H-pyran-4-ylamino)pyrrolidine-1-carbonyl)pyrrolidin-3-yl)thiophene-2-carboxamide 359610 6-(4-chlorophenyl)-3-(1-(4-ethoxyphenyl)-2-methyl-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359619 N-((S)-1-((R)-3-(4,4-dimethylcyclohexylamino)pyrrolidine-1-carbonyl)pyrrolidin-3-yl)-N-methyl-5-(4-(trifluoromethyl)phenyl)thiophene-2-carboxamide 359622 5-(4-methoxyphenyl)-N-methyl-N-((S)-1-((R)-3-(tetrahydro-2H-pyran-4-ylamino)pyrrolidine-1-carbonyl)pyrrolidin-3-yl)thiophene-2-carboxamide 359623 4'-Ethyl-biphenyl-4-carboxylic acid methyl-[(S)-1-((R)-3-piperidin-1-yl-pyrrolidine-1-carbonyl)-pyrrolidin-3-yl]-amide 359644 6-(4-chlorophenyl)-3-((3-((dimethylamino)methyl)quinolin-8-yl)methyl)thieno[3,2-d]pyrimidin-4(3H)-one 359645 N-((S)-1-((R)-3-(4,4-dimethylcyclohexylamino)pyrrolidine-1-carbonyl)pyrrolidin-3-yl)-N-methyl-5-p-tolylthiophene-2-carboxamide 359653 4'-ethyl-biphenyl-4-carboxylic acid methyl-[(S)-1-((R)-3-morpholin-4-yl-pyrrolidine-1-carbonyl)-pyrrolidin-3-yl]-amide 359671 1-(5-((2-(pyrrolidin-1-yl)ethyl)carbamoyl)-2-(m-tolyloxy)phenyl)-3-(3-fluorophenyl)urea 359674 6-(4-chlorophenyl)-3-((3-((diethylamino)methyl)quinolin-8-yl)methyl)thieno[3,2-d]pyrimidin-4(3H)-one 359675 6-(4-chlorophenyl)-3-((3-(pyrrolidin-1-ylmethyl)quinolin-8-yl)methyl)thieno[3,2-d]pyrimidin-4(3H)-one 359676 3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-6-phenoxyquinazolin-4(3H)-one 359677 3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-7-phenoxyquinazolin-4(3H)-one 359686 6-(4-chlorophenyl)-3-(2-(dimethylamino)-1-propyl-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359700 1-(2-(3,4-dimethylphenoxy)-5-((2-(pyrrolidin-1-yl)ethyl)carbamoyl)phenyl)-3-phenylurea 359703 1-(5-((2-(pyrrolidin-1-yl)ethyl)carbamoyl)-2-(p-tolyloxy)phenyl)-3-(3-fluorophenyl)urea 359704 6-(4-chlorophenyl)-3-(2-methyl-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359707 6-(4-chlorophenyl)-3-((3-((4-hydroxypiperidin-1-yl)methyl)quinolin-8-yl)methyl)thieno[3,2-d]pyrimidin-4(3H)-one 359708 3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-7-phenylbenzo[d][1,2,3]triazin-4(3H)-one 359709 3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-6-phenoxybenzo[d][1,2,3]triazin-4(3H)-one 359717 6-(4-chlorophenyl)-3-(2-(dimethylamino)-3-propyl-3H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359718 3-(1-(4-methoxybenzyl)-2-(dimethylamino)-1H-benzo[d]imidazol-5-yl)-6-(4-chlorophenyl)thieno[3,2-d]pyrimidin-4(3H)-one 359732 4-(naphthalen-2-yloxy)-3-(3-phenylpropanamido)-N-(2-(pyrrolidin-1-yl)ethyl)benzamide 359736 1-(2-(4-fluoro-3-methylphenoxy)-5-((2-(pyrrolidin-1-yl)ethyl)carbamoyl)phenyl)-3-(3-fluorophenyl)urea 359739 6-(4-chlorophenyl)-3-((3-((4-(methylsulfonyl)piperazin-1-yl)methyl)quinolin-8-yl)methyl)thieno[3,2-d]pyrimidin-4(3H)-one 359741 3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-7-phenoxybenzo[d][1,2,3]triazin-4(3H)-one 359742 5-(4-ethylphenyl)-N-((S)-1-((R)-3-(isopropylamino)pyrrolidine-1-carbonyl)pyrrolidin-3-yl)-N-methylthiophene-2-carboxamide 359743 4'-ethyl-biphenyl-4-carboxylic acid [(S)-1-((R)-3-isopropylamino-pyrrolidine-1-carbonyl)-pyrrolidin-3-yl]-methyl-amide 359749 3-(3-(4-methoxybenzyl)-2-(dimethylamino)-3H-benzo[d]imidazol-5-yl)-6-(4-chlorophenyl)thieno[3,2-d]pyrimidin-4(3H)-one 359750 6-(4-chlorophenyl)-3-(2-(dimethylamino)-1-(2-hydroxyethyl)-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359763 3-cinnamamido-4-(3,4-dimethylphenoxy)-N-(2-(pyrrolidin-1-yl)ethyl)benzamide 359766 1-(2-(3,4-difluorophenoxy)-5-((2-(pyrrolidin-1-yl)ethyl)carbamoyl)phenyl)-3-(3-fluorophenyl)urea 359767 1-(2-(3-fluorophenoxy)-5-((2-(pyrrolidin-1-yl)ethyl)carbamoyl)phenyl)-3-(3-fluorophenyl)urea 359775 5-(4-ethylphenyl)-N-methyl-N-((S)-1-((R)-3-((tetrahydro-2H-pyran-4-yl)methylamino)pyrrolidine-1-carbonyl)pyrrolidin-3-yl)thiophene-2-carboxamide 359776 4'-ethyl-biphenyl-4-carboxylic acid {(S)-1-[(R)-3-(2-hydroxy-ethylamino)-pyrrolidine-1-carbonyl]-pyrrolidin-3-yl}-methyl-amide 359782 6-(4-chlorophenyl)-3-(2-(dimethylamino)-3-(2-hydroxyethyl)-3H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359807 4-(3,4-dimethylphenoxy)-3-((1R,2R)-2-phenylcyclopropanecarboxamido)-N-(2-(pyrrolidin-1-yl)ethyl)benzamide 359815 6-(4-chlorophenyl)-3-(2-(dimethylamino)-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359816 6-(4-chlorophenyl)-3-(2-(isopropylamino)-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359818 2-(4-(2-(diisopropylamino)ethoxy)-3-methoxyphenyl)-5-phenylisoindoline-1,3-dione 359821 5-(4-ethylphenyl)-N-methyl-N-((S)-1-((R)-3-(methyl(tetrahydro-2H-pyran-4-yl)amino)pyrrolidine-1-carbonyl)pyrrolidin-3-yl)thiophene-2-carboxamide 359822 N-((S)-1-((R)-3-(dimethylamino)pyrrolidine-1-carbonyl)pyrrolidin-3-yl)-5-(4-ethylphenyl)-N-methylthiophene-2-carboxamide 359847 6-(4-chlorophenyl)-3-(2-(cyclopropylamino)-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359848 6-(4-chlorophenyl)-3-(2-(pyrrolidin-1-yl)-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359849 2-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-5-phenoxyisoindoline-1,3-dione 359850 2-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-5-(phenylamino)isoindoline-1,3-dione 359882 3-(2-((6-chloro-5-fluoro-1H-benzo[d]imidazol-2-yl)methyl)-1-(1-(cyclopropylmethyl)piperidin-4-yl)-1,2,3,4-tetrahydroisoquinolin-6-yl)benzonitrile 359887 6-(4-chlorophenyl)-3-(2-(piperidin-1-yl)-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359888 6-(4-chlorophenyl)-3-(2-morpholino-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359889 2-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-5-(phenylthio)isoindoline-1,3-dione 359890 6-(4-chlorophenyl)-3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)quinazolin-4(3H)-one 359892 N-((S)-1-((R)-3-(4,4-dimethylcyclohexylamino)pyrrolidine-1-carbonyl)pyrrolidin-3-yl)-5-(4-ethoxyphenyl)-N-methylthiophene-2-carboxamide 359911 6-(4-chlorophenyl)-3-(1-(4-isopropoxyphenyl)-2-methyl-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359938 Ac-Phe-Orn-Pro-cha-Trp-Arg-OH 359953 Ac-Phe-Orn-Pro-cha-Trp-Arg-NH2 359954 Ac-Phe-Orn-Pro-cha-Trp-Nle-NH2 359956 Ac-Phe-Orn-Pro-cha-Trp-Phe-NH2 359957 Ac-Phe-Orn-Pro-hle-Trp-Phe-NH2 359958 Ac-Phe-Orn-Pro-hle-Bta-Phe-NH2 359966 Ac-Phe-Orn-Pro-hle-Dcf-Phe-NH2 359967 Ac-Phe-Orn-Pro-hle-Mcf-Phe-NH2 359968 Ac-Phe-Orn-Pro-hle-Pff-Phe-NH2 359973 Ac-Phe-[Orn-Pro-cha-Trp-Har] 359974 Ac-Phe-[Orn-Pro-cha-Trp-Lys] 359975 Ac-Phe-[Orn-Pro-cha-Trp-Orn] 359980 Ac-Phe-[Orn-Pro-cha-Trp-Cit] 359981 Ac-Phe-[Orn-Pro-cha-Trp-Arg(NO2)] 359986 Ac-Phe-[Orn-Pro-cha-Trp-Nva] 359987 Ac-Phe-[Orn-Pro-cha-Trp-Nle] 359989 6-(4-chlorophenyl)-3-(2-(2-methoxyethylamino)-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359996 6-(4-chlorophenyl)-3-(2-(2-(pyrrolidin-1-yl)ethylamino)-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 359997 6-(4-chlorophenyl)-3-(2-(methyl(2-(pyrrolidin-1-yl)ethyl)amino)-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 360004 6-(4-chlorophenyl)-3-(2-(dimethylamino)-1-(4-methoxyphenyl)-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 360005 6-(4-chlorophenyl)-3-(2-(dimethylamino)-1-methyl-1H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 360009 Ac-Phe-[Orn-Pro-cha-Trp-Ile] 360014 Ac-Phe-[Orn-Pro-cha-Trp-Leu] 360015 Ac-Phe-[Orn-Pro-cha-Trp-Hle] 360016 Ac-Phe-[Orn-Pro-cha-Trp-Chg] 360020 6-(4-chlorophenyl)-3-(2-(dimethylamino)-3-methyl-3H-benzo[d]imidazol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 360059 Ac-Ala-[Orn-Pro-cha-Trp-Arg] 360060 Ac-Phe-[Orn-Ala-cha-Trp-Arg] 360065 Ac-Phe-[Orn-Pro-ala-Trp-Arg] 360066 Ac-Phe-[Orn-Pro-cha-Ala-Arg] 360067 Ac-Phe-[Orn-Pro-cha-Trp-Ala] 360099 Ac-Phe-[Orn-Pro-cha-Trp-Thi] 360100 Ac-Phe-[Orn-Pro-cha-Trp-1Ni] 360101 Ac-Phe-[Orn-Pro-cha-Trp-2Ni] 360310 5-(4-chlorophenyl)-3-[(E)-2-cyclohexylethenyl]-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole 360349 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-3-[(E)-piperidinoiminomethyl]-1H-pyrazole 360368 1-[2-(5-(4-chlorophenyl)-1(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-yl)-(E)-vinyl]-piperidine 360414 N-cycloheptyl-1-(o-fluorbenzyl)-7-methyl-1,8-naphthyridin-4(1H)-on-3-carboxamide 360436 N-cyclohexyl-1-benzyl-7-chloro-1,8-naphthyridin-4(1H)-on-3-carboxamide 360461 N-cyclohexyl-7-chloro-1-(p-fluorbenzyl)-1,8-naphthyridin-4(1H)-on-3-carboxamide 360468 N-cyclohexyl-7-chloro-1-(o-fluorbenzyl)-1,8-naphthyridin-4(1H)-on-3-carboxamide 360476 N-(4'-methylcyclohexyl)-1-(p-fluorobenzyl)-7-methyl-1,8-naphthyridin-4(1H)-on-3-carboxamide 360477 N-(4'-methylcyclohexyl)-7-chloro-1-(2-morpholin-4-yl-ethyl)-1,8-naphthyridin-4(1H)-on-3-carboxamide 360497 N-cyclohexyl-7-methyl-1-phenethyl-1,8-naphthyridin-4(1H)-on-3-carboxamide 360509 N-cyclohexyl-1-benzylquinolin-4(1H)-on-3-carboxamide 360520 N-cyclohexyl-7-methyl-1-(4-methoxybenzyl)-1,8-naphthyridin-4(1H)-on-3-carboxamide 360534 N-(4'-methylcyclohexyl)-1-(o-fluorobenzyl)-7-methyl-1,8-naphthyridin-4(1H)-on-3-carboxamide 360535 N-cyclohexyl-1-(p-fluorbenzyl)-1,8-naphthyridin-4(1H)-on-3-carboxamide 360536 N-cyclohexyl-7-chloro-1-(2-morpholin-4-ylethyl)-quinolin-4(1H)-on-3-carboxamide 360545 N-cycloheptyl-1-benzyl-7-methyl-1,8-naphthyridin-4(1H)-on-3-carboxamide 360546 N-cyclopentyl-7-methyl-1-(2-morpholin-4-ylethyl)-1,8-naphthyridin-4(1H)-on-3-carboxamide 360555 N-cyclohexyl-1-benzyl-1,8-naphthyridin-4(1H)-on-3-carboxamide 360564 N-cycloheptyl-1-(p-fluorobenzyl)-7-methyl-1,8-naphthyridin-4(1H)-on-3-carboxamide 360565 N-cyclohexyl-1-(2-morpholin-4-yl-ethyl)-1,8-naphthyridin-4(1H)-on-3-carboxamide 360566 N-cyclohexyl-7-methyl-1-benzyl-1,8-naphthyridin-4(1H)-on-3-carboxamide 360572 N-cyclopropylmethyl-14beta-[2'-(4''-chlorophenyl)-ethanamino]-7,8-dihydronormorphinone 360587 (3-ethyl-2-methylquinolin-4-yl)-[4-(4-methylpiperazin-1-yl)-phenyl]amine 360588 MC-CAM 360589 N-cyclopropylmethyl-14beta-[4'-(4''-chlorophenyl)-butanamido]-7,8-dihydronorcodeinone 360590 (1R,5R,13R,17S)-17-{[(2E)-3-(4-chlorophenyl)prop-2-en-1-yl]amino}-4-(cyclopropylmethyl)-10-hydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-14-one 360599 (3-isopropyl-2-methylquinolin-4-yl)-[4-(4-methylpiperazin-1-yl)phenyl]amine 360600 N-cyclopropylmethyl-14beta-[4'-(4''-chlorophenyl)-2'-butenamino]-7,8-dihydronorcodeinone 360601 N-cyclopropylmethyl-14beta-[3'-(4'-chlorophenyl)propylamino]-7,8-dihydronormorphinone 360602 (1S,5R,13R,17S)-4-(cyclopropylmethyl)-17-hydroxy-10-methoxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-14-one 360612 N-cyclopropylmethyl-14beta-[3'-(4'-chlorophenyl)propanamido]-7,8-dihydronorcodeinone 360621 N-cyclopropylmethyl-14beta-[4'-(4''-chlorophenyl)-3'-butenamido]-7,8-dihydronormorphinone 360629 N-cyclopropylmethyl-14beta-[4'-(4''-chlorophenyl)-3'-butenamino]-7,8-dihydronorcodeinone 360639 (1R,5R,13R,17S)-17-{[(2E)-3-(4-chlorophenyl)prop-2-en-1-yl]amino}-4-(cyclopropylmethyl)-10-methoxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-14-one 360646 N-cyclopropylmethyl-14beta-[3'-(4'-chlorophenyl)propylamino]-7,8-dihydronorcodeinone 360647 N-cyclopropylmethyl-14beta-[4'-(4''-chlorophenyl)-butanamido]-7,8-dihydronormorphinone 360659 N-cyclopropylmethyl-14beta-[4'-(4''-chlorophenyl)-butanamino]-7,8-dihydronorcodeinone 360673 N-cyclopropylmethyl-14beta-[4'-(4''-chlorophenyl)-2'-butenamido]-7,8-dihydronorcodeinone 360681 N-cyclopropylmethyl-14beta-[4'-(4''-chlorophenyl)-2'-butenamino]-7,8-dihydronormorphinone 360690 N-cyclopropylmethyl-14beta-[2'-(4''-chlorophenyl)-ethanamido]-7,8-dihydronorcodeinone 360691 N-cyclopropylmethyl-14beta-[4'(4''-chlorophenyl)-3'-butenamino]-7,8-dihydronormorphinone 360695 GNF-Pf-3878 360696 N-cyclopropylmethyl-14beta-[4'-(4''-chlorophenyl)-2'-butenamido]-7,8-dihydronorcodeinone 360697 N-cyclopropylmethyl-14beta-[2'-(4''-chlorophenyl)-ethanamino]-7,8-dihydronorcodeinone 360703 N-(4-(4-methylpiperazin-1-yl)phenyl)quinolin-4-amine 360704 N-cyclopropylmethyl-14beta-[4'-(4''-chlorophenyl)-butanamino]-7,8-dihydronormorphinone 360712 14beta-4'-Chlorocinnamoylaminodihydronormorphinone 360713 N-cyclopropylmethyl-14beta-[2'-(4''-chlorophenyl)-ethanamido]-7,8-dihydronormorphinone 360721 (2,3-dimethylquinolin-4-yl)-[4-(4-methylpiperazin-1-yl)phenyl] amine 360722 N-cyclopropylmethyl-14beta-[3'-(4'-chlorophenyl)propanamido]-7,8-dihydronormorphinone 360740 S-(+)-2beta-carboethoxy-3alpha-[bis(4-chlorophenyl)methoxy]tropane 360741 S-(-)-2beta-{[4-(4'-Aminophenyl)butyryl]oxymethyl}-3alpha-[bis(4-fluorophenyl) methoxy]tropane 360746 1-[2-[(2,1,3-benzothiadiazol-4-ylsulfonyl)amino]-4-(benzoylamino)benzoyl]-piperidine 360747 [4-(3,4-dimethylpiperazin-1-yl)phenyl]-(3-methylquinolin-4-yl)amine 360748 [4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,7,8-tetramethylquinolin-4-yl)amine 360749 [4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,5,8-tetramethylquinolin-4-yl)amine 360751 1-{4-[4-(3,4-dimethylpiperazin-1-yl)phenylamino]-2-methylquinolin-3-yl}ethanol 360752 (R)-{4-[4-(3,4-dimethylpiperazin-1-yl)phenylamino]-3-methylquinolin-2-yl}methanol 360763 S-(+)-N-nor-2beta-carboethoxy-3alpha-[bis(4-fluorophenyl)methoxy]tropane 360774 (2-methyl-3-phenylquinolin-4-yl)-[4-(4-methylpiperazin-1-yl)-phenyl]amine 360775 (R)-[4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,7,8-tetramethylquinolin-4-yl)amine 360776 (5-chloro-2,3-dimethylquinolin-4-yl)-[4-(3,4-dimethylpiperazin-1-yl)phenyl]amine 360777 {4-[4-(3,3,4-trimethylpiperazin-1-yl)phenylamino]quinolin-3-yl}methanol 360783 1,2-dihydro-4-[4-[(5,7-dimethyl-2-ethyl-3H-imidazo[4,5-b]pyridin-3-yl)methyl]phenyl]-2-methyl-1-oxo-3-isoquinolinecarboxylic acid 360787 S-(+)-N-allyl-2beta-carboethoxy-3alpha-[bis(4-fluorophenyl)methoxy]-tropane 360790 (S)-[4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,7,8-tetramethylquinolin-4-yl)amine 360791 [4-(3,4-dimethylpiperazin-1-yl)phenyl]-(6-fluoro-2,3-dimethylquinolin-4-yl)amine 360792 (R)-{4-[4-(3,4-dimethylpiperazin-1-yl)phenylamino]quinolin-3-yl}methanol 360802 S-(+)-N-butyl-2beta-carboethoxy-3alpha-[bis(4-fluorophenyl)methoxy]-tropane 360805 (3-benzyl-2-methylquinolin-4-yl)-[4-(4-methylpiperazin-1-yl)-phenyl]amine 360810 3-[4-[(5,7-dimethyl-2-propyl-3H-imidazo[4,5-b]pyridin-3-yl)-methyl]phenyl]-1-hydroxy-1-methyl-1H-indene-2-carboxylic acid 360815 [4-(4-methylpiperazin-1-yl)phenyl]-(2-methylquinolin-4-yl)-amine 360816 [4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,7-trimethylquinolin-4-yl)amine 360817 4-(3-methyltetrahydropyrimidin-1(2H)-yl)phenyl]-(2,3,8-trimethylquinolin-4-yl)amine 360818 (R)-{4-[4-(3-methylpiperazin-1-yl)phenylamino]quinolin-3-yl}methanol 360828 (R)-[4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,7-trimethylquinolin-4-yl)amine 360829 N-(2-diethylaminoethyl)-N'-(3-ethyl-2,8-dimethylquinolin-4-yl)benzene-1,4-diamine 360830 {7-chloro-4-[4-(3,3,4-trimethylpiperazin-1-yl)phenylamino]-quinolin-3-yl}methanol 360839 (3,5-dimethyl-pyridin-4-yl)-[4-(4-methylpiperazin-1-yl)phenyl]amine 360849 4-(3,4-dimethylpiperazin-1-yl)phenyl]-(3-ethyl-2-methyl-5,6,7,8-tetrahydroquinolin-4-yl)amine 360850 (S)-[4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,7-trimethylquinolin-4-yl)amine 360851 N-(2,3-dimethylquinolin-4-yl)-N'-(2-pyrrolidin-1-ylethyl)benzene-1,4-diamine 360852 {4-[4-(3,4-dimethylpiperazin-1-yl)phenylamino]-6-fluoroquinolin-3-yl}methanol 360858 S-(+)-2beta-Hydroxymethyl-3alpha-[bis(4-fluorophenyl)methoxy]-tropane 360862 [4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2-methyl-3-phenylquinolin-4-yl)amine 360863 [4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,8-trimethylquinolin-4-yl)amine 360864 (3-ethyl-2,8-dimethylquinolin-4-yl)-[4-(4-methyl-[1,4]diazepan-1-yl)phenyl]amine 360865 {6-fluoro-4-[4-(3,3,4-trimethylpiperazin-1-yl)phenylamino]-quinolin-3-yl}methanol 360872 S-(+)-2beta-ethenyl-3alpha-[bis(4-fluorophenyl)methoxy]tropane 360879 S-(+)-2beta-{[4-(4'-nitrophenyl)butryl]oxymethyl}-3alpha-[bis(4-fluorophenyl) methoxy]tropane 360883 (2,3-dimethylquinolin-4-yl)-[4-(octahydro-2H-pyrido[1,2-a]-pyrazin-2-yl)phenyl]amine 360884 [4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,5-trimethylquinolin-4-yl)amine 360885 {4-[4-(3,4-dimethylpiperazin-1-yl)phenylamino]-2-methylquinolin-3-yl}methanol 360886 (R)-{4-[4-(3,4-dimethylpiperazin-1-yl)phenylamino]-6-fluoroquinolin-3-yl}methanol 360891 S-(+)-2beta-(2'-(methoxycarbonyl)eth-1'-enyl)-3alpha-[bis(4-fluorophenyl)methoxy] tropane 360895 (3-methylquinolin-4-yl)-[4-(3,3,4-trimethylpiperazin-1-yl)phenyl]amine 360896 [4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,5,7-tetramethylquinolin-4-yl)amine 360897 {2-methyl-4-[4-(3,3,4-trimethylpiperazin-1-yl)phenylamino]-quinolin-3-yl}methanol 360903 S-(+)-2beta-carbomethoxy-3alpha-[bis(4-chlorophenyl)methoxy]tropane 360904 S-(+)-2beta-(2'-(methoxycarbonyl)ethyl)-3alpha-[bis(4-fluorophenyl)-methoxy] tropane 360920 N-[2-[(1H-indol-2-ylsulfonyl)amino]benzoyl]-phenylalanine 360921 (S)-N-[4-bromo-2-[(1H-indol-2-ylsulfonyl)amino]benzoyl]-phenylalanine 360937 2-((2-phenethylphenoxy)methyl)pyridine 360938 {2-[({[(4-methylphenyl)amino]acetyl}hydrazono)methyl]phenoxy}acetic acid 360939 (2-{[(1H-benzimidazol-1-ylacetyl)hydrazono]methyl}phenoxy)acetic acid 360940 ethyl 4-bromo-2-(1-phenyl-1H-pyrazole-4-carbonyl)phenoxyacetate 360941 4-bromo-2-[1-(4-methoxyphenyl)-1H-pyrazole-4-carbonyl]phenoxyacetic acid 360952 2-{2-[2-(3-methoxy-phenyl)-ethyl]-phenoxymethyl}-pyridine 360954 [2-(({[(3-methyl-1H-pyrazol-5-yl)carbonyl]hydrazono}methyl)phenoxy]acetic acid 360955 4-bromo-2-[1-(4-chlorophenyl)-1H-pyrazole-4-carbonyl]phenoxyacetic acid 360959 1-[2-[(1H-indol-2-ylsulfonyl)amino]benzoyl]-piperidine 360967 3-((2-phenethylphenoxy)methyl)pyridine 360968 2-(2-formylphenoxy)acetic acid 360969 2-(4-bromo-2-formylphenoxy)acetic acid 360970 2-(2-acetyl-4-bromophenoxy)acetic acid 360971 4-bromo-2-[1-(4-bromophenyl)-1H-pyrazole-4-carbonyl]phenoxyacetic acid 360974 1-[4-bromo-2-[(1H-indol-2-ylsulfonyl)amino]benzoyl]-piperidine 360980 3-((2-(3-methoxyphenethyl)phenoxy)methyl)pyridine 360981 2-(2-benzoyl-4-bromophenoxy)acetic acid 360982 4-bromo-2-[1-(3-bromophenyl)-1H-pyrazole-4-carbonyl]phenoxyacetic acid 360991 1-(benzyloxy)-2-phenethylbenzene 360992 2-(4-bromo-2-(isoxazole-5-carbonyl)phenoxy)acetic acid 360993 2-(4-bromo-2-tert-butylphenoxy)acetic acid 360994 4-bromo-2-[1-(2-bromophenyl)-1H-pyrazole-4-carbonyl]phenoxyacetic acid 361004 1-(2-(benzyloxy)phenethyl)-3-methoxybenzene 361005 2-(4-bromo-2-(hydroxymethyl)phenoxy)acetic acid 361006 2-(1-phenyl-1H-pyrazole-4-carbonyl)phenoxyacetic acid 361022 4-fluoro-2-(1-phenyl-1H-pyrazole-4-carbonyl)phenoxyacetic acid 361029 4-chloro-2-(1-phenyl-1H-pyrazole-4-carbonyl)phenoxyacetic acid 361041 1-(2-(3-methoxybenzyloxy)phenethyl)-3-methoxybenzene 361042 4-bromo-2-(1-phenyl-1H-pyrazole-4-carbonyl)phenoxyacetic acid 361051 7-methyl-5,6,7,8,9,10,15,16-octahydroindolo[3,2-g][3]benzazacycloundecine 361052 4-methyl-2-(1-phenyl-1H-pyrazole-4-carbonyl)phenoxyacetic acid 361059 4-methoxy-2-(1-phenyl-1H-pyrazole-4-carbonyl)phenoxyacetic acid 361068 {4-bromo-2-[(quinolin-8-ylhydrazono)methyl]phenoxy}acetic acid 361069 {4-bromo-2-[(pyridin-2-ylhydrazono)methyl]phenoxy}acetic acid 361070 4-nitro-2-(1-phenyl-1H-pyrazole-4-carbonyl)phenoxyacetic acid 361078 8-methyl-5,6,7,8,9,10,15,16-octahydroindolo[3,2-g][4]benzazacycloundecine 361083 [2-({[(2,4-dichlorophenoxy)acetyl]hydrazono}methyl)phenoxy]acetic acid 361084 3-(1-phenyl-1H-pyrazole-4-carbonyl)biphenyl-4-yloxyacetic acid 361092 (4-bromo-2-{[(5-phenyl-1,2,4-triazin-3-yl)hydrazono]methyl}phenoxy)acetic acid 361093 [4'-chloro-3-(1-phenyl-1H-pyrazole-4-carbonyl)biphenyl-4-yloxy]acetic acid 361111 [2-(({[5-(4-methoxyphenyl)-1,2,4-triazin-3-yl]hydrazono}methyl)phenoxy]acetic acid 361112 [3',5'-difluoro-3-(1-phenyl-1H-pyrazole-4-carbonyl)biphenyl-4-yloxy]acetic acid 361128 N-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-yl)-7-fluoro-4-oxo-4H-chromene-2-carboxamide 361129 N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-7-cyano-4-oxo-4H-chromene-2-carboxamide 361130 N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-7-chloro-3-methyl-4-oxo-4H-chromene-2-carboxamide 361131 N-[1-[(2,3-dihydro-1,4-benzodioxin-6-yl)methyl]piperidin-4-yl]-7-fluoro-4-oxo-4H-chromene-2-carboxamide 361132 N-(1-(4-acetamidobenzyl)piperidin-4-yl)-7-fluoro-4-oxo-4H-chromene-2-carboxamide 361143 2-[[(thienyl)carbonyl]-amino]-4-methyl-N-(2-chloro-6-methylphenyl)-1,3-thiazole-5-carboxamide 361144 [4-amino-2-(1-methylpiperidin-4-ylamino)pyrimidin-5-yl](2-methoxyphenyl)methanone 361145 4-[4-amino-5-(2-methoxybenzoyl)pyrimidin-2-ylamino]piperidine-1-carboxylic acid ethylamide 361146 4-amino-2-(1-methanesulfonylpiperidin-4-ylamino)pyrimidin-5-yl](5-fluoro-2-methoxyphenyl)methanone 361148 N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-7-chloro-6-fluoro-4-oxo-4H-chromene-2-carboxamide 361149 N-[1-[(3,4-dimethoxybenzyl)methyl]piperidin-4-yl]-7-fluoro-4-oxo-4H-chromene-2-carboxamide 361156 [4-amino-2-(1-methanesulfonylpiperidin-4-ylamino)pyrimidin-5-yl](5-chloro-2-methoxyphenyl)methanone 361158 N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-7-trifluoromethyl-4-oxo-4H-chromene-2-carboxamide 361159 N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-6-fluoro-7-methoxy-4-oxo-4H-chromene-2-carboxamide 361169 4-[4-amino-5-(2-methoxybenzoyl)pyrimidin-2-ylamino]piperidine-1-carboxylic acid ethyl ester 361170 [4-amino-2-(1-methanesulfonylpiperidin-4-ylamino)pyrimidin-5-yl](2-fluoro-6-methoxyphenyl)methanone 361171 N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-6-chloro-4-oxo-4H-chromene-2-carboxamide 361172 N-[1-[(3-methoxybenzyl)methyl]piperidin-4-yl]-7-fluoro-4-oxo-4H-chromene-2-carboxamide 361179 N-(4-(3-bromophenylamino)quinazolin-6-yl)-1,2-dithiolane-3-carboxamide 361180 1-[4-[4-amino-5-(2-methoxybenzoyl)pyrimidin-2-ylamino]-piperidin-1-yl]ethanone 361182 N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-6,7-difluoro-4-oxo-4H-chromene-2-carboxamide 361183 N-[1-[(4-methoxybenzyl)methyl]piperidin-4-yl]-7-fluoro-4-oxo-4H-chromene-2-carboxamide 361190 2-[[(phenylamino)-carbonyl]amino]-4-methyl-N-(2,4,6-trimethylphenyl)-1,3-thiazole-5-carboxamide 361192 [4-amino-2-(1-methanesulfonylpiperidin-4-ylamino)pyrimidin-5-yl](2,6-difluorophenyl)methanone 361194 4-oxo-7-trifluoromethyl-4H-chromene-2-carboxylic acid (1-benzo[1,3]dioxol-5-ylmethyl-piperidin-4-yl)amide 361195 N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-7,8-difluoro-4-oxo-4H-chromene-2-carboxamide 361202 1-[4-[4-amino-5-(2-methoxybenzoyl)pyrimidin-2-ylamino]-piperidin-1-yl]butan-1-one 361203 [4-amino-2-(1-methanesulfonylpiperidin-4-ylamino)pyrimidin-5-yl](2,3-difluoro-6-methoxyphenyl)methanone 361204 N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-6-bromo-4-oxo-4H-chromene-2-carboxamide 361205 N-[1-[(2-fluorobenzyl)methyl]piperidin-4-yl]-7-fluoro-4-oxo-4H-chromene-2-carboxamide 361212 2-[[(tert-butyloxy)carbonyl]-amino]-4-methyl-N-(2,4-dimethylphenyl)-1,3-thiazole-5-carboxamide 361213 2-[[(tert-butylamino)carbonyl]-amino]-4-methyl-N-(2,4,6-trimethylphenyl)-1,3-thiazole-5-carboxamide 361215 [4-amino-2-(1-methanesulfonylpiperidin-4-ylamino)pyrimidin-5-yl](2-methoxyphenyl)methanone 361216 N-[1-(1,3-benzodioxol-5-ylmethyl)pyrrolidin-3-ylmethyl]-7-methoxy-4-oxo-4H-chromene-2-carboxamide 361218 N-[1-[(3-fluorobenzyl)methyl]piperidin-4-yl]-7-fluoro-4-oxo-4H-chromene-2-carboxamide 361224 2-[[(benzylamino)carbonyl]-amino]-4-methyl-N-(2,4,6-trimethylphenyl)-1,3-thiazole-5-carboxamide 361226 [4-amino-2-(1-methanesulfonylpiperidin-4-ylamino)pyrimidin-5-yl](4,5-difluoro-2-methoxyphenyl)methanone 361227 N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-7-hydroxy-4-oxo-4H-chromene-2-carboxamide 361228 N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-6-methyl-4-oxo-4H-chromene-2-carboxamide 361229 N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-6,7,8-trifluoro-4-oxo-4H-chromene-2-carboxamide 361234 2-[[(benzyloxy)carbonyl]-amino]-4-methyl-N-(2,4,6-trimethylphenyl)-1,3-thiazole-5-carboxamide 361235 [4-amino-2-(1-ethanesulfonylpiperidin-4-ylamino)pyrimidin-5-yl](2-methoxyphenyl)methanone 361236 [4-amino-2-(1-methanesulfonylpiperidin-4-ylamino)pyrimidin-5-yl](2,3,4-trifluoro-6-methoxyphenyl)methanone 361237 N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-6-trifluoromethyl-4-oxo-4H-chromene-2-carboxamide 361238 N-[1-[(4-fluorobenzyl)methyl]piperidin-4-yl]-7-fluoro-4-oxo-4H-chromene-2-carboxamide 361243 2-acetamido-4-methyl-N-(2,4,6-trimethylphenyl)-1,3-thiazole-5-carboxamide 361246 4-[4-amino-5-(2-fluorobenzoyl)pyrimidin-2-ylamino]piperidine-1-carboxylic acid ethyl ester 361247 N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-7-(difluoromethoxy)-4-oxo-4H-chromene-2-carboxamide 361248 N-[1-benzylpiperidin-4-yl]-7-fluoro-4-oxo-4H-chromene-2-carboxamide 361249 N-[1-[(2-fluoro-4-methoxybenzyl)methyl]piperidin-4-yl]-7-fluoro-4-oxo-4H-chromene-2-carboxamide 361254 2-[[(tert-butyl)carbonyl]-amino]-4-methyl-N-(2,4,6-trimethylphenyl)-1,3-thiazole-5-carboxamide 361258 [4-amino-2-(1-methanesulfonylpiperidin-4-ylamino)pyrimidin-5-yl](3,4,5-trifluoro-2-methoxyphenyl)methanone 361259 N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-7-ethyl-4-oxo-4H-chromene-2-carboxamide 361260 N-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-yl)-6-fluoro-4-oxo-4H-chromene-2-carboxamide 361268 4-[4-amino-5-(2-methylbenzoyl)pyrimidin-2-ylamino]piperidine-1-carboxylic acid ethylester 361269 N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-4-oxo-4H-chromene-2-carboxamide 361270 N-(1-(3-fluoro-4-methoxybenzyl)piperidin-4-yl)-7-fluoro-4-oxo-4H-chromene-2-carboxamide 361276 3-[[(furanyl)carbonyl]-amino]-4-methyl-N-(2,4,6-trimethylphenyl)-1,3-thiazole-5-carboxamide 361277 N-(2-chloro-6-methylphenyl)-2-[(2-thienylcarbonyl)amino]-1,3-thiazole-5-carboxamide 361278 [4-amino-2-[4-(4-methylpiperazin-1-yl)phenylamino]pyrimidin-5-yl](2-methoxyphenyl)methanone 361279 1-[4-[4-amino-5-(2-ethoxybenzoyl)pyrimidin-2-ylamino]piperidin-1-yl]ethanone 361280 N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-7-bromo-4-oxo-4H-chromene-2-carboxamide 361281 N-[1-[(2,2-difluoro-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl]-7-fluoro-4-oxo-4H-chromene-2-carboxamide 361282 N-[1-{4-[(4-aminopiperidin-1-yl)methyl]phenyl}ethanonyl]-7-fluoro-4-oxo-4H-chromene-2-carboxamide 361288 3-[[(thienyl)carbonyl]-amino]-4-methyl-N-(2,4,6-trimethylphenyl)-1,3-thiazole-5-carboxamide 361289 N-(2-chloro-6-methylphenyl)-2-[(3-thienylcarbonyl)amino]-1,3-thiazole-5-carboxamide 361290 [4-amino-2-(piperidin-4-ylamino)pyrimidin-5-yl](2-methoxyphenyl)methanone 361291 N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-7-chloro-4-oxo-4H-chromene-2-carboxamide 361292 N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-5-chloro-4-oxo-4H-chromene-2-carboxamide 361293 N-{1-[(6-chloro-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-7-fluoro-4-oxo-4H-chromene-2-carboxamide 361300 3-[[(thienyl)carbonyl]-amino]-4-methyl-N-(2-chloro-6-methylphenyl)-1,3-thiazole-5-carboxamide 361302 [4-amino-2-(1-methanesulfonylpiperidin-4-ylamino)pyrimidin-5-yl](4-fluoro-2-methoxyphenyl)methanone 361310 N-(2-chloro-6-methylphenyl)-2-[(cyclopentylcarbonyl)amino]-1,3-thiazole-5-carboxamide 361311 N-(5-chloro-1,3-benzodioxol-4-yl)-7-[(1-methylpiperidin-4-yl-)methoxy]-5-(tetrahydro-2H-pyran-4-yloxy)quinazolin-4-amine 361312 N-(5-chloro-1,3-benzodioxol-4-yl)-7-isopropoxy-5-[(1-methylpiperidin-4-yl)oxy]quinazolin-4-amine 361313 N-(5-chlorobenzo[d][1,3]dioxol-4-yl)-5-methoxy-7-(3-(pyrrolidin-1-yl)propoxy)quinazolin-4-amine 361326 (R,S)-N-(2-chloro-5-methoxyphenyl)-7-(3-morpholinopropoxy)-5-(tetrahydrofuran-3-yloxy)quinazolin-4-amine 361327 N-(5-chlorobenzo[d][1,3]dioxol-4-yl)-7-(2-(pyridin-4-yl)ethoxy)-5-(tetrahydro-2H-pyran-4-yloxy)quinazolin-4-amine 361328 N-(5-chloro-1,3-benzodioxol-4-yl)-7-(2-fluoroethoxy)-5-[(1-methylpiperidin-4-yl)oxy]quinazolin-4-amine 361329 N-(5-chlorobenzo[d][1,3]dioxol-4-yl)-6-methoxy-7-(3-(pyrrolidin-1-yl)propoxy)quinazolin-4-amine 361330 [4-tert-butyl-Phe9]U-II(4-11) 361331 [Thi6]U-II(4-1 1) 361332 [BzThi6]U-II(4-11) 361333 [4-tert-butyl-Phe6]U-II(4-11) 361335 [Leu6]U-II(4-11) 361336 [Cha6]U-II(4-11) 361343 N-(2-chloro-5-methoxyphenyl)-5-[(1-methylpiperidin-4-yl)oxy]quinazolin-4-amine 361344 N-(2-chloro-5-methoxyphenyl)-6-methoxy-5-[(1-methylpiperidin-4-yl)oxy]quinazolin-4-amine 361350 N-1,3-benzodioxol-4-yl-7-(3-pyrrolidin-1-ylpropoxy)-5-(tetrahydro-2H-pyran-4-yloxy)quinazolin-4-amine 361351 N-(5-chloro-1,3-benzodioxol-4-yl)-5-morpholin-4-yl-7-(2-pyrrolidin-1-ylethoxy)quinazolin-4-amine 361352 N-(5-chlorobenzo[d][1,3]dioxol-4-yl)-7-isobutoxy-5-(1-methylpiperidin-4-yloxy)quinazolin-4-amine 361356 2-(2,6-dimethylpyrimidin-4-ylamino)-N-mesitylthiazole-5-carboxamide 361357 N-(2-chloro-5-methoxyphenyl)-5-(tetrahydro-2H-pyran-4-yloxy)quinazolin-4-amine 361358 N-(5-chloro-1,3-benzodioxol-4-yl)-5-isopropoxy-7-(3-pyrrolidin-1-ylpropoxy)quinazolin-4-amine 361359 N-(2-chloro-5-methoxyphenyl)-5,7-dimethoxyquinazolin-4-amine 361367 Ac-c[Cys-His-D-Phe-N-alpha-guanidinylbutyl-Cys]-Trp-NH2 361369 Ac-c[Cys-His-D-Phe-Cys]-N-alpha-guanidinylbutyl-Trp-NH2 361370 Ac-c[Cys-His-D-Phe-Cys]-N-alpha-guanidinylbutyl-D-Trp-NH2 361372 Ac-c[Glu-His-D-Phe-N-alpha-guanidinylbutyl-Orn]-Trp-NH2 361373 Ac-c[Cys-His-D-Nal(2)'-Cys]-N-alpha-guanidinylbutyl-D-Trp-NH2 361376 N-(5-chloro-1,3-benzodioxol-4-yl)-5-[(1-methylpiperidin-4-yl)oxy]quinazolin-4-amine 361377 N-1,3-benzodioxol-4-yl-7-methoxy-5-[(1-methylpiperidin-4-yl)oxy]quinazolin-4-amine 361378 N-(2-chloro-5-methoxyphenyl)-7-(3-(4-methylpiperazin-1-yl)propoxy)-5-(tetrahydro-2H-pyran-4-yloxy)quinazolin-4-amine 361379 N-(2-chloro-5-methoxyphenyl)-6-[3-(4-methylpiperazin-1-yl)-propoxy]-5-(tetrahydro-2H-pyran-4-yloxy)quinazolin-4-amine 361387 N-(2-chloro-6-methylphenyl)-2-(6-(3-morpholinopropylamino)pyridin-2-ylamino)thiazole-5-carboxamide 361388 N-(2,3-dihydrobenzo[b][1,4]dioxin-5-yl)-7-methoxy-5-(1-methylpiperidin-4-yloxy)quinazolin-4-amine 361389 N-(5-chlorobenzo[d][1,3]dioxol-4-yl)-5-isopropoxy-7-(2-morpholinoethoxy)quinazolin-4-amine 361393 D[CFWKYC]V 361394 [Glu4]U-II(4-11) 361395 [Aib4]U-II(4-1 1) 361397 [N-Me-Asp4]U-II(4-11) 361398 [3-nitro-Tyr9]U-II(4-11) 361399 [4-carboxy-Phe9]U-II4-11 361400 [4-amino-Phe9]U-II(4-11) 361403 N-(2-chloro-5-methoxyphenyl)-7-methoxy-5-(3-morpholin-4-ylpropoxy)quinazolin-4-amine 361404 N-(2-chloro-5-methoxyphenyl)-6,7-dimethoxyquinazolin-4-amine 361405 7-[2-(4-acetylpiperazin-1-yl)ethoxy]-N-(5-fluoro-1,3-benzodioxol-4-yl)-5-isopropoxyquinazolin-4-amine 361414 [Cha6]URP 361416 [Pen5, Cha6]U-II(4-1 1) 361417 [Cha6, 3-iodo-Tyr9] U-II(4-11) 361418 6-(4-chlorophenyl)-3-[2-({4-[2-(1-pyrrolidinyl)ethyl]-1-piperidinyl}methyl)-6-quinolinyl]thieno[3,2-d]pyrimidin-4(3H)-one 361419 6-(4-chlorophenyl)-3-(2-{[4-(4-fluorophenyl)-1-piperidinyl]-methyl}-6-quinolinyl)thieno[3,2-d]pyrimidin-4(3H)-one 361420 6-(4-chlorophenyl)-3-[2-({4-[4-(trifluoromethyl)phenyl]-1-piperidinyl}methyl)-6-quinolinyl]thieno[3,2-d]pyrimidin-4(3H)-one 361421 6-(4-chlorophenyl)-3-[2-({4-[2-(4-morpholinyl)ethyl]-1-piperazinyl}methyl)-6-quinolinyl]thieno[3,2-d]pyrimidin-4(3H)-one 361422 N-(2,6-dimethylphenyl)-2-(pyridin-2-ylamino)thiazole-5-carboxamide 361423 N-(2-chloro-5-methoxyphenyl)-7-methoxy-5-[(1-methylpiperidin-4-yl)oxy]quinazolin-4-amine 361424 N-(benzo[d][1,3]dioxol-4-yl)-7-(2-(pyrrolidin-1-yl)ethoxy)-5-(tetrahydro-2H-pyran-4-yloxy)quinazolin-4-amine 361425 N-(6-chloro-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)-7-(2-(pyrrolidin-1-yl)ethoxy)-5-(tetrahydro-2H-pyran-4-yloxy)quinazolin-4-amine 361433 6-(4-chlorophenyl)-3-[2-({4-[3-(4-morpholinyl)propyl]-1-piperazinyl}methyl)-6-quinolinyl]thieno[3,2-d]pyrimidin-4(3H)-one 361434 N-(2-chloro-6-methylphenyl)-2-(2-methyl-6-morpholinopyrimidin-4-ylamino)thiazole-5-carboxamide 361435 N-(5-chlorobenzo[d][1,3]dioxol-4-yl)-7-(3-(pyrrolidin-1-yl)propoxy)-5-(tetrahydro-2H-pyran-4-yloxy)quinazolin-4-amine 361436 N-(5-chlorobenzo[d][1,3]dioxol-4-yl)-5-(pyridin-4-yloxy)quinazolin-4-amine 361441 N-(2-chloro-6-methylphenyl)-2-(2-methyl-6-(3-morpholinopropylamino)pyrimidin-4-ylamino)thiazole-5-carboxamide 361442 N-(5-chlorobenzo[d][1,3]dioxol-4-yl)-7-methoxy-5-(1-methylpiperidin-4-yloxy)quinazolin-4-amine 361443 N-(5-chloro-1,3-benzodioxol-4-yl)-7-methoxy-5-(piperidin-4-yloxy)quinazolin-4-amine 361444 Saracatinib 361450 N-(2,4,6-trimethylphenyl)-2-[(2-pyridinyl)amino]-1,3-thiazole-5-carboxamide 361451 N-(2-chloro-6-methylphenyl)-2-(6-(2-hydroxyethylamino)-2-methylpyrimidin-4-ylamino)thiazole-5-carboxamide 361452 N-(6-chloro-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)-7-(2-(4-methylpiperazin-1-yl)ethoxy)-5-(tetrahydro-2H-pyran-4-yloxy)quinazolin-4-amine 361460 N-(2-chloro-6-methylphenyl)-2-(pyridazin-3-ylamino)thiazole-5-carboxamide 361461 N-(2-chloro-6-methylphenyl)-2-(6-(4-(hydroxymethyl)piperidin-1-yl)-2-methylpyrimidin-4-ylamino)thiazole-5-carboxamide 361462 N-(5-chlorobenzo[d][1,3]dioxol-4-yl)-7-(2-(pyrrolidin-1-yl)ethoxy)-5-(tetrahydro-2H-pyran-4-yloxy)quinazolin-4-amine 361463 N-(5-chlorobenzo[d][1,3]dioxol-4-yl)-7-(3-(4-methylpiperazin-1-yl)propoxy)-5-(tetrahydro-2H-pyran-4-yloxy)quinazolin-4-amine 361467 N-(2,6-dimethylphenyl)-2-[(3-pyradizinyl)amino]-1,3-thiazole-v 361468 N-(2-chloro-6-methylphenyl)-2-[(3,5-dimethyl-2-pyrazinyl)-amino]-1,3-thiazole-5-carboxamide 361469 Dasatinib 361470 N-(2,3-dihydro-1,4-benzodioxin-5-yl)-7-(2-pyrrolidin-1-ylethoxy)-5-(tetrahydro-2H-pyran-4-yloxy)quinazolin-4-amine 361475 N-mesityl-2-(pyrazin-2-ylamino)thiazole-5-carboxamide 361478 N-(2-chloro-5-methoxyphenyl)-5-(cyclohexyloxy)-7-(3-morpholinopropoxy)quinazolin-4-amine 361479 N-(5-chlorobenzo[d][1,3]dioxol-4-yl)-5-((1-methylpiperidin-4-yl)methoxy)quinazolin-4-amine 361480 N-(2-chloro-5-methoxyphenyl)-6-methoxy-7-((1-methylpiperidin-4-yl)methoxy)quinazolin-4-amine 361499 (R)-2-(4-hydroxybicyclo[2.2.2]octan-1-yl)-8-methyl-4-propyl-7,8-dihydro-1H-imidazo[1,2-g]purin-5(4H)-one 361500 (R)-2-(4-hydroxybicyclo[2.2.2]octan-1-yl)-4,8-dipropyl-7,8-dihydro-1H-imidazo[1,2-g]purin-5(4H)-one 361510 (R)-2-(4-hydroxybicyclo[2.2.2]octan-1-yl)-8-isobutyl-4-propyl-7,8-dihydro-1H-imidazo[1,2-g]purin-5(4H)-one 361516 1-(4-(1-(2,6-difluorobenzyl)-5-((benzyl(methyl)amino)methyl)-2,4-dioxo-3-phenyl-1,2,3,4-tetrahydrothieno[2,3-d]pyrimidin-6-yl)phenyl)-3-benzylurea 361517 1-(2,6-difluorobenzyl)-5-((benzyl(methyl)amino)methyl)-6-(4-(4,5-dihydro-1H-imidazol-2-ylamino)phenyl)-3-phenylthieno[2,3-d]pyrimidine-2,4(1H,3H)-dione 361558 (9R,12R,15S)-12-benzyl-9-(4-hydroxy-benzyl)-15-propyl-6,7,8,9,11,12,14,15,17,18-decahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione 361559 (9R,12R,15S)-15-benzyl-9-(4-hydroxy-benzyl)-12-isopropyl-6,7,8,9,11,12,14,15,17,18-decahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione 361574 (9R,12R,15S)-12-isopropyl-9-naphthalen-2-ylmethyl-15-propyl-6,7,8,9,11,12,14,15,17,18,19,20-dodecahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione 361575 (9R,12R,15S)-12-isopropyl-9-naphthalen-1-ylmethyl-15-propyl-6,7,8,9,11,12,14,15,17,18,19,20-dodecahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione 361576 (9R,12R,15S)-8-acetyl-9-(4-hydroxy-benzyl)-12-isopropyl-15-propyl-6,7,8,9,11,12,14,15,17,18,19,20-dodecahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione 361616 (+/-)-2,3-dihydroxy-6a,7,8,12b-tetrahydro-6H-chromeno[3,4-c]isoquinoline 361617 (6aR,12bS)-(+)-2,3-dihydroxy-6a,7,8,12b-tetrahydro-6H-chromeno[3,4-c]isoquinoline 361625 (6aS,12bR)-(-)-2,3-dihydroxy-6a,7,8,12b-tetrahydro-6H-chromeno[3,4-c]isoquinoline 361643 (R)-8-ethyl-2-(4-hydroxybicyclo[2.2.2]octan-1-yl)-4-propyl-7,8-dihydro-1H-imidazo[1,2-g]purin-5(4H)-one 361664 6-[6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl]-N-[3-(1-pyrrolidinyl)propyl]-2-naphthalenecarboxamide 361665 6-(4-chlorophenyl)-3-[6-(1-piperidinylmethyl)-2-naphthalenyl]thieno[3,2-d]pyrimidin-4(3H)-one 361666 6-(4-chlorophenyl)-3-[2-(morpholin-4-ylmethyl)-1-benzothien-5-yl]thieno[3,2-d]pyrimidin-4(3H)-one 361667 6-(4-methylphenyl)-3-[2-(pyrrolidin-1-ylmethyl)-1-benzofuran-5-yl]thieno[3,2-d]pyrimidin-4(3H)-one 361668 4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-bicyclo[2.2.2]octane-1-carboxylic acid 361669 4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-bicyclo[2.2.2]octane-1-carboxylic Acid (2-dimethylamino-ethyl)-amide 361670 3-noradamantyl-1,3-dipropylxanthine 361679 6-(4-chlorophenyl)-3-{6-[(dimethylamino)methyl]-7,8-dihydro-2-naphthalenyl}thieno[3,2-d]pyrimidin-4(3H)-one 361680 3-(2-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-1-benzofuran-5-yl)-6-(4-methylphenyl)thieno[3,2-d]pyrimidin-4(3H)-one 361681 {[4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-bicyclo[2.2.2]octane-1-carbonyl]-amino}-acetic acid methyl ester 361688 6-(4-chlorophenyl)-3-[6-(1-pyrrolidinylmethyl)-7,8-dihydro-2-naphthalenyl]thieno[3,2-d]pyrimidin-4(3H)-one 361689 6-(4-chlorophenyl)-3-[1-methyl-2-(pyrrolidin-1-ylmethyl)-1Hindol-5-yl]thieno[3,2-d]pyrimidin-4(3H)-one 361690 {[4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-bicyclo[2.2.2]octane-1-carbonyl]-amino}-acetic acid 361693 (R)-2-(4-hydroxybicyclo[2.2.2]octan-1-yl)-7-methyl-4-propyl-7,8-dihydro-1H-imidazo[1,2-g]purin-5(4H)-one 361697 6-(4-chlorophenyl)-3-[6-(1-piperidinylmethyl)-7,8-dihydro-2-naphthalenyl]thieno[3,2-d]pyrimidin-4(3H)-one 361698 6-(4-chlorophenyl)-3-(2-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-1-methyl-1H-indol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 361699 2-((4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)bicyclo[2.2.2]octan-1-yl)(methyl)amino)acetic acid 361702 (S)-2-(4-hydroxybicyclo[2.2.2]octan-1-yl)-7-methyl-4-propyl-7,8-dihydro-1H-imidazo[1,2-g]purin-5(4H)-one 361706 6-(4-chlorophenyl)-3-{6-[(dimethylamino)methyl]-5,6,7,8-tetrahydro-2-naphthalenyl}thieno[3,2-d]pyrimidin-4-(3H)-one 361708 3-{[4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-bicyclo[2.2.2]octane-1-carbonyl]-amino}-propionic acid methy lester 361715 6-(4-chlorophenyl)-3-[6-(1-pyrrolidinylmethyl)-5,6,7,8-tetrahydro-2-naphthalenyl]thieno[3,2-d]pyrimidin-4-(3H)-one 361716 8-(4-hydroxymethyl-cyclohexyl)-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 361717 1-[4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-bicyclo[2.2.2]octane-1-carbonyl]-piperidine-4-carboxylic acid 361724 6-(4-chlorophenyl)-3-[6-(1-piperidinylmethyl)-5,6,7,8-tetrahydro-2-naphthalenyl]thieno[3,2-d]pyrimidin-4-(3H)-one 361725 8-(4-benzyloxymethyl-cyclohexyl)-1,3-dipropyl-3,7-dihydropurine-2,6-dione 361728 (R)-2-(4-hydroxybicyclo[2.2.2]octan-1-yl)-8-isopropyl-4-propyl-7,8-dihydro-1H-imidazo[1,2-g]purin-5(4H)-one 361733 6-(4-chlorophenyl)-3-{2-[(dimethylamino)methyl]-1-benzothien-5-yl}thieno[3,2-d]pyrimidin-4(3H)-one 361734 4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-cyclohexanecarboxylic acid butylamide 361735 4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-bicyclo[2.2.2]octane-1-carboxylic acid methyl ester 361737 (R)-8-tert-butyl-2-(4-hydroxybicyclo[2.2.2]octan-1-yl)-4-propyl-7,8-dihydro-1H-imidazo[1,2-g]purin-5(4H)-one 361741 6-(4-chlorophenyl)-3-[2-(1-pyrrolidinylmethyl)-1-benzothien-5-yl]thieno[3,2-d]pyrimidin-4(3H)-one 361742 4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-cyclohexanecarboxylic acid (2-dimethylamino-ethyl)-amide 361743 8-(4-hydroxymethyl-bicyclo[2.2.2]oct-1-yl)-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 361745 (R)-2-(4-hydroxybicyclo[2.2.2]octan-1-yl)-8-phenyl-4-propyl-7,8-dihydro-1H-imidazo[1,2-g]purin-5(4H)-one 361750 6-(4-chlorophenyl)-3-(2-{[(3R)-3-hydroxypyrrolidin-1-yl]-methyl}-1-benzothien-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 361752 4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-bicyclo[2.2.2]octane-1-carbaldehyde 361754 (R)-8-benzyl-2-(4-hydroxybicyclo[2.2.2]octan-1-yl)-4-propyl-7,8-dihydro-1H-imidazo[1,2-g]purin-5(4H)-one 361759 6-(4-chlorophenyl)-3-[2-(piperidin-1-ylmethyl)-1-benzothien-5-yl]thieno[3,2-d]pyrimidin-4(3H)-one 361761 (E)-3-[4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-bicyclo[2.2.2]oct-1-yl]-acrylic acid 361763 Tonapofylline 361765 6-(4-chlorophenyl)-3-[6-(hydroxymethyl)-2-naphthalenyl]thieno[3,2-d]pyrimidin-4(3H)-one 361766 6-(4-chlorophenyl)-3-{2-[(4-phenylpiperidin-1-yl)methyl]-1-benzothien-5-yl}thieno[3,2-d]pyrimidin-4(3H)-one 361768 3-[4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-bicyclo[2.2.2]oct-1-yl]-propionic acid 361770 8-(4-hydroxybicyclo[2.2.2]octan-1-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 361774 trans-[4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-cyclohexyl]-carbamic acid benzyl ester 361775 [4-(2,6-dioxo-1,3-dipropyl-2,3,6,9-tetrahydro-1H-purin-8-yl)-bicyclo[2.2.2]oct-1-yl]-acetic acid 361777 (R)-3-(4-(8-ethyl-5-oxo-4-propyl-4,5,7,8-tetrahydro-1H-imidazo[1,2-g]purin-2-yl)bicyclo[2.2.2]octan-1-yl)propanoic acid 361781 6-(4-chlorophenyl)-3-{2-[(4-methylpiperazin-1-yl)methyl]-1-benzothien-5-yl}thieno[3,2-d]pyrimidin-4(3H)-one 361783 4-[4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-bicyclo[2.2.2]oct-1-yl]-butyric acid 361785 (R)-3-(4-(8-isopropyl-5-oxo-4-propyl-4,5,7,8-tetrahydro-1H-imidazo[1,2-g]purin-2-yl)bicyclo[2.2.2]octan-1-yl)propanoic acid 361788 6-[6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl]-N-[2-(1-pyrrolidinyl)ethyl]-2-naphthalenecarboxamide 361789 6-(4-chlorophenyl)-3-{2-[(4-phenylpiperazin-1-yl)methyl]-1-benzothien-5-yl}thieno[3,2-d]pyrimidin-4(3H)-one 361791 1,3-dipropyl-8-[2-(5,6-exo-epoxy-(1S,2S)-norborn-2-yl)]-xanthine 361793 (R)-4-(8-ethyl-5-oxo-4-propyl-4,5,7,8-tetrahydro-1H-imidazo[1,2-g]purin-2-yl)bicyclo[2.2.2]octane-1-carboxylic acid 361799 6-(4-fluorophenyl)-3-[2-(4-morpholinylmethyl)-6-quinolinyl]-thieno[3,2-d]pyrimidin-4(3H)-one 361800 6-(4-cyano)-3-[2-(4-morpholinylmethyl)-6-quinolinyl]thieno-[3,2-d]pyrimidin-4(3H)-one 361801 6-(4-chlorophenyl)-3-{2-[(4-phenyl-1-piperidinyl)methyl]-6-quinolinyl}thieno[3,2-d]pyrimidin-4(3H)-one 361802 6-(4-chlorophenyl)-3-{(2S)-2-[(dimethylamino)methyl]-2,3-dihydro-1,4-benzodioxin-6-yl}thieno[3,2-d]pyrimidin-4-(3H)-one 361809 (S)-2-(2,6-dimethoxyphenoxy)-N-((2,3,6,7,8,9-hexahydronaphtho[2,3-b][1,4]dioxin-2-yl)methyl)ethanaminium chloride 361810 (S)-2-[((2-(2-methoxy-5,6,7,8-tetrahydronaphthoxy)ethyl)amino)methyl]-1,4-benzodioxane hydrochloride 361818 3-[2-(4-morpholinylmethyl)-6-quinolinyl]-6-[4-(trifluoromethyl)phenyl]thieno[3,2-d]pyrimidin-4(3H)-one 361819 6-(4-chlorophenyl)-3-{2-[(4-methyl-1-piperazinyl)methyl]-6-quinolinyl}thieno[3,2-d]pyrimidin-4(3H)-one 361820 6-(4-chlorophenyl)-3-{(2R)-2-[(dimethylamino)methyl]-2,3-dihydro-1,4-benzodioxin-6-yl}thieno[3,2-d]pyrimidin-4-(3H)-one 361824 (R)-2-[((2-(2-methoxy-5,6,7,8-tetrahydronaphthoxy)ethyl)amino)methyl]-1,4-benzodioxane hydrochloride 361826 (9R,12R,15S)-9,12-diisopropyl-15-propyl-6,7,8,9,11,12,14,15,17,18-decahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione 361830 6-[4-(methyloxy)phenyl]-3-[2-(4-morpholinylmethyl)-6-quinolinyl]thieno[3,2-d]pyrimidin-4(3H)-one 361831 6-(4-chlorophenyl)-3-{2-[(4-ethyl-1-piperazinyl)methyl]-6-quinolinyl}thieno[3,2-d]pyrimidin-4(3H)-one 361832 6-(4-chlorophenyl)-3-(2-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-1-methyl-1H-indol-5-yl)thieno[3,2-d]pyrimidin-4(3H)-one 361845 6-[4-(1-methylpropyl)phenyl]-3-[2-(4-morpholinylmethyl)-6-quinolinyl]thieno[3,2-d]pyrimidin-4(3H)-one 361846 6-(4-chlorophenyl)-3-{2-[(4-phenyl-1-piperazinyl)methyl]-6-quinolinyl}thieno[3,2-d]pyrimidin-4(3H)-one 361853 (S)-2-[((2-(2-methoxy-6-phenylphenoxy)ethyl)amino)methyl]-1,4-benzodioxane hydrochloride 361859 6-(4-chlorophenyl)-3-[2-(hydroxymethyl)-6-quinolinyl]thieno-[3,2-d]pyrimidin-4(3H)-one 361860 (R)-N-(5-(2-fluoro-2-phenylacetyl)-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl)-4-(4-methylpiperazin-1-yl)benzamide 361868 (S)-2-[((2-(2-methoxy-5-phenylphenoxy)ethyl)amino)methyl]-1,4-benzodioxane hydrochloride 361875 6-[4-(1,1-dimethylethyl)phenyl]-3-[2-(4-morpholinylmethyl)-6-quinolinyl]thieno[3,2-d]pyrimidin-4(3H)-one 361876 6-(4-chlorophenyl)-3-{2-[(dimethylamino)methyl]-3,4-dihydro-2H-1,4-benzoxazin-6-yl}thieno[3,2-d]pyrimidin-4 (3H)-one 361877 (R)-N-(5-(2-hydroxy-2-phenylacetyl)-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl)-4-(4-methylpiperazin-1-yl)benzamide 361885 (S)-2-[((2-(2-methoxy-4-phenylphenoxy)ethyl)amino)methyl]-1,4-benzodioxane hydrochloride 361891 6-(4-chlorophenyl)-3-(6-quinolinyl)thieno[3,2-d]pyrimidin-4(3H)-one 361892 6-(4-chlorophenyl)-3-[2-[(dimethylamino)methyl]-4-(methylsulfonyl)-3,4-dihydro-2H-1,4-benzoxazin-6-yl]thieno[3,2-d]pyrimidin-4(3H)-one 361893 (R)-6-(4-chlorophenyl)-3-(2-(cyclopentylmethyl)-2,3-dihydrobenzo[b][1,4]dioxin-6-yl)thieno[3,2-d]pyrimidin-4(3H)-one 361902 (S)-2-[((2-(2-methoxy-1-naphthoxy)ethyl)amino)methyl]-2,3,6,7,8,9-hexahydronaphtho[2,3-b][1,4]dioxine hydrochloride 361908 6-(4-chlorophenyl)-3-{2-[(dimethylamino)methyl]-6-quinolinyl}thieno[3,2-d]pyrimidin-4(3H)-one 361909 (R)-4-(4-methylpiperazin-1-yl)-N-(5-(2-phenylpropanoyl)-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl)benzamide 361920 (E)-(9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-15-propyl-6,7,8,9,11,12,14,15,17,18-decahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione 361926 6-(4-chlorophenyl)-3-(2-{[methyl(phenyl)amino]methyl}-6-quinolinyl)thieno[3,2-d]pyrimidin-4(3H)-one 361927 6-(4-chlorophenyl)-3-[2-[(dimethylamino)methyl]-4-(phenylsulfonyl)-3,4-dihydro-2H-1,4-benzoxazin-6-yl]thieno[3,2-d]pyrimidin-4(3H)-one 361942 6-(4-chlorophenyl)-3-[2-(1H-imidazol-1-ylmethyl)-6-quinolinyl]thieno[3,2-d]pyrimidin-4(3H)-one 361943 (S)-4-(4-methylpiperazin-1-yl)-N-(5-(2-phenylpropanoyl)-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl)benzamide 361956 3-[2-(4-morpholinylmethyl)-6-quinolinyl]-6-phenylthieno-[3,2-d]pyrimidin-4(3H)-one 361957 6-(4-chlorophenyl)-3-[2-(1-pyrrolidinylmethyl)-6-quinolinyl]-thieno[3,2-d]pyrimidin-4(3H)-one 361958 6-(4-chlorophenyl)-3-[2-(1-pyrrolidinylmethyl)-3,4-dihydro-2H-1,4-benzoxazin-6-yl]thieno[3,2-d]pyrimidin-4 (3H)-one 361959 (S)-N-(5-(2-methoxy-2-phenylacetyl)-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl)-4-(4-methylpiperazin-1-yl)benzamide 361964 (S)-2-(2,6-dimethoxyphenoxy)-ethylaminomethyl-1,4-benzodioxane 361965 (R)-2-[((2-(2-methoxy-6-phenylphenoxy)ethyl)amino)methyl]-1,4-benzodioxane hydrochloride 361969 6-(4-chlorophenyl)-3-[2-(4-morpholinylmethyl)-6-quinolinyl]-thieno[3,2-d]pyrimidin-4(3H)-one 361970 6-(4-chlorophenyl)-3-[2-(1-piperidinylmethyl)-6-quinolinyl]-thieno[3,2-d]pyrimidin-4(3H)-one 361971 6-(4-chlorophenyl)-3-(2-{[(3R)-3-hydroxy-1-pyrrolidinyl]-methyl}-3,4-dihydro-2H-1,4-benzoxazin-6-yl)thieno[3,2-d]pyrimidin-4-(3H)-one 361983 (R)-2-(2,6-dimethoxyphenoxy)-ethylaminomethyl-1,4-benzodioxane 361984 (R)-2-[((2-(2-methoxy-5-phenylphenoxy)ethyl)amino)methyl]-1,4-benzodioxane hydrochloride 361990 6-(3-chlorophenyl)-3-[2-(4-morpholinylmethyl)-6-quinolinyl]-thieno[3,2-d]pyrimidin-4(3H)-one 361991 6-(4-chlorophenyl)-3-(2-{[(3S)-3-hydroxy-1-pyrrolidinyl]-methyl}-3,4-dihydro-2H-1,4-benzoxazin-6-yl)thieno[3,2-d]pyrimidin-4-(3H)-one 361997 (S)-N-((2,3-dihydronaphtho[2,3-b][1,4]dioxin-2-yl)methyl)-2-(2,6-dimethoxyphenoxy)ethanaminium chloride 361998 (R)-2-[((2-(2-methoxy-4-phenylphenoxy)ethyl)amino)methyl]-1,4-benzodioxane hydrochloride 362002 6-(2-chlorophenyl)-3-[2-(4-morpholinylmethyl)-6-quinolinyl]-thieno[3,2-d]pyrimidin-4(3H)-one 362003 6-(4-chlorophenyl)-3-(2-{[4-(1-pyrrolidinyl)-1-piperidinyl]-methyl}-6-quinolinyl)thieno[3,2-d]pyrimidin-4(3H)-one 362004 6-(4-chlorophenyl)-3-[2-(4-morpholinylmethyl)-3,4-dihydro-2H-1,4-benzoxazin-6-yl]thieno[3,2-d]pyrimidin-4-(3H)-one 362008 (R)-N-((2,3-dihydronaphtho[2,3-b][1,4]dioxin-2-yl)methyl)-2-(2,6-dimethoxyphenoxy)ethanaminium chloride 362009 (R)-2-[((2-(2-methoxy-1-naphthoxy)ethyl)amino)methyl]-2,3,6,7,8,9-hexahydronaphtho[2,3-b][1,4]dioxine hydrochloride 362014 6-(4-bromophenyl)-3-[2-(4-morpholinylmethyl)-6-quinolinyl]-thieno[3,2-d]pyrimidin-4(3H)-one 362015 6-(4-chlorophenyl)-3-{2-[(4-methyl-1-piperazinyl)methyl]-3,4-dihydro-2H-1,4-benzoxazin-6-yl}thieno[3,2-d]pyrimidin-4-(3H)-one 362020 (S)-N-((2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)-2-(2-methoxynaphthalen-1-yloxy)ethanaminium chloride 362021 1-(3-methoxybenzyloxy)-2-phenethylbenzene 362022 6-(4-chlorophenyl)-3-{2-[(dimethylamino)methyl]-2,3-dihydro-1,4-benzodioxin-6-yl}thieno[3,2-d]pyrimidin-4-(3H)-one 362025 (R)-N-((2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)-2-(2-methoxynaphthalen-1-yloxy)ethanaminium chloride 362026 (R)-2-(2,6-dimethoxyphenoxy)-N-((2,3,6,7,8,9-hexahydronaphtho[2,3-b][1,4]dioxin-2-yl)methyl)ethanaminium chloride 362055 (9R,12R,15S)-15-(4-amino-butyl)-9-(4-hydroxy-benzyl)-12-isopropyl-6,7,8,9,11,12,14,15,17,18-decahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione 362056 (8R,11R,14S)-8-(4-hydroxy-benzyl)-11-isopropyl-14-propyl-5,7,8,10,11,13,14,16,17,18,19,20-dodecahydro-6H-7,10,13,16-tetraaza-benzocyclooctadecene-9,12,15-trione 362057 (9R,12R,15S)-9-benzyl-12-isopropyl-15-propyl-6,7,8,9,11,12,14,15,17,18,19,20-dodecahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione 362064 (9R,12R,15S)-9-cyclohexylmethyl-12-isopropyl-15-propyl-6,7,8,9,11,12,14,15,17,18,19,20-dodecahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione 362065 (9R,12R,15S)-9-(4-hydroxy-benzyl)-15-isobutyl-12-isopropyl-14-methyl-6,7,8,9,11,12,14,15,17,18,19,20-dodecahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione 362072 (9R,12R,15S)-9-benzyl-12-isopropyl-15-propyl-6,7,8,9,11,12,14,15,17,18-decahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione 362073 (9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-10,13,16-trioxo-7,8,9,10,11,12,13,14,15,16,17,18-dodecahydro-6H-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecen-15-yl]-acetic acid 362074 (E/Z)-(8R,11R,14S)-8-(4-Hydroxy-benzyl)-11-isopropyl-14-propyl-5,6,7,8,10,11,13,14,16,17-decahydro-7,10,13,16-tetraaza-benzocycloheptadecene-9,12,15-trione 362082 (9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-15-propyl-7,8,9,10,11,12,14,15,17,18,19,20-dodecahydro-6H-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-13,16-dione 362087 (9R,12R,15S)-9-(4-hydroxy-benzyl)-12-methyl-15-propyl-6,7,8,9,11,12,14,15,17,18-decahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione 362088 (9R,12R,15S)-9-(4-hydroxy-benzyl)-15-isobutyl-12-isopropyl-6,7,8,9,11,12,14,15,17,18-decahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione 362090 (9R,12R,15S)-12-isopropyl-9-phenethyl-15-propyl-6,7,8,9,11,12,14,15,17,18,19,20-dodecahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione 362099 (9R,13R,16S)-9-(4-hydroxy-benzyl)-13-isopropyl-16-propyl-6,7,8,9,12,13,15,16,18,19,20,21-dodecahydro-11H-5-oxa-8,11,12,15,18-pentaaza-benzocyclononadecene-10,14,17-trione 362107 (E/Z)-(9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-15-propyl-5,6,7,8,9,11,12,14,15,17,18,19-dodecahydro-8,11,14,17-tetraaza-benzocyclononadecene-10,13,16-trione 362109 (9R,12R,15S)-9-(1H-indol-3-ylmethyl)-12-isopropyl-15-propyl-6,7,8,9,11,12,14,15,17,18,19,20-dodecahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione 362117 3-[(9R,12R,15S)-9-(4-hydroxy-benzyl)-10,13,16-trioxo-15-propyl-7,8,9,10,11,12,13,14,15,16,17,18-dodecahydro-6H-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecen-12-yl]-propionic acid 362118 (9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-8-methyl-15-propyl-6,7,8,9,11,12,14,15,17,18,19,20-dodecahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione 362126 (9S,12R,15R)-15-(4-hydroxy-benzyl)-12-isopropyl-9-propyl-6,7,9,10,12,13,15,16,17,18,19,20-dodecahydro-5H-7,10,13,16-tetraaza-benzocyclooctadecene-8,11,14-trione 362127 (9R,12R,15S)-9-benzo[b]thiophen-3-ylmethyl-12-isopropyl-15-propyl-6,7,8,9,11,12,14,15,17,18,19,20-dodecahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione 362143 (9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-15-propyl-6,7,8,9,11,12,14,15,17,18,19,20-dodecahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione 362144 (9R,12R,15S)-12-isopropyl-9-(4-methoxy-benzyl)-15-propyl-6,7,8,9,11,12,14,15,17,18,19,20-dodecahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione 362150 (9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-15-methyl-6,7,8,9,11,12,14,15,17,18-decahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione 362158 (9R,12R,15R)-9-(4-Hydroxy-benzyl)-12-isopropyl-15-propyl-6,7,8,9,11,12,14,15,17,18-decahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione 362160 (9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-15-propyl-6,7,8,9,11,12,14,15,18,19-decahydro-17H-5-oxa-8,11,14,17-tetraaza-benzocycloheptadecene-10,13,16-trione 362161 (9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-15-propyl-6,7,8,9,14,15,17,18,19,20-decahydro-5,11-dioxa-8,14,17-triaza-benzocyclooctadecene-10,13,16-trione 362169 (E)-(3S,6R,9R)-9-(4-hydroxy-benzyl)-6-isopropyl-3-propyl-1,4,7,10tetraaza-cyclopentadec-12-ene-2,5,8-trione 362179 (9R,12R,15S)-9-(4-hydroxy-benzyl)-15-hydroxymethyl-12-isopropyl-6,7,8,9,11,12,14,15,17,18-decahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione 362181 (3S,6R,9R)-9-(4-hydroxy-benzyl)-6-isopropyl-3-propyl-1,4,7,10tetraaza-cyclooctadecane-2,5,8-trione 362182 (9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-15-propyl-6,7,8,9,11,12,17,18,19,20-decahydro-5,14-dioxa-8,11,17-triaza-benzocyclooctadecene-10,13,16-trione 363000 3-hydroxy-N-1-hydroxypropan-2-yl-5-4-phenoxyphenylamino-isothiazole-4-carboximidamide 363002 5-4-benzylphenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363003 5-4-benzoylphenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363004 3-hydroxy-N-1-hydroxypropan-2-yl-5-4-phenylthio-phenylamino-isothiazole-4-carboximidamide 363005 3-hydroxy-N-1-hydroxypropan-2-yl-5-4-phenylsulfonyl-phenylamino-isothiazole-4-carboximidamide 363006 3-hydroxy-N-1-hydroxypropan-2-yl-5-4-2-phenylpropan-2-yl-phenylamino-isothiazole-4-carboximidamide 363007 3-hydroxy-N-1-hydroxypropan-2-yl-5-4-3-trifluoromethyl-phenoxy-phenylamino-isothiazole-4-carboximidamide 363008 5-4-2-fluoro-3-trifluoromethyl-phenoxy-phenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363009 5-4-2-chloro-3-trifluoromethyl-phenoxy-phenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363010 5-4-2-chloro-5-trifluoromethyl-phenoxy-phenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363011 5-4-3-fluoro-5-trifluoromethyl-phenoxy-phenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363012 5-4-3-dimethylamino-phenoxy-phenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363013 5-3-chloro-4-2-chloro-3-trifluoromethyl-phenoxy-phenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363014 5-4-2-chloro-3-trifluoromethyl-phenoxy-3-fluorophenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363015 5-4-2-fluoro-5-trifluoromethyl-phenoxy-phenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363016 5-4-2,5-dichlorophenoxy-phenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363017 5-4-2-chloro-5-fluorophenoxy-phenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363018 5-4-2,5-dichlorophenoxy-3-fluorophenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363019 5-4-2-chloro-5-fluorophenoxy-3-methylphenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363020 5-3-chloro-4-2-chloro-5-fluorophenoxy-phenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363021 5-4-2,3-dichlorophenoxy-phenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363022 5-4-2,3-difluorophenoxy-phenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363023 5-3-chloro-4-2,3-dichlorophenoxy-phenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363024 5-4-3-chloro-2-fluorophenoxy-phenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363025 5-4-3,5-dichlorophenoxy-phenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363026 5-4-3,5-difluorophenoxy-phenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363027 5-4-2-chloro-4-fluorophenoxy-phenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363028 5-3-chloro-4-2-chloro-4-fluorophenoxy-phenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363029 5-4-2,4-dichlorophenoxy-phenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363030 5-4-2,4-difluorophenoxy-phenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363031 5-4-2-chloro-3,5-difluorophenoxy-phenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363032 5-4-2-chloro-3,5-difluorophenoxy-3-fluorophenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363033 5-4-2-chloro-4-fluorophenoxy-2-methylphenylamino-3-hydroxy-N-1-hydroxypropan-2-yl-isothiazole-4-carboximidamide 363034 5-(4-(2,5-dichlorophenoxy)phenylamino)-3-hydroxy-N-morpholinoisothiazole-(4-carboximidamide 363035 5-(4-(2,5-dichlorophenoxy)phenylamino)-3-hydroxy-N-2-morpholinoethyl)isothiazole-(4-carboximidamide 363036 5-(4-(2,5-dichlorophenoxy)phenylamino)-3-hydroxy-N-3-morpholinopropyl)isothiazole-(4-carboximidamide 363037 5-(4-(2,5-dichlorophenoxy)phenylamino)-3-hydroxy-N-(4-methylpiperazin-1-yl)isothiazole-(4-carboximidamide 363038 5-(4-(2,5-dichlorophenoxy)phenylamino)-3-hydroxy-N-2-(4-methylpiperazin-1-yl)ethyl)isothiazole-(4-carboximidamide 363039 5-(4-(2,5-dichlorophenoxy)phenylamino)-3-hydroxy-N-3-(4-methylpiperazin-1-yl)propyl)isothiazole-(4-carboximidamide 363040 5-(4-(2,5-dichlorophenoxy)phenylamino)-3-hydroxy-N-2-piperazin-1-yl)ethyl)isothiazole-(4-carboximidamide 363041 5-(4-(2,5-dichlorophenoxy)phenylamino)-3-hydroxy-N-2-3-oxopiperazin-1-yl)ethyl)isothiazole-(4-carboximidamide 363042 5-(4-(2,5-dichlorophenoxy)phenylamino)-3-hydroxy-N-2-hydroxyethyl)isothiazole-(4-carboximidamide 363043 5-(4-(2,5-dichlorophenoxy)phenylamino)-N-(2,3-dihydroxypropyl)-3-hydroxyisothiazole-(4-carboximidamide 363044 5-(4-(2,5-dichlorophenoxy)phenylamino)-N-1,3-dihydroxypropan-2-yl)-3-hydroxyisothiazole-(4-carboximidamide 363045 5-(4-(2,5-dichlorophenoxy)phenylamino)-N-3,4-dihydroxybutyl)-3-hydroxyisothiazole-(4-carboximidamide 363046 5-(4-(2,5-dichlorophenoxy)phenylamino)-3-hydroxy-N-2-hydroxypropyl)isothiazole-(4-carboximidamide 363047 5-(4-(2,5-dichlorophenoxy)phenylamino)-N-(2,3-dihydroxypropoxy)-3-hydroxyisothiazole-(4-carboximidamide 363048 5-(4-(2,5-dichlorophenoxy)phenylamino)-3-hydroxy-N-1-hydroxy-3-methylbutan-2-yl)isothiazole-(4-carboximidamide 363049 5-(4-(2,5-dichlorophenoxy)phenylamino)-3-hydroxy-N-1-hydroxybutan-2-yl)isothiazole-(4-carboximidamide 363050 5-(4-(2,5-dichlorophenoxy)phenylamino)-3-hydroxy-N-tetrahydrofuran-2-yl)methyl)isothiazole-(4-carboximidamide 363051 5-3-chloro-4-iodophenylamino-3-hydroxy-N-isopropylisothiazole-4-carboximidamide 363052 Cyclopropanecarboxylic acid-(3-(4-(3-trifluoromethyl-phenylamino)-pyrimidin-2-ylamino)-phenyl)-amide 363053 N-3-2-3-trifluoromethyl-phenylamino-pyrimidin-4-ylamino-phenyl-cyclopropanecarboxamide 363054 Cyclopropanecarboxylic acid (3-(6-(3-trifluoromethyl-phenylamino)-pyrimidin-4-ylamino)-phenyl)-amide 363055 2-3-7-3-4-hydroxymethyl-piperidin-1-yl-propoxy-6-methoxyquinazolin-4-ylamino-1H-pyrazol-5-yl-N-phenylacetamide 363056 N-2-fluorophenyl-2-3-7-3-4-hydroxymethyl-piperidin-1-yl-propoxy-6-methoxyquinazolin-4-ylamino-1H-pyrazol-5-yl-acetamide 363057 N-(3-fluorophenyl)-2-(3-(7-(3-(4-(hydroxymethyl)piperidin-1-yl)propoxy)-6-methoxyquinazolin-4-ylamino)-1H-pyrazol-5-yl)acetamide 363058 N-4-fluorophenyl-2-3-7-3-4-hydroxymethyl-piperidin-1-yl-propoxy-6-methoxyquinazolin-4-ylamino-1H-pyrazol-5-yl-acetamide 363059 N-2,3-difluorophenyl-2-3-7-3-4-hydroxymethyl-piperidin-1-yl-propoxy-6-methoxyquinazolin-4-ylamino-1H-pyrazol-5-yl-acetamide 363060 N-3,5-difluorophenyl-2-3-7-3-4-hydroxymethyl-piperidin-1-yl-propoxy-6-methoxyquinazolin-4-ylamino-1H-pyrazol-5-yl-acetamide 363061 N-3-chlorophenyl-2-3-7-3-4-hydroxymethyl-piperidin-1-yl-propoxy-6-methoxyquinazolin-4-ylamino-1H-pyrazol-5-yl-acetamide 363062 N-3-cyanophenyl-2-3-7-3-4-hydroxymethyl-piperidin-1-yl-propoxy-6-methoxyquinazolin-4-ylamino-1H-pyrazol-5-yl-acetamide 363063 2-3-7-3-4-hydroxymethyl-piperidin-1-yl-propoxy-6-methoxyquinazolin-4-ylamino-1H-pyrazol-5-yl-N-3-nitrophenyl-acetamide 363064 2-3-7-3-4-hydroxymethyl-piperidin-1-yl-propoxy-6-methoxyquinazolin-4-ylamino-1H-pyrazol-5-yl-N-3-hydroxyphenyl-acetamide 363065 2-3-7-3-4-hydroxymethyl-piperidin-1-yl-propoxy-6-methoxyquinazolin-4-ylamino-1H-pyrazol-5-yl-N-3-methoxyphenyl-acetamide 363066 2-3-7-3-4-hydroxymethyl-piperidin-1-yl-propoxy-6-methoxyquinazolin-4-ylamino-1H-pyrazol-5-yl-N-3-trifluoromethyl-phenyl-acetamide 363067 (R)-N-2,3-difluorophenyl)-2-3-7-3-2-hydroxymethyl)pyrrolidin-1-yl)propoxy)-6-methoxyquinazolin-4-ylamino)-1H-pyrazol-5-yl)acetamide 363068 S-N-2,3-difluorophenyl-2-3-7-3-2-hydroxymethyl-pyrrolidin-1-yl-propoxy-6-methoxyquinazolin-4-ylamino-1H-pyrazol-5-yl-acetamide 363069 N-2,3-difluorophenyl-2-3-7-3-4-2-hydroxyethyl-piperazin-1-yl-propoxy-6-methoxyquinazolin-4-ylamino-1H-pyrazol-5-yl-acetamide 363070 N-2,3-difluorophenyl-2-3-7-3-4-hydroxypiperidin-1-yl-propoxy-6-methoxyquinazolin-4-ylamino-1H-pyrazol-5-yl-acetamide 363071 N-2,3-difluorophenyl-2-3-7-3-4-2-hydroxyethyl-piperidin-1-yl-propoxy-6-methoxyquinazolin-4-ylamino-1H-pyrazol-5-yl-acetamide 363072 (R)-N-3-fluorophenyl)-2-3-7-3-2-hydroxymethyl)pyrrolidin-1-yl)propoxy)-6-methoxyquinazolin-4-ylamino)-1H-pyrazol-5-yl)acetamide 363073 N-3-fluorophenyl-2-3-7-3-2-hydroxyethylamino-propoxy-6-methoxyquinazolin-4-ylamino-1H-pyrazol-5-yl-acetamide 363074 N-3-fluorophenyl-2-3-7-3-2-hydroxyethyl-methyl-amino-propoxy-6-methoxyquinazolin-4-ylamino-1H-pyrazol-5-yl-acetamide 363075 2-(3-(7-(3-(ethyl(2-hydroxyethyl)amino)propoxy)-6-methoxyquinazolin-4-ylamino)-1H-pyrazol-5-yl)-N-(3-fluorophenyl)acetamide 363076 N-(3-fluorophenyl)-2-(3-(7-(3-((2-hydroxyethyl)(propyl)amino)propoxy)-6-methoxyquinazolin-4-ylamino)-1H-pyrazol-5-yl)acetamide 363077 N-(2,3-difluorophenyl)-2-(3-(7-(3-(ethyl(2-hydroxyethyl)amino)propoxy)-6-methoxyquinazolin-4-ylamino)-1H-pyrazol-5-yl)acetamide 363078 N-(2,3-difluorophenyl)-2-(3-(7-(3-((2-hydroxyethyl)(propyl)amino)propoxy)-6-methoxyquinazolin-4-ylamino)-1H-pyrazol-5-yl)acetamide 363079 N-(2,3-difluorophenyl)-2-(3-(7-(3-((2-hydroxyethyl)(isobutyl)amino)propoxy)-6-methoxyquinazolin-4-ylamino)-1H-pyrazol-5-yl)acetamide 363080 N-(2,3-difluorophenyl)-2-(3-(7-(3-(ethyl(2-hydroxyethyl)amino)propoxy)quinazolin-4-ylamino)-1H-pyrazol-5-yl)acetamide 363081 N-2,3-difluorophenyl-2-3-7-3-2-hydroxyethyl-propyl-amino-propoxy-quinazolin-4-ylamino-1H-pyrazol-5-yl-acetamide 363082 (R)-N-2,3-difluorophenyl)-2-3-7-3-2-hydroxymethyl)pyrrolidin-1-yl)propoxy)quinazolin-4-ylamino)-1H-pyrazol-5-yl)acetamide 363083 2-(3-((7-(3-(ethyl(2-hydroxyethyl)amino)propoxy)quinazolin-4-yl)amino)-1H-pyrazol-5-yl)-N-(3-fluorophenyl)acetamide 363084 N-3-fluorophenyl-2-3-7-3-2-hydroxyethyl-propyl-amino-propoxy-quinazolin-4-ylamino-1H-pyrazol-5-yl-acetamide 363085 (R)-N-3-fluorophenyl)-2-3-7-3-2-hydroxymethyl)pyrrolidin-1-yl)propoxy)quinazolin-4-ylamino)-1H-pyrazol-5-yl)acetamide 363090 4-benzyl-3-bromo-N-5-6-methoxy-7-3-morpholinopropoxy-quinazolin-4-ylamino-pyrimidin-2-yl-benzamide 363091 2-N,N-dipropylsulfamoyl-N-5-6-methoxy-7-3-morpholinopropoxy-quinazolin-4-ylamino-pyrimidin-2-yl-pyrimidine-5-carboxamide 363092 2S,3S,4R,5R-N-6R,9R,12R,15R,18R,21R-1-amino-6-carbamoyl-9,12,15,18,21-pentakis3-guanidinopropyl-1-imino-8,11,14,17,20,23-hexaoxo-2,7,10,13,16,19,22-heptaazaoctacosan-28-yl-5-6-amino-9H-purin-9-yl-3,4-dihydroxytetrahydrofuran-2-carboxamide 363093 2S,3S,4R,5R-5-6-amino-9H-purin-9-yl-N-12R,15R,18R,21R,24R,27R-12,15,18,21,24,27-hexakis3-guanidinopropyl-1-isoquinoline-5-sulfonamido-9,11,14,17,20,23,26,29-octaoxo-3,10,13,16,19,22,25,28-o ctaazatetratriacontan-34-yl-3,4-dihydroxytetrahydrofuran-2-carboxamide 363094 N-((5-(4-(1H-benzo[d][1,2,3]triazol-1-yl)piperidin-1-ylsulfonyl)thiophen-2-yl)methyl)-4-chlorobenzamide 363095 7-cyclohexyl-N-4-4-methylpiperazin-1-yl-phenyl-7H-pyrrolo[2,3-d]pyrimidin-2-amine 363096 7-cyclohexyl-N-4-morpholinophenyl-7H-pyrrolo[2,3-d]pyrimidin-2-amine 363097 7-cyclohexyl-N-4-4-2-methoxyethyl-piperazin-1-yl-phenyl-7H-pyrrolo[2,3-d]pyrimidin-2-amine 363098 2-3-7-cyclohexyl-7H-pyrrolo[2,3-d]pyrimidin-2-ylamino-phenyl-acetic acid 363099 4-[4-({7-cyclohexyl-7H-pyrrolo[2,3-d]pyrimidin-2-yl}amino)phenyl]-1,4-thiomorpholine-1,1-dione 363100 7-bicyclo[2.2.1]heptan-2-yl-N-4-4-methylpiperazin-1-yl-phenyl-7H-pyrrolo[2,3-d]pyrimidin-2-amine 363101 7-3-methoxyphenyl-N-4-4-methylpiperazin-1-yl-phenyl-7H-pyrrolo[2,3-d]pyrimidin-2-amine 363102 N-4-4-methylpiperazin-1-yl-phenyl-7-pyridin-3-yl-7H-pyrrolo[2,3-d]pyrimidin-2-amine 363103 N-4-4-methylpiperazin-1-yl-phenyl-7-3-methylsulfonyl-phenyl-7H-pyrrolo[2,3-d]pyrimidin-2-amine 363104 7-2,3-dihydro-1H-inden-2-yl-N-4-4-methylpiperazin-1-yl-phenyl-7H-pyrrolo[2,3-d]pyrimidin-2-amine 363107 N-(4-amino-2-propylquinolin-6-yl)-4-(4-chlorophenyl)cyclohexanecarboxamide 363108 N-(4-amino-2-propylquinolin-6-yl)-4-(trifluoromethyl)benzamide 363109 N-(4-amino-2-propylquinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363110 N-(4-amino-2-propylquinolin-6-yl)-2-(4-(trifluoromethyl)phenyl)acetamide 363111 N-(4-amino-2-propylquinolin-6-yl)-3-phenylpropanamide 363112 N-(4-amino-2-propylquinolin-6-yl)-N-methyl-3-(4-(trifluoromethyl)phenyl)propanamide 363114 N-(4-amino-2-propylquinolin-6-yl)-4'-(trifluoromethyl)biphenyl-4-carboxamide 363115 (E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-hydroxyphenyl)acrylamide 363116 5,6-difluoro-N-(3-(4-methylpiperazin-1-yl)propyl)-N-((1R,3R,6R)-6-(3-(morpholinomethyl)phenyl)bicyclo[4.1.0]heptan-3-yl)-1H-benzo[d]imidazol-2-amine 363117 5,6-difluoro-N-((1R,3R,6R)-6-(3-((4-methylpiperazin-1-yl)methyl)phenyl)bicyclo[4.1.0]heptan-3-yl)-N-(3-(4-methylpiperazin-1-yl)propyl)-1H-benzo[d]imidazol-2-amine 363118 N-(1-(naphthalen-2-ylmethyl)piperidin-4-yl)benzamide 363119 3-methoxy-N-(1-(naphthalen-2-ylmethyl)piperidin-4-yl)benzamide 363120 3,5-dimethoxy-N-(1-(naphthalen-2-ylmethyl)piperidin-4-yl)benzamide 363121 3,5-diethoxy-N-(1-(naphthalen-2-ylmethyl)piperidin-4-yl)benzamide 363122 3,4-dimethoxy-N-(1-(naphthalen-2-ylmethyl)piperidin-4-yl)benzamide 363123 3,4,5-trimethoxy-N-(1-(naphthalen-2-ylmethyl)piperidin-4-yl)benzamide 363124 N-(4-amino-2-propylquinolin-6-yl)-4'-chlorobiphenyl-4-carboxamide 363125 3,5-dimethoxy-N-((3R,4R)-3-methyl-1-(naphthalen-2-ylmethyl)piperidin-4-yl)benzamide 363127 4-((1S,4R,5S)-4-((5-fluoro-6-(trifluoromethyl)-1H-benzo[d]imidazol-2-yl)(3-(4-methylpiperazin-1-yl)propyl)amino)bicyclo[3.1.0]hexan-1-yl)benzonitrile 363128 3-((1S,4R,5S)-4-((6-chloro-5-fluoro-1H-benzo[d]imidazol-2-yl)(3-(4-methylpiperazin-1-yl)propyl)amino)bicyclo[3.1.0]hexan-1-yl)benzonitrile 363129 3,5-dimethoxy-N-(4-methyl-1-(naphthalen-2-ylmethyl)piperidin-4-yl)benzamide 363130 3,5-dimethoxy-N-((3S,4R)-3-methyl-1-(naphthalen-2-ylmethyl)piperidin-4-yl)benzamide 363131 3-((1R,4R,6R)-4-((6-chloro-5-fluoro-1H-benzo[d]imidazol-2-yl)((1-(methylsulfonyl)piperidin-4-yl)methyl)amino)bicyclo[4.1.0]heptan-1-yl)benzonitrile 363132 (E)-N-(4-amino-2-propylquinolin-6-yl)-3-(2-chlorophenyl)acrylamide 363133 4-fluoro-N-(1-(naphthalen-2-ylmethyl)piperidin-4-yl)benzamide 363134 3-((1R,4R,6R)-4-((5,6-dichloro-1H-benzo[d]imidazol-2-yl)((1-(methylsulfonyl)piperidin-4-yl)methyl)amino)bicyclo[4.1.0]heptan-1-yl)benzonitrile 363135 3-((1R,4R,6R)-4-((5,6-difluoro-1H-benzo[d]imidazol-2-yl)((1-(methylsulfonyl)piperidin-4-yl)methyl)amino)bicyclo[4.1.0]heptan-1-yl)benzonitrile 363136 (1R,5S,6r)-N-(3,4-difluorobenzyl)-3-(naphthalen-2-ylmethyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide 363138 3-((1S,4R,5S)-4-((5,6-dichloro-1H-benzo[d]imidazol-2-yl)(3-(4-methylpiperazin-1-yl)propyl)amino)bicyclo[3.1.0]hexan-1-yl)benzonitrile 363139 3,4-difluoro-N-(1-(naphthalen-2-ylmethyl)piperidin-4-yl)benzamide 363140 3,4,5-trifluoro-N-(1-(naphthalen-2-ylmethyl)piperidin-4-yl)benzamide 363141 3-((1S,4R,5S)-4-((5,6-difluoro-1H-benzo[d]imidazol-2-yl)(3-(4-methylpiperazin-1-yl)propyl)amino)bicyclo[3.1.0]hexan-1-yl)benzonitrile 363142 4-((1S,4R,5S)-4-((5,6-dichloro-1H-benzo[d]imidazol-2-yl)(3-(4-methylpiperazin-1-yl)propyl)amino)bicyclo[3.1.0]hexan-1-yl)benzonitrile 363143 (E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-iodophenyl)acrylamide 363144 (E)-N-(4-amino-2-propylquinolin-6-yl)-3-p-tolylacrylamide 363145 (E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)acrylamide 363146 (E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-ethylphenyl)acrylamide 363147 (E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-propylphenyl)acrylamide 363148 (E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-butylphenyl)acrylamide 363149 4-chloro-N-(1-(naphthalen-2-ylmethyl)piperidin-4-yl)benzamide 363150 (R)-3,5-dimethoxy-N-(1-(naphthalen-2-ylmethyl)pyrrolidin-3-yl)benzamide 363152 (S)-3,5-dimethoxy-N-(1-(naphthalen-2-ylmethyl)pyrrolidin-3-yl)benzamide 363153 (R)-3-methoxy-N-(1-(naphthalen-2-ylmethyl)pyrrolidin-3-yl)benzamide 363154 3,5-difluoro-N-(1-(naphthalen-2-ylmethyl)piperidin-4-yl)benzamide 363155 4-fluoro-3-methoxy-N-(1-(naphthalen-2-ylmethyl)piperidin-4-yl)benzamide 363156 4-((1S,4R,5S)-4-((6-chloro-5-fluoro-1H-benzo[d]imidazol-2-yl)(3-(4-methylpiperazin-1-yl)propyl)amino)bicyclo[3.1.0]hexan-1-yl)benzonitrile 363157 3-((1R,4R,6R)-4-((5,6-dichloro-1H-benzo[d]imidazol-2-yl)(3-(4-methylpiperazin-1-yl)propyl)amino)bicyclo[4.1.0]heptan-1-yl)benzaldehyde 363158 3-((1R,4R,6R)-4-((5,6-difluoro-1H-benzo[d]imidazol-2-yl)(3-(4-methylpiperazin-1-yl)propyl)amino)bicyclo[4.1.0]heptan-1-yl)benzaldehyde 363159 tert-butyl 4-((((1R,3R,6R)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)(5,6-dichloro-1H-benzo[d]imidazol-2-yl)amino)methyl)piperidine-1-carboxylate 363160 5,6-difluoro-N-(3-(4-methylpiperazin-1-yl)propyl)-N-((1R,3R,6R)-6-(3-(piperidin-1-ylmethyl)phenyl)bicyclo[4.1.0]heptan-3-yl)-1H-benzo[d]imidazol-2-amine 363161 (E)-N-(4-amino-2-propylquinolin-6-yl)-3-(3,4-dichlorophenyl)acrylamide 363162 (E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-nitrophenyl)acrylamide 363163 (E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-aminophenyl)acrylamide 363164 N-(1-((6-fluoronaphthalen-2-yl)methyl)piperidin-4-yl)-3,5-dimethoxybenzamide 363165 (R)-4-fluoro-3-methoxy-N-(1-(naphthalen-2-ylmethyl)pyrrolidin-3-yl)benzamide 363166 3,5-dimethoxy-N-((3R)-1-(1-(naphthalen-2-yl)ethyl)pyrrolidin-3-yl)benzamide 363167 (R,E)-N-(1-cinnamylpyrrolidin-3-yl)-3,5-dimethoxybenzamide 363168 (E)-4R,6R)-4-((5,6-difluoro-1H-benzo[d]imidazol-2-yl)(3-(4-methylpiperazin-1-yl)propyl)amino)bicyclo[4.1.0]heptan-1-yl)benzaldehyde O-methyl oxime 363169 (E)-4-(3-(4-amino-2-propylquinolin-6-ylamino)-3-oxoprop-1-enyl)phenyl acetate 363170 3-(dimethylamino)-N-(1-(naphthalen-2-ylmethyl)piperidin-4-yl)benzamide 363171 (E)-N-(4-amino-2-propylquinolin-6-yl)-3-(3-chlorophenyl)acrylamide 363172 (E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-chlorophenyl)acrylamide 363173 (E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-fluorophenyl)acrylamide 363174 (3-((1R,4R,6R)-4-((5,6-difluoro-1H-benzo[d]imidazol-2-yl)(3-(4-methylpiperazin-1-yl)propyl)amino)bicyclo[4.1.0]heptan-1-yl)phenyl)methanol 363175 5,6-dichloro-N-((1R,3R,6R)-6-(3-((dimethylamino)methyl)phenyl)bicyclo[4.1.0]heptan-3-yl)-N-(3-(4-methylpiperazin-1-yl)propyl)-1H-benzo[d]imidazol-2-amine 363176 5,6-difluoro-N-(3-(4-methylpiperazin-1-yl)propyl)-N-((1R,3R,6R)-6-(3-(pyrrolidin-1-ylmethyl)phenyl)bicyclo[4.1.0]heptan-3-yl)-1H-benzo[d]imidazol-2-amine 363177 (S)-1-(difluoro-1H-benzo[d]imidazol-2-yl)(3-(4-methylpiperazin-1-yl)propyl)amino)bicyclo[4.1.0]heptan-1-yl)benzyl)pyrrolidin-3-ol 363178 3,5-dimethoxy-N-(1-(1-(naphthalen-2-yl)ethyl)piperidin-4-yl)benzamide 363179 3,5-dimethoxy-N-(1-(quinolin-2-ylmethyl)piperidin-4-yl)benzamide 363180 3,5-dimethoxy-N-((3R)-1-((E)-4-phenylbut-3-en-2-yl)pyrrolidin-3-yl)benzamide 363181 (R)-N-(1-benzylpyrrolidin-3-yl)-3,5-dimethoxybenzamide 363182 3-((1R,4R,6R)-4-((5,6-difluoro-1H-benzo[d]imidazol-2-yl)(3-(4-methylpiperazin-1-yl)propyl)amino)bicyclo[4.1.0]heptan-1-yl)benzonitrile 363183 (E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-tert-butylphenyl)acrylamide 363184 (E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-(methylthio)phenyl)acrylamide 363185 (E)-N-(4-amino-2-propylquinolin-6-yl)-3-(biphenyl-4-yl)acrylamide 363186 3,5-dimethoxy-N-(1-((1-methyl-1H-indol-2-yl)methyl)piperidin-4-yl)benzamide 363187 3-((1R,4R,6R)-4-((5,6-dichloro-1H-benzo[d]imidazol-2-yl)(3-(4-methylpiperazin-1-yl)propyl)amino)bicyclo[4.1.0]heptan-1-yl)benzonitrile 363188 N-((1R,3R,6R)-6-(3-((dimethylamino)methyl)phenyl)bicyclo[4.1.0]heptan-3-yl)-5,6-difluoro-N-(3-(4-methylpiperazin-1-yl)propyl)-1H-benzo[d]imidazol-2-amine 363189 (E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-isopropylphenyl)acrylamide 363190 5,6-dichloro-N-(3-(4-methylpiperazin-1-yl)propyl)-N-((1R,3R,6R)-6-(3-(morpholinomethyl)phenyl)bicyclo[4.1.0]heptan-3-yl)-1H-benzo[d]imidazol-2-amine 363191 (S)-N-(1-(3-hydroxy-3-phenylpropyl)piperidin-4-yl)-3,5-dimethoxybenzamide 363192 N-(1-benzylpiperidin-4-yl)-3,5-dimethoxybenzamide 363193 3-((1R,4R,6R)-4-((6-chloro-5-fluoro-1H-benzo[d]imidazol-2-yl)(3-(4-methylpiperazin-1-yl)propyl)amino)bicyclo[4.1.0]heptan-1-yl)benzonitrile 363194 3-((1R,4R,6R)-4-((5,6-dichloro-1H-benzo[d]imidazol-2-yl)(piperidin-1-ylmethyl)amino)bicyclo[4.1.0]heptan-1-yl)benzonitrile 363195 N-(1-(3,4-dichlorobenzyl)piperidin-4-yl)-3,5-dimethoxybenzamide 363196 3,5-dimethoxy-N-(1-((1,2,3,4-tetrahydronaphthalen-2-yl)methyl)piperidin-4-yl)benzamide 363198 (R)-N-(5-guanidino-1-oxo-1-(4-(trifluoromethyl)benzylamino)pentan-2-yl)-1-naphthamide 363199 (S)-4-(4-fluorophenethyl)-1-(6-((diethylamino)-methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-2-one 363200 N-(2-(isopropylamino)-1-methyl-1H-benzo[d]imidazol-6-yl)-2-(4-(trifluoromethyl)phenoxy)acetamide 363201 N-(1-methyl-2-(piperazin-1-ylmethyl)-1H-benzo[d]imidazol-6-yl)-2-(4-(trifluoromethyl)phenoxy)acetamide 363202 N-{1-[(6-fluoro-2-naphthyl)methyl]piperidin-4-yl}benzamide 363203 3,5-dimethoxy-N-methyl-N-(1-(naphthalen-2-ylmethyl)piperidin-4-yl)benzamide 363204 N-(2-(methyl(propyl)amino)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363205 N-(2-(isopropyl(methyl)amino)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363206 (E)-N-(4-(azetidin-1-yl)-2-propylquinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)acrylamide 363207 (E)-N-(2-propyl-4-(pyrrolidin-1-yl)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)acrylamide 363209 (S)-4-(4-chlorophenethyl)-1-(6-((diethylamino)-methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-2-one 363210 N-(2-(methylamino)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363211 (S)-4-(2-cyclohexylethyl)-1-(6-((diethylamino)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-2-one 363212 N-(1-(6,7-dihydro-5H-indeno[5,6-d][1,3]dioxol-5-yl)piperidin-4-yl)-6-fluoro-4-oxo-4H-chromene-2-carboxamide 363213 N-(1-(7,8-dihydro-6H-indeno[5,4-d][1,3]dioxol-6-yl)piperidin-4-yl)-6-fluoro-4-oxo-4H-chromene-2-carboxamide 363214 N-(2-(cyclopentyl(methyl)amino)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363215 4-(3-(trifluoromethyl)phenethyl)-1-(6-((diethylamino)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-2-one 363216 (S)-N-(6-((4-acetylpiperazin-1-yl)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)-5-(4-fluorophenyl)-N-methylpicolinamide 363217 (S)-1-(6-((1H-imidazol-1-yl)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)-4-(4-fluorophenethyl)piperazin-2-one 363218 N-(2-(dimethylamino)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363219 (S)-1-(((S)-6-(4'-fluoro-N-methylbiphenyl-4-ylcarboxamido)-5,6,7,8-tetrahydronaphthalen-2-yl)methyl)-N,N-dimethylpyrrolidine-2-carboxamide 363221 7-fluoro-4-oxo-N-(1-(2-oxo-3,5,6,7-tetrahydro-2H-indeno[5,6-d]oxazol-5-yl)piperidin-4-yl)-4H-chromene-2-carboxamide 363222 N-(2-(2-methylpyrrolidin-1-yl)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363223 N-[(2S)-6-[(1,1-dioxo-1,4-thiomorpholin-4-yl)methyl]-1,2,3,4-tetrahydronaphthalen-2-yl]-4-(4-fluorophenyl)-N-methylbenzamid 363224 5-(4-((diethylamino)methyl)phenethyl)-N-(4-fluorophenyl)-4-oxo-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carboxamide 363225 7-fluoro-4-oxo-N-(1-(3-oxo-2,3,4,6,7,8-hexahydroindeno[5,6-b][1,4]oxazin-6-yl)piperidin-4-yl)-4H-chromene-2-carboxamide 363226 (S)-N-(6-((dimethylamino)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)-N-methyl-4-(pyridin-4-yl)benzamide 363227 (S)-4'-fluoro-N-methyl-N-(6-((3-oxopiperazin-1-yl)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)biphenyl-4-carboxamide 363228 N-(1-((2-ethylbenzo[d]oxazol-6-yl)methyl)piperidin-4-yl)-7-fluoro-4-oxo-4H-chromene-2-carboxamide 363229 N-(2-(cyclohexyl(methyl)amino)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363230 (S)-N-(6-(((2-(dimethylamino)-2-oxoethyl)(methyl)amino)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)-4'-fluoro-N-methylbiphenyl-4-carboxamide 363231 1-(4-(piperidin-1-ylmethyl)phenethyl)-4-phenethylpiperazin-2-one 363232 N-(1-((2-ethylbenzo[d]oxazol-5-yl)methyl)piperidin-4-yl)-7-fluoro-4-oxo-4H-chromene-2-carboxamide 363233 N-(2-(methyl(phenyl)amino)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363234 4-{[(6S)-6-{4-[2-(4-fluorophenyl)ethyl]-2-oxopiperazin-1-yl}-5,6,7,8-tetrahydronaphthalen-2-yl]methyl}-1,4-thiomorpholine-1,1-dione 363235 N-(3-fluorophenyl)-4-oxo-5-(4-(piperidin-1-ylmethyl)phenethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carboxamide 363236 7-fluoro-4-oxo-N-(1-((2-oxo-2,3-dihydrobenzo[d]oxazol-5-yl)methyl)piperidin-4-yl)-4H-chromene-2-carboxamide 363237 N-(2-(azetidin-1-yl)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363238 (S)-1-(6-((4-acetylpiperazin-1-yl)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)-4-(4-fluorophenethyl)piperazin-2-one 363239 N-(4-fluorophenyl)-N-methyl-4-oxo-5-(4-(piperidin-1-ylmethyl)phenethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carboxamide 363240 N-(2-(3-methylpyrrolidin-1-yl)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363241 (S)-N-(6-((dimethylamino)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)-6-(4-fluorophenyl)-N-methylnicotinamide 363242 2-((((S)-6-(4-(4-fluorophenethyl)-2-oxopiperazin-1-yl)-5,6,7,8-tetrahydronaphthalen-2-yl)methyl)(methyl)amino)-3-hydroxy-N,N-dimethylpropanamide 363243 N-(1-((1H-indol-5-yl)methyl)piperidin-4-yl)-7-fluoro-4-oxo-4H-chromene-2-carboxamide 363244 methyl 1-(6-(3-(4-(trifluoromethyl)phenyl)propanamido)quinolin-2-yl)pyrrolidine-2-carboxylate 363245 (S)-4-(5-chloropyridin-2-yl)-N-(6-((dimethylamino)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)-N-methylbenzamide 363246 N-(1-((1H-indol-6-yl)methyl)piperidin-4-yl)-7-fluoro-4-oxo-4H-chromene-2-carboxamide 363247 N-(2-(3-phenylpyrrolidin-1-yl)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363248 (S)-N-(6-((dimethylamino)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)-N-methyl-4-(pyridin-2-yl)benzamide 363249 N-(1-(benzofuran-5-ylmethyl)piperidin-4-yl)-7-fluoro-4-oxo-4H-chromene-2-carboxamide 363250 N-(1-(benzo[d]oxazol-6-ylmethyl)piperidin-4-yl)-7-fluoro-4-oxo-4H-chromene-2-carboxamide 363251 N-(2-(3-aminopyrrolidin-1-yl)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363252 (S)-4-(4-fluorophenethyl)-1-(6-((2,2,2-trifluoroethylamino)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-2-one 363253 N-(1-(benzo[b]thiophen-5-ylmethyl)piperidin-4-yl)-7-fluoro-4-oxo-4H-chromene-2-carboxamide 363254 N-(2-(dimethylamino)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363255 (S)-5-(4-chlorophenyl)-N-(6-((dimethylamino)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)-N-methylpicolinamide 363256 1-((S)-6-(((2R,6S)-2,6-dimethylpiperidin-1-yl)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)-4-(4-fluorophenethyl)piperazin-2-one 363257 N-(2-(3-acetamidopyrrolidin-1-yl)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363258 N-(2-(piperidin-1-yl)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363259 (S)-6-(4-chlorophenyl)-N-(6-((dimethylamino)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)-N-methylnicotinamide 363260 (S)-4-(4-fluorophenethyl)-1-(6-(morpholinomethyl)-1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-2-one 363261 (S)-4-(4-fluorophenethyl)-1-(6-((4-(methylsulfonyl)piperazin-1-yl)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-2-one 363262 N-(1-(6-(3-(4-(trifluoromethyl)phenyl)propanamido)quinolin-2-yl)pyrrolidin-3-yl)benzamide 363263 (S)-N-(6-((dimethylamino)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)-5-(4-fluorophenyl)-N-methylpicolinamide 363264 N-(1-(6-acetamido-2,3-dihydro-1H-inden-1-yl)piperidin-4-yl)-7-fluoro-4-oxo-4H-chromene-2-carboxamide 363265 1-((S)-6-((diethylamino)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)-4-(2-(tetrahydrothiophen-2-yl)ethyl)piperazin-2-one 363266 N-(2-(3-isobutyramidopyrrolidin-1-yl)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363267 (S)-N-(6-((4-acetylpiperazin-1-yl)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)-4'-fluoro-N-methylbiphenyl-4-carboxamide 363268 (S)-4-(4-fluorophenethyl)-1-(6-((4-(trifluoromethyl)piperidin-1-yl)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-2-one 363269 N-(2-(2-azabicyclo[2.2.2]octan-2-yl)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363270 (R)-N-(5-guanidino-1-oxo-1-(4-(trifluoromethyl)benzylamino)pentan-2-yl)-7-methoxybenzofuran-2-carboxamide 363272 5-(4-((diethylamino)methyl)phenethyl)-4-oxo-N-(4-(trifluoromethyl)phenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carboxamide 363273 5-(4-((dimethylamino)methyl)phenethyl)-N-(4-fluorophenyl)-4-oxo-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carboxamide 363274 7-fluoro-N-(1-((1-methyl-2-oxo-1,2-dihydroquinolin-7-yl)methyl)piperidin-4-yl)-4-oxo-4H-chromene-2-carboxamide 363275 7-fluoro-4-oxo-N-(1-((2-oxo-2H-chromen-7-yl)methyl)piperidin-4-yl)-4H-chromene-2-carboxamide 363277 7-fluoro-4-oxo-N-(1-((2-oxobenzo[d][1,3]dioxol-5-yl)methyl)piperidin-4-yl)-4H-chromene-2-carboxamide 363278 (E)-N-(4-amino-2-ethylquinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)acrylamide 363279 3-(3-chloro-4-fluorophenyl)-1-(6-cyano-1,2,3,4-tetrahydronaphthalen-2-yl)-1-(3-(4-methylpiperazin-1-yl)propyl)urea 363280 7-fluoro-4-oxo-N-(1-((3-oxo-3,4-dihydro-2H-benzo[b][1,4]oxazin-7-yl)methyl)piperidin-4-yl)-4H-chromene-2-carboxamide 363281 N-(1-(3-acetamidobenzyl)piperidin-4-yl)-7-fluoro-4-oxo-4H-chromene-2-carboxamide 363282 3-(3-chloro-4-fluorophenyl)-1-(6-methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)-1-(3-(4-methylpiperazin-1-yl)propyl)urea 363283 7-fluoro-4-oxo-N-(1-((3-oxo-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)methyl)piperidin-4-yl)-4H-chromene-2-carboxamide 363284 1-(4-amino-2-propylquinolin-6-yl)-3-(4-(trifluoromethyl)benzyl)urea 363285 (E)-N-(4-amino-2-butylquinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)acrylamide 363286 3-(3-chloro-4-fluorophenyl)-1-(7-methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)-1-(3-(4-methylpiperazin-1-yl)propyl)urea 363287 7-fluoro-4-oxo-N-(1-((2-oxo-1,2-dihydroquinolin-7-yl)methyl)piperidin-4-yl)-4H-chromene-2-carboxamide 363288 2-propyl-N6-(3-(4-(trifluoromethyl)phenyl)propyl)quinoline-4,6-diamine 363289 (R)-5-fluoro-N-(5-guanidino-1-oxo-1-(4-(trifluoromethyl)benzylamino)pentan-2-yl)-1H-indole-2-carboxamide 363290 (E)-N-(4-amino-2-tert-butylquinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)acrylamide 363291 N-(2-(3-(3-methylureido)pyrrolidin-1-yl)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363292 4-amino-2-propyl-N-(4-(trifluoromethyl)phenethyl)quinoline-6-carboxamide 363293 (R)-N-(5-guanidino-1-oxo-1-(4-(trifluoromethyl)benzylamino)pentan-2-yl)benzo[b]thiophene-2-carboxamide 363294 (E)-N-(4-amino-2-neopentylquinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)acrylamide 363295 1-(6-(3-(4-(trifluoromethyl)phenyl)propanamido)quinolin-2-yl)pyrrolidin-3-ylsulfamic acid 363296 (R)-N-(5-guanidino-1-oxo-1-(4-(trifluoromethyl)benzylamino)pentan-2-yl)-9,10-dihydroanthracene-9-carboxamide 363297 (E)-N-(4-amino-2-cyclobutylquinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)acrylamide 363298 N-(2-(2-azabicyclo[2.2.1]heptan-2-yl)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363299 (R)-N-(5-guanidino-1-oxo-1-(4-(trifluoromethyl)benzylamino)pentan-2-yl)-1H-indole-2-carboxamide 363300 (E)-N-(4-amino-2-cyclopentylquinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)acrylamide 363301 (R)-N-(5-guanidino-1-oxo-1-(4-(trifluoromethyl)benzylamino)pentan-2-yl)-9H-xanthene-9-carboxamide 363302 7-(4-fluorophenethyl)-2-(4-(piperidin-1-ylmethyl)phenethyl)-3,4-dihydropyrrolo[1,2-a]pyrazin-1(2H)-one 363304 (R)-N-(5-guanidino-1-oxo-1-(4-(trifluoromethyl)benzylamino)pentan-2-yl)quinoline-3-carboxamide 363305 7-(4-fluorophenyl)-2-(4-(piperidin-1-ylmethyl)phenethyl)-3,4-dihydropyrrolo[1,2-a]pyrazin-1(2H)-one 363306 3-(3-chloro-4-fluorophenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)-1-(1,2,3,4-tetrahydronaphthalen-2-yl)urea 363307 (S)-N-(6-((4-acetylpiperazin-1-yl)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)-N-methyl-4-(pyridin-2-yl)benzamide 363308 2-(4-chlorophenoxy)-N-(2-morpholinoquinolin-6-yl)acetamide 363309 1-(6-{13-[4-(trifluoromethyl)phenyl]tridecanamido}quinolin-2-yl)-1-azabicyclo[2.2.2]octan-1-ylium 363310 (R)-N-(5-guanidino-1-oxo-1-(4-(trifluoromethyl)benzylamino)pentan-2-yl)-9H-fluorene-9-carboxamide 363311 1-(6-bromo-1,2,3,4-tetrahydronaphthalen-2-yl)-3-(3-chloro-4-fluorophenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)urea 363313 (E)-N-(4-amino-2-pentylquinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)acrylamide 363314 (S)-6-(4-fluorophenyl)-N-methyl-N-(6-((3-oxopiperazin-1-yl)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)nicotinamide 363315 (R)-2-(2,2-diphenylacetamido)-5-guanidino-N-(4-(trifluoromethyl)benzyl)pentanamide 363316 (E)-N-(4-amino-2-isopropylquinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)acrylamide 363317 5-(4-((diethylamino)methyl)phenethyl)-4-oxo-N-(3-(trifluoromethyl)phenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carboxamide 363319 3-(3-chloro-4-fluorophenyl)-1-((1R,3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(3-(4-methylpiperazin-1-yl)propyl)urea 363320 (E)-N-(4-amino-2-sec-butylquinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)acrylamide 363321 7-(4-fluorobenzoyl)-2-(4-(piperidin-1-ylmethyl)phenethyl)-3,4-dihydropyrrolo[1,2-a]pyrazin-1(2H)-one 363322 (R)-N-(5-guanidino-1-oxo-1-(4-(trifluoromethyl)benzylamino)pentan-2-yl)benzofuran-2-carboxamide 363323 7-(4-fluorobenzyl)-2-(4-(piperidin-1-ylmethyl)phenethyl)-3,4-dihydropyrrolo[1,2-a]pyrazin-1(2H)-one 363324 3-(3-chloro-4-fluorophenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)-1-(7-nitro-1,2,3,4-tetrahydronaphthalen-2-yl)urea 363325 7-(3-(3-chloro-4-fluorophenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)ureido)-N-methyl-5,6,7,8-tetrahydronaphthalene-2-sulfonamide 363326 (R)-N-(5-guanidino-1-oxo-1-(4-(trifluoromethyl)benzylamino)pentan-2-yl)isoquinoline-3-carboxamide 363327 (R)-2-(2-(1H-indol-2-yl)acetamido)-5-guanidino-N-(4-(trifluoromethyl)benzyl)pentanamide 363328 (R)-N-(5-guanidino-1-oxo-1-(4-(trifluoromethyl)benzylamino)pentan-2-yl)benzo[b]thiophene-3-carboxamide 363329 N-(2-(2-oxa-5-azabicyclo[2.2.1]heptan-5-yl)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363330 7-(3-(3-chloro-4-fluorophenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)ureido)-N,N-dimethyl-5,6,7,8-tetrahydronaphthalene-2-sulfonamide 363331 (R)-N-(5-guanidino-1-oxo-1-(4-(trifluoromethyl)benzylamino)pentan-2-yl)-2-naphthamide 363332 N-(2-((2-(dimethylamino)ethyl)(methyl)amino)-4-methylquinazolin-6-yl)-2-(4-(trifluoromethyl)phenoxy)acetamide 363333 N-(2-(2,5-diazabicyclo[2.2.1]heptan-2-yl)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363334 N-(2-(diethylamino)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363335 (R)-5-guanidino-2-(2-(naphthalen-1-yl)acetamido)-N-(4-(trifluoromethyl)benzyl)pentanamide 363336 N-(2-(pyrrolidin-1-yl)-1H-benzo[d]imidazol-6-yl)-2-(4-(trifluoromethyl)phenoxy)acetamide 363337 N-(2-(2,7-diazaspiro[4.4]nonan-2-yl)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363338 (E)-N-(4-amino-2-cyclohexylquinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)acrylamide 363339 2-(2-chlorophenoxy)-N-(4-methyl-2-(pyrrolidin-1-yl)quinazolin-6-yl)acetamide 363340 N-(1-methyl-2-(pyrrolidin-1-yl)-1H-benzo[d]imidazol-6-yl)-2-(4-(trifluoromethyl)phenoxy)acetamide 363342 (E)-N-(4-amino-2-phenylquinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)acrylamide 363343 3-(3-chloro-4-fluorophenyl)-1-(7-cyano-1,2,3,4-tetrahydronaphthalen-2-yl)-1-(3-(4-methylpiperazin-1-yl)propyl)urea 363344 2-(4-methoxyphenoxy)-N-(4-methyl-2-(pyrrolidin-1-yl)quinazolin-6-yl)acetamide 363345 N-(4-(dimethylamino)-2-propylquinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363347 (R)-N-(5-guanidino-1-oxo-1-(4-(trifluoromethyl)benzylamino)pentan-2-yl)quinoline-2-carboxamide 363348 N-(7-(3-(3-chloro-4-fluorophenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)ureido)-5,6,7,8-tetrahydronaphthalen-2-yl)isobutyramide 363349 N-(2-aminoquinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363350 (R)-N-(5-guanidino-1-oxo-1-(4-(trifluoromethyl)benzylamino)pentan-2-yl)quinoline-4-carboxamide 363351 3-hydroxy-N-(1-(naphthalen-2-ylmethyl)piperidin-4-yl)benzamide 363352 N-(4-methyl-2-(pyrrolidin-1-yl)quinazolin-6-yl)-2-(4-(trifluoromethyl)phenoxy)acetamide 363353 N-(7-(3-(3-chloro-4-fluorophenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)ureido)-5,6,7,8-tetrahydronaphthalen-2-yl)methanesulfonamide 363354 (S)-N-(6-((dimethylamino)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)-N-methyl-4-(pyridin-3-yl)benzamide 363355 (R)-4-fluoro-N-(5-guanidino-1-oxo-1-(4-(trifluoromethyl)benzylamino)pentan-2-yl)-1-naphthamide 363356 2-(4-chlorophenoxy)-N-(4-methyl-2-(pyrrolidin-1-yl)quinazolin-6-yl)acetamide 363357 N-(4-fluorophenyl)-1-oxo-2-(4-(piperidin-1-ylmethyl)phenethyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazine-7-carboxamide 363358 (R)-N-(5-guanidino-1-oxo-1-(4-(trifluoromethyl)benzylamino)pentan-2-yl)-6-methoxy-2-naphthamide 363359 1-(7-amino-1,2,3,4-tetrahydronaphthalen-2-yl)-3-(3-chloro-4-fluorophenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)urea 363360 (E)-N-(4-(cyclobutylamino)-2-propylquinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)acrylamide 363362 N-(2-morpholinoquinolin-6-yl)-2-(4-(trifluoromethyl)phenoxy)acetamide 363363 N-(7-(3-(3-chloro-4-fluorophenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)ureido)-5,6,7,8-tetrahydronaphthalen-2-yl)acetamide 363364 (E)-N-(4-(dimethylamino)-2-propylquinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)acrylamide 363365 (S)-N-(6-((dimethylamino)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)-N-methyl-5-phenylpicolinamide 363366 N-(2-(piperazin-1-ylmethyl)quinolin-6-yl)-2-(4-(trifluoromethyl)phenoxy)acetamide 363367 (E)-N-(4-methoxy-2-propylquinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)acrylamide 363368 (E)-N-(4-(diethylamino)-2-propylquinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)acrylamide 363370 3-(3-chloro-4-fluorophenyl)-1-(3-(4-methylpiperazin-1-yl)propyl)-1-(7-(methylsulfonyl)-1,2,3,4-tetrahydronaphthalen-2-yl)urea 363371 (E)-N-(4-(methylamino)-2-propylquinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)acrylamide 363372 (E)-N-(4-(ethylamino)-2-propylquinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)acrylamide 363380 3,5-dimethoxy-N-(1-((6-methoxynaphthalen-2-yl)methyl)piperidin-4-yl)benzamide 363382 ((S)-1-(difluoro-1H-benzo[d]imidazol-2-yl)(3-(4-methylpiperazin-1-yl)propyl)amino)bicyclo[4.1.0]heptan-1-yl)benzyl)pyrrolidin-2-yl)methanol 363383 N-(4-amino-2-propylquinolin-6-yl)cinnamamide 363384 (E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-bromophenyl)acrylamide 363385 (E)-N-(4-amino-2-propylquinolin-6-yl)-3-(2,4-dichlorophenyl)acrylamide 363386 (S)-N-(6-((dimethylamino)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)-4'-fluoro-N-methylbiphenyl-4-carboxamide 363387 (S)-4-((6-(4'-fluoro-N-methylbiphenyl-4-ylcarboxamido)-5,6,7,8-tetrahydronaphthalen-2-yl)methyl)piperazine-1-carboxamide 363388 (R)-N-(5-guanidino-1-oxo-1-(4-(trifluoromethyl)benzylamino)pentan-2-yl)-5-methoxy-1H-indole-2-carboxamide 363389 (R)-2-(2-(benzo[b]thiophen-3-yl)acetamido)-5-guanidino-N-(4-(trifluoromethyl)benzyl)pentanamide 363390 2-(3-chlorophenoxy)-N-(4-methyl-2-(pyrrolidin-1-yl)quinazolin-6-yl)acetamide 363391 N-(2-((2-(dimethylamino)ethyl)(methyl)amino)-1-methyl-1H-benzo[d]imidazol-6-yl)-2-(4-(trifluoromethyl)phenoxy)acetamide 363392 1-(3-chloro-4-fluorophenyl)-3-{7-[(ethylcarbamoyl)amino]-1,2,3,4-tetrahydronaphthalen-2-yl}-3-[3-(4-methylpiperazin-1-yl)propyl]urea 363393 N-(2-(dipropylamino)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363394 N-(2-(azepan-1-yl)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide 363395 (E)-N-(4-(cyclopropylamino)-2-propylquinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)acrylamide 363822 7-amino-19-methyl-3-(2-methylpropyl)-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-14-one 363823 3-{3-ethyl-19-methyl-14-oxo-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl}-1-(4-methoxyphenyl)urea 363831 naphthalen-1-yl(5-phenyl-1-propyl-1H-pyrrol-3-yl)methanone 363832 1-(4-methoxyphenyl)-3-{19-methyl-14-oxo-3-propyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl}urea 363837 (1-butyl-5-phenyl-1H-pyrrol-3-yl)(naphthalen-1-yl)methanone 363838 naphthalen-1-yl(1-pentyl-5-phenyl-1H-pyrrol-3-yl)methanone 363839 3-{19-methyl-14-oxo-3-propyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl}-1-[4-(methylsulfanyl)phenyl]urea 363844 (1-hexyl-5-phenyl-1H-pyrrol-3-yl)(naphthalen-1-yl)methanone 363845 (1-heptyl-5-phenyl-1H-pyrrol-3-yl)(naphthalen-1-yl)methanone 363846 3-{10-carboximidoyl-5-oxo-14-propyl-4,14-diazapentacyclo[11.7.0.0^{2,6}.0^{7,12}.0^{15,20}]icosa-1(13),2(6),7(12),9,15,17,19-heptaen-18-yl}-1-(4-methylphenyl)urea 363852 naphthalen-1-yl(1-pentyl-5-o-tolyl-1H-pyrrol-3-yl)methanone 363853 (5-(2-ethylphenyl)-1-pentyl-1H-pyrrol-3-yl)(naphthalen-1-yl)methanone 363854 3-{19-methyl-14-oxo-3-propyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl}-1-(thiophen-2-yl)urea 363858 (5-(2-butylphenyl)-1-pentyl-1H-pyrrol-3-yl)(naphthalen-1-yl)methanone 363859 (5-(2-methoxyphenyl)-1-pentyl-1H-pyrrol-3-yl)(naphthalen-1-yl)methanone 363860 1-(2-fluoro-5-methylphenyl)-3-{19-methyl-14-oxo-3-propyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl}urea 363864 (5-(2-fluorophenyl)-1-pentyl-1H-pyrrol-3-yl)(naphthalen-1-yl)methanone 363865 (5-(2-chlorophenyl)-1-pentyl-1H-pyrrol-3-yl)(naphthalen-1-yl)methanone 363866 3-{19-methyl-14-oxo-3-propyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl}-1-phenylurea 363871 naphthalen-1-yl(1-pentyl-5-(2-(trifluoromethyl)phenyl)-1H-pyrrol-3-yl)methanone 363872 naphthalen-1-yl(1-pentyl-5-m-tolyl-1H-pyrrol-3-yl)methanone 363873 1-methyl-3-{19-methyl-14-oxo-3-propyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl}-1-phenylurea 363879 (5-(3-methoxyphenyl)-1-pentyl-1H-pyrrol-3-yl)(naphthalen-1-yl)methanone 363880 (5-(3-fluorophenyl)-1-pentyl-1H-pyrrol-3-yl)(naphthalen-1-yl)methanone 363881 1-(4-fluorophenyl)-3-{19-methyl-14-oxo-3-propyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl}urea 363886 (5-(3-chlorophenyl)-1-pentyl-1H-pyrrol-3-yl)(naphthalen-1-yl)methanone 363887 naphthalen-1-yl(1-pentyl-5-(3-(trifluoromethyl)phenyl)-1H-pyrrol-3-yl)methanone 363888 1-(3-fluorophenyl)-3-{19-methyl-14-oxo-3-propyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl}urea 363893 naphthalen-1-yl(5-(3-nitrophenyl)-1-pentyl-1H-pyrrol-3-yl)methanone 363894 naphthalen-1-yl(1-pentyl-5-p-tolyl-1H-pyrrol-3-yl)methanone 363895 1-(2-fluorophenyl)-3-{19-methyl-14-oxo-3-propyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl}urea 363900 (5-(4-ethylphenyl)-1-pentyl-1H-pyrrol-3-yl)(naphthalen-1-yl)methanone 363901 (5-(4-butylphenyl)-1-pentyl-1H-pyrrol-3-yl)(naphthalen-1-yl)methanone 363902 1-(4-chlorophenyl)-3-{19-methyl-14-oxo-3-propyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl}urea 363907 (5-(4-methoxyphenyl)-1-pentyl-1H-pyrrol-3-yl)(naphthalen-1-yl)methanone 363908 (5-(4-fluorophenyl)-1-pentyl-1H-pyrrol-3-yl)(naphthalen-1-yl)methanone 363909 1-(2-chlorophenyl)-3-{19-methyl-14-oxo-3-propyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl}urea 363915 1-(4-methoxyphenyl)-3-[19-methyl-3-(2-methylpropyl)-14-oxo-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl]urea 363916 3-{3-butyl-19-methyl-14-oxo-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl}-1-(4-methoxyphenyl)urea 363917 1-[4-(dimethylamino)phenyl]-3-{19-methyl-14-oxo-3-propyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl}urea 363918 1-[2-fluoro-5-(trifluoromethyl)phenyl]-3-{19-methyl-14-oxo-3-propyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl}urea 363919 1-(3-methoxyphenyl)-3-[19-methyl-3-(2-methylpropyl)-14-oxo-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl]urea 363920 1-(2-methoxyphenyl)-3-[19-methyl-3-(2-methylpropyl)-14-oxo-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl]urea 363921 (5-(4-chlorophenyl)-1-pentyl-1H-pyrrol-3-yl)(naphthalen-1-yl)methanone 363922 naphthalen-1-yl(1-pentyl-5-(4-(trifluoromethyl)phenyl)-1H-pyrrol-3-yl)methanone 363931 naphthalen-1-yl(5-(naphthalen-1-yl)-1-pentyl-1H-pyrrol-3-yl)methanone 363932 naphthalen-1-yl(5-(naphthalen-2-yl)-1-pentyl-1H-pyrrol-3-yl)methanone 363940 naphthalen-1-yl(1-pentyl-5-(pyridin-3-yl)-1H-pyrrol-3-yl)methanone 363941 7-amino-19-methyl-3-propyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-14-one 363948 N-{19-methyl-14-oxo-3-propyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl}furan-2-carboxamide 363955 N-[19-methyl-3-(2-methylpropyl)-14-oxo-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl]furan-2-carboxamide 363962 4-methoxyphenyl N-{19-methyl-14-oxo-3-propyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl}carbamate 363967 4-fluorophenyl N-{19-methyl-14-oxo-3-propyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl}carbamate 363974 propan-2-yl N-{19-methyl-14-oxo-3-propyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl}carbamate 363975 ethyl N-{19-methyl-14-oxo-3-propyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl}carbamate 363984 propyl N-{19-methyl-14-oxo-3-propyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl}carbamate 363990 N-(6-((3S,8aS)-3-benzyl-hexahydropyrrolo[1,2-a]pyrazin-2(1H)-yl)-6-oxohexyl)-3-(1H-indol-3-yl)propanamide 364004 1-((3S,8aS)-3-benzyl-hexahydropyrrolo[1,2-a]pyrazin-2(1H)-yl)-3-(1H-indol-3-yl)propan-1-one 364005 1-((3R,8aS)-3-benzyl-hexahydropyrrolo[1,2-a]pyrazin-2(1H)-yl)-3-(1H-indol-3-yl)propan-1-one 364006 7-amino-3-butyl-19-methyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-14-one 364011 N-[(S)-1-((3S,8aS)-3-benzyl-hexahydro-pyrrolo[1,2-a]pyrazine-2-carbonyl)-4-guanidino-butyl]-3-(1H-indol-3-yl)-propionamide 364017 1-((3S,8aS)-3-benzyl-hexahydropyrrolo[1,2-a]pyrazin-2(1H)-yl)-2-phenylethanone 364018 1-((3R,8aS)-3-benzyl-hexahydropyrrolo[1,2-a]pyrazin-2(1H)-yl)-2-phenylethanone 364024 N-(2-(1H-indol-3-yl)ethyl)-4-((3S,8aS)-3-benzyl-hexahydropyrrolo[1,2-a]pyrazin-2(1H)-yl)-4-oxobutanamide 364025 N-(2-(1H-indol-3-yl)ethyl)-4-((3R,8aS)-3-benzyl-hexahydropyrrolo[1,2-a]pyrazin-2(1H)-yl)-4-oxobutanamide 364038 1-(2-bromophenyl)-3-{19-methyl-14-oxo-3-propyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl}urea 364043 N-{19-methyl-14-oxo-3-propyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl}thiophene-2-carboxamide 364050 N-[19-methyl-3-(2-methylpropyl)-14-oxo-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-7-yl]thiophene-2-carboxamide 364055 (S)-2-pyrrolidin-1-ylmethyl-pyrrolidine-1-carboxylic acid biphenyl-4-ylmethyl-methyl-amide 364056 4-isopropyl-piperazine-1-carboxylic acid biphenyl-4-ylmethyl-methyl-amide 364063 (S)-isoindolin-2-yl(2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl)methanone 364064 isoindolin-2-yl(4-isopropylpiperazin-1-yl)methanone 364065 (4-cyclopropylpiperazin-1-yl)(isoindolin-2-yl)methanone 364072 (4-cyclopentylpiperazin-1-yl)(isoindolin-2-yl)methanone 364073 N-(1-(1-isopropylpiperazine-4-carbonyl)piperidin-4-yl)cyclopentanecarboxamide 364080 [4-(3-Aza-bicyclo[3.2.2]nonane-3-carbonyl)-piperidin-1-yl]-(4-isopropyl-piperazin-1-yl)-methanone 364081 tert-butyl 1-(1-isopropylpiperazine-4-carbonyl)piperidine-4-carboxylate 364088 (4-benzylpiperidin-1-yl)(4-isopropylpiperazin-1-yl)methanone 364089 (4-tert-butylpiperidin-1-yl)(4-isopropylpiperazin-1-yl)methanone 364090 (3,4-dihydroisoquinolin-2(1H)-yl)(4-isopropylpiperazin-1-yl)methanone 364095 (S,E)-1-(2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl)-3-(4-(trifluoromethyl)phenyl)prop-2-en-1-one 364096 (S)-3-(4-chlorophenyl)-1-(2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl)prop-2-en-1-one 364097 (6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)(4-isopropylpiperazin-1-yl)methanone 364098 (4-isopropylpiperazin-1-yl)(4-phenylpiperidin-1-yl)methanone 364099 (4-isopropylpiperazin-1-yl)(4-phenyl-5,6-dihydropyridin-1(2H)-yl)methanone 364104 (S)-1-(2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl)-3-(4-(trifluoromethoxy)phenyl)prop-2-en-1-one 364105 3-biphenyl-4-yl-1-((S)-2-pyrrolidin-1-ylmethyl-pyrrolidin-1-yl)-propenone 364112 (S)-N-(4-(trifluoromethyl)benzyl)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carboxamide 364113 (S)-N-(4-chlorobenzyl)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carboxamide 364119 5-(4-hydroxy-2,6-dimethylstyryl)nicotinic acid 364120 (S)-N-(4-(trifluoromethoxy)benzyl)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carboxamide 364121 (S)-2-pyrrolidin-1-ylmethyl-pyrrolidine-1-carboxylic acid (biphenyl-4-ylmethyl)-amide 364128 3,5-dimethyl-4-{(E)-2-[5-(1H-tetrazol-5-yl)-3-pyridinyl]ethenyl}phenol 364129 (S)-N-benzyl-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carboxamide 364130 (S)-N-(4-methoxybenzyl)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carboxamide 364131 (S)-N-(3-methoxybenzyl)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carboxamide 364138 (S)-N-(3-(trifluoromethyl)benzyl)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carboxamide 364139 (S)-N-(3-(aminomethyl)benzyl)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carboxamide 364140 (S)-N-(4-(aminomethyl)benzyl)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carboxamide 364141 SID26751979 364147 (S)-N-(4-phenoxybenzyl)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carboxamide 364148 (S)-N-(3,4-dichlorobenzyl)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carboxamide 364155 (S)-N-(cyclohexylmethyl)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carboxamide 364156 (S)-N-phenethyl-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carboxamide 364157 (S)-N-(2,3-dihydro-1H-inden-2-yl)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carboxamide 364165 N-benzyl-4-cyclopentylpiperazine-1-carboxamide 364166 4-cyclopentyl-N-(2,3-dihydro-1H-inden-2-yl)piperazine-1-carboxamide 364167 N-(2,3-dihydro-1H-inden-2-yl)-4-isopropylpiperazine-1-carboxamide 364174 N-(2,3-dihydro-1H-inden-2-yl)-4-ethylpiperazine-1-carboxamide 364175 4-ethyl-N-((1R,2S)-2-phenylcyclopropyl)piperazine-1-carboxamide 364176 N-(4-phenoxybenzyl)-4-cyclopentylpiperazine-1-carboxamide 364184 N-(4-phenoxybenzyl)-4-isopropylpiperazine-1-carboxamide 364185 N-(3,4-dichlorobenzyl)-4-cyclopentylpiperazine-1-carboxamide 364186 N-(3,4-dichlorobenzyl)-4-isopropylpiperazine-1-carboxamide 364398 3-((3R,7R,8R,9alpahR)-3-benzyl-7,8-dimethyl-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364399 3-((3S,7R,8R,9alphaR)-3-cyclohexyl-7,8-dimethyl-octahydro-1Hpyrido[1,2-R]pyrazin-8-yl)phenol 364400 3-((7R,8R,9alphaR)-2-(4-(dimethylamino)benzyl)-7,8-dimethyl-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364401 methyl 3-(((7R,8R,9alphaR)-8-(3-hydroxyphenyl)-7,8-dimethylhexahydro-1H-pyrido[1,2-R]pyrazin-2(6H)-yl)methyl)benzoate 364404 3-((3S,7R,8R,9alphaR)-3-isopropyl-7,8-dimethyl-octahydro-1Hpyrido[1,2-R]pyrazin-8-yl)phenol 364406 1-((7R,8R,9alphaR)-8-(3-hydroxyphenyl)-7,8-dimethyl-hexahydro-1H-pyrido[1,2-R]pyrazin-2(6H)-yl)ethanone 364407 3-((7R,8R,9alphaR)-7,8-dimethyl-2-(3-phenoxybenzyl)-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364408 3-((7R,8R,9alphaR)-2-(3-(benzyloxy)benzyl)-7,8-dimethyl-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364410 ((7R,8R,9alphaR)-8-(3-hydroxyphenyl)-7,8-dimethyl-hexahydro-1H-pyrido[1,2-R]pyrazin-2(6H)-yl)(phenyl)methanone 364411 1-((7R,8R,9alphaR)-8-(3-hydroxyphenyl)-7,8-dimethyl-hexahydro-1H-pyrido[1,2-R]pyrazin-2(6H)-yl)-2-phenylethanone 364412 3-((7R,8R,9alphaR)-7,8-dimethyl-2-(naphthalen-2-ylmethyl)-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364413 3-((7R,8R,9alphaR)-7,8-dimethyl-2-(naphthalen-1-ylmethyl)-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364416 1-((7R,8R,9alphaR)-8-(3-hydroxyphenyl)-7,8-dimethyl-hexahydro-1H-pyrido[1,2-R]pyrazin-2(6H)-yl)-3-phenylpropan-1-one 364417 3-((7R,8R,9alphaR)-7,8-dimethyl-2-phenyl-octahydro-1H-pyrido-[1,2-R]pyrazin-8-yl)phenol 364418 3-((7R,8R,9alphaR)-7,8-dimethyl-2-(quinolin-4-ylmethyl)-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364419 3-((7R,8R,9alphaR)-7,8-dimethyl-2-(pyridin-2-ylmethyl)-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364421 3-((7R,8R,9alphaR)-2-benzyl-7,8-dimethyl-octahydro-1H-pyrido-[1,2-R]pyrazin-8-yl)phenol 364422 3-((7R,8R,9alphaR)-7,8-dimethyl-2-phenethyl-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364423 3-((7R,8R,9alphaR)-7,8-dimethyl-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364424 3-((7R,8R,9alphaR)-7,8-dimethyl-2-(pyridin-4-ylmethyl)-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364426 3-((7R,8R,9alphaR)-7,8-dimethyl-2-(3-phenylpropyl)-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364427 3-((8R,9R,10alphaR)-2-benzyl-8,9-dimethyl-decahydropyrido[1,2-R][1,4]diazepin-9-yl)phenol 364428 3-((7R,8R,9alphaR)-2-(furan-2-ylmethyl)-7,8-dimethyl-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364429 3-((7R,8R,9alphaR)-2-(furan-3-ylmethyl)-7,8-dimethyl-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364432 3-((7R,8R,9alphaR)-7,8-dimethyl-2-(phenylsulfonyl)-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364433 3-((7R,8R,9alphaR)-7,8-dimethyl-2-(thiophen-2-ylmethyl)-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364434 3-((7R,8R,9alphaR)-7,8-dimethyl-2-(thiophen-3-ylmethyl)-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364436 (7R,8R,9alphaR)-8-(3-hydroxyphenyl)-7,8-dimethyl-N-phenylhexahydro-1H-pyrido[1,2-R]pyrazine-2(6H)-carboxamide 364437 3-((7R,8R,9alphaR)-7,8-dimethyl-2-(2-methylbenzyl)-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364438 3-((7R,8R,9alphaR)-2-(cyclohexylmethyl)-7,8-dimethyl-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364439 N6-methyl-9-(beta-D-ribofuranosyl)-2-(1,2,3-triazol-1-yl)adenine 364441 3-((7R,8R,9alphaR)-7,8-dimethyl-2-(3-methylbenzyl)-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364442 3-((7R,8R,9alphaR)-7,8-dimethyl-2-(4-methylbenzyl)-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364443 2-(4-ethyl-1,2,3-triazol-1-yl)-N6-methyl-9-(beta-D-ribofuranosyl)-adenine 364444 2-(4-butyl-1,2,3-triazol-1-yl)-N6-methyl-9-(beta-D-ribofuranosyl)-adenine 364447 3-((7R,8R,9alphaR)-7,8-dimethyl-2-(2-chlorobenzyl)-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364448 3-((7R,8R,9alphaR)-7,8-dimethyl-2-(3-chlorobenzyl)-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364449 2-[4-(2-hydroxyethyl)-1,2,3-triazol-1-yl]-N6-methyl-9-(beta-D-ribofuranosyl)adenine 364450 2-(4-dimethylaminomethyl-1,2,3-triazol-1-yl)-N6-methyl-9-(beta-D-ribofuranosyl)adenine 364453 3-((3S,7R,8R,9alphaR)-2-benzyl-7,8-dimethyl-3-phenyl-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364454 3-((7R,8R,9alphaR)-7,8-dimethyl-2-(4-chlorobenzyl)-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364455 2-(((7R,8R,9alphaR)-8-(3-hydroxyphenyl)-7,8-dimethyl-hexahydro-1H-pyrido[1,2-R]pyrazin-2(6H)-yl)methyl)phenol 364456 N6-methyl-2-(4-phenyl-1,2,3-triazol-1-yl)-9-(beta-D-ribofuranosyl) 364457 N6-methyl-2-[4-pyridin-2-yl-1,2,3-triazol-1-yl]-9-(beta-D-ribofuranosyl)adenine 364458 3-((2R,3R,7S,9-alpha-S)-2,3-dimethyl-7-phenyl-octahydro-1H-quinolizin-2-yl)phenol 364459 3-((3S,7R,8R,9alphaR)-7,8-dimethyl-3-phenyl-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364460 (3S,7R,8R,9alphaR)-2-benzyl-7,8-dimethyl-3,8-diphenyl-octahydro-1H-pyrido[1,2-R]pyrazine 364462 3-((7R,8R,9alphaR)-2-(3-hydroxybenzyl)-7,8-dimethyl-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364463 3-((7R,8R,9alphaR)-2-(4-hydroxybenzyl)-7,8-dimethyl-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364464 N6-methyl-2-[4-(4-propoxyphenyl)-1,2,3-triazol-1-yl]-9-(beta-D-ribofuranosyl)adenine 364465 N6-methyl-2-(4-benzyl-1,2,3-triazol-1-yl)-9-(beta-D-ribofuranosyl)adenine 364466 1-((3S,7R,8R,9alphaR)-8-(3-hydroxyphenyl)-7,8-dimethyl-3-phenyl-hexahydro-1H-pyrido[1,2-R]pyrazin-2(6H)-yl)ethanone 364467 3-((3S,7R,8R,9alphaR)-2,7,8-trimethyl-3-phenyl-octahydro-1Hpyrido[1,2-R]pyrazin-8-yl)phenol 364468 3-((3S,7R,8R,9alphaR)-2-benzyl-7,8-dimethyl-3-phenyl-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)benzoic acid 364469 3-((3S,7R,8R,9alphaR)-2-benzyl-7,8-dimethyl-3-phenyl-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)benzamide 364472 3-((3S,7R,8R,9alphaR)-7,8-dimethyl-3-phenyl-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)benzamide 364473 3-((3R,7R,8R,9alphaR)-7,8-dimethyl-3-phenyl-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364476 3-((3S,7R,8R,9alphaR)-3-benzyl-7,8-dimethyl-octahydro-1H-pyrido[1,2-R]pyrazin-8-yl)phenol 364479 9-(5-ethylcarbamoyl-beta-D-ribofuranosyl)-N6-methyl-2-(4-benzyl-1,2,3-triazol-1-yl)adenine 364480 2-(4-cyclopentylmethyl-1,2,3-triazol-1-yl)-9-(5-ethylcarbamoyl-beta-D-ribofuranosyl)-N6-methyladenine 364481 N-(3,3-diphenyl-2-propenyl)cyclobutanecarboxamide 364482 (Z)-N-[3-(3-methoxyphenyl)-3-phenyl-2-propenyl]acetamide 364483 N-(3-(3-methoxyphenyl)-3-phenylallyl)acetamide 364487 1-(2',4'-dichlorophenyl)-6-methyl-N-p-chlorophenyl-1,4-dihydroindeno[1,2-c]pyrazole-3-carboxamide 364489 N6-(5-chloro-2-methoxybenzyl)-2-(4-cyclopentylmethyl-1,2,3-triazol-1-yl)-9-(beta-D-ribofuranosyl)adenine 364490 2-azido-N6-methyl-9-(beta-D-ribofuranosyl)adenine 364491 (Z)-N-[3-(3-methoxyphenyl)-3-phenyl-2-propenyl]cyclobutancarboxamide 364492 (E)-N-[3-(3-methoxyphenyl)-3-phenyl-2-propenyl]cyclobutancarboxamide 364493 N-[3,3-bis-(3-methoxyphenyl)-2-propenyl]acetamide 364499 2-azido-9-(5-ethylcarbamoyl-beta-D-ribofuranosyl)-N6-methyladenine 364500 2-azido-N6-(5-chloro-2-methoxybenzyl)-9-(beta-D-ribofuranosyl)adenine 364501 1-(2',4'-dichlorophenyl)-6-methyl-N-p-methoxyphenyl-1,4-dihydroindeno[1,2-c]pyrazole-3-carbohydrazide 364502 7-chloro-1-(2',4'-dichlorophenyl)-6-methyl-N-cyclohexylamine-1,4-dihydroindeno[1,2-c]pyrazole-3-carboxamide 364511 7-chloro-1-(2',4'-dichlorophenyl)-6-methyl-N-piperidin-1-yl-1,4-dihydroindeno[1,2-c]pyrazole-3-carboxamide 364512 6-chloro-1-(2',4'-dichlorophenyl)-7-methyl-N-piperidin-1-yl-1,4-dihydroindeno[1,2-c]pyrazole-3-carboxamide 364519 1-(2',4'-dichlorophenyl)-6-methyl-N-p-fluorophenyl-1,4-dihydroindeno[1,2-c]pyrazole-3-carboxamide 364523 3-((2R,3R,7S,9RR)-2,3-dimethyl-7-phenyl-octahydro-1H-quinolizin-2-yl)phenol 364525 3-((2R,3R,7R,9-alpha-R)-2,3-dimethyl-7-phenyl-octahydro-1H-quinolizin-2-yl)phenol 364529 6-methyl-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4-dihydroindeno[1,2-c]pyrazole-3-carboxamide 364535 3-((2R,3R,7R,9-alpha-S)-2,3-dimethyl-7-phenyl-octahydro-1H-quinolizin-2-yl)phenol 364536 1-(2',4'-dichlorophenyl)-6-methyl-N-p-methylphenyl-1,4-dihydroindeno[1,2-c]pyrazole-3-carboxamide 364543 3-((1R,2R,7R,9-alpha-S)-1,2-dimethyl-7-phenyl-octahydro-1H-quinolizin-2-yl)phenol 364544 3-((1R,2R,7S,9-alpha-S)-1,2-dimethyl-7-phenyl-octahydro-1H-quinolizin-2-yl)phenol 364547 1,4-dihydroindeno[1,2-c]-pyrazole 364551 3-((1R,2R,7R,9-alpha-R)-1,2-dimethyl-7-phenyl-octahydro-1H-quinolizin-2-yl)phenol 364552 3-((1R,2R,7S,9-alpha-R)-1,2-dimethyl-7-phenyl-octahydro-1H-quinolizin-2-yl)phenol 364554 1-(2',4'-dichlorophenyl)-6-methyl-N-p-methoxyphenyl-1,4-dihydroindeno[1,2-c]pyrazole-3-carboxamide 364560 3-((2R,3R,9-alpha-R)-2,3-dimethyl-octahydro-1H-quinolizin-2-yl)-phenol 364561 3-((2R,3R,9-alpha-S)-2,3-dimethyl-octahydro-1H-quinolizin-2-yl)-phenol 364562 3-((1R,2R,9-alpha-S)-1,2-dimethyl-octahydro-1H-quinolizin-2-yl)phenol 364567 3-((1R,2R,9-alpha-R)-1,2-dimethyl-octahydro-1H-quinolizin-2-yl)phenol 364572 1-(2',4'-dichlorophenyl)-6-methyl-N-o,p-dichlorophenyl-1,4-dihydroindeno[1,2-c]pyrazole-3-carboxamide 364579 1-(2',4'-dichlorophenyl)-6-methyl-N-phenyl-1,4-dihydroindeno[1,2-c]purazole-3-carbohydrazide 364587 1-(2',4'-dichlorphenyl)-6-methyl-N-p-nitrophenyl-1,4-dihydroindeno[1,2-c]pyrazole-3-carbohydrazide 364592 2-(4-cyclopentylmethyl-1,2,3-triazol-1-yl)-N6-methyl-9-(beta-Dribofuranosyl)adenine 364593 2-(4-cyclohexylmethyl-1,2,3-triazol-1-yl)-N6-methyl-9-(beta-D-ribofuranosyl)adenine 364595 N-(2,3-diphenylpropyl)acetamide 364596 N-[2-(3-methoxyphenyl)-3-phenylpropyl]acetamide 364598 N-(3,3-diphenyl-propyl)acetamide 364600 (+/-)-N-[3-(3-methoxyphenyl)-3-phenylpropyl]acetamide 364601 (+/-)-N-[3-(3-methoxyphenyl)-3-phenylpropyl]propanamide 364607 2-(1-benzyl-1,2,3-triazol-4-yl)-N6-methyl-9-(beta-D-ribofuranosyl)adenine 364608 2-[1-(3-methoxybenzyl)-1,2,3-triazol-4-yl)-N6-methyl-9-(beta-D-ribofuranosyl)adenine 364609 N-[2-(3-methoxyphenyl)-3-phenylpropyl]propanamide 364610 (Z)-N-(2,3-diphenyl-2-propenyl)acetamide 364611 (E)-N-(2,3-diphenyl-2-propenyl)acetamide 364613 (+/-)-N-[3-(3-methoxyphenyl)-3-phenylpropyl)butanamide 364615 1-(2',4'-dichlorophenyl)-6-methyl-N-cyclohexylamine-1,4-dihydroindeno[1,2-c]pyrazole-3-carboxamide 364616 1-(2',4'-dichlorophenyl)-6-methyl-N-phenyl-1,4-dihydroindeno-[1,2-c]pyrazole-3-carboxamide 364617 2-[1-(3-chlorobenzyl)-1,2,3-triazol-4-yl)-N6-methyl-9-(beta-D-ribofuranosyl)adenine 364618 9-(5-ethylcarbamoyl-beta-D-ribofuranosyl)-N6-methyl-2-(1,2,3-triazol-1-yl)adenine 364619 N-{2-[(3-benzyl)phenyl]ethyl}propanamide 364620 N-[2-(2-benzyl-5-methoxyphenyl)ethyl]acetamide 364622 N-(3,3-diphenyl-2-propenyl)acetamide 364629 2-(4-butyl-1,2,3-triazol-1-yl)-9-(5-ethylcarbamoyl-beta-D-ribofuranosyl)-N6-methyladenine 364630 9-(5-ethylcarbamoyl-beta-D-ribofuranosyl)-N6-methyl-2-(4-pyridin-2-yl-1,2,3-triazol-1-yl)adenine 364633 N-(3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-ylmethyl)-benzamide 364634 2-methoxy-N-(3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-ylmethyl)-benzamide 364642 3-methyl-N-(3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-ylmethyl)benzamide 364649 6-(4-((1H-benzo[d]imidazol-2-yl)methyl)piperazin-1-yl)pyridin-3-ol 364680 N-(2-methyl-4-fluorophenyl)-2-(1-oxy-3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-yl)acetamide 364685 2-(3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-yl)-N-(m-tolyl)acetamide 364742 methyl-N-(1-oxy-3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'ylmethyl)benzamide 364743 2-(1-oxy-3',4',5',6'-tetrahydro-2'H-[2,4'bipyridine]-1'-yl)-N-(m-tolyl)acetamide 364745 SID4254117 364796 N-[2,3-bis(4-chlorophenyl)-1-methylpropyl]-2-(4-chlorophenyloxy)-2-methylpropanamide 364797 (1S,2S)N-[2,3-bis(4-chlorophenyl)-1-methylpropyl]-2-(4-chlorophenyloxy)-2-methylpropanamide 364832 3-(3,4-dioxo-2-(pentan-3-ylamino)cyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide 364833 3-(2-(benzylamino)-3,4-dioxocyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide 364838 N-[3-(4-chlorophenyl)-1-methyl-2-phenylpropyl]-2-(4-chlorophenyloxy)-2-methylpropanamide 364842 (S)-3-(3,4-dioxo-2-(1-phenylethylamino)cyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide 364843 tri(propylene glycol)(3-methoxy-1,2,5-thiadiazol-4-yl) [3-(1-methyl-1,2,5,6-tetrahydropyrid-3-yl)-1,2,5-thiadiazol-4-yl] ether 364844 tri(propylene glycol)(3-methoxy-1,2,4-thiadiazol-5-yl) [3-(1-methyl-1,2,5,6-tetrahydropyrid-3-yl)-1,2,5-thiadiazol-4-yl] ether 364849 (S)-3-(3,4-dioxo-2-(1-phenylpropylamino)cyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide 364855 (R)-3-(2-(1-(benzo[d][1,3]dioxol-5-yl)propylamino)-3,4-dioxocyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide 364856 N-[(1S,2S)-3-(4-chlorophenyl)-1-methyl-2-phenylpropyl]-2-(5-chloropyridyloxy)-2-methylpropanamide 364860 (R)-3-(3,4-dioxo-2-(1-(thiophen-2-yl)propylamino)cyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide 364861 (R)-3-(2-(1-(furan-2-yl)propylamino)-3,4-dioxocyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide 364874 (R)-2-hydroxy-N,N-dimethyl-3-(2-(1-(5-methylthiophen-2-yl)propylamino)-3,4-dioxocyclobut-1-enylamino)benzamide 364875 (R)-2-hydroxy-N,N-dimethyl-3-(2-(1-(5-methylfuran-2-yl)propylamino)-3,4-dioxocyclobut-1-enylamino)benzamide 364900 N-[(1S,2S)-3-(4-chlorophenyl)-1-methyl-2-phenylpropyl]-2-(3-chlorophenyloxy)-2-methylpropanamide 364904 (R)-2-hydroxy-N,N-dimethyl-3-(2-(1-(5-methylfuran-2-yl)ethylamino)-3,4-dioxocyclobut-1-enylamino)benzamide 364905 (R)-3-(2-(cyclopropyl(5-methylfuran-2-yl)methylamino)-3,4-dioxocyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide 364932 N-((2S,3S)-4-(4-chlorophenyl)-3-phenylbutan-2-yl)-2-methyl-2-phenoxypropanamide 364933 N-[(1S,2S)-3-(4-chlorophenyl)-1-methyl-2-phenylpropyl]-2-(3-fluorophenyloxy)-2-methylpropanamide 364937 (R)-2-hydroxy-N,N-dimethyl-3-(2-(2-methyl-1-(5-methylfuran-2-yl)propylamino)-3,4-dioxocyclobut-1-enylamino)benzamide 364938 (R)-3-(2-(2,2-dimethyl-1-(5-methylfuran-2-yl)propylamino)-3,4-dioxocyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide 364940 N-((2S,3S)-4-(4-chlorophenyl)-3-phenylbutan-2-yl)-2-(3,5-difluorophenoxy)-2-methylpropanamide 364941 N-((2S,3S)-4-(4-chlorophenyl)-3-phenylbutan-2-yl)-2-methyl-2-(pyridin-2-yloxy)propanamide 364953 tetra(ethylene glycol)(3-methoxy-1,2,5-thiadiazol-4-yl)[3-(1-methyl-1,2,5,6-tetrahydropyrid-3-yl)-1,2,5-thiadiazol-4-yl] ether 364954 penta(ethylene glycol)(3-methoxy-1,2,5-thiadiazol-4-yl) [3-(1-methyl-1,2,5,6-tetrahydropyrid-3-yl)-1,2,5-thiadiazol-4-yl] ether 364970 di(ethylene glycol)(3-methoxy-1,2,5-thiadiazol-4-yl) [3-(1-methyl-1,2,5,6-tetrahydropyrid-3-yl)-1,2,5-thiadiazol-4-yl] ether 364971 tri(ethylene glycol)(3-methoxy-1,2,5-thiadiazol-4-yl) [3-(1-methyl-1,2,5,6-tetrahydropyrid-3-yl)-1,2,5-thiadiazol-4-yl] ether 364972 2-(2-(2-(2-(4-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)-1,2,5-thiadiazol-3-yloxy)ethoxy)ethoxy)ethoxy)ethanol 364973 tetra(ethylene glycol)(3-methoxy-1,2,4-thiadiazol-5-yl) [3-(1-methyl-1,2,5,6-tetrahydropyrid-3-yl)-1,2,5-thiadiazol-4-yl] ether 364975 N-[(1S,2S)-3-(4-chlorophenyl)-1-methyl-2-phenylpropyl]-2-[(5-chloro-2-pyridin-2-yl)oxy]-2-methylpropanamide 364976 N-((2S,3S)-4-(4-chlorophenyl)-3-phenylbutan-2-yl)-2-methyl-2-(5-(trifluoromethyl)pyridin-2-yloxy)propanamide 364983 N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)-2-methyl-2-(5-(trifluoromethyl)pyridin-2-yloxy)propanamide 364984 (S)-2-amino-N-hydroxy-3-(4-hydroxyphenyl)propanamide 365291 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-{5-[(4-phenylpiperazin-1-yl)methyl]-3-furyl}-3-quinolinecarbonitrile 365294 3-(3-amino-phenylamino)-6,11-dihydro-dibenzo[b,e]oxepin-11-one 365295 3-(4-amino-2-fluoro-phenylamino)-6,11-dihydro-dibenzo[b,e]oxepin-11-one 365302 3-(2-Amino-4-fluoro-phenylamino)-6H-dibenzo[b,e]oxepin-11-one 365309 8-(2-aminophenylamino)-6,11-dihydrodibenzo[b,e]oxepin-11-one 365310 2-(2-Amino-phenylamino)-10,11-dihydro-dibenzo[a,d]cyclohepten-5-one 365311 4-(2,4-dichloro-5-methoxyphenylamino)-7-(5-((4-methylpiperazin-1-yl)methyl)thiophen-2-yl)quinoline-3-carbonitrile 365317 2-(4-amino-phenylamino)-10,11-dihydro-dibenzo[a,d]cyclohepten-5-one 365318 2-(2-Amino-phenylamino)-dibenzo[a,d]cyclohepten-5-one 365319 4-[(2,4-dichloro-5-methoxyphenyl)amino]-7-{5-[(4-methylpiperazin-1-yl)methyl]-3-furyl}-3-quinolinecarbonitrile 365320 4-[(2,4-dichloro-5-methoxyphenyl)amino]-7-{5-[(4-methyl-1-piperazinyl)methyl]-2-furyl}-3-quinolinecarbonitrile 365326 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-{5-[(4-methylpiperazin-1-yl)methyl]-3-furyl}-3-quinolinecarbonitrile 365331 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-{5-[(4-methyl-1-piperazinyl)methyl]-2-furyl}-3-quinolinecarbonitrile 365332 4-[(2,4-dichlorophenyl)amino]-7-{5-[(4-methylpiperazin-1-yl)methyl]-3-furyl}-3-quinolinecarbonitrile 365339 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-{5-[(4-methyl-1-piperazinyl)methyl]-3-furyl}-3-quinolinecarbonitrile 365340 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[5-(morpholin-4-ylmethyl)-3-furyl]-3-quinolinecarbonitrile 365343 3-(2-amino-phenylamino)-6,11-dihydro-dibenzo[b,e]thiepin-11-one 365344 3-(2,4-Difluoro-phenylamino)-6H-dibenzo[b,e]oxepin-11-one 365347 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-{5-[(dimethylamino)methyl]-3-furyl}-3-quinolinecarbonitrile 365351 3-(2,4-dichloro-phenylamino)-6,11-dihydro-dibenzo[b,e]oxepin-11-one 365361 3-(2-Amino-phenylamino)-6H-dibenzo[b,e]oxepin-11-one 365400 4-(1-ethyl-6-phenoxy-1H-imidazo[4,5-c]pyridin-2-yl)-1,2,5-oxadiazol-3-amine 365401 4-(1-ethyl-6-(3-acetylaminophenoxy)-1H-imidazo[4,5-c]pyridin-2-yl)-1,2,5-oxadiazol-3-amine 365402 4-(1-ethyl-6-(4-acetylaminophenoxy)-1H-imidazo[4,5-c]pyridin-2-yl)-1,2,5-oxadiazol-3-amine 365403 1-(3-{[2-(4-Amino-furazan-3-yl)-1-ethyl-1H-imidazo[4,5-c]pyridin-6-yl]oxy}phenyl)ethanone 365404 4-(1-ethyl-6-{[3-(methylsulfonyl)phenyl]oxy}-1H-imidazo[4,5-c]pyridin-2-yl)-1,2,5-oxadiazol-3-amine 365405 4-{6-[(3-aminophenyl)oxy]-1-ethyl-1H-imidazo[4,5-c]pyridin-2-yl}-1,2,5-oxadiazol-3-amine 365406 N-(3-{[2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-1H-imidazo[4,5-c]pyridin-6-yl]oxy}phenyl)benzamide 365407 N-(3-{[2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-1H-imidazo[4,5-c]pyridin-6-yl]oxy}phenyl)-4-(dimethylamino)benzamide 365408 N-(3-{[2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-1H-imidazo[4,5-c]pyridin-6-yl]oxy}phenyl)-4-{[2-(4-morpholinyl)ethyl]oxy}benzamide 365442 SID11113351 365445 4-(4-fluorophenyl)-N-(1H-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide 365452 4-(4-fluorophenyl)-N-1H-indazol-5-yl-2-methyl-6-oxo-1,4,5,6-tetrahydro-3-pyridinecarboxamide 365453 N-(1H-indazol-5-yl)-2-methyl-6-oxo-4-(4-(trifluoromethyl)phenyl)-1,4,5,6-tetrahydropyridine-3-carboxamide 365460 4-(3,4-dichlorophenyl)-N-1H-indazol-5-yl-2-methyl-6-oxo-1,4,5,6-tetrahydropyridine-3-carboxamide 365461 N-(1H-indazol-5-yl)-2-methyl-4-(naphthalen-2-yl)-6-oxo-1,4,5,6-tetrahydropyridine-3-carboxamide 365469 2-methyl-N-(3-methyl-1H-indazol-5-yl)-6-oxo-4-(4-(trifluoromethyl)phenyl)-1,4,5,6-tetrahydropyridine-3-carboxamide 365470 N-(4-fluoro-1H-indazol-5-yl)-2-methyl-6-oxo-4-(4-(trifluoromethyl)phenyl)-1,4,5,6-tetrahydropyridine-3-carboxamide 365478 N-(6-fluoro-1H-indazol-5-yl)-2-methyl-6-oxo-4-(4-(trifluoromethyl)phenyl)-1,4,5,6-tetrahydropyridine-3-carboxamide 365479 N-(7-chloro-1H-indazol-5-yl)-2-methyl-6-oxo-4-(4-(trifluoromethyl)phenyl)-1,4,5,6-tetrahydropyridine-3-carboxamide 365480 2-amino-4-(2-chlorophenyl)-6-(2-(diethylamino)ethylthio)pyridine-3,5-dicarbonitrile 365540 4-(1-ethyl-6-methoxy-1H-imidazo[4,5-c]pyridin-2-yl)-1,2,5-oxadiazol-3-amine 365548 (-)-(3R,3aS,4S,4aR,6R,8aS,9aR)-decahydro-6-hydroxy-3-methyl-4-[(E)-2-[5-[3-(trifluoromethyl)phenyl]-2-pyridinyl]ethenyl]-naphtho[2,3-c]f uran-1(3H)-one 365549 (3R,3aS,4S,4aR,8aR,9aR)-7,7-difluoro-decahydro-3-methyl-4-[(E)-2-[5-(3-methylphenyl)-2-pyridinyl] ethenyl]naphtho[2,3-c]furan-1(3H)-one 365555 (+)-(3R,3aS,4S,4aR,6S,8aS,9aR)-decahydro-6-hydroxy-3-methyl-4-[(E)-2-[5-[3-(trifluoromethyl)phenyl]-2-pyridinyl]ethenyl]-naphtho[2,3-c]furan-1(3H)-one 365565 (3R,3aS,4S,4aR,8aR,9aR)-7,7-difluoro-decahydro-3-methyl-4-[(E)-2-[5-[3-(trifluoromethyl)phenyl]-2-pyridinyl]ethenyl]naphtho[2,3-c]furan-1(3H)-one 365572 (3R,3aS,4S,4aS,8aS,9aR)-8,8-difluoro-decahydro-3-methyl-4-[(E)-2-[5-[3-(trifluoromethyl)phenyl]-2-pyridinyl]ethenyl]naphtho[2,3-c]furan-1(3H)-one 365580 (3R,3aS,4S,4aR,7R,8aR,9aR)-decahydro-7-hydroxy-3-methyl-4-[(E)-2-[5-(3-fluorophenyl)-2-pyridinyl]ethenyl]naphtho[2,3-c]-furan-1(3H)-one 365589 (3R,3aS,4S,4aR,7R,8aR,9aR)-decahydro-7-hydroxy-3-methyl-4-[(E)-2-[5-(2-fluorophenyl)-2-pyridinyl]ethenyl]naphtho[2,3-c]-furan-1(3H)-one 365590 (3R,3aS,4S,4aR,7R,8aR,9aR)-decahydro-7-hydroxy-3-methyl-4-[(E)-2-[5-(4-fluorophenyl)-2-pyridinyl]ethenyl]naphtho[2,3-c]-furan-1(3H)-one 365598 (3R,3aS,4S,4aR,7R,8aR,9aR)-decahydro-7-hydroxy-3-methyl-4-[(E)-2-[5-(3-chlorophenyl)-2-pyridinyl]ethenyl]naphtho[2,3-c]-furan-1(3H)-one 365605 (3R,3aS,4S,4aR,7R,8aR,9aR)-decahydro-7-hydroxy-3-methyl-4-[(E)-2-[5-(3-methylphenyl)-2-pyridinyl]ethenyl]naphtho[2,3-c]furan-1(3H)-one 365615 (3R,3aS,4S,4aR,7R,8aR,9aR)-decahydro-7-hydroxy-3-methyl-4-[(E)-2-[5-(2-methylphenyl)-2-pyridinyl]ethenyl]naphtho[2,3-c]furan-1(3H)-one 365616 (3R,3aS,4S,4aR,7R,8aR,9aR)-decahydro-7-hydroxy-3-methyl-4-[(E)-2-[5-(4-methylphenyl)-2-pyridinyl]ethenyl]naphtho[2,3-c]furan-1(3H)-one 365626 (3R,3aS,4S,4aR,7R,8aR,9aR)-decahydro-7-hydroxy-3-methyl-4-[(E)-2-[5-(2,5-dichlorophenyl)-2-pyridinyl]ethenyl]naphtho-[2,3-c]furan-1(3H)-one 365633 (3R,3aS,4S,4aR,7R,8aR,9aR)-decahydro-7-hydroxy-3-methyl-4-[(E)-2-[5-(2,3-dichlorophenyl)-2-pyridinyl]ethenyl]naphtho-[2,3-c]furan-1(3H)-one 365642 (3R,3aS,4S,4aR,8aR,9aR)-7,7-difluoro-decahydro-3-methyl-4-[(E)-2-[5-(3-fluorophenyl)-2-pyridinyl]ethenyl]naphtho[2,3-c]furan-1(3H)-one 365649 (3R,3aS,4S,4aS,8S,8aS,9aR)-decahydro-8-hydroxy-3-methyl-4-[(E)-2-[5-[3-(trifluoromethyl)phenyl]-2-pyridinyl]ethenyl]-naphtho[2,3-c]furan-1(3H)-one 365659 (3R,3aS,4S,4aR,7R,8aR,9aR)-decahydro-7-hydroxy-3-methyl-4-[(E)-2-[5-[3-(trifluoromethyl)phenyl]-2-pyridinyl]ethenyl]naphtho[2,3-c]furan-1(3H)-one 365661 (3R,3aS,4S,4aR,8aR,9aR)-7,7-difluoro-decahydro-3-methyl-4-[(E)-2-[5-(2-fluorophenyl)-2-pyridinyl] ethenyl]naphtho[2,3-c]furan-1(3H)-one 365662 (3R,3aS,4S,4aR,8aR,9aR)-7,7-difluoro-decahydro-3-methyl-4-[(E)-2-[5-(3-chlorophenyl)-2-pyridinyl] ethenyl]naphtho[2,3-c]furan-1(3H)-one 365668 (3R,3aS,4S,4aR,7S,8aR,9aR)-decahydro-7-hydroxy-3-methyl-4-[(E)-2-[5-[3-(trifluoromethyl)phenyl]-2-pyridinyl]ethenyl]naphtho[2,3-c]furan-1(3H)-one 365671 (3R,3aS,4S,4aR,8aR,9aR)-7,7-difluoro-decahydro-3-methyl-4-[(E)-2-[5-(2-chlorophenyl)-2-pyridinyl] ethenyl]naphtho[2,3-c]furan-1(3H)-one 365676 (3R,3aS,4S,4aS,8R,8aS,9aR)-decahydro-8-hydroxy-3-methyl-4-[(E)-2-[5-[3-(trifluoromethyl)phenyl]-2-pyridinyl]ethenyl]naphtho[2,3-c]furan-1(3H)-one 365814 cyclo(-D-Tyr-L-Arg-L-Arg-L-Nal-Gly-) 365816 cyclo(-D-Tyr-L-Ala-L-Arg-L-Nal-Gly-) 365819 cyclo(-D-Tyr-D-Arg-L-Arg-L-Nal-Gly-) 365820 cyclo(-D-Ala-D-Arg-L-Arg-L-Nal-Gly-) 365821 cyclo(-D-Tyr-D-Ala-L-Arg-L-Nal-Gly-) 365824 cyclo(-D-Tyr-L-Arg-L-Arg-L-Nal-L-Ala-) 365825 cyclo(-D-Tyr-L-Arg-L-Arg-L-Nal-D-Ala-) 365830 cyclo(-D-Tyr-L-Arg-L-Arg-L-Nal-beta-Ala-) 365831 cyclo(-D-Tyr-D-Arg-L-Arg-L-Nal-L-Ala-) 365832 cyclo(-D-Tyr-D-Arg-L-Arg-L-Nal-D-Ala-) 365835 cyclo(-D-Tyr-D-Arg-L-Arg-L-Nal-L-Pic-) 365837 cyclo(-D-Tyr-D-Arg-L-Arg-L-Nal-beta-Ala-) 365838 cyclo(-D-MeTyr-L-Arg-L-Arg-L-Nal-Gly-) 365839 cyclo(-D-Tyr-L-MeArg-L-Arg-L-Nal-Gly-) 365840 cyclo(-D-Tyr-L-Arg-L-MeArg-L-Nal-Gly-) 365841 cyclo(-D-Tyr-L-Arg-L-Arg-L-MeNal-Gly-) 365842 cyclo(-D-Tyr-L-Arg-L-Arg-L-Ala-Sar-) 365843 cyclo(-D-MeTyr-D-Arg-L-Arg-L-Nal-Gly-) 365844 cyclo(-D-Tyr-D-MeArg-L-Arg-L-Nal-Gly-) 365845 cyclo(-D-Tyr-D-Arg-L-MeArg-L-Nal-Gly-) 365846 cyclo(-D-Tyr-D-Arg-L-Arg-L-MeNal-Gly-) 365847 cyclo(-D-Tyr-D-Arg-L-Arg-L-Nal-Sar-) 365856 N'-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-6-yl)furan-2-carbohydrazide 365857 H-Tyr-D-Ala-Gly-Phe-NH-NH-Trp-D-Nle-D-Asp-D-Phe-Boc 365858 H-Tyr-D-Ala-Gly-Phe-NH-NH-Trp-D-Nle-D-Asp-D-Phe-H 365859 H-Tyr-D-Ala-Gly-Phe-NH-NH-D-Trp-Nle-Asp-Phe-Bo 365860 H-Tyr-D-Ala-Gly-Phe-NH-NH-D-Trp-Nle-Asp-Phe-H 365861 H-Tyr-D-Ala-Gly-Phe-NH-NH-D-Phe-D-Asp-D-Nle-Trp-Boc 365862 H-Tyr-D-Ala-Gly-Phe-NH-NH-D-Phe-D-Asp-D-Nle-Trp-H 365863 (3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(2S)-2-amino-3-carboxypropanamido]-3-[4-(sulfooxy)phenyl]propanamido]-4-(methylsulfanyl)butanamido]acetamido}-3-(1H-indol-3-yl)propanamido]-4-(methylsulfanyl)butanamido]-3-{[(1S)-1-carboxy-2-phenylethyl]carbamoyl}propanoic acid 365870 5-bromo-N'-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-6-yl)furan-2-carbohydrazide 365871 N'-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-6-yl)-5-methylfuran-2-carbohydrazide 365878 N'-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-6-yl)-5-methylthiophene-2-carbohydrazide 365884 N'-(2-chloro-9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-6-yl)furan-2-carbohydrazide 365892 1-deoxy-1-{2-chloro-6-[N'-(5-methyl-thiophene-2-carbonyl)-hydrazino]-9H-purin-9-yl}-N-ethyl-beta-D-ribofuranuronamide 365893 N'-(2-chloro-9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-6-yl)-2-(thiophen-2-yl)acetohydrazide 365898 N'-(2-chloro-9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-6-yl)thiophene-3-carbohydrazide 365899 N'-(2-chloro-9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-6-yl)thiophene-2-carbohydrazide 365905 N'-(2-chloro-9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-6-yl)-1H-pyrrole-2-carbohydrazide 365916 8-Cyclopentyl-6-ethyl-3-thiophen-2-yl-5,8-dihydro-4H-1,2,3a,7,8-pentaaza-as-indacene 365966 H-Dmt-Tic-(2S,3S)-beta-MeCha-Phe-OH 365967 H-Dmt-Tic-(2R,3R)-beta-MeCha-Phe-OH 365968 H-Dmt-Tic-(2S,3R)-beta-MeCha-Phe-OH 365969 H-Dmt-Tic-(2R,3S)-beta-MeCha-Phe-OH 365970 H-Dmt-Tic-(2S,3S)-beta-MeCha-Phe-NH2 365971 H-Dmt-Tic-(2R,3R)-beta-MeCha-Phe-NH2 365972 H-Dmt-Tic-(2S,3R)-beta-MeCha-Phe-NH2 365973 H-Dmt-Tic-(2R,3S)-beta-MeCha-Phe-NH2 365979 (3S)-3-{[(2S)-1-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]propanamido]acetamido}-3-phenylpropanehydrazido]-1-oxo-3-phenylpropan-2-yl]carbamoyl}-3-[(2S)-2-[(2R)-2-{[(tert-butoxy)carbonyl]amino}-3-(1H-indol-2-yl)propanamido]hexanamido]propanoic acid 365980 (3S)-3-[(2S)-2-[(2R)-2-amino-3-(1H-indol-2-yl)propanamido]hexanamido]-3-{[(2S)-1-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]propanamido]acetamido}-3-phenylpropanehydrazido]-1-oxo-3-phenylpropan-2-yl]carbamoyl}propanoic acid 366462 Tyr-Pro-Trp-D-1-Nal-NH2 366463 Tyr-Pro-Trp-D-2-Nal-NH2 366464 Dmt-Pro-Trp-D-1-Nal-NH2 366465 Dmt-Pro-Trp-D-2-Nal-NH2 366470 Dmt-Pro-Phe-D-1-Nal-NH2 366477 N-(5-cyclohexyl-2-methoxyphenyl)-4-methyl-3-(3-(2-(methylamino)pyridin-4-yl)pyridin-2-yloxy)benzamide 366482 3-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-yloxy)-N-(2-(piperidin-1-yl)-5-(trifluoromethyl)phenyl)benzamide 366488 4-fluoro-3-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-yloxy)-N-(2-(piperidin-1-yl)-5-(trifluoromethyl)phenyl)benzamide 366489 3-thia-13,23-diazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,22}]tricosa-1,4(9),5,7,10,15,17(22),18,20-nonaen-14-one 366490 3-thia-13,23-diazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,22}]tricosa-1,4(9),5,7,10,15,17(22),18,20-nonaen-12-one 366492 (2S,3S)-N-hydroxy-2-((R)-3-phenylpyrrolidine-1-carbonyl)piperidine-3-carboxamide 366497 N-(4-phenoxyphenyl)-3-(3-(4-(3,4,5-trimethoxyphenylamino)-1,3,5-triazin-2-yl)pyridin-2-ylamino)benzamide 366498 N-{2-[4-((S)-2-amino-6-guanidino-hexanoyl)-piperazin-1-yl]-1,1-dimethyl-2-oxo-ethyl}-2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonamide 366499 N-{1-[4-((S)-2-amino-6-dimethylamino-hexanoyl)-piperazine-1-carbonyl]-cyclopentyl}-2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonamide 366500 N-{1-[4-((S)-3-amino-6-dimethylamino-hexanoyl)-piperazine-1-carbonyl]-cyclopentyl}-2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonamide 366501 N-{1-[4-((S)-2-amino-6-guanidino-hexanoyl)-piperazine-1-carbonyl]-cyclopentyl}-2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonamide 366502 2,4-dichloro-N-{1-[4-((S)-2,6-diamino-hexanoyl)-piperazine-1-carbonyl]-cyclopentyl}-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonamide 366503 N-{1-[4-((S)-2,6-bis-dimethylamino-hexanoyl)-piperazine-1-carbonyl]-cyclopentyl}-2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonamide 366504 [(S)-5-amino-6-(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazin-1-yl)-6-oxo-hexyl]-trimethyl-ammonium 366506 4-chloro-3-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-yloxy)-N-(2-(piperidin-1-yl)-5-(trifluoromethyl)phenyl)benzamide 366507 3-oxa-13,23-diazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,22}]tricosa-1,4(9),5,7,10,15,17(22),18,20-nonaen-14-one 366508 3-oxa-13,23-diazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,22}]tricosa-1,4(9),5,7,10,15,17(22),18,20-nonaen-12-one 366509 (6S,7S)-N-hydroxy-6-(4-phenylpiperazine-1-carbonyl)-5-azaspiro[2.5]octane-7-carboxamide 366510 (6S,7S)-N-hydroxy-6-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-5-azaspiro[2.5]octane-7-carboxamide 366512 4-(2-(phenylamino)pyridin-3-yl)-N-(3,4,5-trimethoxyphenyl)-1,3,5-triazin-2-amine 366513 [(S)-5-(4-{1-acetyl-4-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-piperidine-4-carbonyl}-piperazin-1-yl)-4-amino-5-oxo-pentyl]-trimethyl-ammonium 366514 4-methyl-3-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-yloxy)-N-(2-(piperidin-1-yl)-5-(trifluoromethyl)phenyl)benzamide 366515 5-(2-(2-aminopyrimidin-5-yl)ethynyl)-2-fluoro-N-(3-(trifluoromethyl)phenyl)benzamide 366516 3-(2-(2-aminopyrimidin-5-yl)ethynyl)-4-methyl-N-(2-(piperidin-1-yl)-5-(trifluoromethyl)phenyl)benzamide 366517 (6S,7S)-6-(4-phenyl-piperidine-1-carbonyl)-5-aza-spiro[2.5]octane-7-carboxylic acid hydroxyamide 366518 (6S,7S)-N-hydroxy-6-[(5-methyl-4-phenyl-3,6-dihydropyridin-1(2H)-yl)carbonyl]-5-azaspiro[2.5]octane-7-carboxamide 366519 N-(4-phenoxyphenyl)-2-(pyridin-4-ylmethylamino)nicotinamide 366520 4-Methyl-3-(3-(pyrimidin-4-yl)pyridin-2-ylamino)-N-(3-(trifluoromethyl)phenyl)benzamide 366521 [(S)-5-amino-6-(4-{4-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-tetrahydro-pyran-4-carbonyl}-piperazin-1-yl)-6-oxo-pentyl]-trimethyl-ammonium 366522 4-fluoro-5-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-yloxy)-N-(2-(piperidin-1-yl)-5-(trifluoromethyl)phenyl)benzamide 366524 indenyl[2,3-c]benzothienyl[2,3-e]isoindol-1-one 366526 (6S,7S)-N-hydroxy-6-{[4-(2-methyl-4-nitrophenyl)piperazin-1-yl]carbonyl}-5-azaspiro[2.5]octane-7-carboxamide 366527 4-methyl-N-phenyl-3-(3-(pyrimidin-4-yl)pyridin-2-ylamino)-benzamide 366528 4-methyl-3-(3-(pyrimidin-4-yl)pyridin-2-ylamino)-N-(4-(trifluoromethyl)phenyl)benzamide 366529 N'-[3-(4-cyclohexyl-piperazin-1-ylmethyl)-2-phenyl-quinoline-4-carbonyl]-N-phenyl-hydrazinecarboxylic acid methyl ester 366530 N-phenyl-N'-{2-phenyl-3-[4-(tetrahydro-pyran-4-yl)-piperazin-1-ylmethyl]-quinoline-4-carbonyl}-hydrazinecarboxylic acid methyl ester 366531 N-phenyl-N'-{2-phenyl-3-[4-(tetrahydro-thiopyran-4-yl)-piperazin-1-ylmethyl]-quinoline-4-carbonyl}-hydrazinecarboxylic acid methyl ester 366532 N'-[3-(4-benzyl-piperazin-1-ylmethyl)-2-phenyl-quinoline-4-carbonyl]-N-phenyl-hydrazinecarboxylic acid methyl ester 366533 N'-[3-(4-benzenesulfonyl-piperazin-1-ylmethyl)-2-phenyl-quinoline-4-carbonyl]-N-phenyl-hydrazinecarboxylic acid methyl ester 366534 N-phenyl-N'-{2-phenyl-3-[1-(tetrahydro-pyran-4-yl)-piperidin-4-ylmethyl]-quinoline-4-carbonyl}-hydrazinecarboxylic acid methyl ester 366535 N'-[3-(4-tert-butyl-piperazin-1-ylmethyl)-8-fluoro-2-phenyl-quinoline-4-carbonyl]-N-phenyl-hydrazinecarboxylic acid methyl ester 366536 N'-{8-fluoro-3-[4-(1-methyl-cyclohexyl)-piperazin-1-ylmethyl]-2-phenyl-quinoline-4-carbonyl}-N-phenyl-hydrazinecarboxylic acid methyl ester 366537 N'-{8-fluoro-2-phenyl-3-[4-(tetrahydro-pyran-4-yl)-piperazin-1-ylmethyl]-quinoline-4-carbonyl}-N-phenyl-hydrazinecarboxylic acid methyl ester 366538 N'-{8-fluoro-3-[4-(4-methyl-tetrahydro-pyran-4-yl)-piperazin-1-ylmethyl]-2-phenyl-quinoline-4-carbonyl}-N-phenyl-hydrazinecarboxylic acid methyl ester 366540 4-methyl-3-(3-(4-(methylamino)-1,3,5-triazin-2-yl)pyridin-2-yloxy)-N-(3-(trifluoromethyl)phenyl)benzamide 366541 3-(2-(6-aminopyridin-3-yl)ethynyl)-4-methyl-N-(3-(trifluoromethyl)phenyl)benzamide 366542 3-(2-(3H-imidazo[4,5-b]pyridin-6-yl)ethynyl)-4-methyl-N-(3-(trifluoromethyl)phenyl)benzamide 366543 (6S,7S)-N-hydroxy-6-{[4-(2-methyl-4-nitrophenyl)-3,6-dihydropyridin-1(2H)-yl]carbonyl}-5-azaspiro[2.5]octane-7-carboxamide 366544 (6S,7S)-N-hydroxy-6-(3,4,10,10a-tetrahydropyrazino[1,2-a]indol-2(1H)-ylcarbonyl)-5-azaspiro[2.5]octane-7-carboxamide 366545 N-(3-(3-(dimethylamino)propyl)-5-(trifluoromethyl)phenyl)-4-methyl-3-(3-(pyrimidin-4-yl)pyridin-2-ylamino)benzamide 366546 2-fluoro-5-(3-(4-(methylamino)-1,3,5-triazin-2-yl)pyridin-2-yloxy)-N-(2-(piperidin-1-yl)-5-(trifluoromethyl)phenyl)benzamide 366549 1H-indenyl[2,3-c]-1H-indenyl[2,3-e]-3H-isoindol-1-one 366550 (6S,7S)-N-hydroxy-6-((R)-3-phenylpyrrolidine-1-carbonyl)-5-azaspiro[2.5]octane-7-carboxamide 366551 (6S,7S)-6-(3-phenyl-2,5-dihydro-pyrrole-1-carbonyl)-5-aza-spiro[2.5]octane-7-carboxylic acid hydroxyamide 366552 N-(2-methoxy-5-(trifluoromethyl)phenyl)-4-methyl-3-(3-(pyrimidin-4-yl)pyridin-2-ylamino)benzamide 366555 Indenyl[2,3-c]benzothienyl[2,3-e]isoindol-3-one 366556 4-methyl-3-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-yloxy)-N-(3-(trifluoromethyl)phenyl)benzamide 366557 (6S,7S)-N-hydroxy-5-methyl-6-(4-phenylpiperazine-1-carbonyl)-5-azaspiro[2.5]octane-7-carboxamide 366558 (6S,7S)-N-hydroxy-5-methyl-6-[(4-phenyl-3,6-dihydropyridin-1(2H)-yl)carbonyl]-5-azaspiro[2.5]octane-7-carboxamide 366559 4-methyl-N-(2-(piperidin-1-yl)-5-(trifluoromethyl)phenyl)-3-(3-(pyrimidin-4-yl)pyridin-2-ylamino)benzamide 366560 4-methyl-3-(3-(pyrimidin-4-yl)pyridin-2-yloxy)-N-(3-(trifluoromethyl)phenyl)benzamide 366563 N-methyl-5-(2-(2-methyl-5-((3-(trifluoromethyl)phenyl)carbamoyl)phenyl)ethynyl)picolinamide 366564 4-methyl-3-(2-(quinolin-3-yl)ethynyl)-N-(3-(trifluoromethyl)-phenyl)benzamide 366565 (6S,7S)-methyl 7-(hydroxycarbamoyl)-6-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-5-azaspiro[2.5]octane-5-carboxylate 366566 4-methyl-3-(3-(pyrimidin-4-yl)pyridin-2-yloxy)-N-(4-(trifluoromethyl)phenyl)benzamide 366567 N-(2-methoxy-5-(trifluoromethyl)phenyl)-4-methyl-3-(3-(pyrimidin-4-yl)pyridin-2-yloxy)benzamide 366574 2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-N-{1-[4-(6-guanidino-hexanoyl)-piperazine-1-carbonyl]-cyclopentyl}-benzenesulfonamide 366575 [6-(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazin-1-yl)-6-oxo-hexyl]-trimethyl-ammonium 366576 [(S)-1-(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazine-1-carbonyl)-5-guanidino-pentyl]-trimethyl-ammonium 366577 N-[1-[4-(2-(S)-trimethylammonium-6-trimethylammoniumhexanoyl)-piperazin-1-yl]-cyclopentyl]-2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonamide 366578 [(S)-5-amino-1-(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazine-1-carbonyl)-pentyl]-trimethyl-ammonium 366579 2,4-dichloro-N-{1-[4-((S)-3,6-diamino-hexanoyl)-piperazine-1-carbonyl]-cyclopentyl}-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonamide 366580 [(S)-4-amino-6-(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazin-1-yl)-6-oxo-hexyl]-trimethyl-ammonium 366581 {(S)-4-amino-1-[2-(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazin-1-yl)-2-oxo-ethyl]-butyl}-trimethyl-ammonium 366582 N-{1-[4-((S)-3-amino-6-guanidino-hexanoyl)-piperazine-1-carbonyl]-cyclopentyl}-2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonamide 366584 [2-(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazin-1-yl)-2-oxo-ethyl]-trimethyl-ammonium 366586 [4-(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazin-1-yl)-4-oxo-butyl]-trimethyl-ammonium 366587 4-methyl-N-(2-(piperidin-1-yl)-5-(trifluoromethyl)phenyl)-3-(3-(pyrimidin-4-yl)pyridin-2-yloxy)benzamide 366590 3-(2-(2-aminopyrimidin-5-yl)ethynyl)-4-methyl-N-(3-(trifluoromethyl)phenyl)benzamide 366594 4-methyl-3-(2-(quinoxalin-2-yl)ethynyl)-N-(3-(trifluoromethyl)phenyl)benzamide 366595 3-(2-(2-aminopyrimidin-5-yl)ethynyl)-N-(3-(trifluoromethyl)-phenyl)benzamide 366598 4-methyl-N-(2-morpholino-5-(trifluoromethyl)phenyl)-3-(3-(pyrimidin-4-yl)pyridin-2-yloxy)benzamide 366603 [(S)-3-amino-4-(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazin-1-yl)-4-oxo-butyl]-trimethyl-ammonium 366604 2-methyl-3-(5-methyl-3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-yloxy)-N-(2-(piperidin-1-yl)-5-(trifluoromethyl)phenyl)benzamide 366605 4-methyl-3-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-yloxy)-N-(2-morpholino-5-(trifluoromethyl)phenyl)benzamide 366607 12,13-dihydro-6H,14H-naphthyl[3,4-a]pyrrolo[3,4-c]carbazole-5,7(5H,7H)dione 366613 [5-(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazin-1-yl)-5-oxo-pentyl]-trimethyl-ammonium 366614 [(S)-4-amino-5-(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazin-1-yl)-5-oxo-pentyl]-trimethyl-ammonium 366615 N-(2-((3-(dimethylamino)propyl)(methyl)amino)-5-(trifluoromethyl)phenyl)-2-fluoro-5-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-yloxy)benzamide 366616 [5-(4-(1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl]-piperazin-1-yl)-4(S)-trimethylammonio-5-oxo-pentyl]trimethyl-ammonium 366617 [(S)-4-amino-1-(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazine-1-carbonyl)-butyl]-trimethyl-ammonium 366618 4-methyl-3-(3-(4-(methylamino)-1,3,5-triazin-2-yl)pyridin-2-yloxy)-N-(2-(piperidin-1-yl)-5-(trifluoromethyl)phenyl)benzamide 366619 4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-N-(3-dimethylamino-propyl)-piperazine-1-carboxamidine 366620 N-(2-((3-(dimethylamino)propyl)(methyl)amino)-5-(trifluoromethyl)phenyl)-4-methyl-3-(3-(4-(methylamino)-1,3,5-triazin-2-yl)pyridin-2-yloxy)benzamide 366621 {3-[(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazine-1-carboximidoyl)-amino]-propyl}-trimethyl-ammonium 366622 N-(2-((3-(dimethylamino)propyl)(methyl)amino)-5-(trifluoromethyl)phenyl)-2-fluoro-5-(3-(4-(methylamino)-1,3,5-triazin-2-yl)pyridin-2-yloxy)benzamide 366623 N-(5-cyclohexyl-2-methoxyphenyl)-4-methyl-3-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-yloxy)benzamide 366624 12,13-dihydro-5H,6H,14H-naphthy[3,4-a]pyrrolo[3,4-c]carbazole-7(7H)one 366625 12,13-dihydro-6H,7H,14H-naphthyl-[3,4-a]pyrrolo[3,4-c]carbazole-5(5H)one 366632 N-(2-((3-(dimethylamino)propyl)(methyl)amino)-5-isopropylphenyl)-2-fluoro-5-(3-(4-(methylamino)-1,3,5-triazin-2-yl)pyridin-2-yloxy)benzamide 366633 [(S)-4-amino-5-(4-{4-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-tetrahydro-thiopyran-4-carbonyl}-piperazin-1-yl)-5-oxo-pentyl]-trimethyl-ammonium 366634 N-(5-cyclopropyl-2-((3-(dimethylamino)propyl)(methyl)amino)phenyl)-2-fluoro-5-(3-(4-(methylamino)-1,3,5-triazin-2-yl)pyridin-2-yloxy)benzamide 366635 [(S)-4-amino-5-(4-{4-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-piperidine-4-carbonyl}-piperazin-1-yl)-5-oxo-pentyl]-trimethyl-ammonium 366636 [(S)-4-amino-5-(4-{4-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-1-methyl-piperidine-4-carbonyl}-piperazin-1-yl)-5-oxo-pentyl]-trimethyl-ammonium 366637 N-(5-cyclohexyl-2-methoxyphenyl)-4-methyl-3-(3-(4-(methylamino)-1,3,5-triazin-2-yl)pyridin-2-yloxy)benzamide 366640 2,6-diphenyl-8-isobutyl-1-deazapurine 366641 2,6-diphenyl-8-(1-ethylpropyl)-1-deazapurine 366642 5-(2-(2-aminopyrimidin-5-yl)ethynyl)-N-(2-(4-(dimethylamino)piperidin-1-yl)-5-(trifluoromethyl)phenyl)-2-fluorobenzamide 366651 2,6-diphenyl-8-tButyl-1-deazapurine 366652 8-cyclopentyl-2,6-diphenyl-1-deazapurin 366653 (R)-5-(2-(2-aminopyrimidin-5-yl)ethynyl)-N-(2-(3-(dimethylamino)piperidin-1-yl)-5-(trifluoromethyl)phenyl)-2-fluorobenzamide 366662 2,6-diphenyl-8-cyclohexyl-1-deazapurine 366663 (S)-5-(2-(2-aminopyrimidin-5-yl)ethynyl)-N-(2-(3-(dimethylamino)piperidin-1-yl)-5-(trifluoromethyl)phenyl)-2-fluorobenzamide 366668 N'-[3-(1-tert-butyl-piperidin-4-yloxy)-2-phenyl-quinoline-4-carbonyl]-N-phenyl-hydrazinecarboxylic acid methyl ester 366669 (S)-5-(2-(2-aminopyrimidin-5-yl)ethynyl)-2-fluoro-N-(2-(3-(methylamino)piperidin-1-yl)-5-(trifluoromethyl)phenyl)benzamide 366670 (S)-N-(2-(3-aminopiperidin-1-yl)-5-(trifluoromethyl)phenyl)-5-(2-(2-aminopyrimidin-5-yl)ethynyl)-2-fluorobenzamide 366678 (R)-5-(2-(2-aminopyrimidin-5-yl)ethynyl)-N-(2-(3-(dimethylamino)pyrrolidin-1-yl)-5-(trifluoromethyl)phenyl)-2-fluorobenzamide 366683 (S)-5-(2-(2-aminopyrimidin-5-yl)ethynyl)-N-(2-(3-(dimethylamino)pyrrolidin-1-yl)-5-(trifluoromethyl)phenyl)-2-fluorobenzamide 366802 N'-[3-(2-dimethylamino-ethoxy)-2-phenyl-quinoline-4-carbonyl]-N-phenyl-hydrazinecarboxylic acid methyl ester 366803 N-phenyl-N'-{2-phenyl-3-[1-(tetrahydro-pyran-4-yl)-piperidin-4-yloxy]-quinoline-4-carbonyl}-hydrazinecarboxylic acid methyl ester 366808 2,6-dimethyl-8-ethyl-1-deazapurine 366809 5,7-diphenyl-3H-imidazo[4,5-b]pyridin-2-ol 366810 3-(2-(2-aminopyrimidin-5-yl)ethynyl)-N-(2-(piperidin-1-yl)-5-(trifluoromethyl)phenyl)benzamide 366811 5-(2-(2-aminopyrimidin-5-yl)ethynyl)-2-fluoro-N-(2-(piperidin-1-yl)-5-(trifluoromethyl)phenyl)benzamide 366822 2,6-diphenyl-1-deazapurine 366824 2,6-diphenyl-8-methyl-1-deazapurine 366825 5-(2-(2-aminopyrimidin-5-yl)ethynyl)-2-methoxy-N-(2-(piperidin-1-yl)-5-(trifluoromethyl)phenyl)benzamide 366826 5-(2-(2-aminopyrimidin-5-yl)ethynyl)-N-(2-((3-(dimethylamino)propyl)(methyl)amino)-5-(trifluoromethyl)phenyl)-2-fluorobenzamide 366832 2,6-diphenyl-8-ethyl-1-deazapurine 366833 2,6-dphenyl-8-propyl-1-deazapurine 366834 2,6-diphenyl-8-isopropyl-1-deazapurine 366835 3-(2-(2-aminopyrimidin-5-yl)ethynyl)-N-(2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl)benzamide 366836 N-[4-(piperidin-4-ylsulfamoyl)-naphthalen-1-yl]-benzamide 366837 4-(4-benzoylamino-naphthalene-1-sulfonylamino)-piperidine-1-carboxylic acid tert-butyl ester 366838 5-bromo-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-1H-indole-2-carboxamide 366839 6-cyano-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-1H-indole-2-carboxamide 366840 N'-[3-(4-isopropyl-piperazin-1-ylmethyl)-2-phenyl-quinoline-4-carbonyl]-N-phenyl-hydrazinecarboxylic acid methyl ester 366844 4-(4-benzoylamino-naphthalene-1-sulfonylamino)-piperidine-1-carboxylic acid ethyl ester 366845 4-[4-(2-methyl-benzoylamino)-naphthalene-1-sulfonylamino]-piperidine-1-carboxylic acid ethyl ester 366846 5-bromo-N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-1H-indole-2-carboxamide 366847 6-cyano-N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-1H-indole-2-carboxamide 366848 N'-[3-(4-acetyl-piperazin-1-ylmethyl)-2-phenyl-quinoline-4-carbonyl]-N-phenyl-hydrazinecarboxylic acid methyl ester 366852 4-(4-cyclohexylcarbamoyl-naphthalene-1-sulfonylamino)-piperidine-1-carboxylic acid ethyl ester 366853 4-(4-o-tolylcarbamoyl-naphthalene-1-sulfonylamino)-piperidine-1-carboxylic acid ethyl ester 366854 N-phenyl-N'-(2-phenyl-3-piperidin-4-ylmethyl-quinoline-4-carbonyl)-hydrazinecarboxylic acid methyl ester 366857 ethyl 4-(1-(benzyloxy)naphthalene-4-sulfonamido)piperidine-1-carboxylate 366858 ethyl 4-({[4-(benzoyloxy)-1-naphthyl]sulfonyl}amino)-piperidine-1-carboxylate 366859 N'-(8-fluoro-2-phenyl-3-piperazin-1-ylmethyl-quinoline-4-carbonyl)-N-phenyl-hydrazinecarboxylic acid methyl ester 366860 arginine vasopressin 366861 (S)-1-((4R,7S,10S,13S,16S)-7-(2-amino-2-oxoethyl)-10-(3-amino-3-oxopropyl)-13-benzyl-16-(4-hydroxybenzyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentaazacycloicosane-4-carbonyl)-N-((S)-1-(2-amino-2-oxoethylamino)-5-guanidino-1-oxopentan-2-yl)pyrrolidine-2-carboxamide 366868 (S)-1-((4R,7S,10S,13S,16S)-7-(2-amino-2-oxoethyl)-10-(3-amino-3-oxopropyl)-13-benzyl-16-(4-hydroxybenzyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentaazacycloicosane-4-carbonyl)-N-((R)-1-(2-amino-2-oxoethylamino)-5-guanidino-1-oxopentan-2-yl)pyrrolidine-2-carboxamide 366869 d[Val4]AVP 366870 dVDAVP 366871 d[D-3-Pal2]AVP 366872 d[Cha4]AVP 366873 d[Cha4,Lys8]VP 366874 d[Cha4,Orn8]VP 366875 d[Cha4,Dab8]VP 366876 d[Cha4,Dap8]VP 366877 d[Leu4]AVP 366878 d[Leu4,Lys8]VP 366879 d[Leu4,Orn8]VP 366880 d[Leu4,Dab8]VP 366881 d[Leu4,Dap8]VP 366882 4-[4-(benzylamino-methyl)-naphthalene-1-sulfonylamino]piperidine-1-carboxylic acid ethyl ester 366883 4-[4-(phenethylamino-methyl)-naphthalene-1-sulfonylamino]-piperidine-1-carboxylic acid ethyl ester 366884 N'-[8-fluoro-3-(4-isopropyl-piperazin-1-ylmethyl)-2-phenyl-quinoline-4-carbonyl]-N-phenyl-hydrazinecarboxylic acid methyl ester 366887 4-{4-[(3-phenyl-propylamino)-methyl]-naphthalene-1-sulfonylamino}-piperidine-1-carboxylic acid ethyl ester 366888 ethyl 4-[({4-[(piperidin-1-ylcarbonyl)amino]-1-naphthyl}-sulfonyl)amino]piperidine-1-carboxylate 366894 ((+/-)-N-(4-{[(1-butyrylpyrrolidin-3-yl)amino]sulfonyl}-1-naphthyl)-2-methylbenzamide 366900 d[Orn4]AVP 366901 d[Orn4,Lys8]VP 366902 d[Orn4,Orn8]VP 366903 d[Arg4]AVP 366904 d[Arg4,Lys8]VP 366905 d[Arg4,Orn8]VP 366906 d[Arg4,Dab8]VP 366907 N-(4-(4-(2-chlorophenyl)piperazin-1-yl)butyl)-2-naphthamide 366908 4-chloro-N-(4-(4-(2-chlorophenyl)piperazin-1-yl)butyl)benzamide 366909 N-(4-{[(1-butyrylazetidin-3-yl)amino]sulfonyl}-1-naphthyl)-2-methylbenzamide 366910 N-(4-{[(1-butyrylpiperidin-4-yl)amino]-sulfonyl}-1-naphthyl)benzamide 366928 N-(4-(4-(2-chlorophenyl)piperazin-1-yl)butyl)-3,4-dimethoxybenzamide 366929 biphenyl-4-carboxylic acid {4-[4-(2-chloro-phenyl)-piperazin-1-yl]-butyl}-amide 366930 N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-3-methylbenzamide 366935 N-[4-(4-methoxy-phenylsulfamoyl)-naphthalen-1-yl]-benzamide 366937 N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-4-methylbenzamide 366947 5-ethynyl-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)benzo[b]thiophene-2-carboxamide 366948 3-((4-(4-chlorophenyl)piperazin-1-yl)methyl)-7-iodoH-pyrazolo[1,5-a]pyridine 366953 5-cyano-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)benzo[b]thiophene-2-carboxamide 366954 6-ethynyl-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)benzo[b]thiophene-2-carboxamide 366955 N-[4-(1-butyryl-piperidin-4-ylsulfamoyl)-naphthalen-1-yl]-2-fluoro-benzamide 366960 N-(4-(morpholinosulfonyl)naphthalen-1-yl)benzamide 366965 N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-2-methylbenzamide 366966 5-bromo-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)benzofuran-2-carboxamide 366967 5-bromo-N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)benzofuran-2-carboxamide 366968 N-phenyl-N'-(2-phenyl-3-piperidin-1-ylmethyl-quinoline-4-carbonyl)-hydrazinecarboxylic acid methyl ester 366973 5-cyano-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)benzofuran-2-carboxamide 366974 N-phenyl-N'-(2-phenyl-3-piperazin-1-ylmethyl-quinoline-4-carbonyl)-hydrazinecarboxylic acid methyl ester 366977 N-(4-phenylsulfamoyl-naphthalen-1-yl)-benzamide 366978 N-{4-[(benzylamino)sulfonyl]-1-naphthyl}benzamide 366979 5-cyano-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-1H-indole-2-carboxamide 366980 4-[4-(2-methyl-benzoylamino)-naphthalene-1-sulfonylamino]-piperidine-1-carboxylic acid ethylamide 366981 N'-[3-(4-methyl-piperazin-1-ylmethyl)-2-phenyl-quinoline-4-carbonyl]-N-phenyl-hydrazinecarboxylic acid methyl ester 366984 N-{4-[(pyridin-4-ylmethyl)-sulfamoyl]-naphthalen-1-yl}-benzamide 366985 N-(4-cyclohexylsulfamoyl-naphthalen-1-yl)-benzamide 366986 cyclobutanecarboxylic acid [4-(1-butyryl-piperidin-4-ylsulfamoyl)-naphthalen-1-yl]-amide 366987 2-methyl-N-{4-[({1-[(2S)-pyrrolidin-2-ylcarbonyl]piperidin-4-yl}amino)sulfonyl]-1-naphthyl}benzamide 366988 N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-4-ethylbenzamide 366989 N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-5-methyl-2-(trifluoromethyl)-3-furamide 366992 N-(4-{[(1-benzoylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-2-methylbenzamide 366993 1-(2-bromobenzyl)-N-(5-(4-(2-methoxyphenyl)piperazin-1-yl)pentyl)-5-methyl-1H-1,2,3-triazole-4-carboxamide 366994 1-(2-bromobenzyl)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-5-propyl-1H-1,2,3-triazole-4-carboxamide 366995 cyclopentanecarboxylic acid [4-(1-butyryl-piperidin-4-ylsulfamoyl)-naphthalen-1-yl]-amide 366997 N-{4-[({1-[4-(dimethylamino)benzoyl]piperidin-4-yl}amino)-sulfonyl]-1-naphthyl}-2-methylbenzamide 366998 4-butyl-N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)benzamide 366999 4-phenyl-1-((1-phenyl-1H-pyrazol-4-yl)methyl)piperidine 367000 N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-1-methyl-1H-imidazole-2-carboxamide 367001 N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-2-chloro-6-methylisonicotinamide 367002 N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-2-cyclopentylacetamide 367003 2-methyl-N-{4-[1-(piperidine-1-carbonyl)-piperidin-4-ylsulfamoyl]-naphthalen-1-yl}-benzamide 367004 4-phenyl-1-((1-phenyl-1H-1,2,3-triazol-4-yl)methyl)piperidine 367005 N-[4-(1-butyryl-piperidin-4-ylsulfamoyl)-naphthalen-1-yl]-2-methyl-nicotinamide 367006 N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-pyrazine-2-carboxamide 367007 cyclohexanecarboxylic acid [4-(1-butyryl-piperidin-4-ylsulfamoyl)-naphthalen-1-yl]-amide 367010 4-tert-butyl-N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)benzamide 367011 N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-pyridine-2-carboxamide 367012 N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-nicotinamide 367014 3-(dimethylamino)propyl 4-[({4-[(2-methylbenzoyl)amino]-1-naphthyl}sulfonyl)amino]piperidine-1-carboxylate 367015 N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-4-pentylbenzamide 367016 N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-3-furamide 367017 ethyl 4-({[4-(Isonicotinoylamino)-1-naphthyl]sulfonyl}amino)-piperidine-1-carboxylate 367019 tetrahydro-pyran-4-carboxylic acid [4-(1-butyryl-piperidin-4-ylsulfamoyl)-naphthalen-1-yl]-amide 367020 N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-2-ethylbutanamide 367021 (R)-3-(naphthalene-7-sulfonamido)-3-phenyl-N-((R)-5-(piperidin-1-ylmethyl)-2,3-dihydro-1H-inden-1-yl)propanamide 367022 (R)-3-(naphthalene-7-sulfonamido)-3-phenyl-N-((S)-5-(piperidin-1-ylmethyl)-2,3-dihydro-1H-inden-1-yl)propanamide 367023 (R)-3-(naphthalene-3-sulfonamido)-3-phenyl-N-((R)-6-(piperidin-1-ylmethyl)-1,2,3,4-tetrahydronaphthalen-1-yl)propanamide 367024 (R)-3-(naphthalene-7-sulfonamido)-3-phenyl-N-((S)-6-(piperidin-1-ylmethyl)-1,2,3,4-tetrahydronaphthalen-1-yl)propanamide 367029 (R)-3-(naphthalene-7-sulfonamido)-3-phenyl-N-((S)-7-(piperidin-1-ylmethyl)-2,2-dioxo-1,2,3,4-tetrahydro-1-methyl-2,1-benzothiazine-4-yl)propanamide 367030 3-(diethylamino)propyl 4-[({4-[(2-methylbenzoyl)amino]-1-naphthyl}sulfonyl)amino]piperidine-1-carboxylate 367031 1-benzyl-N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-5-methyl-1H-1,2,3-triazole-4-carboxamide 367033 1-(2-bromobenzyl)-N-(5-(4-(2-methoxyphenyl)piperazin-1-yl)pentyl)-5-propyl-1H-1,2,3-triazole-4-carboxamide 367035 3-pyrrolidin-1-ylpropyl 4-[({4-[(2-methylbenzoyl)amino]-1-naphthyl}sulfonyl)amino]piperidine-1-carboxylate 367036 3-(2,6-dimethylmorpholin-4-yl)propyl-4-[({4-[(2-methylbenzoyl)amino]-1-naphthyl}sulfonyl)amino]piperidine-1-carboxylate 367037 3-(3,4-dihydroisoquinolin-2(1H)-yl)propyl 4-[({4-[(2-methylbenzoyl)amino]-1-naphthyl}sulfonyl)amino]piperidine-1-carboxylate 367038 1-benzyl-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-5-methyl-1H-1,2,3-triazole-4-carboxamide 367039 1-benzyl-N-(5-(4-(2,3-dichlorophenyl)piperazin-1-yl)pentyl)-5-methyl-1H-1,2,3-triazole-4-carboxamide 367040 N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-3,3-dimethylbutanamide 367041 N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-2-phenylbutanamide 367042 (R)-3-(naphthalene-7-sulfonamido)-3-phenyl-N-((R)-7-(piperidin-1-ylmethyl)-2,2-dioxo-1,2,3,4-tetrahydro-1-methyl-2,1-benzothiazine-4-yl)propanamide 367048 4-(1-(2-methylbenzamido)naphthalene-4-sulfonamido)piperidine-1-carboxamide 367049 4-[4-(2-methyl-benzoylamino)-naphthalene-1-sulfonylamino]-piperidine-1-carboxylic acid methylamide 367050 1-benzyl-N-(5-(4-(2-methoxyphenyl)piperazin-1-yl)pentyl)-5-methyl-1H-1,2,3-triazole-4-carboxamide 367051 N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-1-benzothiophene-2-carboxamide 367053 2-methyl-N-[4-(1-propionyl-piperidin-4-ylsulfamoyl)-naphthalen-1-yl]-benzamide 367054 N-(4-{[(1-acetylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-2-methylbenzamide 367062 4-[({4-[(2-methylbenzoyl)amino]-1-naphthyl}sulfonyl)amino]-N-propylpiperidine-1-carboxamide 367063 N-isopropyl-4-[({4-[(2-methylbenzoyl)amino]-1-naphthyl}-sulfonyl)amino]piperidine-1-carboxamide 367064 1-benzyl-N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-5-propyl-1H-1,2,3-triazole-4-carboxamide 367065 1-benzyl-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-5-propyl-1H-1,2,3-triazole-4-carboxamide 367068 N-[4-(1-cyclopropanecarbonyl-piperidin-4-ylsulfamoyl)-naphthalen-1-yl]-2-methyl-benzamide 367069 N-[4-(1-cyclopentanecarbonyl-piperidin-4-ylsulfamoyl)-naphthalen-1-yl]-2-methyl-benzamide 367070 4-[4-(2-methyl-benzoylamino)-naphthalene-1-sulfonylamino]-piperidine-1-carboxylic acid phenylamide 367071 1-(4-methoxybenzyl)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-5-methyl-1H-1,2,3-triazole-4-carboxamide 367074 N-{4-[1-(2-hydroxy-acetyl)-piperidin-4-ylsulfamoyl]-naphthalen-1-yl}-2-methyl-benzamide 367075 N-{4-[1-(2-methoxy-acetyl)-piperidin-4-ylsulfamoyl]-naphthalen-1-yl}-2-methyl-benzamide 367076 4-({[4-(benzoylamino)-1-naphthyl]sulfonyl}amino)-N,N-dimethylpiperidine-1-carboxamide 367077 N-{4-[1-(azetidine-1-carbonyl)-piperidin-4-ylsulfamoyl]-naphthalen-1-yl}-2-methyl-benzamide 367078 3-tert-butyl-N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-1-methyl-1H-pyrazole-5-carboxamide 367081 N-{4-[1-(2-amino-acetyl)-piperidin-4-ylsulfamoyl]-naphthalen-1-yl}-2-methyl-benzamide 367082 N-{4-[1-(3-amino-propionyl)-piperidin-4-ylsulfamoyl]-naphthalen-1-yl}-2-methyl-benzamide 367083 2-methyl-N-[4-({[1-(pyrrolidin-1-ylcarbonyl)piperidin-4-yl]-amino}sulfonyl)-1-naphthyl]benzamide 367084 1-(4-methoxybenzyl)-N-(5-(4-(2,3-dichlorophenyl)piperazin-1-yl)pentyl)-5-methyl-1H-1,2,3-triazole-4-carboxamide 367085 N-{4-[1-(4-amino-butyryl)-piperidin-4-ylsulfamoyl]-naphthalen-1-yl}-2-methyl-benzamide 367086 N-[4-({[1-(5-aminopentanoyl)piperidin-4-yl]amino}sulfonyl)-1-naphthyl]-2-methyl-benzamide 367087 N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-3-fluorobenzamide 367088 4-(benzyloxy)-N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)benzamide 367089 1-(4-methoxybenzyl)-N-(5-(4-(2-methoxyphenyl)piperazin-1-yl)pentyl)-5-methyl-1H-1,2,3-triazole-4-carboxamide 367090 cyclopropanecarboxylic acid [4-(1-butyryl-piperidin-4-ylsulfamoyl)-naphthalen-1-yl]-amide 367091 N-[4-({[1-(azetidin-3-ylcarbonyl)piperidin-4-yl]amino}sulfonyl)-1-naphthyl]-2-methyl-benzamide 367092 N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-naphthyl)-4-fluorobenzamide 367093 1-(4-methoxybenzyl)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-5-propyl-1H-1,2,3-triazole-4-carboxamide 367094 1-(2-bromobenzyl)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-5-methyl-1H-1,2,3-triazole-4-carboxamide 367098 [2-(benzo[1,3]dioxol-4-yloxy)-ethyl]-(3-cyclopent-1-enyl-benzyl)-amine 367099 (3-cyclopent-1-enyl-benzyl)-[2-(2,2-dimethyl-benzo[1,3]dioxol-4-yloxy)-ethyl]-amine 367100 4-[4-(2-methyl-benzoylamino)-naphthalene-1-sulfonylamino]-piperidine-1-carboxylic acid (3-diethylamino-propyl)-amide 367103 (3-cyclopent-1-enyl-benzyl)-[2-(2,2-dimethyl-2,3-dihydrobenzofuran-7-yloxy)-ethyl]-amine 367104 (3-cyclopenten-1-yl-benzyl)-[2-(2-spiro-cyclopropyl-2,3-dihydro-benzofuran-7-yloxy)-ethyl]-amine 367105 ethyl 4-({[5-(benzoylamino)-1-naphthyl]sulfonyl}amino)-piperidine-1-carboxylate 367106 4-(8-benzoylamino-naphthalene-2-sulfonylamino)-piperidine-1-carboxylic acid ethyl ester 367109 (3-cyclopent-1-enyl-benzyl)-[2-(2-ethyl-2-methyl-2,3-dihydrobenzofuran-7-yloxy)-ethyl]-amine 367110 (3-cyclopent-1-enyl-benzyl)-[2-(3,3-dimethyl-2,3-dihydrobenzofuran-7-yloxy)-ethyl]-amine 367112 4-(6-fluoropyridin-2-yl)-N-{4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl}benzamide 367117 (5-cyclopent-1-enyl-pyridin-3-yl-methyl)-[2-(2,2-dimethyl-2,3-dihydro-benzofuran-7-yloxy)-ethyl]-amine 367118 (5-cyclopent-1-enyl-pyridin-3-ylmethyl)-[2-(2-spiro-cyclopropyl-2,3-dihydro-benzofuran-7-yloxy)]-ethylamine 367119 4-(6-fluoropyridin-3-yl)-N-{4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl}benzamide 367120 3-(RS)-N-(4-(piperidin-1-ylmethyl)benzyl)-3-(naphthalene-7-sulfonamido)-3-phenylpropanamide 367124 (4R)-2-undecylthiazolidine-4-carboxylic acid 367125 (4R)-2-decylthiazolidine-4-carboxylic acid 367129 5-(4-carboxy-2-(4-(4-(heptadecylamino)phenyl)-2,4-dioxobutyl)phenoxy)isophthalic acid 367130 5-(4-carboxy-2-(2,4-dioxo-4-(4-stearamidophenyl)butyl)phenoxy)isophthalic acid 367131 (E)-5-[1-(4-cetyloxy-3-methoxyphenyl)-1-phenylmethylene]-sulfohydrazono isophthalic acid 367132 (Z)-5-[1-(4-cetyloxy-3-methoxyphenyl)-1-phenylmethylene]-sulfohydrazono isophthalic acid 367133 (E)-5-[1-(4-cetyloxyphenyl)-1-phenylmethylene]sulfohydrazonoisophthalic acid 367142 2-(hexadecyloxy)-5-sulfobenzoic acid 367147 (E)-5-[1-(4-octyloxy-3-methoxyphenyl)-1-phenylmethylene]-sulfohydrazono isophthalic acid 367150 (Z)-5-[1-(4-octyloxy-3-methoxyphenyl)-1-phenylmethylene]-sulfohydrazono isophthalic acid 367153 1-(2,3-dihydrobenzo[b][1,4]dioxin-5-yl)-4-((5-(4-fluorophenyl)pyridin-3-yl)methyl)piperazine 367154 (R)-N-((3,4-dihydro-2H-chromen-2-yl)methyl)(5-(4-fluorophenyl)pyridin-3-yl)methanamine 367160 Bifeprunox 367161 [2-(2-isopropoxy-phenoxy)-ethyl]-(3-phenyl-benzyl)-amine 367162 N-(4-(methylsulfonyl)benzyl)-4-amino-6-ethoxy-5-ethynylpicolinamide 367167 2-(2-isopropoxy-phenoxy)-ethyl]-(3-thien-2-yl-benzyl)-amine 367168 2-(2-isopropoxy-phenoxy)-ethyl]-(3-thien-3-yl-benzyl)-amine 367169 N-(4-(methylsulfonyl)benzyl)-4-amino-6-ethoxy-5-(2-(thiophen-3-yl)ethynyl)picolinamide 367170 N-(4-(methylsulfonyl)benzyl)-4-amino-6-ethoxy-5-(3-hydroxyprop-1-ynyl)picolinamide 367174 (3-fur-2-yl-benzyl)-[2-(2-isopropoxy-phenoxy)-ethyl]-amine 367175 3-cyclohept-1-enyl-benzyl)-[2-(2-isopropoxy-phenoxy)-ethyl]-amine 367176 N-(4-(methylsulfonyl)benzyl)-4-amino-6-ethoxy-5-(4-hydroxybut-1-ynyl)picolinamide 367177 N-(4-(methylsulfonyl)benzyl)-4-amino-6-ethoxy-5-(5-hydroxypent-3-en-1-ynyl)picolinamide 367182 3-cyclohex-1-enyl-benzyl)-[2-(2-isopropoxy-phenoxy)-ethyl]-amine 367183 3-cyclopent-1-enyl-benzyl)-[2-(2-isopropoxy-phenoxy)-ethyl]-amine 367184 2-methyl-N-{4-[1-(4-methyl-piperazine-1-carbonyl)-piperidin-4-ylsulfamoyl]-aphthalen-1-yl}-benzamide 367189 3-cyclopentanyl-benzyl)-[2-(2-isopropoxy-phenoxy)-ethyl]-amine 367190 3-cyclopropyl-benzyl)-[2-(2-isopropoxy-phenoxy)-ethyl]-amine 367191 2-methyl-N-[4-({[1-(morpholin-4-ylcarbonyl)piperidin-4-yl]-amino}sulfonyl)-1-naphthyl]benzamide 367195 (3-cyclopent-1-enyl-benzyl)-[2-(2,3-dihydro-benzo[1,4]dioxin-5-yloxy)-ethyl]-amine 367196 4-[4-(2-methyl-benzoylamino)-naphthalene-1-sulfonylamino]-piperidine-1-carboxylic acid (3-morpholin-4-yl-propyl)-amide 367205 N2-(4-(methylsulfonyl)benzyl)-4-amino-6-ethoxy-N5-propylpyridine-2,5-dicarboxamide 367206 N-(4-(methylsulfonyl)benzyl)-4-amino-6-(3-chlorophenyl)-5-cyanopicolinamide 367207 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(phenethylamino)picolinamide 367208 1-(2-(6-((4-(methylsulfonyl)benzyl)carbamoyl)-4-amino-3-cyanopyridin-2-ylamino)ethyl)urea 367213 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(3-hydroxyphenyl)picolinamide 367214 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(3-methoxyphenyl)picolinamide 367215 N-(4-(methylsulfonyl)benzyl)-4-amino-6-(3-amino-3-oxopropylamino)-5-cyanopicolinamide 367216 N-(4-(methylsulfonyl)benzyl)-6-(2-acetamidoethylamino)-4-amino-5-cyanopicolinamide 367221 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(3-(methylsulfonyl)phenyl)picolinamide 367222 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(thiophen-3-yl)picolinamide 367223 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(3-hydroxypropylamino)picolinamide 367224 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(2-hydroxyethylamino)picolinamide 367229 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(furan-3-yl)picolinamide 367230 5-(6-((4-(methylsulfonyl)benzyl)carbamoyl)-4-amino-3-cyanopyridin-2-yl)thiophene-2-carboxylic acid 367231 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(2-methoxyethylamino)picolinamide 367232 N-(4-(methylsulfonyl)benzyl)-4-amino-6-(2-aminoethylamino)-5-cyanopicolinamide 367235 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(2-(hydroxymethyl)thiophen-3-yl)picolinamide 367236 N-(4-(methylsulfonyl)benzyl)-4-amino-6-(2-((benzylamino)methyl)thiophen-3-yl)-5-cyanopicolinamide 367237 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(2-(dimethylamino)ethylamino)picolinamide 367238 (S)-N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(1-hydroxypropan-2-ylamino)picolinamide 367243 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(pyridin-3-yl)picolinamide 367244 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(pyridin-4-yl)picolinamide 367245 (R)-N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(1-hydroxypropan-2-ylamino)picolinamide 367246 (S)-N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(1-hydroxy-3-methylbutan-2-ylamino)picolinamide 367251 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(pyrimidin-5-yl)picolinamide 367252 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(prop-1-enyl)picolinamide 367253 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(1,3-dihydroxypropan-2-ylamino)picolinamide 367258 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(prop-1-enyl)picolinamide 367259 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-styrylpicolinamide 367264 (S)-2-(4-(4-chlorobenzyl)-7-fluoro-5-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid 367267 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(4-hydroxybut-1-enyl)picolinamide 367268 3-(6-((4-(methylsulfonyl)benzyl)carbamoyl)-4-amino-3-cyanopyridin-2-yl)acrylic acid 367275 3-(6-((4-(methylsulfonyl)benzyl)carbamoyl)-4-amino-3-cyanopyridin-2-yl)propanoic acid 367276 N6-(4-(methylsulfonyl)benzyl)-4-amino-3-cyano-N2-isopropylpyridine-2,6-dicarboxamide 367283 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-isopropoxypicolinamide 367284 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(cyclopropylmethoxy)picolinamide 367290 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-isobutoxypicolinamide 367291 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(cyclopentylmethoxy)picolinamide 367298 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(4-methoxyphenoxy)picolinamide 367299 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(isopropylamino)picolinamide 367302 N-(4-(methylsulfonyl)benzyl)-4-amino-6-ethoxy-5-vinylpicolinamide 367303 N-(4-(methylsulfonyl)benzyl)-4-amino-6-ethoxy-5-styrylpicolinamide 367304 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(cyclopropylamino)picolinamide 367305 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(cyclobutylamino)picolinamide 367306 [(3R)-5-bromo-4-(4-chlorobenzyl)-7-fluoro-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl]acetic acid 367309 N-(4-(methylsulfonyl)benzyl)-4-amino-5-(3,3-dimethylbut-1-enyl)-6-ethoxypicolinamide 367310 N-(4-(methylsulfonyl)benzyl)-4-amino-5-(2-cyanovinyl)-6-ethoxypicolinamide 367311 N-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(cyclopentylamino)picolinamide 367312 N-(4-(methylsulfonyl)benzyl)-4-amino-6-(benzylamino)-5-cyanopicolinamide 367313 [(3R)-4-(4-chlorobenzyl)-7-fluoro-5-acetyl-1,2,3,4-tetrahydrocyclopenta-[b]indol-3-yl]acetic acid 367314 [(3R)-4-(4-chlorobenzyl)-7-fluoro-5-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl]-acetic acid 367318 N-(4-(methylsulfonyl)benzyl)-4-amino-5-(but-1-en-3-ynyl)-6-ethoxypicolinamide 367319 N2-(4-(methylsulfonyl)benzyl)-4-amino-6-ethoxypyridine-2,5-dicarboxamide 367354 ((2S,4aR,6aS,7R,9S,10aS,10bR)-9-acetoxy-2-(furan-3-yl)-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-benzo[f]isochromen-7-yl)methyl cyclopropanecarboxylate 367364 (2-methoxy-ethoxy)-acetic acid (3S,4aR,4bS,6S,8R,8aS,10aR)-6-acetoxy-3-furan-3-yl-4a,8a-dimethyl-1,5-dioxo-dodecahydro-2-oxa-phenanthren-8-ylmethyl ester 367469 1-(3-((2S,4R)-4-(4-fluorobenzyl)-1-(2-hydroxyethyl)piperidin-2-yl)propyl)-3-(3,5-diacetylphenyl)urea 367470 1-(3-((2S,4R)-4-(4-fluorobenzyl)-1-(3-hydroxypropyl)piperidin-2-yl)propyl)-3-(3,5-diacetylphenyl)urea 367474 1-(3-((2S,4R)-4-(4-fluorobenzyl)-1-(2-oxopropyl)piperidin-2-yl)propyl)-3-(3,5-diacetylphenyl)urea 367475 1-(3-((2S,4R)-4-(4-fluorobenzyl)-1-(2-amino-2-oxoethyl)piperidin-2-yl)propyl)-3-(3,5-diacetylphenyl)urea 367480 1-(3-((2S,4R)-4-(4-fluorobenzyl)-1-(2-fluoroethyl)piperidin-2-yl)propyl)-3-(3,5-diacetylphenyl)urea 367481 1-(3-((2S,4R)-4-(4-fluorobenzyl)-1-(prop-2-ynyl)piperidin-2-yl)propyl)-3-(3,5-diacetylphenyl)urea 367486 1-(3-((2S,4R)-4-(4-fluorobenzyl)-1-(2,2-difluoroethyl)piperidin-2-yl)propyl)-3-(3,5-diacetylphenyl)urea 367490 1-(3-((2S,4R)-4-(4-fluorobenzyl)-1-(2,2,2-trifluoroethyl)piperidin-2-yl)propyl)-3-(3,5-diacetylphenyl)urea 367491 1-(3-((2S,4R)-4-(4-fluorobenzyl)-1-acetylpiperidin-2-yl)propyl)-3-(3,5-diacetylphenyl)urea 367496 1-(3-((2S,4R)-4-(4-fluorobenzyl)-1-propionylpiperidin-2-yl)propyl)-3-(3,5-diacetylphenyl)urea 367497 (2S,4R)-2-{3-[3-(3,5-diacetyl-phenyl)-ureido]-propyl}-4-(4-fluoro-benzyl)-piperidine-1-carboxamidine 367502 (+/-)1-(3-((2R,4R)-4-benzylpiperidin-2-yl)propyl)-3-(3-cyanophenyl)urea 367508 (-)1-(3-((2S,4R)-4-benzylpiperidin-2-yl)propyl)-3-(3-cyanophenyl)urea 367524 (+/-)1-(2-((2R,4R)-4-benzylpiperidin-2-yl)ethyl)-3-(3-cyanophenyl)urea 367525 (+/-)1-(4-((2S,4R)-4-benzylpiperidin-2-yl)butyl)-3-(3-cyanophenyl)urea 367530 (+/-)1-(3-acetylphenyl)-3-(3-((2S,4R)-4-benzylpiperidin-2-yl)propyl)urea 367531 (+)1-(3-((2S,4R)-4-(4-fluorobenzyl)piperidin-2-yl)propyl)-3-(3-acetylphenyl)urea 367536 (+)1-(3-((2S,4R)-4-(4-fluorobenzyl)piperidin-2-yl)propyl)-3-(3,5-diacetylphenyl)urea 367537 1-(3-((2S,4R)-4-(4-fluorobenzyl)-1-methylpiperidin-2-yl)propyl)-3-(3-acetylphenyl)urea 367542 1-(3-((2S,4R)-4-(4-fluorobenzyl)-1-propylpiperidin-2-yl)propyl)-3-(3-acetylphenyl)urea 367543 1-(3-((2S,4R)-4-(4-fluorobenzyl)-1-(cyclopropylmethyl)piperidin-2-yl)propyl)-3-(3-acetylphenyl)urea 367553 1-(3-((2S,4R)-4-(4-fluorobenzyl)-1-allylpiperidin-2-yl)propyl)-3-(3-acetylphenyl)urea 367554 1-(3-((2S,4R)-4-(4-fluorobenzyl)-1-(2-hydroxyethyl)piperidin-2-yl)propyl)-3-(3-acetylphenyl)urea 367559 1-(3-((2S,4R)-4-(4-fluorobenzyl)-1-propylpiperidin-2-yl)propyl)-3-(3,5-diacetylphenyl)urea 367560 1-(3-((2S,4R)-4-(4-fluorobenzyl)-1-allylpiperidin-2-yl)propyl)-3-(3,5-diacetylphenyl)urea 367565 3-(2-((E)-3-(4-(benzyloxy)-3-methoxyphenyl)prop-1-enyl)phenyl)-N-(thiophen-2-ylsulfonyl)acrylamide 367566 3-(2-(2-(2,6-dichlorobenzyloxy)-5-methylcinnamyl)phenyl)acrylic acid 367567 3-(2-((6-(benzyloxy)naphthalen-2-yl)methyl)phenyl)-N-(5-bromo-2-methoxyphenylsulfonyl)acrylamide 367574 3-(2-(3-(2-(benzyloxy)-5-methylphenyl)propyl)phenyl)propanoic acid 367575 3-(2-(3-(2-(benzyloxy)-5-methylphenyl)propyl)phenyl)-N-(thiophen-2-ylsulfonyl)propanamide 367582 3-(2-(naphthalen-2-ylmethyl)phenyl)-N-(thiophen-2-ylsulfonyl)acrylamide 367588 N-(5-bromo-2-methoxyphenylsulfonyl)-3-(2-(naphthalen-2-ylmethyl)phenyl)acrylamide 367589 3-(2-((6-(benzyloxy)naphthalen-2-yl)methyl)phenyl)acrylic acid 367599 3-(2-((6-(benzyloxy)naphthalen-2-yl)methyl)phenyl)-N-(thiophen-2-ylsulfonyl)acrylamide 367609 7-(naphthalen-2-yl)benzo[e][1,2,4]triazin-3-amine 367610 7-(2,6-dimethylphenyl)benzo[e][1,2,4]triazin-3-amine 367628 7-(2,6-dimethylphenyl)-5-methyl-N-phenylbenzo[e][1,2,4]triazin-3-amine 367629 7-(2,6-dimethylphenyl)-5,6-dimethyl-N-phenylbenzo[e][1,2,4]triazin-3-amine 367635 7-(2,6-dichlorophenyl)-5-methylbenzo[e][1,2,4]triazin-3-amine 367642 3-(2-(2-(benzyloxy)-5-methylcinnamyl)phenyl)acrylic acid 367644 7-(2,6-dimethylphenyl)-5-methylbenzo[e][1,2,4]triazin-3-amine 367645 3-(3-amino-5-methylbenzo[e][1,2,4]triazin-7-yl)-4-chlorophenol 367651 3-(2-((E)-3-(2-(benzyloxy)-5-methylphenyl)prop-1-enyl)phenyl)acrylic acid 367652 3-(2-(2-(benzyloxy)-5-methylcinnamyl)phenyl)-N-(thiophen-2-ylsulfonyl)acrylamide 367660 3-(2-((E)-3-(2-(benzyloxy)-5-methylphenyl)prop-1-enyl)phenyl)-N-(thiophen-2-ylsulfonyl)acrylamide 367661 3-(2-cinnamylphenyl)acrylic acid 367662 3-(3-aminobenzo[e][1,2,4]triazin-7-yl)phenol 367663 7-(benzo[d][1,3]dioxol-5-yl)benzo[e][1,2,4]triazin-3-amine 367668 3-(2-cinnamylphenyl)-N-(thiophen-2-ylsulfonyl)acrylamide 367669 7-(2,6-dimethylphenyl)-N-phenylbenzo[e][1,2,4]triazin-3-amine 367673 3-(2-((E)-3-phenylprop-1-enyl)phenyl)-N-(thiophen-2-ylsulfonyl)acrylamide 367674 3-(2-(4-methoxycinnamyl)phenyl)acrylic acid 367676 N-(3-chlorophenyl)-7-(2,6-dimethylphenyl)-5-methylbenzo[e][1,2,4]triazin-3-amine 367681 3-(2-(4-methoxycinnamyl)phenyl)-N-(thiophen-2-ylsulfonyl)acrylamide 367682 3-(2-((E)-3-(4-methoxyphenyl)prop-1-enyl)phenyl)-N-(thiophen-2-ylsulfonyl)acrylamide 367690 3-(2-(4-(benzyloxy)-3-methoxycinnamyl)phenyl)acrylic acid 367696 3-(2-(4-(benzyloxy)-3-methoxycinnamyl)phenyl)-N-(thiophen-2-ylsulfonyl)acrylamide 367710 7-(2,6-dimethylphenyl)-5-methyl-N-(3-(piperazin-1-ylsulfonyl)phenyl)benzo[e][1,2,4]triazin-3-amine 367711 7-(2,6-dimethylphenyl)-5-methyl-N-(4-(piperazin-1-ylsulfonyl)phenyl)benzo[e][1,2,4]triazin-3-amine 367717 7-(2,6-dimethylphenyl)-N-(3,4-dimethylphenyl)-5-methylbenzo[e][1,2,4]triazin-3-amine 367722 3-(7-(2,6-dimethylphenyl)-5-methylbenzo[e][1,2,4]triazin-3-ylamino)benzenesulfonamide 367730 6-chloro-3-({(cyanoimino)[(2-ethylphenyl)amino]methyl}amino)-2-hydroxy-N,N-dimethylbenzenesulfonamide 367731 1-[4-chloro-3-(dimethylsulfamoyl)-2-hydroxyphenyl]-2-cyano-3-[2-(propan-2-yl)phenyl]guanidine 367732 7-(2,6-dimethylphenyl)-5-methyl-N-(pyridin-4-yl)benzo[e][1,2,4]triazin-3-amine 367742 N-(7-(2,6-dimethylphenyl)-5-methylbenzo[e][1,2,4]triazin-3-yl)benzamide 367743 N-(4-(2-(diethylamino)ethoxy)phenyl)-7-(2,6-dimethylphenyl)-5-methylbenzo[e][1,2,4]triazin-3-amine 367750 N-(3-(2-(diethylamino)ethoxy)phenyl)-7-(2,6-dimethylphenyl)-5-methylbenzo[e][1,2,4]triazin-3-amine 367751 7-(2,6-dimethylphenyl)-N-(4-(2-ethoxymorpholino)phenyl)-5-methylbenzo[e][1,2,4]triazin-3-amine 367758 7-(2,6-dimethylphenyl)-N-(4-(2-ethoxy-4-methylpiperazin-1-yl)phenyl)-5-methylbenzo[e][1,2,4]triazin-3-amine 367759 7-(2,6-dimethylphenyl)-5-methyl-N-(4-(4-methyl-2-propoxypiperazin-1-yl)phenyl)benzo[e][1,2,4]triazin-3-amine 367761 7-(2,6-dimethylphenyl)-5-methyl-N-(3-(4-methyl-2-propoxypiperazin-1-yl)phenyl)benzo[e][1,2,4]triazin-3-amine 367764 7-(2,6-dimethylphenyl)-N-(3-(2-ethoxy-4-methylpiperazin-1-yl)phenyl)-5-methylbenzo[e][1,2,4]triazin-3-amine 367769 7-(2,6-dimethylphenyl)-5-methyl-N-[4-(2-pyrrolidin-1-ylethoxy)phenyl]-1,2,4-benzotriazin-3-amine 367770 7-(2,6-dimethylphenyl)-5-methyl-N-(3-(2-(pyrrolidin-1-yl)ethoxy)phenyl)benzo[e][1,2,4]triazin-3-amine 367776 N-(4-(7-(2,6-dimethylphenyl)-5-methylbenzo[e][1,2,4]triazin-3-ylamino)phenyl)-2-(pyrrolidin-1-yl)ethanesulfonamide 367778 6-chloro-3-({(cyanoimino)[(2-methylphenyl)amino]methyl}amino)-2-hydroxy-N,N-dimethylbenzenesulfonamide 367779 N-(3-(7-(2,6-dimethylphenyl)-5-methylbenzo[e][1,2,4]triazin-3-ylamino)phenyl)-2-(pyrrolidin-1-yl)ethanesulfonamide 367784 6-chloro-3-({(cyanoimino)[(2-fluorophenyl)amino]methyl}amino)-2-hydroxy-N,N-dimethylbenzenesulfonamide 367785 3-{[[(2-bromophenyl)amino](cyanoimino)methyl]amino}-6-chloro-2-hydroxy-N,N-dimethylbenzenesulfonamide 367787 7-(2,6-dimethylphenyl)-5-methyl-N-(3-(4-methylpiperazin-1-ylsulfonyl)phenyl)benzo[e][1,2,4]triazin-3-amine 367793 3-[2-(benzyloxy)phenyl]-1-[4-chloro-3-(dimethylsulfamoyl)-2-hydroxyphenyl]-2-cyanoguanidine 367794 1-[4-chloro-3-(dimethylsulfamoyl)-2-hydroxyphenyl]-2-cyano-3-(2-phenylphenyl)guanidine 367795 7-(2,6-dimethylphenyl)-5-methyl-N-(4-(4-methylpiperazin-1-ylsulfonyl)phenyl)benzo[e][1,2,4]triazin-3-amine 367801 N1-(7-(2,6-dimethylphenyl)-5-methylbenzo[e][1,2,4]triazin-3-yl)-N4,N4-dimethylbenzene-1,4-diamine 367815 7-(2,6-dimethylphenyl)-N-(4-methoxyphenyl)-5-methylbenzo[e][1,2,4]triazin-3-amine 367816 7-(2,6-dimethylphenyl)-N-(4-ethoxyphenyl)-5-methylbenzo[e][1,2,4]triazin-3-amine 367825 7-(2,6-dimethylphenyl)-5-methyl-N-m-tolylbenzo[e][1,2,4]triazin-3-amine 367829 3-(2-bromophenyl)-1-[4-chloro-3-({3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]pentan-3-yl}sulfamoyl)-2-hydroxyphenyl]-2-cyanoguanidine 367830 2-(3H-imidazo[4,5-c]pyridin-3-yl)-6-(4-methylpiperazin-1-yl)-N-((S)-1-phenylethyl)pyrimidin-4-amine 367831 3-(4-(2-chlorophenoxy)-6-(4-methylpiperazin-1-yl)pyrimidin-2-yl)-3H-imidazo[4,5-c]pyridine 367835 1-[4-chloro-3-({3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]pentan-3-yl}sulfamoyl)-2-hydroxyphenyl]-2-cyano-3-(2-methylphenyl)guanidine 367836 3-{[[(2-bromophenyl)amino](cyanoimino)methyl]amino}-2-hydroxy-N,N,6-trimethylbenzenesulfonamide 367842 3-(4-(2,6-difluorophenoxy)-6-(4-methylpiperazin-1-yl)pyrimidin-2-yl)-3H-imidazo[4,5-c]pyridine 367846 3-(2-bromophenyl)-2-cyano-1-(2-hydroxy-4-methyl-3-{[3-(morpholin-4-yl)pentan-3-yl]sulfamoyl}phenyl)guanidine 367847 3-{[[(2-bromophenyl)amino](cyanoimino)methyl]amino}-6-fluoro-2-hydroxy-N,N-dimethylbenzenesulfonamide 367848 N-(2-chlorophenyl)-2-(3H-imidazo[4,5-c]pyridin-3-yl)-6-(4-methylpiperazin-1-yl)pyrimidin-4-amine 367853 3-{[[(2-bromophenyl)amino](cyanoimino)methyl]amino}-2-hydroxy-N,N-dimethyl-6-(trifluoromethyl)benzenesulfonamide 367854 3-(2-bromophenyl)-2-cyano-1-(2-hydroxy-3-{[3-(morpholin-4-yl)pentan-3-yl]sulfamoyl}phenyl)guanidine 367860 3-((3S,4S)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino)piperidin-1-yl)-3-oxopropanenitrile 367867 (R)-1-(2-(3H-imidazo[4,5-c]pyridin-3-yl)-6-((S)-1-phenylethylamino)pyrimidin-4-yl)pyrrolidin-3-ol 367884 2-(3H-imidazo[4,5-c]pyridin-3-yl)-N-((S)-1-phenylethyl)pyrimidin-4-amine 367885 N-((S)-1-(4-fluorophenyl)ethyl)-2-(3H-imidazo[4,5-c]pyridin-3-yl)pyrimidin-4-amine 367886 6-(furan-3-yl)-2-(3H-imidazo[4,5-c]pyridin-3-yl)-N-((S)-1-phenylethyl)pyrimidin-4-amine 367897 N-((S)-1-(4-chlorophenyl)ethyl)-2-(3H-imidazo[4,5-c]pyridin-3-yl)pyrimidin-4-amine 367898 2-(3H-imidazo[4,5-c]pyridin-3-yl)-N-methyl-N-((S)-1-phenylethyl)pyrimidin-4-amine 367900 6-(4-(dimethylamino)phenyl)-2-(3H-imidazo[4,5-c]pyridin-3-yl)-N-((S)-1-phenylethyl)pyrimidin-4-amine 367918 6-(3-(dimethylamino)phenyl)-2-(3H-imidazo[4,5-c]pyridin-3-yl)-N-((S)-1-phenylethyl)pyrimidin-4-amine 367926 2-(3H-imidazo[4,5-c]pyridin-3-yl)-N-((S)-1,2,3,4-tetrahydronaphthalen-1-yl)pyrimidin-4-amine 367927 2-(1H-imidazo[4,5-c]pyridin-1-yl)-N-((S)-1-phenylethyl)pyrimidin-4-amine 367928 6-(3,4-dimethoxyphenyl)-2-(3H-imidazo[4,5-c]pyridin-3-yl)-N-((S)-1-phenylethyl)pyrimidin-4-amine 367935 4-(3H-imidazo[4,5-c]pyridin-3-yl)-N-((R)-1-phenylethyl)pyrimidin-2-amine 367938 2-(3H-imidazo[4,5-c]pyridin-3-yl)-6-(1-methyl-1H-pyrazol-4-yl)-N-((S)-1-phenylethyl)pyrimidin-4-amine 367947 4-(2-(3H-imidazo[4,5-c]pyridin-3-yl)-6-((S)-1-phenylethylamino)pyrimidin-4-yl)benzonitrile 367962 3-(4-((S)-1-methoxypropan-2-ylamino)pyrimidin-2-yl)-3H-benzo[d]imidazole-5-carbonitrile 367964 3-(2-(3H-imidazo[4,5-c]pyridin-3-yl)-6-((S)-1-phenylethylamino)pyrimidin-4-yl)benzonitrile 367967 6-chloro-3-[((cyanoimino){[2-(trifluoromethyl)phenyl]amino}methyl)amino]-2-hydroxy-N,N-dimethylbenzenesulfonamide 367968 6-chloro-3-{[[(3-chloro-2-fluorophenyl)amino](cyanoimino)methyl]amino}-2-hydroxy-N,N-dimethylbenzenesulfonamide 367970 6-(furan-3-yl)-2-(3H-imidazo[4,5-c]pyridin-3-yl)-N-((S)-1-methoxypropan-2-yl)pyrimidin-4-amine 367971 3-(4-(furan-3-yl)-6-((S)-1-phenylethylamino)pyrimidin-2-yl)-3H-benzo[d]imidazole-5-carbonitrile 367983 (R)-1-(3-(3-(3-(2-bromophenyl)-2-cyanoguanidino)-6-chloro-2-hydroxyphenylsulfonamido)pentan-3-yl)pyrrolidine-2-carboxylic acid 367986 N-((S)-1-(4-fluorophenyl)ethyl)-6-(furan-3-yl)-2-(3H-imidazo[4,5-c]pyridin-3-yl)pyrimidin-4-amine 367990 1-(3-{[3-(4-aminopiperidin-1-yl)pentan-3-yl]sulfamoyl}-4-chloro-2-hydroxyphenyl)-3-(2-bromophenyl)-2-cyanoguanidine 367992 2-(3H-imidazo[4,5-c]pyridin-3-yl)-N4,N4-dimethyl-N6-((S)-1-phenylethyl)pyrimidine-4,6-diamine 368007 3-(1-(3-aminopropyl)-1H-indazol-3-yl)-4-(1-(benzo[b]thiophen-3-yl)-1H-indol-3-yl)-1H-pyrrole-2,5-dione 368063 3-[4'-(H-Dmt)-aminobutyl]-6-[3'-(H-Dmt)-aminopropyl]-5-methyl-2(1H)-pyrazinone 368083 SID26753040 368126 H-Tyr-Asn-Trp-Asn-Ser-Phe-Gly-Leu-Arg-Phe-NH2 368127 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]-2-phenylethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368128 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]-2-phenylethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}ethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368129 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]-2-phenylethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368130 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]-2-phenylethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}ethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368131 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]-2-phenylethyl]carbamoyl}ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368132 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]ethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368133 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}ethyl]carbamoyl}-2-phenylethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368134 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}butyl]carbamoyl}ethyl]carbamoyl}methyl)carbamoyl]-2-phenylethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368135 (2S)-2-[(2S)-2-[(2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-3-carbamoylpropanamido]-3-(4-hydroxyphenyl)propanamido]-N-[(1S)-1-{[(1S)-2-carbamoyl-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}ethyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]-2-phenylethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}ethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]butanediamide 368136 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoylethyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]-2-phenylethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368137 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368138 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]-2-(4-hydroxyphenyl)ethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368139 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]-3-methylbutyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368140 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]-2-cyclohexylethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368141 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]-2-(1H-imidazol-5-yl)ethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368142 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]-2-(pyridin-3-yl)ethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368143 (2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-3-carbamoylpropanamido]-3-(4-hydroxyphenyl)propanamido]-3-carbamoylpropanamido]-3-(1H-indol-3-yl)propanamido]-3-carbamoylpropanamido]-3-hydroxypropanamido]-N-({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)pentanediamide 368144 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-4-carbamimidamido-1-[({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]butyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368152 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-(1H-indol-3-yl)ethyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]-2-phenylethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368153 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-(4-hydroxyphenyl)ethyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]-2-phenylethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368154 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-cyclohexylethyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]-2-phenylethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368155 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-(1H-imidazol-4-yl)ethyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]-2-phenylethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368156 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-(pyridin-3-yl)ethyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]-2-phenylethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368157 (2S)-2-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-3-carbamoylpropanamido]-3-(4-hydroxyphenyl)propanamido]-3-carbamoylpropanamido]-3-(1H-indol-3-yl)propanamido]-3-carbamoylpropanamido]-3-hydroxypropanamido]-3-phenylpropanamido]acetamido}-4-methylpentanamido]-5-carbamimidamidopentanamido]pentanediamide 368158 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-4-carbamimidamido-1-carbamoylbutyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]-2-phenylethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368160 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoylethyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]ethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368161 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-4-carbamimidamido-1-carbamoylbutyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]ethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368162 LPNYNWNSFLRF-NH2 368163 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}-3-methylbutyl]carbamoyl}-2-phenylethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368164 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(2S)-1-[(2S)-2-{[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamoyl}pyrrolidin-1-yl]-1-oxo-3-phenylpropan-2-yl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368165 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S,2S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}butyl]carbamoyl}-2-methylbutyl]carbamoyl}methyl)carbamoyl]-2-phenylethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368167 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}butyl]carbamoyl}pentyl]carbamoyl}methyl)carbamoyl]-2-phenylethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368168 (2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-({2-[(2S)-2-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}butyl]carbamoyl}pyrrolidin-1-yl]-2-oxoethyl}carbamoyl)-2-phenylethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide 368169 (2S)-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-5-amino-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}pentyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]-2-phenylethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}butanediamide 368177 (2S)-2-[(2S)-2-[(2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-3-carbamoylpropanamido]-3-(4-hydroxyphenyl)propanamido]-N-[(1S)-1-{[(1S)-2-carbamoyl-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}-4-(carbamoylamino)butyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]-2-phenylethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}ethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]butanediamide 368178 (2S)-2-[(2S)-2-[(2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidin-2-yl]formamido}-3-carbamoylpropanamido]-3-(4-hydroxyphenyl)propanamido]-N-[(1S)-1-{[(1S)-2-carbamoyl-1-{[(1S)-1-{[(1S)-1-[({[(1S)-1-{[(1S)-1-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}-3-phenylpropyl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamoyl]-2-phenylethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}ethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl]butanediamide 368180 LPNYNWNSFGLRF-NH2 368181 LPNYNWNSFGLRF 368203 N'-ethyl-3-methoxy-N',2-diphenylquinoline-4-carbohydrazide 368204 3-methoxy-N',N',2-triphenylquinoline-4-carbohydrazide 368211 N'-acetyl-3-methoxy-N',2-diphenylquinoline-4-carbohydrazide 368212 3-methoxy-N',2-diphenyl-N'-propionylquinoline-4-carbohydrazide 368221 N'-(3-methoxy-2-phenyl-quinoline-4-carbonyl)-N-phenyl-hydrazinecarboxylic acid methyl ester 368222 N'-(3-methoxy-2-phenyl-quinoline-4-carbonyl)-N-phenyl-hydrazinecarboxylic acid ethyl ester 368239 N'-(3-methoxy-2-phenyl-quinoline-4-carbonyl)-N-phenyl-hydrazinecarboxylic acid isobutyl ester 368240 N-phenyl-N'-(2-phenyl-quinoline-4-carbonyl)-hydrazinecarboxylic acid methyl ester 368249 N'-(3-methyl-2-phenyl-quinoline-4-carbonyl)-N-phenyl-hydrazinecarboxylic acid methyl ester 368250 N'-(3-amino-2-phenyl-quinoline-4-carbonyl)-N-phenyl-hydrazinecarboxylic acid methyl ester 368258 N'-(3-hydroxy-2-phenyl-quinoline-4-carbonyl)-N-phenyl-hydrazinecarboxylic acid methyl ester 368259 N-(2-fluoro-phenyl)-N'-(3-methoxy-2-phenyl-quinoline-4-carbonyl)-hydrazinecarboxylic acid methyl ester 368264 2-(2-chlorophenyl)-6-(2-chlorophenylamino)pyridazin-3(2H)-one 368266 N-(3-fluoro-phenyl)-N'-(3-methoxy-2-phenyl-quinoline-4-carbonyl)-hydrazinecarboxylic acid methyl ester 368267 N-(4-fluoro-phenyl)-N'-(3-methoxy-2-phenyl-quinoline-4-carbonyl)-hydrazinecarboxylic acid methyl ester 368272 2-(2-chlorophenyl)-6-(2-ethylphenylamino)pyridazin-3(2H)-one 368273 6-(o-toluidino)-2-(2-chlorophenyl)pyridazin-3(2H)-one 368274 2-(2-chlorophenyl)-6-(2-methoxyphenylamino)pyridazin-3(2H)-one 368275 N'-[2-(2-fluoro-phenyl)-3-methoxy-quinoline-4-carbonyl]-N-phenyl-hydrazinecarboxylic acid methyl ester 368276 N'-[2-(3-fluoro-phenyl)-3-methoxy-quinoline-4-carbonyl]-N-phenyl-hydrazinecarboxylic acid methyl ester 368281 2-(2-chlorophenyl)-6-(2-fluorophenylthio)pyridazin-3(2H)-one 368282 2-(4-chloro-2-methylphenyl)-6-(2,4-difluorophenylthio)pyridazin-3(2H)-one 368283 2-(4-chloro-2-methylphenyl)-6-(4-chlorophenylthio)pyridazin-3(2H)-one 368284 N'-[2-(4-fluoro-phenyl)-3-methoxy-quinoline-4-carbonyl]-N-phenyl-hydrazinecarboxylic acid methyl ester 368285 N'-(5-fluoro-3-methoxy-2-phenyl-quinoline-4-carbonyl)-N-phenyl-hydrazinecarboxylic acid methyl ester 368288 6-[4'-(H-Dmt)-aminobutyl]-3-[3'-(H-Dmt)-aminopropyl]-5-methyl-2(1H)-pyrazinone 368293 2-(2-chlorophenyl)-6-[(2-methylbenzyl)amino]pyridazin-3(2H)-one 368294 N'-(6-fluoro-3-methoxy-2-phenyl-quinoline-4-carbonyl)-N-phenyl-hydrazinecarboxylic acid methyl ester 368295 N'-(7-fluoro-3-methoxy-2-phenyl-quinoline-4-carbonyl)-N-phenyl-hydrazinecarboxylic acid methyl ester 368301 6-((2-chloro-4-fluorophenyl)(2-hydroxyethyl)amino)-2-(2-chlorophenyl)pyridazin-3(2H)-one 368302 N'-(8-fluoro-3-methoxy-2-phenyl-quinoline-4-carbonyl)-N-phenyl-hydrazinecarboxylic acid methyl ester 368303 N'-(8-bromo-3-methoxy-2-phenyl-quinoline-4-carbonyl)-N-phenyl-hydrazinecarboxylic acid methyl ester 368308 6-((3-aminopropyl)(2-chlorophenyl)amino)-2-(2-chlorophenyl)pyridazin-3(2H)-one 368309 6-((3-(2,3,4-trimethoxybenzylamino)propyl)(2-chlorophenyl)amino)-2-(2-chlorophenyl)pyridazin-3(2H)-one 368312 6-[4'-(H-Tyr)-aminobutyl]-3-[3'-(H-tyr)-amino-propyl]-5-methyl-2(1H)-pyrazinone 368316 2-(3-((2-chlorophenyl)(1-(2-chlorophenyl)-6-oxo-1,6-dihydropyridazin-3-yl)amino)propyl)isoindoline-1,3-dione 368317 2-(3-((2-chloro-4-fluorophenyl)(1-(2-chlorophenyl)-6-oxo-1,6-dihydropyridazin-3-yl)amino)propyl)isoindoline-1,3-dione 368325 2-amino-N-(3-((2-chlorophenyl)(1-(2-chlorophenyl)-6-oxo-1,6-dihydropyridazin-3-yl)amino)propyl)acetamide 368326 N-(3-((2-chlorophenyl)(1-(2-chlorophenyl)-6-oxo-1,6-dihydropyridazin-3-yl)amino)propyl)-2-(methylamino)acetamide 368337 N-(3-((2-chlorophenyl)(1-(2-chlorophenyl)-6-oxo-1,6-dihydropyridazin-3-yl)amino)propyl)-2-(pyrrolidin-2-yl)acetamide 368338 N-(3-((2-chlorophenyl)(1-(2-chlorophenyl)-6-oxo-1,6-dihydropyridazin-3-yl)amino)propyl)piperidine-4-carboxamide 368345 N-(3-((2-chlorophenyl)(1-(2-chlorophenyl)-6-oxo-1,6-dihydropyridazin-3-yl)amino)propyl)-4-(trifluoromethyl)cyclohexanecarboxamide 368360 3-methoxy-N',2-diphenylquinoline-4-carbohydrazide 368361 3-methoxy-N'-methyl-N',2-diphenylquinoline-4-carbohydrazide 368473 3-[4'-(H-Tyr)-aminobutyl]-6-[3'-(H-Tyr)-amino-propyl]-5-methyl-2(1H)-pyrazinone 368492 N-tert-butyl-7-(2,4-difluorophenyl)-2,3-dihydro-1H-1,4-diazepin-5-amine 368493 N-ethyl-N-((2-(4-fluorophenyl)-3-(2-((S)-1-phenylethyl)pyrimidin-4-yl)H-imidazo[1,2-a]pyridin-7-yl)methyl)ethanamine 368501 N-tert-butyl-7-(2-chlorophenyl)-2,3-dihydro-1H-1,4-diazepin-5-amine 368502 (2-(4-fluorophenyl)-3-(2-((S)-1-phenylethyl)pyrimidin-4-yl)H-imidazo[1,2-a]pyridin-7-yl)-N-hydroxy-N-methylmethanamine 368509 (2-(4-fluorophenyl)-3-(2-((S)-1-phenylethyl)pyrimidin-4-yl)H-imidazo[1,2-a]pyridin-7-yl)-N-methoxy-N-methylmethanamine 368510 4-(7-(tert-butylamino)-3,4-dihydro-2H-1,4-diazepin-5-yl)benzonitrile 368516 N-((2-(4-fluorophenyl)-3-(2-((S)-1-phenylethyl)pyrimidin-4-yl)H-imidazo[1,2-a]pyridin-7-yl)methyl)acetamide 368517 (2-(4-fluorophenyl)-3-(2-((S)-1-phenylethyl)pyrimidin-4-yl)H-imidazo[1,2-a]pyridin-7-yl)methanamine 368522 N-tert-butyl-7-(3-(trifluoromethyl)phenyl)-2,3-dihydro-1H-1,4-diazepin-5-amine 368529 7-(2-fluorophenyl)-N-neopentyl-2,3-dihydro-1H-1,4-diazepin-5-amine 368530 7-(4-fluorophenyl)-N-(1-methylcyclohexyl)-2,3-dihydro-1H-1,4-diazepin-5-amine 368531 7-(4-fluorophenyl)-N-(3-methylpentan-3-yl)-2,3-dihydro-1H-1,4-diazepin-5-amine 368537 N-(3-methylpentan-3-yl)-7-p-tolyl-2,3-dihydro-1H-1,4-diazepin-5-amine 368544 N-tert-butyl-7-(2-fluoro-4-methylphenyl)-2,3-dihydro-1H-1,4-diazepin-5-amine 368545 N-tert-butyl-7-(2,4-dimethylphenyl)-2,3-dihydro-1H-1,4-diazepin-5-amine 368546 7-(2-fluorophenyl)-N-(3-methylpentan-3-yl)-2,3-dihydro-1H-1,4-diazepin-5-amine 368553 N-tert-butyl-7-phenyl-2,3-dihydro-1H-1,4-diazepin-5-amine 368554 N-tert-butyl-7-p-tolyl-2,3-dihydro-1H-1,4-diazepin-5-amine 368555 N-(1-ethylcyclopentyl)-7-(4-fluorophenyl)-2,3-dihydro-1H-1,4-diazepin-5-amine 368556 7-(2,4-difluorophenyl)-N-(1-ethylcyclopentyl)-2,3-dihydro-1H-1,4-diazepin-5-amine 368557 N-(2-cyclobutylpropan-2-yl)-7-(2,4-difluorophenyl)-2,3-dihydro-1H-1,4-diazepin-5-amine 368563 4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-imidazo[1,2-a]pyridin-3-yl)-N-((R)-1-phenylethyl)pyrimidin-2-amine 368564 4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-imidazo[1,2-a]pyridin-3-yl)-N-((S)-1-phenylethyl)pyrimidin-2-amine 368579 N-benzyl-4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-imidazo[1,2-a]pyridin-3-yl)-N-methylpyrimidin-2-amine 368580 N-tert-butyl-7-o-tolyl-2,3-dihydro-1H-1,4-diazepin-5-amine 368581 7-(2-fluorophenyl)-N-(2-methyl-1-phenylpropan-2-yl)-2,3-dihydro-1H-1,4-diazepin-5-amine 368582 N-(1-ethylcyclopentyl)-7-(2-fluorophenyl)-2,3-dihydro-1H-1,4-diazepin-5-amine 368589 (3-(2-(benzyloxy)pyrimidin-4-yl)-2-(4-fluorophenyl)H-imidazo[1,2-a]pyridin-7-yl)-N,N-dimethylmethanamine 368590 N-tert-butyl-7-(4-methoxyphenyl)-2,3-dihydro-1H-1,4-diazepin-5-amine 368591 7-(2,4-difluorophenyl)-N-(3-ethylpentan-3-yl)-2,3-dihydro-1H-1,4-diazepin-5-amine 368593 N-(2-methyl-1-phenylpropan-2-yl)-7-p-tolyl-2,3-dihydro-1H-1,4-diazepin-5-amine 368599 2-(ethyl((2-(4-fluorophenyl)-3-(2-((S)-1-phenylethyl)pyrimidin-4-yl)H-imidazo[1,2-a]pyridin-7-yl)methyl)amino)ethanol 368600 2-(((2-(4-fluorophenyl)-3-(2-((S)-1-phenylethyl)pyrimidin-4-yl)H-imidazo[1,2-a]pyridin-7-yl)methyl)(methyl)amino)ethanol 368607 N-tert-butyl-7-(2-fluorophenyl)-2,3-dihydro-1H-1,4-diazepin-5-amine 368608 N-((2-(4-fluorophenyl)-3-(2-((S)-1-phenylethyl)pyrimidin-4-yl)H-imidazo[1,2-a]pyridin-7-yl)methyl)-N-methylethanamine 368616 N-((2-(4-fluorophenyl)-3-(2-((S)-1-phenylethyl)pyrimidin-4-yl)H-imidazo[1,2-a]pyridin-7-yl)methyl)ethanamine 368617 (2-(4-fluorophenyl)-3-(2-((S)-1-phenylethyl)pyrimidin-4-yl)H-imidazo[1,2-a]pyridin-7-yl)-N-methylmethanamine 368626 N-tert-butyl-7-(4-fluorophenyl)-2,3-dihydro-1H-1,4-diazepin-5-amine 368627 N-((2-(4-fluorophenyl)-3-(2-((S)-1-phenylethyl)pyrimidin-4-yl)H-imidazo[1,2-a]pyridin-7-yl)methyl)-2-methylpropan-2-amine 368637 3-(5-((4-(aminomethyl)piperidin-1-yl)methyl)-1H-indol-2-yl)-2-oxo-1,2-dihydroquinoline-6-carbonitrile 368638 3-(5-((4-(aminomethyl)piperidin-1-yl)methyl)-1H-indol-2-yl)-2-oxo-1,2-dihydroquinoline-6-carboxamide 368639 2-(1H-benzo[d]imidazol-1-yl)-N-(5-methoxy-2-methylphenyl)pyrimidin-4-amine 368645 2-oxo-3-(5-(piperidin-1-ylmethyl)-1H-indol-2-yl)-1,2-dihydroquinoline-6-carbonitrile 368646 6-bromo-3-(5-(piperidin-1-ylmethyl)-1H-indol-2-yl)quinolin-2(1H)-one 368648 3-(2-(1H-benzo[d]imidazol-1-yl)-6-chloropyrimidin-4-ylamino)-4-methylphenol 368652 2-oxo-3-(5-(piperidin-1-ylmethyl)-1H-indol-2-yl)-1,2-dihydroquinoline-6-carboxamide 368653 3-(5-(piperidin-1-ylmethyl)-1H-indol-2-yl)-6-(1H-pyrazol-4-yl)quinolin-2(1H)-one 368654 3-(6-amino-2-(1H-benzo[d]imidazol-1-yl)pyrimidin-4-ylamino)-4-methylphenol 368655 3-(2-(1H-benzo[d]imidazol-1-yl)-6-(methylamino)pyrimidin-4-ylamino)-4-methylphenol 368658 3-(5-(piperidin-1-ylmethyl)-1H-indol-2-yl)-6-(1H-pyrazol-3-yl)quinolin-2(1H)-one 368659 6-(1H-imidazol-1-yl)-3-(5-(piperidin-1-ylmethyl)-1H-indol-2-yl)quinolin-2(1H)-one 368660 3-(2-(1H-benzo[d]imidazol-1-yl)-6-(dimethylamino)pyrimidin-4-ylamino)-4-methylphenol 368661 3-(2-(1H-benzo[d]imidazol-1-yl)-6-methoxypyrimidin-4-ylamino)-4-methylphenol 368667 6-(1-methyl-1H-pyrazol-4-yl)-3-(5-(piperidin-1-ylmethyl)-1H-indol-2-yl)quinolin-2(1H)-one 368668 3-(2-(1H-benzo[d]imidazol-1-yl)-6-morpholinopyrimidin-4-ylamino)-4-methylphenol 368669 3-(2-(1H-benzo[d]imidazol-1-yl)-6-(4-methylpiperazin-1-yl)pyrimidin-4-ylamino)-4-methylphenol 368674 6-(isothiazol-4-yl)-3-(5-(piperidin-1-ylmethyl)-1H-indol-2-yl)quinolin-2(1H)-one 368675 1-(3-(2,5-dimethylbenzyl)-5-(3-cyclohexylpropyl)phenyl)-1H-indene 368676 2-(1H-benzo[d]imidazol-1-yl)-N-(5-methoxy-2-methylphenyl)-6-(2-morpholinoethoxy)pyrimidin-4-amine 368680 6-(2-methyl-2H-tetrazol-5-yl)-3-(5-(piperidin-1-ylmethyl)-1H-indol-2-yl)quinolin-2(1H)-one 368682 3-(2-(1H-benzo[d]imidazol-1-yl)-6-(2-morpholinoethylamino)pyrimidin-4-ylamino)-4-methylphenol 368683 3-(2-(1H-benzo[d]imidazol-1-yl)-6-(2-(4-methylpiperazin-1-yl)ethoxy)pyrimidin-4-ylamino)-4-methylphenol 368688 3-(5-(piperidin-1-ylmethyl)-1H-indol-2-yl)-6-(1H-1,2,3-triazol-1-yl)quinolin-2(1H)-one 368691 3-(2-(1H-benzo[d]imidazol-1-yl)-6-(2-(diethylamino)ethylamino)pyrimidin-4-ylamino)-4-methylphenol 368692 3-(2-(1H-benzo[d]imidazol-1-yl)-6-(3-(dimethylamino)propylamino)pyrimidin-4-ylamino)-4-methylphenol 368696 3-(5-(piperidin-1-ylmethyl)-1H-indol-2-yl)-6-(2H-1,2,3-triazol-2-yl)quinolin-2(1H)-one 368698 3-(2-(1H-benzo[d]imidazol-1-yl)-6-(3-(piperazin-1-yl)propylamino)pyrimidin-4-ylamino)-4-methylphenol 368699 3-(2-(1H-benzo[d]imidazol-1-yl)-6-(2-(4-methylpiperazin-1-yl)ethylamino)pyrimidin-4-ylamino)-4-methylphenol 368703 6-(3-hydroxyphenyl)-3-(5-(piperidin-1-ylmethyl)-1H-indol-2-yl)quinolin-2(1H)-one 368704 6-(4-hydroxy-3-methoxyphenyl)-3-(5-(piperidin-1-ylmethyl)-1H-indol-2-yl)quinolin-2(1H)-one 368705 3-(2-(1H-benzo[d]imidazol-1-yl)-6-(4-methylpiperazin-1-ylamino)pyrimidin-4-ylamino)-4-methylphenol 368706 3-(2-(1H-benzo[d]imidazol-1-yl)-6-(morpholinoamino)pyrimidin-4-ylamino)-4-methylphenol 368710 3-(5-((4-fluoropiperidin-1-yl)methyl)-1H-indol-2-yl)-6-(1H-pyrazol-4-yl)quinolin-2(1H)-one 368711 3-(5-(morpholinomethyl)-1H-indol-2-yl)-6-(1H-pyrazol-4-yl)quinolin-2(1H)-one 368712 3-(2-(1H-benzo[d]imidazol-1-yl)-6-((1-methylpiperidin-4-yl)methyl)pyrimidin-4-ylamino)-4-methylphenol 368713 3-(5-((4-acetylpiperazin-1-yl)methyl)-1H-indol-2-yl)-6-(1-methyl-1H-pyrazol-4-yl)quinolin-2(1H)-one 368718 3-(5-((4-acetylpiperazin-1-yl)methyl)-1H-indol-2-yl)-6-(1H-pyrazol-4-yl)quinolin-2(1H)-one 368719 3-(5-((4-(2-methoxyacetyl)piperazin-1-yl)methyl)-1H-indol-2-yl)-6-(1H-pyrazol-4-yl)quinolin-2(1H)-one 368720 3-(2-(1H-benzo[d]imidazol-1-yl)-6-(3-(piperidin-4-yl)propyl)pyrimidin-4-ylamino)-4-methylphenol 368725 3-(4-(1H-benzo[d]imidazol-1-yl)pyrimidin-2-ylamino)-4-methylphenol 368727 3-(4-(benzo[d]isoxazol-3-yl)pyrimidin-2-ylamino)-4-methylphenol 368732 3-(5-((4-(aminomethyl)piperidin-1-yl)methyl)-1H-indol-2-yl)-1H-indazole-6-carbonitrile 368733 3-(4-(1H-benzo[d]imidazol-1-yl)pyrimidin-2-ylamino)-4-methylbenzamide 368734 N-(3-(4-(1H-benzo[d]imidazol-1-yl)pyrimidin-2-ylamino)-4-methylphenyl)acetamide 368739 3-(5-((4-(aminomethyl)piperidin-1-yl)methyl)-1H-indol-2-yl)quinolin-2(1H)-one 368740 3-(1H-indol-2-yl)quinolin-2(1H)-one 368742 3-(2-(1H-benzo[d]imidazol-1-yl)pyrimidin-4-ylamino)-4-methylphenol 368743 N1-(4-(benzo[d]isoxazol-3-yl)pyrimidin-2-yl)-6-methylbenzene-1,3-diamine 368747 3-(5-((4-(aminomethyl)piperidin-1-yl)methyl)-1H-indol-2-yl)-2-oxo-1,2-dihydroquinoline-5-carbonitrile 368748 3-(5-((4-(aminomethyl)piperidin-1-yl)methyl)-1H-indol-2-yl)-2-oxo-1,2-dihydroquinoline-7-carbonitrile 368751 1-(4-((2-(6-chloro-1H-indazol-3-yl)-1H-indol-5-yl)methyl)piperazin-1-yl)ethanone 368752 1-(4-((2-(1H-indazol-3-yl)-1H-indol-5-yl)methyl)piperazin-1-yl)ethanone 368754 (E)-4-amino-6-(4-fluoro-2-methyl-1H-indol-5-yloxy)pyrimidine-5-carbaldehyde O-3-hydroxypropoxy oxime 368758 3-(5-(morpholinomethyl)-1H-indol-2-yl)-1H-indazole-6-carbonitrile 368759 methyl 3-(5-(morpholinomethyl)-1H-indol-2-yl)-1H-indazole-6-carboxylate 368764 3-(5-(morpholinomethyl)-1H-indol-2-yl)-1H-indazole-6-carboxamide 368765 N-methyl-3-(5-(morpholinomethyl)-1H-indol-2-yl)-1H-indazole-6-carboxamide 368771 N,N-dimethyl-3-(5-(morpholinomethyl)-1H-indol-2-yl)-1H-indazole-6-carboxamide 368772 3-(5-(morpholinomethyl)-1H-indol-2-yl)-6-(1H-pyrazol-4-yl)-1H-indazole 368778 6-(1-methyl-1H-pyrazol-4-yl)-3-(5-(morpholinomethyl)-1H-indol-2-yl)-1H-indazole 368779 3-(5-(morpholinomethyl)-1H-indol-2-yl)-6-(1H-pyrazol-5-yl)-1H-indazole 368785 6-(isothiazol-4-yl)-3-(5-(piperidin-1-ylmethyl)-1H-indol-2-yl)-1H-indazole 368786 3-(5-(piperidin-1-ylmethyl)-1H-indol-2-yl)-6-(thiazol-2-yl)-1H-indazole 368788 (E)-4-amino-6-(quinolin-6-yloxy)pyrimidine-5-carbaldehyde O-methyl oxime 368800 2-(2-chloro-4-(3-(4-methylpiperazin-1-yl)propoxy)phenyl)-4,5-dimethyl-1H-benzo[d]imidazole 368801 3-(5-(piperidin-1-ylmethyl)-1H-indol-2-yl)-6-(1H-1,2,3-triazol-1-yl)-1H-indazole 368802 6-(5-methyl-1H-1,2,3-triazol-1-yl)-3-(5-(piperidin-1-ylmethyl)-1H-indol-2-yl)-1H-indazole 368803 (E)-4-amino-6-(quinolin-7-yloxy)pyrimidine-5-carbaldehyde O-methyl oxime 368804 (E)-4-(1H-indol-5-yloxy)-6-aminopyrimidine-5-carbaldehyde O-methyl oxime 368805 (E)-4-amino-6-(1-methyl-1H-indol-5-yloxy)pyrimidine-5-carbaldehyde O-methyl oxime 368808 2-(2-chloro-4-(3-(4-methylpiperazin-1-yl)propoxy)phenyl)-4,6-dimethyl-1H-benzo[d]imidazole 368809 5-tert-butyl-2-(2-chloro-4-(3-(4-methylpiperazin-1-yl)propoxy)phenyl)-1H-benzo[d]imidazole 368810 3-(5-(piperidin-1-ylmethyl)-1H-indol-2-yl)-6-(1H-pyrazol-1-yl)-1H-indazole 368811 3-(5-(piperidin-1-ylmethyl)-1H-indol-2-yl)-6-(2H-1,2,3-triazol-2-yl)-1H-indazole 368812 (E)-4-amino-6-(2-methyl-1H-indol-5-yloxy)pyrimidine-5-carbaldehyde O-methyl oxime 368813 (E)-4-amino-6-(3-methyl-1H-indol-5-yloxy)pyrimidine-5-carbaldehyde O-methyl oxime 368814 (E)-4-amino-6-(4-fluoro-1H-indol-5-yloxy)pyrimidine-5-carbaldehyde O-methyl oxime 368817 2-(2-chloro-4-(3-(4-methylpiperazin-1-yl)propoxy)phenyl)-3H-naphtho[2,1-d]imidazole 368818 1-(3-(4-(5-tert-butyl-1H-benzo[d]imidazol-2-yl)-2-chlorophenoxy)propyl)-N,N-dimethylpyrrolidin-3-amine 368819 6-phenyl-3-(5-(piperidin-1-ylmethyl)-1H-indol-2-yl)-1H-indazole 368820 (5-(3-(5-(piperidin-1-ylmethyl)-1H-indol-2-yl)-1H-indazol-6-yl)-1H-1,2,3-triazol-4-yl)methanol 368821 (E)-4-amino-6-(6-fluoro-1H-indol-5-yloxy)pyrimidine-5-carbaldehyde O-methyl oxime 368822 (E)-4-amino-6-(4-fluoro-2-methyl-1H-indol-5-yloxy)pyrimidine-5-carbaldehyde O-ethyl oxime 368823 (E)-4-amino-6-(4-fluoro-2-methyl-1H-indol-5-yloxy)pyrimidine-5-carbaldehyde O-propyl oxime 368826 5-tert-butyl-2-(3-chloro-4-(3-(4-methyl-1,4-diazepan-1-yl)propoxy)phenyl)-1H-benzo[d]imidazole 368827 5-tert-butyl-2-(3-chloro-4-(3-(4-methylpiperazin-1-yl)propoxy)phenyl)-1H-benzo[d]imidazole 368828 (5-(3-(5-((4-fluoropiperidin-1-yl)methyl)-1H-indol-2-yl)-1H-indazol-6-yl)-1H-1,2,3-triazol-4-yl)methanol 368829 (5-(3-(5-((4-fluoropiperidin-1-yl)methyl)-1H-indol-2-yl)-1H-indazol-6-yl)-1H-1,2,3-triazol-4-yl)methanamine 368830 (E)-4-amino-6-(4-fluoro-2-methyl-1H-indol-5-yloxy)pyrimidine-5-carbaldehyde O-butyl oxime 368831 (E)-4-amino-6-(4-fluoro-2-methyl-1H-indol-5-yloxy)pyrimidine-5-carbaldehyde O-allyl oxime 368834 5-tert-butyl-2-(3-methyl-4-(3-(4-methylpiperazin-1-yl)propoxy)phenyl)-1H-benzo[d]imidazole 368835 2-(2-chloro-4-(3-(4-methyl-1,4-diazepan-1-yl)propoxy)phenyl)-4,5-dimethyl-1H-benzo[d]imidazole 368836 2-methoxy-4-(3-(5-(piperidin-1-ylmethyl)-1H-indol-2-yl)-1H-indazol-6-yl)phenol 368838 (E)-4-amino-6-(4-fluoro-2-methyl-1H-indol-5-yloxy)pyrimidine-5-carbaldehyde O-prop-2-ynyl oxime 368839 (E)-4-amino-6-(4-fluoro-2-methyl-1H-indol-5-yloxy)pyrimidine-5-carbaldehyde O-cyclohexylmethyl oxime 368841 2-(2-chloro-4-(3-(4-methyl-1,4-diazepan-1-yl)propoxy)phenyl)-4,6-dimethyl-1H-benzo[d]imidazole 368845 4-amino-6-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]pyrimidine-5-carbaldehyde O-benzyloxime 368846 (E)-4-amino-6-(4-fluoro-2-methyl-1H-indol-5-yloxy)pyrimidine-5-carbaldehyde O-2-(methylamino)ethoxy oxime 368853 (E)-4-amino-6-(4-fluoro-2-methyl-1H-indol-5-yloxy)pyrimidine-5-carbaldehyde O-2-(dimethylamino)ethoxy oxime 368854 (E)-4-amino-6-(4-fluoro-2-methyl-1H-indol-5-yloxy)pyrimidine-5-carbaldehyde O-2-(pyrrolidin-1-yl)ethoxy oxime 368860 (E)-4-amino-6-(4-fluoro-2-methyl-1H-indol-5-yloxy)pyrimidine-5-carbaldehyde O-2-morpholinoethoxy oxime 368861 (E)-4-amino-6-(4-fluoro-2-methyl-1H-indol-5-yloxy)pyrimidine-5-carbaldehyde O-3-(dimethylamino)propoxy oxime 368865 3-(1H-indol-2-yl)-6-(1H-tetrazol-5-yl)-1H-indazole 368867 (E)-4-amino-6-(4-fluoro-2-methyl-1H-indol-5-yloxy)pyrimidine-5-carbaldehyde O-2-methoxyethoxy oxime 368868 (E)-4-amino-6-(4-fluoro-2-methyl-1H-indol-5-yloxy)pyrimidine-5-carbaldehyde O-3-methoxypropoxy oxime 368871 1-(4-((2-(6-(1H-tetrazol-5-yl)-1H-indazol-3-yl)-1H-indol-5-yl)methyl)piperazin-1-yl)ethanone 368872 3-(5-((4-acetylpiperazin-1-yl)methyl)-1H-indol-2-yl)-1H-indazole-6-carbonitrile 368874 (E)-4-amino-6-(4-fluoro-2-methyl-1H-indol-5-yloxy)pyrimidine-5-carbaldehyde oxime 368875 (E)-4-amino-6-(4-fluoro-2-methyl-1H-indol-5-yloxy)pyrimidine-5-carbaldehyde O-2-hydroxyethoxy oxime 368878 4-(3-chloro-4-fluorophenylamino)-6-((2-ethyl-1H-imidazol-4-yl)methylamino)quinoline-3-carbonitrile 368879 4-(3-chloro-4-fluorophenylamino)-6-((1,4-dimethyl-1H-imidazol-5-yl)methylamino)quinoline-3-carbonitrile 368884 6-(benzylamino)-4-(3-chloro-4-fluorophenylamino)quinoline-3-carbonitrile 368886 4-(3-chloro-4-fluorophenylamino)-6-((4-methyl-1-(2-morpholinoethyl)-1H-imidazol-5-yl)methylamino)quinoline-3-carbonitrile 368892 N-(4-(3-chloro-4-fluorophenylamino)-3-cyanoquinolin-6-yl)benzamide 368893 4-(3-chloro-4-fluorophenylamino)-6-((5-methyl-1-(2-morpholinoethyl)-1H-imidazol-4-yl)methylamino)quinoline-3-carbonitrile 368899 N-(4-(3-chloro-4-fluorophenylamino)-3-cyanoquinolin-6-yl)benzenesulfonamide 368900 4-(3-chloro-4-fluorophenylamino)-6-(1-(pyridin-2-yl)ethylamino)quinoline-3-carbonitrile 368907 6-(3-cyanobenzylamino)-4-(3-chloro-4-fluorophenylamino)quinoline-3-carbonitrile 368908 6-(3-aminobenzylamino)-4-(3-chloro-4-fluorophenylamino)quinoline-3-carbonitrile 368909 6-((1H-imidazol-4-yl)methylamino)-4-(3-chloro-4-fluorophenylamino)-7-(3-morpholinopropoxy)quinoline-3-carbonitrile 368910 6-((1H-imidazol-4-yl)methylamino)-4-(3-chloro-4-fluorophenylamino)-2-methylquinoline-3-carbonitrile 368917 4-((4-(3-chloro-4-fluorophenylamino)-3-cyanoquinolin-6-ylamino)methyl)benzenesulfonamide 368925 4-(3-chloro-4-fluorophenylamino)-6-(furan-2-ylmethylamino)quinoline-3-carbonitrile 368926 4-(3-chloro-4-fluorophenylamino)-6-(thiazol-2-ylmethylamino)quinoline-3-carbonitrile 368929 4-(ethylthio)-6-phenyl-1,3,5-triazin-2-amine 368930 4-(3-(6-methoxypyridin-3-yl)phenyl)-6-(methylthio)-1,3,5-triazin-2-amine 368931 4-(3-(1H-indol-5-yl)phenyl)-6-(methylthio)-1,3,5-triazin-2-amine 368934 6-((1H-pyrazol-3-yl)methylamino)-4-(3-chloro-4-fluorophenylamino)quinoline-3-carbonitrile 368935 6-((1H-imidazol-4-yl)methylamino)-4-(3-chloro-4-fluorophenylamino)quinoline-3-carbonitrile 368938 2-amino-4-(4-fluorophenyl)-6-phenylnicotinonitrile 368939 2-amino-4-(2-chlorophenyl)-6-phenylnicotinonitrile 368940 2-amino-6-cyclopropyl-4-(4-fluorophenyl)nicotinonitrile 368945 2-amino-6-phenyl-4-p-tolylnicotinonitrile 368946 SID24801556 368947 2-amino-4-(4-chlorophenyl)-6-phenylnicotinonitrile 368949 4-(3-chloro-4-fluoro-phenylamino)-6-[(1-oxy-pyridin-2-ylmethyl)-amino]-quinoline-3-carbonitrile 368952 2-amino-4-(3,4-dichlorophenyl)-6-(pyridin-3-yl)nicotinonitrile 368953 2-amino-4-(3-ethoxy-4-hydroxyphenyl)-6-(4-hydroxyphenyl)nicotinonitrile 368954 2-amino-6-(2-chlorophenyl)-4-(4-chlorophenyl)nicotinonitrile 368958 4-(3-chloro-4-fluorophenylamino)-6-((tetrahydrofuran-2-yl)methylamino)quinoline-3-carbonitrile 368961 SID26667329 368962 SID24267755 368963 N-(4-fluorobenzyl)-4-(thiophen-2-yl)-6-(trifluoromethyl)pyrimidin-2-amine 368969 4-(3-chloro-4-fluorophenylamino)-6-(pyridin-2-ylmethylamino)-1,7-naphthyridine-3-carbonitrile 368972 4-(3-chloro-4-fluorophenylamino)-6-(pyridin-2-ylmethylamino)quinoline-3-carbonitrile 368973 SID24267445 368974 SID24267413 368977 4-(3-chloro-4-fluorophenylamino)-6-(pyrrolidin-2-ylmethylamino)quinoline-3-carbonitrile 368982 4-[(3-chloro-4-fluorophenyl)amino]-6-[(2-morpholin-4-ylethyl)amino]quinoline-3-carbonitrile 368984 (S)-4-(3-chloro-4-fluorophenylamino)-6-((1-ethylpyrrolidin-2-yl)methylamino)quinoline-3-carbonitrile 368991 (R)-4-(3-chloro-4-fluorophenylamino)-6-((1-ethylpyrrolidin-2-yl)methylamino)quinoline-3-carbonitrile 368999 4-(3-chloro-4-fluorophenylamino)-6-((5-methyl-1H-imidazol-4-yl)methylamino)quinoline-3-carbonitrile 369000 4-(3-chloro-4-fluorophenylamino)-6-((1,5-dimethyl-1H-imidazol-4-yl)methylamino)quinoline-3-carbonitrile 369011 6-chloro-5-(2-fluorophenylamino)-1H-indazole-4,7-dione 369017 6-chloro-5-(3-fluorophenylamino)-1H-indazole-4,7-dione 369023 6-chloro-5-(2,4-difluorophenylamino)-1H-indazole-4,7-dione 369024 6-chloro-5-(4-ethoxyphenylamino)-1H-indazole-4,7-dione 369025 6-chloro-5-(4-(trifluoromethyl)phenylamino)-1H-indazole-4,7-dione 369032 5-(3-bromophenylamino)-6-chloro-1H-indazole-4,7-dione 369034 6-chloro-5-(3,4-dichlorophenylthio)-1H-indazole-4,7-dione 369043 2-thioxo-(1,3)ditholo[4,5-beta][1,4-dithine-5,6-dicarboxylic acid dimethyl ester 369112 1-cyclohexylmethyl-5-(2,4-difluoro-phenylamino)-1,3-dihydro-benzoimidazol-2-one 369131 5-(5,6-dimethoxy-1H-benzo[d]imidazol-1-yl)-3-(2-(trifluoromethyl)benzyloxy)thiophene-2-carbonitrile 369137 3-(2-(trifluoromethyl)benzyloxy)-5-(6-methoxy-5-(2-morpholinoethoxy)-1H-benzo[d]imidazol-1-yl)thiophene-2-carbonitrile 369144 3-(2-(trifluoromethyl)benzyloxy)-5-(5-(3-hydroxypropoxy)-6-methoxy-1H-benzo[d]imidazol-1-yl)thiophene-2-carbonitrile 369145 5-(5,6-dimethoxy-1H-benzo[d]imidazol-1-yl)-3-((R)-1-(2-(trifluoromethyl)phenyl)ethoxy)thiophene-2-carbonitrile 369152 3-(2-(methylsulfonyl)benzyloxy)-5-(5,6-dimethoxy-1H-benzo[d]imidazol-1-yl)thiophene-2-carbonitrile 369153 5-(5,6-dimethoxy-1H-benzo[d]imidazol-1-yl)-3-(2-morpholinoethoxy)thiophene-2-carbonitrile 369161 5-(5,6-dimethoxy-1H-benzo[d]imidazol-1-yl)-3-hydroxythiophene-2-carbonitrile 369162 3-(cyclopropylmethoxy)-5-(5,6-dimethoxy-1H-benzo[d]imidazol-1-yl)thiophene-2-carbonitrile 369163 5-(1H-benzo[d]imidazol-1-yl)-3-(benzyloxy)thiophene-2-carbonitrile 369170 5-(5,6-dimethoxy-1H-benzo[d]imidazol-1-yl)-3-(2-(piperidin-1-yl)ethoxy)thiophene-2-carbonitrile 369171 4-((2-cyano-5-(5,6-dimethoxy-1H-benzo[d]imidazol-1-yl)thiophen-3-yloxy)methyl)benzamide 369180 3-((R)-1-(2-chlorophenyl)ethoxy)-5-(5,6-dimethoxy-1H-benzo[d]imidazol-1-yl)thiophene-2-carbonitrile 369230 5-(5,6-dimethoxy-1H-benzo[d]imidazol-1-yl)-3-(4-(methylsulfonyl)benzyloxy)thiophene-2-carboxamide 369231 3-(4-(methylsulfonyl)benzyloxy)-5-(5,6-dimethoxy-1H-benzo[d]imidazol-1-yl)thiophene-2-carbonitrile 369238 5-(5,6-dimethoxy-1H-benzo[d]imidazol-1-yl)-3-((tetrahydrofuran-2-yl)methoxy)thiophene-2-carboxamide 369239 5-(5,6-dimethoxy-1H-benzo[d]imidazol-1-yl)-3-((tetrahydrofuran-2-yl)methoxy)thiophene-2-carbonitrile 369247 (R)-3-(1-(2-chlorophenyl)ethoxy)-5-(5,6-dimethoxy-1H-benzo[d]imidazol-1-yl)thiophene-2-carboxamide 369248 3-(benzyloxy)-5-(5,6-dimethoxy-1H-benzo[d]imidazol-1-yl)thiophene-2-carboxylic acid 369415 3-{2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-1H-benzo[4,5]thieno[3,2-d]pyrimidine-2,4-dione 369435 3-(2-(4-(5-chloro-2-methoxyphenyl)piperazin-1-yl)ethyl)-1H-pyrimido[5,4-b]indole-2,4(3H,5H)-dione 369440 3-{2-[4-(5-chloro-2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-1H-benzo[4,5]thieno[3,2-d]pyrimidine-2,4-dione 369449 3-{2-[4-(3,4-dichloro-phenyl)-piperazin-1-yl]-ethyl}-1H-benzo[4,5]thieno[3,2-d]pyrimidine-2,4-dione 369450 3-(2-(4-(3,4-dichlorophenyl)piperazin-1-yl)ethyl)-1,5-dimethyl-1H-pyrimido[5,4-b]indole-2,4(3H,5H)-dione 369454 3-(2-(4-(5-chloro-2-methoxyphenyl)piperazin-1-yl)ethyl)-2-methyl-3H-pyrimido[5,4-b]indol-4(5H)-one 369455 3-(2-(4-(3,4-dichlorophenyl)piperazin-1-yl)ethyl)-2-methyl-3H-pyrimido[5,4-b]indol-4(5H)-one 369461 3-{2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-2-methyl[1]benzothieno[3,2-d]pyrimidin-4(3H)-one 369465 3-{2-[4-(5-chloro-2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-2-methyl-3H-benzo[4,5]thieno[3,2-d]pyrimidin-4-one 369555 2-(4-(4-chlorobenzyl)-7-fluoro-5-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid 369755 [2-(hydroxymethyl)-4-(methylethylidene)-5-oxo-2-2,3-dihydrofuryl]methyl 4-[2-(4-ethynylphenyl)ethynyl]benzoate 369756 [2-(hydroxymethyl)-4-(methylethylidene)-5-oxo-2-2,3-dihydrofuryl]methyl 4-(2-{4-[2-(4-ethynylphenyl)ethynyl]phenyl}-ethynyl)benzoate 369762 (2-(hydroxymethyl)-5-oxo-4-(propan-2-ylidene)-tetrahydrofuran-2-yl)methyl 4-(2-(4-(2-(4-methoxyphenyl)ethynyl)phenyl)ethynyl)benzoate 369763 methyl 2-{4-[2-(4-{2-[4-({[2-(hydroxymethyl)-4-(methylethylidene)-5-oxo-2-2,3-dihydrofuryl]methyl}oxycarbonyl)phenyl]-ethynyl}phenyl)ethynyl]phenoxy}acetate 369764 methyl 2-[4-(2-{4-[2-(4-{2-[4-({[2-(hydroxymethyl)-4-(methylethylidene)-5-oxo-2-2,3-dihydrofuryl]methyl}oxycarbonyl)-phenyl]ethynyl}phenyl)ethynyl]phenyl} ethynyl)phenoxy]acetate 369765 methyl 16-{4-[2-(4-{2-[4-({[2-(Hydroxymethyl)-4-(methylethylidene)-5-oxo-2-2,3dihydrofuryl]methyl}oxycarbonyl)phenyl]ethynyl}phenyl)ethynyl]phenoxy}hexadecanoate 369766 tert-butyl 2-({[(tert-Butyl)oxycarbonyl]methyl}{2-[2-(2-{4-[2-(4-{2-[4-({[2-(hydroxymethyl)-4-(methylethylidene)-5-oxo(2-2,3-dihydrofuryl)]methyl}oxycarbonyl)phenyl]ethynyl}phenyl)ethynyl]phenoxy}ethoxy)ethoxy]ethyl}amino)acetate 369767 2-(N-(carboxymethyl){2-[2-(2-{4-[2-(4-{2-[4-({[2-(hydroxymethyl)-4-(methyl ethylidene)-5-oxo(2-2,3-dihydrofuryl)]methyl}-oxycarbonyl)phenyl]ethynyl}phenyl)ethynyl]phenoxy}ethoxy)-ethoxy]ethoxy}carbonylamino)acetic acid 369775 [2-(hydroxymethyl)-4-(methylethylidene)-5-oxo-2-2,3-dihydrofuryl]methyl decanoate 370024 4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-N-((pyridin-3-yl)-methyl)-1H-pyrrole-2-carboxamide 370026 N-((S)-(methylcarbamoyl(phenyl)methyl)-4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-1H-pyrrole-2-carboxamide 370032 4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-N-((pyridin-4-yl)-methyl)-1H-pyrrole-2-carboxamide 370034 4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-N-(2,3-dihydro-2-hydroxy-1H-inden-1-yl)-1H-pyrrole-2-carboxamide 370035 4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-N-(1-(4-fluorophenyl)-2-hydroxyethyl)-1H-pyrrole-2-carboxamide 370038 4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-N-((pyridin-4-yl)-methyl)-1H-pyrrole-2-carboxamide 370039 N-(3,4-difluorobenzyl)-4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-1H-pyrrole-2-carboxamide 370040 4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-N-(1-(4-chlorophenyl)-2-hydroxyethyl)-1H-pyrrole-2-carboxamide 370043 N-(4-methoxybenzyl)-4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-1H-pyrrole-2-carboxamide 370044 4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-1H-pyrrol-2-yl)(3,4-dihydroisoquinolin-2-(1H)-yl)methane 370046 4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-N-(1-(4-(trifluoro-methyl)phenyl)-2-hydroxy-ethyl)-1H-pyrrole-2-carboxamide 370049 4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-N-(1-(2-fluorophenyl)-2-hydroxyethyl)-1H-pyrrole-2-carboxamide 370055 4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-N-(2-(pyridin-3-yl)-ethyl)-1H-pyrrole-2-carboxamide 370057 4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-N-(1-(3-fluorophenyl)-2-hydroxyethyl)-1H-pyrrole-2-carboxamide 370062 N-(benzyloxy)-4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-1Hpyrrole-2-carboxamide 370065 4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-N-(1-(3,4-difluorophenyl)-2-hydroxyethyl)-1H-pyrrole-2-carboxamide 370067 N,N-dimethyl-4-(4-phenyl-1H-pyrazol-5-yl)-1H-pyrrole-2-carboxamide 370068 4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-N-((R)-1-phenylethyl)-1H-pyrrole-2-carboxamide 370069 4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-N-(1-(3,5-dichlorophenyl)-2-hydroxyethyl)-1H-pyrrole-2-carboxamide 370070 N-(1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl)-4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-1H-pyrrole-2-carboxamide 370074 4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-N-ethyl-N-methyl-1H-pyrrole-2-carboxamide 370076 N-((S)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl)-4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-1H-pyrrole-2-carboxamide 370077 N-((R)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl)-4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-1H-pyrrole-2-carboxamide 370082 4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-1H-pyrrol-2-yl)(pyrrolidin-1-yl)methanone 370083 4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-1H-pyrrol-2-yl)(morpholino)methanone 370085 4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-N-((S)-1-phenylethyl)-1H-pyrrole-2-carboxamide 370089 4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-N-((tetrahydrofuran-2-yl)methyl)-1H-pyrrole-2-carboxamide 370099 4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-N-((S)-2-hydroxy-1-phenylethyl)-1H-pyrrole-2-carboxamide 370113 4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-N-phenyl-1H-pyrrole-2-carboxamide 370129 N-benzyl-4-(4-(3-chlorophenyl)-1H-pyrazol-3-yl)-1H-pyrrole-2-carboxamide 370131 N-((S)-carbamoyl(phenyl)methyl)-4-(4-(3-chlorophenyl)-1Hpyrazol-3-yl)-1H-pyrrole-2-carboxamide 370139 1-(6-thiophen-2-yl-pyridazin-3-yl)-piperidine-4-carboxylic acid [1-(4-methyl-benzyl)-pyrrolidin-3-ylmethyl]-amide 370214 3-(4-fluorophenyl)-4-(pyridin-4-yl)quinolin-2(1H)-one 370216 3-(4-fluorophenyl)-5-isopropyl-4-(pyridin-4-yl)isoxazole 370225 5-(4-fluorophenyl)-3-isopropyl-4-(pyridin-4-yl)isoxazole 370240 2-(4-benzyl-5-(2-(piperidin-1-yl)ethyl)-4H-1,2,4-triazol-3-ylthio)-N-(2,4-dimethylphenyl)acetamide 370241 2-(4-oxo-3-(3-(piperidin-1-yl)propyl)-3,4-dihydroquinazolin-2-ylthio)-N-phenethylacetamide 370248 1-((1-(4-fluorobenzyl)-1H-tetrazol-5-yl)(2-fluorophenyl)methyl)-4-cyclohexylpiperazine 370249 1-(3-diethylamino-propylamino)-3-methyl-2-(2-methyl-allyl)-benzo[4,5]imidazo[1,2-a]pyridine-4-carbonitrile 370257 N-(1-benzylpiperidin-4-yl)-2-(5-methyl-4-p-tolyl-4H-1,2,4-triazol-3-ylthio)acetamide 370258 N-(2-methyl-4-((4-methylpiperazin-1-yl)methyl)phenyl)-2-(5-methyl-4-phenyl-4H-1,2,4-triazol-3-ylthio)acetamide 370276 (2S,2'S,5'S)-1-methyl-2-(2-cyclohexyl-2-phenyl-1,3-oxathiolan-5-yl)pirrolidine 370286 (2R,2'R,5'R)-1-methyl-2-(2-cyclohexyl-2-phenyl-1,3-oxathiolan-5-yl)pirrolidine 370289 SID11111827 370307 (S)-2-((S)-2,2-diphenyl-[1,3]oxathiolan-5-yl)-1,1-dimethyl-pyrrolidinium iodide 370327 (R)-2-((R)-2,2-diphenyl-[1,3]oxathiolan-5-yl)-1,1-dimethyl-pyrrolidinium iodide 370335 (S)-2-((2R,5S)-2-cyclohexyl-2-phenyl-[1,3]oxathiolan-5-yl)-1,1-dimethyl-pyrrolidinium iodide 370355 (R)-2-((2S,5R)-2-cyclohexyl-2-phenyl-[1,3]oxathiolan-5-yl)-1,1-dimethyl-pyrrolidinium iodide 370371 (S)-2-((2S,5S)-2-cyclohexyl-2-phenyl-[1,3]oxathiolan-5-yl)-1,1-dimethyl-pyrrolidinium iodide 370380 (2S,5'S)-1-methyl 2-(2,2-diphenyl-1,3-oxathiolan-5-yl)pirrolidine 370382 (R)-2-((2R,5R)-2-cyclohexyl-2-phenyl-[1,3]oxathiolan-5-yl)-1,1-dimethyl-pyrrolidinium iodide 370401 (2R,5'R)-1-methyl2-(2,2-diphenyl-1,3-oxathiolan-5-yl)pirrolidine 370409 (2S,2'R,5'S)-1-methyl-2-(2-cyclohexyl-2-phenyl-1,3-oxathiolan-5-yl)pirrolidine 370418 (2R,2'S,5'R)-1-methyl-2-(2-cyclohexyl-2-phenyl-1,3-oxathiolan-5-yl)pirrolidine 370422 H-Tyr-c[D-Cys-Gly-Phe-D-Cys]NH2 370425 (+/-)-7-methylthio-1,3,4,10b-tetrahydropyrazino[2,1-a]isoindol-6(2H)-one 370436 H-Tyr-c[D-Allylgly-Gly-Phe-L-Allylgly]NH2 370441 H-Tyr-c[D-Allylgly-Gly-Phe-L-Allylgly]NH2 370453 H-Tyr-c[D-Cys-Gly-Phe-L-Cys]NH2 370466 (+/-)-7-hydroxy-1,3,4,10b-tetrahydropyrazino[2,1-a]isoindol-6(2H)-one 370486 H-Tyr-c[D-Allylgly-Gly-Phe-D-Allylgly]NH2 370493 H-Tyr-c[D-Allylgly-Gly-Phe-D-Allylgly]NH2 370496 (+/-)-7-isopropoxy-1,3,4,10b-tetrahydropyrazino[2,1-a]isoindol-6(2H)-one 370503 H-Tyr-c[D-Allylgly-Gly-Phe-D-Allylgly]NH2 370505 1,3,4,10b-tetrahydropyrazino[2,1-a]isoindol-6(2H)-one 370506 (+/-)-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino[2,1-a]isoindol-6(2H)-one 370507 (+/-)-7-methoxy-1,3,4,10b-tetrahydropyrazino[2,1-a]isoindol-6(2H)-one 370508 (+/-)-1,3,4,10b-tetrahydro-7-trifluoromethoxypyrazino[2,1-a]-isoindol-6(2H)-one 370514 H-Tyr-c[D-Allylgly-Gly-Phe-L-Allylgly]NH2 370517 (+/-)-7-fluoro-1,3,4,10b-tetrahydropyrazino[2,1-a]isoindol-6(2H)-one 370519 (+/-)-7-chloro-1,3,4,10b-tetrahydropyrazino[2,1-a]isoindol-6(2H)-one 370520 (+/-)-7-nitrile-1,3,4,10b-tetrahydropyrazino[2,1-a]isoindol-6(2H)-one 370523 N6-methoxy-2-[(4-methylphenyl)ethynyl]-5'-N-methylcarboxamidoadenosine 370528 (R)-9-methyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino-[2,1-a]isoindol-6(2H)-one 370529 (R)-9-ethyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino-[2,1-a]isoindol-6(2H)-one 370530 (R)-9-propyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino-[2,1-a]isoindol-6(2H)-one 370531 N6-methoxy-2-[(4-pentylphenyl)ethynyl]-5'-N-methylcarboxamidoadenosine 370533 (2S,3S,4R,5R)-3,4-dihydroxy-5-(6-(methoxyamino)-2-(phenylethynyl)-9H-purin-9-yl)-N-methyltetrahydrofuran-2-carboxamide 370536 (R)-9-butyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino-[2,1-a]isoindol-6(2H)-one 370537 (R)-9-isopropyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino-[2,1-a]isoindol-6(2H)-one 370538 (R)-9-ethenyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino-[2,1-a]isoindo l-6(2H)-one 370539 (2S,3S,4R,5R)-5-(2-((4-fluorophenyl)ethynyl)-6-(methoxyamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide 370543 (R)-9-ethynyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino-[2,1-a]isoindol-6(2H)-one 370544 (R)-9-cyclopropyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino[2,1-a]isoindol-6(2H)-one 370545 (R)-9-(1-methylcyclopropyl)-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino[2,1-a]isoindol-6(2H)-one 370549 (S)-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino[2,1-a]isoindol-6(2H)-one 370551 (2R,3R,4S,5R)-2-(6-amino-2-(phenylethynyl)-9H-purin-9-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol 370552 (2R,3S,4R)-2-hydroxymethyl-5-((S)-2-iodo-6-methoxyamino-9H-purin-3-yl)-tetrahydro-furan-3,4-diol 370553 (2S,3S,4R,5R)-5-(2-((4-acetylphenyl)ethynyl)-6-(methoxyamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide 370559 N6-methoxy-2-phenylethynyladenosine 370560 2-ethynyl-N6-methoxyadenosine 370561 (2S,3S,4R)-5-((R)-6-amino-2-phenylethynyl-9H-purin-3-yl)-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 370565 (10bR)-2-methyl-7-(trifluoromethyl)-1,3,4,10b-tetrahydropyrazino[2,1-a]isoindol-6(2H)-one 370566 (10bR)-3,3-dimethyl-7-(trifluoromethyl)-1,3,4,10b-tetrahydropyrazino[2,1-a]isoindol-6(2H)-one 370567 (3S,10bR)-3-methyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino[2,1-a]isoindol-6(2H)-one 370569 2-(hex-1-ynyl)-N6-methoxyadenosine 370571 (2S,3S,4R)-3,4-dihydroxy-5-((S)-2-iodo-6-methoxyamino-9H-purin-3-yl)-tetrahydro-furan-2-carboxylic acid ethylamide 370573 (3R,10bR)-3-methyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino[2,1-a]isoindol-6(2H)-one 370574 (4R,10bR)-4-methyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino[2,1-a]isoindol-6(2H)-one 370575 (4S,10bR)-4-methyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino[2,1-a]isoindol-6(2H)-one 370576 N6-methoxy-2-[2-(trimethylsilyl)ethynyl]adenosine 370577 2-(5-cyano-1-pent-1-ynyl)-N6-methoxyadenosine 370582 (1S,10bR)-1-methyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino[2,1-a]isoindol-6(2H)-one 370583 (1S,10bR)-1-ethyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino[2,1-a]isoindol-6(2H)-one 370584 2-(4-hydroxypent-1-yl)-N6-methoxyadenosine 370585 N6-methoxy-2-[2-(1-hydroxycyclohexyl)ethynyl]adenosine 370586 N6-methoxy-2-phenylethynyl-5'-N-ethylcarboxamidoadenosine 370591 ((R)-10-chloro-7-methoxy-1,3,4,10b-tetrahydropyrazino[2,1-a]isoindol-6(2 H)-one 370592 (2R,3S,4R,5R)-2-(hydroxymethyl)-5-(6-(methoxyamino)-2-(pyridin-2-ylethynyl)-9H-purin-9-yl)tetrahydrofuran-3,4-diol 370593 N6-methoxy-2-[(3-pyridinyl)ethynyl]-adenosine 370598 N6-methoxy-2-[(4-pyridinyl)ethynyl]adenosine 370599 N6-methoxy-2-[(4-methylphenyl)ethynyl]adenosine 370600 N6-methoxy-2-[(2-pyridinyl)ethynyl]-5'-N-ethylcarboxamidoadenosine 370606 (R)-7-chloro-10-methyl-1,3,4,10b-tetrahydropyrazino[2,1-a]-isoindol-6(2H)-one 370607 (R)-7-chloro-10-ethyl-1,3,4,10b-tetrahydropyrazino[2,1-a]-isoindol-6(2H)-one 370609 N6-methoxy-2-[(4-pentylphenyl)ethynyl]adenosine 370610 2-[(4-fluorophenyl)ethynyl]-N6-methoxyadenosine 370612 (R)-7-chloro-10-methoxy-1,3,4,10b-tetrahydropyrazino[2,1-a]isoindol-6(2H)-one 370613 (R)-10-chloro-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino-[2,1-a]isoindol-6(2H)-one 370614 (R)-7,8-dichloro-1,3,4,10b-tetrahydropyrazino[2,1-a]isoindol-6(2H)-one 370615 N6-methoxy-2-{[3-(trifluoromethyl)phenyl]ethynyl}adenosine 370616 2-{[4-(cyanomethyl)phenyl]ethynyl}-N6-methoxyadenosine 370617 N6-methoxy-2-(4-methylphenyl)ethynyl-5'-N-ethylcarboxamidoadenosine 370620 (R)-8-chloro-7-methoxy-1,3,4,10b-tetrahydropyrazino[2,1-a]-isoindol-6(2H)-one 370621 (R)-8-ethyl-7-methoxy-1,3,4,10b-tetrahydropyrazino[2,1-a]-isoindol-6(2H)-one 370622 2-[(4-acetylphenyl)ethynyl]-N6-methoxyadenosine 370623 2-[(4-carboxamidophenyl)ethynyl]-N6-methoxyadenosine 370624 N6-methoxy-2-[(4-pentylphenyl)ethynyl]-5'-N-ethylcarboxamidoadenosine 370626 (R)-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino[2,1-a]isoindol-6(2H)-one 370627 (R)-9-chloro-8-methoxy-1,3,4,10b-tetrahydropyrazino[2,1-a]-isoindol-6(2H)-one 370628 (R)-9-ethyl-8-methoxy-1,3,4,10b-tetrahydropyrazino[2,1-a]-isoindol-6(2H)-one 370629 (R)-7-chloro-9-methoxy-1,3,4,10b-tetrahydropyrazino[2,1-a]-isoindol-6(2H)-one 370630 N6-methoxy-2-[(4-methoxyphenyl)ethynyl]adenosine 370631 2-[(4-fuorophenyl)ethynyl]-N6-methoxy-5'-N-ethylcarboxamidoadenosine 370635 (R)-7-chloro-9-ethyl-1,3,4,10b-tetrahydropyrazino[2,1-a]-isoindol-6(2H)-one 370636 (R)-9-chloro-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino-[2,1-a]isoindol-6(2H)-one 370637 (R)-9-acetyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino-[2,1-a]isoindol-6(2H)-one 370638 (2S,3S,4R)-3,4-dihydroxy-5-((S)-2-iodo-6-methoxyamino-9H-purin-3-yl)-tetrahydro-furan-2-carboxylic acid methylamide 370639 (2S,3S,4R,5R)-3,4-dihydroxy-5-(6-(methoxyamino)-2-(pyridin-2-ylethynyl)-9H-purin-9-yl)-N-methyltetrahydrofuran-2-carboxamide 370640 2-[(4-acetylphenyl)ethynyl]-N6-methoxy-5'-N-ethylcarboxamidoadenosine 370644 (R)-9-hydroxymethyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino[2,1-a]isoindol-6(2H)-one 370645 (R)-9-methoxy-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino-[2,1-a]isoindol-6(2H)-one 370646 (R)-9-ethoxy-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino-[2,1-a]isoindol-6(2H)-one 370799 7-chloro-3-oxo-8-(pyridin-3-ylmethoxy)-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370800 7-chloro-3-oxo-8-(pyridin-2-ylmethoxy)-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370807 7-chloro-8-(2-imidazol-1-yl-ethoxy)-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370808 8-amino-7-chloro-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370817 7-chloro-8-methylamino-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370818 7-chloro-8-ethylamino-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370827 8-butylamino-7-chloro-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370828 7-chloro-8-(2-hydroxy-ethylamino)-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370847 7-chloro-8-isopropylamino-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370848 7-chloro-8-isobutylamino-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370869 7-chloro-3-oxo-8-[(pyridin-3-ylmethyl)-amino]-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370870 7-Chloro-3-oxo-8-[(pyridin-4-ylmethyl)-amino]-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0*5,10*]docosa-1(21),5(10),6,8,18(22),19-hexaene-19-carbonitrile 370875 8-benzylamino-7-chloro-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370876 7-chloro-8-[(1H-imidazol-4-ylmethyl)-amino]-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370884 7-Chloro-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0*5,10*]docosa-1(22),5,7,9,18,20-hexaen-3-one 370885 7-chloro-3-oxo-8-[(thiazol-5-ylmethyl)-amino]-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370886 7-chloro-8-[(oxazol-5-ylmethyl)-amino]-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370892 7-chloro-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0*5,10*]docosa-1(22),5,7,9,18,20-hexaene-19-carbonitrile 370893 7-chloro-3-oxo-11,16-dioxa-2,4,19,21-tetraaza-tricyclo[15.3.1.0*5,10*]henicosa-1(21),5,7,9,17,19-hexaene-18-carbonitrile 370894 7-chloro-3-oxo-8-[(thiophen-3-ylmethyl)-amino]-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370895 7-chloro-8-[(3-methyl-3H-imidazol-4-ylmethyl)-amino]-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370907 7-chloro-3-oxo-11,18-dioxa-2,4,21,23-tetraaza-tricyclo[17.3.1.0*5,10*]tricosa-1(23),5,7,9,19,21-hexaene-2-carbonitrile 370908 7-chloro-8-hydroxy-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.05,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370909 N-(7-chloro-19-cyano-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaen-8-yl)-acetamide 370910 N-(7-chloro-19-cyano-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaen-8-yl)-2-dimethylamino-acetamide 370916 7-chloro-8-(3-hydroxy-propoxy)-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.05,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370917 8-(3-amino-propoxy)-7-chloro-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrie 370918 N-(7-chloro-19-cyano-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaen-8-yl)-3-cyclopentylamino-propionamide 370919 N-(7-chloro-19-cyano-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaen-8-yl)-methanesulfonamide 370922 7-chloro-8-(2,3-dihydroxy-propoxy)-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370923 7-chloro-8-(2-hydroxy-ethoxy)-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370924 7-chloro-8-dimethylamino-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370925 7-chloro-8-diethylamino-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370928 7-chloro-8-(2-methoxy-ethoxy)-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370929 7-chloro-8-[2-(2-methoxy-ethoxy)-ethoxy]-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370930 8-[bis-(2-hydroxy-ethyl)-amino]-7-chloro-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370931 7-chloro-8-cyclohexylamino-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370935 7-chloro-8-(2-dimethylamino-ethoxy)-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370936 7-chloro-8-(3-methyl-butoxy)-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370937 7-chloro-8-(3-hydroxy-prop-1-ynyl)-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370938 7-chloro-8-(3-hydroxy-but-1-ynyl)-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370945 7-chloro-8-ethoxy-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370946 7-chloro-8-(3-hydroxy-3-methyl-but-1-ynyl)-3-oxo-11,17-dioxa-2,4,20,22traaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370947 7-chloro-8-(3-diethylamino-prop-1-ynyl)-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370953 7-chloro-8-isopropoxy-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370954 7-chloro-3-oxo-8-(pyridin-4-ylmethoxy)-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370955 7-chloro-8-(3-hydroxy-propyl)-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 370956 7-chloro-8-(2,3-dihydroxy-propyl)-3-oxo-11,17-dioxa-2,4,20,22-tetraaza-tricyclo[16.3.1.0 5,10]docosa-1(22),5(10),6,8,18,20-hexaene-19-carbonitrile 371129 1-(4-(3-amino-1H-indazol-4-yl)phenyl)-3-(3-chlorophenyl)urea 371130 1-(4-(3-amino-1H-indazol-4-yl)phenyl)-3-(3-bromophenyl)urea 371138 1-(4-(3-amino-1H-indazol-4-yl)phenyl)-3-(3-(trifluoromethyl)phenyl)urea 371139 1-(4-(3-amino-1H-indazol-4-yl)phenyl)-3-(3-hydroxyphenyl)urea 371147 1-(4-(3-amino-1H-indazol-4-yl)phenyl)-3-(2-fluoro-5-methylphenyl)urea 371148 1-(4-(3-amino-1H-indazol-4-yl)phenyl)-3-(4-fluoro-3-methylphenyl)urea 371156 1-(4-(3-amino-1H-indazol-4-yl)phenyl)-3-(3-fluoro-4-methylphenyl)urea 371157 1-(4-(3-amino-1H-indazol-4-yl)phenyl)-3-(2-fluoro-5-(trifluoromethyl)phenyl)urea 371169 1-(4-(3-amino-1-(2-methoxyethoxy)-1H-indazol-4-yl)phenyl)-3-(3-chlorophenyl)urea 371180 1-(4-(3-amino-7-methyl-1H-indazol-4-yl)phenyl)-3-m-tolylurea 371181 1-(4-(3-amino-7-methoxy-1H-indazol-4-yl)phenyl)-3-m-tolylurea 371185 1-(4-(3-amino-7-(2-(pyrrolidin-1-yl)ethoxy)-1H-indazol-4-yl)phenyl)-3-m-tolylurea 371186 1-(4-(3-amino-7-(2-morpholinoethoxy)-1H-indazol-4-yl)phenyl)-3-m-tolylurea 371191 N-[4-(3-amino-1-methyl-1H-indazol-4-yl)-phenyl]-N'-(3-methylphenyl)urea 371192 N-{4-[3-amino-1-(2-hydroxyethyl)-1H-indazol-4-yl]phenyl}-N'-(3-methylphenyl)urea 371198 4-(4-aminophenyl)-1H-indazol-3-amine 371200 1-(4-(3-amino-7-fluoro-1H-indazol-4-yl)phenyl)-3-m-tolylurea 371201 1-(4-(3-amino-7-bromo-1H-indazol-4-yl)phenyl)-3-m-tolylurea 371210 1-(4-(3-amino-7-(2-(2-oxopyrrolidin-1-yl)ethoxy)-1H-indazol-4-yl)phenyl)-3-m-tolylurea 371211 1-(4-(3-amino-7-(2-methoxyethoxy)-1H-indazol-4-yl)phenyl)-3-m-tolylurea 371216 N-(4-(3-amino-1H-indazol-4-yl)phenyl)benzenesulfonamide 371217 1-(4-(3-amino-1H-indazol-4-yl)phenyl)-3-phenylurea 371218 N-{4-[3-amino-1-(2-morpholin-4-yl-ethyl)-1H-indazol-4-yl]-phenyl}-N'-(3-methylphenyl)urea 371219 N-{4-[3-amino-1-(2-methoxyethyl)-1H-indazol-4-yl]phenyl}-N'-(2-fluoro-5-methylphenyl)urea 371224 1-(4-(3-amino-1H-indazol-4-yl)phenyl)-3-m-tolylurea 371225 1-(4-(3-amino-1H-indazol-4-yl)phenyl)-3-(thiophen-3-yl)urea 371226 1-(4-(3-amino-7-(2-(dimethylamino)ethoxy)-1H-indazol-4-yl)phenyl)-3-m-tolylurea 371227 1-(4-(3-amino-7-(2-(diethylamino)ethoxy)-1H-indazol-4-yl)phenyl)-3-m-tolylurea 371234 1-(4-(3-amino-1H-indazol-4-yl)phenyl)-3-cyclopentylurea 371235 N-(4-(3-amino-1H-indazol-4-yl)phenyl)cyclohexanecarboxamide 371236 N-{4-[3-amino-7-(4-morpholinylmethyl)-1H-indazol-4-yl]phenyl}-N'-(3-methylphenyl)urea 371237 1-(4-(3-amino-7-((4-methylpiperazin-1-yl)methyl)-1H-indazol-4-yl)phenyl)-3-m-tolylurea 371242 1-(4-(3-amino-1H-indazol-4-yl)phenyl)-3-(2-fluorophenyl)urea 371243 N-[4-(3-amino-1H-indazol-4-yl)phenyl]-N'-(3-fluorophenyl)-urea 371251 1-(4-(3-amino-1H-indazol-4-yl)phenyl)-3-(4-fluorophenyl)urea 371252 1-(4-(3-amino-1H-indazol-4-yl)phenyl)-3-o-tolylurea 371259 1-(4-(3-amino-1H-indazol-4-yl)phenyl)-3-p-tolylurea 371260 1-(4-(3-amino-1H-indazol-4-yl)phenyl)-3-(3-ethylphenyl)urea 371268 1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(2-oxo-2-phenyl-ethyl)-pyrrolidinium 371273 1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-phenylcarbamoylmethyl-pyrrolidinium 371274 1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(3-phenyl-oxiranylmethyl)-pyrrolidinium 371278 1-(4-(3-amino-1-(2-methoxyethoxy)-1H-indazol-4-yl)phenyl)-3-(2-fluoro-5-methylphenyl)urea 371280 1-cyanomethyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(2-phenoxy-ethyl)-pyrrolidinium 371281 1-methoxyethyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(2-phenoxy-ethyl)-pyrrolidinium 371285 1-(4-(3-amino-1-(2-(diethylamino)ethoxy)-1H-indazol-4-yl)phenyl)-3-(2-fluoro-5-methylphenyl)urea 371287 1-methyl-3-(R)-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(2-phenoxy-ethyl)-pyrrolidinium 371288 1-methyl-3-(S)-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(2-phenoxy-ethyl)-pyrrolidinium 371295 1-methyl-3-(R)-[4,4-Bis-(4-fluoro-phenyl)-2-oxo-imidazolidin-1-yl]-1-phenethyl-pyrrolidinium 371296 1-methyl-3-(R)-3-[4,4-bis-(4-fluoro-phenyl)-2-oxo-imidazolidin-1-yl]-1-(2-oxo-2-phenyl-ethyl)-pyrrolidinium 371302 1-methyl-3-(R)-3-[4,4-bis-(4-fluoro-phenyl)-2-oxo-imidazolidin-1-yl]-1-[2-(3-fluoro-phenyl)-2-oxo-ethyl]-pyrrolidinium 371303 1-methyl-3-(R)-3-[4,4-bis-(4-fluoro-phenyl)-2-oxo-imidazolidin-1-yl]-1-(2-oxo-2-thiophen-3-ylethyl)-pyrrolidinium 371307 N-{1-methyl-4-[4-(3-methylphenylureido)phenyl]-1H-indazol-3-yl}acetamide 371309 1-methyl-3-(R)-3-[4,4-bis-(4-fluoro-phenyl)-2-oxo-imidazolidin-1-yl]-1-(2-oxo-2-pyridin-3-ylethyl)-pyrrolidinium 371310 1-methyl-3-(R)-3-[4,4-bis-(4-fluoro-phenyl)-2-oxo-imidazolidin-1-yl]-1-(2-oxo-2-pyridin-2-ylethyl)-pyrrolidinium 371312 N-[4-(3-dimethylamino-1-methyl-1H-indazol-4-yl)phenyl]-N'-(3-methylpheny)urea 371313 N-[4-(1-methyl-1H-indazol-4-yl)-phenyl]-N'-(3-methylphenyl)urea 371315 1-benzyl-1-methyl-4-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-piperidinium 371319 N-[4-(1H-indazol-4-yl)-phenyl]-N'-(3-methylphenyl)urea 371321 1,1-dimethyl-4-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-piperidinium 371322 8-benzyl-8-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-8-azonia-bicyclo[3.2.1]octane 371330 8,8-dimethyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-8-azonia-bicyclo[3.2.1]octane 371331 1-benzyl-1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-pyrrolidinium 371338 1,1-dimethyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-pyrrolidinium 371339 1-methyl-3-(R)-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-benzyl-pyrrolidinium 371346 1-methyl-3-(S)-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-benzyl pyrrolidinium 371347 benzyl-dimethyl-[2-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-ethyl]-ammonium 371353 trimethyl-[2-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-ethyl]-ammonium 371360 trimethyl-[3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-propyl]-ammonium 371361 1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-phenethyl-pyrrolidinium bromide 371369 1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(3-phenyl-propyl)-pyrrolidinium 371370 1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(2-phenoxy-ethyl)-pyrrolidinium 371378 1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(2-benzyloxy-ethyl)-pyrrolidinium 371379 1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(3-phenoxy-propyl)-pyrrolidinium 371387 3-(1-(3-fluorobenzyl)-piperidin-4-yl)-5,5-di-(2-thienyl)-imidazolidin-2-one 371394 3-(1-phenylethyl-piperidin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371395 3-(1-phenylpropyl-piperidin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371400 3-(1-phenoxyethyl-piperidin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371401 3-(1-(3-pyridylmethyl)-piperidin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371404 3-(1-(2-thienylmethyl)-piperidin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371405 3-(1-(4-imidazolylmethyl)-piperidin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371409 3-(1-(2-chlorobenzyl)-piperidin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371410 3-(1-(3-chlorobenzyl)-piperidin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371413 3-(1-benzylpiperidin-4-yl)-5,5-diphenyl-imidazolidin-2,4-dione 371414 3-(1-benzylpiperidin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371427 3-(1-(4-chlorobenzyl)-piperidin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371432 1-(1-benzyl-piperidin-4-yl)-3-methyl-4,4-diphenyl-imidazolidin-2-one 371433 3-(1-benzyl-piperidin-4-yl)-5,5-diphenyl-oxazolidin-2-one 371434 3-(1-(2-methoxybenzyl)-piperidin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371435 3-(1-(3-methoxybenzyl)-piperidin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371439 1-(1-benzyl-piperidin-4-yl)-3-benzyl-4-phenyl-imidazolidin-2-one 371440 3-(1-benzyl-piperidin-3-yl)-5,5-diphenyl-imidazolidin-2-one 371441 3-(1-(4-methoxybenzyl)-piperidin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371442 3-(1-(3-hydroxybenzyl)-piperidin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371447 3-(1-benzyl-tropin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371448 3-(1-benzyl-azepin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371449 3-(1-(3-methylbenzyl)-piperidin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371450 3-(1-(3-aminobenzyl)-piperidin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371454 (R)-3-(1-benzyl-pyrrolidin-3-yl)-5,5-diphenyl-imidazolidin-2-one 371455 (S)-3-(1-benzyl-pyrrolidin-3-yl)-5,5-diphenyl-imidazolidin-2-one 371456 3-(1-(3-trifluoromethoxybenzyl)-piperidin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371457 3-(1-(3-cyanobenzyl)-piperidin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371460 3-(1-benzyl-piperidin-4-yl)-5,5-di-(4-fluorophenyl)-imidazolidin-2-one 371461 3-(1-benzyl-piperidin-4-yl)-5,5-di-(4-methoxyphenyl)-imidazolidin-2-one 371463 3-(1-(3-trifluoromethylbenzyl)-piperidin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371481 3-(1-benzyl-piperidin-4-yl)-5-phenyl-5-cyclohexyl-imidazolidin-2-one 371483 3-(1-(3-fluorobenzyl)-piperidin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371484 3-(1-(3-chlorobenzyl)-piperidin-4-yl)-5,5-di-(4-fluorophenyl)-imidazolidin-2-one 371488 3-(1-benzyl-piperidin-4-yl)-5,5-di-(2-thienyl)-imidazolidin-2-one 371489 3-(1-benzyl-piperidin-4-yl)-5,5-dibenzyl-imidazolidine-2,4-dione 371491 3-(1-(3-fluorobenzyl)-piperidin-4-yl)-5,5-di-(4-fluorophenyl)-imidazolidin-2-one 371497 3-(1-methyl-piperidin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371498 3-(1-(3-methylbenzyl)-piperidin-4-yl)-5-phenyl-5-cyclohexyl-imidazolidin-2-one 371499 3-(1-(3-chlorobenzyl)-piperidin-4-yl)-5-phenyl-5-cyclohexyl-imidazolidin-2-one 371504 3-(1-Phenyl-piperidin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371505 3-(1-cyclohexylmethyl-piperidin-4-yl)-5,5-diphenyl-imidazolidin-2-one 371515 3-(1-(3-methylbenzyl)-piperidin-4-yl)-5,5-di-(2-thienyl)-imidazolidin-2-one 371750 2-(3''-(4''-bromo-indolyl)ethyloxy)adenosine 371755 (2R,3R,4S,5R)-2-(6-amino-2-(2-(thiophen-2-yl)ethoxy)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 371756 (2R,3R,4S,5R)-2-(6-amino-2-(2-(thiophen-3-yl)ethoxy)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 371758 2-(3''(7''-bromo-indolyl)ethyloxy)adenosine 371765 (2R,3R,4S,5R)-2-(2-(2-(1H-indol-3-yl)ethoxy)-6-amino-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 371766 (2R,3R,4S,5R)-2-(2-(2-(1H-pyrrol-3-yl)ethoxy)-6-amino-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 371767 2-(3''-(5''-methoxy-2''-methylindolyl)ethyloxy)adenosine 371778 2-(2''-indolylethyloxy)adenosine 371780 2-(2''-(1''-(p-toluenesulfonyl)indolyl)ethyloxy)adenosine 371781 (2R,3R,4S,5R)-2-(6-amino-2-(2-(5-methoxy-1H-indol-3-yl)ethoxy)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 371782 (2R,3R,4S,5R)-2-(6-amino-2-(2-(5-hydroxy-1H-indol-3-yl)ethoxy)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 371788 (2R,3R,4S,5R)-2-(6-amino-2-(2-(5-fluoro-1H-indol-3-yl)ethoxy)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 371790 2-(3''-(benzoimidazole-1''-yl)ethyloxy)adenosine 371791 2-(3''-(benzotriazole-1''-yl)ethyloxy)adenosine 371795 (2R,3R,4S,5R)-2-(6-amino-2-(2-(5-chloro-1H-indol-3-yl)ethoxy)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 371804 (2R,3R,4S,5R)-2-(6-amino-2-(2-(5-bromo-1H-indol-3-yl)ethoxy)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 371806 (2S,3S,4R,5R)-5-(2-(2-(1H-indol-3-yl)ethoxy)-6-amino-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 371813 (2R,3R,4S,5R)-2-(6-amino-2-(2-(5-iodo-1H-indol-3-yl)ethoxy)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 371815 2-(3''-(5''-bromo-1''-(p-toluenesulfonyl)indolyl)ethyloxy)adenosine 371826 (2R,3R,4S,5R)-2-(6-amino-2-(2-(6-chloro-1H-indol-3-yl)ethoxy)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 371844 (2S,3S,4R,5R)-N-ethyl-5-(6-guanidino-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 371845 (2S,3S,4R,5R)-5-(6-amino-2-((S)-3-hydroxy-3-phenylprop-1-ynyl)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 371846 (2R,3R,4S,5R)-2-(6-amino-2-(2-(6-bromo-1H-indol-3-yl)ethoxy)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 371855 (2R,3R,4S,5R)-2-(6-amino-2-ethoxy-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 371856 (2R,3R,4S,5R)-2-(6-amino-2-(2-cyclohexylethoxy)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 371865 (2R,3R,4S,5R)-2-(6-amino-2-phenethoxy-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 371866 2-phenylpropoxyadenosine 371876 (2R,3R,4S,5R)-2-(6-amino-2-(4-phenylbutoxy)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 371877 (2R,3R,4S,5R)-2-(6-amino-2-((S)-3-phenylbutoxy)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 371888 (2R,3R,4S,5R)-2-(2-(2-fluorophenethoxy)-6-amino-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 371889 (2R,3R,4S,5R)-2-(2-(3-fluorophenethoxy)-6-amino-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 371900 (2R,3R,4S,5R)-2-(2-(4-fluorophenethoxy)-6-amino-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 371901 (2R,3R,4S,5R)-2-(6-amino-2-(2-(naphthalen-2-yl)ethoxy)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 371902 2-(3''-(1''-(p-toluenesulfonyl)indolyl)ethyloxy)adenosine 372037 cis-((+/-)-Methyl(1R,2S/1S,2R)-2-[(4-Hydroxy-4-phenylpiperidin-1-yl)methyl]-1-(4-methylphenyl)cyclopropanecarboxylate 372051 6-isopropyl-2-morpholin-4-yl-4H-thiopyran-4-one 372052 6-tert-Butyl-2-morpholin-4-yl-4H-thiopyran-4-one 372068 2-morpholin-4-yl-6-thianthren-1-yl-4H-thiopyran-4-one 372077 6-(4-cyanophenyl)-2-morpholin-4-yl-4H-thiopyran-4-one 372084 2-morpholin-4-yl-5,6,7,8-tetrahydrothiochromen-4-one 372091 6-(4-chlorophenyl)-2-morpholin-4-ylpyridin-4-ol 372124 N-[3'-(6-morpholin-4-yl-4-oxo-4H-thiopyran-2-yl)-biphenyl-3-yl]-acetamide 372130 6-(2-fluorophenyl)-2-(4-morpholin-4-yl)pyran-4-one 372159 4-morpholino-6-phenyl-2H-pyran-2-one 372160 6-(4-methoxyphenyl)-4-morpholino-2H-pyran-2-one 372161 6-(4-chlorophenyl)-4-morpholino-2H-pyran-2-one 372166 6-(4-tert-butylphenyl)-4-morpholino-2H-pyran-2-one 372176 2-morpholino-6-(thiophen-2-yl)-4H-pyran-4-one 372177 2-morpholino-6-(thiophen-3-yl)-4H-pyran-4-one 372178 2-(furan-2-yl)-6-morpholino-4H-pyran-4-one 372184 3-(6-morpholino-4-oxo-4H-pyran-2-yl)thiophene-2-carbaldehyde 372186 2-(1H-indol-5-yl)-6-morpholino-4H-pyran-4-one 372193 6-(4-benzo[b]thiophen-3-ylphenyl)-2-morpholin-4-yl-4H-thiopyran-4-one 372194 2-(benzo[b]thiophen-2-yl)-6-morpholino-4H-pyran-4-one 372195 2-(benzofuran-2-yl)-6-morpholino-4H-pyran-4-one 372202 2-morpholino-6-(naphthalen-1-yl)-4H-pyran-4-one 372203 2-morpholino-6-(naphthalen-2-yl)-4H-pyran-4-one 372204 2-(4-methylnaphthalen-1-yl)-6-morpholino-4H-pyran-4-one 372209 2-morpholino-6-styryl-4H-pyran-4-one 372210 2-morpholino-6-(2-(trifluoromethyl)phenyl)-4H-pyran-4-one 372211 2-(2-aminophenyl)-6-morpholino-4H-pyran-4-one 372212 4-(6-morpholino-4-oxo-4H-pyran-2-yl)-1-naphthaldehyde 372217 tert-butyl 4-(6-morpholino-4-oxo-4H-pyran-2-yl)phenylcarbamate 372218 benzyl 4-(6-morpholino-4-oxo-4H-pyran-2-yl)phenylcarbamate 372219 2-morpholino-6-(quinolin-8-yl)-4H-pyran-4-one 372224 3-(6-morpholino-4-oxo-4H-pyran-2-yl)benzonitrile 372225 4-(6-morpholino-4-oxo-4H-pyran-2-yl)benzonitrile 372226 2-morpholino-6-(3-(trifluoromethoxy)phenyl)-4H-pyran-4-one 372227 2-dibenzofuran-4-yl-6-morpholin-4-yl-pyran-4-one 372228 2-morpholino-6-(thianthren-1-yl)-4H-pyran-4-one 372233 2-morpholino-6-(4-(trifluoromethoxy)phenyl)-4H-pyran-4-one 372234 2-(2-(benzyloxy)phenyl)-6-morpholino-4H-pyran-4-one 372239 2-(3-(benzyloxy)phenyl)-6-morpholino-4H-pyran-4-one 372240 2-(4-(benzyloxy)phenyl)-6-morpholino-4H-pyran-4-one 372247 2-(3-acetylphenyl)-6-morpholino-4H-pyran-4-one 372249 3-(6-morpholino-4-oxo-4H-pyran-2-yl)benzaldehyde 372254 3-(6-morpholino-4-oxo-4H-pyran-2-yl)benzoic acid 372255 methyl 2-(6-morpholino-4-oxo-4H-pyran-2-yl)benzoate 372256 methyl 3-(6-morpholino-4-oxo-4H-pyran-2-yl)benzoate 372261 benzyl 4-(6-morpholino-4-oxo-4H-pyran-2-yl)benzoate 372267 2-biphenyl-4-yl-6-morpholin-4-yl-pyran-4-one 372272 methyl 3-amino-4-(6-morpholino-4-oxo-4H-pyran-2-yl)benzoate 372273 3-(6-morpholino-4-oxo-4H-pyran-2-yl)benzyl acetate 372281 methyl 3-(3-(6-morpholino-4-oxo-4H-pyran-2-yl)phenyl)acrylate 372288 2-(3-(6-morpholino-4-oxo-4H-pyran-2-yl)benzyl)isoindoline-1,3-dione 372289 2-(4-(6-morpholino-4-oxo-4H-pyran-2-yl)benzyl)isoindoline-1,3-dione 372354 benzyl-dimethyl-[3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-propyl]-ammonium 372609 (R)-N-(1-(4-(2,4-dimethoxybenzyl)-5-benzyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372619 (R)-N-(1-(4-(3,5-dimethoxybenzyl)-5-benzyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372626 (R)-N-(1-(4-(3-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372635 (R)-N-(1-(4-(4-methoxybenzyl)-5-(3-phenylpropyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372638 (R)-N-(1-(4-(2-methoxybenzyl)-5-benzyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372639 (R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(2-methoxy)benzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372645 (R)-N-(1-(4-(3-methoxybenzyl)-5-benzyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372646 (R)-N-(1-(5-((1H-indol-3-yl)methyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372648 (R)-N-(1-(4-(4-methoxybenzyl)-5-benzyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372649 (R)-N-(1-(5-(3-(1H-indol-3-yl)propyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372658 (R)-N-(1-(4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372659 (R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372671 (R)-N-(1-(4-(2-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372689 (R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(2,4-dimethoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372690 (R)-N-(1-(5-(3-(1H-indol-3-yl)propyl)-4-(2,4-dimethoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372691 (R)-N-(1-(4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372692 (R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(3,5-dimethoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372694 (R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(3-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372695 (R)-N-(1-(5-(3-(1H-indol-3-yl)propyl)-4-(3-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372719 2-amino-N-((R)-1-(4,5-dibenzyl-4H-1,2,4-triazol-3-yl)-2-(1Hindol-3-yl)ethyl)-2-methylpropanamide 372720 (R)-N-(1-(4-(4-ethylbenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372721 N-((R)-1-(4-(4-bromobenzyl)-5-benzyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372723 (R)-N-(1-(4-(4-fluorobenzyl)-5-benzyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372725 N-((R)-1-(4-(4-fluorobenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372726 N-((R)-1-(4-(4-methoxyphenethyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372727 N-((R)-1-(4-(3,4-dichlorobenzyl)-5-benzyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372728 (R)-N-(2-(1H-indol-3-yl)-1-(5-phenethyl-4-(thiophen-2-ylmethyl)-4H-1,2,4-triazol-3-yl)ethyl)-2-amino-2-methylpropanamide 372729 N-((R)-1-(4-(3,4-dichlorobenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372730 (R)-2-amino-N-(1-(4-(furan-2-ylmethyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-methylpropanamide 372732 (R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-phenyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372734 N-((R)-2-(1H-indol-3-yl)-1-(4,5-diphenethyl-4H-1,2,4-triazol-3-yl)ethyl)-2-amino-2-methylpropanamide 372736 (R)-N-(1-(4-(2-(1H-indol-3-yl)ethyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372738 2-amino-N-((R)-1-(5-benzyl-4-hexyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-methylpropanamide 372740 (R)-N-(1-(5-((1H-indol-3-yl)methyl)-4-methyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372743 (R)-N-(1-(5-((1H-indol-3-yl)methyl)-4-(2,4-dimethoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372747 (R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-hexyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372748 N-((R)-1-(4-(2-(1H-indol-3-yl)ethyl)-5-benzyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372749 (R)-N-(1-(4,5-bis(2-(1H-indol-3-yl)ethyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372750 (R)-N-(1-(4-(2-(1H-indol-3-yl)ethyl)-5-(3-(1H-indol-3-yl)propyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372751 (R)-N-(1-(5-(2-(1H-indol-2-yl)ethyl)-4-(4-methylbenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372754 (R)-N-(1-(5-(3-(1H-indol-3-yl)propyl)-4-hexyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372756 (R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-methyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372757 (R)-N-(1-(4-(4-methylbenzyl)-5-(3-phenylpropyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372761 (R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-benzyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372762 (R)-N-(1-(4-(4-methylbenzyl)-5-(3-benzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372763 (R)-N-(1-(5-((1H-indol-3-yl)methyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372764 (R)-N-(1-(5-(3-(1H-indol-3-yl)propyl)-4-benzyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372765 (R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-bromobenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372766 (R)-N-(1-(5-(3-(1H-indol-3-yl)propyl)-4-(4-bromobenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372767 (R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-fluorobenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372768 (R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(3,4-dichlorobenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372769 (R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372770 N-((R)-1-(5-((1H-indol-3-yl)methyl)-4-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372771 (R)-N-(1-(5-(3-(1H-indol-3-yl)propyl)-4-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372773 N-((R)-1-(5-(2-(1H-indol-3-yl)ethyl)-4-(2,2-diphenylethyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372774 (R)-2-amino-N-(1-(5-benzyl-4-(naphthalen-1-ylmethyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-methylpropanamide 372775 (R)-N-(1-(5-(3-(1H-indol-3-yl)propyl)-4-(naphthalen-1-ylmethyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372776 (R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(naphthalen-1-ylmethyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372777 (R)-N-(2-(1H-indol-3-yl)-1-(4-(naphthalen-1-ylmethyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)ethyl)-2-amino-2-methylpropanamide 372778 (R)-N-(1-(4-(4-methylbenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide 372875 2-(2-{4-[1-(2-[1,3]dioxolan-2-yl-ethyl)-1H-indol-3-yl]piperidin-1-yl}ethoxy)benzoic acid 372876 3-(2-(4-(1-(2-ethoxyethyl)-1H-indol-3-yl)piperidin-1-yl)ethoxy)thiophene-2-carboxylic acid 372877 2-(1-(2-(thiophen-2-yl)phenoxy)ethyl)-4,5-dihydro-1H-imidazole 372878 rac-2-(1-(2-(thiophen-3-yl)phenoxy)ethyl)-4,5-dihydro-1H-imidazole 372879 2-[1-(2'-methyl-biphenyl-2-yloxy)-ethyl]-4,5-dihydro-1H-imidazole 372882 2-(2-(4-(1-(furan-2-ylmethyl)-1H-indol-3-yl)piperidin-1-yl)ethoxy)benzoic acid 372883 2-{2-[4-(6-fluoro-1-furan-2-ylmethyl-1H-indol-3-yl)piperidin-1-yl]ethoxy}benzoic acid 372884 (+/-)-2-furan-2-yl-5-(octahydropyrido[1,2-a]pyrazin-2-yl)[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 372885 2-{2-[4-(1-butyl-6-fluoro-1H-indol-3-yl)piperidin-1-yl]-ethoxy}benzoic acid 372886 2-[1-(3'-methyl-biphenyl-2-yloxy)-ethyl]-4,5-dihydro-1H-imidazole 372887 2-[1-(4'-methyl-biphenyl-2-yloxy)-ethyl]-4,5-dihydro-1H-imidazole 372888 2'-[1-(4,5-dihydro-1H-imidazol-2-yl)-ethoxy]-biphenyl-2-ol 372891 2-(2-(4-(1-(thiophen-2-ylmethyl)-1H-indol-3-yl)piperidin-1-yl)ethoxy)benzoic acid 372892 2-{2-[4-(6-fluoro-1-furan-3-ylmethyl-1H-indol-3-yl)piperidin-1-yl]ethoxy}benzoic acid 372893 (R)-2-furan-2-yl-7-(hexahydropyrrolo[1,2-a]pyrazin-2-yl)[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 372894 rac-2'-(1-(4,5-dihydro-1H-imidazol-2-yl)ethoxy)biphenyl-3-ol 372895 2'-[1-(4,5-dihydro-1H-imidazol-2-yl)ethoxy]-biphenyl-4-ol 372896 2-[1-(2'-nitro-biphenyl-2-yloxy)-ethyl]-4,5-dihydro-1H-imidazole 372900 2-(2-(4-(1-((5-chlorothiophen-2-yl)methyl)-6-fluoro-1H-indol-3-yl)piperidin-1-yl)ethoxy)benzoic acid 372901 3-{4-[6-fluoro-1-(2-methoxyethyl)-1H-indol-3-yl]piperidin-1-ylmethyl}benzoic acid 372902 3-{4-[1-(2-ethoxyethyl)-5-methoxy-1H-indol-3-yl]piperidin-1-ylmethyl}benzoic acid 372903 rac-2-(1-(3'-nitrobiphenyl-2-yloxy)ethyl)-4,5-dihydro-1H-imidazole 372904 2-[1-(4'-nitro-biphenyl-2-yloxy)-ethyl]-4,5-dihydro-1H-imidazole 372905 2'-[1-(4,5-dihydro-1H-imidazol-2-yl)ethoxy]-biphenyl-3-ylamine 372907 2-(2-(4-(1-(2-(1,4-dioxan-2-yl)ethyl)-1H-indol-3-yl)piperidin-1-yl)ethoxy)benzoic acid 372909 3-(4-(1,4-diazepan-1-yl)-6-(((1S,2R,5S)-6,6-dimethylbicyclo[3.1.1]heptan-2-yl)methylamino)-1,3,5-triazin-2-ylamino)-4-methylbenzamide 372910 (7RS,9aRS)-[2-(5-amino-2-furan-2-yl[1,2,4]triazolo-[1,5-c]pyrimidin-7-yl)octahydropyrido[1,2-a]pyrazin-7-yl]methanol 372911 2-{1-[(3'-fluoro-1,1'-biphenyl-2-yl)oxy]ethyl}-4,5-dihydro-1H-imidazole 372912 SID29215339 372913 2-(2-{4-[1-(2-ethoxyethyl)-5-methoxy-1H-indol-3-yl]piperidin-1-yl}ethoxy)benzoic acid 372914 2-(2-(4-(1-(2-(pyridin-2-yl)ethyl)-1H-indol-3-yl)piperidin-1-yl)ethoxy)benzoic acid 372915 3-(2-(4-(1-(2-ethoxyethyl)-1H-indol-3-yl)piperidin-1-yl)ethoxy)benzoic acid 372916 2-methoxy-5-{4-[1-(2-methoxyethyl)-1H-indol-3-yl]piperidin-1-ylmethyl}benzoic acid 372917 5-{4-[6-fluoro-1-(2-methoxyethyl)-1H-indol-3-yl]piperidin-1-ylmethyl}-2-methoxybenzoic acid 372918 2-[1-(biphenyl-2-ylsulfanyl)-ethyl]-4,5-dihydro-1H-imidazole 372919 cis-2-(3-biphenyl-2-yl-oxiranyl)-4,5-dihydro-1H-imidazole 372921 2-(2-(4-(1-(2-ethoxyethyl)-5-fluoro-1H-indol-3-yl)piperidin-1-yl)ethoxy)benzoic acid 372922 4-(2-(4-(1-(2-ethoxyethyl)-1H-indol-3-yl)piperidin-1-yl)ethoxy)benzoic acid 372923 5-[4-(6-fluoro-1-thiophen-2-ylmethyl-1H-indol-3-yl)piperidin-1-ylmethyl]-2-methoxybenzoic acid 372924 (S)-2-furan-2-yl-5-(hexahydropyrrolo[1,2-a]pyrazin-2-yl)[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 372925 2-[1-(biphenyl-2-yloxy)ethyl]-4,5-dihydrooxazole 372927 5-[1-(biphenyl-2-yloxy)ethyl]-3,4-dihydro-2H-pyrrole 372928 2-(2-(4-(1-(2-ethoxyethyl)-6-fluoro-1H-indol-3-yl)piperidin-1-yl)ethoxy)benzoic acid 372929 2-(2-(4-(5-bromo-1-(2-ethoxyethyl)-1H-indol-3-yl)piperidin-1-yl)ethoxy)benzoic acid 372930 2-((4-(1-(2-ethoxyethyl)-1H-indol-3-yl)piperidin-1-yl)methyl)benzoic acid 372931 3-[4-(1-furan-2-ylmethyl-1H-indol-3-yl)piperidin-1-ylmethyl]benzoic acid 372932 3-[4-(1-thiophen-2-ylmethyl-1H-indol-3-yl)piperidin-1-ylmethyl]benzoic acid 372935 2-(2-(4-(7-bromo-1-(2-ethoxyethyl)-1H-indol-3-yl)piperidin-1-yl)ethoxy)benzoic acid 372936 2-(2-(4-(1-(2-ethoxyethyl)-7-methyl-1H-indol-3-yl)piperidin-1-yl)ethoxy)benzoic acid 372939 5-[4-(6-fluoro-1-furan-3-ylmethyl-1H-indol-3-yl)piperidin-1-ylmethyl]-2-methoxybenzoic acid 372944 2-(2-(4-(1-(2-ethoxyethyl)-6-(trifluoromethyl)-1H-indol-3-yl)piperidin-1-yl)ethoxy)benzoic acid 372946 2-(2-((4-(1-(2-ethoxyethyl)-1H-indol-3-yl)piperidin-1-yl)methyl)phenoxy)acetic acid 372947 5-{4-[1-(5-chlorothiophen-2-ylmethyl)-6-fluoro-1H-indol-3-yl]piperidin-1-ylmethyl}-2-methoxybenzoic acid 372950 2-(2-(4-(1-(2-ethoxyethyl)-1H-indol-3-yl)piperidin-1-yl)ethoxy)-6-fluorobenzoic acid 372952 (+/-)-2-furan-2-yl-7-(octahydro-pyrido[1,2-a]pyrazin-2-yl)-[1,2,4]triazolo[1,5-c]pyrimidin-5-yl-amine 372953 2-(3-((4-(1-(2-ethoxyethyl)-1H-indol-3-yl)piperidin-1-yl)methyl)phenoxy)acetic acid 372957 2-(2-(4-(1-(2-ethoxyethyl)-1H-indol-3-yl)piperidin-1-yl)ethoxy)-3,5-dibromobenzoic acid 372958 2-(2-(4-(1-(2-ethoxyethyl)-1H-indol-3-yl)piperidin-1-yl)ethoxy)-5-methylbenzoic acid 372960 (+/-)-2-furan-2-yl-5-(octahydro-pyrido[1,2-a]pyrazin-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl-amine 372961 2-methoxy-5-[4-(1-thiophen-2-ylmethyl-1H-indol-3-yl)-piperidin-1-ylmethyl]benzoic acid 372962 (S)-2-furan-2-yl-7-(hexahydro-pyrrolo[1,2-a]pyrazin-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-5-ylamine 372964 5-acetyl-2-(2-(4-(1-(2-ethoxyethyl)-1H-indol-3-yl)piperidin-1-yl)ethoxy)benzoic acid 372967 2-(4-((4-(1-(2-ethoxyethyl)-1H-indol-3-yl)piperidin-1-yl)methyl)phenoxy)acetic acid 372968 (S,S)-5-(3-benzyl-hexahydro-pyrrolo[1,2-a]pyrazin-2-yl)-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 372971 2-(2-(4-(1-(2-methoxyethyl)-1H-indol-3-yl)piperidin-1-yl)ethoxy)benzoic acid 372974 2-(2-{4-[6-fluoro-1-(2-methoxyethyl)-1H-indol-3-yl]piperidin-1-yl}ethoxy)benzoic acid 372976 5-{4-[1-(2-ethoxyethyl)-1H-indol-3-yl]piperidin-1-ylmethyl}-2-fluorobenzoic acid 372981 2-{2-[4-(1-cyclopropylmethyl-1H-indol-3-yl)piperidin-1-yl]ethoxy}benzoic acid 372982 4-bromo-3-((4-(1-(2-ethoxyethyl)-1H-indol-3-yl)piperidin-1-yl)methyl)benzoic acid 372984 2-{2-[1-(4,5-dihydro-1H-imidazol-2-yl)-ethoxy]phenyl}pyridine 372985 3-(2-(1-(4,5-dihydro-1H-imidazol-2-yl)ethoxy)phenyl)pyridine 372986 4-(2-(1-(4,5-dihydro-1H-imidazol-2-yl)ethoxy)phenyl)pyridine 372989 2-{2-[4-(1-cyclopropylmethyl-6-fluoro-1H-indol-3-yl)piperidin-1-yl]ethoxy}benzoic acid 372990 2-{2-[4-(1-allyl-1H-indol-3-yl)piperidin-1-yl]ethoxy}-benzoic acid 372991 4-(2-((R)-2-((S)-3-hydroxyoct-1-enyl)-5-oxopyrrolidin-1-yl)ethyl)benzoate 372992 (7RS,9aRS)-2-furan-2-yl-5-[7-(quinazolin-2-yloxymethyl)-octahydro-pyrido[1,2-a]pyrazin-2-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 372994 4-methyl-3-(4-(methyl(2-phenylpropyl)amino)-6-((S)-pyrrolidin-3-ylamino)-1,3,5-triazin-2-ylamino)benzamide 372995 (S)-3-(4-(isobutylamino)-6-(pyrrolidin-3-ylamino)-1,3,5-triazin-2-ylamino)-4-methylbenzamide 372996 (7RS,9aSR)-2-furan-2-yl-5-(7-phenoxymethyl-octahydro-pyrido[1,2-a]pyrazin-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 372997 (6RS,9aRS)-2-furan-2-yl-5-(6-phenoxymethyl-octahydro-pyrido[1,2-a]pyrazin-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 372998 4-(2-((S)-2-((S)-3-hydroxyoctyl)-5-oxopyrrolidin-1-yl)ethyl)benzoic acid 372999 5-(2-((R)-2-((S,E)-3-hydroxyoct-1-enyl)-5-oxopyrrolidin-1-yl)ethyl)thiophene-2-carboxylic acid 373000 (7RS,9aRS)-2-furan-2-yl-5-(7-{[(pyridin-4-ylmethyl)-amino]methyl}octahydropyrido[1,2-a]pyrazin-2-yl)[1,2,4]-triazolo[1,5-a][1,3,5]triazin-7-ylamine 373002 7-((7R,9aS)-7-(aminomethyl)-hexahydro-1H-pyrido[1,2-a]pyrazin-2(6H)-yl)-2-(furan-2-yl)-[1,2,4]triazolo[1,5-f]pyrimidin-5-amine 373003 5-((7R,9aS)-7-(aminomethyl)-hexahydro-1H-pyrido[1,2-a]pyrazin-2(6H)-yl)-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine 373004 (7RS,9aRS)-2-furan-2-yl-5-[7-(4-methoxy-phenoxymethyl)-octahydro-pyrido[1,2-a]pyrazin-2-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 373005 (7RS,9aSR)-2-furan-2-yl-5-[7-(4-methoxy-phenoxymethyl)-octahydro-pyrido[1,2-a]pyrazin-2-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 373006 4-(2-((R)-2-((S,E)-5-cyclobutyl-3-hydroxypent-1-enyl)-5-oxopyrrolidin-1-yl)ethyl)benzoic acid 373010 (7RS,9aRS)-5-(7-aminomethyloctahydropyrido[1,2-a]-pyrazin-2-yl)-2-furan-2-yl[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 373011 (7RS,9aRS)-[2-(5-amino-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin-7-yl)-octahydro-pyrido[1,2-a]pyrazin-7-yl]-methanol 373012 (7RS,9aRS)-5-[7-(2-fluoro-phenoxymethyl)-octahydro-pyrido[1,2-a]pyrazin-2-yl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 373013 5-((7S,9aS)-7-((3-fluorophenoxy)methyl)-hexahydro-1H-pyrido[1,2-a]pyrazin-2(6H)-yl)-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-amine 373014 4-(2-((S)-2-((S)-5-cyclobutyl-3-hydroxypentyl)-5-oxopyrrolidin-1-yl)ethyl)benzoic acid 373015 4-(2-((R)-2-((S,E)-3-hydroxy-4-(3-(methoxymethyl)phenyl)but-1-enyl)-5-oxopyrrolidin-1-yl)ethyl)benzoic acid 373018 (S)-3-(4-(isobutyl(methyl)amino)-6-(pyrrolidin-3-ylamino)-1,3,5-triazin-2-ylamino)-4-methylbenzamide 373019 (S)-4-methyl-3-(4-(methyl(neopentyl)amino)-6-(pyrrolidin-3-ylamino)-1,3,5-triazin-2-ylamino)benzamide 373020 (7RS,9aSR)-5-[7-(3-fluoro-phenoxymethyl)-octahydro-pyrido[1,2-a]pyrazin-2-yl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 373021 (7RS,9aRS)-5-[7-(3-fluoro-phenoxymethyl)-octahydro-pyrido[1,2-a]pyrazin-2-yl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 373022 (7RS,9aSR)-2-furan-2-yl-5-[7-(quinazolin-2-yloxymethyl)-octahydro-pyrido[1,2-a]pyrazin-2-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 373023 4-{2-[(2S)-2-[(3R)-3-[3-(4-chloro-2-methylphenyl)phenyl]-3-hydroxypropyl]-5-oxopyrrolidin-1-yl]ethyl}benzoic acid 373026 (7RS,9aRS)-[2-(5-amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)-octahydropyrido[1,2-a]pyrazin-7-yl]-methanol 373027 (S)-3-(4-(cyclohexyl(methyl)amino)-6-(pyrrolidin-3-ylamino)-1,3,5-triazin-2-ylamino)-4-methylbenzamide 373028 (7RS,9aSR)-5-[7-(2, 4-difluoro-phenoxymethyl)-octahydro-pyrido[1,2-a]pyrazin-2-yl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 373030 2-(2-((R)-2-((S,E)-3-hydroxyoct-1-enyl)-5-oxopyrrolidin-1-yl)ethylthio)acetic acid 373031 4-(2-((R)-2-((S,E)-3-hydroxyoct-1-enyl)-5-oxopyrrolidin-1-yl)ethylthio)butanoic acid 373032 (7RS,9aRS)-2-furan-2-yl-5-[7-(pyrimidin-2-ylaminomethyl)octahydropyrido[1,2-a]pyrazin-2-yl][1,2,4]triazolo-[1,5-a][1,3,5]triazin-7-ylamine 373034 (7RS,9aSR)-[2-(7-amino-2-furan-2-yl[1,2,4]triazolo[1,5-a][1,3,5]triazin-5-yl)octahydropyrido[1,2-a]pyrazin-7-yl]-methanol 373035 (S)-N-ethyl-4-methyl-3-(4-(methyl(neopentyl)amino)-6-(pyrrolidin-3-ylamino)-1,3,5-triazin-2-ylamino)benzamide 373036 2-(furan-2-yl)-5-((7S,9aS)-7-((quinolin-6-yloxy)methyl)-hexahydro-1H-pyrido[1,2-a]pyrazin-2(6H)-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-amine 373038 2-(4-((R)-2-((S,E)-3-hydroxy-4-(3-(trifluoromethyl)phenyl)but-1-enyl)-5-oxopyrrolidin-1-yl)butoxy)acetic acid 373041 (S)-N-(2-methoxyethyl)-4-methyl-3-(4-(methyl(neopentyl)amino)-6-(pyrrolidin-3-ylamino)-1,3,5-triazin-2-ylamino)benzamide 373042 (S)-N-benzyl-4-methyl-3-(4-(methyl(neopentyl)amino)-6-(pyrrolidin-3-ylamino)-1,3,5-triazin-2-ylamino)benzamide 373043 (6RS,9aRS)-2-furan-2-yl-5-[6-(quinolin-6-yloxymethyl)-octahydro-pyrido[1,2-a]pyrazin-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-ylamine 373045 (7RS,9aRS)-2-furan-2-yl-5-(7-imidazol-1-ylmethyloctahydropyrido[1,2-a]pyrazin-2-yl)[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 373047 2-(furan-2-yl)-5-((7S,9aS)-7-((pyrimidin-2-ylamino)methyl)-hexahydro-1H-pyrido[1,2-a]pyrazin-2(6H)-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-amine 373048 (S)-methyl-4-methyl-3-(4-(methyl(neopentyl)amino)-6-(pyrrolidin-3-ylamino)-1,3,5-triazin-2-ylamino)benzoate 373049 5-((7S,9aS)-7-(aminomethyl)-hexahydro-1H-pyrido[1,2-a]pyrazin-2(6H)-yl)-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine 373050 (6RS,9aSR)-2-furan-2-yl-5-[6-(1H-indol-5-yloxymethyl)-octahydro-pyrido[1,2-a]pyrazin-2-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 373051 (7RS,9aRS)-2-furan-2-yl-5-(7-[1,2,4]triazol-1-ylmethyl-octahydro-pyrido[1,2-a]pyrazin-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 373052 (7RS,9aRS)-2-furan-2-yl-5-(7-tetrazol-1-ylmethyl-octahydro-pyrido[1,2-a]pyrazin-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 373055 (S)-N-cyclopentyl-4-methyl-3-(4-(methyl(neopentyl)-amino)-6-(pyrrolidin-3-ylamino)-1,3,5-triazin-2-ylamino)-benzamide 373056 5-((7S,9aS)-7-(aminomethyl)-hexahydro-1H-pyrido[1,2-a]pyrazin-2(6H)-yl)-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-amine 373057 (7RS,9aRS)-2-furan-2-yl-5-[7-(isoquinolin-5-yloxymethyl)-octahydro-pyrido[1,2-a]pyrazin-2-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 373061 2-(furan-2-yl)-7-((7R,9aS)-7-((pyrimidin-2-ylamino)methyl)-hexahydro-1H-pyrido[1,2-a]pyrazin-2(6H)-yl)-[1,2,4]triazolo[1,5-f]pyrimidin-5-amine 373063 (S)-N-methoxy-4-methyl-3-(4-(methyl(neopentyl)amino)-6-(pyrrolidin-3-ylamino)-1,3,5-triazin-2-ylamino)benzamide 373064 (S)-N-hydroxy-4-methyl-3-(4-(methyl(neopentyl)amino)-6-(pyrrolidin-3-ylamino)-1,3,5-triazin-2-ylamino)benzamide 373065 (7RS,9aSR)-2-furan-2-yl-5-[7-(isoquinolin-5-yloxymethyl)-octahydro-pyrido[1,2-a]pyrazin-2-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 373066 (7RS,9aRS)-2-furan-2-yl-5-[7-(pyridin-2-yloxymethyl)-octahydro-pyrido[1,2-a]pyrazin-2-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 373067 5-((7R,9aS)-7-((2,4-difluorobenzylamino)methyl)-hexahydro-1H-pyrido[1,2-a]pyrazin-2(6H)-yl)-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-amine 373069 5-((7R,9aS)-7-((bis((5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl)amino)methyl)-hexahydro-1H-pyrido[1,2-a]pyrazin-2(6H)-yl)-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-amine 373070 SID26753546 373072 (6RS,9aRS)-[2-(5-amino-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin-7-yl)-octahydro-pyrido[1,2-a]pyrazin-6-yl]-methanol 373073 (S)-N-isopropyl-4-methyl-3-(4-(methyl(neopentyl)-amino)-6-(pyrrolidin-3-ylamino)-1,3,5-triazin-2-ylamino)-benzamide 373074 (7RS,9aSR)-2-furan-2-yl-5-[7-(pyridin-2-yloxymethyl)-octahydro-pyrido[1,2-a]pyrazin-2-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 373075 2-(furan-2-yl)-5-((7R,9aS)-7-((quinolin-2-yloxy)methyl)-hexahydro-1H-pyrido[1,2-a]pyrazin-2(6H)-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-amine 373076 5-((7R,9aS)-7-(((5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methylamino)methyl)-hexahydro-1H-pyrido[1,2-a]pyrazin-2(6H)-yl)-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-amine 373081 N-methoxy-4-methyl-3-(4-(methyl(neopentyl)amino)-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-ylamino)benzamide 373082 N-methoxy-4-methyl-3-(4-(methyl(neopentyl)amino)-6-(piperazin-1-yl)-1,3,5-triazin-2-ylamino)benzamide 373083 (7RS,9aRS)-2-furan-2-yl-5-[7-(isoquinolin-3-yloxymethyl)-octahydro-pyrido[1,2-a]pyrazin-2-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 373084 5-((7R,9aS)-7-((bis(furan-2-ylmethyl)amino)methyl)-hexahydro-1H-pyrido[1,2-a]pyrazin-2(6H)-yl)-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-amine 373088 N-methoxy-4-methyl-3-(4-(methyl(neopentyl)amino)-6-(4-methyl-1,4-diazepan-1-yl)-1,3,5-triazin-2-ylamino)-benzamide 373089 3-(4-(1,4-diazepan-1-yl)-6-(methyl(neopentyl)amino)-1,3,5-triazin-2-ylamino)-N-methoxy-4-methylbenzamide 373090 (7RS,9aSR)-2-furan-2-yl-5-[7-(isoquinolin-3-yloxymethyl)-octahydro-pyrido[1,2-a]pyrazin-2-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 373091 (7RS,9aRS)-2-furan-2-yl-5-[7-(pyridin-3-yloxymethyl)-octahydro-pyrido[1,2-a]pyrazin-2-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 373093 5-((7R,9aS)-7-((bis(pyridin-2-ylmethyl)amino)methyl)-hexahydro-1H-pyrido[1,2-a]pyrazin-2(6H)-yl)-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-amine 373095 5-((7R,9aS)-7-((bis(pyridin-3-ylmethyl)amino)methyl)-hexahydro-1H-pyrido[1,2-a]pyrazin-2(6H)-yl)-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-amine 373098 (7RS,9aRS)-[2-(7-amino-2-furan-2-yl[1,2,4]triazolo-[1,5-a]pyrimidin-5-yl)octahydropyrido[1,2-a]pyrazin-7-yl]methanol 373099 3-(4-(((1S,2R,5S)-6,6-dimethylbicyclo[3.1.1]heptan-2-yl)-methylamino)-6-(4-methyl-1,4-diazepan-1-yl)-1,3,5-triazin-2-ylamino)-4-methylbenzamide 373100 (6RS,9aRS)-[2-(5-amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)-octahydropyrido[1,2-a]pyrazin-6-yl]-methanol 373101 (6RS,9aRS)-[2-(7-amino-2-furan-2-yl[1,2,4]triazolo[1,5-a][1,3,5]triazin-5-yl)octahydropyrido[1,2-a]pyrazin-6-yl]-methanol 373102 (6RS,9aRS)-2-furan-2-yl-5-[6-(pyridin-3-yloxymethyl)-octahydro-pyrido[1,2-a]pyrazin-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-ylamine 373103 (7RS,9aRS)-2-furan-2-yl-5-[7-(pyridin-4-yloxymethyl)-octahydro-pyrido[1,2-a]pyrazin-2-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 373105 5-((7S,9aS)-7-((bis(pyridin-3-ylmethyl)amino)methyl)-hexahydro-1H-pyrido[1,2-a]pyrazin-2(6H)-yl)-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-amine 373107 2-(furan-2-yl)-5-((7R,9aS)-7-((pyridin-3-ylmethylamino)methyl)-hexahydro-1H-pyrido[1,2-a]pyrazin-2(6H)-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-amine 373108 (7RS,9aRS)-[2-(7-amino-2-furan-2-yl[1,2,4]triazolo[1,5-a][1,3,5]triazin-5-yl)octahydropyrido[1,2-a]pyrazin-7-yl]-methanol 373109 3-(4-amino-6-(((1S,2R,5S)-6,6-dimethylbicyclo[3.1.1]heptan-2-yl)methylamino)-1,3,5-triazin-2-ylamino)-4-methylbenzamide 373110 (7RS,9aRS)-2-furan-2-yl-5-[7-(quinolin-6-yloxymethyl)octahydropyrido[1,2-a]pyrazin-2-yl][1,2,4]triazolo-[1,5-a][1,3,5]triazin-7-ylamine 373111 (7RS,9aRS)-2-furan-2-yl-5-(7-phenoxymethyl-octahydro-pyrido[1,2-a]pyrazin-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-ylamine 373112 (7RS,9aSR)-2-furan-2-yl-5-[7-(pyridin-4-yloxymethyl)-octahydro-pyrido[1,2-a]pyrazin-2-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 373113 3-(3-((R)-2-((S,E)-3-hydroxyoct-1-enyl)-5-oxopyrrolidin-1-yl)propyl)benzoic acid 373116 (7RS,9aRS)-5-{7-[(bispyridin-4-ylmethylamino)-methyl]octahydropyrido[1,2-a]pyrazin-2-yl}-2-furan-2-yl[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 373118 3-(4-(((1S,2R,5S)-6,6-dimethylbicyclo[3.1.1]heptan-2-yl)methylamino)-6-((S)-pyrrolidin-3-ylamino)-1,3,5-triazin-2-ylamino)-4-methylbenzamide 373119 (S)-3-(4-(4-fluorophenethylamino)-6-(pyrrolidin-3-ylamino)-1,3,5-triazin-2-ylamino)-4-methylbenzamide 373125 N-{4-[5-(4-fluorophenyl)-2-(4-methylsulfinylbenzylsulfanyl)-3-(2-methoxyethyl)-3H-imidazol-4-yl]pyridin-2-yl}acetamide 373129 N7-(((7S,9aR)-2-(2,4-difluorobenzyl)-octahydro-1H-pyrido[1,2-a]pyrazin-7-yl)methyl)-2-(furan-2-yl)-[1,2,4]triazolo[1,5-f]pyrimidine-5,7-diamine 373130 N-{4-[5-(4-fluorophenyl)-2-(4-methylsulfinylbenzylsulfanyl)-3-(3-methoxypropyl)-3H-imidazol-4-yl]pyridin-2-yl}acetamide 373134 (7RS,9aRS)-3-amino-5-{7-[(7-amino-2-furan-2-yl[1,2,4]-triazolo[1,5-a][1,3,5]triazin-5-ylamino)methyl]octahydropyrido[1,2-a]pyrazin-2-yl}-6-chloropyrazine-2-carboxylic acid methyl ester 373139 (7RS,9aRS)-2-furan-2-yl-N5-(2-pyrimidin-2-yloctahydropyrido[1,2-a]pyrazin-7-ylmethyl)[1,2,4]triazolo[1,5-a]-[1,3,5]triazine-5,7-diamine 373144 (7RS,9aSR)-N5-[2-(5-chloro-1-methyl-3-trifluoromethyl-1H-pyrazol-4-ylmethyl)octahydropyrido[1,2-a]pyrazin-7-ylmethyl]-2-furan-2-yl[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 373160 N-(4-(4-(4-fluorophenyl)-1-(2-hydroxyethyl)-2-(methylthio)-1H-imidazol-5-yl)pyridin-2-yl)acetamide 373161 N-(4-(4-(4-fluorophenyl)-1-(2-methoxyethyl)-2-(methylthio)-1H-imidazol-5-yl)pyridin-2-yl)acetamide 373162 N-{4-[5-(4-fluorophenyl)-2-(4-methylsulfinylbenzylsulfanyl)-3-(2-prop-2-ynyloxyethyl)-3H-imidazol-4-yl]pyridin-2-yl}acetamide 373172 N-(4-(4-(4-fluorophenyl)-1-(3-hydroxypropyl)-2-(methylthio)-1H-imidazol-5-yl)pyridin-2-yl)acetamide 373173 N-{4-[5-(4-fluorophenyl)-3-(3-methoxypropyl)-2-methylsulfanyl-3H-imidazol-4-yl]pyridin-2-yl}acetamide 373174 N-{4-[5-(4-fluorophenyl)-2-(4-methylsulfinylbenzylsulfanyl)-3-(2-methylsulfanylethyl)-3H-imidazol-4-yl]pyridin-2-yl}acetamide 373179 N-{4-[5-(4-fluorophenyl)-3-[2-(2-hydroxyethoxy)ethyl]-2-methylsulfanyl-3H-imidazol-4-yl]pyridin-2-yl}acetamide 373180 N-{4-[5-(4-fluorophenyl)-3-(2-hydroxypropyl)-2-methylsulfanyl-3H-imidazol-4-yl]pyridin-2-yl}acetamide 373181 N-{4-[5-(4-fluorophenyl)-2-(4-methylsulfinylbenzylsulfanyl)-3-(2-piperidin-1-ylethyl)-3H-imidazol-4-yl]pyridin-2-yl}acetamide 373187 N-{4-[3-(2-acetylaminoethyl)-5-(4-fluorophenyl)-2-methylsulfanyl-3H-imidazol-4-yl]pyridin-2-yl}acetamide 373188 N-{4-[3-(2-dimethylaminoethyl)-5-(4-fluorophenyl)-2-methylsulfanyl-3H-imidazol-4-yl]pyridin-2-yl}acetamide 373189 N-{4-[5-(4-fluorophenyl)-3-(2-hydroxyethyl)-2-(3-morpholin-4-yl-3-oxopropylsulfanyl)-3H-imidazol-4-yl]pyridin-2-yl}acetamide 373190 N-{4-[5-(4-fluorophenyl)-3-(2-hydroxyethyl)-2-(4-morpholin-4-yl-4-oxobutylsulfanyl)-3H-imidazol-4-yl]pyridin-2-yl}acetamide 373194 N-{4-[3-(2-allyloxyethyl)-5-(4-fluorophenyl)-2-methylsulfanyl-3H-imidazol-4-yl]pyridin-2-yl}acetamide 373195 N-{4-[5-(4-fluorophenyl)-2-methylsulfanyl-3-(2-prop-2-ynyloxyethyl)-3H-imidazol-4-yl]pyridin-2-yl}acetamide 373196 N-{4-[5-(4-fluorophenyl)-3-(3-hydroxypropyl)-2-(4-morpholin-4-yl-3-oxopropylsulfanyl)-3H-imidazol-4-yl]pyridin-2-yl}acetamide 373200 N-{4-[5-(4-fluorophenyl)-2-methylsulfanyl-3-(2-methylsulfanylethyl)-3H-imidazol-4-yl]pyridin-2-yl}acetamide 373201 N-{4-[3-(2,2-dimethoxyethyl)-5-(4-fluorophenyl)-2-methylsulfanyl3H-imidazol-4-yl]pyridin-2-yl}acetamide 373202 N-{4-[5-(4-fluorophenyl)-3-(2-methoxyethyl)-2-(3-morpholin-4-yl-3-oxopropylsulfanyl)-3H-imidazol-4-yl]pyridin-2-yl}acetamide 373207 N-{4-[3-(2,2-dimethyl[1,3]dioxolan-4-ylmethyl)-5-(4-fluorophenyl)-2-methylsulfanyl-3H-imidazol-4-yl]pyridin-2-yl}acetamide 373208 N-{4-[5-(4-fluorophenyl)-3-(2-morpholin-4-ylethyl)-2-methylsulfanyl-3H-imidazol-4-yl]pyridin-2-yl}acetamide 373214 N-{4-[5-(4-fluorophenyl)-3-(3-morpholin-4-ylpropyl)-2-methylsulfanyl-3H-imidazol-4-yl]pyridin-2-yl}-acetamide 373215 N-{4-[5-(4-fluorophenyl)-2-methylsulfanyl-3-(2-piperidin-1-ylethyl)-3H-imidazol-4-yl]pyridin-2-yl}acetamide 373220 (7RS,9aRS)-N5-[2-(3,5-difluorophenyl)octahydropyrido-[1,2-a]pyrazin-7-ylmethyl]-2-furan-2-yl[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 373228 (7RS,9aRS)-N5-[2-(2,4-difluorobenzyl)octahydropyrido-[1,2-a]pyrazin-7-ylmethyl]-2-furan-2-yl[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 373230 N-{4-[5-(4-fluorophenyl)-2-(4-methylsulfinylbenzylsulfanyl)-3-methyl-3H-imidazol-4-yl]pyridin-2-yl}acetamide 373231 N-{4-[5-(4-fluorophenyl)-3-(2-hydroxyethyl)-2-(4-methylsulfinylbenzylsulfanyl)-3H-imidazol-4-yl]pyridin-2-yl}acetamide 373233 4-({2-[(5-cyano-1,3-thiazol-2-yl)amino]-4-pyridinyl}-methyl)-N,N-dimethyl-1-piperazinecarboxamide 373234 4-[2-(5-cyanothiazol-2-ylamino)pyridin-4-ylmethyl]piperazine-1-carboxylic acid methylamide 373247 2-{4-[4-(2-hydroxyethanoyl)piperazin-1-ylmethyl]pyridin-2-ylamino}thiazole-5-carbonitrile 373255 2-[(4-{[4-(methylsulfonyl)piperidin-1-yl]methyl}pyridin-2-yl)amino]-1,3-thiazole-5-carbonitrile 373268 4-[2-(5-cyanothiazol-2-ylamino)-3-methylpyridin-4-ylmethyl]piperazine-1-carboxylic acid methylamide 373297 N-(2,6-diphenylpyrimidin-4-yl)benzamide 373304 N-(2,6-diphenylpyrimidin-4-yl)-4-methoxybenzamide) 373305 N-(2,6-diphenylpyrimidin-4-yl)acetamide 373313 N-(2,6-diphenylpyrimidin-4-yl)propionamide 373314 N-(2,6-diphenylpyrimidin-4-yl)butyramide 373315 hexanoic Acid (2,6-diphenylpyrimidin-4-yl)amide 373323 N-(2,6-diphenylpyrimidin-4-yl)isobutyramide 373324 N-(2,6-diphenylpyrimidin-4-yl)-3-methylbutyramide 373331 N-(2,6-diphenylpyrimidin-4-yl)-2-ethylbutyramide 373332 N-(2,6-diphenylpyrimidin-4-yl)-2-methylbutyramide 373345 N-(2,6-diphenylpyrimidin-4-yl)-2,2-dimethylpropionamide 373346 N-(2,6-diphenylpyrimidin-4-yl)-3,3-dimethylbutyramide 373352 cyclopropanecarboxylic acid (2,6-diphenylpyrimidin-4-yl)amide 373353 cyclobutanecarboxylic acid (2,6-diphenylpyrimidin-4-yl)amide 373366 cyclopentanecarboxylic acid (2,6-diphenylpyrimidin-4-yl)amide 373367 cyclohexanecarboxylic acid (2,6-diphenylpyrimidin-4-yl)amide 373371 (5-phenylthiazol-2-yl)(4-pyrrolidin-1-ylmethylpyridin-2-yl)amine 373372 1-{4-[2-(5-phenylthiazol-2-ylamino)pyridin-4-ylmethyl]piperazin-1-yl}ethanone 373378 4-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-N-(5-phenyl-1,3-thiazol-2-yl)pyridin-2-amine 373379 2-[4-(4-acetylpiperazin-1-ylmethyl)pyridin-2-ylamino]-thiazole-5-carbonitrile 373381 SID26755745 373386 2-(4-piperazin-1-ylmethylpyridin-2-ylamino)thiazole-5-carbonitrile 373387 2-(4-morpholin-4-ylmethylpyridin-2-ylamino)thiazole-5-carbonitrile 373388 4-({2-[(5-cyano-1,3-thiazol-2-yl)amino]-4-pyridinyl}-methyl)-1-piperazinecarboxamide 373399 N-(4,5-diphenylpyrimidin-2-yl)acetamide 373400 N-(4,6-diphenylpyrimidin-2-yl)propionamide 373401 N-(4,6-diphenylpyrimidin-2-yl)butyramide 373409 pentanoic acid (4,6-diphenylpyrimidin-2-yl)amide 373416 N-(4,6-diphenylpyrimidin-2-yl)isobutyramide 373417 N-(4,6-diphenylpyrimidin-2-yl)-2,2-dimethylpropionamide 373424 N-(4,6-diphenylpyrimidin-2-yl)-3-methylbutyramide 373425 N-(4,6-diphenylpyrimidin-2-yl)-2-ethylbutyramide 373432 cyclopropane carboxylic acid (4,6-diphenylpyrimidin-2-yl)amide 373433 cyclobutane carboxylic acid (4,6-diphenylpyrimidin-2-yl)amide 373439 N-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-2-(4-(2-methoxyphenyl)piperazin-1-yl)acetamide 373441 cyclopentane carboxylic acid (4,6diphenylpyrimidin-2-yl)amide 373459 N-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-4-(2-methoxyphenyl)-1-piperazinebutanamide 373461 cyclohexanecarboxylic acid (4,6-diphenylpyrimidin-2-yl)amide 373476 N-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-4-(2-methoxyphenyl)-1-piperazinepentanamide 373477 N-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-4-(2-methoxyphenyl)-1-piperazinehexanamide 373490 N-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-4-(2-methoxyphenyl)-1-piperazinebutanamide 373491 N-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-4-(2-methoxyphenyl)-1-piperazinepentanamide 373497 N-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-4-(2-methoxyphenyl)-1-piperazinehexanamide 373498 N-(7-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-4-(2-methoxyphenyl)-1-piperazinebutanamide 373501 N-(7-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-4-(2-methoxyphenyl)-1-piperazinepentanamide 373502 N-(7-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-4-(2-methoxyphenyl)-1-piperazinehexanamide 373506 N-(8-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-4-(4-(2-methoxyphenyl)piperazin-1-yl)butanamide 373507 N-(8-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-4-(2-methoxyphenyl)-1-piperazinepentanamide 373512 N-(8-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-4-(2-methoxyphenyl)-1-piperazinehexanamide 373533 N-(4,6-diphenylpyrimidin-2-yl)benzamide 373534 N-(4,6-diphenylpyrimidin-2-yl)-4-chlorobenzamide 373557 N-(4,6-diphenylpyrimidin-2-yl)-3-chlorobenzamide 373568 6-(4-(2-methoxyphenyl)piperazin-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)hexanamide 373570 6-(4-(2-acetylphenyl)piperazin-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)hexanamide 373571 4-(4-chloro-2-methoxyphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 373576 4-(2,5-dimethoxyphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 373577 4-(3-methoxyphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 373584 4-(4-methoxyphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 373585 4-(3-cyanophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 373588 SID26755678 373590 4-(4-cyanophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 373591 4-(3-acetylphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 373596 4-(4-acetylphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 373597 2-(4-(6-oxo-6-(1,2,3,4-tetrahydronaphthalen-1-ylamino)hexyl)piperazin-1-yl)benzamide 373599 7-[(2,4-dichloro-5-methoxyanilino)amino]thieno[3,2-b]pyridine-6-carbonitrile 373604 6-(4-(2-(methylthio)phenyl)piperazin-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)hexanamide 373606 7-[(2,4-dichloro-5-methoxyphenyl)amino]-2-phenylthieno[3,2-b]pyridine-6-carbonitrile 373609 6-(4-(2-(methylsulfonyl)phenyl)piperazin-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)hexanamide 373615 6-(4-(2-hydroxyphenyl)piperazin-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)hexanamide 373617 7-[(2,4-dichloro-5-methoxyphenyl)amino]-2-[4-(4-methylpiperazin-1-ylmethyl)phenyl]thieno[3,2-b]pyridine-6-carbonitrile 373622 6-(4-(2-chlorophenyl)piperazin-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)hexanamide 373623 6-(4-(2-nitrophenyl)piperazin-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)hexanamide 373625 7-[(2,4-dichloro-5-methoxyphenyl)amino]-2-{3-[(4-methylpiperazine-1-yl)methyl]phenyl}thieno[3,2-b]pyridine-6-carbonitrile 373628 N-(1,2,3,4-tetrahydronaphthalen-1-yl)-6-(4-o-tolylpiperazin-1-yl)hexanamide 373634 6-(4-phenylpiperazin-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)hexanamide 373640 4-(1,2-benzisoxazol-3-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 373648 4-[(2,4-dichloro-5-methoxyphenyl)amino]-2-[4-(morpholin-4-ylmethyl)phenyl]thieno[2,3-b]pyridine-5-carbonitrile 373651 4-(2-benzoxazolyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 373669 4-(4-(2-methoxyphenyl)piperazin-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)butanamide 373671 4-(1H-benzimidazol-2-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 373672 4-(5-methoxybenzoxazol-2-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 373675 7-(2,4-dichlorophenoxy)-2-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}thieno[3,2-b]pyridine-6-carbonitrile 373678 5-(4-(2-methoxyphenyl)piperazin-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)pentanamide 373680 6-(4-(2-cyanophenyl)piperazin-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)hexanamide 373682 7-[2,4-dichlorobenzyl)amino]-2-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}thieno[3,2-b]pyridine-6-carbonitrile 373724 (+/-)isobutyl 8-chloro-2-((4-(diethylamino)phenyl)carbamoyl)-1,2,3,4-tetrahydronaphthalen-2-ylcarbamate 373745 (1S,2S,9R)-18-(cyclopropylmethyl)-7-methyl-5-phenyl-10-oxa-7,18-diazahexacyclo[9.9.1.0^{1,9}.0^{2,17}.0^{4,8}.0^{15,21}]henicosa-4(8),5,11,13,15(21)-pentaene-2,12-diol 373752 (1S,2S,9R)-18-(cyclopropylmethyl)-7-ethyl-5-phenyl-10-oxa-7,18-diazahexacyclo[9.9.1.0^{1,9}.0^{2,17}.0^{4,8}.0^{15,21}]henicosa-4(8),5,11,13,15(21)-pentaene-2,12-diol 373764 17-cyclopropylmethyl-6-7-didehydro-3,14-dihydroxy-4,5alpha-epoxy-1'-ethyl-4',5',6',7'-tetrahydroindolo[2',3';6,7]morphinan 373765 l',17-dicyclopropylmethyl-6-7-didehydro-3,14-dihydroxy-4,5alpha-epoxy-4',5',6',7'-tetrahydroindolo[2',3';6,7]morphinan 373774 (1S,2S,13R)-11-benzyl-22-(cyclopropylmethyl)-14-oxa-11,22-diazaheptacyclo[13.9.1.0^{1,13}.0^{2,21}.0^{4,12}.0^{5,10}.0^{19,25}]pentacosa-4(12),5(10),15,17,19(25)-pentaene-2,16-diol 373785 1'-cyclohexylmethyl-17-cyclopropylmethyl-6-7-didehydro-3,14-dihydroxy-4,5alpha-epoxy-4',5',6',7'-tetrahydroindolo[2',3';6,7]morphinan 373791 17-cyclopropylmethyl-6-7-didehydro-3,14-dihydroxy-4,5alpha-epoxy-1'-phenylethyl-4',5',6',7'-tetrahydroindolo[2',3';6,7]morphinan 373792 6,7-didehydro-3,14-dihydroxy-1'17-dimethyl-4,5 alpha-epoxy-4',5',6',7'-tetrahydroindolo[2',3';6,7]morphinan 373801 6,7-didehydro-3,14-dihydroxy-4,5alpha-epoxy-1'-ethyl-17-methyl-4',5',6',7'-tetrahydroindolo'2',3';6,7]morphinan 373802 1'-benzyl-6,7-didehydro-3,14-dihydroxy-4,5alpha-epoxy-17-methyl-4',5',6',7'-tetrahydroindolo[2',3':6,7]morphinan 373812 1'-cyclohexylmethyl-6,7-didehydro-3,14-dihydroxy-4,5alpha-epoxy-17-methyl-4',5',6',7'-tetrahydroindolo[2',3':6,7]morphinan 373824 6,7-didehydro-3,14-dihydroxy-4,5alpha-epoxy-17-methyl-1'phenylethyl-4',5',6',7'-tetrahydroindolo[2',3':6,7]morphinan 373854 H-Dmt-Tic-Glu-NH-(CH2)5-NH2 373855 5-[({5-[(2S)-2-({2-[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]-1,2,3,4-tetrahydroisoquinolin-3-yl}formamido)-4-carboxybutanamido]pentyl}carbamothioyl)amino]-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic acid 374088 (2R)-[2-aminoacetamido]-3-(4-chlorophenyl)propionyl-1-2-[(2-thienyl)ethylaminomethyl]phenyl piperazine 374109 3-phenyl-5-(4-phenyl-5-(trifluoromethyl)thiophen-2-yl)-1,2,4-oxadiazole 374110 3-(2,4-dichlorophenyl)-5-(4-phenyl-5-(trifluoromethyl)thiophen-2-yl)-1,2,4-oxadiazole 374115 SID26753263 374116 1-(4-(5-(4-phenyl-5-(trifluoromethyl)thiophen-2-yl)-1,2,4-oxadiazol-3-yl)benzyl)azetidine-3-carboxylic acid 374122 1-(4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)benzyl)pyrrolidine-3-carboxylic acid 374130 26-tert-butyl-13-(2,4,4-trimethylpentan-2-yl)-3,6,9,16,19,22-hexaoxatricyclo[22.3.1.0^{10,15}]octacosa-1(28),10(15),11,13,24,26-hexaene-28-carboxylic acid 374131 1-(3-bromo-4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)benzyl)azetidine-3-carboxylic acid 374140 1-(3-chloro-4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)benzyl)azetidine-3-carboxylic acid 374141 1-(3-fluoro-4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)benzyl)azetidine-3-carboxylic acid 374151 1-(3-methyl-4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)benzyl)azetidine-3-carboxylic acid 374152 1-(3-ethyl-4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)benzyl)azetidine-3-carboxylic acid 374167 1-(3-methoxy-4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)benzyl)azetidine-3-carboxylic acid 374168 1-(3,5-dimethyl-4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)benzyl)azetidine-3-carboxylic acid 374176 1-(3,5-dichloro-4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)benzyl)azetidine-3-carboxylic acid 374212 SID26754965 374225 1-(4-nonylbenzyl)pyrrolidine-3-carboxylic acid 374226 1-(4-nonylbenzyl)azetidine-3-carboxylic acid 374253 12-(R)-amino-5-(S),8-(R)-dibenzyl-2-(S)-(1Hindol-3-ylmethyl)-1,4,7,10-tetraaza-cyclotetradecane-3,6,11,14-tetraone 374255 (2S,5S,8R,13R)-13-amino-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 374257 5-(S)-benzyl-8-(R)-(3,4-dichloro-benzyl)-2-(S)-(1H-indol-3-ylmethyl)-1,4,7,10-tetraaza-cyclotetradecane-3,6,11,14-tetraone 374258 (2S,5S,8R,12S)-12-amino-5-benzyl-8-(3,4-dichloro-benzyl)-2-(1H-indol-3-ylmethyl)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 374259 5-(S),8-(R)-dibenzyl-2-(S)-(1H-indol-3-ylmethyl)-12-(R)-(tetrahydro-pyran-4-ylamino)-1,4,7,10-tetraaza-cyclotetradecane-3,6,11,14-tetraone trifluoroacetate 374260 (2S,5S,8R,12S)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-12-(tetrahydro-pyran-4-ylamino)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 374261 (2S,5S,8R,13R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-13-(tetrahydro-pyran-4-ylamino)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 374267 (2S,5S,8R,13S)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-13-(tetrahydro-pyran-4-ylamino)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 374268 (2S,5S,8R,12R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-12-morpholin-4-yl-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 374269 (2S,5S,8R,12S)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-12-morpholin-4-yl-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 374270 (2S,5S,8R,12R)-5-benzyl-8-(3,4-dichloro-benzyl)-2-(1H-indol-3-ylmethyl)-12-morpholin-4-yl-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 374271 (2S,5S,8R,12R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-12-piperidin-1-yl-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 374272 (2S,5S,8R,12R)-12-(4-amino-piperidin-1-yl)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 374273 (2S,5S,8R,12R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-12-piperazin-1-yl-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 374274 (2S,5S,8R,12R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-12-(4-methyl-piperazin-1-yl)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 374275 (2S,5S,8R,12R)-12-(4-acetyl-piperazin-1-yl)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 374276 (2S,5S,8R,12R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-12-(4-methanesulfonyl-piperazin-1-yl)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 374277 (2S,5S,8R,12R)-5,8-dibenzyl-12-[1,4']bipiperidinyl-1'-yl-2-(1H-indol-3-ylmethyl)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 374278 (2S,5S,8R,12R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-12-(4-morpholin-4-yl-piperidin-1-yl)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 374279 (2S,5S,8R,12R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-12-(tetrahydro-thiopyran-4-ylamino)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 374280 (2S,5S,8R,12R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-12-(1-oxo-hexahydro-1lambda*4*-thiopyran-4-ylamino)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 374281 (2S,5S,8R,12R)-5,8-dibenzyl-12-(1,1-dioxo-hexahydro-1lambda*6*-thiopyran-4-ylamino)-2-(1H-indol-3-ylmethyl)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 374282 (2S,5S,8R,12R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-12-[methyl-(tetrahydro-pyran-4-yl)-amino]-1,4,7,10tetaaza-cyclotetradecane-3,6,11,14-tetraone 374283 (2S,5S,8R,12R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-12-(1-methanesulfonyl-piperidin-4-ylamino)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 374284 4-[(2S,5S,8R,12R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-3,6,11,14-tetraoxo-1,4,7,10tetraaza-cyclotetradec-12-ylamino]-piperidine-1-sulfonic acid amide 374285 (2S,5S,8R,12R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-12-(1-methyl-piperidin-4-ylamino)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 374286 N-(3-(R)-acetylamino-4-(R),5-(R)-dihydroxy-6-(R)-hydroxymethyl-tetrahydro-pyran-2-(R)-yl)-N'-[5-(S),8-(R)-dibenzyl-2-(S)-(1H-indol-3-ylmethyl)-3,6,11,14-tetraoxo-1,4,7,10-tetraaza-cyclotetradec-12-(R)-yl]-succinamide 374287 2-(S)-acetylamino-N4-(3-(R)-acetylamino-4-(R),5-(R)-dihydroxy-6-(R)-hydroxymethyl-tetrahydro-pyran-2-(R)-yl)-N'-[5-(S),8-(R)-dibenzyl-2-(S)-(1H-indol-3-ylmethyl)-3,6,11,14-tetraoxo-1,4,7,10-tetraaza-cyclotetradec-12-(R)-yl]-succinamide 374288 N-((1S,2R,3S,4R)-1-{[(2S,5S,8R,12R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-3,6,11,14-tetraoxo-1,4,7,10tetraaza-cyclotetradec-12-ylamino]-methyl}-2,3,4,5-tetrahydroxy-pentyl)-acetamide 374289 (2S,5S,8R,12R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-12-((2S,3R,4R,5R)-2,3,4,5,6-pentahydroxy-hexylamino)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 374290 (2S,5S,8R,12R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-12-[(2S,3R,4R,5R)-2,3,5,6-tetrahydroxy-4-((2S,3R,4S,5R,6R)-3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-hexylamino]-1,4,7,10tetraaza-cyclotetrad 374291 (2S,5S,8R,12R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-12-[(2S,3R,4S,5R)-2,3,5,6-tetrahydroxy-4-((2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-hexylamino]-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetrone 374308 (2S,5S,8R,12R)-5,8-dibenzyl-12-{[(2S,3S,4S,5R)-4-{[(2R,3R,4R,5S,6R)-3,4-dihydroxy-6-(hydroxymethyl)-5-{[(2S,3S,4R,5R,6S)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy}oxan-2-yl]oxy}-2,3,5,6-tetrahydroxyhexyl]amino}-2-(1H-indol-3-ylmethyl)-1,4,7,10-tetraazacyclotetradecane-3,6,11,14-tetrone 374317 2-(S),3-(R),5-(R),6-tetrahydroxy-4-(R)-(O-r-D-glucopyranosyl)-hexanoic acid [5-(S),8-(R)-dibenzyl-2-(S)-(1-Hindol-3-ylmethyl)-3,6,11,14-tetraoxo-1,4,7,10-tetraaza-cyclotetradec-12-(R)-yl]-amide 374319 N-[(2S,5S,8R,12R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-3,6,11,14-tetraoxo-1,4,7,10tetraaza-cyclotetradec-12-yl]-2-(4-hydroxy-piperidin-1-yl)-acetamide 374320 N-[(2S,5S,8R,12R)-5,8-Dibenzyl-2-(1H-indol-3-ylmethyl)-3,6,11,14-tetraoxo-1,4,7,10tetraaza-cyclotetradec-12-yl]-2-((S)-2-hydroxymethyl-pyrrolidin-1-yl)-acetamide 374321 N-[(2S,5S,8R,12R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-3,6,11,14-tetraoxo-1,4,7,10tetraaza-cyclotetradec-12-yl]-2-(4-methyl-piperazin-1-yl)-acetamide 374322 1-{[(2S,5S,8R,12R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-3,6,11,14-tetraoxo-1,4,7,10tetraaza-cyclotetradec-12-ylcarbamoyl]-methyl}-piperidine-4-carboxylic acid amide 374323 N-[(2S,5S,8R,12R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-3,6,11,14-tetraoxo-1,4,7,10tetraaza-cyclotetradec-12-yl]-2-(1-oxo-1lambda*4*-thiomorpholin-4-yl)-acetamide 374324 N-((2S,5S,8R,12R)-5,8-dibenzyl-2-indan-1-ylmethyl-3,6,11,14-tetraoxo-1,4,7,10tetraaza-cyclotetradec-12-yl)-2-(4-sulfamoyl-piperazin-1-yl)-acetamide 374325 2-[1,4']bipiperidinyl-1'-yl-N-((2S,5S,8R,12R)-5,8-dibenzyl-2-indan-1-ylmethyl-3,6,11,14-tetraoxo-1,4,7,10tetraaza-cyclotetradec-12-yl)-acetamide 374326 N-[(2S,5S,8R,12R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-3,6,11,14-tetraoxo-1,4,7,10tetraaza-cyclotetradec-12-yl]-2-[4-(1-oxo-1lambda*4*-thiomorpholin-4-yl)-piperidin-1-yl]-acetamide 374327 N-[(2S,5S,8R,12R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-3,6,11,14-tetraoxo-1,4,7,10tetraaza-cyclotetradec-12-yl]-2-(4-morpholin-4-yl-piperidin-1-yl)-acetamide 374399 2S,5S,8R)-5,8-dibenzyl-2-(1H-indol-3-ylmethyl)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 374400 (2S,5S,8R)-5-benzyl-8-(3,4-dichloro-benzyl)-2-(1H-indol-3-ylmethyl)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 374442 6-(2-hexyl-5-hydroxyphenoxy)hexanoic acid cyclopropylamide 374449 11-(2-hexyl-5-hydroxyphenoxy)undecanoic acid (2-hydroxyethyl)amide 374450 11-(2-hexyl-5-hydroxyphenoxy)undecanoic acid cyclopropylamide 374455 6-(3-hydroxy-5-pentylphenoxy)hexanoic acid cyclopropylamide 374457 11-(2-hexyl-5-hydroxyphenoxy)undecanoic acid (4-hydroxyphenyl)amide 374462 11-(3-hydroxy-5-pentylphenoxy)undecanoic acid (2-hydroxyethyl)amide 374463 N-cyclopropyl-11-(3-hydroxy-5-pentylphenoxy)undecanamide 374464 16-(2-hexyl-5-hydroxyphenoxy)hexadecanoic acid cyclopropylamide 374465 16-(2-hexyl-5-hydroxyphenoxy)hexadecanoic acid (4-hydroxyphenyl)amide 374470 11-(3-hydroxy-5-pentylphenoxy)undecanoic acid (4-hydroxyphenyl)amide 374471 16-(3-hydroxy-5-pentylphenoxy)hexadecanoic acid (2-hydroxyethyl)amide 374473 SID26754856 374502 11-(3-hydroxyphenoxy)undecanoic acid cyclopropilamide 374513 16-(3-hydroxyphenoxy)hexadecanoic acid cyclopropylamide 374514 16-(3-hydroxyphenoxy)hexadecanoic acid (4-hydroxyphenyl)amide 374518 6-(3-hydroxy-4-hexylphenoxy)hexanoic acid (2-hydroxyethyl)amide 374519 6-(3-hydroxy-4-hexylphenoxy)hexanoic acid cyclopropylamide 374524 11-(3-hydroxy-4-hexylphenoxy)undecanoic acid (2-hydroxyethyl)amide 374530 11-(3-hydroxy-4-hexylphenoxy)undecanoic acid cyclopropylamide 374561 7-chloro-1-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-4,5-dihydro-1H-benzo[g]indazole-3-carboxamide 374562 8-Chloro-1-(2,4-dichloro-phenyl)-1,3a,4,5,6,10b-hexahydro-1,2-diaza-benzo[e]azulene-3-carboxylic acid piperidin-1-ylamide 374568 8-chloro-1-(2',4'-dichlorophenyl)-N-pyrrolidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide 374569 8-chloro-1-(2',4'-dichlorophenyl)-N-homopiperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide 374576 8-chloro-1-(2',4'-dichlorophenyl)-N-cyclohexyl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide 374577 8-chloro-1-(2',4'-dichlorophenyl)-N-phenyl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide 374581 1-(bis(4-chlorophenyl)methyl)-3-phenylurea 374582 8-chloro-1-(2',4'-dichlorophenyl)-N-p-chlorophenyl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide 374583 8-chloro-1-(2',4'-dichlorophenyl)-N-m,p-dichlorophenyl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide 374588 1-(bis(4-bromophenyl)methyl)-3-phenylurea 374589 1-[bis(4-chlorophenyl)methyl]-3-(4-chlorophenyl)- 374590 8-chloro-1-(2',4'-dichlorophenyl)-N-p-methylphenyl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide 374591 8-chloro-1-(2',4'-dichlorophenyl)-N-p-methoxylphenyl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide 374595 1-(bis(4-chlorophenyl)methyl)-3-(4-bromophenyl)urea 374596 1-[bis(4-bromophenyl)methyl]-3-(4-chlorophenyl)-urea 374597 7-chloro-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide 374598 9-chloro-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide 374602 1-(bis(4-bromophenyl)methyl)-3-(4-bromophenyl)urea 374603 1-[bis(4-iodophenyl)methyl]-3-(4-bromophenyl)urea 374604 8-bromo-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide 374605 8-methyl-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide 374611 8-methyl-1-(2',4'-dichlorophenyl)-N-pyrrolidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide 374612 1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide 374615 1-[bis(4-chlorophenyl)methyl]-3-phenylthiourea 374620 1-[bis(4-bromophenyl)methyl]-3-phenylthiourea 374621 1-[bis(4-chlorophenyl)methyl]-3-(4-chlorophenyl)thiourea 374626 1-[bis(4-bromophenyl)methyl]-3-(4-chlorophenyl)thiourea 374643 5,5'-bis(4-bromophenyl)-3-phenyl-2-thioxoimidazolidin-4-one 374651 5,5'-bis(4-bromophenyl)-3-(4-chlorophenyl)-2-thioxoimidazolidin-4-one 374747 isopropyl 4-(4-methoxyphenethylamino)-1-(2-chloro-2-phenylethyl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374748 isopropyl 4-(2-chlorophenethylamino)-1-(2-chloro-2-phenylethyl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374750 isopropyl 4-(3-chlorophenethylamino)-1-(2-chloro-2-phenylethyl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374751 isopropyl 4-(4-chlorophenethylamino)-1-(2-chloro-2-phenylethyl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374752 methyl 1-(2-chloro-2-phenylethyl)-4-(cyclopropylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374753 butyl 1-(2-chloro-2-phenylethyl)-4-(cyclopropylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374754 butyl 1-(2-chloro-2-phenylethyl)-4-(propylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374756 methyl 1-(2-chloro-2-phenylethyl)-4-(propylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374757 methyl 1-(2-chloro-2-phenylethyl)-4-(pyrrolidin-1-yl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374758 butyl 1-(2-chloro-2-phenylethyl)-4-(pyrrolidin-1-yl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374763 methyl 4-(benzylamino)-1-(2-chloro-2-phenylethyl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374765 sec-butyl 1-(2-chloro-2-phenylethyl)-4-(cyclopropylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374768 methyl 1-(2-chloro-2-phenylethyl)-4-(phenethylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374769 1-(2-chloro-2-phenyl-ethyl)-4-(2-p-tolyl-ethylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid methyl ester 374770 sec-butyl 1-(2-chloro-2-phenylethyl)-4-(propylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374771 sec-butyl 1-(2-chloro-2-phenylethyl)-4-(phenethylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374773 methyl 4-(4-methoxyphenethylamino)-1-(2-chloro-2-phenylethyl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374774 1-(2-chloro-2-phenyl-ethyl)-4-(2-p-tolyl-ethylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid ethyl ester 374775 4-butyl-5-(4-cyclopropylbut-1-en-2-yl)-1-(2-phenylpropyl)-1H-indene 374776 cyclopropylmethyl 1-(2-chloro-2-phenylethyl)-4-(phenethylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374780 ethyl 4-(4-methoxyphenethylamino)-1-(2-chloro-2-phenylethyl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374781 ethyl 4-(2-fluorophenethylamino)-1-(2-chloro-2-phenylethyl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374782 1-(2-chloro-2-phenyl-ethyl)-4-(2-p-tolyl-ethylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid cyclopropylmethyl ester 374786 ethyl 4-(3-fluorophenethylamino)-1-(2-chloro-2-phenylethyl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374787 ethyl 4-(4-fluorophenethylamino)-1-(2-chloro-2-phenylethyl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374792 ethyl 4-(2-chlorophenethylamino)-1-(2-chloro-2-phenylethyl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374793 ethyl 4-(3-chlorophenethylamino)-1-(2-chloro-2-phenylethyl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374799 ethyl 4-(4-chlorophenethylamino)-1-(2-chloro-2-phenylethyl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374800 propyl 1-(2-chloro-2-phenylethyl)-4-(cyclopropylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374804 propyl 1-(2-chloro-2-phenylethyl)-4-(propylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374805 propyl 1-(2-chloro-2-phenylethyl)-4-(pyrrolidin-1-yl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374806 propyl 1-(2-chloro-2-phenylethyl)-4-morpholino-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374807 propyl 4-(benzylamino)-1-(2-chloro-2-phenylethyl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374811 propyl 1-(2-chloro-2-phenylethyl)-4-(phenethylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374812 isopropyl 1-(2-chloro-2-phenylethyl)-4-(cyclopropylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374823 isopropyl 1-(2-chloro-2-phenylethyl)-4-(propylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374824 isopropyl 1-(2-chloro-2-phenylethyl)-4-(pyrrolidin-1-yl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374829 isopropyl 1-(2-chloro-2-phenylethyl)-4-morpholino-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374830 isopropyl 4-(benzylamino)-1-(2-chloro-2-phenylethyl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374833 isopropyl 1-(2-chloro-2-phenylethyl)-4-(phenethylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 374834 1-(2-chloro-2-phenyl-ethyl)-4-(2-p-tolyl-ethylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid isopropyl ester 374948 (S)-4-((4R,7S,10S,13S,16S,19S)-13-((1H-indol-3-yl)methyl)-10-(4-aminobutyl)-16-benzyl-4-((S)-1-carboxy-2-methylpropylcarbamoyl)-7-(4-hydroxybenzyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentaazacycloicosan-19-ylamino)-3-amino-4-oxobutanoic acid 374949 H-Asp-c[Pen-Phe-Trp-Lys-Tyr-Cys]-Val-OH 374950 H-asp-cyclo[pen-phe-Dtrp-lys-tyr-cys]-val-OH 374951 H-asp-cyclo[cys-phe-Dtrp-lys-tyr-cys]-val-OH 374952 H-asp-cyclo[pen-phe-trp-orn-tyr-cys]-val-OH 374953 H-asp-cyclo[cys-phe-trp-orn-tyr-cys]-val-OH 374954 H-Asp-c[Pen-Phe-DTrp-Orn-Tyr-Cys]-Val-OH 374955 H-asp-cyclo[cys-phe-Dtrp-orn-tyr-cys]-val-OH 374956 H-asp-cyclo[Dpen-phe-Dtrp-orn-tyr-cys]-val-OH 374957 H-asp-cyclo[pen-phe-Dtrp-Dorn-tyr-cys]-val-OH 375127 bis(4-hydroxybenzyl)sulfide 375129 N6-(4-hydroxybenzyl)adenine riboside 375204 4-(4-(3-(4-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)prop-2-ynyloxy)benzyl)-morpholine 375209 6-((4-methylpiperazin-1-yl)methyl)-3-(5-(3-phenoxyprop-1-ynyl)thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole 375210 6-((4-methylpiperazin-1-yl)methyl)-3-(5-(3-phenoxyprop-1-ynyl)thiophen-2-yl)-1,4-dihydroindeno[1,2-c]pyrazole 375211 4-((3-(5-(3-phenoxyprop-1-ynyl)thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazol-6-yl)methyl)piperazine-1-carbaldehyde 375212 6-((4-methylpiperazin-1-yl)methyl)-3-(4-(3-phenoxyprop-1-ynyl)thiophen-2-yl)-1,4-dihydroindeno[1,2-c]pyrazole 375213 6-((4-methylpiperazin-1-yl)methyl)-3-(3-(3-phenoxyprop-1-ynyl)phenyl)-1,4-dihydroindeno[1,2-c]pyrazole 375214 1-methyl-4-((3-(5-(3-phenoxyprop-1-ynyl)thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazol-6-yl)methyl)piperazin-2-one 375215 4-methyl-1-((3-(5-(3-phenoxyprop-1-ynyl)thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazol-6-yl)methyl)piperazin-2-one 375216 6-((4-methylpiperazin-1-yl)methyl)-3-(4-(3-phenoxyprop-1-ynyl)phenyl)-1,4-dihydroindeno[1,2-c]pyrazole 375217 7-((4-methylpiperazin-1-yl)methyl)-3-(5-(3-phenoxyprop-1-ynyl)thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole 375218 (4-methylpiperazin-1-yl)(3-(5-(3-phenoxyprop-1-ynyl)thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazol-6-yl)methanone 375219 3-((3-(5-(3-phenoxyprop-1-ynyl)thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazol-6-yl)methyl)thiazolidine 375220 3-(5-ethynylthiophen-3-yl)-6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazole 375221 6-((4-methylpiperazin-1-yl)methyl)-3-(5-(pent-1-ynyl)thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole 375222 6-(2-methoxyethoxy)-3-(5-(3-phenoxyprop-1-ynyl)thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole 375223 N,N-dimethyl-2-(3-(5-(3-phenoxyprop-1-ynyl)thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazol-6-yloxy)acetamide 375224 4-(4-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno-[1,2-c]pyrazol-3-yl)thiophen-2-yl)but-3-yn-1-ol 375225 2-methyl-5-(4-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)pent-4-yn-2-ol 375226 6-((1H-imidazol-1-yl)methyl)-3-(5-(3-phenoxyprop-1-ynyl)thiophen-3-yl)-1, 4-dihydroindeno[1,2-c]pyrazole 375227 6-((1H-pyrazol-1-yl)methyl)-3-(5-(3-phenoxyprop-1-ynyl)thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole 375228 3-(5-(3-methoxyprop-1-ynyl)thiophen-3-yl)-6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazole 375229 6-((4-methylpiperazin-1-yl)methyl)-3-(5-(4-phenoxybut-1-ynyl)thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole 375230 6-((1H-1,2,3-triazol-1-yl)methyl)-3-(5-(3-phenoxyprop-1-ynyl)-thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole 375231 6-((1H-1,2,4-triazol-1-yl)methyl)-3-(5-(3-phenoxyprop-1-ynyl)-thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole 375232 3-(5-(3-(2-chlorophenoxy)prop-1-ynyl)thiophen-3-yl)-6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazole 375233 3-(5-(3-(3-chlorophenoxy)prop-1-ynyl)thiophen-3-yl)-6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazole 375234 2-(3-(4-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno-[1,2-c]pyrazol-3-yl)thiophen-2-yl)prop-2-ynyloxy)acetamide 375235 3-(5-(3-(2-methoxyethoxy)prop-1-ynyl)thiophen-3-yl)-6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazole 375236 3-(5-(3-(4-chlorophenoxy)prop-1-ynyl)thiophen-3-yl)-6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazole 375237 3-(5-(3-(2-methoxyethoxy)prop-1-ynyl)thiophen-3-yl)-7-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazole 375238 6-((1H-1,2,4-triazol-1-yl)methyl)-3-(5-(3-(2-methoxyethoxy)-prop-1-ynyl)thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole 375239 3-(5-(3-(3,4-dimethylphenoxy)prop-1-ynyl)thiophen-3-yl)-6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazole 375240 6-((4-methylpiperazin-1-yl)methyl)-3-(5-(3-(pyridin-3-yloxy)-prop-1-ynyl)thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole 375241 7-((1H-1,2,4-triazol-1-yl)methyl)-3-(5-(3-(2-methoxyethoxy)-prop-1-ynyl)thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole 375242 3-(5-(3-(2-methoxyethoxy)prop-1-ynyl)thiophen-3-yl)-6-((4-methylpiperazin-1-yl)methyl)indeno[1,2-c]pyrazol-4(1H)-one 375243 6-((4-methylpiperazin-1-yl)methyl)-3-(5-(4-phenylbut-1-ynyl)-thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole 375244 N-(3-(4-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno-[1,2-c]pyrazol-3-yl)thiophen-2-yl)prop-2-ynyl)aniline 375247 N-(3-(4-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno-[1,2-c]pyrazol-3-yl)thiophen-2-yl)prop-2-ynyl)benzamide 375249 N-(3-(4-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno-[1,2-c]pyrazol-3-yl)thiophen-2-yl)prop-2-ynyl)benzenesulfonamide 375252 phenyl 3-(4-(6-((4-Methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)prop-2-ynylcarbamate 375255 1-methyl-1-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-m-tolylurea 375256 1-(3-(4-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno-[1,2-c]pyrazol-3-yl)thiophen-2-yl)prop-2-ynyl)-3-phenylurea 375257 3-(5-(3-phenoxyprop-1-ynyl)thiophen-3-yl)-1,4-dihydroindeno-[1,2-c]pyrazole 375258 6-(4-methylpiperazin-1-yl)-3-(5-(3-phenoxyprop-1-ynyl)-thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole 375259 6-(2-(4-methylpiperazin-1-yl)ethyl)-3-(5-(3-phenoxyprop-1-ynyl)thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole 375260 1-methyl-1-((5-(7-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-m-tolylurea 375261 6-((4-methylpiperidin-1-yl)methyl)-3-(5-(3-phenoxyprop-1-ynyl)thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole 375262 6-((1-methylpiperidin-4-yl)methyl)-3-(5-(3-phenoxyprop-1-ynyl)thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole 375514 N-(1-(pyridin-3-ylmethyl)piperidin-3-yl)-1H-indazol-5-amine 375519 N-(1-((1H-pyrrol-2-yl)methyl)piperidin-3-yl)-1H-indazol-5-amine 375521 N-(1-(thiophen-2-ylmethyl)piperidin-3-yl)-1H-indazol-5-amine 375528 N-(1-(thiophen-3-ylmethyl)piperidin-3-yl)-1H-indazol-5-amine 375529 N-(1-(furan-2-ylmethyl)piperidin-3-yl)-1H-indazol-5-amine 375553 5-(1-benzylpiperidin-4-yloxy)-1H-indazole 375554 5-(1-benzylpiperidin-3-yloxy)-1H-indazole 375563 N-(1-benzylpiperidin-3-yl)-1H-indazol-5-amine 375589 N-(1-(2-chlorobenzyl)pyrrolidin-3-yl)-1H-indazol-5-amine 375590 N-(1-(3-chlorobenzyl)pyrrolidin-3-yl)-1H-indazol-5-amine 375597 N-(1-(4-chlorobenzyl)pyrrolidin-3-yl)-1H-indazol-5-amine 375598 N-(1-(2-chlorobenzyl)piperidin-3-yl)-1H-indazol-5-amine 375599 N-(1-(3-chlorobenzyl)piperidin-3-yl)-1H-indazol-5-amine 375602 N-(1-benzylpiperidin-4-yl)-1H-indazol-5-amine 375603 N-(1-benzylpyrrolidin-3-yl)-1H-indazol-5-amine 375604 N-(1-(4-chlorobenzyl)piperidin-3-yl)-1H-indazol-5-amine 375613 N-(1-(4-fluorobenzyl)piperidin-3-yl)-1H-indazol-5-amine 375614 N-(1-(3,4-difluorobenzyl)piperidin-3-yl)-1H-indazol-5-amine 375617 1-benzyl-N-(1H-indazol-5-yl)piperidine-3-carboxamide 375618 N-(1-(4-methylbenzyl)piperidin-3-yl)-1H-indazol-5-amine 375619 N-(1-(4-methoxybenzyl)piperidin-3-yl)-1H-indazol-5-amine 375626 N-(1-(2-aminobenzyl)piperidin-3-yl)-1H-indazol-5-amine 375632 N-(1-(3-aminobenzyl)piperidin-3-yl)-1H-indazol-5-amine 375633 N-(1-(4-aminobenzyl)piperidin-3-yl)-1H-indazol-5-amine 375641 5-((3-(3-(prop-1-en-2-yl)benzyl)cyclohexyl)methyl)-1H-indene 375642 N-(1-(4-nitrobenzyl)piperidin-3-yl)-1H-indazol-5-amine 376242 N-(1-(4-fluorobenzyl)pyrrolidin-3-yl)isoquinolin-5-amine 376243 N-(1-(2,6-difluorobenzyl)pyrrolidin-3-yl)isoquinolin-5-amine 376249 8-[(3-dimethylamino-propyl)-methyl-amino]-6-methoxy-4-oxo-1,4-dihydroquinoline-2-carboxylic acid(4-morpholin-4-yl-phenyl)amide 376250 6-methoxy-8-(4-methyl-piperazin-1-yl)-4-oxo-1,4-dihydroquinoline-2-carboxylic acid (4-morpholin-4-ylphenyl)amide 376251 N-(1-(2-aminobenzyl)pyrrolidin-3-yl)isoquinolin-5-amine 376252 N-(1-(3-aminobenzyl)pyrrolidin-3-yl)isoquinolin-5-amine 376258 8-[(2-dimethylamino-ethyl)-methyl-amino]-6-methoxy-4-oxo-1,4-dihydroquinoline-2-carboxylic acid(4-morpholin-4-yl-phenyl)amide 376259 8-((3R)-(+)-3-dimethylamino-pyrrolidin-1-yl)-6-methoxy-4-oxo-1,4-dihydroquinoline-2-carboxylic acid(4-morpholin-4-yl-phenyl)amide 376260 N-(1-(4-aminobenzyl)pyrrolidin-3-yl)isoquinolin-5-amine 376261 (3R)-N-[1-(3-aminobenzyl)-3-pyrrolidyl]-N-(5-isoquinolyl)amine 376267 (3S)-N-[1-(3-aminobenzyl)-3-pyrrolidyl]-N-(5-isoquinolyl)amine 376273 8-[ethyl-(1-ethyl-pyrrolidin-3-yl)-amino]-6-methoxy-4-oxo-1,4-dihydroquinoline-2-carboxylic acid (4-morpholin-4-yl-phenyl)amide 376281 6-fluoro-8-(4-methyl-piperazin-1-yl)-4-oxo-1,4-dihydroquinoline-2-carboxylic acid (4-morpholin-4-ylphenyl)amide 376288 4-dimethylamino-6-methoxy-8-(4-methyl-piperazin-1-yl)-quinoline-2-carboxylic acid (4-morpholin-4-ylphenyl)amide 376289 6-methoxy-4-methylamino-8-(4-methyl-piperazin-1-yl)-quinoline-2-carboxylic acid (4-morpholin-4-yl-phenyl)amide 376296 6-fluoro-4-methoxy-8-(4-methyl-piperazin-1-yl)-quinoline-2-carboxylic acid (4-morpholin-4-yl-phenyl)amide 376377 N-(1-(4-chlorobenzyl)piperidin-3-yl)isoquinolin-5-amine 376378 N-(1-(2-chlorobenzyl)pyrrolidin-3-yl)isoquinolin-5-amine 376384 6-methoxy-8-(4-methyl-[1,4]diazepan-1-yl)-4-oxo-1,4-dihydroquinoline-2-carboxylic acid (4-morpholin-4-phenyl)amide 376385 N-(1-(3-chlorobenzyl)pyrrolidin-3-yl)isoquinolin-5-amine 376386 N-(1-(4-chlorobenzyl)pyrrolidin-3-yl)isoquinolin-5-amine 376481 N-(2,6-dimethyl-phenyl)-5-phenylimidazo[1,5-a]pyrazine-8-amine 376482 N-Phenyl-5-phenylimidazo[1,5-a]pyrazin-8-amine 376490 N-(2,6-dichlorophenyl)-5-phenylimidazo[1,5-a]pyrazin-8-amine 376491 N-(2,6-difluorophenyl)-5-phenylimidazo[1,5-a]pyrazin-8-amine 376499 N-(5-phenylimidazo[1,5-a]pyrazin-8-yl)-2,4,6-trimethylphenylamine 376500 N-(2-methoxy-6-methylphenyl)-5-phenylimidazo[1,5-a]pyrazin-8-amine 376504 N-methyl-N-phenyl-5-phenylimidazo[1,5-a]pyrazin-8-amine 376505 N-(2,6-dimethylphenyl)-5-(4-methoxyphenyl)imidazo[1,5-a]pyrazin-8-amine 376513 N-[5-(4-methoxyphenyl)imidazo[1,5-a]pyrazin-8-yl]-o-tolylamine 376514 N-[5-(4-methoxyphenyl)imidazo[1,5-a]pyrazin-8-yl]phenylamine 376560 4-[8-(2,6-dimethylphenylamino)imidazo[1,5-a]-pyrazin-5-yl]benzoic acid 376561 4-[8-(2,6-dimethylphenylamino)imidazo[1,5-a]-pyrazin-5-yl]-N,N-dimethylbenzamide 376570 N-(2,6-dimethylphenyl)-5-pyridin-4-ylimidazo[1,5-a]-pyrazin-8-amine 376571 N-(2,6-dimethylphenyl)-5-thiophen-2-ylimidazo[1,5-a]pyrazin-8-amine 376591 N-(2-chloro-6-methylphenyl)-6-(3-methoxyphenyl)imidazo[1,5-a]pyrazin-8-amine 376592 N-(2-chloro-6-methylphenyl)-6-(4-fluorophenyl)-imidazo[1,5-a]pyrazin-8-amine 376598 N-(2,6-dimethylphenyl)-5-(4-fluorophenyl)imidazo[1,5-a]pyrazin-8-amine 376599 N-(2,6-dimethylphenyl)-5-[4-(2-morpholin-4-ylethoxy)phenyl]imidazo[1,5-a]pyrazin-8-amine 376606 N-(2,6-dimethylphenyl)-5-[4-(2-pyrrolidin-1-ylethoxy)phenyl]imidazo[1,5-a]pyrazin-8-amine 376607 N-(2,6-dimethylphenyl)-5-[4-(1-methylpiperidin-3-ylmethoxy)phenyl]imidazo[1,5-a]pyrazin-8-amine 376618 N-(2,6-dimethylphenyl)-5-[3-(1-methylpiperidin-3-ylmethoxy)phenyl]imidazo[1,5-a]pyrazin-8-amine 376627 SID26752156 376638 [3-amino-3-(3-octylphenylcarbamoyl)propyl]-phosphonic acid 376659 (R)-2-amino-3-(4-octylphenylamino)-3-oxopropyl dihydrogen phosphate 376686 N-(2,6-dimethylphenyl)-5-(3-methoxyphenyl)imidazo[1,5-a]pyrazin-8-amine 376687 4-[8-(2,6-dimethylphenylamino)imidazo[1,5-a]pyrazin-5-yl]benzonitrile 376693 N-[5-(3,4-dimethoxyphenyl)imidazo[1,5-a]pyrazin-8-yl]-2,6-dimethylphenylamine 376694 N-(2,6-dimethylphenyl)imidazo[1,5-a]pyrazin-8-amine 376703 N-(2,6-dimethylphenyl)-5-(4-trifluoromethylphenyl)imidazo[1,5-a]pyrazin-8-amine 376704 N-[5-(4-dimethylaminophenyl)imidazo[1,5-a]pyrazin-8-yl]-2,6-dimethylphenylamine 377125 (5alpha,6alpha)-17-(cyclobutylmethyl)-6,14-dihydroxy-4,5-epoxymorphinan-3-yl-17-(cyclobutylmethyl)morphinan-3-yl sebacoylate 377126 17-(cyclopropylmethyl)morphinan-3-yl(5alpha)-17-(cyclopropylmethyl)-14-hydroxy-6-oxo-4,5-epoxymorphiana-3-yl sebacoylate 377142 17-(cyclopropylmethyl)-6,7-didehydro-4,5alpha-epoxy-3,14-dihydroxy-1'-(10'''-[3''-propyl]-[1''',4''',7''',10'''-tetraazacyclododecane-1''',4''',7'''-triacetic acid])indolo[6,7:2',3']morphinan 377143 17-cyclopropylmethyl)-6,7-didehydro-4,5alpha-epoxy-3,14-dihydroxy-1'-(10'''-[6''-hexyl]-[1''',4''',7''',10'''-tetraazacyclododecane-1''',4''',7'''-triacetic acid])indolo[6,7:2',3']morphinan 377278 (2S)-2-[(2S)-2-[(2S,3R)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2-aminophenyl)formamido]-5-carbamimidamidopentanamido]-3-(1H-imidazol-5-yl)propanamido]-3-(4-hydroxyphenyl)propanamido]-4-methylpentanamido]-3-carbamoylpropanamido]-4-methylpentanamido]-3-methylbutanamido]-3-hydroxybutanamido]-5-carbamimidamidopentanamido]-N-[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-(4-hydroxyphenyl)ethyl]carbamoyl}butyl]pentanediamide 377279 (2S)-N-[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-(4-hydroxyphenyl)ethyl]carbamoyl}butyl]-2-[(2S)-5-carbamimidamido-2-[(2S,3R)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-5-carbamimidamido-2-{[2-(methylsulfanyl)pyridin-3-yl]formamido}pentanamido]-3-(1H-imidazol-5-yl)propanamido]-3-(4-hydroxyphenyl)propanamido]-4-methylpentanamido]-3-carbamoylpropanamido]-4-methylpentanamido]-4-methylpentanamido]-3-hydroxybutanamido]pentanamido]pentanediamide 377518 N-(2-(2-(4-chlorobenzyloxy)ethylamino)ethyl)isoquinoline-5-sulfonamide 377555 1-(4-(9H-purin-6-yl)phenyl)-2-phenylethanamine 377563 5-methyl-4-phenyl-1H-pyrazole 377566 (4-(9H-purin-6-yl)phenyl)(4-chlorophenyl)methanamine 377572 (4-(5-methyl-1H-pyrazol-4-yl)phenyl)methanamine 377573 2-(4-(5-methyl-1H-pyrazol-4-yl)phenyl)ethanamine 377574 3-(4-(1H-pyrazol-4-yl)phenyl)propan-1-amine 377575 4-phenyl-1H-pyrazole 377577 (4-(9H-purin-6-yl)phenyl)(4-chlorophenyl)-N-methylmethanamine 377584 6-(4-(4-(4-chlorophenyl)piperidin-4-yl)phenyl)-9H-purine 377586 2-(4-(1H-pyrazol-4-yl)phenyl)-2-phenylethanamine 377587 4-(4-(1H-pyrazol-4-yl)phenyl)-4-phenylpiperidine 377588 2-(4-chloro-phenyl)-2-[4-(1H-pyrazol-4-yl)-phenyl]-ethylamine 377594 4-(4-(1H-pyrazol-4-yl)phenyl)-4-(4-chlorophenyl)piperidine 377595 (R)-2-(4-Chloro-phenyl)-2-[4-(1H-pyrazol-4-yl)-phenyl]-ethylamine 377596 (S)-2-(4-chloro-phenyl)-2-[4-(1H-pyrazol-4-yl)-phenyl]-ethylamine 377613 [D-Ncy(2-naphthyl)1]acyline 377614 [Ncy(2-naphthyl)1]acyline 377615 [Ncy(methyl)4]acyline 377616 [Ncy(SO,methyl)4]acyline 377617 [D-Ncy(methyl)4]acyline 377618 [D-Ncy(SO,methyl)4]acyline 377619 [Ncy(isopropyl)7]acyline 377620 [Ncy(SO,isopropyl)7]acyline 377621 [D-Ncy(isopropyl)7]acyline 377622 [D-Ncy(SO,isopropyl)7]acyline 377637 Ac-Nle4-cyclo(Asp5-His6-L-Phe-Pro8-Trp9-Lys10)-NH2 377675 [Ncy(methyl)10]acyline 377682 [Ncy(SO,methyl)10]acyline 377683 [D-Ncy(methyl)10] acyline 377685 [D-Ncy(SO,methyl)10]acyline 377686 [D-Gln3,Ncy(isopropyl)7]acyline 377687 [D-Gln3,Ncy(SO,isopropyl)7]acyline 377688 [D-Gln3,Ncy(SO2,isopropyl)7]acyline 377689 [D-Gln3,D-Ncy(isopropyl)7]acyline 377690 [D-Gln3,D-Ncy(SO,isopropyl)7]acyline 377691 [D-Gln3,D-Ncy(SO2,isopropyl)7]acyline 377696 (4-(9H-purin-6-yl)phenyl)-N-methylmethanamine 377702 (3-(9H-purin-6-yl)phenyl)-N-methylmethanamine 377703 2-(4-(9H-purin-6-yl)phenyl)ethanamine 377704 2-(3-(9H-purin-6-yl)phenyl)ethanamine 377709 (4-(9H-purin-6-yl)phenyl)(phenyl)methanamine 377808 Ac-Nle4-cyclo(Asp5-His6-D-Phe(No2)-Pro8-Trp9-Lys10)-NH2 377811 Ac-Nle4-cyclo(Asp5-His6-D-Phe(4-Cl)-Pro8-Trp9-Lys10)-NH2 377812 Ac-Nle4-cyclo(Asp5-His6-D-Bth-Pro8-Trp9-Lys10)-NH2 377813 Ac-Nle4-cyclo(Asp5-His6-D-4,4'-Bip-Pro8-Trp9-Lys10)-NH2 377848 Ac-Nle4-cyclo(Asp5-His6-D-Phe-Pro8-Trp9-Lys10)-NH2 377849 Ac-Nle4-cyclo(Asp5-His6-D-Nal(2)-Pro8-Trp9-Lys10)-NH2 377850 Ac-Nle4-cyclo(Asp5-His6-D-Tyr-Pro8-Trp9-Lys10)-NH2 377853 Ac-Nle4-cyclo(Asp5-His6-D-Tyr(Me)-Pro8-Trp9-Lys10)-NH2 377854 Ac-Nle4-cyclo(Asp5-His6-D-Tyr(Et)-Pro8-Trp9-Lys10)-NH2 377859 3-(2-fluorobenzyl)-N-methyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377860 3-(2-fluorobenzyl)-N-ethyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377868 3-(2-fluorobenzyl)-5-phenyl-N-propyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377869 3-(2-fluorobenzyl)-N-butyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377877 3-(2-fluorobenzyl)-N-hexyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377879 3-(2-fluorobenzyl)-N-cyclopropyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377887 3-(2-fluorobenzyl)-N-cyclopentyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377888 3-(2-fluorobenzyl)-N-cyclohexyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377897 2-(3-(2-fluorobenzyl)-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-ylamino)ethanol 377898 1-(3-(2-fluorobenzyl)-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-ylamino)propan-2-ol 377903 3-benzyl-N-methyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377904 3-(3-(2-fluorobenzyl)-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-ylamino)propan-1-ol 377905 3-(2-(trifluoromethyl)benzyl)-N-methyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377908 3-benzyl-N-ethyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377909 3-benzyl-5-phenyl-N-propyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377915 3-benzyl-N-butyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377916 3-benzyl-N-hexyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377917 3-(2-(trifluoromethyl)benzyl)-N-butyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377924 3-benzyl-N-cyclopropyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377925 3-benzyl-N-cyclobutyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377926 3-(2-(trifluoromethyl)benzyl)-N-cyclopropyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377927 3-(2-(trifluoromethyl)benzyl)-N-cyclopentyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377937 3-benzyl-N-cyclopentyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377938 3-benzyl-N-cyclohexyl-5-phenyl-3H-[1,2,3]triazolo[4,5-b]pyridin-7-amine 377939 3-(2-(trifluoromethyl)benzyl)-N-cyclohexyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377946 2-(3-benzyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-ylamino)ethanol 377947 1-(3-benzyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-ylamino)propan-2-ol 377949 3-(3-(2-(trifluoromethyl)benzyl)-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-ylamino)propan-1-ol 377953 3-(3-benzyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-ylamino)propan-1-ol 377954 3-(2-chlorobenzyl)-N-methyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377955 2-(3-(2-chlorobenzyl)-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-ylamino)ethanol 377956 1-(3-(2-chlorobenzyl)-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-ylamino)propan-2-ol 377961 3-(2-chlorobenzyl)-N-ethyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377962 3-(2-chlorobenzyl)-5-phenyl-N-propyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377963 3-(3-(2-chlorobenzyl)-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-ylamino)propan-1-ol 377971 3-(2-chlorobenzyl)-N-butyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377972 3-(2-chlorobenzyl)-N-hexyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377980 3-(2-chlorobenzyl)-N-cyclopropyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377981 3-(2-chlorobenzyl)-N-cyclobutyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377988 3-(2-chlorobenzyl)-N-cyclopentyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 377989 3-(2-chlorobenzyl)-N-cyclohexyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine 378538 4'-(furan-2-yl)-N-(pyridin-3-yl)-4,5'-bipyrimidin-2'-amine 378539 4'-(2-furyl)-N-pyrimidin-5-yl-4,5'-bipyrimidin-2'-amine 378540 4'-(2-furyl)-N-pyrazin-2-yl-4,5'-bipyrimidin-2'-amine 378541 4'-(2-furyl)-N-(6-methoxypyridin-3-yl)-4,5'-bipyrimidin-2'-amine 378542 4'-(2-furyl)-N-(2-methoxypyrimidin-5-yl)-4,5'-bipyrimidin-2'-amine 378543 5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}nicotinonitrile 378544 4'-(2-furyl)-N-(1-oxidopyridin-3-yl)-4,5'-bipyrimidin-2'-amine 378546 5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}pyridin-2(1H)-one 378547 5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}-1-methylpyridin-2(1H)-one 378548 1-(cyclopropylmethyl)-5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}pyridin-2(1H)-one 378588 N-(3,5-bis(trifluoromethyl)benzyl)-3-(4-phenylpiperidin-1-yl)cyclopentanecarboxamide 378593 cis-(1S,3R)-N-(3,5-bis(trifluoromethyl)benzyl)-3-(4-phenylpiperidin-1-yl)cyclopentanecarboxamide 378601 (1S,3R)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-3-{spiro[indene-1,4'-piperidine]-1'-yl}cyclopentane-1-carboxamide 378603 (1S,3R)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-3-[(1R,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]cyclopentane-1-carboxamide 378605 (1S,3R)-N-[3,5-bis(trifluoromethyl)benzyl]-1-methyl-3-[(1R,3'R)-methyl-1'H-spiro[indene-1,4'-piperidin]-1'-yl]cyclopentanecarboxamide 378609 (1S,3R)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-1-methyl-3-{spiro[indene-1,4'-piperidine]-1'-yl}cyclopentane-1-carboxamide 378628 2-(pyridin-4-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 378630 2-(2-chloropyridin-4-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 378631 2-(2-phenylpyridin-4-yl)-1,5,6,7-tetrahydro-4H-pyrrolo[3,2- 378633 2-(2,4'-bipyridin-4-yl)-1,5,6,7-tetrahydro-4H-pyrrolo[3,2-c]-pyridin-4-one 378636 2-(2,3'-bipyridin-4-yl)-1,5,6,7-tetrahydro-4H-pyrrolo[3,2-c]-pyridin-4-one 378639 2-(2-pyrimidin-5-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4H-pyrrolo[3,2-c]pyridin-4-one 378644 2-(2-thien-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4H-pyrrolo-[3,2-c]pyridin-4-one 378646 2-[2-(2-naphthyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4H-pyrrolo-[3,2-c]pyridin-4-one 378648 2-[2-(1-benzothien-2-yl)pyridin-4-yl]-1,5,6,7-tetrahydro-4Hpyrrolo[3,2-c]pyridin-4-one 378650 2-(2-(quinolin-3-yl)pyridin-4-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 378653 2-[2-(2-hydroxyphenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4Hpyrrolo[3,2-c]pyridin-4-one 378654 2-[2-(3-hydroxyphenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4Hpyrrolo[3,2-c]pyridin-4-one 378656 2-[2-(4-hydroxyphenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4Hpyrrolo[3,2-c]pyridin-4-one 378657 2-[2-(2-chlorophenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4Hpyrrolo[3,2-c]pyridin-4-one 378659 2-[2-(3-chlorophenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4Hpyrrolo[3,2-c]pyridin-4-one 378662 2-[2-(4-chlorophenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4Hpyrrolo[3,2-c]pyridin-4-one 378664 2-[2-(2-fluorophenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4H-pyrrolo[3,2-c]pyridin-4-one 378665 2-[2-(3-fluorophenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4H-pyrrolo[3,2-c]pyridin-4-one 378667 2-[2-(4-fluorophenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4H-pyrrolo[3,2-c]pyridin-4-one 378668 2-{2-[4-(trifluoromethyl)phenyl]pyridin-4-yl}-1,5,6,7-tetrahydro-4H-pyrrolo[3,2-c]pyridin-4-one 378670 4-[4-(4-oxo-4,5,6,7-tetrahydro-1H-pyrrolo[3,2-c]pyridin-2-yl)-pyridin-2-yl]benzonitrile 378672 2-[2-(4-acetylphenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4H-pyrrolo[3,2-c]pyridin-4-one 378673 2-[2-(4-methoxyphenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4Hpyrrolo[3,2-c]pyridin-4-one 378675 2-[2-(4-aminophenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4H-pyrrolo[3,2-c]pyridin-4-one 378677 4-[4-(4-oxo-4,5,6,7-tetrahydro-1H-pyrrolo[3,2-c]pyridin-2-yl)-pyridin-2-yl]benzoic acid 378679 N-cyclopropyl-4-[4-(4-oxo-4,5,6,7-tetrahydro-1H-pyrrolo[3,2-c]pyridin-2-yl)pyridin-2-yl]benzamide 378680 N-cyclopentyl-4-[4-(4-oxo-4,5,6,7-tetrahydro-1H-pyrrolo[3,2-c]pyridin-2-yl)pyridin-2-yl]benzamide 378682 N-cyclohexyl-4-[4-(4-oxo-4,5,6,7-tetrahydro-1H-pyrrolo[3,2-c]pyridin-2-yl)pyridin-2-yl]benzamide 378684 N-benzyl-4-[4-[4-oxo-4,5,6,7-tetrahydro-1H-pyrrolo[3,2-c]pyridin-2-yl]benzamide 378685 4-(4-(4,5,6,7-tetrahydro-4-oxo-1H-pyrrolo[3,2-c]pyridin-2-yl)pyridin-2-yl)-N-phenethylbenzamide 378688 N-benzyl-4-(4-(4,5,6,7-tetrahydro-4-oxo-1H-pyrrolo[3,2-c]pyridin-2-yl)-N-methylbenzamide 378898 (+/-)-1-[2-(4-fluorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]-4-(1-naphthylmethyl)piperazine 378899 (+/-)-1-[2-(4-fluorophenyl)-2-(4-methylpiperazin-1-yl)-ethyl]-4-[2-(1-naphthyl)ethyl]piperazine 378900 1-[2-(4-fluorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]-4-[3-(1-naphthyl)propyl]piperazine 378901 (+/-)-1-[2-(4-fluorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]-4-[4-(1-naphthyl)butyl]piperazine 378905 (+/-)-1-[2-(4-fluorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]-4-[5-(1-naphthyl)pentyl]piperazine 378906 (+/-)-1-[2-(4-fluorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]-4-[6-(1-naphthyl)hexyl]piperazine 378907 (+/-)-1-[2-(4-fluorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]-4-(2-naphthylmethyl)piperazine 378908 (+/-)-1-[2-(4-fluorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]-4-[2-(2-naphthyl)ethyl]piperazine 378909 (+/-)-1-[2-(4-fluorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]-4-[3-(2-naphthyl)propyl]piperazine 378910 (+/-)-1-[2-(4-fluorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]-4-[4-(2-naphthyl)butyl]piperazine 378911 (+/-)-1-[2-(4-fluorophenyl)-2-piperazin-1-ylethyl]-4-[4-(1-naphthyl)butyl]piperazine 378912 (+/-)-1-ethyl-4-(1-(4-fluorophenyl)-2-{4-[4-(1-naphthyl)butyl]piperazin-1-yl}ethyl)piperazine 378913 (+/-)-1-(1-(4-fluorophenyl)-2-{4-[4-(1-naphthyl)butyl]piperazin-1-yl}ethyl)-4-propylpiperazine 378914 (+/-)-1-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]-4-[4-(1-naphthyl)butyl]piperazine 378915 (+/-)-1-cyclopropyl-4-(1-(4-fluorophenyl)-2-{4-[4-(1-naphthyl)butyl]piperazin-1-yl}ethyl)piperazine 378916 (+/-)-1-cyclohexyl-4-(1-(4-fluorophenyl)-2-{4-[4-(1-naphthyl)butyl]piperazin-1-yl}ethyl)piperazine 378918 (+/-)-1-methyl-4-(2-{4-[4-(1-naphthyl)butyl]piperazin-1-yl}-1-phenylethyl)piperazine 378919 (+/-)-1-[2-(3-fluorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]-4-[4-(1-naphthyl)butyl]piperazine 378920 (+/-)-1-[2-(4-chlorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]-4-[4-(1-naphthyl)butyl]piperazine 378921 (+/-)-1-[2-(2-bromophenyl)-2-(4-methylpiperazin-1-yl)ethyl]-4-[4-(1-naphthyl)butyl]piperazine 378922 (+-)-1-[2-(3-bromophenyl)-2-(4-methylpiperazin-1-yl)ethyl]-4-[4-(1-naphthyl)butyl]piperazine 378923 (+/-)-1-[2-(4-bromophenyl)-2-(4-methylpiperazin-1-yl)ethyl]-4-[4-(1-naphthyl)butyl]piperazine 378924 (+/-)-1-methyl-4-(1-(4-methylphenyl)-2-{4-[4-(1-naphthyl)butyl]piperazin-1-yl}ethyl)piperazine 378925 (+/-)-1-[2-(4-methoxyphenyl)-2-(4-methylpiperazin-1-yl)ethyl]-4-[4-(1-naphthyl)butyl]piperazine 378926 (+/-)-1-methyl-4-{2-{4-[4-(1-naphthyl)butyl]piperazin-1-yl}-1-[4-(trifluoromethyl)phenyl]ethyl}piperazine 378927 (+/-)-1-methyl-4-[2-{4-[4-(1-naphthyl)butyl]piperazin-1-yl}-1-(4-nitrophenyl)ethyl]piperazine 378928 (+/-)-1-[2-biphenyl-4-yl-2-(4-methylpiperazin-1-yl)ethyl]-4-[4-(1-naphthyl)butyl]piperazine 378929 (+/-)-4-(1-(4-methylpiperazin-1-yl)-2-{4-[4-(1-naphthyl)butyl]piperazin-1-yl}ethyl)aniline 378930 (+/-)-1-[4-(2-bromo-1-naphthyl)butyl]-4-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]piperazine 378931 (+/-)-1-(1-(4-fluorophenyl)-2-{4-[4-(4-methoxy-1-naphthyl)butyl]piperazin-1-yl}ethyl)-4-methylpiperazine 378932 (+/-)-1-(4-{4-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]piperazin-1-yl}butyl)-2-naphthol 378933 (+/-)-1-[4-(2-ethoxy-1-naphthyl)butyl]-4-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]piperazine 378934 1-(1-(4-fluorophenyl)-2-{4-[4-(2-isopropoxy-1-naphthyl)butyl]piperazin-1-yl}ethyl)-4-isopropylpiperazine 378935 (+/-)-1-(1-ethylpropyl)-4-(1-(4-fluorophenyl)-2-{4-[4-(2-methoxy-1-naphthyl)butyl]piperazin-1-yl}ethyl)piperazine 378936 (+/-)-1-cyclopentyl-4-(1-(4-fluorophenyl)-2-{4-[4-(2-methoxy-1-naphthyl)butyl]piperazin-1-yl}ethyl)piperazine 378937 (+/-)-1-tert-butyl-4-(1-(4-fluorophenyl)-2-{4-[4-(2-methoxy-1-naphthyl)butyl]piperazin-1-yl}ethyl)piperazine 378938 (+/-)-1-(2-biphenyl-2-ylethyl)-4-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]piperazine 378939 (+/-)-1-(3-biphenyl-2-ylpropyl)-4-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]piperazine 378940 (+/-)-1-(4-biphenyl-2-ylbutyl)-4-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]piperazine 378941 (+/-)-1-(3-biphenyl-3-ylpropyl)-4-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]piperazine 378942 (+/-)-1-(3-biphenyl-4-ylpropyl)-4-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]piperazine 378943 (+/-)-1-[3-(6-fluorobiphenyl-2-yl)propyl]-4-[2-(4-fluorophenyl)-2-4-isopropylpiperazin-1-yl)ethyl]piperazine 378944 (+/-)-1-[3-(5-fluorobiphenyl-2-yl)propyl]-4-[2-(4-fluorophenyl)-2-4-isopropylpiperazin-1-yl)ethyl]piperazine 378945 (+/-)-1-[3-(4-fluorobiphenyl-2-yl)propyl]-4-[2-(4-fluorophenyl)-2-4-isopropylpiperazin-1-yl)ethyl]piperazine 378946 (+/-)-1-[3-(3-fluorobiphenyl-2-yl)propyl]-4-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]piperazine 378947 (+/-)-1-[3-(3-chlorobiphenyl-2-yl)propyl]-4-[2-(4-fluorophenyl)-2-4-isopropylpiperazin-1-yl)ethyl]piperazine 378948 (+/-)-1-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]-4-[3-(3-methylbiphenyl-2-yl)propyl]piperazine 378949 (+/-)-1-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]-4-[3-(3-methoxybiphenyl-2-yl)propyl]piperazine 378950 (+/-)-1-[3-(2'-fluorobiphenyl-2-yl)propyl]-4-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]piperazine 378951 (+/-)-1-[3-(3'-fluorobiphenyl-2-yl)propyl]-4-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]piperazine 378952 (+/-)-1-[3-(4'-fluorobiphenyl-2-yl)propyl]-4-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]piperazine 378953 (+/-)-1-[3-(4'-chlorobiphenyl-2-yl)propyl]-4-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]piperazine 378954 (+/-)-1-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]-4-[3-(40-methylbiphenyl-2-yl)propyl]piperazine 378955 (+/-)-1-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]-4-[3-(40-methoxybiphenyl-2-yl)propyl]piperazine 378956 (+/-)-1-[3-(4'-tert-Butylbiphenyl-2-yl)propyl]-4-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]piperazine 378957 (+/-)-1-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]-4-[3-(1,1':4',1''-terphenyl-2-yl)propyl]piperazine 378958 (+/-)-1-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]-4-{3-[4'-(trifluoromethyl)biphenyl-2-yl]propyl}-piperazine 378959 (+/-)-1-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]-4-{3-[4'-(trifluoromethoxy)biphenyl-2-yl]propyl}-piperazine 378960 (+/-)-2'-(3-{4-[2-(4-fluorophenyl)-2-(4-isopropylpiperazin-1-yl)ethyl]piperazin-1-yl}propyl)-N,N-dimethylbiphenyl-4-amine 379003 1-{4-[(3-chlorophenyl)amino-6-quinazolinyl}-3-{2-[N-(2-chloroethyl)-N-methylethylenamine]}triazene 379004 1-{4-[(3-chlorophenyl)amino-6-quinazolinyl}-3-{2-[N-(2-chloroethyl)-N-benzylethylenamine]}triazene 379005 1-{4-[(3-chlorophenyl)amino-6-quinazolinyl}-3-{2-[N-(2-chloroethyl)-N-4-methoxyphenylethylenamine]} triazene 379006 1-{4-[(3-chlorophenyl)amino-6-quinazolinyl}-3-{2-[N-(2-chloroethyl)-N-4-chlorophenylethylenamine]} triazene 379007 N-(3-chlorophenyl)-6-(3-(2-(dimethylamino)ethyl)triaz-1-enyl)quinazolin-4-amine 379008 1-{4-[(3-chlorophenyl)amino-6-quinazolinyl}-3-{2-[N-(2-chloropropyl)-N-4-methoxyphenylethylenamine]} triazene 379037 (1S,13R,14R)-19-methoxy-24-methyl-4,24-diazahexacyclo[12.7.3.0^{1,13}.0^{3,11}.0^{5,10}.0^{16,21}]tetracosa-3(11),5(10),6,8,16(21),17,19-heptaene 379038 (1S,13R,14R)-24-(cyclopropylmethyl)-19-methoxy-4,24-diazahexacyclo[12.7.3.0^{1,13}.0^{3,11}.0^{5,10}.0^{16,21}]tetracosa-3(11),5(10),6,8,16(21),17,19-heptaene 379039 (1S,13R,14R)-24-(cyclobutylmethyl)-19-methoxy-4,24-diazahexacyclo[12.7.3.0^{1,13}.0^{3,11}.0^{5,10}.0^{16,21}]tetracosa-3(11),5(10),6,8,16(21),17,19-heptaene 379040 (1S,13R,14R)-24-methyl-4,24-diazahexacyclo[12.7.3.0^{1,13}.0^{3,11}.0^{5,10}.0^{16,21}]tetracosa-3(11),5(10),6,8,16(21),17,19-heptaen-19-ol 379041 (1S,13R,14R)-24-(cyclopropylmethyl)-4,24-diazahexacyclo[12.7.3.0^{1,13}.0^{3,11}.0^{5,10}.0^{16,21}]tetracosa-3(11),5(10),6,8,16(21),17,19-heptaen-19-ol 379042 (1S,13R,14R)-24-(cyclobutylmethyl)-4,24-diazahexacyclo[12.7.3.0^{1,13}.0^{3,11}.0^{5,10}.0^{16,21}]tetracosa-3(11),5(10),6,8,16(21),17,19-heptaen-19-ol 379043 (1S,9R,10R)-5-amino-20-methyl-6-thia-4,20-diazapentacyclo[8.7.3.0^{1,9}.0^{3,7}.0^{12,17}]icosa-3(7),4,12(17),13,15-pentaen-15-ol 379044 (1S,9R,10R)-5-amino-20-(cyclopropylmethyl)-6-thia-4,20-diazapentacyclo[8.7.3.0^{1,9}.0^{3,7}.0^{12,17}]icosa-3(7),4,12(17),13,15-pentaen-15-ol 379045 (1S,9R,10R)-5-amino-20-(cyclobutylmethyl)-6-thia-4,20-diazapentacyclo[8.7.3.0^{1,9}.0^{3,7}.0^{12,17}]icosa-3(7),4,12(17),13,15-pentaen-15-ol 379241 (S,R)-(-)-{4-[2-{[2-(3-bromoisoxazol-5-yl)-2-hydroxyethyl]-amino}propyl]phenoxy}acetic acid 379242 (R,R)-(+)-{4-[2-{[2-(3-bromoisoxazol-5-yl)-2-hydroxyethyl]-amino}propyl]phenoxy}acetic acid 379245 (S,R)-(-)-ethyl {4-[2-{[2-(3-bromoisoxazol-5-yl)-2-hydroxyethyl]amino}propyl]phenoxy} acetate 379246 (R,R)-(+)-ethyl {4-[2-{[2-(3-bromoisoxazol-5-yl)-2-hydroxyethyl]amino}propyl]phenoxy} acetate 379247 (S,R)-(-)-1-(3-bromoisoxazol-5-yl)-2-{[2-(4-butoxyphenyl)-1-methylethyl]amino}ethanol 379248 (R,R)-(+)-1-(3-bromoisoxazol-5-yl)-2-{[2-(4-butoxyphenyl)-1-methylethyl]amino}ethanol 379356 (S)-1-(5-(1H-indazol-5-yl)pyridin-3-yloxy)-3-(1H-indol-3-yl)propan-2-amine 379357 (S)-1-(5-(3-chloro-1H-indazol-5-yl)pyridin-3-yloxy)-3-(1H-indol-3-yl)propan-2-amine 379358 (S)-1-(1H-indol-3-yl)-3-(5-(3-(trifluoromethyl)-1H-indazol-5-yl)pyridin-3-yloxy)propan-2-amine 379359 (S)-1-(1H-indol-3-yl)-3-(5-(6-nitro-1H-indazol-5-yl)pyridin-3-yloxy)propan-2-amine 379360 (S)-5-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)-1H-indazol-6-amine 379361 (S)-5-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin-3-yl)-3-chloro-1H-indazol-6-amine 379362 (S)-1-(5-(1H-pyrazolo[3,4-c]pyridin-5-yl)pyridin-3-yloxy)-3-(1H-indol-3-yl)propan-2-amine 379363 (S)-1-(1H-indol-3-yl)-3-(5-(3-methyl-1H-pyrazolo[3,4-c]pyridin-5-yl)pyridin-3-yloxy)propan-2-amine 379364 (S)-1-(5-(1H-pyrazolo[3,4-c]pyridin-5-yl)pyridin-3-yloxy)-3-phenylpropan-2-amine 379365 (S)-1-(5-(3-methyl-1H-pyrazolo[3,4-c]pyridin-5-yl)pyridin-3-yloxy)-3-phenylpropan-2-amine 379366 (S)-1-(5-(3-chloro-1H-pyrazolo[3,4-c]pyridin-5-yl)pyridin-3-yloxy)-3-phenylpropan-2-amine 379367 (S)-5-(5-(2-amino-3-phenylpropoxy)pyridin-3-yl)-3-methyl-1H-pyrazolo[3,4-c]pyridine 6-oxide 379368 (S)-1-phenyl-3-(5-(3-vinyl-1H-pyrazolo[3,4-c]pyridin-5-yl)pyridin-3-yloxy)propan-2-amine 379369 (S)-1-(5-(3-(furan-2-yl)-1H-pyrazolo[3,4-c]pyridin-5-yl)pyridin-3-yloxy)-3-phenylpropan-2-amine 379370 (2S)-1-(5-(3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazolo[3,4-c]pyridin-5-yl)pyridin-3-yloxy)-3-phenylpropan-2-amine 379371 (S)-1-phenyl-3-(5-(3-phenyl-1H-pyrazolo[3,4-c]pyridin-5-yl)pyridin-3-yloxy)propan-2-amine 379544 (2S,3S,4R,5R)-N-ethyl-3,4-dihydroxy-5-(6-(4-(2-oxo-2-(phenylamino)ethoxy)phenylamino)-9H-purin-9-yl)-tetrahydrofuran-2-carboxamide 379545 (2S,3S,4R,5R)-N-ethyl-5-(6-(4-(2-(4-fluorophenylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 379546 (2S,3S,4R,5R)-5-(6-(4-(2-(4-chlorophenylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 379547 (2S,3S,4R,5R)-5-(6-(4-(2-(4-bromophenylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 379548 (2S,3S,4R,5R)-N-ethyl-3,4-dihydroxy-5-(6-(4-(2-(4-iodophenylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-tetrahydrofuran-2-carboxamide 379549 1-deoxy-1-[6-{4-[(2-trifluoromethyl-phenylcarbamoyl)-methoxy]-phenylamino}-9H-purin-9-yl]-N-ethyl-beta-D-ribofuranuronamide 379550 (2S,3S,4R,5R)-N-ethyl-3,4-dihydroxy-5-(6-(4-(2-(4-methoxyphenylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-tetrahydrofuran-2-carboxamide 379551 (2S,3S,4R,5R)-5-(6-(4-(2-(3,4-dimethoxyphenylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 379552 (2S,3S,4R,5R)-5-(6-(4-(2-(3,5-dimethoxyphenylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 379553 (2S,3S,4R,5R)-5-(6-(4-(2-(benzo[d][1,3]dioxol-5-ylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 379554 (2S,3S,4R,5R)-5-(6-(4-(2-(4-tert-butylphenylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 379555 (2S,3S,4R,5R)-N-ethyl-3,4-dihydroxy-5-(6-(4-(2-(4-morpholinophenylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-tetrahydrofuran-2-carboxamide 379556 (2S,3S,4R,5R)-N-ethyl-3,4-dihydroxy-5-(6-(4-(2-oxo-2-(pyridin-4-ylamino)ethoxy)phenylamino)-9H-purin-9-yl)-tetrahydrofuran-2-carboxamide 379557 (2S,3S,4R,5R)-5-(6-(4-(2-(benzylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 379558 (2S,3S,4R,5R)-5-(6-(4-(2-(4-methoxybenzylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 379559 (2S,3S,4R,5R)-5-(6-(4-(2-(cyclohexylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 379560 (2S,3S,4R,5R)-5-(2-chloro-6-(4-(2-oxo-2-(phenylamino)ethoxy)phenylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 379561 (2S,3S,4R,5R)-5-(2-chloro-6-(4-(2-(4-methoxyphenylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 379571 (2S,3S,4R,5R)-5-(6-(4-(2-(benzylamino)-2-oxoethoxy)phenylamino)-2-chloro-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 379572 (2S,3S,4R,5R)-5-(2-chloro-6-(4-(2-(cyclohexylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 379677 SID26754275 379891 5-(4-chloro-phenyl)-6-(2,4-dichloro-phenyl)-pyrazine-2-carboxylic acid piperidin-1-ylamide 379892 6-(4-chloro-phenyl)-5-(2,4-dichloro-phenyl)-pyrazine-2-carboxylic acid piperidin-1-ylamide 379893 5,6-diphenyl-N-(piperidin-1-yl)pyrazine-2-carboxamide 379894 5,6-bis-(4-bromo-phenyl)-pyrazine-2-carboxylic acid piperidin-1-ylamide 379895 N-(piperidin-1-yl)-5,6-dip-tolylpyrazine-2-carboxamide 379896 5,6-bis(4-methoxyphenyl)-N-(piperidin-1-yl)pyrazine-2-carboxamide 379897 5,6-bis(4-chlorophenyl)-N-(piperidin-1-yl)pyrazine-2-carboxamide 379898 5,6-bis(2-chlorophenyl)-N-(piperidin-1-yl)pyrazine-2-carboxamide 379899 5,6-bis-(4-bromo-phenyl)-pyrazine-2-carboxylic acid cyclohexylamide 379900 5,6-di-p-tolyl-pyrazine-2-carboxylic acid cyclohexylamide 379901 N-cyclohexyl-5,6-bis(4-methoxyphenyl)pyrazine-2-carboxamide 379902 5,6-bis(4-chlorophenyl)-N-cyclohexylpyrazine-2-carboxamide 379903 3-(3-(2-acetamidoethyl)-5-methoxy-1H-indole-2-carbonyloxy)propyl 3-(2-acetamidoethyl)-5-methoxy-1H-indole-2-carboxylate 379904 5,6-bis-(2-chloro-phenyl)-pyrazine-2-carboxylic acid cyclohexylamide 379905 5-(3-(2-acetamidoethyl)-5-methoxy-1H-indole-2-carbonyloxy)pentyl 3-(2-acetamidoethyl)-5-methoxy-1Hindole-2-carboxylate 379906 N,5,6-triphenylpyrazine-2-carboxamide 379907 N-phenyl-5,6-dip-tolylpyrazine-2-carboxamide 379908 7-(3-(2-acetamidoethyl)-5-methoxy-1H-indole-2-carbonyloxy)heptyl 3-(2-acetamidoethyl)-5-methoxy-1Hindole-2-carboxylate 379909 8-(3-(2-acetamidoethyl)-5-methoxy-1H-indole-2-carbonyloxy)octyl 3-(2-acetamidoethyl)-5-methoxy-1Hindole-2-carboxylate 379910 5,6-bis(4-methoxyphenyl)-N-phenylpyrazine-2-carboxamide 379911 9-(3-(2-acetamidoethyl)-5-methoxy-1H-indole-2-carbonyloxy)nonyl 3-(2-acetamidoethyl)-5-methoxy-1Hindole-2-carboxylate 379912 5,6-bis-(4-chloro-phenyl)-pyrazine-2-carboxylic acid phenylamide 379913 10-(3-(2-acetamidoethyl)-5-methoxy-1H-indole-2-carbonyloxy)decyl 3-(2-acetamidoethyl)-5-methoxy-1Hindole-2-carboxylate 379914 12-(3-(2-acetamidoethyl)-5-methoxy-1H-indole-2-carbonyloxy)dodecyl 3-(2-acetamidoethyl)-5-methoxy-1Hindole-2-carboxylate 379915 5,6-bis-(2-chloro-phenyl)-pyrazine-2-carboxylic acid phenylamide 379916 pentyl 3-(2-acetamidoethyl)-5-methoxy-1Hindole-2-carboxylate 379917 9-(benzoyloxy)nonyl 3-(2-acetamidoethyl)-5-methoxy-1H-indole-2-carboxylate 379918 N1,N7-bis(2-(5-methoxy-1H-indol-3-yl)ethyl)heptanediamide 379919 N1,N10-bis(2-(5-methoxy-1H-indol-3-yl)ethyl)decanediamide 379995 (S)-1-(6-((diethylamino)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)-4-phenethylpiperazin-2-one 379996 (S)-4-(3-fluorophenethyl)-1-(6-((diethylamino)-methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-2-one 379997 (S)-4-(2-fluorophenethyl)-1-(6-((diethylamino)-methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-2-one 379998 (S)-4-(3-chlorophenethyl)-1-(6-((diethylamino)-methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-2-one 379999 (S)-4-(2-chlorophenethyl)-1-(6-((diethylamino)-methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-2-one 380000 (S)-4-(4-bromophenethyl)-1-(6-((diethylamino)-methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-2-one 380001 (S)-4-(4-(trifluoromethyl)phenethyl)-1-(6-((diethylamino)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-2-one 380002 (S)-4-(2-(trifluoromethyl)phenethyl)-1-(6-((diethylamino)methyl)-1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-2-one 380003 4'-fluoro-biphenyl-4-carboxylic acid [2-(4-dimethylaminomethyl-phenyl)-ethyl]-amide 380004 4'-fluoro-biphenyl-4-carboxylic acid [2-(4-dimethylaminomethyl-phenyl)-ethyl]-methyl-amide 380005 N-(4'-fluoro-biphenyl-4-yl)-3-(4-piperidin-1-ylmethyl-phenyl)-propionamide 380006 (4'-fluoro-biphenyl-4-ylmethyl)-[2-(4-piperidin-1-ylmethyl-phenyl)-ethyl]-amine 380007 1-(4-(piperidin-1-ylmethyl)phenethyl)-4-(2-(4-trifluoromethylphenyl)acetyl) piperazin-2-one 380008 8-(3-hydroxy-5-pentyl-phenoxy)-octanoic acid (2-hydroxy-ethyl)-amide 380009 8-(3-hydroxy-5-pentyl-phenoxy)-octanoic acid cyclopropylamide 380010 11-(3-hydroxy-5-pentyl-phenoxy)-undecanoic acid cyclopropylmethyl-amide 380011 11-(3-hydroxy-5-pentyl-phenoxy)-undecanoic acid [2-(3,4-dihydroxy-phenyl)-ethyl]-amide 380012 11-(3-hydroxy-5-pentyl-phenoxy)-undecanoic acid (3-methoxy-4-hydroxy-phenyl)-amide 380013 12-(3-hydroxy-5-pentyl-phenoxy)-dodecanoic acid(2-hydroxy-ethyl)-amide 380014 12-(3-hydroxy-5-pentyl-phenoxy)-dodecanoic acidcyclopropylamide 380015 8-(2-hexyl-5-hydroxy-phenoxy)-octanoic acid (2-hydroxy-ethyl)-amide 380016 8-(2-hexyl-5-hydroxy-phenoxy)-octanoic acidcyclopropylamide 380017 11-(2-hexyl-5-hydroxy-phenoxy)-undecanoic acidcyclopropylmethyl-amide 380018 11-(2-hexyl-5-hydroxy-phenoxy)-undecanoic acid[2-(3,4-dihydroxy-phenyl)-ethyl]-amide 380019 11-(2-hexyl-5-hydroxy-phenoxy)-undecanoic acid(3-methoxy-4-hydroxy-phenyl)-amide 380020 12-(2-hexyl-5-hydroxy-phenoxy)-dodecanoic acid(2-hydroxy-ethyl)-amide 380021 12-(2-hexyl-5-hydroxy-phenoxy)-dodecanoic acidcyclopropylamide 380022 8-(4-hexyl-3-hydroxy-phenoxy)-octanoic acid (2-hydroxy-ethyl)-amide 380023 8-(4-hexyl-3-hydroxy-phenoxy)-octanoic acidcyclopropylamide 380024 11-(4-hexyl-3-hydroxy-phenoxy)-undecanoic acid cyclopropylmethyl-amide 380028 12-(4-hexyl-3-hydroxy-phenoxy)-dodecanoic acidcyclopropylamide 380029 N-cyclopropyl-11-(3-hydroxy-4-pentylphenoxy)undecanamide 380143 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-((R)-3-hydroxypyrrolidin-1-yl)ethyl)-3-phenylurea 380144 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-3-(2-fluorophenyl)-1-(2-((R)-3-hydroxypyrrolidin-1-yl)ethyl)urea 380145 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-3-(3-fluorophenyl)-1-(2-((R)-3-hydroxypyrrolidin-1-yl)ethyl)urea 380146 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-((R)-3-hydroxypyrrolidin-1-yl)ethyl)-3-(3-methoxyphenyl)urea 380147 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-3-(4-fluorophenyl)-1-(2-((R)-3-hydroxypyrrolidin-1-yl)ethyl)urea 380148 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-3-(3,5-difluorophenyl)-1-(2-((R)-3-hydroxypyrrolidin-1-yl)ethyl)urea 380149 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-3-(3,4-difluorophenyl)-1-(2-((R)-3-hydroxypyrrolidin-1-yl)ethyl)urea 380150 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-3-(3-fluoro-4-methylphenyl)-1-(2-((R)-3-hydroxypyrrolidin-1-yl)ethyl)urea 380151 3-(benzo[d][1,3]dioxol-5-yl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-((R)-3-hydroxypyrrolidin-1-yl)ethyl)urea 380152 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-3-(3,5-dimethylphenyl)-1-(2-((R)-3-hydroxypyrrolidin-1-yl)ethyl)urea 380153 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-3-cyclohexyl-1-(2-((R)-3-hydroxypyrrolidin-1-yl)ethyl)urea 380154 3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-(2-methylpyrrolidin-1-yl)ethyl)urea 380155 1-(2-(3-acetamidopyrrolidin-1-yl)ethyl)-3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)urea 380156 3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-((R)-2-(hydroxymethyl)pyrrolidin-1-yl)ethyl)urea 380157 3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-((S)-2-(hydroxymethyl)pyrrolidin-1-yl)ethyl)urea 380158 3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-(2-methylpiperidin-1-yl)ethyl)urea 380159 3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-(3-(hydroxymethyl)piperidin-1-yl)ethyl)urea 380160 3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-(4-hydroxypiperidin-1-yl)ethyl)urea 380161 3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-morpholinoethyl)urea 380162 1-(2-(azepan-1-yl)ethyl)-3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)urea 380163 3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-(ethyl(2-hydroxyethyl)amino)ethyl)urea 380164 3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-(diisopropylamino)ethyl)urea 380165 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-(diisopropylamino)ethyl)-3-(3-nitrophenyl)urea 380166 3-(3-bromophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-(diisopropylamino)ethyl)urea 380167 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-(diisopropylamino)ethyl)-3-(3-fluorophenyl)urea 380168 3-(3-chlorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-(diisopropylamino)ethyl)urea 380169 3-(3-cyanophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-(diisopropylamino)ethyl)urea 380170 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-3-(3,5-difluorophenyl)-1-(2-(diisopropylamino)ethyl)urea 380171 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-3-(3,4-difluorophenyl)-1-(2-(diisopropylamino)ethyl)urea 380172 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-(diisopropylamino)ethyl)-3-(4-fluorophenyl)urea 380173 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-3-(2,6-dichloropyridin-4-yl)-1-(2-(diisopropylamino)ethyl)urea 380174 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-((R)-3-hydroxypyrrolidin-1-yl)ethyl)-3-(3-nitrophenyl)urea 380175 3-(3-bromophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-((R)-3-hydroxypyrrolidin-1-yl)ethyl)urea 380176 3-(3-chlorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-((R)-3-hydroxypyrrolidin-1-yl)ethyl)urea 380177 3-(3-cyanophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-((R)-3-hydroxypyrrolidin-1-yl)ethyl)urea 380178 3-(3,4-difluorophenyl)-1-(2-(diisopropylamino)ethyl)-1-((3R,6S)-6-phenylbicyclo[4.1.0]heptan-3-yl)urea 380179 1-((3R,6S)-6-(3-bromophenyl)bicyclo[4.1.0]heptan-3-yl)-3-(3,4-difluorophenyl)-1-(2-(diisopropylamino)ethyl)urea 380180 1-((3R,6S)-6-(3-carbamoylphenyl)bicyclo[4.1.0]heptan-3-yl)-3-(3-chloro-4-fluorophenyl)-1-(2-(diisopropylamino)ethyl)urea 380181 methyl 3-((1S,4R)-4-(3-(3,4-difluorophenyl)-1-(2-(diisopropylamino)ethyl)ureido)bicyclo[4.1.0]heptan-1-yl)benzoate 380182 3-(3-chloro-4-fluorophenyl)-1-(2-(diisopropylamino)ethyl)-1-((3R,6S)-6-(3-(hydroxymethyl)phenyl)bicyclo[4.1.0]heptan-3-yl)urea 380183 3-(3-chloro-4-fluorophenyl)-1-(2-(diisopropylamino)ethyl)-1-((3R,6S)-6-(3-((E)-(methoxyimino)methyl)phenyl)bicyclo[4.1.0]heptan-3-yl)urea 380184 3-(3-chloro-4-fluorophenyl)-1-(2-(diisopropylamino)ethyl)-1-((3R,6S)-6-(3-((E)-(ethoxyimino)methyl)phenyl)bicyclo[4.1.0]heptan-3-yl)urea 380186 3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-((2-hydroxyethyl)(isopropyl)amino)ethyl)urea 380187 3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-(((R)-1-hydroxypropan-2-yl)(isopropyl)amino)ethyl)urea 380189 3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-(((S)-1-hydroxypropan-2-yl)(isopropyl)amino)ethyl)urea 380190 3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-((2-fluoroethyl)(isopropyl)amino)ethyl)urea 380191 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-3-(2,6-dichloropyridin-4-yl)-1-(2-((2-hydroxyethyl)(isopropyl)amino)ethyl)urea 380192 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-3-(2,6-dichloropyridin-4-yl)-1-(2-(((S)-1-hydroxypropan-2-yl)(isopropyl)amino)ethyl)urea 380193 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-3-(2,6-dichloropyridin-4-yl)-1-(2-((2-fluoroethyl)(isopropyl)amino)ethyl)urea 380194 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-3-(2,6-dichloropyridin-4-yl)-1-(2-(isopropylamino)ethyl)urea 380195 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-3-(2,6-dichloropyridin-4-yl)-1-(2-(2-fluoroethylamino)ethyl)urea 380196 3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-((2S)-2-(hydroxymethyl)-5-methylpyrrolidin-1-yl)ethyl)urea 380197 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-3-(2,6-dichloropyridin-4-yl)-1-(2-((2S)-2-(hydroxymethyl)-5-methylpyrrolidin-1-yl)ethyl)urea 380203 3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-((1-(tetrahydro-2H-pyran-4-yl)piperidin-4-yl)methyl)urea 380204 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-3-(4-fluoro-3-(trifluoromethyl)phenyl)-1-((1-(methylcarbamoyl)piperidin-4-yl)methyl)urea 380207 1-((1-acetylpiperidin-4-yl)methyl)-3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)urea 380208 3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-((1-(methylsulfonyl)piperidin-4-yl)methyl)urea 380210 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-3-(3,4-difluorophenyl)-1-((1-(methylsulfonyl)piperidin-4-yl)methyl)urea 380211 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-3-(3,4-difluorophenyl)-1-((1-(ethylsulfonyl)piperidin-4-yl)methyl)urea 380212 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-3-(4-fluoro-3-(trifluoromethyl)phenyl)-1-((1-(methylsulfonyl)piperidin-4-yl)methyl)urea 380213 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-3-(3-fluorophenyl)-1-((1-(methylsulfonyl)piperidin-4-yl)methyl)urea 380214 1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-3-(4-fluoro-3-(trifluoromethyl)phenyl)-1-(2-(1-(methylsulfonyl)piperidin-4-yl)ethyl)urea 380215 3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-((1-(methylsulfonyl)piperidin-3-yl)methyl)urea 380216 3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-((1-(methylsulfonyl)piperidin-2-yl)methyl)urea 380217 3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-1-(((S)-1-(methylsulfonyl)pyrrolidin-2-yl)methyl)urea 380223 1-((3R,6S)-6-(3-(aminomethyl)phenyl)bicyclo[4.1.0]heptan-3-yl)-3-(3-chloro-4-fluorophenyl)-1-(2-(diisopropylamino)ethyl)urea 380225 3-(3-chloro-4-fluorophenyl)-1-(2-(diisopropylamino)ethyl)-1-((3R,6S)-6-(3-(methylsulfonamidomethyl)phenyl)bicyclo[4.1.0]heptan-3-yl)urea 380226 1-((3R,6S)-6-(3-(acetamidomethyl)phenyl)bicyclo[4.1.0]heptan-3-yl)-3-(3-chloro-4-fluorophenyl)-1-(2-(diisopropylamino)ethyl)urea 380228 3-(3-chloro-4-fluorophenyl)-1-(2-(diisopropylamino)ethyl)-1-((3R,6S)-6-(3-(((S)-3-hydroxypyrrolidin-1-yl)methyl)phenyl)bicyclo[4.1.0]heptan-3-yl)urea 380229 3-(3-chloro-4-fluorophenyl)-1-(2-(diisopropylamino)ethyl)-1-((3R,6S)-6-(3-((4-methylpiperazin-1-yl)methyl)phenyl)bicyclo[4.1.0]heptan-3-yl)urea 380231 3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-((diethylamino)methyl)phenyl)bicyclo[4.1.0]heptan-3-yl)-1-(2-(diisopropylamino)ethyl)urea 380232 3-(3-chloro-4-fluorophenyl)-1-(2-(diisopropylamino)ethyl)-1-((3R,6S)-6-(3-((dimethylamino)methyl)phenyl)bicyclo[4.1.0]heptan-3-yl)urea 380233 1-((3R,6S)-6-(3-(aminomethyl)phenyl)bicyclo[4.1.0]heptan-3-yl)-3-(3-chloro-4-fluorophenyl)-1-((1-(methylsulfonyl)piperidin-4-yl)methyl)urea 380234 3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-((dimethylamino)methyl)phenyl)bicyclo[4.1.0]heptan-3-yl)-1-((1-(methylsulfonyl)piperidin-4-yl)methyl)urea 380235 1-((3R,6S)-6-(3-(aminomethyl)phenyl)bicyclo[4.1.0]heptan-3-yl)-3-(2,6-dichloropyridin-4-yl)-1-((1-(methylsulfonyl)piperidin-4-yl)methyl)urea 380237 3-(2,6-dichloropyridin-4-yl)-1-((3R,6S)-6-(3-((dimethylamino)methyl)phenyl)bicyclo[4.1.0]heptan-3-yl)-1-((1-(methylsulfonyl)piperidin-4-yl)methyl)urea 380238 3-(2,6-dichloropyridin-4-yl)-1-((3R,6S)-6-(3-(((S)-3-hydroxypyrrolidin-1-yl)methyl)phenyl)bicyclo[4.1.0]heptan-3-yl)-1-((1-(methylsulfonyl)piperidin-4-yl)methyl)urea 380239 3-(3-chloro-4-fluorophenyl)-1-(4-(pyrimidin-5-yl)cyclohex-3-enyl)-1-(2-(pyrrolidin-1-yl)ethyl)urea 380240 3-(3-chloro-4-fluorophenyl)-1-(4-(pyridin-3-yl)cyclohex-3-enyl)-1-(2-(pyrrolidin-1-yl)ethyl)urea 380241 1-(4-(1H-pyrrol-2-yl)cyclohex-3-enyl)-3-(3-chloro-4-fluorophenyl)-1-(2-(pyrrolidin-1-yl)ethyl)urea 380242 3-(3-chloro-4-fluorophenyl)-1-(4-(furan-2-yl)cyclohex-3-enyl)-1-(2-(pyrrolidin-1-yl)ethyl)urea 380244 3-(3-chloro-4-fluorophenyl)-1-(4-(5-formylfuran-2-yl)cyclohex-3-enyl)-1-(2-(pyrrolidin-1-yl)ethyl)urea 380245 1-(4-(benzofuran-2-yl)cyclohex-3-enyl)-3-(3-chloro-4-fluorophenyl)-1-(2-(pyrrolidin-1-yl)ethyl)urea 380246 3-(3-chloro-4-fluorophenyl)-1-(4-(5-methylthiophen-2-yl)cyclohex-3-enyl)-1-(2-(pyrrolidin-1-yl)ethyl)urea 380247 1-(4-(5-acetylthiophen-2-yl)cyclohex-3-enyl)-3-(3-chloro-4-fluorophenyl)-1-(2-(pyrrolidin-1-yl)ethyl)urea 380248 3-(3-chloro-4-fluorophenyl)-1-(4-(5-cyanothiophen-2-yl)cyclohex-3-enyl)-1-(2-(pyrrolidin-1-yl)ethyl)urea 380249 1-(4-(5-(aminomethyl)thiophen-2-yl)cyclohex-3-enyl)-3-(3-chloro-4-fluorophenyl)-1-(2-(pyrrolidin-1-yl)ethyl)urea 380250 3-(3-chloro-4-fluorophenyl)-1-(4-(2-cyanothiazol-5-yl)cyclohex-3-enyl)-1-(2-(pyrrolidin-1-yl)ethyl)urea 380251 1-(4-(2-(aminomethyl)thiazol-5-yl)cyclohex-3-enyl)-3-(3-chloro-4-fluorophenyl)-1-(2-(pyrrolidin-1-yl)ethyl)urea 380252 3-(3-chloro-4-fluorophenyl)-1-(4-(2-((dimethylamino)methyl)thiazol-5-yl)cyclohex-3-enyl)-1-(2-(pyrrolidin-1-yl)ethyl)urea 380253 1-(4-(5-(aminomethyl)thiazol-2-yl)cyclohex-3-enyl)-3-(3-chloro-4-fluorophenyl)-1-(2-(pyrrolidin-1-yl)ethyl)urea 380840 (R,R)-(-)-fenoterol 380841 (R,S)-(-)-fenoterol 380842 (S,R)-(+)-fenoterol 380856 SID11112629 380877 (R,R)-(-)-1-p-methoxyphenyl-2-(beta-3',5'-dihydroxyphenyl-beta-oxy)ethylamino-propane 380881 (R,S)-(-)-1-p-methoxyphenyl-2-(beta-3',5'-dihydroxyphenyl-beta-oxy)ethylaminopropane 380884 (S,R)-(+)-1-p-methoxyphenyl-2-(beta-3',5'-dihydroxyphenyl-beta-oxy)ethylaminopropane 380895 (S,S)-(+)-1-p-methoxyphenyl-2-(beta-3',5'-dihydroxyphenyl-beta-oxy)ethylamino-propane 380898 (R,R)-(-)-5-{2-[2-(4-aminophenyl)-1-methylethylamino]-1-hydroxyethyl}-1,3-benzenediol 380900 (R,S)-(-)-5-{2-[2-(4-aminophenyl)-1-methylethylamino]-1-hydroxyethyl}-1,3-benzenediol 380902 (S,R)-(+)-5-{2-[2-(4-aminophenyl)-1-methylethylamino]-1-hydroxyethyl}-1,3-benzenediol 380904 (S,S)-(+)-5-{2-[2-(4-aminophenyl)-1-methylethylamino]-1-hydroxyethyl}-1,3-benzenediol 380906 (R,R)-(-)-5-[1-hydroxy-2-(1-methyl-2-phenylethylamino)ethyl]-1,3-benzenediol 380907 (R,S)-(-)-5-[1-hydroxy-2-(1-methyl-2-phenylethylamino)ethyl]-1,3-benzenediol 380908 (S,R)-(+)-5-[1-hydroxy-2-(1-methyl-2-phenylethylamino)ethyl]-1,3-benzenediol 380909 (S,S)-(+)-5-[1-hydroxy-2-(1-methyl-2-phenylethylamino)ethyl]-1,3-benzenediol 380911 (R,R)-(-)-5-{1-hydroxy-2-[1-methyl-2-(1-naphthyl)ethylamino]ethyl}-1,3-benzenediol 380912 (R,S)-(-)-5-{1-hydroxy-2-[1-methyl-2-(1-naphthyl)ethylamino]ethyl}-1,3-benzenediol 380913 (S,R)-(+)-5-{1-hydroxy-2-[1-methyl-2-(1-naphthyl)ethylamino]ethyl}-1,3-benzenediol 380914 (S,S)-(+)-5-{1-hydroxy-2-[1-methyl-2-(1-naphthyl)ethylamino]ethyl}-1,3-benzenediol 380915 (R,R)-(-)-5-[1-hydroxy-2-(1-methylhexylamino)ethyl]-1,3-benzenediol 380916 (R,S)-(-)-5-[1-hydroxy-2-(1-methylhexylamino)ethyl]-1,3-benzenediol 380917 (S,R)-(+)-5-[1-hydroxy-2-(1-methylhexylamino)ethyl]-1,3-benzenediol 380918 (S,S)-(+)-5-[1-hydroxy-2-(1-methylhexylamino)ethyl]-1,3-benzenediol 380919 (R)-(-)-5-(1-hydroxy-2-phenethylaminoethyl)-1,3-benzenediol 380920 (S)-(+)-5-(1-hydroxy-2-phenethylaminoethyl)-1,3-benzenediol 381045 7-[3-(4-phenylpiperazin-1-yl)-propyl]-8-ethoxy-1,3-dimethyl-3,7-dihydropurine-2,6-dione 381047 7-{3-[4-(2-methoxyphenyl)-piperazin-1-yl]-propyl}-8-ethoxy-1,3-dimethyl-3,7-dihydropurine-2,6-dione 381049 7-{3-[4-(3-chlorophenyl)-piperazin-1-yl]-propyl}-8-ethoxy-1,3-dimethyl-3,7-dihydropurine-2,6-dione 381050 7-[3-(4-phenylpiperazin-1-yl)-propyl]-8-propoxy-1,3-dimethyl-3,7-dihydropurine-2,6-dione 381051 7-{3-[4-(2-methoxyphenyl)-piperazin-1-yl]-propyl}-8-propoxy-1,3-dimethyl-3,7-dihydropurine-2,6-dione 381052 7-{3-[4-(3-chlorophenyl)-piperazin-1-yl]-propyl}-8-propoxy-1,3-dimethyl-3,7-dihydropurine-2,6-dione 381053 7-[4-(4-phenylpiperazin-1-yl)-butyl]-8-ethoxy-1,3-dimethyl-3,7-dihydropurine-2,6-dione 381065 7-[4-(4-phenylpiperazin-1-yl)-butyl]-8-propoxy-1,3-dimethyl-3,7-dihydropurine-2,6-dione 381067 7-{4-[4-(2-methoxyphenyl)-piperazin-1-yl]-butyl}-8-propoxy-1,3-dimethyl-3,7-dihydropurine-2,6-dione 381068 7-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-8-ethoxy-1,3-dimethyl-3,7-dihydropurine-2,6-dione 381071 7-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-8-ethoxy-1,3-dimethyl-3,7-dihydropurine-2,6-dione 381072 7-[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)-propyl]-8-propoxy-1,3-dimethyl-3,7-dihydropurine-2,6-dione 381073 7-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)-butyl]-8-ethoxy-1,3-dimethyl-3,7-dihydropurine-2,6-dione 381074 7-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)-butyl]-8-propoxy-1,3-dimethyl-3,7-dihydropurine-2,6-dione 381075 7-[3-(4-phenylpiperazin-1-yl)-propyl]-1,3-dimethyl-7,9-dihydro-3H-purine-2,6,8-trione 381076 7-{3-[4-(3-chlorophenyl)-piperazin-1-yl]-propyl}-1,3-dimethyl-7,9-dihydro-3H-purine-2,6,8-trione 381077 7-[4-(4-phenylpiperazin-1-yl)-butyl]-1,3-dimethyl-7,9-dihydro-3H-purine-2,6,8-trione 381078 7-{4-[4-(3-chlorophenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-7,9-dihydro-3H-purine-2,6,8-trione 381079 7-{3-[1,2,3,4-tetrahydroisoquinolin-2-yl]-propyl}-1,3-dimethyl-7,9-dihydro-3H-purine-2,6,8-trione 381096 N-Isobutyl-2E,4E-dodeca-2,4-dienamide 381327 H-Tyr-D-Ala-Gly-Phe-Gly-Pro-Leu-Trp-O-3,5-Bzl(CF3)2 381328 H-Tyr-D-Ala-Gly-Phe-Leu-Pro-Leu-Trp-O-3,5-Bzl(CF3)2 381329 Tyr-D-Ala-Gly-Phe-Met-Pro-Leu-Trp-O-3,5-Bzl(CF 3) 2 381330 H-Tyr-D-Ala-Gly-Phe-Met(O)-Pro-Leu-Trp-O-3,5-Bzl(CF3)2 381331 H-Tyr-D-Ala-Gly-Phe-Nle-Pro-Leu-Trp-O-3,5-Bzl(CF3)2 381332 H-Tyr-D-Ala-Gly-Phe-N-Me-Nle-Pro-Leu-Trp-O-3,5-Bzl(CF3)2 381502 Tyr-Pro-Mmp-Phe-NH 381503 Dmt-Pro-Mmp-Phe-NH2 381504 Tyr-Pro-3,5Dmp-Phe-NH2 381505 Dmt-Pro-3,5Dmp-Phe-NH2 381506 Tyr-Pro-Dmp-Phe-NH2 381509 Dmt-Pro-Dmp-Phe-NH2 381510 Tyr-Pro-Dmt-Phe-NH2 381512 Dmt-Pro-Dmt-Phe-NH2 381515 Tyr-Pro-Tmp-Phe-NH 381517 Dmt-Pro-Tmp-Phe-NH2 381520 Tyr-Pro-Emp-Phe-NH2 381521 Dmt-Pro-Emp-Phe-NH2 381522 Tyr-Pro-Imp-Phe-NH2 381527 Dmt-Pro-Imp-Phe-NH2 381672 cis-(-)-7,8-dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 381674 cis-(-)-7,8-dimethoxy-3-[4-(3-(4-fluoro)phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole 381693 SID17389715 381933 (1S)-1-(3-fluoro-benzyl)-2-(5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy)-ethylamine 381934 (1S)-1-(2,3-difluoro-benzyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381935 (1S)-1-(2,4-difluoro-benzyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381936 (1S)-1-(2,6-difluoro-benzyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381937 (1S)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-1-(2,3,4-trifluoro-benzyl)-ethylamine 381938 (1S)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-1-(2,4,6-trifluoro-benzyl)-ethylamine 381939 (1S)-1-(2-chloro-benzyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381940 (1S)-1-(3-chloro-benzyl)-2-(5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy)-ethylamine 381941 (1S)-1-(4-chloro-benzyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381942 (1S)-bromo-benzyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381943 (1S)-1-(3-bromo-benzyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381944 (1S)-1-(4-bromo-benzyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381945 (1S)-1-(3-iodo-benzyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381946 (1S)-1-(3-chloro-4-fluoro-benzyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381947 (1S)-1-(4-chloro-3-fluoro-benzyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381948 (1S)-1-(2,3-dichloro-benzyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381949 (1S)-1-(3,4-dichloro-benzyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381950 (1S)-1-(3,5-dichloro-benzyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381972 (1S)-1-(4-bromo-2-fluoro-benzyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381973 (1S)-1-(4-bromo-3-fluoro-benzyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381974 (1S)-1-(2-bromo-4,6-difluoro-benzyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381975 (1S)-1-(5-fluoro-2-methyl-benzyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381976 (1S)-1-(4-bromo-3-methyl-benzyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381977 (1S)-1-(4-fluoro-3-methyl-benzyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381978 (1S)-1-(4-fluoro-2-methyl-benzyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381979 (1S)-1-(3-fluoro-4-methyl-benzyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381980 (1S)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-1-(2,4,6-trimethyl-benzyl)-ethylamine 381981 (1S)-1-(5-fluoro-2-methoxy-benzyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381982 (1S)-2-(5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy)-1-(3-trifluoromethyl-benzyl)-ethylamine 381983 (1S)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-1-(4-trifluoromethyl-benzyl)-ethylamine 381984 (1S)-1-(3,5-bis-trifluoromethyl-benzyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381985 (1S)-1-(4-fluoro-3-trifluoromethyl-benzyl)-2-[5-(3-methyl-1Hindazol-5-yl)-pyridin-3-yloxy]-ethylamine 381986 (1S)-1-(3-fluoro-5-trifluoromethyl-benzyl)-2-[5-(3-methyl-1Hindazol-5-yl)-pyridin-3-yloxy]-ethylamine 381987 ((1S)-1-(2-fluoro-5-trifluoromethyl-benzyl)-2-[5-(3-methyl-1Hindazol-5-yl)-pyridin-3-yloxy]-ethylamine 381988 (1S)-1-(3-fluoro-4-trifluoromethyl-benzyl)-2-[5-(3-methyl-1Hindazol-5-yl)-pyridin-3-yloxy]-ethylamine 381989 (1S)-1-(2-fluoro-4-trifluoromethyl-benzyl)-2-[5-(3-methyl-1Hindazol-5-yl)-pyridin-3-yloxy]-ethylamine 381990 (1S)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-1-(2-trifluoromethoxy-benzyl)-ethylamine 381991 (1S)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-1-(3-trifluoromethoxy-benzyl)-ethylamine 381992 (1S)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-1-(4-trifluoromethoxy-benzyl)-ethylamine 381993 (1S)-1-biphenyl-3-ylmethyl-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381994 (1S)-1-benzo1,3dioxol-5-ylmethyl-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381995 (1S)-1-(2,2-difluoro-benzo1,3dioxol-4-ylmethyl)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-ethylamine 381996 (1S)-2-[5-(3-methyl-1H-indazol-5-yl)-pyridin-3-yloxy]-1-(2,2,3,3-tetrafluoro-2,3-dihydro-benzo1,4dioxin-6-ylmethyl)-ethylamine 381997 (S)-1-(5-(3-methyl-1H-indazol-5-yl)pyridin-3-yloxy)-3-(3-(2-morpholinoethoxy)phenyl)propan-2-amine 381998 (S)-1-(5-(3-methyl-1H-indazol-5-yl)pyridin-3-yloxy)-3-(3-(2-(piperidin-4-yl)ethoxy)phenyl)-propan-2-amine 381999 (S)-1-(5-(3-methyl-1H-indazol-5-yl)pyridin-3-yloxy)-3-(3-(piperidin-4-ylmethoxy)phenyl)-propan-2-amine 382000 (S)-1-(3-cyclohexylmethoxy-benzyl)-2-[5-(3-methyl-1H-indazol-6-yl)-pyridin-3-yloxy]-ethylamine 382001 (S)-2-[5-(3-methyl-1H-indazol-6-yl)-pyridin-3-yloxy]-1-[3-(1-methyl-piperidin-4-ylmethoxy)-benzyl]-ethylamine 382002 (S)-1-[3-(2-amino-ethoxy)-benzyl]-2-[5-(3-methyl-1H-indazol-6-yl)-pyridin-3-yloxy]-ethylamine 382003 (S)-5-(5-(2-amino-3-phenylpropoxy)pyridin-3-yl)indolin-2-one 382004 (S,Z)-3-((1H-pyrrol-2-yl)methylene)-5-(5-(2-amino-3-phenylpropoxy)pyridin-3-yl)indolin-2-one 382005 (S)-5-(5-(2-amino-3-phenylpropoxy)pyridin-3-yl)-3-(furan-2-ylmethylene)indolin-2-one 382006 (S)-1-(5-(1H-pyrazolo[3,4-c]pyridin-5-yl)pyridin-3-yloxy)-3-(3-(trifluoromethyl)phenyl)propan-2-amine 382007 (S)-1-(5-(3-chloro-1H-pyrazolo[3,4-c]pyridin-5-yl)pyridin-3-yloxy)-3-(3-(trifluoromethyl)-phenyl)propan-2-amine 382008 (S)-1-(5-(3-methyl-1H-pyrazolo[3,4-c]pyridin-5-yl)pyridin-3-yloxy)-3-(3-(trifluoromethyl)-phenyl)propan-2-amine 382009 (S)-1-(2,3-difluorophenyl)-3-(5-(3-methyl-1H-pyrazolo[3,4-c]-pyridin-5-yl)pyridin-3-yloxy)propan-2-amine 382118 3-(2-(1-(3,3-dimethyl-2-oxo-butyl)-5-isobutyl-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-benzoic acid 382120 3-(2-(5-cycloheptyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-benzoic acid 382121 3-(2-(5-adamantan-1-yl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-benzoic acid 382127 3-(2-(1-(2-adamantan-1-yl-2-oxo-ethyl)-5-cyclohexyl-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-benzoic acid 382128 3-(2-(5-cyclohexyl-1-(2-oxo-2-o-tolyl-ethyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-benzoic acid 382129 3-(2-(5-cyclohexyl-1-(2-cyclopentyl-2-oxo-ethyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-benzoic acid 382130 3-(2-(1-(2-cyclohexyl-2-oxo-ethyl)-5-cyclohexyl-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-benzoic acid 382131 3-(2-(5-cyclohexyl-1-(2-(1-methyl-cyclopentyl)-2-oxo-ethyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-benzoic acid 382132 (3-(2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-phenyl)-acetic acid 382134 (3-(2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-phenylsulfanyl)-acetic acid 382135 ((3-(2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-phenyl)-methyl-amino)-acetic acid 382137 (3-(2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-phenoxy)-acetic acid 382139 2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(3-methanesulfonylaminocarbonyl-phenyl)-acetamide 382140 2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(3-(2H-tetrazol-5-yl)-phenyl)-acetamide 382141 2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(3-(5-oxo-2,5-dihydro-1,2,4oxadiazol-3-yl)-phenyl)-acetamide 382142 2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(4-(methyl-(2H-tetrazol-5-yl)-amino)-phenyl)-acetamide 382144 2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(3-(1H-tetrazol-5-ylmethylsulfanyl)-phenyl)-acetamide 382145 3'-(2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-biphenyl-3-carboxylic acid 382147 2-(3-(2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-phenyl)-oxazole-4-carboxylic acid 382148 5-(3-(2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-phenyl)-furan-2-carboxylic acid 382151 (3-(2-(5-cyclohexyl-1-(2-cyclopentyl-2-oxo-ethyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-phenyl)-acetic acid 382152 3-(3-(2-(5-cyclohexyl-1-(2-cyclopentyl-2-oxo-ethyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-phenyl)-propionic acid 382153 2-(5-cyclohexyl-1-(2-cyclopentyl-2-oxo-ethyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(3-(5-oxo-2,5-dihydro-[1,2,4]-oxadiazol-3-yl)-phenyl)-acetamide 382154 (3-(2-(5-cyclohexyl-1-(2-cyclopentyl-2-oxo-ethyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-phenylsulfanyl)-acetic acid 382155 3-{[5-(adamantan-1-yloxymethyl)-2-cyclohexyl-1H-imidazole-4-carbonyl]-amino}-benzoic acid 382156 (6-(2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-indol-1-yl)-acetic acid 382158 (6-(2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-indazol-1-yl)-acetic acid 382159 (5-(2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-indol-1-yl)-acetic acid 382160 (5-(2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-indazol-1-yl)-acetic acid 382253 (2R,3R,4S)-2-(6-(3-fluorobenzylamino)-2-chloro-9H-purin-9-yl)-tetrahydrothiophene-3,4-diol 382255 (2R,3R,4S)-2-(6-(3-chlorobenzylamino)-2-chloro-9H-purin-9-yl)-tetrahydrothiophene-3,4-diol 382257 (2R,3R,4S)-2-(6-(3-bromobenzylamino)-2-chloro-9H-purin-9-yl)-tetrahydrothiophene-3,4-diol 382259 (2R,3R,4S)-2-(2-chloro-6-(3-iodobenzylamino)-9H-purin-9-yl)tetrahydrothiophene-3,4-diol 382261 (2R,3R,4S)-2-(2-chloro-6-(2-chlorobenzylamino)-9H-purin-9-yl)tetrahydrothiophene-3,4-diol 382263 (2R,3R,4S)-2-(2-chloro-6-(5-chloro-2-methoxybenzylamino)-9H-purin-9-yl)tetrahydrothiophene-3,4-diol 382265 (2R,3R,4S)-2-(2-chloro-6-(2-methoxybenzylamino)-9H-purin-9-yl)tetrahydrothiophene-3,4-diol 382267 (2R,3R,4S)-2-(2-chloro-6-(naphthalen-1-ylmethylamino)-9H-purin-9-yl)tetrahydrothiophene-3,4-diol 382271 (2R,3R,4S)-2-(2-chloro-6-(methylamino)-9H-purin-9-yl)-tetrahydrothiophene-3,4-diol 382323 cis-H-Tyr-c[D-AllylGly-Gly-Phe-D-Allylgly]-OH 382324 trans-H-Tyr-c[D-AllylGly-Gly-Phe-D-Allylgly]-OH 382325 H-Tyr-c[D-Allylgly-Gly-Phe-D-Allylgly]-OH 382326 H-butyloxycarbonyl-L-tyrosinyl-D-allylglycyl-glycyl-L-phenylalanyl-D-allylglycine- 382327 3-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-methylpyridin-2-yl)-1H-imidazol-2-yl)methylamino)benzonitrile 382328 4-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-methylpyridin-2-yl)-1H-imidazol-2-yl)methylamino)benzonitrile 382329 3-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-ethylpyridin-2-yl)-1H-imidazol-2-yl)methylamino)benzonitrile 382330 4-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-ethylpyridin-2-yl)-1H-imidazol-2-yl)methylamino)benzonitrile 382331 3-((5-(6-methylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H-imidazol-2-yl)methylamino)benzonitrile 382332 4-((5-(6-methylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H-imidazol-2-yl)methylamino)benzonitrile 382333 3-((5-(6-ethylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H-imidazol-2-yl)methylamino)benzonitrile 382334 4-((5-(6-ethylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H-imidazol-2-yl)methylamino)benzonitrile 382335 3-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-methylpyridin-2-yl)-1H-imidazol-2-yl)methylamino)benzamide 382336 4-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-methylpyridin-2-yl)-1H-imidazol-2-yl)methylamino)benzamide 382337 3-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-ethylpyridin-2-yl)-1H-imidazol-2-yl)methylamino)benzamide 382338 4-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-ethylpyridin-2-yl)-1H-imidazol-2-yl)methylamino)benzamide 382339 3-((5-(6-methylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H-imidazol-2-yl)methylamino)benzamide 382340 4-((5-(6-methylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H-imidazol-2-yl)methylamino)benzamide 382341 3-((5-(6-ethylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H-imidazol-2-yl)methylamino)benzamide 382342 4-((5-(6-ethylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H-imidazol-2-yl)methylamino)benzamide 382343 3-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-methylpyridin-2-yl)-1H-imidazol-2-ylamino)methyl)benzonitrile 382344 4-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-methylpyridin-2-yl)-1H-imidazol-2-ylamino)methyl)benzonitrile 382367 (1'R,2'S,4'R,5'S)-phosphoric acid mono-[4-(2-cyano-6-methylaminopurin-9-yl)-1-phosphonooxymethyl-bicyclo[3.1.0]hex-2-yl]ester 382368 (1'R,2'S,4'R,5'S)-phosphoric acid mono-[4-(2-carbamoyl-6-methylaminopurin-9-yl)-1-phosphonooxymethyl-bicyclo-[3.1.0]hex-2-yl] ester 382374 (1'R,2'S,4'R,5'S)-6-methylamino-9-(4-phosphonooxy-5-phosphonooxymethyl-bicyclo[3.1.0]hex-2-yl)-9H-purine-2-carboxylic acid 382376 5-[4-(6-fluorobenzisoxazol-3-yl)piperidinylmethyl]-6-phenyl-4,5-dihydro-2H-pyridazin-3-one 382379 5-(piperazin-1-ylmethyl)-6-phenyl-4,5-dihydro-2H-pyridazin-3-one 382385 5-[4-(3-(p-fluorobenzoyl)butyl)piperazin-1-ylmethyl]-6-phenyl-4,5-dihydro-2Hpyridazin-3-one 382392 (1'R,2'S,4'S,5'S)-4-(2-ethynyl-6-methylaminopurin-9-yl)-1-[(phosphato)-methyl]-2-(phosphato)-bicyclo[3.1.0]hexane 382401 1-[(4-oxo-4,5,6,7-tetrahydrobenzofuran-5-yl)ethyl]-4-(4-fluorobenzoyl)piperazine 382405 (1'R,2'S,4'R,5'S)-phosphoric acid mono-[4-(6-methylamino-2-phenylpurin-9-yl)-1-phosphonooxymethyl-bicyclo[3.1.0]hex-2-yl] ester 382406 (1'R,2'S,4'S,5'S)-phosphoric acid mono-[1-hydroxymethyl-4-(2-iodo-6-methylaminopurin-9-yl)-bicyclo[3.1.0]hex-2-yl] ester 382407 [3-(2-iodo-6-methylaminopurin-9-yl)-2-phosphonomethylpropyl]-phosphonic acid 382478 5-[(4R)-3-oxo-4-[(phenylacetyl)amino]-3,4,5,10-tetrahydroazepino[3,4-b]indol-2(1H)-yl]pentan-1-aminium 382479 N-[(4R)-2-(5-aminopentyl)-3-oxo-1,2,3,4,5,10-hexahydroazepino[3,4-b]indol-4-yl]-3,3-diphenylpropanamide 382480 (2S)-6-amino-N-benzyl-2-[(4R)-3-oxo-4-[(phenylacetyl)amino]-3,4,5,10-tetrahydroazepino[3,4-b]indol-2(1H)-yl]hexanamide 382481 (2S)-6-amino-N-benzyl-2-[(4R)-4-[(3,3-diphenylpropanoyl)amino]-3-oxo-3,4,5,10-tetrahydroazepino[3,4-b]indol-2(1H)-yl]hexanamide 382704 N-[(1S,2S)-2-(3-cyano-5-fluorophenyl)-3-(4-methoxyphenyl)-1-methylpropyl]-2-methyl-2-{[5-(trifluoromethyl)pyridin-2-yl]oxy}propanamide 382705 N-[(1S,2S)-2-(3-cyano-5-fluorophenyl)-3-[4-(fluoromethoxy)phenyl)]-1-methylpropyl]-2-methyl-2-{[5-(trifluoromethyl)pyridin-2-yl]oxy}propanamide 382708 N-{(1S,2S)-2-(3-cyano-5-fluorophenyl)-3-[4-(2-fluoroethoxy)phenyl)]-1-methylpropyl}-2-methyl-2-{[5-(trifluoromethyl)pyridin-2-yl]oxy}propanamide 382709 N-{(1S,2S)-2-(3-cyanophenyl)-3-[4-(2-fluoroethoxy)phenyl)]-1-methylpropyl}-2-methyl-2-{[5-(trifluoromethyl)pyridin-2-yl]oxy}propanamide 382710 N-{(1S,2S)-2-(3-cyanophenyl)-3-[4-(2-fluoroethoxy)phenyl)]-1-methylpropyl}-2-methyl-2-{[4-(trifluoromethyl)pyridin-2-yl]oxy}propanamide 382711 N-{(1S,2S)-2-(3-cyanophenyl)-3-[4-(2-fluoroethoxy)phenyl]-1-methylpropyl}-2-methyl-2-(pyridin-2-yloxy)propanamide 382713 N-{(1S,2S)-2-(3-cyanophenyl)-3-[4-(2-fluoroethoxy)phenyl)]-1-methylpropyl}-2-methyl-2-[(5-chloropyridin-2-yl)oxy]propanamide 382714 N-{(1S,2S)-2-(3-cyanophenyl)-3-[4-(2-fluoroethoxy)phenyl)]-1-methylpropyl}-2-methyl-2-[(5-cyanopyridin-2-yl)oxy]propanamide 382715 N-{(1S,2S)-2-(3-cyanophenyl)-3-[4-(2-fluoroethoxy)phenyl)]-1-methylpropyl}-2-methyl-2-[(4-methylpyridin-2-yl)oxy]propanamide 382716 N-{(1S,2S)-2-(3-cyanophenyl)-3-[4-(2-fluoroethoxy)phenyl)]-1-methylpropyl}-2-methyl-2-[(5-methylpyridin-2-yl)oxy]propanamide 382718 N-{(1S,2S)-2-(3-cyanophenyl)-3-[4-(2-fluoroethoxy)phenyl]-1-methylpropyl}-2-(6-trifluoromethyl-4-pyrimidyloxy)-2-methylpropanamide 382723 N-[(2S,3S)-3-(3-cyanophenyl)-4-[4-(2-fluoroethoxy)phenyl]butan-2-yl]-2-methyl-2-[(5-methylpyridin-2-yl)oxy]propanamide 382885 (2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 9-acetoxy-2-(2-bromofuran-3-yl)-6a,10b-dimethyl-4,10-dioxododecahydro-1H-benzo[f]isochromene-7-carboxylate 382886 (2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 9-acetoxy-2-(2-bromo-5-methoxy-2,5-dihydrofuran-3-yl)-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 382888 (2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 9-acetoxy-6a,10b-dimethyl-4,10-dioxo-2-((R)-tetrahydrofuran-3-yl)-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 382889 (1R,2R,4aR,5R,7S,8aR)-7-acetoxy-5-(methoxycarbonyl)-4a-methyl-8-oxo-1-(2-(tetrahydrofuran-3-yl)ethyl)-decahydronaphthalene-2-carboxylic acid 382890 (4aR,6aR,7R,9S,10aS,10bR)-methyl 9-acetoxy-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 382891 (2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 9-acetoxy-2-(4,5-dihydrooxazol-2-yl)-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 382892 (2S,4aS,6aR,7R,9S,10aS,10bR)-methyl 9-acetoxy-6a,10b-dimethyl-2-(3-methyl-1,2,4-oxadiazol-5-yl)-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 382893 (4aR,6aR,7R,9S,10aS,10bR)-methyl 9-acetoxy-2-((2S,5S)-2,5-dimethoxy-2,5-dihydrofuran-3-yl)dodecahydro-6a,10b-dimethyl-4,10-dioxo-2H-naphtho[2,1-c]pyran-7-carboxylic acid 382894 (4aR,6aR,7R,9S,10aS,10bR)-methyl 9-acetoxy-2-((2R,5S)-2,5-dimethoxy-2,5-dihydrofuran-3-yl)dodecahydro-6a,10b-dimethyl-4,10-dioxo-2H-naphtho[2,1-c]pyran-7-carboxylic acid 382895 (2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 9-acetoxy-2-((2S,3S,5S)-2,5-dimethoxy-tetrahydrofuran-3-yl)dodecahydro-6a,10b-dimethyl-4,10-dioxo-2H-naphtho[2,1-c]pyran-7-carboxylic acid methyl ester 382896 (2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 9-acetoxy-2-((2R,3S,5S)-2,5-dimethoxy-tetrahydrofuran-3-yl)dodecahydro-6a,10b-dimethyl-4,10-dioxo-2H-naphtho[2,1-c]pyran-7-carboxylic acid methyl ester 383076 N-cyclohexyl-2-(2,4-dichlorophenyl)-1-p-tolyl-1H-imidazole-4-carboxamide 383077 N-cyclohexyl-2-(2,4-dichlorophenyl)-1-(4-methoxyphenyl)-1H-imidazole-4-carboxamide 383078 N-cyclohexyl-2-(2,4-dichlorophenyl)-1-(4-fluorophenyl)-1H-imidazole-4-carboxamide 383079 1-(4-chlorophenyl)-N-cyclohexyl-2-(2,5-dichlorophenyl)-1H-imidazole-4-carboxamide 383080 1-(4-chlorophenyl)-N-cyclohexyl-2-phenyl-1H-imidazole-4-carboxamide 383081 1-(4-chlorophenyl)-N-cyclohexyl-2-(2,4-dimethylphenyl)-1H-imidazole-4-carboxamide 383082 1-(4-chlorophenyl)-N-cyclohexyl-2-(2,4-difluorophenyl)-1H-imidazole-4-carboxamide 383083 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-cyclohexyl-1H-imidazole-4-carboxamide 383084 2-(2-chlorophenyl)-N-cyclohexyl-1-p-tolyl-1H-imidazole-4-carboxamide 383085 2-(2-chlorophenyl)-N-cyclohexyl-1-(4-methoxyphenyl)-1H-imidazole-4-carboxamide 383086 2-(2-chlorophenyl)-N-cyclohexyl-1-(4-fluorophenyl)-1H-imidazole-4-carboxamide 383087 1-(4-chlorophenyl)-N-cyclohexyl-2-o-tolyl-1H-imidazole-4-carboxamide 383088 1-(4-chlorophenyl)-N-cyclohexyl-2-(2-ethylphenyl)-1H-imidazole-4-carboxamide 383089 1-(4-chlorophenyl)-N-cyclohexyl-2-(2-methoxyphenyl)-1H-imidazole-4-carboxamide 383090 2-(2-chlorophenyl)-N-cyclohexyl-1-(4-methylcyclohexyl)-1H-imidazole-4-carboxamide 383091 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-cyclohexyl-N-methyl-1H-imidazole-4-carboxamide 383092 2-(2-chlorophenyl)-N-cyclohexyl-1-(pyridin-3-yl)-1H-imidazole-4-carboxamide 383094 N-((1S,2S)-2-aminocyclohexyl)-1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-1H-imidazole-4-carboxamide 383095 N-((1R,2R)-2-aminocyclohexyl)-1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-1H-imidazole-4-carboxamide 383096 1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-N-((1S,2S)-2-(methylamino)cyclohexyl)-1H-imidazole-4-carboxamide 383097 1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-N-((1R,2R)-2-(methylamino)cyclohexyl)-1H-imidazole-4-carboxamide 383098 rac-1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-N-(2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide 383099 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide 383100 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1R,2R)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide 383101 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclopentyl)-1H-imidazole-4-carboxamide 383102 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1R,2R)-2-hydroxycyclopentyl)-1H-imidazole-4-carboxamide 383103 rac-2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl)-1H-imidazole-4-carboxamide 383104 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl)-1H-imidazole-4-carboxamide 383105 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl)-1H-imidazole-4-carboxamide 383106 rac-2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-1-hydroxy-2,3-dihydro-1H-inden-2-yl)-1H-imidazole-4-carboxamide 383107 rac-2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1R,2S)-1-hydroxy-2,3-dihydro-1H-inden-2-yl)-1H-imidazole-4-carboxamide 383108 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-5-methyl-1H-imidazole-4-carboxamide 383112 2-(2-chlorophenyl)-1-(4-chlorophenyl)-5-ethyl-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide 383114 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-5-propyl-1H-imidazole-4-carboxamide 383115 5-butyl-2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide 383117 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-5-isopropyl-1H-imidazole-4-carboxamide 383119 5-bromo-2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide 383121 1-(4-bromophenyl)-2-(2-chlorophenyl)-5-ethyl-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide 383178 N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-aminothiazol-4-yl)-4-(4-phenylpiperidin-1-yl)butanamide 383179 N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-aminothiazol-4-yl)-4-(4-(4-fluorophenyl)piperidin-1-yl)butanamide 383180 4-(4-(1H-benzo[d]imidazol-1-yl)piperidin-1-yl)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-aminothiazol-4-yl)butanamide 383181 2-(2-amino-1,3-thiazol-4-yl)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-4-{spiro[indene-1,4'-piperidine]-1'-yl}butanamide 383182 2-(2-amino-1,3-thiazol-4-yl)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-4-[(5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]butanamide 383184 N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-aminothiazol-4-yl)-4-(4-o-tolylpiperazin-1-yl)butanamide 383186 7-phenyl-5-methyl-N-[4-(2-pyrrolidin-1-ylethoxy)phenyl]-1,2,4-benzotriazin- 383187 ([7-(2,6-dichloro-phenyl)-5-methyl-benzo[1,2,4]triazin-3-yl]-[4-(2-pyrrolidin-1-yl-ethoxy)-phenyl]-amine) 383188 N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-acetamidothiazol-4-yl)-4-(4-phenylpiperidin-1-yl)butanamide 383189 7-(2-chlorophenyl)-5-methyl-N-[4-(2-pyrrolidin-1-ylethoxy)phenyl]-1,2,4-benzotriazin-3-amine 383190 N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-acetamidothiazol-4-yl)-4-(4-(4-fluorophenyl)piperidin-1-yl)butanamide 383192 4-(4-(1H-benzo[d]imidazol-1-yl)piperidin-1-yl)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-acetamidothiazol-4-yl)butanamide 383193 7-(2-chloro-6-methoxyphenyl)-5-methyl-N-(4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)benzo[e][1,2,4]triazin-3-amine 383194 N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-2-(2-acetamido-1,3-thiazol-4-yl)-4-{spiro[indene-1,4'-piperidine]-1'-yl}butanamide 383195 7-(2-chloro-5-methoxyphenyl)-5-methyl-N-(4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)benzo[e][1,2,4]triazin-3-amine 383196 N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-2-(2-acetamido-1,3-thiazol-4-yl)-4-[(5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]butanamide 383197 N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-acetamidothiazol-4-yl)-4-(4-(4-fluorophenyl)piperazin-1-yl)butanamide 383198 7-(5-chloro-2-methoxyphenyl)-5-methyl-N-(4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)benzo[e][1,2,4]triazin-3-amine 383199 N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-acetamidothiazol-4-yl)-4-(4-o-tolylpiperazin-1-yl)butanamide 383200 7-(2-fluoro-5-methylpyridin-4-yl)-5-methyl-N-(4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)benzo[e][1,2,4]triazin-3-amine 383201 7-(3,5-dimethylisoxazol-4-yl)-5-methyl-N-(4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)benzo[e][1,2,4]triazin-3-amine 383202 5-methyl-7-(pyrimidin-4-yl)-N-(4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)benzo[e][1,2,4]triazin-3-amine 383203 5-methyl-7-(pyridin-2-yl)-N-(4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)benzo[e][1,2,4]triazin-3-amine 383204 7-(2,6-dimethylphenyl)-N-(4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)benzo[e][1,2,4]triazin-3-amine 383205 7-(2,6-dichlorophenyl)-N-(4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)benzo[e][1,2,4]triazin-3-amine 383207 7-(2,6-dimethylphenyl)-6-methyl-N-(4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)benzo[e][1,2,4]triazin-3-amine 383208 4-(7-(2,6-dimethylphenyl)-5-methylbenzo[e][1,2,4]triazin-3-ylamino)-N-(2-(pyrrolidin-1-yl)ethyl)benzenesulfonamide 383209 4-(7-(2,6-dichlorophenyl)-5-methylbenzo[e][1,2,4]triazin-3-ylamino)-N-(2-(pyrrolidin-1-yl)ethyl)benzenesulfonamide 383210 4-(7-(2-chloro-6-hydroxyphenyl)-5-methylbenzo[e][1,2,4]triazin-3-ylamino)-N-(2-(pyrrolidin-1-yl)ethyl)benzenesulfonamide 383211 4-(7-(5-cyano-2-methylphenyl)-5-methylbenzo[e][1,2,4]triazin-3-ylamino)-N-(2-(pyrrolidin-1-yl)ethyl)benzenesulfonamide 383212 4-(7-(5-amino-2-chlorophenyl)-5-methylbenzo[e][1,2,4]triazin-3-ylamino)-N-(2-(pyrrolidin-1-yl)ethyl)benzenesulfonamide 383213 4-(7-(3-aminophenyl)-5-methylbenzo[e][1,2,4]triazin-3-ylamino)-N-(2-(pyrrolidin-1-yl)ethyl)benzenesulfonamide 383214 4-(7-(5-(aminomethyl)-2-methylphenyl)-5-methylbenzo[e][1,2,4]triazin-3-ylamino)-N-(2-(pyrrolidin-1-yl)ethyl)benzenesulfonamide 383215 4-(5-methyl-7-(3-(methylamino)phenyl)benzo[e][1,2,4]triazin-3-ylamino)-N-(2-(pyrrolidin-1-yl)ethyl)benzenesulfonamide 383216 4-(5-methyl-7-(3-(methylsulfonamido)phenyl)benzo[e][1,2,4]triazin-3-ylamino)-N-(2-(pyrrolidin-1-yl)ethyl)benzenesulfonamide 383217 N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-formamidothiazol-4-yl)-4-(4-phenylpiperidin-1-yl)butanamide 383218 N-(3,5-bis(trifluoromethyl)benzyl)-4-(4-phenylpiperidin-1-yl)-2-(2-propionamidothiazol-4-yl)butanamide 383219 N-(4-(1-(3,5-bis(trifluoromethyl)benzylamino)-1-oxo-4-(4-phenylpiperidin-1-yl)butan-2-yl)thiazol-2-yl)cyclopropanecarboxamide 383220 N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-isobutyramidothiazol-4-yl)-4-(4-phenylpiperidin-1-yl)butanamide 383221 4-(7-(2,6-dimethylphenyl)-6-methylbenzo[e][1,2,4]triazin-3-ylamino)-N-(2-(pyrrolidin-1-yl)ethyl)benzenesulfonamide 383222 N-(3,5-bis(trifluoromethyl)benzyl)-4-(4-phenylpiperidin-1-yl)-2-(2-pivalamidothiazol-4-yl)butanamide 383223 N-(4-(1-(3,5-bis(trifluoromethyl)benzylamino)-1-oxo-4-(4-phenylpiperidin-1-yl)butan-2-yl)thiazol-2-yl)benzamide 383224 1-(4-(1-(3,5-bis(trifluoromethyl)benzylamino)-1-oxo-4-(4-phenylpiperidin-1-yl)butan-2-yl)thiazol-2-yl)-3-methylurea 383225 3-(4-(1-(3,5-bis(trifluoromethyl)benzylamino)-1-oxo-4-(4-phenylpiperidin-1-yl)butan-2-yl)thiazol-2-yl)-1,1-dimethylurea 383226 4-(6-methyl-7-phenylbenzo[e][1,2,4]triazin-3-ylamino)-N-(2-(pyrrolidin-1-yl)ethyl)benzenesulfonamide 383227 methyl 4-(1-(3,5-bis(trifluoromethyl)benzylamino)-1-oxo-4-(4-phenylpiperidin-1-yl)butan-2-yl)thiazol-2-ylcarbamate 383229 N-(3,5-bis-trifluoromethyl-benzyl)-2-(2-guanidino-thiazol-4-yl)-4-(4-phenyl-piperidin-1-yl)-butyramide 383231 N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-(methylsulfonamido)thiazol-4-yl)-4-(4-phenylpiperidin-1-yl)butanamide 383232 4-(6-methyl-7-o-tolylbenzo[e][1,2,4]triazin-3-ylamino)-N-(2-(pyrrolidin-1-yl)ethyl)benzenesulfonamide 383233 4-(6-methyl-7-(2-(trifluoromethyl)phenyl)benzo[e][1,2,4]triazin-3-ylamino)-N-(2-(pyrrolidin-1-yl)ethyl)benzenesulfonamide 383234 (S)-tert-butyl 4-(1-(3,5-bis(trifluoromethyl)benzylamino)-1-oxo-4-(4-phenylpiperidin-1-yl)butan-2-yl)thiazol-2-ylcarbamate 383235 4-(7-(5-cyano-2-methylphenyl)-6-methylbenzo[e][1,2,4]triazin-3-ylamino)-N-(2-(pyrrolidin-1-yl)ethyl)benzenesulfonamide 383236 4-(7-(4-fluoro-2-methylphenyl)-6-methylbenzo[e][1,2,4]triazin-3-ylamino)-N-(2-(pyrrolidin-1-yl)ethyl)benzenesulfonamide 383237 (S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-aminothiazol-4-yl)-4-(4-phenylpiperidin-1-yl)butanamide 383238 4-(7-amino-6-methylbenzo[e][1,2,4]triazin-3-ylamino)-N-(2-(pyrrolidin-1-yl)ethyl)benzenesulfonamide 383239 (S)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-acetamidothiazol-4-yl)-4-(4-phenylpiperidin-1-yl)butanamide 383240 (S)-methyl 4-(1-(3,5-bis(trifluoromethyl)benzylamino)-1-oxo-4-(4-phenylpiperidin-1-yl)butan-2-yl)thiazol-2-ylcarbamate 383241 4-(7-(2-(hydroxymethyl)phenyl)-6-methylbenzo[e][1,2,4]triazin-3-ylamino)-N-(2-(pyrrolidin-1-yl)ethyl)benzenesulfonamide 383242 (S)-1-(4-(1-(3,5-bis(trifluoromethyl)benzylamino)-1-oxo-4-(4-phenylpiperidin-1-yl)butan-2-yl)thiazol-2-yl)-3-methylurea 383243 (2S)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-2-(2-acetamido-1,3-thiazol-4-yl)-4-{spiro[indene-1,4'-piperidine]-1'-yl}butanamide 383244 (2S)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-2-{2-[(methylcarbamoyl)amino]-1,3-thiazol-4-yl}-4-{spiro[indene-1,4'-piperidine]-1'-yl}butanamide 383245 7-(2,6-dimethylphenyl)-5-methyl-N-(3-(2-morpholinoethoxy)phenyl)benzo[e][1,2,4]triazin-3-amine 383246 7-(2,6-dimethylphenyl)-5-methyl-N-(4-(3-(pyrrolidin-1-yl)propoxy)phenyl)benzo[e][1,2,4]triazin-3-amine 383247 7-(2,6-dimethylphenyl)-5-methyl-N-(4-(2-(4-methylpiperazin-1-yl)ethoxy)phenyl)benzo[e][1,2,4]triazin-3-amine 383248 7-(2,6-dimethylphenyl)-5-methyl-N-(3-(2-(4-methylpiperazin-1-yl)ethoxy)phenyl)benzo[e][1,2,4]triazin-3-amine 383249 7-(2,6-dimethylphenyl)-5-methyl-N-(4-(2-(4-methylpiperazin-1-yl)propoxy)phenyl)benzo[e][1,2,4]triazin-3-amine 383250 7-(2,6-dimethylphenyl)-5-methyl-N-(3-(2-(4-methylpiperazin-1-yl)propoxy)phenyl)benzo[e][1,2,4]triazin-3-amine 383251 4-(7-(2,6-dimethylphenyl)-5-methylbenzo[e][1,2,4]triazin-3-ylamino)-N-(4-methylpiperazin-1-yl)benzamide 383252 4-(7-(2,6-dimethylphenyl)-5-methylbenzo[e][1,2,4]triazin-3-ylamino)-N-(piperazin-1-yl)benzamide 383253 N-(4-(7-(2,6-dimethylphenyl)-5-methylbenzo[e][1,2,4]triazin-3-ylamino)phenyl)-N-(2-(pyrrolidin-1-yl)ethyl)benzamide 383254 N-(3-(7-(2,6-dimethylphenyl)-5-methylbenzo[e][1,2,4]triazin-3-ylamino)phenyl)-N-(2-(pyrrolidin-1-yl)ethyl)benzamide 383255 7-(2,6-dimethylphenyl)-5-methyl-N-(2-(2-(pyrrolidin-1-yl)ethoxy)pyridin-4-yl)benzo[e][1,2,4]triazin-3-amine 383256 (R)-tert-butyl 4-(1-(3,5-bis(trifluoromethyl)benzylamino)-1-oxo-4-(4-phenylpiperidin-1-yl)butan-2-yl)thiazol-2-ylcarbamate 383257 (R)-N-(3,5-bis(trifluoromethyl)benzyl)-4-(4-phenylpiperidin-1-yl)-2-(thiazol-4-yl)butanamide 383258 (R)-N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-acetamidothiazol-4-yl)-4-(4-phenylpiperidin-1-yl)butanamide 383260 (R)-1-(4-(1-(3,5-bis(trifluoromethyl)benzylamino)-1-oxo-4-(4-phenylpiperidin-1-yl)butan-2-yl)thiazol-2-yl)-3-methylurea 383261 (2R)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-2-(2-acetamido-1,3-thiazol-4-yl)-4-{spiro[indene-1,4'-piperidine]-1'-yl}butanamide 383262 (2R)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-2-{2-[(methylcarbamoyl)amino]-1,3-thiazol-4-yl}-4-{spiro[indene-1,4'-piperidine]-1'-yl}butanamide 383263 7-(2,6-dimethylphenyl)-N3-(4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)benzo[e][1,2,4]triazine-3,5-diamine 383264 7-(2,6-dimethylphenyl)-N5-methyl-N3-(4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)benzo[e][1,2,4]triazine-3,5-diamine 383265 N-(7-(2,6-dimethylphenyl)-3-(4-(2-(pyrrolidin-1-yl)ethoxy)phenylamino)benzo[e][1,2,4]triazin-5-yl)acetamide 383266 N-(7-(2,6-dimethylphenyl)-3-(4-(2-(pyrrolidin-1-yl)ethoxy)phenylamino)benzo[e][1,2,4]triazin-5-yl)methanesulfonamide 383267 N-(3,5-bis(trifluoromethyl)benzyl)-2-(2-acetamidothiazol-4-yl)-4-(piperidin-1-yl)butanamide 383268 N-{4-[1-({[3,5-bis(trifluoromethyl)phenyl]methyl}carbamoyl)-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]propyl]-1,3-thiazol-2-yl}benzamide 383269 N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-4-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]-2-[2-(2-phenylacetamido)-1,3-thiazol-4-yl]butanamide 383270 N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-4-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]-2-{2-[2-(thiophen-2-yl)acetamido]-1,3-thiazol-4-yl}butanamide 383271 N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-4-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]-2-{2-[2-(pyridin-2-yl)acetamido]-1,3-thiazol-4-yl}butanamide 383272 N-{4-[1-({[3,5-bis(trifluoromethyl)phenyl]methyl}carbamoyl)-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]propyl]-1,3-thiazol-2-yl}pyridine-3-carboxamide 383273 N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-4-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]-2-[2-(2-phenylpropanamido)-1,3-thiazol-4-yl]butanamide 383274 N-{4-[1-({[3,5-bis(trifluoromethyl)phenyl]methyl}carbamoyl)-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]propyl]-1,3-thiazol-2-yl}bicyclo[4.2.0]octa-1(6),2,4-triene-7-carboxamide 383367 N-(1-((2S,3S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)butanoyl)piperidin-4-yl)-N-phenylpropionamide 383368 N-(1-((2S,3R)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)butanoyl)piperidin-4-yl)-N-phenylpropionamide 383369 (S)-N-(1-(2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)piperidin-4-yl)-N-phenylpropionamide 383370 (S)-N-(1-(2-amino-3-(4-hydroxyphenyl)propanoyl)piperidin-4-yl)-N-phenylpropionamide 383371 (S)-N-(1-(2-amino-3-phenylpropanoyl)piperidin-4-yl)-N-phenylpropionamide 383372 (R)-N-(1-(2-amino-3-(4-chlorophenyl)propanoyl)piperidin-4-yl)-N-phenylpropionamide 383373 (S)-N-(1-(2-amino-3-(thiazol-4-yl)propanoyl)piperidin-4-yl)-N-phenylpropionamide 383374 (S)-N-(1-(2-amino-3-(benzo[b]thiophen-3-yl)propanoyl)piperidin-4-yl)-N-phenylpropionamide 383375 (S)-N-(1-(2-amino-3-(naphthalen-2-yl)propanoyl)piperidin-4-yl)-N-phenylpropionamide 383376 (S)-N-(1-(2-amino-3,3-diphenylpropanoyl)piperidin-4-yl)-N-phenylpropionamide 383377 N-(1-(3-amino-3-(4-chlorophenyl)propanoyl)piperidin-4-yl)-N-phenylpropionamide 383378 N-(1-(3-amino-3-p-tolylpropanoyl)piperidin-4-yl)-N-phenylpropionamide 383379 N-(1-(3-amino-3-(4-methoxyphenyl)propanoyl)piperidin-4-yl)-N-phenylpropionamide 383380 N-(1-(3-(3-bromophenyl)propanoyl)piperidin-4-yl)-N-phenylpropionamide 383381 N-(1-(3-(3-chloro-4-methoxyphenyl)propanoyl)piperidin-4-yl)-N-phenylpropionamide 383382 (S)-N-(1-(2-amino-2-phenylacetyl)piperidin-4-yl)-N-phenylpropionamide 383383 (R)-N-(1-(2-amino-2-phenylacetyl)piperidin-4-yl)-N-phenylpropionamide 383384 (S)-N-(1-(2-amino-2-(2,3-dihydro-1H-inden-2-yl)acetyl)piperidin-4-yl)-N-phenylpropionamide 383579 2-thiosalvinorin B 383581 2-epi-2-thiosalvinorin A 383582 2-epi-2-thiosalvinorin B 383638 3-(5-(1H-imidazol-1-yl)-7-methyl-1H-benzo[d]imidazol-2-yl)pyridin-2(1H)-one 383639 3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-(2-hydroxyethylamino)pyridin-2(1H)-one 383640 3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-(phenethylamino)pyridin-2(1H)-one 383641 3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-(2-hydroxy-2-phenylethylamino)pyridin-2(1H)-one 383642 3-(5-(1H-imidazol-1-yl)-7-methyl-1H-benzo[d]imidazol-2-yl)-4-(2-(2-chlorophenyl)-2-hydroxyethylamino)pyridin-2(1H)-one 383643 N-(2-(2-(3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-2-oxo-1,2-dihydropyridin-4-ylamino)-1-hydroxyethyl)phenyl)methanesulfonamide 383644 3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-(2-(3-fluorophenyl)-2-hydroxyethylamino)pyridin-2(1H)-one 383645 3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-(2-(3-chlorophenyl)-2-hydroxyethylamino)pyridin-2(1H)-one 383646 3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-(2-(3-bromophenyl)-2-hydroxyethylamino)pyridin-2(1H)-one 383647 3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-(2-hydroxy-2-(3-hydroxyphenyl)ethylamino)pyridin-2(1H)-one 383648 3-(2-(3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-2-oxo-1,2-dihydropyridin-4-ylamino)-1-hydroxyethyl)benzonitrile 383653 N-(3-(2-(3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-2-oxo-1,2-dihydropyridin-4-ylamino)-1-hydroxyethyl)phenyl)methanesulfonamide 383676 3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-(2-hydroxy-2-m-tolylethylamino)pyridin-2(1H)-one 383677 3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-(2-hydroxy-2-(3-(trifluoromethyl)phenyl)ethylamino)pyridin-2(1H)-one 383678 3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-(2-hydroxy-2-(3-methoxyphenyl)ethylamino)pyridin-2(1H)-one 383679 N-(4-(2-(3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-2-oxo-1,2-dihydropyridin-4-ylamino)-1-hydroxyethyl)phenyl)methanesulfonamide 383680 3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-(2-hydroxy-2-p-tolylethylamino)pyridin-2(1H)-one 383681 3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-(2-hydroxy-2-(4-methoxyphenyl)ethylamino)pyridin-2(1H)-one 383683 3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-(2-(3,5-dichlorophenyl)-2-hydroxyethylamino)pyridin-2(1H)-one 383684 3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-(2-(3,4-dichlorophenyl)-2-hydroxyethylamino)pyridin-2(1H)-one 383685 3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-(2-(3-chloro-4-fluorophenyl)-2-hydroxyethylamino)pyridin-2(1H)-one 383686 3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-(2-(3-chloro-4-methoxyphenyl)-2-hydroxyethylamino)pyridin-2(1H)-one 383688 3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-(2-(3-chlorophenyl)-2-methoxyethylamino)pyridin-2(1H)-one 383689 3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-(2-(3-bromophenyl)propylamino)pyridin-2(1H)-one 383690 3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-((S)-2-(3-chlorophenyl)-2-hydroxyethylamino)pyridin-2(1H)-one 383691 3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-((R)-2-(3-chlorophenyl)-2-hydroxyethylamino)pyridin-2(1H)-one 383716 N-(2-((dimethylamino)methyl)-4-(3-(dimethylamino)propoxy)phenyl)quinazolin-4-amine 383717 N-(2-((dimethylamino)methyl)-4-(3-(piperidin-1-yl)propoxy)phenyl)quinazolin-4-amine 383718 5-(3-(dimethylamino)propoxy)-N,N-dimethyl-2-(quinazolin-4-yloxy)benzamide 383719 (2-(2-chlorobenzyloxy)-5-((1-methylpiperidin-3-yl)methoxy)phenyl)-N,N-dimethylmethanamine 383720 (2-(2-chlorobenzyloxy)-5-(1-isopropylpyrrolidin-3-yloxy)phenyl)-N,N-dimethylmethanamine 383721 3-(4-(2-chlorobenzyloxy)-3-((dimethylamino)methyl)phenoxy)-N,N-dimethylpropan-1-amine 383722 (2-(2-chlorobenzyloxy)-5-(3-(piperidin-1-yl)propoxy)phenyl)-N,N-dimethylmethanamine 383724 2-(2-chlorobenzyloxy)-N,N-dimethyl-5-(3-(piperidin-1-yl)propoxy)benzamide 383726 2-(2-chlorobenzyloxy)-N,N-dimethyl-5-(3-morpholinopropoxy)benzamide 383727 2-(2-chlorobenzyloxy)-N,N-dimethyl-5-(2-(1-methylpyrrolidin-2-yl)ethoxy)benzamide 383728 2-(2-methoxybenzyloxy)-N,N-dimethyl-5-(3-morpholinopropoxy)benzamide 383729 2-(2-methoxybenzyloxy)-N,N-dimethyl-5-(3-(piperidin-1-yl)propoxy)benzamide 383731 3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-(pyridin-2-ylmethylamino)pyridin-2(1H)-one 383732 3-(6-(1H-imidazol-1-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-((S)-1-hydroxy-3-phenylpropan-2-ylamino)pyridin-2(1H)-one 383733 (S)-3-(6-bromo-4-methyl-1H-benzo[d]imidazol-2-yl)-4-(1-hydroxy-3-phenylpropan-2-ylamino)pyridin-2(1H)-one 383734 (S)-4-(1-hydroxy-3-phenylpropan-2-ylamino)-3-(4-methyl-6-phenyl-1H-benzo[d]imidazol-2-yl)pyridin-2(1H)-one 383735 (S)-3-(6-(4-fluorophenyl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-(1-hydroxy-3-phenylpropan-2-ylamino)pyridin-2(1H)-one 383736 (S)-4-(1-hydroxy-3-phenylpropan-2-ylamino)-3-(6-(4-methoxyphenyl)-4-methyl-1H-benzo[d]imidazol-2-yl)pyridin-2(1H)-one 383737 4-(2-(3-chlorophenyl)-2-hydroxyethylamino)-3-(4-methyl-1H-benzo[d]imidazol-2-yl)pyridin-2(1H)-one 383738 2-(4-(2-(3-chlorophenyl)-2-hydroxyethylamino)-2-oxo-1,2-dihydropyridin-3-yl)-7-methyl-3H-benzo[d]imidazole-5-carboxamide 383739 2-(4-(2-(3-chlorophenyl)-2-hydroxyethylamino)-2-oxo-1,2-dihydropyridin-3-yl)-N,7-dimethyl-3H-benzo[d]imidazole-5-carboxamide 383740 2-(4-(2-(3-chlorophenyl)-2-hydroxyethylamino)-2-oxo-1,2-dihydropyridin-3-yl)-N,N,7-trimethyl-3H-benzo[d]imidazole-5-carboxamide 383741 2-(4-(2-(3-chlorophenyl)-2-hydroxyethylamino)-2-oxo-1,2-dihydropyridin-3-yl)-N-cyclopropyl-7-methyl-3H-benzo[d]imidazole-5-carboxamide 383742 2-(4-(2-(3-chlorophenyl)-2-hydroxyethylamino)-2-oxo-1,2-dihydropyridin-3-yl)-N-cyclopentyl-7-methyl-3H-benzo[d]imidazole-5-carboxamide 383743 2-(4-(2-(3-chlorophenyl)-2-hydroxyethylamino)-2-oxo-1,2-dihydropyridin-3-yl)-N-cyclohexyl-7-methyl-3H-benzo[d]imidazole-5-carboxamide 383744 4-(2-(3-chlorophenyl)-2-hydroxyethylamino)-3-(4-methyl-6-(1-methyl-4,5-dihydro-1H-imidazol-2-yl)-1H-benzo[d]imidazol-2-yl)pyridin-2(1H)-one 383745 4-(2-(3-chlorophenyl)-2-hydroxyethylamino)-3-(4-methyl-6-(4-methyl-4,5-dihydro-1H-imidazol-2-yl)-1H-benzo[d]imidazol-2-yl)pyridin-2(1H)-one 383746 4-(2-(3-chlorophenyl)-2-hydroxyethylamino)-3-(6-(4,4-dimethyl-4,5-dihydro-1H-imidazol-2-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)pyridin-2(1H)-one 383747 4-(2-(3-chlorophenyl)-2-hydroxyethylamino)-3-(4-methyl-6-(1,4,5,6-tetrahydropyrimidin-2-yl)-1H-benzo[d]imidazol-2-yl)pyridin-2(1H)-one 383748 2-(4-{[2-(3-chlorophenyl)-2-hydroxyethyl]amino}-2-oxo-1,2-dihydropyridin-3-yl)-N,4-dimethyl-1H-1,3-benzodiazole-6-carboximidamide 383751 4-(2-(3-chlorophenyl)-2-hydroxyethylamino)-3-(4-methyl-6-(5-methyl-1H-imidazol-2-yl)-1H-benzo[d]imidazol-2-yl)pyridin-2(1H)-one 383762 4-amino-4'-fluoro-5-pyridin-4-yl-biphenyl-3-carboxylic acid amide 383768 4'-amino-4-fluoro-4''-(pyrrolidine-1-sulfonyl)-[1,1',3',1'']terphenyl-5'-carboxylic acid amide 383775 4'-amino-4-fluoro-4''-sulfamoyl-[1,1',3',1'']terphenyl-5'-carboxylic acid amide 383781 4'-amino-4-chloro-4''-sulfamoyl-[1,1',3',1'']terphenyl-5'-carboxylic acid amide 383785 4'-amino-4-chloro-4''-methanesulfonylamino-[1,1',3',1'']terphenyl-5'-carboxylic acid amide 383788 4'-amino-4''-methanesulfonylamino-[1,1',3',1'']terphenyl-5'-carboxylic acid amide 383791 4'-amino-3''-methanesulfonylamino-[1,1',3',1'']terphenyl-5'-carboxylic acid amide 383794 4'-Amino-4''-sulfamoyl-[1,1',3',1'']terphenyl-5'-carboxylic acid amide 383795 4'-amino-3''-sulfamoyl-[1,1',3',1'']terphenyl-5'-carboxylic acid amide 383796 4'-amino-4''-sulfamoylmethyl-[1,1',3',1'']terphenyl-5'-carboxylic acid amide 383798 2-Amino-5-pyridin-4-yl-biphenyl-3-carboxylic acid amide 383799 2-amino-5-pyridin-4-yl-4'-sulfamoyl-biphenyl-3-carboxylic acid amide 383800 4'-amino-4-methanesulfonyl-4''-sulfamoyl-[1,1',3',1'']terphenyl-5'-carboxylic acid amide 383801 4-amino-4-methanesulfonyl-4''-(pyrrolidine-1-sulfonyl)-[1,1',3',1']terphenyl-5'-carboxylic acid amide 383808 1-(4-(4-amino-7-(pyridin-3-yl)thieno[3,2-c]pyridin-3-yl)phenyl)-3-m-tolylurea 383810 3-(4-aminophenyl)thieno[3,2-c]pyridin-4-amine 383811 N-(4-(4-aminothieno[3,2-c]pyridin-3-yl)phenyl)benzamide 383812 1-(4-(4-aminothieno[3,2-c]pyridin-3-yl)phenyl)-3-phenylurea 383813 1-(4-(4-aminothieno[3,2-c]pyridin-3-yl)phenyl)-3-m-tolylurea 383814 3-(4-(4-aminothieno[3,2-c]pyridin-3-yl)phenyl)-1-methyl-1-m-tolylurea 383815 1-(4-(4-aminothieno[3,2-c]pyridin-3-yl)phenyl)-1-methyl-3-m-tolylurea 383816 N-(4-(4-aminothieno[3,2-c]pyridin-3-yl)phenyl)-2-m-tolylacetamide 383817 2-(4-(4-aminothieno[3,2-c]pyridin-3-yl)phenyl)-N-m-tolylacetamide 383818 1-(4-(4-aminothieno[3,2-c]pyridin-3-yl)phenyl)-3-m-tolylthiourea 383819 1-(3-(4-aminothieno[3,2-c]pyridin-3-yl)phenyl)-3-m-tolylurea 383821 1-(4-(4-amino-2-methylthieno[3,2-c]pyridin-3-yl)phenyl)-3-m-tolylurea 383822 1-(4-(4-aminothieno[3,2-c]pyridin-3-yl)phenyl)-3-p-tolylurea 383823 2-Hydroxy-5-pyridin-4-yl-benzamide 383824 4-chloro-4'-hydroxy-4''-sulfamoyl-[1,1',3',1'']terphenyl-5'-carboxylic acid amide 383825 1-(4-(4-aminothieno[3,2-c]pyridin-3-yl)phenyl)-3-o-tolylurea 383826 1-(4-(4-aminothieno[3,2-c]pyridin-3-yl)phenyl)-3-(3-ethylphenyl)urea 383827 1-(4-(4-aminothieno[3,2-c]pyridin-3-yl)phenyl)-3-(3-fluorophenyl)urea 383828 1-(4-(4-aminothieno[3,2-c]pyridin-3-yl)phenyl)-3-(3-chlorophenyl)urea 383829 4'-hydroxy-4''-methylsulfamoyl-[1,1',3',1'']terphenyl-5'-carboxylic acid amide 383830 1-(4-(4-aminothieno[3,2-c]pyridin-3-yl)phenyl)-3-(3-cyanophenyl)urea 383831 4'-dimethylsulfamoyl-2-hydroxy-5-pyridin-4-yl-biphenyl-3-carboxylic acid amide 383832 1-(4-(4-aminothieno[3,2-c]pyridin-3-yl)phenyl)-3-(3,4-dimethylphenyl)urea 383833 1-(4-(4-aminothieno[3,2-c]pyridin-3-yl)phenyl)-3-(3,5-dimethylphenyl)urea 383834 1-(4-(4-aminothieno[3,2-c]pyridin-3-yl)phenyl)-3-cyclopentylurea 383835 1-(4-(4-aminothieno[3,2-c]pyridin-3-yl)phenyl)-3-cyclohexylurea 383836 1-(4-(4-aminothieno[3,2-c]pyridin-3-yl)phenyl)-3-(naphthalen-1-yl)urea 383837 1-(4-(4-aminothieno[3,2-c]pyridin-3-yl)phenyl)-3-(naphthalen-2-yl)urea 383838 1-(4-(4-aminothieno[3,2-c]pyridin-3-yl)phenyl)-3-(thiophen-2-yl)urea 383839 1-(4-(4-aminothieno[3,2-c]pyridin-3-yl)phenyl)-3-(thiophen-3-yl)urea 383840 1-(4-(4-amino-7-phenylthieno[3,2-c]pyridin-3-yl)phenyl)-3-m-tolylurea 383841 1-(4-(4-amino-7-(4-hydroxyphenyl)thieno[3,2-c]pyridin-3-yl)phenyl)-3-m-tolylurea 383842 2'-amino-3'-(aminocarbonyl)-5'-phenyl-N'-[3-(dimethylamino)propyl]-1,1'-biphenyl-4-sulfonohydrazide 383844 1-(4-(4-amino-7-(3-(methylcarbamoyl)phenyl)thieno[3,2-c]pyridin-3-yl)phenyl)-3-m-tolylurea 383846 2'-amino-3'-(aminocarbonyl)-5'-phenyl-N'-[3-(morpholino)propyl]-1,1'-biphenyl-4-sulfonohydrazide 383852 2'-amino-3'-(aminocarbonyl)-5'-phenyl-N'-[2-aminoethyl]-1,1'-biphenyl-4-sulfonohydrazide 383855 2'-amino-3'-(aminocarbonyl)-5'-phenyl-N'-[3-(methoxy)propyl]-1,1'-biphenyl-4-sulfonohydrazide 383860 1-(4-(4-amino-7-(pyridin-4-yl)thieno[3,2-c]pyridin-3-yl)phenyl)-3-m-tolylurea 383861 2'-amino-3'-(aminocarbonyl)-5'-phenyl-N'-cyclopropyl-1,1'-biphenyl-4-sulfonohydrazide 383868 1-(4-(4-amino-7-(pyrimidin-5-yl)thieno[3,2-c]pyridin-3-yl)phenyl)-3-m-tolylurea 383869 1-(4-(4-amino-7-(isoquinolin-4-yl)thieno[3,2-c]pyridin-3-yl)phenyl)-3-m-tolylurea 383871 2'-amino-3'-(aminocarbonyl)-5'-phenyl-N'-[2-(1-pyrrolidino)ethyl]-1,1'-biphenyl-4-sulfonohydrazide 383897 (1S,3R)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]cyclopentane-1-carboxamide 383898 (1S,3R)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-1-methyl-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]cyclopentane-1-carboxamide 383899 N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-1-ethyl-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]cyclopentane-1-carboxamide 383901 (1S,3R)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]-1-(propan-2-yl)cyclopentane-1-carboxamide 383902 (1S,3R)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]-1-propylcyclopentane-1-carboxamide 383903 (1R,3R)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-1-(2-methylpropyl)-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]cyclopentane-1-carboxamide 383904 N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-1-(cyclopropylmethyl)-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]cyclopentane-1-carboxamide 383905 (1R,3R)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-1-(cyclobutylmethyl)-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]cyclopentane-1-carboxamide 383906 N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-1-hexyl-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]cyclopentane-1-carboxamide 383907 N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-1-(methoxymethyl)-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]cyclopentane-1-carboxamide 383908 N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-1-cyclopropyl-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]cyclopentane-1-carboxamide 383909 (1R,3R)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]-1-[(methylsulfanyl)methyl]cyclopentane-1-carboxamide 383910 (1R,3R)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]-1-(methylsulfanyl)cyclopentane-1-carboxamide 383911 (1S,3R)-N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-1-methyl-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]cyclopentane-1-carboxamide 383912 1-ethyl-N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]cyclopentane-1-carboxamide 383913 (1S,3R)-N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]-1-(propan-2-yl)cyclopentane-1-carboxamide 383914 N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]-1-propylcyclopentane-1-carboxamide 383915 (1R,3R)-N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-1-(2-methylpropyl)-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]cyclopentane-1-carboxamide 383916 1-(cyclopropylmethyl)-N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]cyclopentane-1-carboxamide 383917 1-(cyclobutylmethyl)-N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]cyclopentane-1-carboxamide 383918 N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-1-hexyl-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]cyclopentane-1-carboxamide 383919 N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-1-(methoxymethyl)-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]cyclopentane-1-carboxamide 383920 (1S,3R)-1-cyclopropyl-N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]cyclopentane-1-carboxamide 383921 (1R,3R)-N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]-1-[(methylsulfanyl)methyl]cyclopentane-1-carboxamide 383922 (1R,3R)-N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-[(1S,5'R)-5'-methylspiro[indene-1,4'-piperidine]-1'-yl]-1-(methylsulfanyl)cyclopentane-1-carboxamide 383959 4-butyl-N-(isoindolin-5-yl)benzenesulfonamide 383960 4-butyl-N-(2-methylisoindolin-5-yl)benzenesulfonamide 383961 4-butyl-N-(1,2,3,4-tetrahydroisoquinolin-6-yl)benzenesulfonamide 383962 4-butyl-N-(2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)benzenesulfonamide 383963 4-butyl-N-(2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)benzenesulfonamide 383964 4-butyl-N-(3-methyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)benzenesulfonamide 383965 4'-chloro-biphenyl-4-sulfonic acid (3-methyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)-amide 383966 3'-chloro-4'-fluoro-biphenyl-4-sulfonic acid (3-methyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)-amide 383967 4'-cyano-biphenyl-4-sulfonic acid (3-methyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)-amide 383968 4'-chloro-2-methyl-biphenyl-4-sulfonic acid (3-methyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)-amide 383969 5-(4-chlorophenyl)-N-(3-methyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)thiophene-2-sulfonamide 383970 N-(3-methyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)-4-(5-methylthiophen-2-yl)benzenesulfonamide 383971 4-(3,5-dimethylisoxazol-4-yl)-N-(3-methyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)benzenesulfonamide 383972 4'-chloro-biphenyl-4-sulfonic acid (3,8-dimethyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)-amide 383974 4'-chloro-biphenyl-4-sulfonic acid (8-isopropyl-3-methyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)-amide 383977 4'-chloro-biphenyl-4-sulfonic acid (8-bromo-3-methyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)-amide 383980 4'-chloro-biphenyl-4-sulfonic acid (8-chloro-3-methyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)-amide 383983 4'-chloro-biphenyl-4-sulfonic acid (8-methoxy-3-methyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)-amide 383985 4'-chloro-biphenyl-4-sulfonic acid (8-isopropoxy-3-methyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)-amide 383987 4'-chloro-biphenyl-4-sulfonic acid (8-isopropylamino-3-methyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)-amide 384021 Z-{2-(Hydroxymethyl)-4-[5-methyl-3-(2-methylpropyl)hexylidene]-5-oxo-2-(2,3-dihydrofuryl)}methyl 3-Methylbutanoate 384022 Z-[2-(Hydroxymethyl)-4-(3-methylbutylidene)-5-oxo-2-(2,3-dihydrofuryl)]methyl 5-Methyl-3-(2-methylpropyl)hexanoate 384023 {2-(hydroxymethyl)-5-[5-methyl-3-(2-methylpropyl)hexylidene]-4-oxo-1,3-dioxolan-2-yl}methyl 2,2-dimethylpropanoate 384062 methyl-(1-methyl-3,5,11b-triaza-cyclopenta[a]anthracen-4-yl)-amine 384066 2-(1-methyl-3,5,11b-triaza-cyclopenta[a]anthracen-4-ylamino)-ethanol 384067 (1-methyl-3,5,11b-triaza-cyclopenta[a]anthracen-4-yl)-(2-piperidin-1-yl-ethyl)-amine 384068 methyl-(1-methyl-3,3a,5-triaza-cyclopenta[a]anthracen-4-yl)-amine 384069 N-methyl-N'-(1-methyl-3,3a,5-triaza-cyclopenta[a]anthracen-4-yl)-ethane-1,2-diamine 384070 methyl-(1-methyl-1H-1,3,5-triaza-cyclopenta[a]anthracen-4-yl)-amine 384071 N*1*-(1-methyl-1H-1,3,5-triaza-cyclopenta[a]anthracen-4-yl)-ethane-1,2-diamine 384072 (Z)-3-((4-(2-carboxyethyl)-4,5,6,7-tetrahydro-1H-indol-2-yl)methylene)-2-oxoindoline-5-carboxylic acid 384074 {2-(hydroxymethyl)-5-[5-methyl-3-(2-methylpropyl)hexylidene]-4-oxo-1,3-dioxolan-2-yl}methyl 3-methylbutanoate 384075 {2-(hydroxymethyl)-5-[5-methyl-3-(2-methylpropyl)hexylidene]-4-oxo-1,3-dioxolan-2-yl}methyl 3-methylbutanoate 384076 (Z)-3-(2-((5-bromo-2-oxoindolin-3-ylidene)methyl)-4,5,6,7-tetrahydro-1H-indol-4-yl)propanoic acid 384077 1-(2-fluoro-benzyl)-8-(4-imidazol-1-yl-benzyl)-3-(3-methoxy-phenyl)-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384078 1-(2-fluoro-benzyl)-8-(4-imidazol-1-yl-benzyl)-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384079 3-(2-((2-oxoindolin-3-ylidene)methyl)-4,5,6,7-tetrahydro-1H-indol-4-yl)propanoic acid 384080 3-ethyl-1-(2-fluoro-benzyl)-8-(4-imidazol-1-yl-benzyl)-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384081 2-chloro-4-fluoro-5-(7-(2-methoxyethoxy)quinazolin-4-ylamino)phenol 384082 3-butyl-1-(2-fluoro-benzyl)-8-(4-imidazol-1-yl-benzyl)-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384083 3-cyclohexyl-1-(2-fluoro-benzyl)-8-(4-imidazol-1-yl-benzyl)-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384084 1-(2-fluoro-benzyl)-8-(4-imidazol-1-yl-benzyl)-3-phenyl-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384085 3-benzyl-1-(2-fluoro-benzyl)-8-(4-imidazol-1-yl-benzyl)-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384086 1-(2-fluoro-benzyl)-8-(4-imidazol-1-yl-benzyl)-3-phenethyl-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384087 3-((1H-pyrrol-2-yl)methylene)-4-methylindolin-2-one 384088 1-(2-fluoro-benzyl)-8-(4-imidazol-1-yl-benzyl)-3-naphthalen-1-yl-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384089 1-(2-fluoro-benzyl)-8-(4-imidazol-1-yl-benzyl)-3-(1,2,3,4-tetrahydro-naphthalen-1-yl)-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384090 1-(2-fluoro-benzyl)-3-(3-methoxy-phenyl)-8-[4-(2-methyl-imidazol-1-yl)-benzyl]-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384091 1-(2-fluoro-benzyl)-3-(3-methoxy-phenyl)-8-(4-pyrrol-1-yl-benzyl)-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384092 1-(2-fluoro-benzyl)-3-(3-methoxy-phenyl)-8-(4-pyridin-3-yl-benzyl)-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384093 1-(2-fluoro-benzyl)-3-(3-methoxy-phenyl)-8-(4-pyridin-4-yl-benzyl)-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384094 1-(2-fluoro-benzyl)-3-(3-methoxy-phenyl)-8-(4-pyrimidin-5-yl-benzyl)-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384095 1-(2-fluoro-benzyl)-3-(3-methoxy-phenyl)-8-[4-(6-methyl-pyridin-3-yl)-benzyl]-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384096 1-(2-fluoro-benzyl)-3-(3-methoxy-phenyl)-8-[4-(6-methoxy-pyridin-3-yl)-benzyl]-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384097 8-[4-(6-amino-pyridin-3-yl)-benzyl]-1-(2-fluoro-benzyl)-3-(3-methoxy-phenyl)-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384098 ethyl 5-isopropyl-4-(5-(methoxycarbamoyl)-2,4-dimethylphenylamino)pyrrolo[1,2-f][1,2,4]triazine-6-carboxylate 384099 1-(2-fluoro-benzyl)-3-(3-methoxy-phenyl)-8-[4-(5-methoxy-pyridin-3-yl)-benzyl]-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384100 5-{4-[1-(2-fluoro-benzyl)-3-(3-methoxy-phenyl)-2,4-dioxo-1,3,8-triaza-spiro[4.5]dec-8-ylmethyl]-phenyl}-nicotinonitrile 384101 1-(2-fluoro-benzyl)-3-(3-methoxy-phenyl)-8-[4-(4-methoxy-pyridin-3-yl)-benzyl]-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384102 8-[4-(4-chloro-pyridin-3-yl)-benzyl]-1-(2-fluoro-benzyl)-3-(3-methoxy-phenyl)-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384103 5-(6,7-bis(2-methoxyethoxy)quinazolin-4-ylamino)-2-chloro-4-fluorophenol 384104 8-biphenyl-4-ylmethyl-1-(2-fluoro-benzyl)-3-(3-methoxy-phenyl)-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384106 (Z)-3-(2-((6-methoxy-2-oxoindolin-3-ylidene)methyl)-4,5,6,7-tetrahydro-1H-indol-4-yl)propanoic acid 384107 4'-[1-(2-fluoro-benzyl)-3-(3-methoxy-phenyl)-2,4-dioxo-1,3,8-triaza-spiro[4.5]dec-8-ylmethyl]-biphenyl-3-carbonitrile 384108 4'-[1-(2-fluoro-benzyl)-3-(3-methoxy-phenyl)-2,4-dioxo-1,3,8-triaza-spiro[4.5]dec-8-ylmethyl]-biphenyl-4-carbonitrile 384109 8-methyl-4H,7H-indolo[6,5,4-cd]indol-5-one 384110 1-(2-fluoro-benzyl)-8-(3'-methoxy-biphenyl-4-ylmethyl)-3-(3-methoxy-phenyl)-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384111 N-(2,4-dimethylphenyl)-6,7-dimethoxyquinazolin-4-amine 384112 N-{4'-[1-(2-fluoro-benzyl)-3-(3-methoxy-phenyl)-2,4-dioxo-1,3,8-triaza-spiro[4.5]dec-8-ylmethyl]-biphenyl-3-yl}-acetamide 384113 3-((3-bromothiophen-2-yl)methylene)indolin-2-one 384114 N-{4'-[1-(2-fluoro-benzyl)-3-(3-methoxy-phenyl)-2,4-dioxo-1,3,8-triaza-spiro[4.5]dec-8-ylmethyl]-biphenyl-3-yl}-methanesulfonamide 384115 1-(2-fluoro-benzyl)-8-(3'-hydroxy-biphenyl-4-ylmethyl)-3-(3-methoxy-phenyl)-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384116 8-(3'-acetyl-biphenyl-4-ylmethyl)-1-(2-fluoro-benzyl)-3-(3-methoxy-phenyl)-1,3,8-triaza-spiro[4.5]decane-2,4-dione 384117 3-({4'-[1-(2-fluoro-benzyl)-3-(3-methoxy-phenyl)-2,4-dioxo-1,3,8-triaza-spiro[4.5]dec-8-ylmethyl]-biphenyl-3-yl}-methyl-amino)-propionitrile 384118 4'-[3-(3-methoxy-phenyl)-2,4-dioxo-1,3,8-triaza-spiro[4.5]dec-8-ylmethyl]-biphenyl-3-carbonitrile 384119 4'-[3-(3-methoxy-phenyl)-1-methyl-2,4-dioxo-1,3,8-triaza-spiro[4.5]dec-8-ylmethyl]-biphenyl-3-carbonitrile 384120 4'-[1-cyclopropyl-3-(3-methoxy-phenyl)-2,4-dioxo-1,3,8-triaza-spiro[4.5]dec-8-ylmethyl]-biphenyl-3-carbonitrile 384122 4'-[1-cyclopropylmethyl-3-(3-methoxy-phenyl)-2,4-dioxo-1,3,8-triaza-spiro[4.5]dec-8-ylmethyl]-biphenyl-3-carbonitrile 384124 4'-[1-cyclohexyl-3-(3-methoxy-phenyl)-2,4-dioxo-1,3,8-triaza-spiro[4.5]dec-8-ylmethyl]-biphenyl-3-carbonitrile 384126 4'-[1-cyclohexylmethyl-3-(3-methoxy-phenyl)-2,4-dioxo-1,3,8-triaza-spiro[4.5]dec-8-ylmethyl]-biphenyl-3-carbonitrile 384127 4'-[3-(3-methoxy-phenyl)-2,4-dioxo-1-phenyl-1,3,8-triaza-spiro[4.5]dec-8-ylmethyl]-biphenyl-3-carbonitrile 384129 4'-(2,4-dioxo-1-phenyl-1,3,8-triaza-spiro[4.5]dec-8-ylmethyl)-biphenyl-3-carbonitrile 384131 4'-(2,4-dioxo-1-phenyl-3-m-tolyl-1,3,8-triaza-spiro[4.5]dec-8-ylmethyl)-biphenyl-3-carbonitrile 384133 5-chloro-4'-(2,4-dioxo-1-phenyl-1,3,8-triaza-spiro[4.5]dec-8-ylmethyl)-biphenyl-3-carbonitrile 384184 3-(5-((6-(3,5-dimethoxyphenyl)-2-oxoindolin-3-ylidene)methyl)-2,4-dimethyl-1H-pyrrol-3-yl)propanoic acid 384195 4-(bis(2-chloroethyl)amino)-N-(4-methyl-3-(4-(pyridin-3-yl)pyrimidin-2-ylamino)phenyl)benzamide 384197 4-(((2-chloroethyl)(methyl)amino)methyl)-N-(4-methyl-3-(4-(pyridin-3-yl)pyrimidin-2-ylamino)phenyl)benzamide 384200 4-amino-N-(4-methyl-3-(4-(pyridin-3-yl)pyrimidin-2-ylamino)phenyl)-3-(trifluoromethyl)benzamide 384202 N-(4-methyl-3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)-4-(3-methyltriaz-1-en-1-yl)-3-(trifluoromethyl)benzamide 384204 4-(3,3-dimethyltriaz-1-en-1-yl)-N-(4-methyl-3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)-3-(trifluoromethyl)benzamide 384207 4-[3-(hydroxymethyl)-3-methyltriaz-1-en-1-yl]-N-(4-methyl-3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)-3-(trifluoromethyl)benzamide 384208 3-chloro-N-(4-methyl-3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)-4-(3-methyltriaz-1-en-1-yl)benzamide 384209 4-[3-(hydroxymethyl)-3-methyltriaz-1-en-1-yl]-N-(4-methyl-3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamide 384311 N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)-2-methyl-2-(5-(trifluoromethyl)pyridin-3-yloxy)propanamide 384319 N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)butane-1-sulfonamide 384321 N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)-2-methylpropane-2-sulfonamide 384322 N1-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N1-methyl-N3-phenylmalonamide 384324 N1-benzyl-N3-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N3-methylmalonamide 384326 N1-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N1-methyl-N3-(4-(methylsulfonamido)phenyl)malonamide 384327 N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)benzenesulfonamide 384328 N1-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N1-methyl-N3-(4-(methylsulfonamidomethyl)phenyl)malonamide 384331 N1-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N1-methyl-N4-phenylsuccinamide 384332 1-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-1-methyl-3-(2-oxo-2-(phenylamino)ethyl)urea 384334 N1-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N1-methyl-N3-(thiazol-2-yl)malonamide 384336 N1-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N1-methyl-N4-(thiazol-2-yl)succinamide 384338 N1-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N1-methyl-N3-(pyridin-3-yl)malonamide 384339 N1-((S)-2-((S)-3-hydroxypyrrolidin-1-yl)-1-phenylethyl)-N1-methyl-N4-(pyridin-3-yl)succinamide 384341 2-chloro-N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)benzenesulfonamide 384344 3-chloro-N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)benzenesulfonamide 384348 4-chloro-N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)benzenesulfonamide 384351 2,3-dichloro-N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)benzenesulfonamide 384357 2,4-dichloro-N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)benzenesulfonamide 384370 2,5-dichloro-N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)benzenesulfonamide 384372 2,6-dichloro-N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)benzenesulfonamide 384373 3,5-dichloro-N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)benzenesulfonamide 384376 2,4,5-trichloro-N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)benzenesulfonamide 384378 N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)-3,5-bis(trifluoromethyl)benzenesulfonamide 384380 N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)-3,5-difluorobenzenesulfonamide 384382 biphenyl-3-sulfonic acid [(1S,2S)-3-(4-chloro-phenyl)-2-(3-cyano-phenyl)-1-methyl-propyl]-amide 384383 biphenyl-4-sulfonic acid [(1S,2S)-3-(4-chloro-phenyl)-2-(3-cyano-phenyl)-1-methyl-propyl]-amide 384385 N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)naphthalene-1-sulfonamide 384386 N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)naphthalene-2-sulfonamide 384389 N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)(phenyl)methanesulfonamide 384394 (2-chlorophenyl)-N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)methanesulfonamide 384399 (3-chlorophenyl)-N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)methanesulfonamide 384400 (4-chlorophenyl)-N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)methanesulfonamide 384401 N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)-2-phenylethanesulfonamide 384405 (E)-N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)-2-phenylethenesulfonamide 384418 N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)benzamide 384422 3,5-dichloro-N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)benzamide 384430 2,6-dichloro-N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)benzamide 384432 N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)-2-phenylacetamide 384437 N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)-3-phenylpropanamide 384893 N-(3-{4-[4-(1-Cyclobutanecarbonyl-piperidin-4-yloxy)-3-methyl-phenylamino]-quinazolin-6-yl}-prop-2-ynyl)-2-methoxy-acetamide 384894 N-[3-(4-{4-[1-(3-Chloro-benzoyl)-piperidin-4-yloxy]-3-methyl-phenylamino}-quinazolin-6-yl)-prop-2-ynyl]-2-methoxy-acetamide 384895 N-(3-(4-(4-(1-(3,3-dimethylbutanoyl)piperidin-4-yloxy)-3-methylphenylamino)quinazolin-6-yl)prop-2-ynyl)-2-methoxyacetamide 384897 2-methoxy-N-[3-(4-{3-methyl-4-[1-(tetrahydro-furan-2-carbonyl)-piperidin-4-yloxy]-phenylamino}-quinazolin-6-yl)-prop-2-ynyl]-acetamide 384898 N-(2,6-difluorophenyl)-4-(4-(6-(3-(2-methoxyacetamido)prop-1-ynyl)quinazolin-4-ylamino)-2-methylphenoxy)piperidine-1-carboxamide 384901 3-(4-(6-(3-(2-methoxyacetamido)prop-1-ynyl)quinazolin-4-ylamino)-2-methylphenoxy)-N-phenylbenzamide 384902 N-cyclobutyl-3-(4-(6-(3-(2-methoxyacetamido)prop-1-ynyl)quinazolin-4-ylamino)-2-methylphenoxy)benzamide 384903 N-tert-butyl-3-(4-(6-(3-(2-methoxyacetamido)prop-1-ynyl)quinazolin-4-ylamino)-2-methylphenoxy)benzamide 384904 3-(4-(6-(3-(2-methoxyacetamido)prop-1-ynyl)quinazolin-4-ylamino)-2-methylphenoxy)-N-neopentylbenzamide 384909 4-(4-(6-(3-(2-methoxyacetamido)prop-1-ynyl)quinazolin-4-ylamino)-2-methylphenoxy)-N-neopentylbenzamide 384910 1-(4-(4-(6,7-dimethoxyquinazolin-4-ylamino)-2-methylphenoxy)piperidin-1-yl)-3,3-dimethylbutan-1-one 384911 1-(4-(4-(6,7-bis(2-methoxyethoxy)quinazolin-4-ylamino)-2-methylphenoxy)piperidin-1-yl)-3,3-dimethylbutan-1-one 384912 1-(4-(4-(6-methoxyquinazolin-4-ylamino)-2-methylphenoxy)piperidin-1-yl)-3,3-dimethylbutan-1-one 384913 1-(4-(4-(6-(2-methoxyethoxy)quinazolin-4-ylamino)-2-methylphenoxy)piperidin-1-yl)-3,3-dimethylbutan-1-one 384914 N-(3-methyl-4-(1-methylpiperidin-4-yloxy)phenyl)-6-(3-morpholinopropoxy)quinazolin-4-amine 384915 1-(4-(4-(6-(dimethylamino)pyrido[3,4-d]pyrimidin-4-ylamino)-2-methylphenoxy)piperidin-1-yl)-3,3-dimethylbutan-1-one 384916 3,3-dimethyl-1-(4-(2-methyl-4-(6-morpholinopyrido[3,4-d]pyrimidin-4-ylamino)phenoxy)piperidin-1-yl)butan-1-one 384917 N-(2,6-difluorophenyl)-4-(4-(6,7-dimethoxyquinazolin-4-ylamino)-2-methylphenoxy)piperidine-1-carboxamide 384918 4-(4-(6,7-bis(2-methoxyethoxy)quinazolin-4-ylamino)-2-methylphenoxy)-N-(2,6-difluorophenyl)piperidine-1-carboxamide 384919 N-(2,6-difluorophenyl)-4-(4-(6-methoxyquinazolin-4-ylamino)-2-methylphenoxy)piperidine-1-carboxamide 384920 N-(2,6-difluorophenyl)-4-(4-(6-(2-methoxyethoxy)quinazolin-4-ylamino)-2-methylphenoxy)piperidine-1-carboxamide 384921 N-(2,6-difluorophenyl)-4-(2-methyl-4-(6-(3-morpholinopropoxy)quinazolin-4-ylamino)phenoxy)piperidine-1-carboxamide 384922 N-(2,6-difluorophenyl)-4-(2-methyl-4-(6-(methylamino)pyrido[3,4-d]pyrimidin-4-ylamino)phenoxy)piperidine-1-carboxamide 384923 N-(2,6-difluorophenyl)-4-(4-(6-(dimethylamino)pyrido[3,4-d]pyrimidin-4-ylamino)-2-methylphenoxy)piperidine-1-carboxamide 384924 N-(2,6-difluorophenyl)-4-(2-methyl-4-(6-morpholinopyrido[3,4-d]pyrimidin-4-ylamino)phenoxy)piperidine-1-carboxamide 384925 (4-(4-(6,7-bis(2-methoxyethoxy)quinazolin-4-ylamino)-2-methylphenoxy)piperidin-1-yl)(cyclopentyl)methanone 384926 cyclopentyl(4-(4-(6-(2-methoxyethoxy)quinazolin-4-ylamino)-2-methylphenoxy)piperidin-1-yl)methanone 384927 cyclopentyl(4-(2-methyl-4-(6-morpholinopyrido[3,4-d]pyrimidin-4-ylamino)phenoxy)piperidin-1-yl)methanone 384928 4-(4-(6,7-dimethoxyquinazolin-4-ylamino)-2-methylphenoxy)-N-neopentylbenzamide 384929 4-(2-methyl-4-(6-(methylamino)pyrido[3,4-d]pyrimidin-4-ylamino)phenoxy)-N-neopentylbenzamide 384930 4-(2-methyl-4-(6-(2-morpholinoethylamino)pyrido[3,4-d]pyrimidin-4-ylamino)phenoxy)-N-neopentylbenzamide 384931 4-(4-(6-(dimethylamino)pyrido[3,4-d]pyrimidin-4-ylamino)-2-methylphenoxy)-N-neopentylbenzamide 384932 4-(2-methyl-4-(6-(pyrrolidin-1-yl)pyrido[3,4-d]pyrimidin-4-ylamino)phenoxy)-N-neopentylbenzamide 384933 4-(2-methyl-4-(6-morpholinopyrido[3,4-d]pyrimidin-4-ylamino)phenoxy)-N-neopentylbenzamide 384934 4-(2-methyl-4-(6-(4-methylpiperazin-1-yl)pyrido[3,4-d]pyrimidin-4-ylamino)phenoxy)-N-neopentylbenzamide 384960 2-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-methyl-5-(piperidin-1-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384961 2-(4-chlorophenyl)-5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384964 5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-2-phenyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384965 5-cyclohexyl-1-(2,4-dichlorophenyl)-2-(4-fluorophenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384966 5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-2-p-tolyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384967 5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-2-(4-(trifluoromethyl)phenyl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384968 5-cyclohexyl-1-(2,4-dichlorophenyl)-2-(4-methoxyphenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384969 5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-2-(4-vinylphenyl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384970 2-(4-aminophenyl)-5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384973 5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-2-m-tolyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384974 5-cyclohexyl-1-(2,4-dichlorophenyl)-2-(3-methoxyphenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384975 5-cyclohexyl-1-(2,4-dichlorophenyl)-2-(3,4-dimethoxyphenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384976 2-(benzo[d][1,3]dioxol-5-yl)-5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384977 5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-2-(3-(trifluoromethyl)phenyl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384978 2-(3-aminophenyl)-5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384979 5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-2-(thiophen-3-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384980 5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-2-(thiophen-2-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384981 5-cyclohexyl-1-(2,4-dichlorophenyl)-2-(furan-2-yl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384982 2-(benzo[b]thiophen-2-yl)-5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384983 5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-2-(pyridin-3-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384984 5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384985 1-(2-chlorophenyl)-2-(4-chlorophenyl)-5-cyclohexyl-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384986 2-(4-chlorophenyl)-5-cyclohexyl-1-(2,6-dichlorophenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384987 1-(2-chlorophenyl)-5-cyclohexyl-2-(4-methoxyphenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384988 5-cyclohexyl-2-(4-methoxyphenyl)-3-methyl-1-o-tolyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384989 5-cyclohexyl-3-methyl-1-o-tolyl-2-(4-(trifluoromethyl)phenyl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384990 5-cyclohexyl-2-(4-fluorophenyl)-3-methyl-1-o-tolyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384991 1-(2-chlorophenyl)-2-(4-chlorophenyl)-3-methyl-5-(piperidin-1-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384992 1-(2-chlorophenyl)-2-(4-methoxyphenyl)-3-methyl-5-(piperidin-1-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 384993 2-(4-methoxyphenyl)-3-methyl-5-(piperidin-1-yl)-1-o-tolyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 385053 2,6-dihydroxy-3',5'-dimethyl-biphenyl-4-carboxylic acid pentyl ester 385054 2-hydroxy-6-methoxy-3',5'-dimethyl-biphenyl-4-carboxylic acid pentyl ester 385058 2,6-dihydroxy-biphenyl-4-carboxylic acid pentyl ester 385060 2,6-dihydroxy-3',5'-dimethyl-biphenyl-4-carboxylic acid butyl ester 385061 2,6-dihydroxy-3',5'-dimethyl-biphenyl-4-carboxylic acid methyl ester 385062 2-hydroxy-6-methoxy-3',5'-dimethyl-biphenyl-4-carboxylic acid methyl ester 385065 2,6-dimethoxy-3',5'-dimethyl-biphenyl-4-carboxylic acid 385087 N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide 385089 N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide 385092 3,4-difluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 385093 3,4-difluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 385094 N-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide 385095 N-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide 385096 5-chloro-N-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 385097 5-chloro-N-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 385098 5-chloro-N-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-fluorobenzenesulfonamide 385099 5-chloro-N-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-fluorobenzenesulfonamide 385100 N-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzo[d][1,3]dioxole-5-sulfonamide 385101 N-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzo[d][1,3]dioxole-5-sulfonamide 385102 3,4-dimethoxy-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 385103 3,4-dimethoxy-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 385104 N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-2,3-dihydrobenzo[b][1,4]dioxine-6-sulfonamide 385105 N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-2,3-dihydrobenzo[b][1,4]dioxine-6-sulfonamide 385107 5-chloro-2-methoxy-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 385108 5-chloro-2-methoxy-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 385110 5-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 385111 5-chloro-2-fluoro-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 385113 3-(difluoromethoxy)-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 385114 3-(difluoromethoxy)-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 385115 4-(difluoromethoxy)-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 385116 4-(difluoromethoxy)-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 385117 N-((1s,4s)-4-(4-(2-(2-fluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide 385118 N-((1r,4r)-4-(4-(2-(2-fluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide 385119 N-((1s,4s)-4-(4-(2-(2,2-difluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide 385120 N-((1r,4r)-4-(4-(2-(2,2-difluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide 385121 N-((1s,4s)-4-(4-(4-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide 385122 N-((1r,4r)-4-(4-(4-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide 385123 N-((1s,4s)-4-(4-(5-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide 385124 N-((1r,4r)-4-(4-(5-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide 385208 N2-[(2,2-diphenylethoxy)acetyl]-L-arginine 385209 (S)-2-(2-benzhydrylfuran-5-carboxamido)-5-guanidinopentanoic acid 385210 (2R)-2-(2-(3-fluorophenyl)furan-5-carboxamido)-5-guanidinopentanoic acid 385211 (2R)-5-guanidino-2-(2-m-tolylfuran-5-carboxamido)pentanoic acid 385212 (2R)-5-guanidino-2-(2-(3-methoxyphenyl)furan-5-carboxamido)pentanoic acid 385213 (2R)-2-(2-(3-ethoxyphenyl)furan-5-carboxamido)-5-guanidinopentanoic acid 385214 (2R)-5-guanidino-2-(2-(3-(hydroxymethyl)phenyl)furan-5-carboxamido)pentanoic acid 385215 (2R)-2-(2-(3-cyanophenyl)furan-5-carboxamido)-5-guanidinopentanoic acid 385216 (2R)-2-(2-(3-chlorophenyl)furan-5-carboxamido)-5-guanidinopentanoic acid 385217 (2R)-2-(2-(3-chloro-4-fluorophenyl)furan-5-carboxamido)-5-guanidinopentanoic acid 385218 (2R)-2-(2-(5-chloro-2-methylphenyl)furan-5-carboxamido)-5-guanidinopentanoic acid 385220 (2R)-2-(2-(2,5-dichlorophenyl)furan-5-carboxamido)-5-guanidinopentanoic acid 385223 (2R)-2-(2-(benzo[b]thiophen-3-yl)furan-5-carboxamido)-5-guanidinopentanoic acid 385224 (R)-2-[(5-dibenzofuran-4-yl-furan-2-carbonyl)-amino]-5-guanidino-pentanoic acid 385225 (R)-2-[(3'-chloro-biphenyl-4-carbonyl)-amino]-5-guanidino-pentanoic acid 385226 (R)-2-[(3'-chloro-biphenyl-3-carbonyl)-amino]-5-guanidino-pentanoic acid 385228 (2R)-2-(2-(3-chlorophenyl)thiophene-5-carboxamido)-5-guanidinopentanoic acid 385230 (R)-2-(1-benzhydrylpiperazine-4-carboxamido)-5-guanidinopentanoic acid 385232 (R)-2-(4-benzhydrylbenzamido)-5-guanidinopentanoic acid 385241 (R)-2-(2-(bis(3-fluorophenyl)methyl)furan-5-carboxamido)-5-guanidinopentanoic acid 385242 (R)-2-(2-(bis(3-chlorophenyl)methyl)furan-5-carboxamido)-5-guanidinopentanoic acid 385243 (R)-2-(2-(bis(4-chlorophenyl)methyl)furan-5-carboxamido)-5-guanidinopentanoic acid 385254 N-(1-benzylpiperidine-4-yl)-1-naphthamide 385256 N-(1-phenethylpiperidin-4-yl)-1-naphthamide 385257 N-(1-(1-phenylethyl)piperidin-4-yl)-1-naphthamide 385258 N-(1-(3-phenylpropyl)piperidin-4-yl)-1-naphthamide 385259 (S)-N-(1-(1-hydroxy-1-phenylpropyl)piperidin-4-yl)-1-naphthamide 385262 N-(1-(4-phenylbutyl)piperidin-4-yl)-1-naphthamide 385264 naphthalen-1-yl(4-(phenethylamino)piperidin-1-yl)methanone 385268 N-(1-benzylpiperidine-4-yl)-2-naphthamide 385269 N-(1-phenethylpiperidin-4-yl)-2-naphthamide 385270 N-(1-(1-phenylethyl)piperidin-4-yl)-2-naphthamide 385271 N-(1-(3-phenylpropyl)piperidin-4-yl)-2-naphthamide 385272 N-(1-(4-phenylbutyl)piperidin-4-yl)-2-naphthamide 385273 (4-(benzylamino)piperidin-1-yl)(naphthalen-2-yl)methanone 385274 naphthalen-2-yl(4-(phenethylamino)piperidin-1-yl)methanone 385275 naphthalen-2-yl(4-(3-phenylpropylamino)piperidin-1-yl)methanone 385359 (R)-N-(2-(dimethylamino)ethyl)-N-(1-(3-(4-fluorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)decanamide 385468 Ser-Tyr-Ser-Nle-Glu-His-Dphe-Arg 385469 (4S)-4-{[(1S)-1-{[(1R)-1-{[(1S)-1-{[(1S)-1-[({[(2S)-6-amino-1-[(2S)-2-{[(1S)-1-carbamoyl-2-methylpropyl]carbamoyl}pyrrolidin-1-yl]-1-oxohexan-2-yl]carbamoyl}methyl)carbamoyl]-2-(1H-indol-3-yl)ethyl]carbamoyl}-4-carbamimidamidobutyl]carbamoyl}-2-phenylethyl]carbamoyl}-2-(1H-imidazol-5-yl)ethyl]carbamoyl}-4-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-(hex-5-ynamido)-3-hydroxypropanamido]-3-(4-hydroxyphenyl)propanamido]-3-hydroxypropanamido]hexanamido]butanoic acid 385470 (4S)-4-{[(1S)-1-{[(1R)-1-{[(1S)-1-{[(1S)-1-[({[(2S)-6-amino-1-[(2S)-2-{[(1S)-1-carboxy-2-methylpropyl]carbamoyl}pyrrolidin-1-yl]-1-oxohexan-2-yl]carbamoyl}methyl)carbamoyl]-2-(1H-indol-3-yl)ethyl]carbamoyl}-4-carbamimidamidobutyl]carbamoyl}-2-phenylethyl]carbamoyl}-2-(1H-imidazol-5-yl)ethyl]carbamoyl}-4-[(2S)-2-[(2S)-3-hydroxy-2-[(2S)-2-[(2S)-3-hydroxy-2-[4-(1-{6-[(3,7,14,18,22-pentahydroxy-2,6,10,15,19,23-hexamethyltetracosan-11-yl)oxy]hexyl}-1H-1,2,3-triazol-4-yl)butanamido]propanamido]-3-(4-hydroxyphenyl)propanamido]propanamido]hexanamido]butanoic acid 385472 (4S)-4-{[(1S)-1-{[(1R)-1-{[(1S)-1-{[(1S)-1-[({[(2S)-6-amino-1-[(2S)-2-{[(1S)-1-carboxy-2-methylpropyl]carbamoyl}pyrrolidin-1-yl]-1-oxohexan-2-yl]carbamoyl}methyl)carbamoyl]-2-(1H-indol-3-yl)ethyl]carbamoyl}-4-carbamimidamidobutyl]carbamoyl}-2-phenylethyl]carbamoyl}-2-(1H-imidazol-5-yl)ethyl]carbamoyl}-4-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-{4-[1-(6-{[14-({6-[4-(3-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1R)-1-{[(1S)-1-{[(1S)-1-[({[(2S)-6-amino-1-[(2S)-2-{[(1S)-1-carboxy-2-methylpropyl]carbamoyl}pyrrolidin-1-yl]-1-oxohexan-2-yl]carbamoyl}methyl)carbamoyl]-2-(1H-indol-3-yl)ethyl]carbamoyl}-4-carbamimidamidobutyl]carbamoyl}-2-phenylethyl]carbamoyl}-2-(1H-imidazol-5-yl)ethyl]carbamoyl}-3-carboxypropyl]carbamoyl}pentyl]carbamoyl}-2-hydroxyethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]carbamoyl}-2-hydroxyethyl]carbamoyl}propyl)-1H-1,2,3-triazol-1-yl]hexyl}oxy)-7,11,18,22-tetrahydroxy-2,6,10,15,19,23-hexamethyltetracosan-3-yl]oxy}hexyl)-1H-1,2,3-triazol-4-yl]butanamido}-3-hydroxypropanamido]-3-(4-hydroxypheny 385473 His-DPhe-Arg-Trp 385476 N-[(1S)-1-{[(1R)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-(1H-indol-3-yl)ethyl]carbamoyl}butyl]carbamoyl}-2-phenylethyl]carbamoyl}-2-(1H-imidazol-5-yl)ethyl]hex-5-ynamide 385480 (2S)-5-carbamimidamido-2-[(2S)-2-[(2S)-2-{4-[1-(6-{[14-({6-[4-(3-{[(1S)-1-{[(1S)-1-{[(1R)-4-carbamimidamido-1-{[(1S)-1-carbamoyl-2-(1H-indol-3-yl)ethyl]carbamoyl}butyl]carbamoyl}-2-phenylethyl]carbamoyl}-2-(1H-imidazol-5-yl)ethyl]carbamoyl}propyl)-1H-1,2,3-triazol-1-yl]hexyl}oxy)-7,11,18,22-tetrahydroxy-2,6,10,15,19,23-hexamethyltetracosan-3-yl]oxy}hexyl)-1H-1,2,3-triazol-4-yl]butanamido}-3-(1H-imidazol-5-yl)propanamido]-3-phenylpropanamido]-N-[(1S)-1-carbamoyl-2-(1H-indol-3-yl)ethyl]pentanamide 385495 5-(2-(2-(4-fluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-2-fluorobenzoic acid 385496 5-(2-(2-(benzyloxy)-5-(trifluoromethyl)phenyl)-5-methyl-1H-pyrrol-1-yl)-2-fluorobenzoic acid 385497 5-(2-(2-(4-fluorobenzyloxy)-5-(trifluoromethyl)phenyl)-5-methyl-1H-pyrrol-1-yl)-2-fluorobenzoic acid 385498 5-(2-(2-(4-fluorobenzyloxy)-5-methylphenyl)-5-methyl-1H-pyrrol-1-yl)-2-fluorobenzoic acid 385499 5-(2-(2-(4-fluorobenzyloxy)-5-fluorophenyl)-5-methyl-1H-pyrrol-1-yl)-2-fluorobenzoic acid 385500 5-(2-(2-(4-fluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-2-chlorobenzoic acid 385510 5-(2-(2-(4-fluorobenzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-2-methylbenzoic acid 385514 5-(2-(2-(2,4-difluorobenzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-2-methylbenzoic acid 385517 5-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-2-methylbenzoic acid 385520 5-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-2-hydroxybenzoic acid 385523 5-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-2-methoxybenzoic acid 385525 5-(2-(2-(benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-2-(difluoromethoxy)benzoic acid 385527 5-(2-(2-(4-fluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-2-(difluoromethoxy)benzoic acid 385529 5-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-2-(difluoromethoxy)benzoic acid 385531 5-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-2-acetamidobenzoic acid 385532 3-amino-5-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-2-methylbenzoic acid 385548 3-amino-5-(2-(2-(benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-2-methylbenzoic acid 385549 3-amino-5-(2-(2-(benzyloxy)-5-(trifluoromethyl)phenyl)-5-methyl-1H-pyrrol-1-yl)-2-methylbenzoic acid 385550 5-(2-(2-(4-fluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-3-amino-2-methylbenzoic acid 385551 5-(2-(2-(4-fluorobenzyloxy)-5-(trifluoromethyl)phenyl)-5-methyl-1H-pyrrol-1-yl)-3-amino-2-methylbenzoic acid 385552 5-(2-(2-(4-fluorobenzyloxy)-5-methylphenyl)-5-methyl-1H-pyrrol-1-yl)-3-amino-2-methylbenzoic acid 385555 3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-1-naphthoic acid 385556 3-(2-(2-(benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-1-naphthoic acid 385559 3-(2-(2-(4-fluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-1-naphthoic acid 385565 3-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-1-naphthoic acid 385566 3-(2-(2-(4-fluorobenzyloxy)-5-methylphenyl)-5-methyl-1H-pyrrol-1-yl)-1-naphthoic acid 385567 3-(2-(2-(4-fluorobenzyloxy)-5-fluorophenyl)-5-methyl-1H-pyrrol-1-yl)-1-naphthoic acid 385568 (R)-N-(2-(dimethylamino)ethyl)-N-(1-(3-(4-fluorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)dodecanamide 385569 (R)-N-(2-(dimethylamino)ethyl)-N-(1-(3-(4-fluorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)octanamide 385571 (R)-2-(1-((2-(dimethylamino)ethyl)(nonyl)amino)ethyl)-3-(4-fluorophenyl)quinazolin-4(3H)-one 385572 (R)-2-(1-((2-(dimethylamino)ethyl)(octyl)amino)ethyl)-3-(4-fluorophenyl)quinazolin-4(3H)-one 385573 (R)-N-(2-(dimethylamino)ethyl)-N-(1-(3-(4-fluorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)decane-1-sulfonamide 385574 (R)-N-(2-(dimethylamino)ethyl)-N-(1-(3-(4-fluorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)octane-1-sulfonamide 385576 2-biphenyl-4-yl-N-(2-dimethylamino-ethyl)-N-{(R)-1-[3-(4-fluoro-phenyl)-4-oxo-3,4-dihydro-quinazolin-2-yl]-ethyl}-acetamide 385582 (R)-N-(2-(dimethylamino)ethyl)-N-(1-(3-(4-fluorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)-2-(4-(trifluoromethyl)phenyl)acetamide 385583 (R)-N-(2-(dimethylamino)ethyl)-N-(1-(3-(4-fluorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)-2-(4-(trifluoromethoxy)phenyl)acetamide 385585 (R)-N-(1-(3-(4-fluorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)-N-(2-methoxyethyl)-2-(4-(trifluoromethyl)phenyl)acetamide 385586 (R)-N-(2-ethoxyethyl)-N-(1-(3-(4-fluorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)-2-(4-(trifluoromethyl)phenyl)acetamide 385589 (R)-N-(1-(3-(4-fluorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)-N-(thiazol-2-ylmethyl)-2-(4-(trifluoromethyl)phenyl)acetamide 385590 (R)-N-(2-(1H-imidazol-2-yl)-2-oxoethyl)-N-(1-(3-(4-fluorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)-2-(4-(trifluoromethyl)phenyl)acetamide 385592 (R)-N-(2-(1H-imidazol-4-yl)-2-oxoethyl)-N-(1-(3-(4-fluorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)-2-(4-(trifluoromethyl)phenyl)acetamide 385594 (R)-N-(1-(3-(4-fluorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)-N-(2-(1-methyl-1H-imidazol-4-yl)-2-oxoethyl)-2-(4-(trifluoromethyl)phenyl)acetamide 385596 (R)-N-(1-(3-(4-fluorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)-N-(pyridin-2-ylmethyl)-2-(4-(trifluoromethyl)phenyl)acetamide 385597 (R)-N-(1-(3-(4-fluorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)-N-(pyridin-3-ylmethyl)-2-(4-(trifluoromethyl)phenyl)acetamide 385599 (R)-N-(1-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)ethyl)-N-(pyridin-3-ylmethyl)-2-(4-(trifluoromethyl)phenyl)acetamide 385601 (R)-N-(1-(3-(4-chlorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)-N-(pyridin-3-ylmethyl)-2-(4-(trifluoromethyl)phenyl)acetamide 385602 (R)-N-(1-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)ethyl)-N-(pyridin-3-ylmethyl)-2-(4-(trifluoromethyl)phenyl)acetamide 385603 (R)-N-(1-(3-(4-methoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)-N-(pyridin-3-ylmethyl)-2-(4-(trifluoromethyl)phenyl)acetamide 385604 (R)-N-(1-(3-(4-ethoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)-N-(pyridin-3-ylmethyl)-2-(4-(trifluoromethyl)phenyl)acetamide 385605 (R)-N-(1-(4-oxo-3-(4-(prop-1-ynyl)phenyl)-3,4-dihydroquinazolin-2-yl)ethyl)-N-(pyridin-3-ylmethyl)-2-(4-(trifluoromethyl)phenyl)acetamide 385606 (R)-N-(1-(3-(4-nitrophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)-N-(pyridin-3-ylmethyl)-2-(4-(trifluoromethyl)phenyl)acetamide 385607 (R)-N-(1-(3-(4-cyanophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)-N-(pyridin-3-ylmethyl)-2-(4-(trifluoromethyl)phenyl)acetamide 385608 (R)-N-(1-(3-(4-(methylsulfonyl)phenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)-N-(pyridin-3-ylmethyl)-2-(4-(trifluoromethyl)phenyl)acetamide 385609 (R)-4-(4-oxo-2-(1-(N-(pyridin-3-ylmethyl)-2-(4-(trifluoromethyl)phenyl)acetamido)ethyl)quinazolin-3(4H)-yl)benzoic acid 385610 N-{(R)-1-[3-(4-acetylamino-phenyl)-4-oxo-3,4-dihydro-quinazolin-2-yl]-ethyl}-N-pyridin-3-ylmethyl-2-(4-trifluoromethyl-phenyl)-acetamide 385611 2-biphenyl-4-yl-N-(2-ethoxy-ethyl)-N-[3-(4-ethoxy-phenyl)-4-oxo-3,4-dihydro-quinazolin-2-ylmethyl]-acetamide 385612 2-biphenyl-4-yl-N-(2-ethoxy-ethyl)-N-{(R)-1-[3-(4-ethoxy-phenyl)-4-oxo-3,4-dihydro-quinazolin-2-yl]-ethyl}-acetamide 385614 2-biphenyl-4-yl-N-(2-ethoxy-ethyl)-N-{(R)-1-[3-(4-ethoxy-phenyl)-4-oxo-3,4-dihydro-quinazolin-2-yl]-propyl}-acetamide 385615 2-biphenyl-4-yl-N-(2-ethoxy-ethyl)-N-{(R)-[3-(4-ethoxy-phenyl)-4-oxo-3,4-dihydro-quinazolin-2-yl]-phenyl-methyl}-acetamide 385616 (R)-N-(1-(3-(4-ethoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)-N-(pyridin-3-ylmethyl)-2-(4-(trifluoromethoxy)phenyl)acetamide 385617 (R)-N-(1-(3-(4-ethoxyphenyl)-4-oxo-3,4-dihydropyrido[2,3-d]pyrimidin-2-yl)ethyl)-N-(pyridin-3-ylmethyl)-2-(4-(trifluoromethoxy)phenyl)acetamide 385618 (R)-N-(1-(3-(4-ethoxyphenyl)-4-oxo-3,4-dihydropyrido[3,4-d]pyrimidin-2-yl)ethyl)-N-(pyridin-3-ylmethyl)-2-(4-(trifluoromethoxy)phenyl)acetamide 385619 (R)-N-(1-(3-(4-ethoxyphenyl)-4-oxo-3,4-dihydropyrido[3,2-d]pyrimidin-2-yl)ethyl)-N-(pyridin-3-ylmethyl)-2-(4-(trifluoromethoxy)phenyl)acetamide 385620 (R)-N-(1-(3-(4-ethoxyphenyl)-4-oxo-3,4-dihydropteridin-2-yl)ethyl)-N-(pyridin-3-ylmethyl)-2-(4-(trifluoromethoxy)phenyl)acetamide 385678 2-(methyl(phenyl)amino)-4-(phenylamino)pyrazolo[1,5-a][1,3,5]triazine-8-carbonitrile 385679 4-(phenylamino)-2-(pyridin-3-ylamino)pyrazolo[1,5-a][1,3,5]triazine-8-carbonitrile 385680 2-(p-toluidino)-4-(phenylamino)pyrazolo[1,5-a][1,3,5]triazine-8-carbonitrile 385681 2-(3,4-dimethoxyphenylamino)-4-(phenylamino)pyrazolo[1,5-a][1,3,5]triazine-8-carbonitrile 385682 2-(4-(diethylamino)phenylamino)-4-(phenylamino)pyrazolo[1,5-a][1,3,5]triazine-8-carbonitrile 385684 2-(1H-imidazol-2-ylamino)-4-(phenylamino)pyrazolo[1,5-a][1,3,5]triazine-8-carbonitrile 385685 2-(cyclohexylmethylamino)-4-(phenylamino)pyrazolo[1,5-a][1,3,5]triazine-8-carbonitrile 385686 2-(4-chlorobenzylamino)-4-(phenylamino)pyrazolo[1,5-a][1,3,5]triazine-8-carbonitrile 385688 2-(benzyl(methyl)amino)-4-(phenylamino)pyrazolo[1,5-a][1,3,5]triazine-8-carbonitrile 385689 2-(isopentylamino)-4-(phenylamino)pyrazolo[1,5-a][1,3,5]triazine-8-carbonitrile 385690 2-(2,3-dihydro-1H-inden-2-ylamino)-4-(phenylamino)pyrazolo[1,5-a][1,3,5]triazine-8-carbonitrile 385692 4-(phenylamino)-2-(pyrrolidin-1-yl)pyrazolo[1,5-a][1,3,5]triazine-8-carbonitrile 385694 2-(1H-imidazol-1-yl)-4-(phenylamino)pyrazolo[1,5-a][1,3,5]triazine-8-carbonitrile 385696 2-(3,4-dihydroisoquinolin-2(1H)-yl)-4-(phenylamino)pyrazolo[1,5-a][1,3,5]triazine-8-carbonitrile 385697 2-(4-ethylpiperazin-1-yl)-4-(phenylamino)pyrazolo[1,5-a][1,3,5]triazine-8-carbonitrile 385698 4-(phenylamino)-2-(4-(pyridin-2-yl)piperazin-1-yl)pyrazolo[1,5-a][1,3,5]triazine-8-carbonitrile 385700 4-(2-(1H-imidazol-4-yl)ethylamino)-2-(phenylamino)pyrazolo[1,5-a][1,3,5]triazine-8-carbonitrile 385703 2-(p-toluidino)-4-(phenethylamino)pyrazolo[1,5-a][1,3,5]triazine-8-carbonitrile 385704 4-(phenethylamino)-2-(pyridin-3-ylamino)pyrazolo[1,5-a][1,3,5]triazine-8-carbonitrile 385706 N-(3-(8-cyano-4-(phenethylamino)pyrazolo[1,5-a][1,3,5]triazin-2-ylamino)phenyl)acetamide 385707 N-(3-(8-cyano-4-(phenylamino)pyrazolo[1,5-a][1,3,5]triazin-2-ylamino)phenyl)acetamide 385709 N-(3-(8-cyano-4-(cyclopropylamino)pyrazolo[1,5-a][1,3,5]triazin-2-ylamino)phenyl)acetamide 385710 N-(3-(8-cyano-4-(cyclobutylamino)pyrazolo[1,5-a][1,3,5]triazin-2-ylamino)phenyl)acetamide 385712 N-(3-(4-(cyclopropylamino)-8-methylpyrazolo[1,5-a][1,3,5]triazin-2-ylamino)phenyl)acetamide 385713 N-(3-(8-methyl-4-(phenylamino)pyrazolo[1,5-a][1,3,5]triazin-2-ylamino)phenyl)acetamide 385714 N-(3-(4-(cyclopropylamino)-8-ethylpyrazolo[1,5-a][1,3,5]triazin-2-ylamino)phenyl)acetamide 385716 N-(3-(8-bromo-4-(cyclopropylamino)pyrazolo[1,5-a][1,3,5]triazin-2-ylamino)phenyl)acetamide 385717 N-(3-(8-cyano-4-(4-(piperazin-1-ylmethyl)phenylamino)pyrazolo[1,5-a][1,3,5]triazin-2-ylamino)phenyl)acetamide 385718 N-(3-(8-cyano-4-(3-(diethylamino)phenylamino)pyrazolo[1,5-a][1,3,5]triazin-2-ylamino)phenyl)acetamide 385720 N-(3-(8-cyano-4-(4-((diethylamino)methyl)phenylamino)pyrazolo[1,5-a][1,3,5]triazin-2-ylamino)phenyl)acetamide 385721 3-(2-(3-acetamidophenylamino)-8-cyanopyrazolo[1,5-a][1,3,5]triazin-4-ylamino)benzoic acid 385723 3-(2-(3-acetamidophenylamino)-8-cyanopyrazolo[1,5-a][1,3,5]triazin-4-ylamino)-N-(2-(dimethylamino)ethyl)benzamide 385724 N-(3-(8-cyano-4-(3-(pyrrolidine-1-carbonyl)phenylamino)pyrazolo[1,5-a][1,3,5]triazin-2-ylamino)phenyl)acetamide 385726 3-(2-(3-acetamidophenylamino)-8-cyanopyrazolo[1,5-a][1,3,5]triazin-4-ylamino)-N,N-diethylbenzamide 385728 N-(3-(8-cyano-4-(3-ethoxyphenylamino)pyrazolo[1,5-a][1,3,5]triazin-2-ylamino)phenyl)acetamide 385729 N-(3-(8-cyano-4-(3-(difluoromethoxy)phenylamino)pyrazolo[1,5-a][1,3,5]triazin-2-ylamino)phenyl)acetamide 385736 N2,N4-diphenylpyrazolo[1,5-a][1,3,5]triazine-2,4-diamine 385737 2,4-bis(phenylamino)pyrazolo[1,5-a][1,3,5]triazine-8-carbonitrile 385766 1-(3,3-diphenylpropyl)-4-phenylpiperidin-4-ol 385771 1-benzyl-4-phenylpiperidin-4-ol 385774 4-phenyl-1-(1-phenylethyl)piperidin-4-ol 385775 4-phenyl-1-(1-phenylpropyl)piperidin-4-ol 385778 4-phenyl-1-(1-phenylbutyl)piperidin-4-ol 385780 4-phenyl-1-(1-phenylpentyl)piperidin-4-ol 385782 4-phenyl-1-(1-phenylhexyl)piperidin-4-ol 385784 1-(4-methyl-1-phenylpentyl)-4-phenylpiperidin-4-ol 385785 4-phenyl-1-(1-phenylheptyl)piperidin-4-ol 385786 1-(cyclopentyl(phenyl)methyl)-4-phenylpiperidin-4-ol 385787 1-(1,2-diphenylethyl)-4-phenylpiperidin-4-ol 385788 1-(2-hydroxy-1-phenylethyl)-4-phenylpiperidin-4-ol 385789 1-(2-methoxy-1-phenylethyl)-4-phenylpiperidin-4-ol 385790 1-(2-ethoxy-1-phenylethyl)-4-phenylpiperidin-4-ol 385791 methyl 2-(4-hydroxy-4-phenylpiperidin-1-yl)-2-phenylacetate 385792 2-(4-hydroxy-4-phenylpiperidin-1-yl)-2-phenylacetonitrile 385794 N-(2,6-difluorophenyl)-2-(4-hydroxy-4-phenylpiperidin-1-yl)-2-phenylacetamide 385795 1-benzhydryl-4-phenylpiperidin-4-ol 385796 4-phenyl-1-(phenyl(pyridin-2-yl)methyl)piperidin-4-ol 385798 4-phenyl-1-(phenyl(pyridin-3-yl)methyl)piperidin-4-ol 385799 4-phenyl-1-(phenyl(thiophen-2-yl)methyl)piperidin-4-ol 385802 4-phenyl-1-(phenyl(m-tolyl)methyl)piperidin-4-ol 385803 4-phenyl-1-(phenyl(p-tolyl)methyl)piperidin-4-ol 385804 4-phenyl-1-(phenyl(2-(trifluoromethyl)phenyl)methyl)piperidin-4-ol 385805 4-phenyl-1-(phenyl(3-(trifluoromethyl)phenyl)methyl)piperidin-4-ol 385806 4-phenyl-1-(phenyl(4-(trifluoromethyl)phenyl)methyl)piperidin-4-ol 385807 1-((2-ethylphenyl)(phenyl)methyl)-4-phenylpiperidin-4-ol 385808 1-((2-chlorophenyl)(phenyl)methyl)-4-phenylpiperidin-4-ol 385809 1-((3-chlorophenyl)(phenyl)methyl)-4-phenylpiperidin-4-ol 385810 1-((4-chlorophenyl)(phenyl)methyl)-4-phenylpiperidin-4-ol 385812 1-((2-fluorophenyl)(phenyl)methyl)-4-phenylpiperidin-4-ol 385813 1-((2-bromophenyl)(phenyl)methyl)-4-phenylpiperidin-4-ol 385814 1-((4-bromophenyl)(phenyl)methyl)-4-phenylpiperidin-4-ol 385815 1-((2-methoxyphenyl)(phenyl)methyl)-4-phenylpiperidin-4-ol 385816 1-((2-(hydroxymethyl)phenyl)(phenyl)methyl)-4-phenylpiperidin-4-ol 385817 2-((4-hydroxy-4-phenylpiperidin-1-yl)(phenyl)methyl)benzoic acid 385818 1-(dio-tolylmethyl)-4-phenylpiperidin-4-ol 385819 1-(bis(2-chlorophenyl)methyl)-4-phenylpiperidin-4-ol 385820 1-(bis(2-fluorophenyl)methyl)-4-phenylpiperidin-4-ol 385821 1-(bis(4-fluorophenyl)methyl)-4-phenylpiperidin-4-ol 385822 1-(bis(2-bromophenyl)methyl)-4-phenylpiperidin-4-ol 385823 6-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-1H-indole-4-carboxylic acid 385824 1-(bis(2-methoxyphenyl)methyl)-4-phenylpiperidin-4-ol 385825 1-(bis(4-methoxyphenyl)methyl)-4-phenylpiperidin-4-ol 385826 1-benzhydryl-4-methoxy-4-phenylpiperidine 385827 1-benzhydryl-4-ethoxy-4-phenylpiperidine 385828 1-benzhydryl-4-phenyl-4-propoxypiperidine 385829 1-benzhydryl-4-(benzyloxy)-4-phenylpiperidine 385830 4-phenyl-1-(phenyl(o-tolyl)methyl)piperidin-4-ol 385868 (Z)-1-(3-((1H-pyrrol-2-yl)methylene)-2-oxoindolin-5-yl)urea 385869 5-((2-oxo-5-ureidoindolin-3-ylidene)methyl)-1H-pyrrole-3-carboxylic acid 385870 4-methyl-5-((2-oxo-5-ureidoindolin-3-ylidene)methyl)-1H-pyrrole-3-carboxylic acid 385871 3-(4-methyl-5-((2-oxo-5-ureidoindolin-3-ylidene)methyl)-1H-pyrrol-3-yl)propanoic acid 385872 3-(2,4-dimethyl-5-((2-oxo-5-ureidoindolin-3-ylidene)methyl)-1H-pyrrol-3-yl)propanoic acid 385873 1-(3-((4-((2-(dimethylamino)ethyl)carbamoyl)-1H-pyrrol-2-yl)methylene)-2-oxoindolin-5-yl)urea 385874 1-(3-((4-((2-(piperidin-1-yl)ethyl)carbamoyl)-1H-pyrrol-2-yl)methylene)-2-oxoindolin-5-yl)urea 385875 1-(3-((4-((2-morpholinoethyl)carbamoyl)-1H-pyrrol-2-yl)methylene)-2-oxoindolin-5-yl)urea 385876 1-(3-((4-(3-(dimethylamino)pyrrolidine-1-carbonyl)-1H-pyrrol-2-yl)methylene)-2-oxoindolin-5-yl)urea 385877 1-(3-((4-((2-(1H-imidazol-5-yl)ethyl)carbamoyl)-1H-pyrrol-2-yl)methylene)-2-oxoindolin-5-yl)urea 385878 1-(3-((4-((2-(pyridin-4-yl)ethyl)carbamoyl)-1H-pyrrol-2-yl)methylene)-2-oxoindolin-5-yl)urea 385879 1-(2-oxo-3-((4-phenyl-1H-pyrrol-2-yl)methylene)indolin-5-yl)urea 385880 1-(2-oxo-3-((4-(pyridin-3-yl)-1H-pyrrol-2-yl)methylene)indolin-5-yl)urea 385881 3-(5-((2-oxo-5-ureidoindolin-3-ylidene)methyl)-1H-pyrrol-3-yl)benzoic acid 385882 1-(3-((4-(3-((2-(dimethylamino)ethyl)carbamoyl)phenyl)-1H-pyrrol-2-yl)methylene)-2-oxoindolin-5-yl)urea 385885 1-(3-((4-(3-((2-(piperidin-1-yl)ethyl)carbamoyl)phenyl)-1H-pyrrol-2-yl)methylene)-2-oxoindolin-5-yl)urea 385888 1-(3-((4-(3-hydroxyphenyl)-1H-pyrrol-2-yl)methylene)-2-oxoindolin-5-yl)urea 385891 1-(3-((4-(3-methoxyphenyl)-1H-pyrrol-2-yl)methylene)-2-oxoindolin-5-yl)urea 385893 1-(3-((4-(3-fluorophenyl)-1H-pyrrol-2-yl)methylene)-2-oxoindolin-5-yl)urea 385896 1-(2-oxo-3-((4-m-tolyl-1H-pyrrol-2-yl)methylene)indolin-5-yl)urea 385899 1-(3-((4-(3-carbamoylphenyl)-1H-pyrrol-2-yl)methylene)-2-oxoindolin-5-yl)urea 385901 1-(3-((4-(3-acetamidophenyl)-1H-pyrrol-2-yl)methylene)-2-oxoindolin-5-yl)urea 385904 1-(3-((4-(3-(aminomethyl)phenyl)-1H-pyrrol-2-yl)methylene)-2-oxoindolin-5-yl)urea 385907 (Z)-1-(3-(1-(1h-pyrrol-2-yl)ethylidene)-2-oxoindolin-5-yl)urea 385910 1-(3-(1-(4-(aminomethyl)-1H-pyrrol-2-yl)ethylidene)-2-oxoindolin-5-yl)urea 385913 1-(3-(1-(4-(acetamidomethyl)-1H-pyrrol-2-yl)ethylidene)-2-oxoindolin-5-yl)urea 385914 (Z)-1-(3-(1-(4-(isonicotinamidomethyl)-1H-pyrrol-2-yl)ethylidene)-2-oxoindolin-5-yl)urea 385915 1-(3-(1-(4-(nicotinamidomethyl)-1H-pyrrol-2-yl)ethylidene)-2-oxoindolin-5-yl)urea 385916 1-(2-oxo-3-(1-(4-((piperidine-4-carboxamido)methyl)-1H-pyrrol-2-yl)ethylidene)indolin-5-yl)urea(Z)-1-(2-oxo-3-(1-(4-((piperidine-4-carboxamido)methyl)-1H-pyrrol-2-yl)ethylidene)indolin-5-yl)urea 385917 1-(3-(1-(4-((1-methylpiperidine-4-carboxamido)methyl)-1H-pyrrol-2-yl)ethylidene)-2-oxoindolin-5-yl)urea 385918 1-(2-oxo-3-(1-(4-((piperazine-3-carboxamido)methyl)-1H-pyrrol-2-yl)ethylidene)indolin-5-yl)urea 385919 1-(3-(1-(4-((2-aminoacetamido)methyl)-1H-pyrrol-2-yl)ethylidene)-2-oxoindolin-5-yl)urea 385920 1-(3-(1-(4-((2-hydroxyacetamido)methyl)-1H-pyrrol-2-yl)ethylidene)-2-oxoindolin-5-yl)urea 385921 1-(2-oxo-3-(1-(4-((3-(piperidin-1-yl)propanamido)methyl)-1H-pyrrol-2-yl)ethylidene)indolin-5-yl)urea 386060 (E)-1-(1-(cyclooctenylmethyl)piperidin-4-yl)-3-(naphthalen-2-yl)urea 386064 1-(1-(cyclooctenylmethyl)piperidin-4-yl)-3-(3-(trifluoromethyl)phenyl)urea 386066 1-(3-chlorophenyl)-3-(1-(cyclooctenylmethyl)piperidin-4-yl)urea 386067 1-(1-(cyclooctenylmethyl)piperidin-4-yl)-3-(3-(trifluoromethoxy)phenyl)urea 386068 1-(3-acetylphenyl)-3-(1-(cyclooctenylmethyl)piperidin-4-yl)urea 386070 1-(3,5-bis(trifluoromethyl)phenyl)-3-(1-(cyclooctenylmethyl)piperidin-4-yl)urea 386071 1-(1-(cyclooctenylmethyl)piperidin-4-yl)-3-(3-fluoro-5-(trifluoromethyl)phenyl)urea 386073 1-(1-(cyclooctenylmethyl)piperidin-4-yl)-3-(3,5-dichlorophenyl)urea 386076 1-(1-(cyclooctenylmethyl)piperidin-4-yl)-3-(4-phenoxyphenyl)urea 386087 1-(4-tert-butylphenyl)-3-(1-(cyclooctenylmethyl)piperidin-4-yl)urea 386088 1-(1-(cyclooctenylmethyl)piperidin-4-yl)-3-(3,5-dichloropyridin-4-yl)urea 386090 methyl 3-(3-(1-(cyclooctenylmethyl)piperidin-4-yl)ureido)benzoate 386091 1-(1-(cyclooctenylmethyl)piperidin-4-yl)-3-(5-phenylthiophen-2-yl)urea 386103 (1-(2-chloro-4-fluorophenyl)-6,7-dihydro-1H-pyrazolo[4,3-c]pyridin-5(4H)-yl)(2,6-difluorophenyl)methanone 386104 (1-(2-chlorophenyl)-6,7-dihydro-1H-pyrazolo[4,3-c]pyridin-5(4H)-yl)(2,6-difluorophenyl)methanone 386105 (1-(2-chlorophenyl)-6,7-dihydro-1H-pyrazolo[4,3-c]pyridin-5(4H)-yl)(2,6-dichlorophenyl)methanone 386106 (1-(2-chlorophenyl)-6,7-dihydro-1H-pyrazolo[4,3-c]pyridin-5(4H)-yl)(1H-indol-2-yl)methanone 386107 (1-(2-chlorophenyl)-6,7-dihydro-1H-pyrazolo[4,3-c]pyridin-5(4H)-yl)(1H-indol-3-yl)methanone 386108 (1-(2-chlorophenyl)-6,7-dihydro-1H-pyrazolo[4,3-c]pyridin-5(4H)-yl)(1-methyl-1H-indol-3-yl)methanone 386109 (1-(2-chlorophenyl)-6,7-dihydro-1H-pyrazolo[4,3-c]pyridin-5(4H)-yl)(1H-indol-4-yl)methanone 386110 (1-(2-chlorophenyl)-6,7-dihydro-1H-pyrazolo[4,3-c]pyridin-5(4H)-yl)(1H-indol-6-yl)methanone 386111 (1-(2-chlorophenyl)-6,7-dihydro-1H-pyrazolo[4,3-c]pyridin-5(4H)-yl)(1-methyl-1H-indol-5-yl)methanone 386118 (6-chloro-1-methyl-1H-indol-5-yl)(1-(2-chlorophenyl)-6,7-dihydro-1H-pyrazolo[4,3-c]pyridin-5(4H)-yl)methanone 386119 (1-(2-chlorophenyl)-6,7-dihydro-1H-pyrazolo[4,3-c]pyridin-5(4H)-yl)(1-isopropyl-1H-indol-5-yl)methanone 386121 (1-(2-chlorophenyl)-6,7-dihydro-1H-pyrazolo[4,3-c]pyridin-5(4H)-yl)(6-methoxy-1H-pyrrolo[2,3-b]pyridin-5-yl)methanone 386123 (2,4-difluorophenyl)(3-(2,4-difluorophenyl)-5,6-dihydroimidazo[1,5-a]pyrazin-7(8H)-yl)methanone 386125 (2,6-difluorophenyl)(3-(2,4-difluorophenyl)-5,6-dihydroimidazo[1,5-a]pyrazin-7(8H)-yl)methanone 386127 (3-(2,4-difluorophenyl)-5,6-dihydroimidazo[1,5-a]pyrazin-7(8H)-yl)(6-methoxy-1-methyl-1H-indol-5-yl)methanone 386130 (6-chloro-1-methyl-1H-indol-5-yl)(3-(2,4-difluorophenyl)-5,6-dihydroimidazo[1,5-a]pyrazin-7(8H)-yl)methanone 386131 (3-(2,4-difluorophenyl)-5,6-dihydroimidazo[1,5-a]pyrazin-7(8H)-yl)(6-methoxy-1H-pyrrolo[2,3-b]pyridin-5-yl)methanone 386134 2-(5-(3-(2,4-difluorophenyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine-7-carbonyl)-6-methoxy-1-methyl-1H-indol-3-yl)-N,N-dimethyl-2-oxoacetamide 386136 2-(6-chloro-5-(3-(2,4-difluorophenyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine-7-carbonyl)-1H-indol-3-yl)-N,N-dimethyl-2-oxoacetamide 386138 2-(6-chloro-5-(3-(2,4-difluorophenyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine-7-carbonyl)-1-methyl-1H-indol-3-yl)-N,N-dimethyl-2-oxoacetamide 386140 2-(5-(3-(2,4-difluorophenyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine-7-carbonyl)-6-methoxy-1H-pyrrolo[2,3-b]pyridin-3-yl)-N,N-dimethyl-2-oxoacetamide 386142 1-(5-(3-(2,4-difluorophenyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine-7-carbonyl)-6-methoxy-1H-pyrrolo[2,3-b]pyridin-3-yl)-2-(3-hydroxypyrrolidin-1-yl)ethane-1,2-dione 386144 1-(5-(3-(2,4-difluorophenyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine-7-carbonyl)-6-methoxy-1-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)-2-(3-hydroxypyrrolidin-1-yl)ethane-1,2-dione 386152 1-(1-(2-(6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl)ethyl)piperidin-4-yl)-3-(naphthalen-2-yl)urea 386154 1-(naphthalen-2-yl)-3-(1-phenethylpiperidin-4-yl)urea 386155 1-(naphthalen-2-yl)-3-(1-(3-phenylpropyl)piperidin-4-yl)urea 386156 1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl)methyl)piperidin-4-yl)-3-phenylurea 386157 1-(3,5-bis(trifluoromethyl)phenyl)-3-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl)methyl)piperidin-4-yl)urea 386158 1-(3-acetylphenyl)-3-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl)methyl)piperidin-4-yl)urea 386159 2-(5-(1-(2-chlorophenyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridine-5-carbonyl)-6-methoxy-1H-pyrrolo[2,3-b]pyridin-3-yl)-N,N-dimethyl-2-oxoacetamide 386160 2-(6-chloro-5-(1-(2-chlorophenyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridine-5-carbonyl)-1-methyl-1H-indol-3-yl)-N,N-dimethyl-2-oxoacetamide 386161 2-(5-(1-(2-chlorophenyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridine-5-carbonyl)-1H-indol-3-yl)-N,N-dimethyl-2-oxoacetamide 386162 2-(6-chloro-5-(4-(2,4-difluorophenyl)-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidine-7-carbonyl)-1-methyl-1H-indol-3-yl)-N,N-dimethyl-2-oxoacetamide 386163 1-(3,5-difluorophenyl)-3-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl)methyl)piperidin-4-yl)urea 386164 1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl)methyl)piperidin-4-yl)-3-(3-methoxyphenyl)urea 386165 1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl)methyl)piperidin-4-yl)-3-(3-(trifluoromethoxy)phenyl)urea 386166 1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl)methyl)piperidin-4-yl)-3-(4-(trifluoromethoxy)phenyl)urea 386167 1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl)methyl)piperidin-4-yl)-3-(5-phenylthiophen-2-yl)urea 386168 1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl)methyl)piperidin-4-yl)-3-(5-(4-(trifluoromethyl)phenyl)thiophen-2-yl)urea 386169 1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl)methyl)piperidin-4-yl)-3-(5-(3-methoxyphenyl)thiophen-2-yl)urea 386170 1-(5-(2-chlorophenyl)thiophen-2-yl)-3-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl)methyl)piperidin-4-yl)urea 386171 1-(5-bromopyridin-3-yl)-3-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl)methyl)piperidin-4-yl)urea 386172 1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl)methyl)piperidin-4-yl)-3-(5-(thiophen-2-yl)pyridin-3-yl)urea 386173 1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl)methyl)piperidin-4-yl)-3-(5-(thiophen-3-yl)pyridin-3-yl)urea 386174 1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl)methyl)piperidin-4-yl)-3-(3-(tetrahydrofuran-3-yloxy)phenyl)urea 386175 1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl)methyl)piperidin-4-yl)-3-(3-fluoro-5-(tetrahydrofuran-3-yloxy)phenyl)urea 386176 1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl)methyl)piperidin-4-yl)-3-(3-(tetrahydro-2H-pyran-4-yloxy)phenyl)urea 386178 1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl)methyl)piperidin-4-yl)-3-(2-fluoro-5-(trifluoromethyl)phenyl)urea 386179 1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl)methyl)piperidin-4-yl)-3-(3-fluoro-5-(trifluoromethyl)phenyl)urea 386180 1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl)methyl)piperidin-4-yl)-3-(4-fluoro-3-(trifluoromethyl)phenyl)urea 386181 methyl 3-(3-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl)methyl)piperidin-4-yl)ureido)benzoate 386184 1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-({[3-fluoro-5-(trifluoromethyl)phenyl]carbamoyl}amino)-1-methylpiperidin-1-ium iodide 386421 2-(2-butoxypyrimidin-4-ylamino)benzoic acid 386422 2-(2-ethoxypyrimidin-4-ylamino)benzoic acid 386423 2-(2-propoxypyrimidin-4-ylamino)benzoic acid 386424 2-(2-(pentyloxy)pyrimidin-4-ylamino)benzoic acid 386426 2-(2-sec-butoxypyrimidin-4-ylamino)benzoic acid 386427 2-(2-(cyclohexylmethoxy)pyrimidin-4-ylamino)benzoic acid 386428 2-(2-phenoxypyrimidin-4-ylamino)benzoic acid 386429 2-(2-(butylamino)pyrimidin-4-ylamino)benzoic acid 386430 2-(2-(benzylamino)pyrimidin-4-ylamino)benzoic acid 386431 2-(2-(cyclohexylamino)pyrimidin-4-ylamino)benzoic acid 386432 2-(2-(azepan-1-yl)pyrimidin-4-ylamino)benzoic acid 386434 2-(2-(phenylamino)pyrimidin-4-ylamino)benzoic acid 386435 2-(2-(2-hydroxyphenylamino)pyrimidin-4-ylamino)benzoic acid 386436 2-(2-(3-hydroxyphenylamino)pyrimidin-4-ylamino)benzoic acid 386437 2-(2-(4-hydroxyphenylamino)pyrimidin-4-ylamino)benzoic acid 386438 2-(2-(2-fluorophenylamino)pyrimidin-4-ylamino)benzoic acid 386439 2-(2-(3-fluorophenylamino)pyrimidin-4-ylamino)benzoic acid 386440 2-(2-(4-fluorophenylamino)pyrimidin-4-ylamino)benzoic acid 386441 2-(2-(m-toluidino)pyrimidin-4-ylamino)benzoic acid 386442 2-(2-(3-fluoro-4-methylphenylamino)pyrimidin-4-ylamino)benzoic acid 386443 2-(2-(3-hydroxy-2-methylphenylamino)pyrimidin-4-ylamino)benzoic acid 386444 2-(2-(3-(trifluoromethyl)phenylamino)pyrimidin-4-ylamino)benzoic acid 386445 2-(2-(4-(trifluoromethyl)phenylamino)pyrimidin-4-ylamino)benzoic acid 386446 2-(2-(4-nitrophenylamino)pyrimidin-4-ylamino)benzoic acid 386447 2-(2-(4-morpholinophenylamino)pyrimidin-4-ylamino)benzoic acid 386448 2-(2-(1H-indazol-6-ylamino)pyrimidin-4-ylamino)benzoic acid 386449 2-(2-(1H-indazol-5-ylamino)pyrimidin-4-ylamino)benzoic acid 386450 2-(2-(quinolin-6-ylamino)pyrimidin-4-ylamino)benzoic acid 386451 3-(2-(phenylamino)pyrimidin-4-ylamino)-2-naphthoic acid 386452 3-(2-(3-hydroxyphenylamino)pyrimidin-4-ylamino)-2-naphthoic acid 386453 2-(5-fluoro-2-(phenylamino)pyrimidin-4-ylamino)benzoic acid 386454 2-(5-fluoro-2-(3-hydroxyphenylamino)pyrimidin-4-ylamino)benzoic acid 386455 2-(5-bromo-2-(phenylamino)pyrimidin-4-ylamino)benzoic acid 386456 2-(5-bromo-2-(3-hydroxyphenylamino)pyrimidin-4-ylamino)benzoic acid 386465 2-(2-(phenylamino)pyrimidin-4-ylamino)benzamide 386467 2-[2-(3-hydroxy-phenylamino)-pyrimidin-4-ylamino]-benzamide 386529 MCL-433 386530 MCL-431 386531 MCL-434 386532 MCL-449 386533 MCL-429 386534 MCL-444 386535 MCL-435 386537 MCL-432 386538 MCL-428 386539 MCL-443 387060 (1R,5R)-(+)-5-(3-hydroxyphenyl)-9-oxo-2-phenylethyl-2-azabicyclo[3.3.1]nonane 387061 (1S,5S,9S)-(-)-9-hydroxy-5-(3-hydroxyphenyl-2-phenylethyl-2-azabicyclo[3.3.1]nonane 387062 (1R,5R,9R)-(+)-9-hydroxy-5-(3-hydroxyphenyl-2-phenylethyl-2-azabicyclo[3.3.1]nonane 387063 (1R,5R,9S)-(-)-9-hydroxy-5-(3-hydroxyphenyl-2-phenylethyl-2-azabicyclo[3.3.1]nonane 387064 (1S,5S,9R)-(+)-9-hydroxy-5-(3-hydroxyphenyl-2-phenylethyl-2-azabicyclo[3.3.1]nonane 387065 (1S,5R)-(-)-5-(3-hydroxyphenyl)-9-methylene-2-phenethyl-2-azabicyclo[3.3.1]nonane 387066 (1R,5S)-(+)-5-(3-hydroxyphenyl)-9-methylene-2-phenethyl-2-azabicyclo[3.3.1]nonane 387067 (1S,5R,9S)-(-)-5-(3-hydroxyphenyl)-9-methyl-2-phenethyl-2-azabicyclo[3.3.1]nonane 387068 (1R,5S,9R)-(+)-5-(3-hydroxyphenyl)-9-methyl-2-phenethyl-2-azabicyclo[3.3.1]nonane 387163 (R)-(+)-2-(1-(biphenyl-2-yloxy)ethyl)-4,5-dihydro-1H-imidazole 387164 (S)-(-)-2-(1-(biphenyl-2-yloxy)ethyl)-4,5-dihydro-1H-imidazole 387169 N-isopropyl-N'-[2-(2-methylphenoxy)-5-nitrobenzenesulfonyl]-urea 387170 N-n-butyl-N'-[2-(2-methylphenoxy)-5-nitrobenzenesulfonyl]-urea 387171 N-tert-butyl-N'-[2-(2-methylphenoxy)-5-nitrobenzenesulfonyl]-urea 387172 N-isopropyl-N'-[2-(3-methylphenoxy)-5-nitrobenzenesulfonyl]-urea 387173 (R)-(+)-2-(1-(3'-nitrobiphenyl-2-yloxy)ethyl)-4,5-dihydro-1H-imidazole 387174 N-n-butyl-N'-[2-(3-methylphenoxy)-5-nitrobenzenesulfonyl]-urea 387175 N-tert-butyl-N'-[2-(3-methylphenoxy)-5-nitrobenzenesulfonyl]-urea 387176 N-isopropyl-N'-[2-(4-methylphenoxy)-5-nitrobenzenesulfonyl]-urea 387178 N-n-propyl-N'-[2-(4-methylphenoxy)-5-nitrobenzenesulfonyl]-urea 387179 (S)-(-)-2-(1-(3'-nitrobiphenyl-2-yloxy)ethyl)-4,5-dihydro-1H-imidazole 387180 N-tert-butyl-N'-[2-(2-bromophenoxy)-5-nitrobenzenesulfonyl]-urea 387181 N-n-pentyl-N'-[2-(2-bromophenoxy)-5-nitrobenzenesulfonyl]-urea 387182 N-tert-butyl-N'-[2-(3-bromophenoxy)-5-nitrobenzenesulfonyl]-urea 387183 N-n-pentyl-N'-[2-(3-bromophenoxy)-5-nitrobenzenesulfonyl]-urea 387185 N-tert-butyl-N'-[2-(4-bromophenoxy)-5-nitrobenzenesulfonyl]-urea 387186 N-n-pentyl-N'-[2-(4-bromophenoxy)-5-nitrobenzenesulfonyl]-urea 387188 N-tert-butyl-N'-[2-(2-chlorophenoxy)-5-nitrobenzenesulfonyl]-urea 387189 N-n-pentyl-N'-[2-(2-chlorophenoxy)-5-nitrobenzenesulfonyl]-urea 387190 N-tert-butyl-N'-[2-(3-chlorophenoxy)-5-nitrobenzenesulfonyl]-urea 387193 N-n-pentyl-N'-[2-(3-chlorophenoxy)-5-nitrobenzenesulfonyl]-urea 387195 N-tert-butyl-N'-[2-(4-chlorophenoxy)-5-nitrobenzenesulfonyl]-urea 387196 N-n-pentyl-N'-[2-(4-chloroxyphenoxy)-5-nitrobenzenesulfonyl]urea 387198 [4-(2-morpholin-4-ylethoxy)naphthalen-1-yl]naphthalene-1-ylmethanone 387200 N-tert-butyl-N'-[2-(3-iodophenoxy)-5-nitrobenzenesulfonyl]-urea 387201 naphthalen-1-yl-(4-propoxynaphthalen-1-yl)methanone 387202 N-n-pentyl-N'-[2-(3-iodophenoxy)-5-nitrobenzenesulfonyl]-urea 387203 naphthalen-1-yl-(4-butoxynaphthalen-1-yl)methanone 387204 N-tert-butyl-N'-[2-(4-iodophenoxy)-5-nitrobenzenesulfonyl]-urea 387205 naphthalen-1-yl-(4-pentyloxynaphthalen-1-yl)methanone 387206 (4-hexyloxynaphthalen-1-yl)naphthalen-1-ylmethanone 387207 naphthalen-1-yl-(4-phenethyloxynaphthalen-1-yl)methanone 387208 N-n-pentyl-N'-[2-(4-iodophenoxy)-5-nitrobenzenesulfonyl]-urea 387209 naphthalen-1-yl-(4-pentylaminonaphthalen-1-yl)methanone 387210 N-tert-butyl-N'-[2-(4-methoxyphenoxy)-5-nitrobenzenesulfonyl]urea 387211 N-n-pentyl-N'-[2-(4-methoxyphenoxy)-5-nitrobenzenesulfonyl]urea 387213 N-tert-butyl-N'-[2-(4-propoxyphenoxy)-5-nitrobenzenesulfonyl]urea 387214 N-n-pentyl-N'-[2-(4-propoxyphenoxy)-5-nitrobenzenesulfonyl]urea 387215 N-tert-butyl-N'-[2-(4-ethoxyphenoxy)-5-nitrobenzenesulfonyl]-urea 387217 N-n-pentyl-N'-[2-(4-ethoxyphenoxy)-5-nitrobenzenesulfonyl]-urea 387219 N-tert-butyl-N'-[2-(3-methoxyphenoxy)-5-nitrobenzenesulfonyl]urea 387220 N-tert-butyl-N'-[2-(3-methyl-4-chlorophenoxy)-5-nitrobenzenesulfonyl]urea 387222 N-n-pentyl-N'-[2-(3-methyl-4-chlorophenoxy)-5-nitrobenzenesulfonyl]urea 387223 N-tert-butyl-N'-[2-(2-methoxy-4-methylphenoxy)-5-nitrobenzenesulfonyl]urea 387243 N-tert-butyl-N'-[2-(4-methylphenoxy)-5-nitrobenzenesulfonyl]-N''-cyanoguanidine 387296 N-(3-{1-[4-(4-chlorophenyl)-4-oxobutyl)-4-piperidinyl]phenyl}-acetamide 387300 N-(3-{1-[4-(3,4-dimethylphenyl)-4-oxobutyl]-4-piperidinyl}phenyl)-acetamide 387301 N-(3-{1-[4-(4-chlorophenyl)-4-oxobutyl]-4-piperidinyl}phenyl)-2-methylpropanamide 387309 4-(2-ethylphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 387310 4-(2-propylphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 387311 4-(2-butylphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 387312 4-[2-(1-methylethyl)phenyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 387314 4-[2-(1,1-dimethylethyl)phenyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 387316 4-(2-diphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 387317 4-(2-dimethylaminophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 387318 4-(2-methylaminophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 387319 4-(2-aminophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 387320 4-(2-acetylaminophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 387322 N-(3-{1-[4-(4-chlorophenyl)-4-oxobutyl]-4-piperidinyl}phenyl)-2-phenylacetamide 387324 4-(2-methylsulfonamidophenyl)-N-(1,2,3,tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 387325 2-methyl-N-(3-{1-[3-(4-methylphenoxy)benzyl]-4-piperidinyl}phenyl)-propanamide 387327 4-(2-fluorophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 387328 N-(3-{1-[3-(4-methoxyphenoxy)benzyl]-4-piperidinyl}phenyl)-2methylpropanamide 387332 4-(2-pyridinyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 387333 4-(2-pyridinyl-N-oxide)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 387335 2-methyl-N-{3-[1-(4-phenoxybenzyl)-4-piperidinyl]phenyl}-propanamide 387337 N-(3-{1-[4-(4-chlorophenoxy)benzyl]-4-piperidinyl}phenyl)-2-methylpropanamide 387338 N-(3-{1-[4-(4-methoxyphenoxy)benzyl]-4-piperidinyl}phenyl)-2-methylpropanamide 387340 N-(3-{1-[4-(3,4-dichlorophenoxy)benzyl]-4-piperidinyl}phenyl)-2-methylpropanamide 387341 N-(3-(1-(4-(3,4-difluorophenoxy)benzyl)piperidin-4-yl)phenyl)isobutyramide 387342 N-(5-{1-[4-(3,4-difluorophenoxy)benzyl]-4-piperidinyl}-4-methylphenyl)-2-methylpropanamide 387343 N-(3-{1-4-(3,4-difluorophenoxy)benzyl]-4-piperidinyl}-4-methylphenyl)-2-methylpropanamide 387588 3-(2-methoxy-phenyl)-5,10-dihydro-dibenzo[b,e][1,4]diazepin-11-one 387589 3-(3-methoxy-phenyl)-5,10-dihydro-dibenzo[b,e][1,4]diazepin-11-one 387591 3-(3-cyano-phenyl)-5,10-dihydro-dibenzo[b,e][1,4]diazepin-11-one 387593 3-(2-acetyl-phenyl)-5,10-dihydro-dibenzo[b,e][1,4]diazepin-11-one 387594 3-(3-acetyl-phenyl)-5,10-dihydro-dibenzo[b,e][1,4]diazepin-11-one 387596 3-(4-hydroxy-3-methoxyphenyl)-5H-dibenzo[b,e][1,4]diazepin-11(10H)-one 387598 3-(3-methoxy-4-nitrophenyl)-5H-dibenzo[b,e][1,4]diazepin-11(10H)-one 387600 2-methoxy-4-(11-oxo-10,11-dihydro-5H-dibenzo[b,e][1,4]-diazepin-3-yl)-benzonitrile 387601 3-(4-chloro-3-methoxy-phenyl)-5,10-dihydro-dibenzo[b,e][1,4]-diazepin-11-one 387603 3-(4-acetyl-3-methoxy-phenyl)-5,10-dihydro-dibenzo[b,e][1,4]-diazepin-11-one 387604 methyl 2-methoxy-4-(11-oxo-10,11-dihydro-5H-dibenzo[b,e]-[1,4]diazepin-3-yl)benzoate 387605 2-methoxy-4-(11-oxo-10,11-dihydro-5H-dibenzo[b,e][1,4]-diazepin-3-yl)benzamide 387608 9-hydroxy-3-(3-methoxy-4-nitrophenyl)-5H-dibenzo[b,e][1,4]-diazepin-11(10H)-one 387609 8-hydroxy-3-(3-methoxy-4-nitrophenyl)-5H-dibenzo[b,e][1,4]-diazepin-11(10H)-one 387611 8-methoxy-3-(3-methoxy-4-nitrophenyl)-5H-dibenzo[b,e][1,4]-diazepin-11(10H)-one 387612 6-methoxy-3-(3-methoxy-4-nitrophenyl)-5H-dibenzo[b,e][1,4]-diazepin-11(10H)-one 387614 3-(3-methoxy-4-nitrophenyl)-6-(pyridin-4-ylmethoxy)-5Hdibenzo[b,e][1,4]diazepin-11(10H)-one 387615 8-amino-3-(3-methoxy-4-nitrophenyl)-5H-dibenzo[b,e][1,4]-diazepin-11(10H)-one 387617 8-(1,1-dioxo-1l6-isothiazolidin-2-yl)-3-(3-methoxy-4-nitrophenyl)-5,10-dihydro-dibenzo[b,e][1,4]diazepin-11-one 387618 3-(3-methoxy-4-nitrophenyl)-8-(2-oxopyrrolidin-1-yl)-5,10-dihydro-11H-dibenzo[b,e][1,4]diazepin-11-one 387621 7-amino-3-(4-amino-3-methoxy-phenyl)-5,10-dihydro-dibenzo[b,e][1,4]diazepin-11-one 387623 3-(4-amino-3-methoxy-phenyl)-7-morpholin-4-yl-5,10-dihydro-dibenzo[b,e][1,4]diazepin-11-one 387624 methyl [3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5H-dibenzo[b,e][1,4]diazepin-8-yl]acetate 387626 2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5Hdibenzo[b,e][1,4]diazepin-8-yl]-N,N-dimethylacetamide 387627 2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5Hdibenzo[b,e][1,4]diazepin-8-yl]-N-[4-(4-morpholinyl)phenyl]acetamide 387628 2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5Hdibenzo[b,e][1,4]diazepin-8-yl]-2-methyl-N-(4-morpholin-4-ylphenyl)propanamide 387629 3-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5Hdibenzo[b,e][1,4]diazepin-8-yl]-N,N-dimethylpropanamide 387631 3-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5Hdibenzo[b,e][1,4]diazepin-8-yl]-N-(4-morpholin-4-ylphenyl)propanamide 387632 2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5Hdibenzo[b,e][1,4]diazepin-7-yl]-N,N-dimethylacetamide 387633 2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5Hdibenzo[b,e][1,4]diazepin-7-yl]-2-methyl-N-(4-morpholin-4-ylphenyl)propanamide 387635 3-(3-methoxy-4-nitrophenyl)-5-methyl-5H-dibenzo[b,e][1,4]-diazepin-11(10H)-one 387636 methyl 2-(3-(3-Methoxy-4-nitrophenyl)-11-oxo-10,11-dihydrodibenzo[b,f][1,4]oxazepin-8-yl)acetate 387818 2-phenyl-2H-pyrazolo[3,4-c]quinolin-4(5H)-one 387819 2-m-tolyl-2H-pyrazolo[3,4-c]quinolin-4(5H)-one 387820 2-p-tolyl-2H-pyrazolo[3,4-c]quinolin-4(5H)-one 387821 2-(4-methoxyphenyl)-2H-pyrazolo[3,4-c]quinolin-4(5H)-one 387822 2-(3-methoxyphenyl)-2H-pyrazolo[3,4-c]quinolin-4(5H)-one 387823 2-(4-nitrophenyl)-2H-pyrazolo[3,4-c]quinolin-4(5H)-one 387824 2-benzyl-2H-pyrazolo[3,4-c]quinolin-4(5H)-one 387825 2-(3-methoxyphenyl)-2H-pyrazolo[3,4-c]quinolin-4-amine 387826 N-(2-m-tolyl-2H-pyrazolo[3,4-c]quinolin-4-yl)acetamide 387827 N-(2-p-tolyl-2H-pyrazolo[3,4-c]quinolin-4-yl)acetamide 387828 N-(2-(4-methoxyphenyl)-2H-pyrazolo[3,4-c]quinolin-4-yl)acetamide 387829 N-(2-m-tolyl-2H-pyrazolo[3,4-c]quinolin-4-yl)benzamide 387830 N-(2-p-tolyl-2H-pyrazolo[3,4-c]quinolin-4-yl)benzamide 387831 N-(2-(4-methoxyphenyl)-2H-pyrazolo[3,4-c]quinolin-4-yl)benzamide 387832 2-phenyl-N-(2-m-tolyl-2H-pyrazolo[3,4-c]quinolin-4-yl)acetamide 387833 2-phenyl-N-(2-p-tolyl-2H-pyrazolo[3,4-c]quinolin-4-yl)acetamide 387834 N-(2-(4-methoxyphenyl)-2H-pyrazolo[3,4-c]quinolin-4-yl)-2-phenylacetamide 387835 2,2-diphenyl-N-(2-phenyl-2H-pyrazolo[3,4-c]quinolin-4-yl)acetamide 387837 2,2-diphenyl-N-(2-m-tolyl-2H-pyrazolo[3,4-c]quinolin-4-yl)acetamide 387838 2,2-diphenyl-N-(2-p-tolyl-2H-pyrazolo[3,4-c]quinolin-4-yl)acetamide 387841 N-(2-(4-methoxyphenyl)-2H-pyrazolo[3,4-c]quinolin-4-yl)-2,2-diphenylacetamide 387842 1-benzyl-3-(2-m-tolyl-2H-pyrazolo[3,4-c]quinolin-4-yl)urea 387844 1-benzyl-3-(2-p-tolyl-2H-pyrazolo[3,4-c]quinolin-4-yl)urea 387846 N-benzoyl-N-(2-phenyl-2H-pyrazolo[3,4-c]quinolin-4-yl)benzamide 387847 N-benzoyl-N-(2-phenyl-2H-pyrazolo[3,4-c]quinolin-4-yl)-benzamide 387848 N-benzoyl-N-(2-p-tolyl-2H-pyrazolo[3,4-c]quinolin-4-yl)-benzamide 387849 N-benzoyl-N-[2-(4-methoxy-phenyl)-2H-pyrazolo[3,4-c]quinolin-4-yl]-benzamide 388114 [Aib5]hNPS 388171 (6aR-trans)-3-(1-hexylcyclobutyl)-6a,7,10,10a-tetrahydro-6,6,9-trimethyl-6H-dibenzo[b,d]pyran-1-ol 388172 (6aR-trans)-3-(1-hexylcyclohexyl)-6a,7,10,10a-tetrahydro-6,6,9-trimethyl-6H-dibenzo[b,d]pyran-1-ol 388173 (6aR-trans)-3-(1-heptylcyclopropyl)-6a,7,10,10a-tetrahydro-6,6,9-trimethyl-6H-dibenzo[b,d]pyran-1-ol 388174 (6aR-trans)-3-(1-heptylcyclobutyl)-6a,7,10,10a-tetrahydro-6,6,9-trimethyl-6H-dibenzo[b,d]pyran-1-ol 388175 (6aR-trans)-3-(1-heptylcyclopentyl)-6a,7,10,10a-tetrahydro-6,6,9-trimethyl-6H-dibenzo[b,d]pyran-1-ol 388176 (6aR-trans)-3-(1-heptylcyclohexyl)-6a,7,10,10a-tetrahydro-6,6,9-trimethyl-6H-dibenzo[b,d]pyran-1-ol 388177 (6aR-trans)-3-[1-[(1Z)-1-hexenyl]cyclopropyl]-6a,7,10,10a-tetrahydro-6,6,9-trimethyl-6H-dibenzo[b,d]pyran-1-ol 388178 (6aR-trans)-3-[1-[(1Z)-1-hexenyl]cyclobutyl]-6a,7,10,10a-tetrahydro-6,6,9-trimethyl-6H-dibenzo[b,d]pyran-1-ol 388179 (6aR-trans)-3-[1-[(1Z)-1-hexenyl]cyclopentyl]-6a,7,10,10a-tetrahydro-6,6,9-trimethyl-6H-dibenzo[b,d]pyran-1-ol 388180 (6aR-trans)-3-[1-[(1Z)-1-hexenyl]cyclohexyl]-6a,7,10,10a-tetrahydro-6,6,9-trimethyl-6H-dibenzo[b,d]pyran-1-ol 388293 2-(4-{4-[N-(3-{3-[3-(N-{3-[(1-{2-[(4-amino-5-chloro-2-methoxyphenyl)carbonyloxy]ethyl}piperidin-4-yl)carbamoyl]propyl}-2,2-dimethylpropanamido)propyl]phenyl}propyl)-2,2-dimethylpropanamido]butanamido}piperidin-1-yl)ethyl 4-amino-5-chloro-2-methoxybenzoate 388298 2-[4-({5-[(1-{2-[(4-amino-5-chloro-2-methoxyphenyl)carbonyloxy]ethyl}piperidin-4-yl)carbamoyl]pentyl}carbamoyl)piperidin-1-yl]ethyl 4-amino-5-chloro-2-methoxybenzoate 388301 2-[4-({10-[(1-{2-[(4-amino-5-chloro-2-methoxyphenyl)carbonyloxy]ethyl}piperidin-4-yl)carbamoyl]decyl}carbamoyl)piperidin-1-yl]ethyl 4-amino-5-chloro-2-methoxybenzoate 388319 N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-4-pyridin-2-ylbenzamide 388321 N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)-trans-but-2-enyl)-4-(6-oxo-1,6-dihydropyridin-2-yl)benzamide 388322 N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)-trans-but-2-enyl)-4-(6-methylpyridin-2-yl)benzamide 388323 N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)-trans-but-2-enyl)-4-(3-methylpyridin-2-yl)benzamide 388324 N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)-trans-but-2-enyl)-4-(pyridin-N-oxide-2-yl)benzamide 388325 4-(2,3-dichlorophenyl)-1-(4-(4-(pyridin-2-yl)benzamido)-transbut-2-enyl)piperazine 1-oxide 388326 N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)-trans-but-2-enyl)-4-pyridin-2-ylbenzamide 388327 N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)-trans-but-2-enyl)-9H-fluorene-2-carboxamide 388328 N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)-3-hydroxybutyl)-4-pyridin-2-ylbenzamide 388330 N-(3-(4-(2,3-dichlorophenyl)piperazin-1-yl)-3-hydroxybutyl)-9H-fluorene-2-carboxamide 388332 N-(3-hydroxy-4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-4-pyridin-2-ylbenzamide 388336 N-(3-hydroxy-4-(4-(2-methoxyphenyl)piperazin-1-yl)-butyl)-9H-fluorene-2-carboxamide 388337 1-(4-(2,3-dichlorophenyl)piperazin-1-yl)-4-(4-(pyridin-2-yl)-benzamido)butan-2-yl acetate 388338 N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)-2-hydroxybutyl)-4-(pyridin-2-yl)benzamide 388341 N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)-2-hydroxybutyl)-9H-fluorene-2-carboxamide 388342 N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)-2-hydroxybutyl)-9H-fluorene-2-carboxamide 388343 N-(2-(4-(2,3-dichlorophenyl)piperazin-1-ylmethyl)-trans-cyclopropylmethyl)-4-pyridin-2-ylbenzamide 388344 N-(2-(4-(2,3-dichlorophenyl)piperazin-1-ylmethyl)-cis-cyclopropylmethyl)-4-pyridin-2-ylbenzamide 388399 4-(2-(4-chloro-3-(trifluoromethyl)phenylamino)-1H-benzo[d]imidazol-5-yloxy)-N-methylpicolinamide 388400 (4-chloro-3-trifluoromethyl-phenyl)-[5-(pyridin-4-yloxy)-1H-benzimidazol-2-yl]-amine 388401 (4-chloro-phenyl)-[5-(6,7-dimethoxy-quinazolin-4-yloxy)-1Hbenzoimidazol-2-yl]-amine 388402 (4-chloro-3-trifluoromethyl-phenyl)-[6-(1H-pyrrolo[2,3-b]pyridin-4-yloxy)-1H-benzimidazol-2-yl]-amine 388403 4-{2-[4-chloro-3-(4-methyl-piperazin-1-ylmethyl)-phenylamino]-1H-benzimidazol-5-yloxy}-pyridine-2-carboxylic acid methylamide 388404 4-((2-((3-((2-(dimethylamino)ethyl)oxy)-4-(trifluoromethyl)-phenyl)amino)-1H-benzimidazol-5-yl)oxy)-N-methyl-2-pyridinecarboxamide 388405 N-methyl-4-((2-((3-((((2R)-1-methyl-2-pyrrolidinyl)methyl)-oxy)-4-(trifluoromethyl)phenyl)amino)-1H-benzimidazol-5-yl)-oxy)-2-pyridinecarboxamide 388406 (R)-4-{2-[3-(1-methyl-pyrrolidin-2-ylmethoxy)-4-pentafluoroethyl-phenylamino]-1H-benzimidazol-5-yloxy}-pyridine-2-carboxylic acid methylamide 388407 N-methyl-4-((2-((3-((2-(1-pyrrolidinyl)ethyl)oxy)-5-(trifluoromethyl)phenyl)amino)-1H-benzimidazol-5-yl)oxy)-2-pyridinecarboxamide 388408 N-(3-((((2R)-1-methyl-2-pyrrolidinyl)methyl)oxy)-4-(trifluoromethyl)phenyl)-5-(4-quinolinyloxy)-1H-benzimidazol-2-amine 388409 [4-chloro-3-(4-methyl-piperazin-1-ylmethyl)-phenyl]-[5-(quinolin-4-yloxy)-1H-benzimidazol-2-yl]-amine 388410 [4-chloro-3-(4-methylpiperazin-1-ylmethyl)-phenyl]-[5-(6,7-dimethoxyquinolin-4-yloxy)-1H-benzimidazol-2-yl]-amine 388411 [4-chloro-3-(4-methyl-piperazin-1-ylmethyl)-phenyl]-[6-(7Hpyrrolo[2,3-d]pyrimidin-4-yloxy)-1H-benzimidazol-2-yl]-amine 388412 [4-chloro-3-(4-methyl-piperazin-1-ylmethyl)-phenyl]-[6-(1Hpyrrolo[2,3-b]pyridin-4-yloxy)-1H-benzimidazol-2-yl]-amine 388413 [4-chloro-3-(4-methylpiperazin-1-ylmethyl)phenyl]-[5-(2-methylamino-pyrimidin-4-yloxy)-1H-benzimidazol-2-yl]-amine 388414 [4-chloro-3-(4-methyl-piperazin-1-ylmethyl)-phenyl]-[5-(2-methylsulfanyl-pyrimidin-4-yloxy)-1H-benzimidazol-2-yl]-amine 388415 4-{2-[4-chloro-3-(4-methyl-piperazin-1-ylmethyl)-phenylamino]-1-methyl-1H-benzimidazol-5-yloxy}-pyridine-2-carboxylic acid methylamide 388416 4-{2-[4-chloro-3-(4-methyl-piperazin-1-ylmethyl)-phenylamino]-benzoxazol-5-yloxy}-pyridine-2-carboxylic acid methylamide 388417 4-((2-((4-Chloro-3-((((2S)-1-methyl-2-pyrrolidinyl)methyl)oxy)-phenyl)amino)-1,3-benzoxazol-5-yl)oxy)-N-methyl-2-pyridinecarboxamide 388418 4-{2-[4-chloro-3-(2-dimethylamino-ethoxy)-phenylamino]-benzoxazol-5-yloxy}-pyridine-2-carboxylic acid methylamide 388419 4-{2-[4-chloro-3-(2-diethylamino-ethoxy)-phenylamino]-benzoxazol-5-yloxy}-pyridine-2-carboxylic acid methylamide 388420 4-((2-((4-chloro-3-(4-morpholinylmethyl)phenyl)amino)-1,3-benzoxazol-5-yl)oxy)-N-methyl-2-pyridinecarboxamide 388421 4-{2-[4-chloro-3-(piperidin-4-ylmethoxy)-phenylamino]-benzoxazol-5-yloxy}-pyridine-2-carboxylic acid methylamide 388422 4-{2-[4-chloro-3-((2S)-1-methyl-pyrrolidin-2-ylmethoxy)-phenylamino]-benzooxazol-5-yloxy}-pyridine-2-carboxylic acid amide 388423 S-[4-chloro-3-(1-methyl-pyrrolidin-2-ylmethoxy)-phenyl]-[5-(6,7-dimethoxy-quinazolin-4-yloxy)-benzoxazol-2-yl]-amine 388424 S-[4-chloro-3-(1-methylpyrrolidin-2-ylmethoxy)-phenyl]-[5-(6,7-dimethoxyquinolin-4-yloxy)-benzoxazol-2-yl]-amine 388425 5-((6,7-bis(methoxy)-4-quinolinyl)oxy)-N-(4-chloro-3-((4-methyl-1-piperazinyl)methyl)phenyl)-1,3-benzoxazol-2-amine 388426 [4-chloro-3-(4-methyl-piperazin-1-ylmethyl)-phenyl]-[5-(quinolin-4-yloxy)-benzoxazol-2-yl]-amine 388427 [4-chloro-3-(4-methyl-piperazin-1-ylmethyl)-phenyl]-[5-(2-methylamino-pyrimidin-4-yloxy)-benzoxazol-2-yl]-amine 388428 [4-chloro-3-(4-methyl-piperazin-1-ylmethyl)-phenyl]-[5-(6-methylamino-pyrimidin-4-yloxy)-benzoxazol-2-yl]-amine 388429 N-(4-chloro-3-(((2S)-1-methyl-2-pyrrolidinyl)methoxy)phenyl)-5-(1H-pyrrolo[2,3-b]pyridin-4-yloxy)-1,3-benzoxazol-2-amine 388430 N-(4-chloro-3-((4-methyl-1-piperazinyl)methyl)phenyl)-5-(1H-pyrrolo[2,3-b]pyridin-4-yloxy)-1,3-benzoxazol-2-amine 388431 4-((2-((4-chloro-3-(((2S)-1-methyl-2-pyrrolidinyl)methoxy)-phenyl)amino)-7-fluoro-1,3-benzoxazol-5-yl)oxy)-N-methyl-2-pyridinecarboxamide 388432 4-{7-chloro-2-[4-chloro-3-(4-methyl-piperazin-1-ylmethyl)-phenylamino]-benzoxazol-5-yloxy}-pyridine-2-carboxylic acid methylamide 388433 [4-chloro-3-(4-methylpiperazin-1-ylmethyl)-phenyl]-[7-chloro-5-(quinolin-4-yloxy)-benzoxazol-2-yl]-amine 388441 4-[(3-chloro-4-fluorophenyl)amino]-8-fluoro-6-[(1H-imidazol-5-ylmethyl)amino]quinoline-3-carbonitrile 388445 8-chloro-quinoline-3-carbonitrile 388447 8-bromo-4-[(3-chloro-4-fluorophenyl)amino]-6-[(1H-imidazol-5-ylmethyl)amino]quinoline-3-carbonitrile 388448 4-[(3-chloro-4-fluorophenyl)amino]-6-[(1H-imidazol-5-ylmethyl)amino]-8-(trifluoromethyl)quinoline-3-carbonitrile 388449 6-((1H-imidazol-5-yl)methylamino)-4-(3-chloro-4-fluorophenylamino)-8-hydroxyquinoline-3-carbonitrile 388450 4-(3-chloro-4-fluorophenylamino)-6-[(3H-imidazol-4-ylmethyl)-amino]-8-methoxyquinoline-3-carbonitrile 388451 4-[(3-chloro-4-fluorophenyl)amino]-6-[(1H-imidazol-5-ylmethyl)amino]-8-(methylsulfinyl)quinoline-3-carbonitrile 388453 4-[(3-chloro-4-fluorophenyl)amino]-6-[(1H-imidazol-5-ylmethyl)amino]-8-(methylsulfonyl)quinoline-3-carbonitrile 388454 4-[(3-chloro-4-fluorophenyl)amino]-3-cyano-6-[(1H-imidazol-5-ylmethyl)amino]-N,N-dimethylquinoline-8-carboxamide 388455 8-acetyl-4-[(3-chloro-4-fluorophenyl)amino]-6-[(1H-imidazol-5-ylmethyl)amino]quinoline-3-carbonitrile 388456 4-[(3-chloro-4-fluorophenyl)amino]-8-(2,3-dihydroxypropyl)-6-[(1H-imidazol-5-ylmethyl)amino]quinoline-3-carbonitrile 388457 4-[(3-chloro-4-fluorophenyl)amino]-8-(2,3-dihydroxypropoxy)-6-[(1H-imidazol-5-ylmethyl)amino]quinoline-3-carbonitrile 388458 8-chloro-4-[(3-chloro-4-fluorophenyl)amino]-6-{[2-(1H-imidazol-5-yl)ethyl]amino}quinoline-3-carbonitrile 388460 8-chloro-4-[(3-chloro-4-fluorophenyl)amino]-6-{[(1-methyl-1H-pyrazol-4-yl)methyl]amino}quinoline-3-carbonitrile 388461 8-bromo-4-(3-chloro-4-fluorophenylamino)-6-[(2-phenyl-2Hpyrazol-3-ylmethyl)amino]quinoline-3-carbonitrile 388462 8-bromo-4-[(3-chloro-4-fluorophenyl)amino]-6-[(imidazo[1,2-a]pyridin-3-ylmethyl)amino]quinoline-3-carbonitrile 388463 8-chloro-4-(3-chloro-4-fluorophenylamino)-6-(pyridin-3-ylmethylamino)quinoline-3-carbonitrile 388469 8-chloro-4-[(3-chloro-4-fluorophenyl)amino]-6-({[5-(4-hydroxy-1-isopropylpiperidin-4-yl)pyridin-3-yl]methyl}amino)quinoline-3-carbonitrile 388472 8-chloro-4-[(3-chloro-4-fluorophenyl)amino]-6-{[(6-methylpyridin-2-yl)methyl]amino}quinoline-3-carbonitrile 388480 8-chloro-4-[(3-chloro-4-fluorophenyl)amino]-6-{[(6-morpholin-4-ylpyridin-2-yl)methyl]amino}quinoline-3-carbonitrile 388482 8-chloro-4-[(3-chloro-4-fluorophenyl)amino]-6-{[(1-oxidopyridin-2-yl)methyl]amino}quinoline-3-carbonitrile 388484 8-chloro-4-[(3-chloro-4-fluorophenyl)amino]-6-[(2,3-dihydroxypropyl)amino]quinoline-3-carbonitrile 388485 8-chloro-4-[(3-chloro-4-fluorophenyl)amino]-6-[(1H-tetrazol-5-ylmethyl)amino]quinoline-3-carbonitrile 388487 2-(8-chloro-4-(3-chloro-4-fluorophenylamino)-3-cyanoquinolin-6-ylamino) acetic acid 388489 N2-{8-chloro-4-[(3-chloro-4-fluorophenyl)amino]-3-cyanoquinolin-6-yl}-N-pyridin-3-ylglycinamide 388492 6-((1H-1,2,3-triazol-4-yl)methylamino)-8-bromo-4-(3-chloro-4-fluorophenylamino)quinoline-3-carbonitrile 388496 8-bromo-4-(3-chloro-4-fluorophenylamino)-6-((1-(3-(dimethylamino)propyl)-1H-1,2,3-triazol-4-yl)methylamino)quinoline-3-carbonitrile 388503 8-bromo-4-[(3-chloro-4-fluorophenyl)amino]-6-{[(4-isopropyl-1H-imidazol-5-yl)methyl]amino}quinoline-3-carbonitrile 388504 8-chloro-4-[(3-chloro-4-fluorophenyl)amino]-6-{[(5-isopropyl-1H-imidazol-4-yl)methyl]amino}quinoline-3-carbonitrile 388505 8-chloro-4-[(3-chloro-4-fluorophenyl)amino]-6-{[(5-propyl-1H-imidazol-4-yl)methyl]amino}quinoline-3-carbonitrile 388506 8-chloro-4-[(3-chloro-4-fluorophenyl)amino]-6-{[(5-ethyl-1H-imidazol-4-yl)methyl]amino}quinoline-3-carbonitrile 388507 methyl 5-[({8-bromo-4-[(3-chloro-4-fluorophenyl)amino]-3-cyanoquinolin-6-yl}amino)methyl]-1H-imidazole-4-carboxylate 388508 8-chloro-4-[(3-chloro-4-fluorophenyl)amino]-6-[({4-[3-(dimethylamino)propyl]-1H-imidazol-5-yl}methyl)amino]quinoline-3-carbonitrile 388509 8-bromo-4-(3-chloro-4-fluorophenylamino)-6-((1-methyl-1H-imidazol-4-yl)methylamino)quinoline-3-carbonitrile 388510 8-chloro-4-(3-chloro-4-fluorophenylamino)-6-((2-ethyl-5-methyl-1H-imidazol-4-yl)methylamino)quinoline-3-carbonitrile 388511 8-chloro-4-[(3-chloro-4-fluorophenyl)amino]-6-{[(2,5-dimethyl-1H-imidazol-4-yl)methyl]amino}quinoline-3-carbonitrile 388512 8-bromo-4-(3-chloro-4-fluorophenylamino)-6-((2-phenyl-1H-imidazol-5-yl)methylamino)quinoline-3-carbonitrile 388513 8-bromo-4-[(3-chloro-4-fluorophenyl)amino]-6-({[1-(2-morpholin-4-ylethyl)-1H-imidazol-4-yl]methyl}amino)quinoline-3-carbonitrile 388515 8-bromo-4-[(3-chloro-4-fluorophenyl)amino]-6-[({1-[2-(methylsulfonyl)ethyl]-1H-imidazol-4-yl}methyl)amino]quinoline-3-carbonitrile 388516 (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propoxy]phenyl)-imidazo[1,2-a]pyridine 388517 (4-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]propoxy]phenyl)imidazo[1,2-a]pyridine 388518 (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propoxy]phenyl)-6-methylimidazo[1,2-a]pyridine 388520 (4-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]propoxy]phenyl)-6-methylimidazo[1,2-a]pyridine 388521 (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propoxy]phenyl)-7-methylimidazo[1,2-a]pyridine 388522 (4-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]propoxy]phenyl)-7-methylimidazo[1,2-a]pyridine 388523 (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propoxy]phenyl)-8-methylimidazo[1,2-a]pyridine 388524 (4-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]propoxy]phenyl)-8-methylimidazo[1,2-a]pyridine 388525 (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]butoxy]phenyl)imidazo[1,2-a]pyridine 388526 (4-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy]phenyl)imidazo[1,2-a]pyridine 388527 (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]butoxy]phenyl)-6-methylimidazo[1,2-a]pyridine 388528 (4-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy]phenyl)-6-methylimidazo[1,2-a]pyridine 388531 (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]butoxy]phenyl)-7-methylimidazo[1,2-a]pyridine 388532 (4-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy]phenyl)-7-methylimidazo[1,2-a]pyridine 388535 (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]butoxy]phenyl)-8-methylimidazo[1,2-a]pyridine 388540 (4-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy]phenyl)-8-methylimidazo[1,2-a]pyridine 388665 8-chloro-5H-dibenzo[b,e][1,4]diazepin-11(10H)-one 388782 (R)-N-(1-((1-(3-morpholinopropylamino)-1-oxo-3-phenylpropan-2-yl)carbamoyl)cyclopentyl)benzo[b]thiophene-2-carboxamide 388784 benzo[b]thiophene-2-carboxylic acid {1-methyl-1-[1-(R)-(3-morpholin-4-yl-propylcarbamoyl)-ethyl}-amide 388785 benzo[b]thiophene-2-carboxylic acid {1-[1-(R)-(3-morpholin-4-yl-propylcarbamoyl)-2-phenylethylcarbamoyl]-cyclopropyl}-amide 388786 benzo[b]thiophene-2-carboxylic acid {1-[1-(R)-(3-morpholin-4-yl-propylcarbamoyl)-2-phenylethylcarbamoyl]-cyclopent-3-enyl}-amide 388787 benzo[b]thiophene-2-carboxylic acid methyl-{[1-(R)-(3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethylcarbamoyl]-methyl}-amide 388788 benzo[b]thiophene-2-carboxylic acid methyl-{1-[1-(R)-(3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethylcarbamoyl]-cyclopentyl}-amide 388789 benzo[b]thiophene-2-carboxylic acid methyl-{1-[1-(3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethylcarbamoyl]-cyclohexyl}-amide 388790 3-chloro-N-{1-[1-(R)-(3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethylcarbamoyl]-cyclopentyl}-benzamide 388791 N-{1-[1-(R)-(3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethylcarbamoyl]-cyclopentyl}-4-nitro-benzamide 388792 4-iodo-N-{1-[1-(R)-(3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethylcarbamoyl]-cyclopentyl}-benzamide 388793 1-[3-(4-bromo-phenyl)-ureido]-cyclopentanecarboxylic acid [1-(R)-(3-morpholin-4-ylpropylcarbamoyl)-2-phenyl-ethyl]-amide 388794 1-[3-(4-methylsulfanyl-phenyl)-ureido]-cyclopentanecarboxylic acid [1-(R)-(3-morpholin-4-ylpropylcarbamoyl)-2-phenyl-ethyl]-amide 388795 1-[3-(4-iodo-phenyl)-ureido]-cyclopentanecarboxylic acid [1-(R)-(3-morpholin-4-ylpropylcarbamoyl)-2-phenyl-ethyl]-amide 388796 1-[3-(3,4-difluoro-phenyl)-ureido]-cyclopentanecarboxylic acid [1-(R)-(3-morpholin-4-ylpropylcarbamoyl)-2-phenyl-ethyl]-amide 388797 1-[3-(4-bromo-3-methyl-phenyl)-ureido]-cyclopentanecarboxylic acid [1-(R)-(3-morpholin-4-ylpropylcarbamoyl)-2-phenyl-ethyl]-amide 388798 1-[3-(4-iodo-phenyl)-thioureido]-cyclopentanecarboxylic acid [1-(R)-(3-morpholin-4-ylpropylcarbamoyl)-2-phenyl-ethyl]-amide 388799 1-[3-(3,4-dichloro-phenyl)-thioureido]-cyclopentanecarboxylic acid [1-(3-morpholin-4-ylpropylcarbamoyl)-2-phenyl-ethyl]-amide 388800 benzofuran-2-carboxylic acid {1-[1-(R)-(3-morpholin-4-yl-propylcarbamoyl)-2-phenylethylcarbamoyl]-cyclopentyl}-amide 388802 1H-indole-2-carboxylic acid {1-[1-(R)-(3-morpholin-4-yl-propylcarbamoyl)-2-phenylethylcarbamoyl]-cyclopentyl}-amide 388803 3-chloro-4-fluorophenyl-(4-fluoro-4-{[(5-hydroxymethylpyridin-2-ylmethyl)-amino]-methyl}-piperidin-1-yl)-methanone 388804 1-methyl-1H-indole-2-carboxylic acid {1-[1-(R)-(3-morpholin-4-yl-propylcarbamoyl)-2-phenylethylcarbamoyl]-cyclopentyl}-amide 388805 naphthalene-2-carboxylic acid {1-[1-(R)-(3-morpholin-4-yl-propylcarbamoyl)-2-phenylethylcarbamoyl]-cyclopentyl}-amide 388806 3-chloro-4-fluorophenyl-(4-fluoro-4-{[(5-fluoromethylpyridin-2-ylmethyl)-amino]-methyl}-piperidin-1-yl)-methanone 388807 quinoline-6-carboxylic acid {1-[1-(R)-(3-morpholin-4-yl-propylcarbamoyl)-2-phenylethylcarbamoyl]-cyclopentyl}-amide 388808 3-chloro-4-fluorophenyl-(4-fluoro-4-{[(5-difluoromethylpyridin-2-ylmethyl)-amino]-methyl}-piperidin-1-yl)-methanone 388809 biphenyl-4-carboxylic acid {1-[1-(R)-(3-morpholin-4-yl-propylcarbamoyl)-2-phenylethylcarbamoyl]-cyclopentyl}-amide 388810 5-phenyl-thiophene-2-carboxylic acid {1-(R)-[1-(3-morpholin-4-yl-propylcarbamoyl)-2-phenylethylcarbamoyl]-cyclopentyl}-amide 388811 1-(3-phenyl-acryloylamino)-cyclopentanecarboxylic acid [1-(R)-(3-morpholin-4-ylpropylcarbamoyl)-2-phenyl-ethyl]-amide 388812 3-chloro-4-fluorophenyl-(4-fluoro-4-{[(5-chloropyridin-2-ylmethyl)-amino]-methyl}-piperidin-1-yl)-methanone 388813 benzo[b]thiophene-2-carboxylic acid {1-[2-phenyl-(R)-1-(3-thiomorpholin-4-ylpropylcarbamoyl)-ethylcarbamoyl]-cyclopentyl}-amide 388814 3-chloro-4-fluorophenyl-(4-fluoro-4-{[(6-methylpyridazin-3-ylmethyl)-amino]-methyl}-piperidin-1-yl)-methanone 388816 3-chloro-4-fluorophenyl-(4-fluoro-4-{[(5-methylpyrazin-2-ylmethyl)-amino]-methyl}-piperidin-1-yl)-methanone 388817 3-chloro-4-fluorophenyl-(4-fluoro-4-{[(5-methylpyrimidin-2-ylmethyl)-amino]-methyl}-piperidin-1-yl)-methanone 388818 7-methyl-6,7,8,9,10,15-hexahydro-5H-dibenzo[d,g]azacycloundecene-12-ol 388819 1-(2-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)ethyl)-1H-benzo[d]imidazol-2(3H)-one 388820 12-methoxy-7-methyl-6,7,8,9,10,15-hexahydro-5H-dibenzo[d,g]azacycloundecine 388821 3-chloro-4-fluorophenyl-(4-fluoro-4-{[(pyrimidin-2-ylmethyl)-amino]-methyl}-piperidin-1-yl)-methanone 388822 7-methyl-6,7,8,9,10,15-hexahydro-5H-dibenzo[d,g]azacycloundecin-3-ol 388823 3-methoxy-7-methyl-6,7,8,9,10,15-hexahydro-5H-dibenzo[d,g]azacycloundecine 388824 3-chloro-4-fluorophenyl-(4-fluoro-4-{[(5-carbomethoxypyrimidin-2-ylmethyl)-amino]-methyl}-piperidin-1-yl)-methanone 388825 8-methyl-5,6,7,8,9,10,11,16-octahydrodibenzo[e,h]azacyclododecene-3-ol 388826 3-methoxy-8-methyl-5,6,7,8,9,10,11,16-octahydrodibenzo[e,h]azacyclododecene 388827 3-chloro-4-fluorophenyl-(4-fluoro-4-{[(5-hydroxymethylpyrimidin-2-ylmethyl)-amino]-methyl}-piperidin-1-yl)-methanone 388829 3-chloro-4-fluorophenyl-(4-fluoro-4-{[(5-ethylpyrimidin-2-ylmethyl)-amino]-methyl}-piperidin-1-yl)-methanone 388830 6,7,8,9,10,15-hexahydro-5H-dibenzo[d,g]azacycloundecin-12-ol 388831 3-chloro-4-fluorophenyl-(4-fluoro-4-{[(5-difluoromethylpyrimidin-2-ylmethyl)-amino]-methyl}-piperidin-1-yl)-methanone 388832 3-chloro-4-fluorophenyl-(4-fluoro-4-{[(5-chloropyrimidin-2-ylmethyl)-amino]-methyl}-piperidin-1-yl)-methanone 388834 3-chloro-4-fluorophenyl-(4-fluoro-4-{[(4-methoxypyrimidin-2-ylmethyl)-amino]-methyl}-piperidin-1-yl)-methanone 388836 3-chloro-4-fluorophenyl-(4-fluoro-4-{[(4-methylaminopyrimidin-2-ylmethyl)-amino]-methyl}-piperidin-1-yl)-methanone 388837 2-methoxy-7-methyl-6,7,8,9,10,15-hexahydro-5H-dibenzo[d,g]azacycloundecene 388838 3-chloro-4-fluorophenyl-(4-fluoro-4-{[(4-dimethylaminopyrimidin-2-ylmethyl)-amino]-methyl}-piperidin-1-yl)-methanone 388839 7-methyl-6,7,8,9,10,15-hexahydro-5H-dibenzo[d,g]azacycloundecene-2-ol 388841 3-chloro-4-fluorophenyl-(4-fluoro-4-{[(4-fur-2-yl-pyrimidin-2-ylmethyl)-amino]-methyl}-piperidin-1-yl)-methanone 388843 5,6-dimethoxy-11-methyl-11-aza-tricyclo[13.4.0.0.3,8]nonadeca-1(15),3(8),4,6,16,18-hexaene 388844 3-chloro-4-fluorophenyl-(4-fluoro-4-{[(4-methylamino-5-methylpyrimidin-2-ylmethyl)-amino]-methyl}-piperidin-1-yl)-methanone 388847 3-chloro-4-fluorophenyl-(4-fluoro-4-{[(4-methylamino-5-chloropyrimidin-2-ylmethyl)-amino]-methyl}-piperidin-1-yl)-methanone 388855 benzo[b]thiophene-2-carboxylic acid (1-{1-(R)-[3-(4-hydroxy-piperidin-1-yl)-propylcarbamoyl]-2-phenyl-ethylcarbamoyl}-cyclopentyl)-amide 388857 benzo[b]thiophene-2-carboxylic acid (1-{2-phenyl-1-(R)-[3-(4-sulfamoyl-piperazin-1-yl)-propylcarbamoyl]-ethylcarbamoyl}-cyclopentyl)-amide 388858 benzo[b]thiophene-2-carboxylic acid (1-{1-(R)-[3-(4-morpholin-4-yl-piperidin-1-yl)-propylcarbamoyl]-2-phenyl-ethylcarbamoyl}-cyclopentyl)-amide 388859 benzo[b]thiophene-2-carboxylic acid (1-{2-phenyl-1-(R)-[3-(tetrahydro-pyran-4-ylamino)-propylcarbamoyl]-ethylcarbamoyl}-cyclopentyl)-amide 388860 benzo[b]thiophene-2-carboxylic acid (1-{1-(R)-[3-(2-hydroxy-1-hydroxymethyl-ethylamino)-propylcarbamoyl]-2-phenyl-ethylcarbamoyl}-cyclopentyl)-amide 388861 benzo[b]thiophene-2-carboxylic acid [1-(1-(R)-{3-[bis-(2-hydroxy-ethyl)-amino]-propylcarbamoyl}-2-phenyl-ethylcarbamoyl)-cyclopentyl]-amide 388862 benzo[b]thiophene-2-carboxylic acid(1-{1-(R)-[4-(4-morpholin-4-yl-piperidin-1-yl)-4-oxobutylcarbamoyl]-2-phenylethylcarbamoyl}-cyclopentyl)-amide 388863 benzo[b]thiophene-2-carboxylic acid (1-{1-(R)-[3-(4-morpholin-4-yl-piperidin-1-yl)-3-oxopropylcarbamoyl]-2-phenyl-ethylcarbamoyl}-cyclopentyl)-amide 388864 benzo[b]thiophene-2-carboxylic acid (1-{1-(R)-[3-(4-methyl-piperazin-1-yl)-3-oxopropylcarbamoyl]-2-phenyl-ethylcarbamoyl}-cyclopentyl)-amide 388865 benzo[b]thiophene-2-carboxylic acid (1-{1-(R)-[3-oxo-3-(4-pyridin-2-yl-piperazin-1-yl)-propylcarbamoyl]-2-phenyl-ethylcarbamoyl}-cyclopentyl)-amide 388866 benzo[b]thiophene-2-carboxylic acid [1-(1-(R)-{3-oxo-3-[4-(tetrahydro-pyran-4-ylmethyl)-piperazin-1-yl]-propylcarbamoyl}-2-phenyl-ethylcarbamoyl)-cyclopentyl]-amide 388867 benzo[b]thiophene-2-carboxylic acid [1-(1-(R)-{3-oxo-3-[4-(tetrahydro-pyran-4-yl)-piperazin-1-yl]-propylcarbamoyl}-2-phenyl-ethylcarbamoyl)-cyclopentyl]-amide 388868 benzo[b]thiophene-2-carboxylic acid (1-{2-phenyl-1-(R)-[1-(tetrahydro-pyran-4-ylmethyl)-piperidin-4-ylcarbamoyl]-ethylcarbamoyl}-cyclopentyl)-amide 388869 benzo[b]thiophene-2-carboxylic acid [1-(2-phenyl-1-(R)-{[1-(tetrahydro-pyran-4-ylmethyl)-piperidin-4-ylmethyl]-carbamoyl}-ethylcarbamoyl)-cyclopentyl]-amide 388870 benzo[b]thiophene-2-carboxylic acid [1-(2-phenyl-1-(R)-{2-[1-(tetrahydro-pyran-4-ylmethyl)-piperidin-4-yl]-ethylcarbamoyl}-ethylcarbamoyl)-cyclopentyl]-amide 388871 benzo[b]thiophene-2-carboxylic acid [1-(2-phenyl-1-(R)-{[1-(tetrahydro-pyran-4-yl)-piperidin-4-ylmethyl]-carbamoyl}-ethylcarbamoyl)-cyclopentyl]-amide 388872 benzo[b]thiophene-2-carboxylic acid [1-(2-phenyl-1-(R)-{2-[1-(tetrahydro-pyran-4-yl)-piperidin-4-yl]-ethylcarbamoyl}-ethylcarbamoyl)-cyclopentyl]-amide 388873 4-chloro-benzo[b]thiophene-2-carboxylic acid {1-[1-(R)-(3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethylcarbamoyl]-cyclopentyl}-amide 388874 5-chloro-benzo[b]thiophene-2-carboxylic acid {1-[1-(R)-(3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethylcarbamoyl]-cyclopentyl}-amide 388875 6-chloro-benzo[b]thiophene-2-carboxylic acid {1-[1-(R)-(3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethylcarbamoyl]-cyclopentyl}-amide 388876 7-chloro-benzo[b]thiophene-2-carboxylic acid {1-[1-(R)-(3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethylcarbamoyl]-cyclopentyl}-amide 388877 3-chloro-benzo[b]thiophene-2-carboxylic acid {1-[1-(R)-(3-morpholin-4-yl-propylcarbamoyl)-2-phenyl-ethylcarbamoyl]-cyclopentyl}-amide 388879 6-chloro-benzo[b]thiophene-2-carboxylic acid [1-(2-phenyl-1(R)-{[1-(tetrahydro-pyran-4-ylmethyl)-piperidin-4-ylmethyl]-carbamoyl}-ethylcarbamoyl)-ciclopentyl]-amide 388880 6-fluoro-benzo[b]thiophene-2-carboxylic acid [1-(2-phenyl-1(R)-{[1-(tetrahydro-pyran-4-ylmethyl)-piperidin-4-ylmethyl]-carbamoyl}-ethylcarbamoyl)-ciclopentyl]-amide 388883 6-bromo-benzo[b]thiophene-2-carboxylic acid [1-(2-phenyl-1(R)-{[1-(tetrahydro-pyran-4-ylmethyl)-piperidin-4-ylmethyl]-carbamoyl}-ethylcarbamoyl)-ciclopentyl]-amide 388885 6-trifluoromethyl-benzo[b]thiophene-2-carboxylic acid [1-(2-phenyl-1(R)-{[1-(tetrahydropyran-4-ylmethyl)-piperidin-4-ylmethyl]-carbamoyl}-ethylcarbamoyl)-ciclopentyl]-amide 388887 6-methoxy-benzo[b]thiophene-2-carboxylic acid [1-(2-phenyl-1(R)-{[1-(tetrahydro-pyran-4-ylmethyl)-piperidin-4-ylmethyl]-carbamoyl}-ethylcarbamoyl)-ciclopentyl]-amide 388891 6-methyl-benzo[b]thiophene-2-carboxylic acid [1-(2-phenyl-1(R)-{[1-(tetrahydro-pyran-4-ylmethyl)-piperidin-4-ylmethyl]-carbamoyl}-ethylcarbamoyl)-ciclopentyl]-amide 388893 6-cyano-benzo[b]thiophene-2-carboxylic acid [1-(2-phenyl-1(R)-{[1-(tetrahydro-pyran-4-ylmethyl)-piperidin-4-ylmethyl]-carbamoyl}-ethylcarbamoyl)-ciclopentyl]-amide 388895 6-dimethylamino-benzo[b]thiophene-2-carboxylic acid [1-(2-phenyl-1(R)-{[1-(tetrahydro-pyran-4-ylmethyl)-piperidin-4-ylmethyl]-carbamoyl}-ethylcarbamoyl)-ciclopentyl]-amide 389011 SID26753203 389153 3-[(1-isopropylpiperidin-3-yl)methyl]-2-(2-methylphenyl)-quinazolin-4(3H)-one 389156 3-[(1-ethylpiperidin-3-yl)methyl]-6-methoxy-2-(2-methoxyphenyl)quinazolin-4(3H)-one 389158 3-[(1-ethylpiperidin-3-yl)methyl]-2-(2-methylphenyl)-6-(trifluoromethoxy)quinazolin-4(3H)-one 389160 6-(4-fluorophenoxy)-2-(2-methylphenyl)-3-(piperidin-3-ylmethyl)quinazolin-4(3H)-one 389163 6-(4-fluorophenoxy)-3-[(1-isopropylpiperidin-3-yl)methyl]-2-(2-methylphenyl)quinazolin-4(3H)-one 389164 6-(4-chlorophenyl)-2-(2-methylphenyl)-3-(piperidin-3-ylmethyl)-quinazolin-4(3H)-one 389166 6-(4-chlorophenyl)-3-[(-1-ethylpiperidin-3-yl)methyl]-2-(2-methylphenyl)quinazolin-4(3H)-one 389171 6-(4-chlorophenyl)-3-{[(3S)-1-ethylpiperidin-3-yl]methyl}-2-(2-methylphenyl)quinazolin-4(3H)-one 389173 6-(4-chlorophenyl)-3-{[(3R)-1-ethylpiperidin-3-yl]methyl}-2-(2-methylphenyl)quinazolin-4(3H)-one 389180 6-(4-chlorophenyl)-3-[(1-isopropylpiperidin-3-yl)methyl]-2-(2-methylphenyl)quinazolin-4(3H)-one 389182 6-(4-chlorophenyl)-3-[(1-cyclobutylpiperidin-3-yl)methyl]-2-(2-methylphenyl)quinazolin-4(3H)-one 389184 6-(4-chlorophenyl)-3-{[1-(2-methoxyethyl)piperidin-3-yl]-methyl}-2-(2-methylphenyl)quinazolin-4(3H)-one 389185 6-(4-chlorophenyl)-3-{[1-(2-fluoroethyl)piperidin-3-yl]methyl}-2-(2-methylphenyl)quinazolin-4(3H)-one 389186 6-(4-chlorophenyl)-2-(2-methylphenyl)-3-{[1-(2,2,2-trifluoroethyl)piperidin-3-yl]methyl}quinazolin-4(3H)-one 389188 6-(4-chlorophenyl)-2-(2-methylphenyl)-3-{[1-(3,3,3-trifluoropropyl)piperidin-3-yl]methyl}quinazolin-4(3H)-one 389191 6-(4-chlorophenyl)-3-[(1-ethyl-1,2,5,6-tetrahydropyridin-3-yl)-methyl]-2-(2-methylphenyl)quinazolin-4(3H)-one 389194 6-(4-chlorophenyl)-3-[(4-isopropylmorpholin-2-yl)methyl]-2-(2-methylphenyl)quinazolin-4(3H)-one 389195 6-(4-fluorophenyl)-2-isopropyl-3-[(1-isopropylpiperidin-3-yl)-methyl]quinazolin-4(3H)-one 389199 6-(4-chlorophenyl)-2-isopropyl-3-{[(3S)-1-isopropylpiperidin-3-yl]methyl}quinazolin-4(3H)-one 389218 6-(4-chlorophenyl)-3-{[(3S)-1-isopropylpiperidin-3-yl]methyl}-2-methylquinazolin-4(3H)-one 389221 6-(4-chlorophenyl)-3-[(1-isopropylpiperidin-3-yl)methyl]-quinazolin-4(3H)-one 389232 (S)-6-(4-fluorophenoxy)-3-((1-isopropylpiperidin-3-yl)methyl)-2-o-tolylquinazolin-4(3H)-one 389235 6-(4-fluorophenoxy)-2-isopropyl-3-[(1-isopropylpiperidin-3-yl)methyl]quinazolin-4(3H)-one 389238 6-(4-fluorophenoxy)-3-{[(3S)-1-isopropylpiperidin-3-yl]methyl}-2-methylquinazolin-4(3H)-one 389252 6-(4-luorophenoxy)-3-{[(3S)-1-isopropylpiperidin-3-yl]-methyl}quinazolin-4(3H)-one 389347 methyl N-(5-(4-(phenylaminocarbonylamino)phenoxy)-1H-benzimidazol-2-yl)carbamate 389348 methyl N-(5-(4-((3-(trifluoromethyl)phenyl)aminocarbonylamino)phenoxy)-1H-benzimidazol-2-yl)carbamate 389349 methyl 5-(4-(3-(2-fluoro-5-(trifluoromethyl)phenyl)ureido)phenoxy)-1H-benzo[d]imidazol-2-ylcarbamate 389350 methyl N-(5-(4-((2-chloro-5-(trifluoromethyl)phenyl)aminocarbonylamino)phenoxy)-1H-benzimidazol-2-yl)carbamate 389352 methyl N-(5-(4-((3-ethylphenyl)aminocarbonylamino)phenoxy)-1H-benzimidazol-2-yl)carbamate 389353 methyl N-(5-(4-((3-bromophenyl)aminocarbonylamino)phenoxy)-1H-benzimidazol-2-yl)carbamate 389354 methyl N-(5-(4-((3-chlorophenyl)aminocarbonylamino)phenoxy)-1H-benzimidazol-2-yl)carbamate 389355 methyl N-(5-(4-((2,5-difluorophenyl)aminocarbonylamino)-phenoxy)-1H-benzimidazol-2-yl)carbamate 389356 methyl N-(5-(4-((3-(trifluoromethylthio)phenyl)aminocarbonylamino)phenoxy)-1H-benzimidazol-2-yl)carbamate 389357 methyl N-(5-(4-((3-methylthiophenyl)aminocarbonylamino)-phenoxy)-1H-benzimidazol-2-yl)carbamate 389358 methyl N-(5-(4-((2-fluoro-5-aminophenyl)aminocarbonylamino)phenoxy)-1H-benzimidazol-2-yl)carbamate 389359 methyl N-(5-(4-((3-carboxyphenyl)aminocarbonylamino)-phenoxy)-1H-benzimidazol-2-yl)carbamate 389360 methyl N-(5-(4-((3-(trifluoromethyl)phenyl)aminothiocarbonylamino)phenoxy)-1H-benzimidazol-2-yl)carbamate 389363 methyl (5-(4-((2-(3-trifluoromethyl)phenyl)acetylamido)-phenoxy)-1H-benzoimidazol-2-yl)carbamate 389364 methyl (6-(4-(2-(2-fluoro-5-(trifluoromethyl)phenylamino)-2-oxoethyl)phenoxy)-1H-benzoimidazol-2-yl)carbamate 389365 methyl N-(5-(3-((2-fluoro-5-(trifluoromethyl)phenyl)aminocarbonylamino)phenoxy)-1H-benzimidazol-2-yl)carbamate 389367 methyl N-(5-(5-((2-fluoro-5-(trifluoromethyl)phenyl)aminocarbonylamino)-2-pyridyloxy)-1H-benzimidazol-2-yl)carbamate 389368 methyl N-(5-(5-((2-fluoro-5-(trifluoromethyl)phenyl)aminocarbonylamino)-1-oxo-2-pyridyloxy)-1H-benzimidazol-2-yl)-carbamate 389369 N-(5-(2-((2-fluoro-5-(trifluoromethyl)phenyl)aminocarbonylamino)-5-pyridyloxy)-1H-benzimidazol-2-yl)acetamide 389370 methyl N-(5-(4-((2-fluoro-5-(trifluoromethyl)phenyl)aminocarbonylamino)phenylthio)-1H-benzimidazol-2-yl)carbamate 389371 methyl N-(5-(4-((2-fluoro-5-(trifluoromethyl)phenyl)aminocarbonylamino)phenylsulfinyl)-1H-benzimidazol-2-yl)carbamate 389373 methyl N-(5-(4-((2-fluoro-5-(trifluoromethyl)phenyl)aminocarbonylamino)phenylsulfonyl)-1H-benzimidazol-2-yl)carbamate 389374 methyl N-(5-(4-((2-fluoro-5-(trifluoromethyl)phenyl)aminocarbonylamino)phenylcarbonyl)-1H-benzimidazol-2-yl)carbamate 389375 (1R,3aR,4aS,8aS,9S,9aS)-decahydro-1-methyl-9-[(1E)-2-[5-[3-(trifluoromethyl)phenyl]-2-pyridinyl]ethenyl]-3H-thiopyrano-[3,4-f]isobenzofuran-3-one 389376 (1R,3aR,4aS,8aS,9S,9aS)-decahydro-1-methyl-9-[(1E)-2-[5-[3-(trifluoromethyl)phenyl]-2-pyridinyl]ethenyl]-3H-thiopyrano-[3,4-f]isobenzofuran-3-one-6,6-dioxide 389377 methyl N-(6-(4-((2-fluoro-5-(trifluoromethyl)phenyl)aminocarbonylamino)phenoxy)-1-methyl-1H-benzimidazol-2-yl)-carbamate 389378 methyl N-(5-(4-((2-fluoro-5-(trifluoromethyl)phenyl)aminocarbonylamino)phenoxy)-1-methyl-1H-benzimidazol-2-yl)-carbamate 389380 methyl N-(6-(4-((2-fluoro-5-(trifluoromethyl)phenyl)aminocarbonylamino)phenoxy)-benzthiazol-2-yl)carbamate 389381 (1R,3aR,4aS,8aS,9S,9aS)-decahydro-1-methyl-9-[(1E)-2-[5-[3-(trifluoromethyl)phenyl]-2-pyridinyl]ethenyl]-3H-thiopyrano[3,4-f]isobenzofuran-3-one-6-oxide 389382 (1R,3aR,4aS,8aS,9S,9aS)-decahydro-1-methyl-9-[(e)-2-[5-[3-(trifluoromethyl)phenyl]-2-pyridinyl]ethenyl]-3H-furo[3,4-g][2]-benzopyran-3-one 389383 (1R,3aR,4aS,8aS,9S,9aS)-9-[(E)-2-[5-(3-fluorophenyl)-2-pyridinyl]ethenyl]-decahydro-1-methyl-3H-furo[3,4-g][2]benzopyran-3-one 389384 methyl N-(6-(4-((2-fluoro-5-(trifluoromethyl)phenyl)aminocarbonylamino)phenoxy) benzoxazol-2-yl)carbamate 389385 methyl N-(5-(4-((2-fluoro-5-(trifluoromethyl)phenyl)aminocarbonylamino)phenoxy)-3a-aza-2-indolyl)carbamate 389386 methyl N-(5-(4-((2-fluoro-5-(trifluoromethyl)phenyl)aminocarbonylamino)phenoxy)-3,4-diazaindole-2-yl)carbamate 389387 (1R,3aR,4aS,8aS,9S,9aS)-9-[(E)-2-[5-(2-fluorophenyl)-2-pyridinyl]ethenyl]-decahydro-1-methyl-3H-furo[3,4-g][2]benzopyran-3-one 389388 (1R,3aR,4aS,8aS,9S,9aS)-9-[(E)-2-[5-(2,3-difluorophenyl)-2-pyridinyl]ethenyl]-decahydro-1-methyl-3H-furo[3,4-g][2]-benzopyran-3-one 389389 (1R,3aR,4aS,8aS,9S,9aS)-9-[(E)-2-[5-(3-chlorophenyl)-2-pyridinyl]ethenyl]-decahydro-1-methyl-3H-furo[3,4-g][2]benzopyran-3-one 389390 methyl N-(6-(4-((2-fluoro-5-(trifluoromethyl)phenyl)aminocarbonylamino)phenoxy)-3,4-diaza-1H-indole-2-yl)carbamate 389391 (1R,3aR,4aS,8aS,9S,9aS)-9-[(E)-2-[5-(2-chlorophenyl)-2-pyridinyl]ethenyl]-decahydro-1-methyl-3H-furo[3,4-g][2]benzopyran-3-one 389392 (1R,3aR,4aS,8aS,9S,9aS)-9-[(E)-2-[5-(2,3-dichlorophenyl)-2-pyridinyl]ethenyl]-decahydro-1-methyl-3H-furo[3,4-g][2]-benzopyran-3-one 389393 (1R,3aR,4aS,8aS,9S,9aS)-decahydro-1-methyl-3-oxo-9-[(1E)-2-[5-[3-(trifluoromethyl)phenyl]-2-pyridinyl]ethenyl]-furo[3,4-g]isoquinoline-6(3H)-carboxylic acid ethyl ester 389394 2-amino-5-(4-((2-fluoro-5-(trifluoromethyl)phenyl)aminocarbonylamino)phenoxy)-1H-benzimidazole 389395 ethyl (4aS,5S,5aS,6R,8aR,9aS)-5-[(E)-2-[5-(3-fluorophenyl)-2-pyridinyl]ethenyl]-decahydro-6-methyl-8-oxofuro[3,4-g]quinoline-1(2H)-carboxylate 389396 ethyl (4aS,5S,5aS,6R,8aR,9aS)-5-[(E)-2-[5-(2-fluorophenyl)-2-pyridinyl]ethenyl]-decahydro-6-methyl-8-oxofuro[3,4-g]quinoline-1(2H)-carboxylate 389397 ethyl (4aS,5S,5aS,6R,8aR,9aS)-5-[(E)-2-[5-(2-methylphenyl)-2-pyridinyl]ethenyl]-decahydro-6-methyl-8-oxofuro[3,4-g]quinoline-1(2H)-carboxylate 389398 N-(5-(4-((2-fluoro-5-(trifluoromethyl)-phenyl)aminocarbonylamino)phenoxy)-1H-benzimidazol-2-yl)-acetamide 389400 ethyl (4aS,5S,5aS,6R,8aR,9aS)-5-[(E)-2-[5-(3-cyanophenyl)-2-pyridinyl]ethenyl]-decahydro-6-methyl-8-oxofuro[3,4-g]quinoline-1(2H)-carboxylate 389401 N-(5-(4-((2-fluoro-5-(trifluoromethyl)phenyl)aminocarbonylamino)phenoxy)-1H-benzimidazol-2-yl)benzamide 389403 N-(6-(4-((2-fluoro-5(trifluoromethyl)phenyl)aminocarbonylamino)phenoxy)-1H-benzimidazol-2-yl)-2-(1H-pyrrol-1-yl)benzamide 389404 (1R,3aR,4aS,8aS,9S,9aS)-decahydro-1-methyl-3-oxo-9-[(1E)-2-[5-(3-fluorophenyl)-2-pyridinyl]ethenyl]-furo[3,4-g]isoquinoline-6(3H)-carboxylic acid ethyl ester 389405 (1R,3aR,4aS,8aS,9S,9aS)-ethyl decahydro-1-methyl-3-oxo-9-[(e)-2-[5-(2-fluorophenyl)-2-pyridinyl]ethenyl]furo[3,4-g]isoquinoline-6(3H)-carboxylate 389406 N-(5-(4-((2-fluoro-5-(trifluoromethyl)phenyl)aminocarbonylamino)phenoxy)-1H-benzimidazol-2-yl)-2-furylcarboxamide 389407 (1R,3aR,4aS,8aS,9S,9aS)-ethyl 9-[(e)-2-[[2,3'-bipyridin]-6'-yl]-ethenyl]-decahydro-1-methyl-3-oxofuro[3,4-g]isoquinoline-6(3H)-carboxylate 389408 N-(5-(4-((2-fluoro-5-(trifluoromethyl)phenyl)aminocarbonylamino)phenoxy)-1H-benzimidazol-2-yl)-3-pyridinecarboxamide 389409 (1R,3aR,4aS,8aS,9S,9aS)-decahydro-1-methyl-9-[(e)-2-[5-[3-(trifluoromethyl)phenyl]-2-pyridinyl]ethenyl]furo[3,4-g]isoquinolin-3(1H)-one 389410 (1R,3aR,4aS,8aS,9S,9aS)-decahydro-6-methyl-1-methyl-9-[(e)-2-[5-[3-(trifluoromethyl)phenyl]-2-pyridinyl]ethenyl]furo-[3,4-g]isoquinolin-3(1H)-one 389411 N-(5-(4-((2-fluoro-5-(trifluoromethyl)phenyl)aminocarbonylamino)phenoxy)-1H-benzimidazol-2-yl)-2-(2-methoxyethoxy)-acetamide 389412 (1R,3aR,4aS,8aS,9S,9aS)-6-acetyl-decahydro-1-methyl-9-[(e)-2-[5-[3-(trifluoromethyl)phenyl]-2-pyridinyl]ethenyl]furo[3,4-g]-isoquinolin-3(1H)-one 389413 (1R,3aR,4aS,8aS,9S,9aS)-decahydro-1-methyl-6-(2-methyl-1-oxopropyl)-9-[(e)-2-[5-[3-(trifluoromethyl)phenyl]-2-pyridinyl]-ethenyl]furo[3,4-g]isoquinolin-3(1H)-one 389414 (1R,3aR,4aS,8aS,9S,9aS)-6-(cyclopropylcarbonyl)-decahydro-1-methyl-9-[(e)-2-[5-[3-(trifluoromethyl)phenyl]-2-pyridinyl]-ethenyl]furo[3,4-g]isoquinolin-3(1H)-one 389415 (1R,3aR,4aS,8aS,9S,9aS)-6-(cyclopropylcarbonyl)-9-[(e)-2-[5-(3-fluorophenyl)-2-pyridinyl]ethenyl]-decahydro-1-methylfuro-[3,4-g]isoquinolin-3(1H)-one 389416 1R,3aR,4aS,8aS,9S,9aS)-6-(cyclopropylcarbonyl)-9-[(e)-2-[5-(2-fluorophenyl)-2-pyridinyl]ethenyl]-decahydro-1-methylfuro-[3,4-g]isoquinolin-3(1H)-one 389417 (1R,3aR,4aS,8aS,9S,9aS)-dodecahydro-1-methyl-3-oxo-9-[(e)-2-[5-(3-fluorophenyl)-2-pyridinyl]ethenyl]furo[3,4-g]isoquinoline-6-carboxamide 389419 N-(5-(4-((2-fluoro-5-(trifluoromethyl)phenyl)aminocarbonylamino)phenoxy)-1H-benzimidazol-2-yl)-2-(4-methylpiperazin-1-yl)acetamide 389420 2-(2-(4-methyl-1-piperazino)ethylamino)-5-(4-((2-fluoro-5-(trifluoromethyl)phenyl)aminocarbonylamino)phenoxy)-1Hbenzimidazole 389421 (1R,3aR,4aS,8aS,9S,9aS)-N-ethyl-dodecahydro-1-methyl-3-oxo-9-[(e)-2-[5-(3-fluorophenyl)-2-pyridinyl]ethenyl]furo[3,4-g]-isoquinoline-6-carboxamide 389423 N-(6-(4-((2-fluoro-5-(trifluoromethyl)phenyl)aminocarbonylamino)phenoxy)benzthiazol-2-yl)methanesulfonamide 389426 HO-LVA 389427 (1R,3aR,4aS,8aS,9S,9aS)-9-[(E)-2-[5-(3-fluorophenyl)-2-pyridinyl]ethenyl]-decahydro-1-methyl-6-(methylsulfonyl)furo[3,4-g]isoquinolin-3(1H)-one 389428 (1R,3aR,4aS,8aS,9S,9aS)-9-[(E)-2-[5-(3-fluorophenyl)-2-pyridinyl]ethenyl]-decahydro-1-methyl-6-(propylsulfonyl)furo[3,4-g]isoquinolin-3(1H)-one 389429 (1R,3aR,4aS,8aS,9S,9aS)-phenylmethyl decahydro-1-methyl-3-oxo-9-[(e)-2-[5-[3-(trifluoromethyl)phenyl]-2-pyridinyl] ethenyl]furo[3,4-g]isoquinoline-6(3H)-carboxylate 389430 (1R,3aR,4aS,8aS,9S,9aS)-2-methoxyethyl 9-[(e)-2-[5-(3-fluorophenyl)-2-pyridinyl]ethenyl]-decahydro-1-methyl-3-oxo-furo-[3,4-g]isoquinoline-6(3H)-carboxylate 389499 6-(butyl(methyl)amino)-3-((1-ethylpiperidin-3-yl)methyl)-2-(2-methoxyphenyl)quinazolin-4(3H)-one 389500 6-(butyl(methyl)amino)-2-(2-methoxyphenyl)-3-(piperidin-3-ylmethyl)quinazolin-4(3H)-one 389956 trans-3-(2-(4-((3-(3-(5-methyl-1,2,4-oxadiazolyl))phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro-1H-3-benzazepine 389958 7-(5-methyl-1,3-oxazol-2-yl)-3-(3-{[4-methyl-5-(2-thienyl)-4H-1,2,4-triazol-3-yl]thio}propyl)-2,3,4,5-tetrahydro-1H-3-benzazepine 389959 3-(3-{[5-(1H-indol-2-yl)-4-methyl-4H-1,2,4-triazol-3-yl]thio}-propyl)-7-(5-methyl-1,3-oxazol-2-yl)-2,3,4,5-tetrahydro-1H-3-benzazepine 389960 3-(3-{[5-(1H-indol-5-yl)-4-methyl-4H-1,2,4-triazol-3-yl]thio}-propyl)-7-(5-methyl-1,3-oxazol-2-yl)-2,3,4,5-tetrahydro-1H-3-benzazepine 389961 3-(3-{[4-methyl-5-(1-methyl-1H-pyrrol-2-yl)-4H-1,2,4-triazol-3-yl]thio}propyl)-7-(5-methyl-1,3-oxazol-2-yl)-2,3,4,5-tetrahydro-1H-3-benzazepine 389962 7-(5-methyl-3-isoxazolyl)-3-(3-{[4-methyl-5-(2-methyl-5-quinolinyl)-4H-1,2,4-triazol-3-yl]thio}propyl)-2,3,4,5-tetrahydro-1H-3-benzazepine 389963 7-(5-methyl-3-isoxazolyl)-3-(3-{[4-methyl-5-(2-methyl-6-quinolinyl)-4H-1,2,4-triazol-3-yl]thio}propyl)-2,3,4,5-tetrahydro-1H-3-benzazepine 389964 3-(3-{[5-(2,3-dimethyl-6-quinoxalinyl)-4-methyl-4H-1,2,4-triazol-3-yl]thio}propyl)-7-(5-methyl-3-isoxazolyl)-2,3,4,5-tetrahydro-1H-3-benzazepine 389965 7-(5-methyl-3-isoxazolyl)-3-{3-[(4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio]propyl}-2,3,4,5-tetrahydro-1H-3-benzazepine 389966 4-[4-methyl-5-({3-[7-(5-methyl-3-isoxazolyl)-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]propyl}thio)-4H-1,2,4-triazol-3-yl]-benzonitrile 389967 7-(5-methyl-3-isoxazolyl)-3-[3-({4-methyl-5-[4-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}thio)propyl]-2,3,4,5-tetrahydro-1H-3-benzazepine 389968 7-(5-methyl-3-isoxazolyl)-3-(3-{[4-methyl-5-(4-methylphenyl)-4H-1,2,4-triazol-3-yl]thio}propyl)-2,3,4,5-tetrahydro-1H-3-benzazepine 389970 7-(5-methyl-3-isoxazolyl)-3-(3-{[4-methyl-5-(4-pyridinyl)-4H-1,2,4-triazol-3-yl]thio}propyl)-2,3,4,5-tetrahydro-1H-3-benzazepine 389971 7-(5-methyl-3-isoxazolyl)-3-(3-{[4-methyl-5-(2-thienyl)-4H-1,2,4-triazol-3-yl]thio}propyl)-2,3,4,5-tetrahydro-1H-3-benzazepine 389973 3-(3-{[5-(2-chlorophenyl)-4-methyl-4H-1,2,4-triazol-3-yl]thio}-propyl)-7-(5-methyl-3-isoxazolyl)-2,3,4,5-tetrahydro-1H-3-benzazepine 389974 3-(3-{[5-(3-chlorophenyl)-4-methyl-4H-1,2,4-triazol-3-yl]thio}-propyl)-7-(5-methyl-3-isoxazolyl)-2,3,4,5-tetrahydro-1H-3-benzazepine 389975 3-(3-{[5-(4-chlorophenyl)-4-methyl-4H-1,2,4-triazol-3-yl]thio}-propyl)-7-(5-methyl-3-isoxazolyl)-2,3,4,5-tetrahydro-1H-3-benzazepine 389976 3-(3-{[5-(3,4-dichlorophenyl)-4-methyl-4H-1,2,4-triazol-3-yl]-thio}propyl)-7-(5-methyl-3-isoxazolyl)-2,3,4,5-tetrahydro-1H-3-benzazepine 389977 3-(3-{[5-(3-fluorophenyl)-4-methyl-4H-1,2,4-triazol-3-yl]thio}-propyl)-7-(5-methyl-3-isoxazolyl)-2,3,4,5-tetrahydro-1H-3-benzazepine 389980 7-(5-methyl-3-isoxazolyl)-3-(3-{[4-methyl-5-(trifluoromethyl)-4H-1,2,4-triazol-3-yl]thio}propyl)-2,3,4,5-tetrahydro-1H-3-benzazepine 389981 7-(5-methyl-3-isoxazolyl)-3-(3-{[4-methyl-5-(1-methylethyl)-4H-1,2,4-triazol-3-yl]thio}propyl)-2,3,4,5-tetrahydro-1H-3-benzazepine 389982 3-(3-{[5-(1,1-dimethylethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-thio}propyl)-7-(5-methyl-3-isoxazolyl)-2,3,4,5-tetrahydro-1H-3-benzazepine 390001 3-{3-[(5-cyclopentyl-4-methyl-4H-1,2,4-triazol-3-yl)thio]propyl}-7-(5-methyl-3-isoxazolyl)-2,3,4,5-tetrahydro-1H-3-benzazepine 390002 7-(5-methyl-3-isoxazolyl)-3-(3-{[4-methyl-5-(4-methylcyclohexyl)-4H-1,2,4-triazol-3-yl]thio}propyl)-2,3,4,5-tetrahydro-1H-3-benzazepine 390003 7-(5-methyl-3-isoxazolyl)-3-(3-{[4-methyl-5-(tetrahydro-2Hpyran-4-yl)-4H-1,2,4-triazol-3-yl]thio}propyl)-2,3,4,5-tetrahydro-1H-3-benzazepine 390004 7-(5-methyl-3-isoxazolyl)-3-[3-({4-methyl-5-[2-(methyloxy)-phenyl]-4H-1,2,4-triazol-3-yl}thio)propyl]-2,3,4,5-tetrahydro-1H-3-benzazepine 390005 7-(5-methyl-3-isoxazolyl)-3-[3-({4-methyl-5-[3-(methyloxy)-phenyl]-4H-1,2,4-triazol-3-yl}thio)propyl]-2,3,4,5-tetrahydro-1H-3-benzazepine 390006 7-(5-methyl-3-isoxazolyl)-3-[3-({4-methyl-5-[4-(methyloxy)-phenyl]-4H-1,2,4-triazol-3-yl}thio)propyl]-2,3,4,5-tetrahydro-1H-3-benzazepine 390007 7-(5-methyl-3-isoxazolyl)-3-[3-({4-methyl-5-[6-(methyloxy)-3-pyridinyl]-4H-1,2,4-triazol-3-yl}thio)propyl]-2,3,4,5-tetrahydro-1H-3-benzazepine 390008 7-(1,3-dimethyl-1H-pyrazol-5-yl)-3-(3-{[4-methyl-5-(2-methyl-5-quinolinyl)-4H-1,2,4-triazol-3-yl]thio}propyl)-2,3,4,5-tetrahydro-1H-3-benzazepine 390010 7-(1,3-dimethyl-1H-pyrazol-5-yl)-3-[3-({4-methyl-5-[4-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}thio)propyl]-2,3,4,5-tetrahydro-1H-3-benzazepine 390101 N-(2,3-dihydro-1H-pyrrolo[3,2,1-ij]-quinolin-6-ethyl)acetamide 390104 N-(2,3-dihydro-1H-pyrrolo-[3,2,1-ij]quinolin-6-ethyl)propionamide 390106 N-(2,3-dihydro-1H-pyrrolo-[3,2,1-ij]quinolin-6-ethyl)butyramide 390108 N-cyclopropanecarboxamido (2,3-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-6-yl)ethanamine 390112 N-[3-[2,3-dihydro-1H-pyrrolo-[3,2,1-ij]quinolin-6-propyl]acetamide 390114 N-[3-[2,3-dihydro-1H-pyrrolo-[3,2,1-ij]quinolin-6-propyl]propionamide 390116 N-[3-[2,3-dihydro-1H-pyrrolo-[3,2,1-ij]quinolin-6-propyl]butyramide 390119 N-cyclopropanecarboxamido-3-(2,3-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-6-yl)-propylamine 390121 N-cyclobutanecarboxamido-3-(2,3-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-6-yl)-propylamine 390124 N-[2-methyl-2-(2,3-dihydro-1Hpyrrolo[3,2,1-ij]quinolin-6-yl)propyl]acetamide 390125 N-[1-(2,3-dihydro-1H-pyrrolo-[3,2,1-ij]quinolin-6-yl)cyclohexanemethyl]acetamide 390126 N-[1-(2,3-dihydro-1H-pyrrolo-[3,2,1-ij]quinolin-6-yl)cyclohexanemethyl]-butyramide 390342 (R)-1-(bis(4-fluorophenyl)methyl)-4-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)piperazine 390347 (S)-1-(bis(4-fluorophenyl)methyl)-4-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)piperazine 390349 (R)-1-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)-4-(2-ethoxyphenyl)piperazine 390350 (S)-1-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)-4-(2-ethoxyphenyl)piperazine 390519 6-benzyl-8-butyl-6,8-diaza-bicyclo[3.2.2]nonan-2-ol 390521 (1R,2S,5S)-6-Benzyl-8-(2-phenylethyl)-6,8-diazabidiazabicyclo 390522 (1R,2R,5S)-6-benzyl-8-(2-phenylethyl)-6,8-diazabicyclo[3.2.2]nonan-2-ol 390523 (1R,2R,5S)-6-benzyl-2-methoxy-8-methyl-6,8-diazabicyclo[3.2.2]nonane 390525 6-benzyl-8-butyl-2-methoxy-6,8-diaza-bicyclo[3.2.2]nonane 390527 6-benzyl-2-methoxy-8-phenethyl-6,8-diaza-bicyclo[3.2.2]nonane 390531 (1R,2R,5S)-6-benzyl-2-benzyloxy-8-methyl-6,8-diazabicyclo[3.2.2]nonane 390534 6-benzyl-2-(benzyloxy)-8-butyl-6,8-diaza-bicyclo[3.2.2]nonane 390536 6-benzyl-2-(benzyloxy)-8-phenethyl-6,8-diaza-bicyclo[3.2.2]nonane 390557 N alpha-amidino-Tyr(Me)-Pro-Trp-p-Cl-Phe-NH2 390558 N alpha-amidino-Tyr(Me)-Pro-Trp-Phe-NH2 390559 N alpha-amidino-Tyr(Me)-D-Pro-Gly-Trp-p-Cl-Phe-NH2 390560 N alpha-amidino-Tyr(Me)-D-Pro-Gly-Trp-Phe-NH2 390883 benzyl 2-(2-methyl-1,3-dioxolan-2-yl)-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)acetate 390885 benzyl 2-((3S,4R)-3-(1,3-dioxoisoindolin-2-yl)-2-oxo-4-((E)-styryl)azetidin-1-yl)-2-(2-methyl-1,3-dioxolan-2-yl)acetate 390896 benzyl 2-((2R,3S)-2-((E)-2-(furan-2-yl)vinyl)-4-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)azetidin-1-yl)-4,4-dimethyl-3-oxopentanoate 390899 benzyl 4,4-dimethyl-3-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)pentanoate 390900 benzyl 3-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)-3-phenylpropanoate 390901 benzyl 2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)acetate 390902 benzyl 3-hydroxy-4,4-dimethyl-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)pentanoate 390903 (S)-benzyl 4-methyl-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)pentanoate 390905 2-(trimethylsilyl)ethyl 2-(2-methyl-1,3-dioxolan-2-yl)-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)acetate 390907 N-benzyl-2-(2-methyl-1,3-dioxolan-2-yl)-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)acetamide 390908 (S)-3-((3S,4R)-1-((S)-4-methyl-1-oxo-1-(4-(2-(piperidin-1-yl)ethyl)piperidin-1-yl)pentan-2-yl)-2-oxo-4-((E)-styryl)azetidin-3-yl)-4-phenyloxazolidin-2-one 390909 (S)-3-((3S,4R)-1-((S)-4-methyl-1-oxo-1-(4-(piperidin-1-yl)piperidin-1-yl)pentan-2-yl)-2-oxo-4-((E)-styryl)azetidin-3-yl)-4-phenyloxazolidin-2-one 390910 (S)-N-benzyl-4-methyl-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)pentanamide 390911 (S)-N-(2-chlorobenzyl)-4-methyl-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)pentanamide 390912 (S)-N-(3-chlorobenzyl)-4-methyl-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)pentanamide 390913 (S)-N-(3-(trifluoromethyl)benzyl)-4-methyl-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)pentanamide 390914 (S)-N-(4-chlorobenzyl)-4-methyl-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)pentanamide 390915 (S)-3-((3S,4R)-1-(4,4-dimethyl-1,3-dioxo-1-(4-(2-(piperidin-1-yl)ethyl)piperidin-1-yl)pentan-2-yl)-2-oxo-4-((E)-styryl)azetidin-3-yl)-4-phenyloxazolidin-2-one 390986 N-(3-(trifluoromethyl)benzyl)-3-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)-3-(4-(2-(piperidin-1-yl)ethyl)piperidin-1-yl)propanamide 390987 N-(3-(trifluoromethyl)benzyl)-3-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)-3-(4-(piperidin-1-yl)piperidin-1-yl)propanamide 390989 4-amino-1-benzyl-1-{2-[(3S,4R)-2-oxo-3-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]-4-[(E)-2-phenylethenyl]azetidin-1-yl]-2-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)acetyl}piperidin-1-ium 390991 N-(3-(trifluoromethyl)benzyl)-3-(4-isopropylpiperazin-1-yl)-3-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)propanamide 390992 N-(3-(trifluoromethyl)benzyl)-3-(4-cyclohexylpiperazin-1-yl)-3-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)propanamide 390993 N-(3-(trifluoromethyl)benzyl)-3-(2-(2-aminoethyl)piperidin-1-yl)-3-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)propanamide 390994 4-amino-1-benzyl-1-[(3S)-3-[(3S,4R)-2-oxo-3-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]-4-[(E)-2-phenylethenyl]azetidin-1-yl]-3-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)propanoyl]piperidin-1-ium 390995 (S)-N-(3-(trifluoromethyl)benzyl)-4-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)-4-(4-(piperidin-1-yl)piperidin-1-yl)butanamide 390996 (3S)-3-amino-1-benzyl-1-[(3S)-3-[(3S,4R)-2-oxo-3-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]-4-[(E)-2-phenylethenyl]azetidin-1-yl]-3-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)propanoyl]pyrrolidin-1-ium 390997 (S)-N-(3-(trifluoromethyl)benzyl)-4-(4-benzyl-1,4-diazepan-1-yl)-4-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)butanamide 390998 (S)-N-(3-(trifluoromethyl)benzyl)-4-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)-4-(4-(2-(piperidin-1-yl)ethyl)piperidin-1-yl)butanamide 390999 (S)-N-(3-(trifluoromethyl)benzyl)-4-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)-4-(4-(pyrrolidin-1-yl)piperazin-1-yl)butanamide 391000 (S)-N-(3-(trifluoromethyl)benzyl)-4-(4-cyclohexylpiperazin-1-yl)-4-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)butanamide 391005 (S)-N-(3-(trifluoromethyl)benzyl)-4-oxo-3-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)-4-(4-phenethylpiperazin-1-yl)butanamide 391011 2(R)-[[4-(piperidin-1-yl)piperidin-1-yl]carbonylmethyl]-2-[3(S)-(4(S)-phenyloxazolidin-2-on-3-yl)-4(R)-(2-styryl)azetidin-2-on-1-yl]acetic acid N-(3-trifluoromethylbenzyl)amide 391012 (R)-N-(3-(trifluoromethyl)benzyl)-4-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)-4-(4-(piperidin-1-ylmethyl)piperidin-1-yl)butanamide 391014 4-amino-1-benzyl-1-[(3R)-3-[(3S,4R)-2-oxo-3-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]-4-[(E)-2-phenylethenyl]azetidin-1-yl]-3-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)propanoyl]piperidin-1-ium 391015 (R)-N-(3-(trifluoromethyl)benzyl)-4-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)-4-(4-(2-(piperidin-1-yl)ethyl)piperidin-1-yl)butanamide 391017 (R)-N-(3-(trifluoromethyl)benzyl)-4-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)-4-(4-(pyrrolidin-1-yl)piperazin-1-yl)butanamide 391021 (S)-N-(3-(trifluoromethyl)benzyl)-5-(4-cyclohexylpiperazin-1-yl)-5-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)pentanamide 391023 (S)-N-(3-(trifluoromethyl)benzyl)-5-(4-(cyclohexylmethyl)piperazin-1-yl)-5-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)pentanamide 391025 (S)-N-(3-(trifluoromethyl)benzyl)-5-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)-5-(4-phenethylpiperazin-1-yl)pentanamide 391027 (S)-N-(3-(trifluoromethyl)benzyl)-5-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)-5-(4-(piperidin-1-yl)piperidin-1-yl)pentanamide 391034 (S)-N-(3-(trifluoromethyl)benzyl)-5-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)-5-(4-propylpiperazin-1-yl)pentanamide 391036 (S)-N-(3-(trifluoromethyl)benzyl)-5-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)-5-(4-(piperidin-1-ylmethyl)piperidin-1-yl)pentanamide 391038 (S)-N1-(3-(trifluoromethyl)benzyl)-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)-N5-(2-(piperidin-1-yl)ethyl)pentanediamide 391040 (S)-N-(3-(trifluoromethyl)benzyl)-5-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)-5-(4-(2-(piperidin-1-yl)ethyl)piperidin-1-yl)pentanamide 391042 (S)-N-(2-fluoro-3-(trifluoromethyl)benzyl)-5-(4-cyclohexylpiperazin-1-yl)-5-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)pentanamide 391043 (S)-N-(2,3-dichlorobenzyl)-5-(4-cyclohexylpiperazin-1-yl)-5-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)pentanamide 391045 (S)-N-(2-fluoro-5-(trifluoromethyl)benzyl)-5-(4-cyclohexylpiperazin-1-yl)-5-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)pentanamide 391046 (S)-N-(3-fluoro-5-(trifluoromethyl)benzyl)-5-(4-cyclohexylpiperazin-1-yl)-5-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)pentanamide 391047 (S)-N-(3-chlorobenzyl)-5-(4-cyclohexylpiperazin-1-yl)-5-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)pentanamide 391048 (S)-N-(3,5-difluorobenzyl)-5-(4-cyclohexylpiperazin-1-yl)-5-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)pentanamide 391049 (S)-N-(2-(trifluoromethyl)benzyl)-5-(4-cyclohexylpiperazin-1-yl)-5-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)pentanamide 391050 (S)-N-(3,5-bis(trifluoromethyl)benzyl)-5-(4-cyclohexylpiperazin-1-yl)-5-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)pentanamide 391052 (R)-N-(3-(trifluoromethyl)benzyl)-5-(4-cyclohexylpiperazin-1-yl)-5-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)pentanamide 391053 (R)-N-(3-(trifluoromethyl)benzyl)-5-(4-butylpiperazin-1-yl)-5-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)pentanamide 391054 (R)-N-(3-(trifluoromethyl)benzyl)-5-(4-isopropylpiperazin-1-yl)-5-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)pentanamide 391055 (R)-N-(3-(trifluoromethyl)benzyl)-5-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)-5-(4-phenethylpiperazin-1-yl)pentanamide 391057 (R)-N-(3-(trifluoromethyl)benzyl)-5-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)-5-(4-(piperidin-1-yl)piperidin-1-yl)pentanamide 391059 2(R)-[[4-(piperidin-1-yl)piperidin-1-yl]carbonylmethyl]-2-[3(S)-(4(S)-phenyloxazolidin-2-on-3-yl)-4(R)-(2-styryl)azetidin-2-on-1-yl]acetic acid N-[(R)-alpha-methylbenzyl]amide 391060 2(R)-[[4-(piperidin-1-yl)piperidin-1-yl]carbonylmethyl]-2-[3(S)-(4(S)-phenyloxazolidin-2-on-3-yl)-4(R)-(2-styryl)azetidin-2-on-1-yl]acetic acid N-methyl-N-(3-trifluoromethylbenzyl)amide 391061 2(R)-[[4-(piperidin-1-yl)piperidin-1-yl]carbonylmethyl]-2-[3(S)-(4(S)-phenyloxazolidin-2-on-3-yl)-4(R)-(2-styryl)azetidin-2-on-1-yl]acetic acid N-[(R)-alpha-methyl-3-trifluoromethylbenzyl]amide 391068 N-(3-(trifluoromethyl)benzyl)-3-(4-butylpiperazin-1-yl)-3-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)propanamide 391084 2(R)-[[4-(piperidin-1-yl)piperidin-1-yl]carbonylmethyl]-2-[3(S)-(4(S)-phenyloxazolidin-2-on-3-yl)-4(R)-(2-styryl)azetidin-2-on-1-yl]acetic acid N-(2-fluoro-3-tri-fluoromethylbenzyl)amide 391085 2(R)-[[4-[2-(1-piperidinyl)ethyl]piperidin-1-yl]carbonylmethyl]-2-[3(S)-(4(S)-phenyloxazolidin-2-on-3-yl)-4(R)-(2-styryl)azetidin-2-on-1-yl]acetic acid N-[(R)-alpha-methylbenzyl]amide 391097 2(R)-[[4-[2-(1-piperidinyl)ethyl]piperidin-1-yl]carbonylmethyl]-2-[3(S)-(4(S)-phenyloxazolidin-2-on-3-yl)-4(R)-(2-styryl)azetidin-2-on-1-yl]acetic acid N-[(S)-alpha-methylbenzyl]amide 391283 (S)-6-(4-chlorophenyl)-3-((1-ethylpiperidin-3-yl)methyl)-2-(4-(trifluoromethyl)phenyl)quinazolin-4(3H)-one 391284 (R)-6-(4-chlorophenyl)-3-((1-ethylpiperidin-3-yl)methyl)-2-(4-(trifluoromethyl)phenyl)quinazolin-4(3H)-one 391288 (R)-6-(4-fluorophenoxy)-3-((1-isopropylpiperidin-3-yl)methyl)-2-o-tolylquinazolin-4(3H)-one 391290 (S)-3-((1-ethylpiperidin-3-yl)methyl)-2-o-tolyl-6-(trifluoromethoxy)quinazolin-4(3H)-one 391291 (R)-3-((1-ethylpiperidin-3-yl)methyl)-2-o-tolyl-6-(trifluoromethoxy)quinazolin-4(3H)-one 391294 6-(2-chlorophenyl)-2-isopropyl-3-(((S)-1-isopropylpiperidin-3-yl)methyl)quinazolin-4(3H)-one 391297 6-(2-chlorophenyl)-2-isopropyl-3-(((R)-1-isopropylpiperidin-3-yl)methyl)quinazolin-4(3H)-one 391304 (S)-3-((1-ethylpiperidin-3-yl)methyl)-6-(4-fluorophenyl)-2-isopropylquinazolin-4(3H)-one 391307 (R)-3-((1-ethylpiperidin-3-yl)methyl)-6-(4-fluorophenyl)-2-isopropylquinazolin-4(3H)-one 391418 6,6'-(4,4'-(ethane-1,2-diyl)bis(piperidine-4,1-diyl))bis(N-(2-methoxybenzyl)hexan-1-amine) 391596 (+)-2-[(4aS,8aR)-4-(5-bromo-2-furoyl)octahydroquinoxalin-1(2H)-yl]-6,7-dimethoxyquinazolin-4-amine 391597 (+)-6,7-dimethoxy-2-[(4aS,8aR)-4-(5-methyl-2-furoyl)octahydroquinoxalin-1(2H)-yl]quinazolin-4-amine 391598 (+)-6,7-dimethoxy-2-[(4aS,8aR)-4-(5-methoxy-2-furoyl)octahydroquinoxalin-1(2H)-yl]quinazolin-4-amine 391599 (+)-1-(5-{[(4aR,8aS)-4-(4-amino-6,7-dimethoxyquinazolin-2-yl)octahydroquinoxalin-1(2H)-yl]carbonyl}-2-furyl)ethanone 391600 (+)-6,7-dimethoxy-2-[(4aS,8aR)-4-(2-thienylcarbonyl)octahydroquinoxalin-1(2H)-yl]quinazolin-4-amine 391601 (+)-6,7-dimethoxy-2-[(4aS,8aR)-4-(1H-pyrrol-2-ylcarbonyl)octahydroquinoxalin-1(2H)-yl]quinazolin-4-amine 391602 (+)-6,7-dimethoxy-2-[(4aS,8aR)-4-(pyridin-2-ylcarbonyl)octahydroquinoxalin-1(2H)-yl]quinazolin-4-amine 391603 (+)-2-[(4aS,8aR)-4-benzoyloctahydroquinoxalin-1(2H)-yl]-6,7-dimethoxyquinazolin-4-amine 391631 H-Tyr-Pro-Ala-Phe-NH2 391633 (S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-ylamino)-3-methyl-1-oxobutan-2-yl)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)pyrrolidine-2-carboxamide 391635 (S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-ylamino)-4-methyl-1-oxopentan-2-yl)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)pyrrolidine-2-carboxamide 391636 (S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-ylamino)-1-oxohexan-2-yl)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)pyrrolidine-2-carboxamide 391637 (S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-ylamino)-3-cyclohexyl-1-oxopropan-2-yl)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)pyrrolidine-2-carboxamide 391638 (S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-ylamino)-1-oxo-3-(perfluorophenyl)propan-2-yl)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)pyrrolidine-2-carboxamide 391646 (S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-ylamino)-3-(1H-imidazol-4-yl)-1-oxopropan-2-yl)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)pyrrolidine-2-carboxamide 391651 (S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-ylamino)-3-(4-hydroxyphenyl)-1-oxopropan-2-yl)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)pyrrolidine-2-carboxamide 391657 H-Tyr-Pro-Phe-Ala-NH2 391658 (S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-N-((S)-1-((S)-1-amino-3-methyl-1-oxobutan-2-ylamino)-1-oxo-3-phenylpropan-2-yl)pyrrolidine-2-carboxamide 391659 (S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-N-((S)-1-((S)-1-amino-4-methyl-1-oxopentan-2-ylamino)-1-oxo-3-phenylpropan-2-yl)pyrrolidine-2-carboxamide 391660 (S)-N-((S)-1-((S)-1-amino-1-oxohexan-2-ylamino)-1-oxo-3-phenylpropan-2-yl)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)pyrrolidine-2-carboxamide 391662 (S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-N-((S)-1-((S)-1-amino-3-cyclohexyl-1-oxopropan-2-ylamino)-1-oxo-3-phenylpropan-2-yl)pyrrolidine-2-carboxamide 391663 (S)-N-((S)-1-((S)-1-amino-1-oxo-3-(perfluorophenyl)propan-2-ylamino)-1-oxo-3-phenylpropan-2-yl)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)pyrrolidine-2-carboxamide 391664 (S)-N-((S)-1-((S)-1-amino-3-(1H-imidazol-4-yl)-1-oxopropan-2-ylamino)-1-oxo-3-phenylpropan-2-yl)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)pyrrolidine-2-carboxamide 391665 (S)-N-((S)-1-((S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-ylamino)-1-oxo-3-phenylpropan-2-yl)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)pyrrolidine-2-carboxamide 391689 2-(benzyloxy)-5-(6-methoxy-7-(2-methoxyethoxy)quinazolin-4-ylamino)cyclohexa-2,5-diene-1,4-dione 391690 2-(3-fluorobenzyloxy)-5-(6-methoxy-7-(2-methoxyethoxy)quinazolin-4-ylamino)cyclohexa-2,5-diene-1,4-dione 391780 [3-(4-fluoro-phenyl)-1,4-dihydro-indeno[1,2-c]pyrazol-6-ylmethyl]-(cis-4-methyl-cyclohexyl)-amine 391781 (1r,4r)-N-((3-(4-fluorophenyl)-1,4-dihydroindeno[1,2-c]pyrazol-6-yl)methyl)-4-methylcyclohexanamine 391782 (1r,4r)-4-methyl-N-((3-phenyl-1,4-dihydroindeno[1,2-c]pyrazol-6-yl)methyl)cyclohexanamine 391783 (1r,4r)-N-((3-(4-chlorophenyl)-1,4-dihydroindeno[1,2-c]pyrazol-6-yl)methyl)-4-methylcyclohexanamine 391784 4-(6-(((1r,4r)-4-methylcyclohexylamino)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzenamine 391785 1-(4-(6-(((1r,4r)-4-methylcyclohexylamino)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenyl)propan-2-one 391786 (4-(6-(((1r,4r)-4-methylcyclohexylamino)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenyl)methanol 391787 (1r,4r)-4-methyl-N-((3-p-tolyl-1,4-dihydroindeno[1,2-c]pyrazol-6-yl)methyl)cyclohexanamine 391788 (1r,4r)-N-((3-(4-ethoxyphenyl)-1,4-dihydroindeno[1,2-c]pyrazol-6-yl)methyl)-4-methylcyclohexanamine 391789 (1r,4r)-4-methyl-N-((3-(4-(trifluoromethoxy)phenyl)-1,4-dihydroindeno[1,2-c]pyrazol-6-yl)methyl)cyclohexanamine 391790 N,N-dimethyl-4-(6-(((1r,4r)-4-methylcyclohexylamino)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzenamine 391791 methyl 4-(6-(((1r,4r)-4-methylcyclohexylamino)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoate 391792 4-(6-(((1r,4r)-4-methylcyclohexylamino)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenol 391793 trans-4-(6-((4-methylcyclohexylamino)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid 391795 cis-4-(6-((4-methylcyclohexylamino)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid 391796 4-(6-((4-hydroxypiperidin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid 391798 4-(6-(morpholinomethyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid 391799 4-{6-[(trans-4-hydroxy-cyclohexylamino)-methyl]-1,4-dihydro-indeno[1,2-c]pyrazol-3-yl}-benzoic acid 391801 4-(6-((neopentylamino)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid 391802 4-(6-(((1r,4r)-4-hydroxycyclohexyl)carbamoyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid 391803 4-(6-(neopentylcarbamoyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid 391804 4-(6-(morpholinomethyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzamide 391805 4-(6-((4-hydroxypiperidin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzamide 391807 4-(6-(((1r,4r)-4-methylcyclohexylamino)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzenesulfonamide 391808 N-(2-hydroxyethyl)-4-(6-(((1r,4r)-4-methylcyclohexylamino)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzenesulfonamide 391809 N-(4-(6-(((1r,4r)-4-methylcyclohexylamino)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenyl)acetamide 391811 (1r,4r)-N-((3-(4-(aminomethyl)phenyl)-1,4-dihydroindeno[1,2-c]pyrazol-6-yl)methyl)-4-methylcyclohexanamine 391812 4-(6-(((1r,4r)-4-hydroxycyclohexylamino)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)-N-(phenylsulfonyl)benzamide 391813 2-(4-(6-(((1s,4s)-4-methylcyclohexylamino)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenyl)acetonitrile 391814 2-(4-(6-(((1s,4s)-4-methylcyclohexylamino)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenyl)acetic acid 391816 4'-[6-(4-Hydroxy-cyclohexylmethyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl]-biphenyl-4-ol 391817 4'-{6-[(2-hydroxy-ethylamino)-methyl]-1,4-dihydro-indeno[1,2-c]pyrazol-3-yl}-biphenyl-4-ol 391819 4'-{6-[(trans-4-hydroxy-cyclohexylamino)-methyl]-1,4-dihydro-indeno[1,2-c]pyrazol-3-yl}-biphenyl-4-ol 391820 4'-(6-{[(5-methyl-pyrazin-2-ylmethyl)-amino]-methyl}-1,4-dihydro-indeno[1,2-c]pyrazol-3-yl)-biphenyl-4-ol 391822 3-(4'-hydroxybiphenyl-4-yl)-N-(trans-4-hydroxycyclohexyl)-2,4-dihydroindeno[1,2-c]pyrazole-6-carboxamide 391824 3-(4'-hydroxy-biphenyl-4-yl)-1,4-dihydro-indeno[1,2-c]pyrazole-6-carboxylic acid (2-dimethylamino-ethyl)-amide 391825 3-(4'-hydroxy-biphenyl-4-yl)-1,4-dihydro-indeno[1,2-c]pyrazole-6-carboxylic acid (pyridin-4-ylmethyl)-amide 391827 [3-(4'-hydroxy-biphenyl-4-yl)-1,4-dihydro-indeno[1,2-c]pyrazol-6-yl]-(4-hydroxy-piperidin-1-yl)-methanone 391927 MCL-147 391928 MCL-183 391929 2'-amino oxazole[5,4-b]-N-cyclopropylmethylmorphinan 391930 2'-amino oxazole[5,4-b]-N-cyclobutylmethylmorphinan 391931 oxazole-2-one-N-cyclopropylmethylmorphinan 391932 oxazole-2-one-N-cyclobutylmethylmorphinan 391933 N-cyclopropylmethylmorphinan-3-amino-urea 391934 N-cyclobutylmethylmorphinan-3-amino-urea 391935 3-methylurea-N-cyclobutylmethylmorphinan 391936 3-methylurea-N-cyclopropylmethylmorphinan 392195 Oxytocin 392198 [Pip7]OT 392203 [L-Tic7]OT 392204 [D-Tic7]OT 392213 [Aib7]OT 392215 [Gly(But)7]OT 392217 [Gly(But)3, Gly(But)7]OT 392230 [Mpa1, L-Tic7]OT 392232 [Mpa1, D-Tic7]OT 392245 [Mpa1, D-Tyr(Et)2, L-Tic7]OT 392247 [Mpa1, D-Tyr(Et)2, D-Tic7]OT 392251 [Mpa1, D-Tyr(Et)2, D-Tic7, D-Tic9]OT 392252 [Mpa1, D-Tyr(Et)2, D-Tic7, Aib9]OT 392255 [Mpa1, D-Tyr(Et)2, Pip7]OT 392256 [Mpa1, D-Tyr(Et)2, Gly(But)7]OT 392257 [Mpa1, D-Tyr(Et)2, Gly(But)3, Gly(But)7]OT 392260 [Mpa1, D-Tyr(Et)2, Aib7]OT 392261 [Mpa1, D-Tyr(Et)2, Aib7, D-Tic9]OT 392267 [Mpa1, D-Tic2, Aib7]OT 392528 7-methylmelatonin (N-acetyl 5-methoxy-7-methyltryptamine) 392531 N-propanoyl 5-methoxy-7-methyltryptamine 392532 N-butanoyl 5-methoxy-7-methyltryptamine 392534 1,7-dimethylmelatonin (N-acetyl 5-methoxy-1,7-dimethyltryptamine) 392535 N-propanoyl 5-methoxy-1,7-dimethyltryptamine 392537 N-butanoyl 5-methoxy-1,7-dimethyltryptamine 392538 7-bromomelatonin (N-acetyl 7-bromo-5-methoxytryptamine) 392539 N-propanoyl 7-bromo-5-methoxytryptamine 392540 N-butanoyl 7-bromo-5-methoxytryptamine 392541 7-bromo-1-methylmelatonin (N-acetyl 7-bromo-5-methoxy-1-methyltryptamine) 392543 N-propanoyl 7-bromo-5-methoxy-1-methyltryptamine 392544 N-butanoyl 7-bromo-5-methoxy-1-methyltryptamine 392545 7-phenylmelatonin (N-acetyl 5-methoxy-7-phenyltryptamine) 392546 N-propanoyl 5-methoxy-7-phenyltryptamine 392548 N-butanoyl 5-methoxy-7-phenyltryptamine 392549 1-methyl-7-phenylmelatonin (N-acetyl 1-methyl-5-methoxy-7-phenyltryptamine) 392551 N-propanoyl 5-methoxy-1-methyl-7-phenyltryptamine 392554 N-butanoyl 5-methoxy-1-methyl-7-phenyltryptamine 393375 (S)-N-((S)-1-((S)-1-(allylamino)-1-oxo-3-phenylpropan-2-ylamino)-1-oxo-3-phenylpropan-2-yl)-1-((S)-2-(allylamino)-3-(4-hydroxyphenyl)propanoyl)pyrrolidine-2-carboxamide 393376 (S)-1-((S)-2-(allylamino)-3-(4-hydroxyphenyl)propanoyl)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-ylamino)-1-oxo-3-phenylpropan-2-yl)pyrrolidine-2-carboxamide 393377 (S)-N-((S)-1-((S)-1-(allylamino)-1-oxo-3-phenylpropan-2-ylamino)-1-oxo-3-phenylpropan-2-yl)-1-((S)-2-(allylamino)-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)pyrrolidine-2-carboxamide 393378 (S)-1-((S)-2-(allylamino)-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-ylamino)-1-oxo-3-phenylpropan-2-yl)pyrrolidine-2-carboxamide 393379 (S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-ylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-yl)-1-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)pyrrolidine-2-carboxamide 393380 (S)-N-((S)-1-((S)-1-(allylamino)-1-oxo-3-phenylpropan-2-ylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-yl)-1-((S)-2-(allylamino)-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)pyrrolidine-2-carboxamide 393381 (S)-1-((S)-2-(allylamino)-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-ylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-yl)pyrrolidine-2-carboxamide 393382 (S)-2-allylamino-N-{6-[(S)-2-allylamino-3-(4-hydroxy-phenyl)-propionylamino]-hexyl}-3-(4-hydroxy-phenyl)-propionamide 393383 (S)-2-allylamino-N-(5-{[(S)-2-allylamino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionyl]-propyl-amino}-3-oxo-3,4-dihydro-pyrazin-2-yl)-3-(4-hydroxy-2,6-dimethyl-phenyl)-N-propyl-propionamide 393443 1-benzhydryl-4-(2-fluorophenyl)piperidin-4-ol 393444 1-benzhydryl-4-(3-fluorophenyl)piperidin-4-ol 393445 1-benzhydryl-4-(4-fluorophenyl)piperidin-4-ol 393446 1-benzhydryl-4-(4-chlorophenyl)piperidin-4-ol 393447 1-benzhydryl-4-(4-bromophenyl)piperidin-4-ol 393448 1-benzhydryl-4-o-tolylpiperidin-4-ol 393449 1-benzhydryl-4-m-tolylpiperidin-4-ol 393454 1-benzhydryl-4-p-tolylpiperidin-4-ol 393455 1-benzhydryl-4-(4-ethylphenyl)piperidin-4-ol 393456 1-benzhydryl-4-(4-propylphenyl)piperidin-4-ol 393457 1-benzhydryl-4-(4-butylphenyl)piperidin-4-ol 393459 1-benzhydryl-4-(2-methoxyphenyl)piperidin-4-ol 393461 1-benzhydryl-4-(3-methoxyphenyl)piperidin-4-ol 393463 1-benzhydryl-4-(4-methoxyphenyl)piperidin-4-ol 393466 1-benzhydryl-4-(4-(dimethylamino)phenyl)piperidin-4-ol 393468 4-(1-benzhydryl-4-hydroxypiperidin-4-yl)benzonitrile 393469 1-benzhydryl-4-(2-(hydroxymethyl)phenyl)piperidin-4-ol 393470 4-(2-(aminomethyl)phenyl)-1-benzhydrylpiperidin-4-ol 393472 1-benzhydryl-4-cyclopropylpiperidin-4-ol 393474 1-benzhydryl-4-isopropylpiperidin-4-ol 393475 1-benzhydryl-4-butylpiperidin-4-ol 393477 1-benzhydryl-4-tert-butylpiperidin-4-ol 393480 1-benzhydryl-4-hexylpiperidin-4-ol 393481 1-benzhydryl-4-cyclohexylpiperidin-4-ol 393483 1-benzhydryl-4-benzylpiperidin-4-ol 393484 1-benzhydryl-4-(3-phenylpropyl)piperidin-4-ol 393486 1-benzhydryl-4-(furan-2-yl)piperidin-4-ol 393498 1-benzhydryl-4-(thiophen-2-yl)piperidin-4-ol 393500 1-benzhydryl-4-(3-methylthiophen-2-yl)piperidin-4-ol 393504 1-benzhydryl-4-(pyridin-2-yl)piperidin-4-ol 393506 4-(2-(aminomethyl)phenyl)-1-benzylpiperidin-4-ol 393508 4-(2-(aminomethyl)phenyl)-1-(1-phenylpentyl)piperidin-4-ol 393509 4-(2-(aminomethyl)phenyl)-1-(1-phenylhexyl)piperidin-4-ol 393511 4-(2-(aminomethyl)phenyl)-1-(phenyl(o-tolyl)methyl)piperidin-4-ol 393514 4-(2-(aminomethyl)phenyl)-1-((2-chlorophenyl)(phenyl)methyl)piperidin-4-ol 393515 4-(2-(aminomethyl)phenyl)-1-((2-bromophenyl)(phenyl)methyl)piperidin-4-ol 393516 4-(2-(aminomethyl)phenyl)-1-(dio-tolylmethyl)piperidin-4-ol 393517 4-(2-(aminomethyl)phenyl)-1-(dip-tolylmethyl)piperidin-4-ol 393518 4-(2-(aminomethyl)phenyl)-1-(bis(4-chlorophenyl)methyl)piperidin-4-ol 393519 4-(2-(aminomethyl)phenyl)-1-(bis(2-chlorophenyl)methyl)piperidin-4-ol 393520 4-(2-(aminomethyl)phenyl)-1-(bis(2-fluorophenyl)methyl)piperidin-4-ol 393521 4-(2-(aminomethyl)phenyl)-1-(bis(3-fluorophenyl)methyl)piperidin-4-ol 393522 4-(2-(aminomethyl)phenyl)-1-(bis(2-bromophenyl)methyl)piperidin-4-ol 393523 4-(2-(aminomethyl)phenyl)-1-(cycloheptylmethyl)piperidin-4-ol 393524 4-(2-(aminomethyl)phenyl)-1-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)piperidin-4-ol 393525 1-(bis(2-chlorophenyl)methyl)-4-(2-((methylamino)methyl)phenyl)piperidin-4-ol 393526 N-(2-(1-(bis(2-chlorophenyl)methyl)-4-hydroxypiperidin-4-yl)benzyl)propane-1-sulfonamide 393567 N-(2-(1-(bis(2-chlorophenyl)methyl)-4-hydroxypiperidin-4-yl)benzyl)propane-2-sulfonamide 393568 1-(2-(1-(bis(2-chlorophenyl)methyl)-4-hydroxypiperidin-4-yl)benzyl)-3-methylurea 393569 1-(2-(1-(bis(2-chlorophenyl)methyl)-4-hydroxypiperidin-4-yl)benzyl)-3-ethylurea 393570 1-(bis(2-chlorophenyl)methyl)-4-(2-(morpholinomethyl)phenyl)piperidin-4-ol 393572 1-(bis(2-chlorophenyl)methyl)-4-(2-(piperazin-1-ylmethyl)phenyl)piperidin-4-ol 393573 1-(bis(2-chlorophenyl)methyl)-4-(2-((4-methylpiperazin-1-yl)methyl)phenyl)piperidin-4-ol 393574 1-(bis(2-chlorophenyl)methyl)-4-(2-((4-(ethylsulfonyl)piperazin-1-yl)methyl)phenyl)piperidin-4-ol 393576 1-(bis(2-chlorophenyl)methyl)-4-(2-((4-(isopropylsulfonyl)piperazin-1-yl)methyl)phenyl)piperidin-4-ol 393693 1-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-6-(methylamino)-9H-purin-2-yl)-N-methyl-1H-pyrazole-4-carboxamide 393694 (2R,3S,4R,5R)-2-(hydroxymethyl)-5-(2-(4-(4-methoxyphenyl)-1H-pyrazol-1-yl)-6-(methylamino)-9H-purin-9-yl)-tetrahydrofuran-3,4-diol 393696 (2R,3R,4S,5R)-2-(6-(ethylamino)-2-(4-(4-methoxyphenyl)-1H-pyrazol-1-yl)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 393698 (2R,3S,4R,5R)-2-(hydroxymethyl)-5-(6-(methylamino)-2-(4-(pyridin-2-yl)-1H-pyrazol-1-yl)-9H-purin-9-yl)-tetrahydrofuran-3,4-diol 393700 (2R,3R,4S,5R)-2-(6-(ethylamino)-2-(4-(pyridin-2-yl)-1H-pyrazol-1-yl)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 393703 ethyl 1-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-6-((R)-tetrahydrofuran-2-ylamino)-9H-purin-2-yl)-1H-pyrazole-4-carboxylate 393705 1-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-6-((R)-tetrahydrofuran-2-ylamino)-9H-purin-2-yl)-N-methyl-1H-pyrazole-4-carboxamide 393707 1-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-6-((R)-tetrahydrofuran-2-ylamino)-9H-purin-2-yl)-N-ethyl-1H-pyrazole-4-carboxamide 393709 1-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-6-((R)-tetrahydrofuran-2-ylamino)-9H-purin-2-yl)-N-propyl-1H-pyrazole-4-carboxamide 393712 1-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-6-((R)-tetrahydrofuran-2-ylamino)-9H-purin-2-yl)-1H-pyrazole-4-carboxylic acid 393714 N-benzyl-1-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-6-((R)-tetrahydrofuran-2-ylamino)-9H-purin-2-yl)-1H-pyrazole-4-carboxamide 393717 N-(4-fluorobenzyl)-1-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-6-((R)-tetrahydrofuran-2-ylamino)-9H-purin-2-yl)-1H-pyrazole-4-carboxamide 393718 N-(4-chlorobenzyl)-1-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-6-((R)-tetrahydrofuran-2-ylamino)-9H-purin-2-yl)-1H-pyrazole-4-carboxamide 393719 ethyl 4-((1-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-6-((R)-tetrahydrofuran-2-ylamino)-9H-purin-2-yl)-1H-pyrazole-4-carboxamido)methyl)benzoate 393721 4-((1-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-6-((R)-tetrahydrofuran-2-ylamino)-9H-purin-2-yl)-1H-pyrazole-4-carboxamido)methyl)benzoic acid 393724 1-(6-(cyclopentylamino)-9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-9H-purin-2-yl)-N-methyl-1H-pyrazole-4-carboxamide 393726 1-(6-(cyclopentylamino)-9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-9H-purin-2-yl)-N-ethyl-1H-pyrazole-4-carboxamide 393731 1-(6-(cyclopentylamino)-9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-9H-purin-2-yl)-1H-pyrazole-4-carboxylic acid 393734 1-(6-(cyclopentylamino)-9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-9H-purin-2-yl)-1H-pyrazole-4-carboxamide 393736 ethyl 1-(6-(cyclopentylamino)-9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-9H-purin-2-yl)-1H-pyrazole-4-carboxylate 393738 (2R,3R,4S,5R)-2-(6-(cyclopentylamino)-2-(1H-pyrazol-1-yl)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 393740 ethyl 1-(6-(bicyclo[2.2.1]heptan-1-ylamino)-9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-9H-purin-2-yl)-1H-pyrazole-4-carboxylate 393744 (2R,3R,4S,5R)-2-(6-(bicyclo[2.2.1]heptan-1-ylamino)-2-(1H-pyrazol-1-yl)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 393746 ethyl 1-(6-(cyclohexylamino)-9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-9H-purin-2-yl)-1H-pyrazole-4-carboxylate 393748 1-(6-(cyclohexylamino)-9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-9H-purin-2-yl)-N-methyl-1H-pyrazole-4-carboxamide 393751 (2R,3R,4S,5R)-2-(6-(p-toluidino)-2-(4-(hydroxymethyl)-1H-pyrazol-1-yl)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 393756 (2R,3S,4R,5R)-2-(hydroxymethyl)-5-(2-(4-(hydroxymethyl)-1H-pyrazol-1-yl)-6-(4-(trifluoromethyl)phenylamino)-9H-purin-9-yl)-tetrahydrofuran-3,4-diol 393759 (2R,3S,4R,5R)-2-(hydroxymethyl)-5-(2-(4-(hydroxymethyl)-1H-pyrazol-1-yl)-6-(pyridin-2-ylamino)-9H-purin-9-yl)-tetrahydrofuran-3,4-diol 393762 (2R,3S,4R,5R)-2-(hydroxymethyl)-5-(2-(4-(hydroxymethyl)-1H-pyrazol-1-yl)-6-(pyridin-4-ylamino)-9H-purin-9-yl)-tetrahydrofuran-3,4-diol 393785 (2R,3S,4R,5R)-2-(hydroxymethyl)-5-(2-(4-(hydroxymethyl)-1H-pyrazol-1-yl)-6-(quinolin-2-ylamino)-9H-purin-9-yl)-tetrahydrofuran-3,4-diol 393786 (2R,3S,4R,5R)-2-(hydroxymethyl)-5-(2-(4-(hydroxymethyl)-1H-pyrazol-1-yl)-6-(pyrazin-2-ylamino)-9H-purin-9-yl)-tetrahydrofuran-3,4-diol 393789 (2R,3S,4R,5R)-2-(hydroxymethyl)-5-(2-(4-(hydroxymethyl)-1H-pyrazol-1-yl)-6-(quinazolin-2-ylamino)-9H-purin-9-yl)-tetrahydrofuran-3,4-diol 393790 2-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-2-(4-(hydroxymethyl)-1H-pyrazol-1-yl)-9H-purin-6-ylamino)isonicotinic acid 393793 1-(6-(p-toluidino)-9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-9H-purin-2-yl)-N-ethyl-1H-pyrazole-4-carboxamide 393795 1-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-6-(quinolin-2-ylamino)-9H-purin-2-yl)-N-ethyl-1H-pyrazole-4-carboxamide 393862 N2-(2,4-dichlorobenzyl)-N6-(5-(diethylamino)pentan-2-yl)-7H-purine-2,6-diamine 393863 N6-(2,4-dichlorobenzyl)-N2-(5-(diethylamino)pentan-2-yl)-7H-purine-2,6-diamine 393864 N6-(2,4-dichlorobenzyl)-N2-(5-(diethylamino)pentan-2-yl)-7-ethyl-7H-purine-2,6-diamine 393865 N2-(2,4-dichlorobenzyl)-N6-(5-(diethylamino)pentan-2-yl)-7-ethyl-7H-purine-2,6-diamine 393866 9-(2,4-dichlorobenzyl)-N-(5-(diethylamino)pentan-2-yl)-9H-purin-2-amine 393867 7-(2,4-dichlorobenzyl)-N-(5-(diethylamino)pentan-2-yl)-7H-purin-2-amine 393868 1-(2,4-dichlorobenzyl)-N-(5-(diethylamino)pentan-2-yl)-1H-pyrazolo[3,4-b]pyridin-6-amine 393869 N2-(2,4-dichlorobenzyl)-N4-(5-(diethylamino)pentan-2-yl)quinazoline-2,4-diamine 393870 N4-(2,4-dichlorobenzyl)-N2-(5-(diethylamino)pentan-2-yl)quinazoline-2,4-diamine 393871 N4-(2,4-dichlorobenzyl)-N2-(5-(diethylamino)pentan-2-yl)pyrido[2,3-d]pyrimidine-2,4-diamine 393872 (S)-(4-(4-(2,4-dichlorobenzylamino)pyrido[2,3-d]pyrimidin-2-yl)piperazin-1-yl)(piperidin-2-yl)methanone 393873 (S)-(4-(4-(2,4-dichlorobenzylamino)pyrido[2,3-d]pyrimidin-2-yl)piperazin-1-yl)(pyrrolidin-2-yl)methanone 393874 N4-(2,4-dichlorobenzyl)-N2-(4-(diethylamino)pentyl)pyrimidine-2,4-diamine 393876 N2-(2,4-dichlorobenzyl)-N4-(5-(diethylamino)pentan-2-yl)-N6-methyl-1,3,5-triazine-2,4,6-triamine 393960 4-(4-methoxyphenyl)-2-methyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 393961 4-(4-methoxyphenyl)-2-methyl-7-(3-morpholinopropoxy)-1,2,3,4-tetrahydroisoquinoline 393962 7-(3-(4-fluoropiperidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline 393963 7-(3-(4,4-difluoropiperidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline 393964 7-(3-(3,3-difluoropiperidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline 393965 1-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperidin-4-ol 393966 (1-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperidin-4-yl)methanol 393967 1-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperidine-4-carbonitrile 393968 4-(4-methoxyphenyl)-2-methyl-7-(3-(4-(trifluoromethyl)piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 393971 7-[3-(1,1-dioxo-1lambda*6*-thiomorpholin-4-yl)-propoxy]-4-(4-methoxy-phenyl)-2-methyl-1,2,3,4-tetrahydro-isoquinoline 393973 7-(3-(azetidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline 393974 7-(3-(3,3-difluoroazetidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline 393976 7-(3-(3,3-difluoropyrrolidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline 393977 N-ethyl-3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propan-1-amine 393979 N,N-diethyl-3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propan-1-amine 393982 N-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)cyclopropanamine 393984 N-cyclopropyl-N-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)cyclopropanamine 393986 7-(3-(4-ethylpiperazin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline 393987 7-(3-(4-isopropylpiperazin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline 393990 7-(3-(4-cyclopropylpiperazin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline 393992 2-(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)phenol 393994 4-(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)benzonitrile 393998 4-(4-methoxyphenyl)-2-methyl-7-(3-(4-(thiazol-2-yl)piperazin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 394000 4-(4-methoxyphenyl)-2-methyl-7-(3-(4-(pyridin-4-yl)piperazin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 394002 4-(4-methoxyphenyl)-2-methyl-7-(3-(4-(4-(trifluoromethyl)phenyl)piperazin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 394004 1-(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)ethanone 394006 1-(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)-2-methylpropan-1-one 394008 (4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)(1-methyl-1H-pyrrol-2-yl)methanone 394010 1-(4-ethylphenyl)-3-methyl-6-(4-(4-(1-phenylvinyl)cyclohexyl)butyl)-1,2,3,4-tetrahydronaphthalene 394141 (S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-methyl-N-((S)-pyrrolidin-3-yl)pyrrolidine-1-carboxamide 394142 (S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-methyl-N-((S)-1-(3-phenylpropyl)pyrrolidin-3-yl)pyrrolidine-1-carboxamide 394143 (S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-methyl-N-((S)-1-methylpyrrolidin-3-yl)pyrrolidine-1-carboxamide 394145 1-(2-cyclopropyl-5-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl)azepane 394147 (S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-((S)-1-isopropylpyrrolidin-3-yl)-N-methylpyrrolidine-1-carboxamide 394148 1-(2-cyclopropyl-5-methyl-6-(piperidin-1-yl)pyrimidin-4-yl)azepane 394150 1-(6-(azepan-1-yl)-2-cyclopropyl-5-methylpyrimidin-4-yl)azepane 394152 (S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-((S)-1-cyclobutylpyrrolidin-3-yl)-N-methylpyrrolidine-1-carboxamide 394154 (S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-((S)-1-cyclopentylpyrrolidin-3-yl)-N-methylpyrrolidine-1-carboxamide 394155 (S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-((S)-1-(4,4-dimethylcyclohexyl)pyrrolidin-3-yl)-N-methylpyrrolidine-1-carboxamide 394157 1-(2-cyclopropyl-5-methyl-6-(3-methylazetidin-1-yl)pyrimidin-4-yl)azepane 394158 1-(2-cyclopropyl-6-(3,3-dimethylazetidin-1-yl)-5-methylpyrimidin-4-yl)azepane 394159 1-(6-(azepan-1-yl)-2-cyclopropyl-5-methylpyrimidin-4-yl)azetidin-3-ol 394160 (S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-((S)-1-(cyclopropylmethyl)pyrrolidin-3-yl)-N-methylpyrrolidine-1-carboxamide 394161 1-(6-(3-bromoazetidin-1-yl)-2-cyclopropyl-5-methylpyrimidin-4-yl)azepane 394163 (S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-((S)-1-(cyclohexylmethyl)pyrrolidin-3-yl)-N-methylpyrrolidine-1-carboxamide 394166 1-(6-(azepan-1-yl)-2-cyclopropyl-5-methylpyrimidin-4-yl)azetidine-3-carbonitrile 394167 1-(2-cyclopropyl-6-(3-fluoroazetidin-1-yl)-5-methylpyrimidin-4-yl)azepane 394168 (S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-((S)-1-(furan-3-ylmethyl)pyrrolidin-3-yl)-N-methylpyrrolidine-1-carboxamide 394169 1-(6-(azepan-1-yl)-2-cyclopropyl-5-methylpyrimidin-4-yl)azetidin-3-one 394170 1-(2-cyclopropyl-6-(3-methoxyazetidin-1-yl)-5-methylpyrimidin-4-yl)azepane 394172 (S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-methyl-N-((S)-1-((tetrahydrofuran-3-yl)methyl)pyrrolidin-3-yl)pyrrolidine-1-carboxamide 394173 1-(6-(azetidin-1-yl)-2-cyclopropylpyrimidin-4-yl)azepane 394174 1-(2-cyclopropyl-6-(3-methylazetidin-1-yl)pyrimidin-4-yl)azepane 394175 1-(2-cyclopropyl-6-(3-fluoroazetidin-1-yl)pyrimidin-4-yl)azepane 394181 (S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-methyl-N-((S)-1-(tetrahydro-2H-pyran-4-yl)pyrrolidin-3-yl)pyrrolidine-1-carboxamide 394183 (S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-methyl-N-((S)-1-((tetrahydro-2H-pyran-4-yl)methyl)pyrrolidin-3-yl)pyrrolidine-1-carboxamide 394184 (S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-methyl-N-((S)-1-(2-(tetrahydro-2H-pyran-4-yl)ethyl)pyrrolidin-3-yl)pyrrolidine-1-carboxamide 394186 (S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-((S)-1-(3,3-dimethyl-2-oxobutyl)pyrrolidin-3-yl)-N-methylpyrrolidine-1-carboxamide 394189 (S)-3-[6-(4-chloro-phenyl)-4-oxo-4H-thieno[3,2-d]pyrimidin-3-yl]-pyrrolidine-1-carboxylic acid methyl-{(S)-1-[2-oxo-2-(4-trifluoromethoxy-phenyl)-ethyl]-pyrrolidin-3-yl}-amide 394198 (R)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-methyl-N-((R)-1-(tetrahydro-2H-pyran-4-yl)pyrrolidin-3-yl)pyrrolidine-1-carboxamide 394199 (R)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-methyl-N-((S)-1-(tetrahydro-2H-pyran-4-yl)pyrrolidin-3-yl)pyrrolidine-1-carboxamide 394200 (S)-N-methyl-N-((S)-1-methylpyrrolidin-3-yl)-3-(4-oxo-6-p-tolylthieno[3,2-d]pyrimidin-3(4H)-yl)pyrrolidine-1-carboxamide 394201 (S)-3-(6-(4-ethylphenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-methyl-N-((S)-1-methylpyrrolidin-3-yl)pyrrolidine-1-carboxamide 394202 (S)-3-(6-(2,4-dimethylphenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-methyl-N-((S)-1-methylpyrrolidin-3-yl)pyrrolidine-1-carboxamide 394203 (S)-N-methyl-N-((S)-1-methylpyrrolidin-3-yl)-3-(4-oxo-6-(4-(trifluoromethyl)phenyl)thieno[3,2-d]pyrimidin-3(4H)-yl)pyrrolidine-1-carboxamide 394204 (S)-N-methyl-N-((S)-1-methylpyrrolidin-3-yl)-3-(4-oxo-6-(4-(trifluoromethoxy)phenyl)thieno[3,2-d]pyrimidin-3(4H)-yl)pyrrolidine-1-carboxamide 394205 (S)-3-(6-(4-methoxyphenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-methyl-N-((S)-1-methylpyrrolidin-3-yl)pyrrolidine-1-carboxamide 394208 (S)-3-(6-(4-methoxy-2-methylphenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-methyl-N-((S)-1-methylpyrrolidin-3-yl)pyrrolidine-1-carboxamide 394210 (S)-3-(6-(2-chloro-4-ethoxyphenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-methyl-N-((S)-1-methylpyrrolidin-3-yl)pyrrolidine-1-carboxamide 394212 (S)-3-(6-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-methyl-N-((S)-1-methylpyrrolidin-3-yl)pyrrolidine-1-carboxamide 394215 (S)-N-methyl-3-(4-oxo-6-p-tolylthieno[3,2-d]pyrimidin-3(4H)-yl)-N-((S)-1-(tetrahydro-2H-pyran-4-yl)pyrrolidin-3-yl)pyrrolidine-1-carboxamide 394216 (S)-3-(6-(4-ethylphenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-methyl-N-((S)-1-(tetrahydro-2H-pyran-4-yl)pyrrolidin-3-yl)pyrrolidine-1-carboxamide 394217 (S)-3-(6-(2,4-dimethylphenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-methyl-N-((S)-1-(tetrahydro-2H-pyran-4-yl)pyrrolidin-3-yl)pyrrolidine-1-carboxamide 394218 (S)-N-methyl-3-(4-oxo-6-(4-(trifluoromethyl)phenyl)thieno[3,2-d]pyrimidin-3(4H)-yl)-N-((S)-1-(tetrahydro-2H-pyran-4-yl)pyrrolidin-3-yl)pyrrolidine-1-carboxamide 394220 (S)-N-methyl-3-(4-oxo-6-(4-(trifluoromethoxy)phenyl)thieno[3,2-d]pyrimidin-3(4H)-yl)-N-((S)-1-(tetrahydro-2H-pyran-4-yl)pyrrolidin-3-yl)pyrrolidine-1-carboxamide 394221 (S)-3-(6-(4-methoxy-2-methylphenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-methyl-N-((S)-1-(tetrahydro-2H-pyran-4-yl)pyrrolidin-3-yl)pyrrolidine-1-carboxamide 394222 (S)-3-(6-(2-chloro-4-ethoxyphenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-methyl-N-((S)-1-(tetrahydro-2H-pyran-4-yl)pyrrolidin-3-yl)pyrrolidine-1-carboxamide 394223 (S)-3-(6-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-methyl-N-((S)-1-(tetrahydro-2H-pyran-4-yl)pyrrolidin-3-yl)pyrrolidine-1-carboxamide 394242 2,7-dichloro-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)-9H-xanthene-9-carboxamide 394245 N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)-9,10-dihydroanthracene-10-carboxamide 394246 2,2-diphenyl-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)acetamide 394248 2,2-bis(4-chlorophenyl)-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)acetamide 394251 2-cyclohexyl-2-phenyl-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)acetamide 394259 2-(4,4-dimethylcyclohexyl)-2-phenyl-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)acetamide 394260 1-(6-(azetidin-1-yl)-2-cyclopropyl-5-methylpyrimidin-4-yl)azepane 394261 2-(4,4-difluorocyclohexyl)-2-phenyl-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)acetamide 394262 2-phenyl-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)-2-(3,3,5,5-tetramethylcyclohexyl)acetamide 394263 (E)-3-cyclohexyl-2-phenyl-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)acrylamide 394264 3-cyclohexyl-2-phenyl-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)propanamide 394265 2-cyclopentyl-2-phenyl-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)acetamide 394266 2-(cyclopent-3-enyl)-2-phenyl-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)acetamide 394268 2-cyclohexyl-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)-2-p-tolylacetamide 394285 2-cyclohexyl-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)-2-o-tolylacetamide 394288 2-cyclohexyl-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)-2-m-tolylacetamide 394290 2-cyclohexyl-2-(3,5-dimethylphenyl)-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)acetamide 394294 2-cyclohexyl-2-(4-methoxyphenyl)-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)acetamide 394301 2-(4-chlorophenyl)-2-cyclohexyl-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)acetamide 394308 2-(2-chlorophenyl)-2-(cyclohex-2-enyl)-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)acetamide 394309 2-(3-chlorophenyl)-2-(cyclohex-2-enyl)-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)acetamide 394310 2-cyclohexyl-2-(4-fluorophenyl)-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)acetamide 394311 2-cyclohexyl-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)-2-(3,4,5-trifluorophenyl)acetamide 394312 2-cyclohexyl-2-(4-nitrophenyl)-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)acetamide 394313 2-cyclohexyl-2-(naphthalen-2-yl)-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)acetamide 394314 2,2-dicyclohexyl-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)acetamide 394315 2-cyclohexyl-N-(1-(3-(2-methoxypyridin-3-yl)propanoyl)piperidin-4-yl)-2-phenylacetamide 394316 2-cyclohexyl-N-(1-(3-(2-fluoropyridin-3-yl)propanoyl)piperidin-4-yl)-2-phenylacetamide 394317 2-cyclohexyl-N-(1-(3-(6-fluoropyridin-3-yl)propanoyl)piperidin-4-yl)-2-phenylacetamide 394318 (E)-2-cyclohexyl-2-phenyl-N-(1-(3-(pyridin-3-yl)acryloyl)piperidin-4-yl)acetamide 394319 (E)-2-cyclohexyl-N-(1-(3-(5-methylpyridin-3-yl)acryloyl)piperidin-4-yl)-2-phenylacetamide 394320 2-cyclohexyl-N-(1-(3-(2-fluorophenyl)propanoyl)piperidin-4-yl)-2-phenylacetamide 394321 2-cyclohexyl-N-(1-(2-(2,3-difluorophenyl)acetyl)piperidin-4-yl)-2-phenylacetamide 394322 (E)-2-cyclohexyl-N-(1-(3-(2-fluorophenyl)acryloyl)piperidin-4-yl)-2-phenylacetamide 394323 6,7-dichloro-2-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-4-methyl-2,3-dihydropyrrolo[3,4-b]indol-1(4H)-one 394324 6-chloro-2-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-4-methyl-2,3-dihydropyrrolo[3,4-b]indol-1(4H)-one 394325 7-chloro-2-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-4-methyl-2,3-dihydropyrrolo[3,4-b]indol-1(4H)-one 394327 6-fluoro-2-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-4-methyl-2,3-dihydropyrrolo[3,4-b]indol-1(4H)-one 394329 7-methoxy-2-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-4-methyl-2,3-dihydropyrrolo[3,4-b]indol-1(4H)-one 394332 6-chloro-2-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)-4-methyl-2,3-dihydropyrrolo[3,4-b]indol-1(4H)-one 394333 7-chloro-2-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)-4-methyl-2,3-dihydropyrrolo[3,4-b]indol-1(4H)-one 394334 5-fluoro-2-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)-4-methyl-2,3-dihydropyrrolo[3,4-b]indol-1(4H)-one 394335 6-fluoro-2-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)-4-methyl-2,3-dihydropyrrolo[3,4-b]indol-1(4H)-one 394336 7-fluoro-2-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)-4-methyl-2,3-dihydropyrrolo[3,4-b]indol-1(4H)-one 394344 3-hydroxy-2-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)-4-methyl-2,3-dihydropyrrolo[3,4-b]indol-1(4H)-one 394359 2-[4-methoxy-3-(2-piperidin-1-yl-ethoxy)-phenyl]-2,3-dihydro-benzo[4,5]thieno[2,3-c]pyrrol-1-one 394360 2-{4-methoxy-3-[2-(4-methyl-piperidin-1-yl)-ethoxy]-phenyl}-2,3-dihydro-benzo[4,5]thieno[2,3-c]pyrrol-1-one 394456 [Nphe1Aib7Arg14Lys15]N/OFQ-NH2 394457 [(pF)Phe4Aib7Arg14Lys15]N/OFQ-NH2 394466 [Arg(14),Lys(15)]Nociceptin 394532 3-(2-(2-(2,4-difluorobenzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-4-fluorobenzoic acid 394533 3-(2-(2-(benzyloxy)-5-(trifluoromethyl)phenyl)-5-methyl-1H-pyrrol-1-yl)-4-fluorobenzoic acid 394534 3-(2-(2-(4-fluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-4-fluorobenzoic acid 394535 3-(2-(2-(4-fluorobenzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-4-chlorobenzoic acid 394536 3-(2-(2-(2,4-difluorobenzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-4-chlorobenzoic acid 394537 3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-4-methoxybenzoic acid 394538 3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-4-ethoxybenzoic acid 394553 3-(2-(2-(2,4-difluorobenzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-5-chlorobenzoic acid 394554 3-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-5-chlorobenzoic acid 394555 3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-5-bromobenzoic acid 394557 3-(2-(2-(2,4-difluorobenzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-5-bromobenzoic acid 394559 3-(2-(2-(2,4-difluorobenzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-5-(trifluoromethyl)benzoic acid 394561 3-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-5-(trifluoromethyl)benzoic acid 394563 3-amino-5-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 394564 3-amino-5-(2-(2-(benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 394565 3-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-5-aminobenzoic acid 394566 3-(2-(2-(4-fluorobenzyloxy)-5-fluorophenyl)-5-methyl-1H-pyrrol-1-yl)-5-acetamidobenzoic acid 394567 3-acetamido-5-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 394568 3-(2-(2-(4-fluorobenzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-5-acetamidobenzoic acid 394569 3-acetamido-5-(2-(2-(benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 394570 3-(2-(2-(4-fluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-5-acetamidobenzoic acid 394571 3-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-5-acetamidobenzoic acid 394572 3-(2-(2-(2,4-difluorobenzyloxy)-5-iodophenyl)-5-methyl-1H-pyrrol-1-yl)-5-acetamidobenzoic acid 394573 3-acetamido-5-(2-(2-(benzyloxy)-5-(trifluoromethyl)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid 394574 3-(2-(2-(4-fluorobenzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-5-(methylsulfonamido)benzoic acid 394575 3-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-5-(N-methylacetamido)benzoic acid 394576 3-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-5-(2-oxopyrrolidin-1-yl)benzoic acid 394577 3-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-5-(2-oxopiperidin-1-yl)benzoic acid 394578 3-[2-(2-benzyloxy-5-chloro-phenyl)-5-methyl-pyrrol-1-yl]-5-(1,1-dioxo-1lambda*6*-isothiazolidin-2-yl)-benzoic acid 394579 3-(1,1-dioxo-1lambda*6*-isothiazolidin-2-yl)-5-{2-[2-(4-fluoro-benzyloxy)-5-trifluoromethyl-phenyl]-5-methyl-pyrrol-1-yl}-benzoic acid 394580 3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-5-(methoxycarbonyl)benzoic acid 394581 (R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-chlorophenylamino)-4-(methylamino)cyclobut-3-ene-1,2-dione 394582 (R)-3-(2-(2-(4-benzyl-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-chlorophenylamino)-4-(methylamino)cyclobut-3-ene-1,2-dione 394583 (R)-3-(2-(2-(4-(4-chlorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-chlorophenylamino)-4-(methylamino)cyclobut-3-ene-1,2-dione 394584 (R)-3-(2-(2-(4-(4-bromobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-chlorophenylamino)-4-(methylamino)cyclobut-3-ene-1,2-dione 394585 (R)-3-(2-(2-(4-(3,4-difluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-chlorophenylamino)-4-(methylamino)cyclobut-3-ene-1,2-dione 394586 (R)-3-(2-(2-(4-(2-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-chlorophenylamino)-4-(methylamino)cyclobut-3-ene-1,2-dione 394588 (R)-3-(2-(2-(4-(3-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-chlorophenylamino)-4-(methylamino)cyclobut-3-ene-1,2-dione 394589 3-(2-(2-(4-(4-chlorobenzyl)piperazin-1-yl)-2-oxoethoxy)-5-chlorophenylamino)-4-(methylamino)cyclobut-3-ene-1,2-dione 394590 (R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)phenylamino)-4-(methylamino)cyclobut-3-ene-1,2-dione 394591 (R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-bromophenylamino)-4-(methylamino)cyclobut-3-ene-1,2-dione 394592 (R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-fluorophenylamino)-4-(methylamino)cyclobut-3-ene-1,2-dione 394593 (R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-methylphenylamino)-4-(methylamino)cyclobut-3-ene-1,2-dione 394594 (R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-4,5-difluorophenylamino)-4-(methylamino)cyclobut-3-ene-1,2-dione 394601 (R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-chlorophenylamino)-4-(ethylamino)cyclobut-3-ene-1,2-dione 394604 (R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-chlorophenylamino)-4-(propylamino)cyclobut-3-ene-1,2-dione 394605 (R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-chlorophenylamino)-4-(benzylamino)cyclobut-3-ene-1,2-dione 394608 (R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-chlorophenylamino)-4-aminocyclobut-3-ene-1,2-dione 394612 (R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-chlorophenylamino)-4-(2-(dimethylamino)ethylamino)cyclobut-3-ene-1,2-dione 394615 (R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-chlorophenylamino)-4-(2-methoxyethylamino)cyclobut-3-ene-1,2-dione 394616 (R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-chlorophenylamino)-4-(2-hydroxyethylamino)cyclobut-3-ene-1,2-dione 394618 (R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-chlorophenylamino)-4-(2-aminoethylamino)cyclobut-3-ene-1,2-dione 394620 (R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-chlorophenylamino)-4-(2-(pyrrolidin-1-yl)ethylamino)cyclobut-3-ene-1,2-dione 394622 (R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-chlorophenylamino)-4-(2-morpholinoethylamino)cyclobut-3-ene-1,2-dione 394623 (R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-chlorophenylamino)-4-(2-(piperazin-1-yl)ethylamino)cyclobut-3-ene-1,2-dione 394624 (R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-chlorophenylamino)-4-(pyridin-2-ylmethylamino)cyclobut-3-ene-1,2-dione 394625 (R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-chlorophenylamino)-4-(pyridin-3-ylmethylamino)cyclobut-3-ene-1,2-dione 394626 (R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-chlorophenylamino)-4-(pyridin-4-ylmethylamino)cyclobut-3-ene-1,2-dione 394629 (R,E)-3-(2-(3-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-3-oxoprop-1-enyl)-5-chlorophenylamino)-4-aminocyclobut-3-ene-1,2-dione 394630 (R,E)-3-(2-(3-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-3-oxoprop-1-enyl)-5-chlorophenylamino)-4-(methylamino)cyclobut-3-ene-1,2-dione 394632 (R)-1-(5-chloro-2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)phenyl)urea 394668 3-(2-(2-(benzyloxy)phenyl)cyclopent-1-enyl)benzoic acid 394669 3-(2-(2-(2,4-difluorobenzyloxy)phenyl)cyclopent-1-enyl)benzoic acid 394670 3-(2-(2-(3,4-dichlorobenzyloxy)phenyl)cyclopent-1-enyl)benzoic acid 394671 3-(2-(2-(4-chloro-2-fluorobenzyloxy)phenyl)cyclopent-1-enyl)benzoic acid 394672 3-(2-(2-(4-methoxybenzyloxy)phenyl)cyclopent-1-enyl)benzoic acid 394673 3-(2-(2-(benzyloxy)-5-bromophenyl)cyclopent-1-enyl)benzoic acid 394674 3-(2-(2-(4-chlorobenzyloxy)-5-bromophenyl)cyclopent-1-enyl)benzoic acid 394675 3-(2-(2-(4-fluorobenzyloxy)-5-bromophenyl)cyclopent-1-enyl)benzoic acid 394676 3-(2-(2-(3,4-dichlorobenzyloxy)-5-bromophenyl)cyclopent-1-enyl)benzoic acid 394677 3-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)cyclopent-1-enyl)benzoic acid 394678 3-(2-(2-(4-chloro-2-fluorobenzyloxy)-5-bromophenyl)cyclopent-1-enyl)benzoic acid 394679 3-(2-(2-(4-methoxybenzyloxy)-5-bromophenyl)cyclopent-1-enyl)benzoic acid 394680 3-(2-(2-(benzyloxy)-5-(methylthio)phenyl)cyclopent-1-enyl)benzoic acid 394681 3-(2-(2-(4-fluorobenzyloxy)-5-(methylthio)phenyl)cyclopent-1-enyl)benzoic acid 394682 3-(2-(2-(2,4-difluorobenzyloxy)-5-(methylthio)phenyl)cyclopent-1-enyl)benzoic acid 394683 3-(2-(2-(benzyloxy)-5-(methylsulfonyl)phenyl)cyclopent-1-enyl)benzoic acid 394684 3-(2-(2-(4-fluorobenzyloxy)-5-(methylsulfonyl)phenyl)cyclopent-1-enyl)benzoic acid 394685 3-(2-(2-(2,4-difluorobenzyloxy)-5-(methylsulfonyl)phenyl)cyclopent-1-enyl)benzoic acid 394686 3-(2-(2-(benzyloxy)-5-cyanophenyl)cyclopent-1-enyl)benzoic acid 394687 3-(2-(2-(4-fluorobenzyloxy)-5-cyanophenyl)cyclopent-1-enyl)benzoic acid 394688 3-(2-(2-(2,4-difluorobenzyloxy)-5-cyanophenyl)cyclopent-1-enyl)benzoic acid 394689 3-(2-(2-(4-chlorobenzyloxy)-5-cyanophenyl)cyclopent-1-enyl)benzoic acid 394690 4-(2-(2-(benzyloxy)-5-(trifluoromethyl)phenyl)cyclopent-1-enyl)picolinic acid 394691 2-(2-(2-(4-fluorobenzyloxy)-5-bromophenyl)cyclopent-1-enyl)isonicotinic acid 394692 5-(2-(2-(benzyloxy)-5-(trifluoromethyl)phenyl)cyclopent-1-enyl)nicotinic acid 394693 5-(2-(2-(4-fluorobenzyloxy)-5-chlorophenyl)cyclopent-1-enyl)-2-methylnicotinic acid 394694 5-(2-(2-(benzyloxy)-5-chlorophenyl)cyclopent-1-enyl)pyridazine-3-carboxylic acid 394695 6-(2-(2-(2,4-difluorobenzyloxy)-5-chlorophenyl)cyclopent-1-enyl)pyridazine-4-carboxylic acid 394696 6-(2-(2-(benzyloxy)-5-chlorophenyl)cyclopent-1-enyl)pyrimidine-4-carboxylic acid 394697 2-(2-(2-(benzyloxy)-5-chlorophenyl)cyclopent-1-enyl)pyrimidine-4-carboxylic acid 394698 6-(2-(2-(2,4-difluorobenzyloxy)-5-chlorophenyl)cyclopent-1-enyl)pyrazine-2-carboxylic acid 394699 6-(2-(5-chloro-2-(2,4-difluorobenzyloxy)phenyl)cyclopent-1-enyl)picolinic acid 394768 (R)-3-(5-chloro-2-(2-(4-((5-chlorothiophen-2-yl)methyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)phenylamino)-4-(methylamino)cyclobut-3-ene-1,2-dione 394806 4-phenyl-2-(phenylamino)pyrimidine-5-carbonitrile 394807 4-phenyl-2-(4-(pyrrolidin-1-ylmethyl)phenylamino)pyrimidine-5-carbonitrile 394808 2-(3-methoxy-4-(pyrrolidin-1-ylmethyl)phenylamino)-4-phenylpyrimidine-5-carbonitrile 394809 4-phenyl-2-(4-(2-(pyrrolidin-1-yl)ethyl)phenylamino)pyrimidine-5-carbonitrile 394810 2-(4-(3-morpholino-3-oxopropyl)phenylamino)-4-phenylpyrimidine-5-carbonitrile 394811 2-(3-(morpholinomethyl)phenylamino)-4-phenylpyrimidine-5-carbonitrile 394812 2-(4-(2-hydroxyethyl)phenylamino)-4-phenylpyrimidine-5-carbonitrile 394813 2-(3-methoxyphenylamino)-4-phenylpyrimidine-5-carbonitrile 394814 2-(2-methyl-1H-indol-5-ylamino)-4-phenylpyrimidine-5-carbonitrile 394815 2-(4-methoxyphenylamino)-4-phenylpyrimidine-5-carbonitrile 394816 2-(p-toluidino)-4-phenylpyrimidine-5-carbonitrile 394817 2-(naphthalen-2-ylamino)-4-phenylpyrimidine-5-carbonitrile 394818 2-(1H-benzo[d]imidazol-2-ylamino)-4-phenylpyrimidine-5-carbonitrile 394825 16-hydroxy-4,14,18-triazaheptacyclo[12.10.2.0^{2,6}.0^{7,26}.0^{8,13}.0^{18,25}.0^{19,24}]hexacosa-1(25),2(6),7(26),8,10,12,19(24),20,22-nonaen-3-one 394827 16,16-bis(hydroxymethyl)-4,14,18-triazaheptacyclo[12.10.2.0^{2,6}.0^{7,26}.0^{8,13}.0^{18,25}.0^{19,24}]hexacosa-1(25),2(6),7(26),8,10,12,19(24),20,22-nonaen-3-one 394829 16-(1,3-dihydroxypropan-2-ylidene)-4,14,18-triazaheptacyclo[12.10.2.0^{2,6}.0^{7,26}.0^{8,13}.0^{18,25}.0^{19,24}]hexacosa-1(25),2(6),7(26),8,10,12,19(24),20,22-nonaen-3-one 394831 16-methylidene-4,14,18-triazaheptacyclo[12.10.2.0^{2,6}.0^{7,26}.0^{8,13}.0^{18,25}.0^{19,24}]hexacosa-1(25),2(6),7(26),8,10,12,19(24),20,22-nonaen-3-one 394833 16-hydroxy-16-(hydroxymethyl)-4,14,18-triazaheptacyclo[12.10.2.0^{2,6}.0^{7,26}.0^{8,13}.0^{18,25}.0^{19,24}]hexacosa-1(25),2(6),7(26),8,10,12,19(24),20,22-nonaen-3-one 394834 16-(hydroxymethyl)-4,14,18-triazaheptacyclo[12.10.2.0^{2,6}.0^{7,26}.0^{8,13}.0^{18,25}.0^{19,24}]hexacosa-1(25),2(6),7(26),8,10,12,19(24),20,22-nonaen-3-one 394836 10,16-bis(hydroxymethyl)-4,14,18-triazaheptacyclo[12.10.2.0^{2,6}.0^{7,26}.0^{8,13}.0^{18,25}.0^{19,24}]hexacosa-1(25),2(6),7(26),8,10,12,19(24),20,22-nonaen-3-one 394837 16-(hydroxymethyl)-10-[(propan-2-yloxy)methyl]-4,14,18-triazaheptacyclo[12.10.2.0^{2,6}.0^{7,26}.0^{8,13}.0^{18,25}.0^{19,24}]hexacosa-1(25),2(6),7(26),8,10,12,19(24),20,22-nonaen-3-one 394838 10-[(dimethylamino)methyl]-16-(hydroxymethyl)-4,14,18-triazaheptacyclo[12.10.2.0^{2,6}.0^{7,26}.0^{8,13}.0^{18,25}.0^{19,24}]hexacosa-1(25),2(6),7(26),8,10,12,19(24),20,22-nonaen-3-one 394840 22-bromo-16-(hydroxymethyl)-4,14,18-triazaheptacyclo[12.10.2.0^{2,6}.0^{7,26}.0^{8,13}.0^{18,25}.0^{19,24}]hexacosa-1(25),2(6),7(26),8,10,12,19(24),20,22-nonaen-3-one 394842 22-bromo-16-(hydroxymethyl)-3-oxo-4,14,18-triazaheptacyclo[12.10.2.0^{2,6}.0^{7,26}.0^{8,13}.0^{18,25}.0^{19,24}]hexacosa-1(25),2(6),7(26),8,10,12,19(24),20,22-nonaene-10-carbaldehyde 394844 22-bromo-16-(hydroxymethyl)-10-[(propan-2-yloxy)methyl]-4,14,18-triazaheptacyclo[12.10.2.0^{2,6}.0^{7,26}.0^{8,13}.0^{18,25}.0^{19,24}]hexacosa-1(25),2(6),7(26),8,10,12,19(24),20,22-nonaen-3-one 394846 22-bromo-16-(hydroxymethyl)-10-(morpholin-4-ylmethyl)-4,14,18-triazaheptacyclo[12.10.2.0^{2,6}.0^{7,26}.0^{8,13}.0^{18,25}.0^{19,24}]hexacosa-1(25),2(6),7(26),8,10,12,19(24),20,22-nonaen-3-one 394848 10,16,22-tris(hydroxymethyl)-4,14,18-triazaheptacyclo[12.10.2.0^{2,6}.0^{7,26}.0^{8,13}.0^{18,25}.0^{19,24}]hexacosa-1(25),2(6),7(26),8,10,12,19(24),20,22-nonaen-3-one 394850 16-(hydroxymethyl)-10,22-bis[(propan-2-yloxy)methyl]-4,14,18-triazaheptacyclo[12.10.2.0^{2,6}.0^{7,26}.0^{8,13}.0^{18,25}.0^{19,24}]hexacosa-1(25),2(6),7(26),8,10,12,19(24),20,22-nonaen-3-one 394853 16-(hydroxymethyl)-22-[(E)-2-(pyridin-2-yl)ethenyl]-4,14,18-triazaheptacyclo[12.10.2.0^{2,6}.0^{7,26}.0^{8,13}.0^{18,25}.0^{19,24}]hexacosa-1(25),2(6),7(26),8,10,12,19(24),20,22-nonaen-3-one 394854 4-(4-(2-aminopropan-2-yl)phenyl)-2-(4-(2-hydroxyethyl)phenylamino)pyrimidine-5-carbonitrile 394856 16-(hydroxymethyl)-22-[(E)-2-(4-methyl-1,3-thiazol-5-yl)ethenyl]-4,14,18-triazaheptacyclo[12.10.2.0^{2,6}.0^{7,26}.0^{8,13}.0^{18,25}.0^{19,24}]hexacosa-1(25),2(6),7(26),8,10,12,19(24),20,22-nonaen-3-one 394858 2-[5-((E)-2-biphenyl-4-yl-vinyl)-2-hydroxy-benzo[4,5]imidazo[1,2-a]quinolin-1-ylmethyl]-isoindole-1,3-dione 394859 16-(hydroxymethyl)-22-[(E)-2-(1H-imidazol-1-yl)ethenyl]-4,14,18-triazaheptacyclo[12.10.2.0^{2,6}.0^{7,26}.0^{8,13}.0^{18,25}.0^{19,24}]hexacosa-1(25),2(6),7(26),8,10,12,19(24),20,22-nonaen-3-one 394860 2-(4-(2-hydroxyethyl)phenylamino)-4-(thiophen-2-yl)pyrimidine-5-carbonitrile 394861 16-(hydroxymethyl)-22-[(1E)-3-(1H-imidazol-1-yl)prop-1-en-1-yl]-4,14,18-triazaheptacyclo[12.10.2.0^{2,6}.0^{7,26}.0^{8,13}.0^{18,25}.0^{19,24}]hexacosa-1(25),2(6),7(26),8,10,12,19(24),20,22-nonaen-3-one 394863 22-[(1E)-3-(4,5-dihydro-1H-imidazol-2-ylamino)prop-1-en-1-yl]-16-(hydroxymethyl)-4,14,18-triazaheptacyclo[12.10.2.0^{2,6}.0^{7,26}.0^{8,13}.0^{18,25}.0^{19,24}]hexacosa-1(25),2(6),7(26),8,10,12,19(24),20,22-nonaen-3-one 394864 2-[2-hydroxy-5-((E)-styryl)-benzo[4,5]imidazo[1,2-a]quinolin-1-ylmethyl]-isoindole-1,3-dione 394865 2-(4-(2-hydroxyethyl)phenylamino)-4-(1H-indol-5-yl)pyrimidine-5-carbonitrile 394866 (2E)-3-[16-(hydroxymethyl)-5-oxo-4,14,18-triazaheptacyclo[12.10.2.0^{2,6}.0^{7,26}.0^{8,13}.0^{18,25}.0^{19,24}]hexacosa-1(25),2(6),7(26),8(13),9,11,19,21,23-nonaen-10-yl]prop-2-enoic acid 394868 (2E)-N-[3-(dimethylamino)propyl]-3-[16-(hydroxymethyl)-5-oxo-4,14,18-triazaheptacyclo[12.10.2.0^{2,6}.0^{7,26}.0^{8,13}.0^{18,25}.0^{19,24}]hexacosa-1(25),2(6),7(26),8(13),9,11,19,21,23-nonaen-10-yl]prop-2-enamide 394870 2-(4-(2-hydroxyethyl)phenylamino)-4-(4-methoxyphenyl)pyrimidine-5-carbonitrile 394871 10,16-bis(hydroxymethyl)-22-[(1E)-3-(1H-imidazol-1-yl)prop-1-en-1-yl]-4,14,18-triazaheptacyclo[12.10.2.0^{2,6}.0^{7,26}.0^{8,13}.0^{18,25}.0^{19,24}]hexacosa-1(25),2(6),7(26),8,10,12,19(24),20,22-nonaen-3-one 394872 2-{2-hydroxy-5-[(E)-2-(4-hydroxy-phenyl)-vinyl]-benzo[4,5]imidazo[1,2-a]quinolin-1-ylmethyl}-isoindole-1,3-dione 394873 4-(4-bromophenyl)-2-(4-(2-hydroxyethyl)phenylamino)pyrimidine-5-carbonitrile 394876 4-(5-cyano-2-(4-(2-hydroxyethyl)phenylamino)pyrimidin-4-yl)benzenesulfonamide 394878 4-(benzo[d]thiazol-2-yl)-2-(4-(2-hydroxyethyl)phenylamino)pyrimidine-5-carbonitrile 394881 2-(4-(2-hydroxyethyl)phenylamino)-4-(4-(2-hydroxypropan-2-yl)phenyl)pyrimidine-5-carbonitrile 394882 2-(4-(2-hydroxyethyl)phenylamino)-4-(1H-indol-2-yl)pyrimidine-5-carbonitrile 394884 4-tert-butyl-2-(4-(2-hydroxyethyl)phenylamino)pyrimidine-5-carbonitrile 394890 4-(4-(2-aminopropan-2-yl)phenyl)-2-(4-(2-morpholinoethyl)phenylamino)pyrimidine-5-carbonitrile 394891 4-(4-(2-aminopropan-2-yl)phenyl)-2-(3-(2-morpholinoethyl)phenylamino)pyrimidine-5-carbonitrile 394893 4-(4-(2-aminopropan-2-yl)phenyl)-2-(4-(2-(2-ethyl-1H-imidazol-1-yl)ethyl)phenylamino)pyrimidine-5-carbonitrile 394894 4-(4-(2-aminopropan-2-yl)phenyl)-2-(4-(2-(4-methylpiperazin-1-yl)ethyl)phenylamino)pyrimidine-5-carbonitrile 394896 4-(4-(2-aminopropan-2-yl)phenyl)-2-(4-(2-morpholinoethoxy)phenylamino)pyrimidine-5-carbonitrile 394925 2-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)isoindolin-1-one 394927 4-chloro-2-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)isoindolin-1-one 394928 5-chloro-2-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)isoindolin-1-one 394929 6-chloro-2-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)isoindolin-1-one 394930 7-chloro-2-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)isoindolin-1-one 394931 4-chloro-2-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)isoindolin-1-one 394932 5-chloro-2-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)isoindolin-1-one 394933 6-chloro-2-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)isoindolin-1-one 394934 7-chloro-2-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)isoindolin-1-one 394935 7-fluoro-2-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)isoindolin-1-one 394936 7-bromo-2-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)isoindolin-1-one 394937 2-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)-7-(trifluoromethyl)isoindolin-1-one 394939 2-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)-3-oxoisoindoline-4-carbonitrile 394940 7-methoxy-2-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)isoindolin-1-one 394942 7-chloro-2-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)-3-methylisoindolin-1-one 394949 4-fluoro-2-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)-7-(trifluoromethyl)isoindolin-1-one 394950 7-chloro-4,5-difluoro-2-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)isoindolin-1-one 394951 5,6-dichloro-2-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)isoindolin-1-one 394953 5,7-dichloro-2-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)isoindolin-1-one 394955 6,7-dichloro-2-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)isoindolin-1-one 394957 5,6-dichloro-2-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)-7-methylisoindolin-1-one 394959 5,7-dichloro-2-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)-6-methylisoindolin-1-one 394961 5-fluoro-2-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)-7-(trifluoromethyl)isoindolin-1-one 394963 2-(4-methoxy-3-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)-5,7-dimethylisoindolin-1-one 394967 2-{4-methoxy-3-[2-(4-methyl-piperidin-1-yl)-ethoxy]-phenyl}-5,7-dimethyl-2,3-dihydro-isoindol-1-ylideneamine 394969 5,7-dichloro-2-(4-methoxy-3-(2-(3-methylpiperidin-1-yl)ethoxy)phenyl)isoindolin-1-one 394971 5,7-dichloro-2-(4-methoxy-3-(2-(2-methylpiperidin-1-yl)ethoxy)phenyl)isoindolin-1-one 394973 5,7-dichloro-2-(3-(2-((2R,6S)-2,6-dimethylpiperidin-1-yl)ethoxy)-4-methoxyphenyl)isoindolin-1-one 394976 5,7-dichloro-2-(3-(2-(4,4-dimethylpiperidin-1-yl)ethoxy)-4-methoxyphenyl)isoindolin-1-one 394977 2-(3-(2-(azepan-1-yl)ethoxy)-4-methoxyphenyl)-5,7-dichloroisoindolin-1-one 394980 5,7-dichloro-2-(4-methoxy-3-(2-morpholinoethoxy)phenyl)isoindolin-1-one 395015 1-(4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)pyrrolidine-2,5-dione 395025 N-((S)-1-{4-[4-(3-chlorophenyl)piperazin-1-yl]butyl}pyrrolidin-2,5-dion-yl)cyclopentanecarboxamide 395026 (S)-N-(1-(4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)-2,5-dioxopyrrolidin-3-yl)cyclohexanecarboxamide 395029 N-((S)-1-{4-[4-(3-chlorophenyl)piperazin-1-yl]butyl}pyrrolidin-2,5-dion-3-yl)-2-(bicyclo[2.2.1]heptan-2-yl)acetamide 395032 N-((S)-1-{4-[4-(3-chlorophenyl)piperazin-1-yl]butyl}pyrrolidin-2,5-dion-yl)-1-adamantanecarboxamide 395033 1-(cyclohexylcarbonyl)-N-{4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl}-L-prolinamide 395036 1-((bicyclo[2.2.1]heptan-2-yl)acetyl)-N-{4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl}-L-prolinamide 395039 1-(adamantylcarbonyl)-N-{4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl}-L-prolinamide 395040 1-(cyclohexylcarbonyl)-N-{4-[4-(3-chlorophenyl)piperazin-1-yl]butyl}-L-prolinamide 395041 1-((bicyclo[2.2.1]heptan-2-yl)acetyl)-N-{4-[4-(3-chlorophenyl)piperazin-1-yl]butyl}-L-prolinamide 395044 1-(adamantylcarbonyl)-N-{4-[4-(3-chlorophenyl)piperazin-1-yl]butyl}-L-prolinamide 395315 (2R,3R)-2-(5-(2,3-difluorobenzylthio)-2-aminothiazolo[4,5-d]pyrimidin-7-ylamino)butane-1,3-diol 395318 2-(5-(2,3-difluorobenzylthio)-2-aminothiazolo[4,5-d]pyrimidin-7-ylamino)-2-methylpropane-1,3-diol 395320 2-(5-(2,3-difluorobenzylthio)-2-aminothiazolo[4,5-d]pyrimidin-7-ylamino)propane-1,3-diol 395322 4,5,6,7-tetrafluoro-2-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)isoindoline-1,3-dione 395324 (R)-2-(5-(2,3-difluorobenzylthio)-2-aminothiazolo[4,5-d]pyrimidin-7-ylamino)propan-1-ol 395325 5,6-dichloro-2-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)isoindoline-1,3-dione 395326 (S)-2-(5-(2,3-difluorobenzylthio)-2-aminothiazolo[4,5-d]pyrimidin-7-ylamino)propan-1-ol 395328 4-fluoro-2-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)isoindoline-1,3-dione 395335 2-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2H-benzo[e]isoindole-1,3-dione 395337 (R)-2-(5-(2,3-difluorobenzylthio)-2-(cyclopropylamino)thiazolo[4,5-d]pyrimidin-7-ylamino)propan-1-ol 395339 8-fluoro-2-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2H-benzo[e]isoindole-1,3-dione 395342 2-(5-(2,3-difluorobenzylthio)-2-(cyclopropylamino)thiazolo[4,5-d]pyrimidin-7-ylamino)propane-1,3-diol 395345 (R)-2-(5-(2,3-difluorobenzylthio)-2-(isopropylamino)thiazolo[4,5-d]pyrimidin-7-ylamino)propan-1-ol 395348 6-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-6H-pyrrolo[3,4-b]pyridine-5,7-dione 395349 (R)-2-(5-(2,3-difluorobenzylthio)-2-(isopropylamino)thiazolo[4,5-d]pyrimidin-7-ylamino)butan-1-ol 395351 2-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2H-pyrrolo[3,4-c]pyridine-1,3-dione 395352 (R)-2-(5-(2,3-difluorobenzylthio)-2-(methylamino)thiazolo[4,5-d]pyrimidin-7-ylamino)propan-1-ol 395353 (R)-2-(5-(2,3-difluorobenzylthio)-2-(diethylamino)thiazolo[4,5-d]pyrimidin-7-ylamino)propan-1-ol 395355 2-(5-(2,3-difluorobenzylthio)-2-(diethylamino)thiazolo[4,5-d]pyrimidin-7-ylamino)propane-1,3-diol 395365 (R)-2-(5-(2-fluorobenzylthio)-2-aminothiazolo[4,5-d]pyrimidin-7-ylamino)propan-1-ol 395367 (R)-2-(5-(3-fluorobenzylthio)-2-aminothiazolo[4,5-d]pyrimidin-7-ylamino)propan-1-ol 395368 (R)-2-(5-(2-chlorobenzylthio)-2-aminothiazolo[4,5-d]pyrimidin-7-ylamino)propan-1-ol 395369 (R)-2-(5-(3-chlorobenzylthio)-2-aminothiazolo[4,5-d]pyrimidin-7-ylamino)propan-1-ol 395370 (R)-2-(5-(3-chloro-2-fluorobenzylthio)-2-aminothiazolo[4,5-d]pyrimidin-7-ylamino)propan-1-ol 395371 (R)-2-(5-(2,3-dichlorobenzylthio)-2-aminothiazolo[4,5-d]pyrimidin-7-ylamino)propan-1-ol 395372 2-(2-amino-5-(furan-2-ylmethylthio)thiazolo[4,5-d]pyrimidin-7-ylamino)-2-methylpropan-1-ol 395373 (R)-2-(2-amino-5-(furan-2-ylmethylthio)thiazolo[4,5-d]pyrimidin-7-ylamino)propan-1-ol 395374 2-(2-amino-5-((2-methylthiazol-4-yl)methylthio)thiazolo[4,5-d]pyrimidin-7-ylamino)-2-methylpropan-1-ol 395375 (R)-2-(2-amino-5-((2-methylthiazol-4-yl)methylthio)thiazolo[4,5-d]pyrimidin-7-ylamino)propan-1-ol 395488 benzyl (S)-6-((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamido)-1-(benzylamino)-1-oxohexan-2-ylcarbamate 395495 (S)-N-((S)-5-acetamido-6-(benzylamino)-6-oxohexyl)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 395501 (S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-N-((S)-5-amino-6-(benzylamino)-6-oxohexyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 395502 benzyl (S)-6-((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamido)-1-oxo-1-(phenylamino)hexan-2-ylcarbamate 395503 (S)-N-((S)-5-acetamido-6-oxo-6-(phenylamino)hexyl)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 395504 (S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-N-((S)-5-amino-6-oxo-6-(phenylamino)hexyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 395506 benzyl (S)-5-((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamido)-1-(1H-benzo[d]imidazol-2-yl)pentylcarbamate 395508 (S)-N-((S)-5-acetamido-5-(1H-benzo[d]imidazol-2-yl)pentyl)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 395516 (S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-N-((S)-5-amino-5-(1H-benzo[d]imidazol-2-yl)pentyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 395640 (Z)-2-amino-5-(quinolin-6-ylmethylene)thiazol-4(5H)-one 395646 N,N-dimethyl-3-((phenethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 395648 dimethyl-{3-[(2-p-tolyl-ethylamino)-methyl]-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl}-amine 395649 3-((4-chlorophenethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 395651 3-((4-isopropylphenethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 395654 3-((2,6-dichlorophenethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 395655 3-((2-fluorophenethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 395657 (Z)-5-(quinolin-6-ylmethylene)-2-(thiophen-2-ylmethylamino)thiazol-4(5H)-one 395660 3-((cyclohexylmethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 395662 3-((2-cyclopentylethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 395663 3-((2-cyclohexylethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 395664 3-((2-cycloheptylethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 395665 {3-[(2-adamantan-1-yl-ethylamino)-methyl]-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl}-dimethyl-amine 395666 N,N-dimethyl-3-((2-(tetrahydro-2H-pyran-4-yl)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 395668 N,N-dimethyl-3-((2-(tetrahydropyran-4-ylidene)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 395669 N,N-dimethyl-3-((2-(tetrahydro-2H-thiopyran-4-yl)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 395670 3-((2-(3,6-dihydro-2H-thiopyran-4-yl)ethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 395672 4-(2-((3-(dimethylamino)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl)methylamino)ethyl)cyclohexanol 395674 (4-(2-((3-(dimethylamino)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl)methylamino)ethyl)cyclohexyl)methanol 395675 7-fluoro-N,N-dimethyl-3-((2-(tetrahydro-2H-pyran-4-yl)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 395677 7,8-dichloro-N,N-dimethyl-3-((2-(tetrahydro-2H-pyran-4-yl)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 395703 (R,Z)-2-(1-hydroxy-3-phenylpropan-2-ylamino)-5-(quinolin-6-ylmethylene)thiazol-4(5H)-one 395709 (Z)-2-((1R,2S)-2-phenylcyclopropylamino)-5-(quinolin-6-ylmethylene)thiazol-4(5H)-one 395762 N-(1-(2-chlorobenzyl)piperidin-4-yl)-1-naphthamide 395766 N-(1-(3-chlorobenzyl)piperidin-4-yl)-1-naphthamide 395767 N-(1-(4-chlorobenzyl)piperidin-4-yl)-1-naphthamide 395769 N-(1-(3-bromobenzyl)piperidin-4-yl)-1-naphthamide 395770 N-(1-(4-bromobenzyl)piperidin-4-yl)-1-naphthamide 395772 N-(1-(3-(trifluoromethyl)benzyl)piperidin-4-yl)-1-naphthamide 395774 N-(1-(4-(trifluoromethyl)benzyl)piperidin-4-yl)-1-naphthamide 395776 N-(1-(perfluorobenzyl)piperidin-4-yl)-1-naphthamide 395780 N-(1-(3-methoxybenzyl)piperidin-4-yl)-1-naphthamide 395782 N-(1-(4-methoxybenzyl)piperidin-4-yl)-1-naphthamide 395783 naphthalene-1-carboxylic acid [1-(2-methyl-benzyl)-piperidin-4-yl]-amide 395784 naphthalene-1-carboxylic acid [1-(3-methyl-benzyl)-piperidin-4-yl]-amide 395787 naphthalene-1-carboxylic acid [1-(4-methyl-benzyl)-piperidin-4-yl]-amide 395789 N-(1-(2-chlorobenzyl)piperidin-4-yl)-2-naphthamide 395790 N-(1-(3-chlorobenzyl)piperidin-4-yl)-2-naphthamide 395791 N-(1-(4-chlorobenzyl)piperidin-4-yl)-2-naphthamide 395793 N-(1-(3-bromobenzyl)piperidin-4-yl)-2-naphthamide 395794 N-(1-(4-bromobenzyl)piperidin-4-yl)-2-naphthamide 395795 N-(1-(3-(trifluoromethyl)benzyl)piperidin-4-yl)-2-naphthamide 395796 N-(1-(4-(trifluoromethyl)benzyl)piperidin-4-yl)-2-naphthamide 395798 N-(1-(4-nitrobenzyl)piperidin-4-yl)-2-naphthamide 395799 N-(1-(3-methoxybenzyl)piperidin-4-yl)-2-naphthamide 395800 N-(1-(4-methoxybenzyl)piperidin-4-yl)-2-naphthamide 395801 naphthalene-2-carboxylic acid [1-(2-methyl-benzyl)-piperidin-4-yl]-amide 395802 naphthalene-2-carboxylic acid [1-(3-methyl-benzyl)-piperidin-4-yl]-amide 395803 naphthalene-2-carboxylic acid [1-(4-methyl-benzyl)-piperidin-4-yl]-amide 395805 N-(1-(pyridin-2-ylmethyl)piperidin-4-yl)-2-naphthamide 395807 N-(1-(pyridin-3-ylmethyl)piperidin-4-yl)-2-naphthamide 395808 N-(1-(pyridin-4-ylmethyl)piperidin-4-yl)-2-naphthamide 395876 (2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-2-benzyl-5-(3-carbamimidamidopropyl)-8-(1H-indol-3-ylmethyl)-3,6,9,17,20,31-hexaoxo-1,4,7,10,16,21-hexaazatricyclo[20.8.1.0^{24,29}]hentriaconta-24(29),25,27-triene-11-carboxamide 395880 (2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-5-(3-carbamimidamidopropyl)-2-[(4-chlorophenyl)methyl]-8-(1H-indol-3-ylmethyl)-3,6,9,17,20,31-hexaoxo-1,4,7,10,16,21-hexaazatricyclo[20.8.1.0^{24,29}]hentriaconta-24(29),25,27-triene-11-carboxamide 395885 (2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-5-(3-carbamimidamidopropyl)-8-(1H-indol-3-ylmethyl)-2-(naphthalen-2-ylmethyl)-3,6,9,17,20,31-hexaoxo-1,4,7,10,16,21-hexaazatricyclo[20.8.1.0^{24,29}]hentriaconta-24(29),25,27-triene-11-carboxamide 395888 (3S,6S,9R,12S,15S,23S)-15-[(2S)-2-aminohexanamido]-6-(3-carbamimidamidopropyl)-12-(1H-imidazol-5-ylmethyl)-3-(1H-indol-3-ylmethyl)-9-(naphthalen-2-ylmethyl)-2,5,8,11,14,17-hexaoxo-1,4,7,10,13,18-hexaazacyclotricosane-23-carboxamide 395931 1-(2-((R)-4-(6-fluoronaphthalen-1-yl)-2-methylpiperazin-1-yl)ethyl)-3,4-dihydro-1H-isochromene-6-carboxamide 395932 (S)-1-(2-((R)-4-(6-fluoronaphthalen-1-yl)-2-methylpiperazin-1-yl)ethyl)-3,4-dihydro-1H-isochromene-6-carboxamide 395933 (R)-1-(2-((R)-4-(6-fluoronaphthalen-1-yl)-2-methylpiperazin-1-yl)ethyl)-3,4-dihydro-1H-isochromene-6-carboxamide 395934 (S)-1-(2-((S)-4-(6-fluoronaphthalen-2-yl)-2-methylpiperazin-1-yl)ethyl)isochroman-6-carboxamide 395935 (S)-1-(2-(4-(6-fluoronaphthalen-2-yl)piperazin-1-yl)ethyl)isochroman-6-carboxamide 395936 (S)-1-(2-((S)-4-(6-cyanonaphthalen-1-yl)-2-methylpiperazin-1-yl)ethyl)-3,4-dihydro-1H-isochromene-6-carboxamide 395937 (S)-1-(2-(4-(6-cyanonaphthalen-1-yl)piperazin-1-yl)ethyl)-3,4-dihydro-1H-isochromene-6-carboxamide 395953 N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 395954 N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 395955 2-cyano-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 395956 2-cyano-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 395957 2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 395958 2-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 395959 N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-nitrobenzenesulfonamide 395960 N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-nitrobenzenesulfonamide 395963 N-(3-(5-fluoro-1H-indol-3-yl)propyl)-5-methoxy-3,4-dihydro-2H-chromen-3-amine 395964 N-(3-(5-fluoro-1H-indol-3-yl)propyl)-2,3-dihydro-1H-pyrano[3,2-f]quinolin-2-amine 395965 3-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 395966 3-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 395968 N-(3-(5-fluoro-1H-indol-3-yl)propyl)-N-propyl-2,3-dihydro-1H-pyrano[3,2-f]quinolin-2-amine 395969 N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(trifluoromethyl)benzenesulfonamide 395970 N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(trifluoromethyl)benzenesulfonamide 395971 4-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 395972 4-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 395973 N-(2-(5-fluoro-1H-indol-3-yl)ethyl)-2,3-dihydro-1H-pyrano[3,2-f]quinolin-2-amine 395974 N-(2-(5-fluoro-1H-indol-3-yl)ethyl)-N-propyl-2,3-dihydro-1H-pyrano[3,2-f]quinolin-2-amine 395975 N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(methylsulfonyl)benzenesulfonamide 395976 N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(methylsulfonyl)benzenesulfonamide 395978 N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(trifluoromethoxy)benzenesulfonamide 395980 N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(trifluoromethoxy)benzenesulfonamide 395982 N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide 395984 N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide 395985 N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2,5-dimethoxybenzenesulfonamide 395986 N-(3-(5-fluoro-1H-indol-3-yl)propyl)-3,4-dihydro-2H-pyrano[2,3-f]quinolin-3-amine 395987 N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2,5-dimethoxybenzenesulfonamide 395989 N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-methylbenzenesulfonamide 395993 N-(3-(5-fluoro-1H-indol-3-yl)propyl)-N-propyl-3,4-dihydro-2H-pyrano[2,3-f]quinolin-3-amine 395996 N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-methylbenzenesulfonamide 396000 N-(4-(5-fluoro-1H-indol-3-yl)butyl)-3,4-dihydro-2H-pyrano[2,3-f]quinolin-3-amine 396002 5-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 396005 5-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 396006 N-(4-(5-fluoro-1H-indol-3-yl)butyl)-N-propyl-3,4-dihydro-2H-pyrano[2,3-f]quinolin-3-amine 396008 5-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 396010 5-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 396019 5-bromo-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 396020 5-bromo-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 396023 N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-(trifluoromethyl)benzenesulfonamide 396026 N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-(trifluoromethyl)benzenesulfonamide 396028 N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-nitrobenzenesulfonamide 396031 N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-nitrobenzenesulfonamide 396035 3-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methylbenzenesulfonamide 396036 3-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methylbenzenesulfonamide 396039 2,4-dichloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 396042 2,4-dichloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 396045 3-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 396049 3-chloro-2-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 396050 4-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 396051 4-chloro-2-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 396052 5-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 396054 N-((1s,4s)-4-(4-(2-(cyclopropylmethoxy)phenyl)piperazin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide 396056 5-chloro-N-((1s,4s)-4-(4-(2-(cyclopropylmethoxy)phenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 396058 5-chloro-N-((1s,4s)-4-(4-(2-(cyclopropylmethoxy)phenyl)piperazin-1-yl)cyclohexyl)-2-fluorobenzenesulfonamide 396060 N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)(phenyl)methanesulfonamide 396061 N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)(phenyl)methanesulfonamide 396062 N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide 396063 N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide 396064 N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methoxypyridine-3-sulfonamide 396066 N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methoxypyridine-3-sulfonamide 396067 5-bromo-6-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide 396070 5-bromo-6-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide 396149 2-fluorophenyl 6-(2-methyl-4,5-diphenyl-1H-imidazol-1-yl)hexylcarbamate 396209 [8-((R)-2-amino-propyl)-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']difuran-4-yl]-methanol 396210 (R)-2-(8-methoxymethyl-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']difuran-4-yl)-1-methyl-ethylamine 396211 (R)-2-[8-(2-methoxy-ethoxymethyl)-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']difuran-4-yl]-1-methyl-ethylamine 396212 [8-((R)-2-amino-propyl)-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']difuran-4-ylmethoxy]-acetic acid phenyl ester 396213 8-((R)-2-amino-propyl)-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']difuran-4-carboxylic acid methyl ester 396214 3-[8-((R)-2-amino-propyl)-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']difuran-4-yl]-propionic acid methyl ester 396215 [8-((R)-2-amino-propyl)-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']difuran-4-yl]-acetic acid 396220 3-[8-((R)-2-amino-propyl)-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']difuran-4-yl]-propionic acid 396221 (R)-1-methyl-2-[8-(3-methyl-[1,2,4]oxadiazol-5-yl)-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']difuran-4-yl]-ethylamine 396222 (R)-1-methyl-2-[8-(3-methyl-[1,2,4]oxadiazol-5-ylmethyl)-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']difuran-4-yl]-ethylamine 396223 (R)-1-methyl-2-{8-[2-(3-methyl-[1,2,4]oxadiazol-5-yl)-ethyl]-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']difuran-4-yl}-ethylamine 396224 (R)-1-methyl-2-[8-(3-methyl-[1,2,4]oxadiazol-5-ylmethyl)-benzo[1,2-b;4,5-b']difuran-4-yl]-ethylamine 396225 [8-((R)-2-amino-propyl)-benzo[1,2-b;4,5-b']difuran-4-yl]-methanol 396226 (R)-2-(8-methoxymethyl-benzo[1,2-b;4,5-b']difuran-4-yl)-1-methyl-ethylamine 396227 (1S,2R)-2-amino-1-(8-bromo-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']difuran-4-yl)-propan-1-ol 396228 (1R,2R)-2-amino-1-(8-bromo-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']difuran-4-yl)-propan-1-ol 396241 [2-(2',6'-dimethoxy-biphenyl-3-yl)-ethyl]-dimethyl-amine 396242 N,N-dimethyl-2-(2'-methylbiphenyl-3-yl)ethanamine 396243 [2-(2'-methoxy-biphenyl-3-yl)-ethyl]-dimethyl-amine 396244 [2-(2',6'-dimethyl-biphenyl-3-yl)-ethyl]-dimethyl-amine 396250 2-(2'-methyl-biphenyl-3-yl)-ethylamine 396330 8-bromo-4-(3-chloro-4-fluorophenylamino)-6-[(2-methyl-2Hpyrazol-3-ylmethyl)amino]quinoline-3-carbonitrile 396331 8-chloro-4-[(3-chloro-4-fluorophenyl)amino]-6-{[(1-methyl-1H-imidazol-5-yl)methyl]amino}quinoline-3-carbonitrile 396366 1-benzhydryl-4-(2H-1lambda*4*-thiazol-2-yl)-piperidin-4-ol 396367 2-cyclohexyl-N-[1-(3-pyridin-3-yl-propionyl)-piperidin-4-yl]-2-(2H-1lambda*4*-thiophen-3-yl)-acetamide 396368 2-{4-methoxy-3-[2-(4-methyl-pyridin-1-yl)-ethoxy]-phenyl}-7-methyl-2,3-dihydro-isoindol-1-one 396388 LRHYLNLLTRQRY-NH2 396389 (S)-2-((S)-2-((2S,3R)-2-((S)-2-((S)-2-((S)-2-((S)-2-((S)-2-((S)-2-((S)-2-((S)-2-acetamido-4-methylpentanamido)-5-guanidinopentanamido)-3-(1H-imidazol-5-yl)propanamido)-3-(4-hydroxyphenyl)propanamido)-4-methylpentanamido)-4-amino-4-oxobutanamido)-4-methylp 396390 (S)-2-((S)-2-((2S,3R)-2-((S)-2-((S)-2-((S)-2-((S)-2-((S)-2-((S)-2-((S)-2-((S)-2-((R)-2-acetamido-3-mercaptopropanamido)-4-methylpentanamido)-5-guanidinopentanamido)-3-(1H-imidazol-5-yl)propanamido)-3-(4-hydroxyphenyl)propanamido)-4-methylpentanamido)-4-am 396492 (2-(4-chlorobenzyloxy)-5-bromophenyl)methanamine 396493 N-(2-(4-chlorobenzyloxy)-5-bromobenzyl)ethanamine 396495 (2-(4-chlorobenzyloxy)-5-bromophenyl)-N,N-dimethylmethanamine 396500 N-(2-(4-chlorobenzyloxy)-5-bromobenzyl)-N-ethylethanamine 396569 4-(1-hexyl-cyclopropyl)-3',5'-dimethyl-biphenyl-2-ol 396570 4-(1-hexyl-cyclopentyl)-3',5'-dimethyl-biphenyl-2-ol 396571 N-(2-(4-chlorobenzyloxy)-5-bromobenzyl)-N-methyl(phenyl)methanamine 396572 4-(1-hexyl-cyclohexyl)-3',5'-dimethyl-biphenyl-2-ol 396574 1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)pyrrolidine 396576 4-(2-(4-chlorobenzyloxy)-5-bromobenzyl)morpholine 396578 2-(2-hydroxy-3',5'-dimethyl-biphenyl-4-yl)-2-methyl-propionic acid methyl ester 396582 4-(2-hydroxy-3',5'-dimethyl-biphenyl-4-yl)-4-methyl-pentanoic acid methyl ester 396586 1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)piperidin-4-one 396587 6-(2-hydroxy-3',5'-dimethyl-biphenyl-4-yl)-6-methyl-heptanoic acid methyl ester 396588 1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)pyrrolidin-3-ol 396589 1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)piperidin-4-ol 396593 1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)piperidin-3-ol 396596 1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)-4-ethoxypiperidine 396597 4-(2-hydroxy-1,1-dimethyl-ethyl)-3',5'-dimethyl-biphenyl-2-ol 396598 1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)-4-fluoropiperidine 396599 1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)piperidin-4-amine 396600 4-(4-hydroxy-1,1-dimethyl-butyl)-3',5'-dimethyl-biphenyl-2-ol 396601 1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)-N-ethylpiperidin-4-amine 396602 4-(6-hydroxy-1,1-dimethyl-hexyl)-3',5'-dimethyl-biphenyl-2-ol 396604 N-(1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)piperidin-4-yl)acetamide 396605 4-(2-hydroxy-3',5'-dimethyl-biphenyl-4-yl)-4-methyl-pentanoic acid methylamide 396606 methyl 1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)piperidin-4-ylcarbamate 396607 6-(2-hydroxy-3',5'-dimethyl-biphenyl-4-yl)-6-methyl-heptanoic acid methylamide 396608 (1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)piperidin-4-yl)methanamine 396609 1-(1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)piperidin-4-yl)piperazine 396610 4-(1,1-dimethyl-heptyl)-2',6'-dimethyl-biphenyl-2-ol 396611 4-(1,1-dimethyl-heptyl)-2',5'-dimethyl-biphenyl-2-ol 396612 ethyl 1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)piperidine-4-carboxylate 396613 4-(1,1-dimethyl-heptyl)-2',3'-dimethyl-biphenyl-2-ol 396614 1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)piperidine-4-carboxylic acid 396615 4-(1,1-dimethyl-heptyl)-3',4'-dimethyl-biphenyl-2-ol 396616 4-(1,1-dimethyl-heptyl)-2'-methoxy-biphenyl-2-ol 396617 1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)-4-(trifluoromethyl)piperidin-4-ol 396618 4-(1,1-dimethyl-heptyl)-2',3'-dimethoxy-biphenyl-2-ol 396619 1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)-4-(4-bromophenyl)piperidin-4-ol 396620 4-(1,1-dimethyl-heptyl)-3'-methoxy-biphenyl-2-ol 396621 1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)-4-(aminomethyl)piperidin-4-ol 396622 4-(1,1-dimethyl-heptyl)-3',4'-dimethoxy-biphenyl-2-ol 396623 2'-amino-4-(1,1-dimethyl-heptyl)-biphenyl-2-ol 396624 1-[5-bromo-2-(4-chloro-benzyloxy)-benzyl]-4-(4-hydroxy-piperidin-1-ylmethyl)-piperidin-4-ol 396625 3'-amino-4-(1,1-dimethyl-heptyl)-biphenyl-2-ol 396626 1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)-4-((4-methylpiperazin-1-yl)methyl)piperidin-4-ol 396627 4'-amino-4-(1,1-dimethyl-heptyl)-biphenyl-2-ol 396628 1-((1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)-4-hydroxypiperidin-4-yl)methyl)-3-(4-fluorophenyl)urea 396629 4'-(1,1-dimethyl-heptyl)-2'-hydroxy-biphenyl-3-carbonitrile 396630 1-((1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)-4-hydroxypiperidin-4-yl)methyl)-3-(2,6-difluorophenyl)urea 396631 1-((1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)-4-hydroxypiperidin-4-yl)methyl)-3-(2,6-dichlorophenyl)urea 396634 1-((1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)-4-hydroxypiperidin-4-yl)methyl)-3-(2,4,6-trichlorophenyl)urea 396635 5-(1,1-dimethyl-heptyl)-2-pyridin-3-yl-phenol 396636 1-((1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)-4-hydroxypiperidin-4-yl)methyl)-3-(4-bromo-2,6-dimethylphenyl)urea 396637 1-((1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)-4-hydroxypiperidin-4-yl)methyl)-3-mesitylurea 396638 4-(1,1-dimethyl-heptyl)-2-methoxy-3',5'-dimethyl-biphenyl 396639 1-((1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)-4-hydroxypiperidin-4-yl)methyl)-3-(2,6-dimethylphenyl)urea 396640 1-((1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)-4-hydroxypiperidin-4-yl)methyl)-3-(2,6-diethylphenyl)urea 396645 4-(1,1-dimethyl-heptyl)-3',5'-dimethyl-biphenyl-2-ylamine 396646 1-((1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)-4-hydroxypiperidin-4-yl)methyl)-3-(2,6-diisopropylphenyl)urea 396648 1-((1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)-4-hydroxypiperidin-4-yl)methyl)-3-(2,6-dimethoxyphenyl)urea 396649 4-(1,1-dimethyl-heptyl)-3',5'-dimethyl-biphenyl-2-carboxylic acid methyl ester 396651 4-(1,1-dimethyl-heptyl)-3',5'-dimethyl-biphenyl-2-carboxylic acid amide 396658 [4-(1,1-dimethyl-heptyl)-3',5'-dimethyl-biphenyl-2-yl]-methanol 396662 c-[4-(1,1-dimethyl-heptyl)-3',5'-dimethyl-biphenyl-2-yl]-methylamine 396665 morpholin-4-yl-acetic acid 4-(1,1-dimethyl-heptyl)-3',5'-dimethyl-biphenyl-2-ylmethyl ester 396667 4-[4-(1,1-dimethyl-heptyl)-3',5'-dimethyl-biphenyl-2-ylmethyl]-morpholine 397165 (Z)-methyl 2-(2-isopropylphenylimino)-5,5-dimethyl-1,3-thiazinane-3-carbodithioate 397170 (Z)-methyl 5,5-diethyl-2-(2-isopropylphenylimino)-1,3-thiazinane-3-carbodithioate 397173 6-[(Z)-2-isopropyl-phenylimino]-5-thia-7-aza-spiro[2.5]octane-7-carbodithioic acid methyl ester 397177 8-[(Z)-2-isopropyl-phenylimino]-7-thia-9-aza-spiro[4.5]decane-9-carbodithioic acid methyl ester 397179 3-[(Z)-2-isopropyl-phenylimino]-2-thia-4-aza-spiro[5.5]undecane-4-carbodithioic acid methyl ester 397181 3-[(Z)-3-isopropyl-phenylimino]-2-thia-4-aza-spiro[5.5]undecane-4-carbodithioic acid methyl ester 397184 3-[(Z)-4-isopropyl-phenylimino]-2-thia-4-aza-spiro[5.5]undecane-4-carbodithioic acid methyl ester 397185 3-[(Z)-2-methoxy-phenylimino]-2-thia-4-aza-spiro[5.5]undecane-4-carbodithioic acid methyl ester 397186 3-[(Z)-3-methoxy-phenylimino]-2-thia-4-aza-spiro[5.5]undecane-4-carbodithioic acid methyl ester 397187 3-[(Z)-4-methoxy-phenylimino]-2-thia-4-aza-spiro[5.5]undecane-4-carbodithioic acid methyl ester 397188 3-[(Z)-4-ethyl-phenylimino]-2-thia-4-aza-spiro[5.5]undecane-4-carbodithioic acid methyl ester 397189 3-[(Z)-4-propyl-phenylimino]-2-thia-4-aza-spiro[5.5]undecane-4-carbodithioic acid methyl ester 397190 3-[(Z)-4-trifluoromethyl-phenylimino]-2-thia-4-aza-spiro[5.5]undecane-4-carbodithioic acid methyl ester 397191 3-[(Z)-4-trifluoromethoxy-phenylimino]-2-thia-4-aza-spiro[5.5]undecane-4-carbodithioic acid methyl ester 397192 3-[(Z)-4-cyano-phenylimino]-2-thia-4-aza-spiro[5.5]undecane-4-carbodithioic acid methyl ester 397193 3-[(Z)-2-ethoxy-phenylimino]-2-thia-4-aza-spiro[5.5]undecane-4-carbodithioic acid methyl ester 397194 3-[(Z)-2-trifluoromethyl-phenylimino]-2-thia-4-aza-spiro[5.5]undecane-4-carbodithioic acid methyl ester 397195 3-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-N-(methylsulfonyl)benzamide 397196 3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-N-(phenylsulfonyl)benzamide 397197 3-(2-(2-(benzyloxy)phenyl)-5-methyl-1H-pyrrol-1-yl)-N-(phenylsulfonyl)benzamide 397198 3-(2-(2-(benzyloxy)phenyl)-5-methyl-1H-pyrrol-1-yl)-N-(3,5-dimethylisoxazol-4-ylsulfonyl)benzamide 397199 N-(3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)phenylsulfonyl)benzamide 397200 N-(4-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)phenylsulfonyl)benzamide 397201 2-(3-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)phenyl)-1,1,1,3,3,3-hexafluoropropan-2-ol 397203 2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1-(3-(methylsulfonyl)phenyl)-1H-pyrrole 397204 2-(2-(benzyloxy)-5-bromophenyl)-5-methyl-1-(3-(methylsulfonyl)phenyl)-1H-pyrrole 397205 2-(2-(benzyloxy)phenyl)-5-methyl-1-(4-(methylsulfonyl)phenyl)-1H-pyrrole 397206 2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1-(4-(methylsulfonyl)phenyl)-1H-pyrrole 397207 2-(2-(benzyloxy)-5-bromophenyl)-5-methyl-1-(4-(methylsulfonyl)phenyl)-1H-pyrrole 397208 4-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)benzenesulfonamide 397209 4-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzamide 397210 4-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-N-methylbenzamide 397211 3-[(Z)-2-trifluoromethoxy-phenylimino]-2-thia-4-aza-spiro[5.5]undecane-4-carbodithioic acid methyl ester 397212 4-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-N,N-dimethylbenzamide 397213 3-[(Z)-2,3-dimethyl-phenylimino]-2-thia-4-aza-spiro[5.5]undecane-4-carbodithioic acid methyl ester 397214 4-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-N,N-diethylbenzamide 397215 4-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-N-tert-butylbenzamide 397216 3-[(Z)-indan-4-ylimino]-2-thia-4-aza-spiro[5.5]undecane-4-carbodithioic acid methyl ester 397217 N-benzyl-4-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)benzamide 397218 3-[(Z)-5,6,7,8-tetrahydro-naphthalen-1-ylimino]-2-thia-4-aza-spiro[5.5]undecane-4-carbodithioic acid methyl ester 397219 4-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-N-(pyridin-2-ylmethyl)benzamide 397220 3-[(Z)-5,6,7,8-tetrahydro-naphthalen-2-ylimino]-2-thia-4-aza-spiro[5.5]undecane-4-carbodithioic acid methyl ester 397221 4-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-N-(pyridin-3-ylmethyl)benzamide 397222 methyl 3-(naphthalen-1-ylimino)-2-thia-4-azaspiro[5.5]undecane-4-carbodithioate 397223 3-[(Z)-quinolin-5-ylimino]-2-thia-4-aza-spiro[5.5]undecane-4-carbodithioic acid methyl ester 397224 3-[(Z)-benzo[1,2,5]thiadiazol-4-ylimino]-2-thia-4-aza-spiro[5.5]undecane-4-carbodithioic acid methyl ester 397225 4-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-N-(pyridin-4-ylmethyl)benzamide 397226 3-[(Z)-benzo[1,2,5]oxadiazol-4-ylimino]-2-thia-4-aza-spiro[5.5]undecane-4-carbodithioic acid methyl ester 397227 4-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-N-((S)-1-phenylethyl)benzamide 397228 3-[(Z)-1-methyl-1,2,3,4-tetrahydro-quinolin-5-ylimino]-2-thia-4-aza-spiro[5.5]undecane-4-carbodithioic acid methyl ester 397229 3-(2-(2-(2,4-difluorobenzyloxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzamide 397230 3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)benzamide 397231 3-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-N-methylbenzamide 397232 3-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-N,N-dimethylbenzamide 397233 3-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)-N-phenylbenzamide 397235 N-benzyl-3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)benzamide 397236 3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-N-(pyridin-2-ylmethyl)benzamide 397237 3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-N-(pyridin-3-ylmethyl)benzamide 397240 3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-N-(pyridin-4-ylmethyl)benzamide 397241 3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-N-((S)-1-phenylethyl)benzamide 397245 3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-N-((R)-1-phenylethyl)benzamide 397246 4-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-N-((R)-1-phenylethyl)benzamide 397247 6-(2-(2-(2,4-difluorobenzyloxy)phenyl)-5-methyl-1H-pyrrol-1-yl)-1H-benzo[d][1,2,3]triazole 397248 6-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-1H-benzo[d][1,2,3]triazole 397249 6-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-1H-indazole 397250 5-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-1H-indazole 397251 3-(3-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)phenyl)pyridine 397252 2-(3-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)phenyl)pyridine 397253 2-(3-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)phenyl)pyrimidine 397254 2-(3-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)phenyl)-1H-benzo[d]imidazole 397255 2-(3-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)phenyl)-5-methyl-1,3,4-oxadiazole 397257 3-(3-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)phenyl)-5-methyl-1,2,4-oxadiazole 397260 N-(3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)phenyl)acetamide 397263 7-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)-4-methylquinolin-2(1H)-one 397264 5-(4-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)phenyl)-1H-imidazole 397265 1-(4-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)phenyl)-1H-1,2,4-triazole 397266 5-(2-(2-(2,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)isoindoline-1,3-dione 397275 7-chloro-1,1-dioxo-3-phenylamino-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397276 7-chloro-3-(2-fluoro-phenylamino)-1,1-dioxo-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397278 7-chloro-3-(2-chloro-phenylamino)-1,1-dioxo-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397279 3-(2-bromo-phenylamino)-7-chloro-1,1-dioxo-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397281 3-(3-bromo-phenylamino)-7-chloro-1,1-dioxo-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397284 3-(4-bromo-phenylamino)-7-chloro-1,1-dioxo-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397285 7-chloro-3-(2-chloro-3-fluoro-phenylamino)-1,1-dioxo-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397286 3-(2-bromo-4-fluoro-phenylamino)-7-chloro-1,1-dioxo-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397287 3-(2-bromo-5-fluoro-phenylamino)-7-chloro-1,1-dioxo-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397289 3-(2-bromo-6-fluoro-phenylamino)-7-chloro-1,1-dioxo-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397292 7-chloro-1,1-dioxo-3-o-tolylamino-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397294 3-(biphenyl-2-ylamino)-7-chloro-1,1-dioxo-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397319 7-chloro-3-(2-methoxy-phenylamino)-1,1-dioxo-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397320 7-chloro-1,1-dioxo-3-(2-phenoxy-phenylamino)-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397321 7-chloro-1,1-dioxo-3-(2-trifluoromethyl-phenylamino)-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397322 7-chloro-1,1-dioxo-3-(2-trifluoromethoxy-phenylamino)-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397324 1-[2-(7-chloro-5-hydroxy-1,1-dioxo-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-3-ylamino)-phenyl]-ethanone 397326 3-(2-chloro-phenylamino)-1,1-dioxo-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397327 3-(2-bromo-phenylamino)-7-fluoro-1,1-dioxo-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397329 rac-5-(3'-acetylamino-biphenyl-4-ylmethyl)-oxazole-4-carboxylic acid (2-phenyl-propyl)-amide 397330 7-bromo-3-(2-bromo-phenylamino)-1,1-dioxo-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397334 5-(3'-acetylamino-biphenyl-4-ylmethyl)-oxazole-4-carboxylic acid benzylamide 397337 5-(3'-acetylamino-biphenyl-4-ylmethyl)-oxazole-4-carboxylic acid phenethyl-amide 397345 rac-5-(3'-acetylamino-biphenyl-4-ylmethyl)-oxazole-4-carboxylic acid (1-phenyl-ethyl)-amide 397347 5-(3'-acetylamino-biphenyl-4-ylmethyl)-oxazole-4-carboxylic acid methyl-phenethyl-amide 397351 5-(3'-acetylamino-biphenyl-4-ylmethyl)-oxazole-4-carboxylic acid ((1S,2R)-2-phenyl-cyclopropyl)-amide 397353 5-(3'-acetylamino-biphenyl-4-ylmethyl)-oxazole-4-carboxylic acid ((R)-2-phenyl-propyl)-amide 397357 5-(3'-acetylamino-biphenyl-4-ylmethyl)-oxazole-4-carboxylic acid ((S)-2-phenyl-propyl)-amide 397358 (R)-2-{[5-(3'-acetylamino-biphenyl-4-ylmethyl)-oxazole-4-carbonyl]-amino}-3-phenyl-propionic acid 397359 (S)-2-{[5-(3'-acetylamino-biphenyl-4-ylmethyl)-oxazole-4-carbonyl]-amino}-3-phenyl-propionic acid 397361 5-(3'-acetylamino-biphenyl-4-ylmethyl)-oxazole-4-carboxylic acid (2-pyridin-2-yl-ethyl)-amide 397364 5-(3'-acetylamino-biphenyl-4-ylmethyl)-oxazole-4-carboxylic acid (2-pyridin-3-yl-ethyl)-amide 397367 3-(2-bromo-phenylamino)-7-nitro-1,1-dioxo-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397368 5-(3'-acetylamino-biphenyl-4-ylmethyl)-oxazole-4-carboxylic acid (2-pyridin-4-yl-ethyl)-amide 397374 5-(3'-acetylamino-biphenyl-4-ylmethyl)-oxazole-4-carboxylic acid phenylamide 397376 5-(3'-acetylamino-biphenyl-4-ylmethyl)-oxazole-4-carboxylic acid methylamide 397377 5-(3'-acetylamino-biphenyl-4-ylmethyl)-oxazole-4-carboxylic acid dimethylamide 397378 5-(3'-acetylamino-biphenyl-4-ylmethyl)-oxazole-4-carboxylic acid (2-dimethylamino-ethyl)-amide 397379 3-(2-bromo-phenylamino)-7-methyl-1,1-dioxo-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397380 3-(2-bromo-phenylamino)-8-fluoro-1,1-dioxo-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397381 3-(2-bromo-phenylamino)-8-chloro-1,1-dioxo-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397382 7-nitro-1,1-dioxo-3-(2-phenoxy-phenylamino)-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397384 3-(2-chloro-phenylamino)-7-nitro-1,1-dioxo-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397393 3-benzylamino-7-chloro-1,1-dioxo-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397399 3-((R)-sec-butylamino)-7-chloro-1,1-dioxo-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397400 7-chloro-3-cyclopentylamino-1,1-dioxo-1,4-dihydro-1lambda6-benzo[1,2,4]thiadiazin-5-ol 397543 1-(4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidin-1-yl)ethanone 397544 1-(4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidin-1-yl)propan-1-one 397545 1-(4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidin-1-yl)-2-methylpropan-1-one 397546 (4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidin-1-yl)(cyclopropyl)methanone 397547 1-(4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidin-1-yl)-2,2-dimethylpropan-1-one 397548 1-(4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidin-1-yl)-2-methoxyethanone 397549 1-(4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidin-1-yl)-2-phenylethanone 397550 (4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidin-1-yl)(phenyl)methanone 397551 (4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidin-1-yl)(3,5-dimethylphenyl)methanone 397552 (4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidin-1-yl)(mesityl)methanone 397553 (3,5-bis(trifluoromethyl)phenyl)(4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidin-1-yl)methanone 397554 2-methoxy-1-(4-phenyl-4-(1-(1-phenylethyl)-1H-imidazol-2-yl)piperidin-1-yl)ethanone 397568 methyl 4-((2-(1-(2-methoxyacetyl)-4-phenylpiperidin-4-yl)-1H-imidazol-1-yl)methyl)benzoate 397570 phenyl(4-phenyl-4-(1-(1-phenylethyl)-1H-imidazol-2-yl)piperidin-1-yl)methanone 397574 methyl 3-((2-(1-benzoyl-4-phenylpiperidin-4-yl)-1H-imidazol-1-yl)methyl)benzoate 397578 methyl 4-((2-(1-benzoyl-4-phenylpiperidin-4-yl)-1H-imidazol-1-yl)methyl)benzoate 397581 4-((2-(1-benzoyl-4-phenylpiperidin-4-yl)-1H-imidazol-1-yl)methyl)-N,N-diethylbenzamide 397583 methyl 4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidine-1-carboxylate 397585 ethyl 4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidine-1-carboxylate 397589 propyl 4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidine-1-carboxylate 397591 butyl 4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidine-1-carboxylate 397593 isopropyl 4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidine-1-carboxylate 397594 cyclohexyl 4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidine-1-carboxylate 397601 tert-butyl 4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidine-1-carboxylate 397603 benzyl 4-(1-benzyl-1H-imidazol-2-yl)-4-phenylpiperidine-1-carboxylate 397604 ethyl 4-phenyl-4-(1-(1-phenylethyl)-1H-imidazol-2-yl)piperidine-1-carboxylate 397607 ethyl 4-(1-(3-methoxybenzyl)-1H-imidazol-2-yl)-4-phenylpiperidine-1-carboxylate 397610 ethyl 4-(1-(4-methoxybenzyl)-1H-imidazol-2-yl)-4-phenylpiperidine-1-carboxylate 397613 ethyl 4-(1-(3-fluorobenzyl)-1H-imidazol-2-yl)-4-phenylpiperidine-1-carboxylate 397616 ethyl 4-(1-(4-fluorobenzyl)-1H-imidazol-2-yl)-4-phenylpiperidine-1-carboxylate 397620 ethyl 4-(1-(4-hydroxybenzyl)-1H-imidazol-2-yl)-4-phenylpiperidine-1-carboxylate 397624 ethyl 4-(1-(4-(methoxycarbonyl)benzyl)-1H-imidazol-2-yl)-4-phenylpiperidine-1-carboxylate 397627 ethyl 4-(1-(1-methylnaphthalen-2-yl)-1H-imidazol-2-yl)-4-phenylpiperidine-1-carboxylate 397636 ethyl 4-(1-(cyclohexylmethyl)-1H-imidazol-2-yl)-4-phenylpiperidine-1-carboxylate 397637 (E)-ethyl 4-(1-cinnamyl-1H-imidazol-2-yl)-4-phenylpiperidine-1-carboxylate 397656 (S)-1-(2-(3,5-dimethylphenyl)-3-(1-(2-(pyridin-4-yl)ethylamino)propan-2-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-5(4H)-yl)ethanone 397657 (S)-cyclopentyl(2-(3,5-dimethylphenyl)-3-(1-(2-(pyridin-4-yl)ethylamino)propan-2-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-5(4H)-yl)methanone 397663 (S)-(2-(3,5-dimethylphenyl)-3-(1-(2-(pyridin-4-yl)ethylamino)propan-2-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-5(4H)-yl)(2,2,3,3-tetramethylcyclopropyl)methanone 397664 adamantan-1-yl-{2-(3,5-dimethyl-phenyl)-3-[(S)-1-methyl-2-(2-pyridin-4-yl-ethylamino)-ethyl]-1,4,6,7-tetrahydro-pyrrolo[3,2-c]pyridin-5-yl}-methanone 397665 (S)-(2-(3,5-dimethylphenyl)-3-(1-(2-(pyridin-4-yl)ethylamino)propan-2-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-5(4H)-yl)(phenyl)methanone 397666 (S)-1-(2-(3,5-dimethylphenyl)-3-(1-(2-(pyridin-4-yl)ethylamino)propan-2-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-5(4H)-yl)-2-phenylethanone 397667 (S)-1-(2-(3,5-dimethylphenyl)-3-(1-(2-(pyridin-4-yl)ethylamino)propan-2-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-5(4H)-yl)-2-(2-methoxyphenyl)ethanone 397669 (S)-1-(2-(3,5-dimethylphenyl)-3-(1-(2-(pyridin-4-yl)ethylamino)propan-2-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-5(4H)-yl)-2-(2-fluorophenyl)ethanone 397670 (S)-2-(2-chlorophenyl)-1-(2-(3,5-dimethylphenyl)-3-(1-(2-(pyridin-4-yl)ethylamino)propan-2-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-5(4H)-yl)ethanone 397671 (S)-1-(2-(3,5-dimethylphenyl)-3-(1-(2-(pyridin-4-yl)ethylamino)propan-2-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-5(4H)-yl)-2-(2-(trifluoromethyl)phenyl)ethanone 397674 (S)-1-(2-(3,5-dimethylphenyl)-3-(1-(2-(pyridin-4-yl)ethylamino)propan-2-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-5(4H)-yl)-2-(2-fluoro-6-(trifluoromethyl)phenyl)ethanone 397678 (S)-1-(3-(1-aminopropan-2-yl)-2-(3,5-dimethylphenyl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-5(4H)-yl)-2-(2-fluoro-6-(trifluoromethyl)phenyl)ethanone 397680 (S)-1-(2-(3,5-dimethylphenyl)-3-(1-(2-(tetrahydro-2H-pyran-4-yl)ethylamino)propan-2-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-5(4H)-yl)-2-(2-(trifluoromethyl)phenyl)ethanone 397681 (S)-5-(2-(2-(2-(3,5-dimethylphenyl)-5-(2-(2-fluoro-6-(trifluoromethyl)phenyl)acetyl)-4,5,6,7-tetrahydro-1H-pyrrolo[3,2-c]pyridin-3-yl)propylamino)ethyl)-1-methylpyridin-2(1H)-one 397682 (S)-1-(2-(3,5-dimethylphenyl)-3-(1-(2-(quinoxalin-6-yl)ethylamino)propan-2-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-5(4H)-yl)-2-(2-fluoro-6-(trifluoromethyl)phenyl)ethanone 397683 (S)-1-(2-(3,5-dimethylphenyl)-3-(1-(2-(2-methyl-1H-benzo[d]imidazol-5-yl)ethylamino)propan-2-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-5(4H)-yl)-2-(2-fluoro-6-(trifluoromethyl)phenyl)ethanone 397684 (S)-7-(2-(2-(2-(3,5-dimethylphenyl)-5-(2-(2-fluoro-6-(trifluoromethyl)phenyl)acetyl)-4,5,6,7-tetrahydro-1H-pyrrolo[3,2-c]pyridin-3-yl)propylamino)ethyl)-3-ethylquinazoline-2,4(1H,3H)-dione 397685 (S)-1-(3-(1-(2-(1H-benzo[d][1,2,3]triazol-5-yl)ethylamino)propan-2-yl)-2-(3,5-dimethylphenyl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-5(4H)-yl)-2-(2-fluoro-6-(trifluoromethyl)phenyl)ethanone 397686 (S)-1-(3-(1-(2-(3H-[1,2,3]triazolo[4,5-b]pyridin-6-yl)ethylamino)propan-2-yl)-2-(3,5-dimethylphenyl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-5(4H)-yl)-2-(2-fluoro-6-(trifluoromethyl)phenyl)ethanone 397687 (S)-1-(2-(3,5-dimethylphenyl)-3-(1-(2-(6-fluoro-1H-benzo[d][1,2,3]triazol-5-yl)ethylamino)propan-2-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-5(4H)-yl)-2-(2-fluoro-6-(trifluoromethyl)phenyl)ethanone 397688 (S)-1-(3-(1-(4-(1H-tetrazol-5-yl)phenethylamino)propan-2-yl)-2-(3,5-dimethylphenyl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-5(4H)-yl)-2-(2-fluoro-6-(trifluoromethyl)phenyl)ethanone 397689 1-(3-((S)-1-(2-(6-(1H-tetrazol-5-yl)pyridin-3-yl)ethylamino)propan-2-yl)-2-(3,5-dimethylphenyl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-5(4H)-yl)-2-(2-fluoro-6-(trifluoromethyl)phenyl)ethanone 397690 (S)-1-(3-(1-(2-(4-(1H-tetrazol-5-yl)phenoxy)ethylamino)propan-2-yl)-2-(3,5-dimethylphenyl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-5(4H)-yl)-2-(2-fluoro-6-(trifluoromethyl)phenyl)ethanone 397691 (S)-1-(3-(1-(4-(1H-tetrazol-5-yl)benzylamino)propan-2-yl)-2-(3,5-dimethylphenyl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-5(4H)-yl)-2-(2-fluoro-6-(trifluoromethyl)phenyl)ethanone 397692 (S)-4-(2-(2-(2-(3,5-dimethylphenyl)-5-(2-(2-fluoro-6-(trifluoromethyl)phenyl)acetyl)-4,5,6,7-tetrahydro-1H-pyrrolo[3,2-c]pyridin-3-yl)propylamino)ethyl)benzoic acid 397732 (3R,3aS,4S,4aS,9aR,E)-3-methyl-4-(2-(pyridin-2-yl)vinyl)-3,3a,4,4a,5,6,7,8-octahydronaphtho[2,3-c]furan-1(9aH)-one 397733 (3R,3aS,4S,4aS,9aR,E)-3-methyl-4-(2-(6-methylpyridin-2-yl)vinyl)-3,3a,4,4a,5,6,7,8-octahydronaphtho[2,3-c]furan-1(9aH)-one 397735 (3R,3aS,4S,4aS,9aR,E)-3-methyl-4-(2-(5-phenylpyridin-2-yl)vinyl)-3,3a,4,4a,5,6,7,8-octahydronaphtho[2,3-c]furan-1(9aH)-one 397748 (3R,3aS,4S,4aS,9aR,E)-3-methyl-4-(2-(6-methyl-5-phenylpyridin-2-yl)vinyl)-3,3a,4,4a,5,6,7,8-octahydronaphtho[2,3-c]furan-1(9aH)-one 397749 (3R,3aS,4S,4aS,9aR,E)-4-(2-(6-ethyl-5-phenylpyridin-2-yl)vinyl)-3-methyl-3,3a,4,4a,5,6,7,8-octahydronaphtho[2,3-c]furan-1(9aH)-one 397756 (3R,3aS,4S,4aR,8aS,9aR,E)-4-(2-(5-ethylpyridin-2-yl)vinyl)-3-methyl-decahydronaphtho[2,3-c]furan-1(3H)-one 397758 (3R,3aS,4S,4aR,8aS,9aR,E)-4-(2-(5-cyclopentylpyridin-2-yl)vinyl)-3-methyl-decahydronaphtho[2,3-c]furan-1(3H)-one 397760 (3R,3aS,4S,4aR,8aS,9aR,E)-3-methyl-4-(2-(5-(pyrrolidin-1-yl)pyridin-2-yl)vinyl)-decahydronaphtho[2,3-c]furan-1(3H)-one 397763 (3R,3aS,4S,4aR,8aS,9aR,E)-3-methyl-4-(2-(5-(4-phenylpiperazin-1-yl)pyridin-2-yl)vinyl)-decahydronaphtho[2,3-c]furan-1(3H)-one 397764 (3R,3aS,4S,4aR,8aS,9aR,E)-4-(2-(5-(furan-2-yl)pyridin-2-yl)vinyl)-3-methyl-decahydronaphtho[2,3-c]furan-1(3H)-one 397766 (3R,3aS,4S,4aR,8aS,9aR,E)-3-methyl-4-(2-(5-(thiophen-2-yl)pyridin-2-yl)vinyl)-decahydronaphtho[2,3-c]furan-1(3H)-one 397767 (3R,3aS,4S,4aR,8aS,9aR,E)-4-(2-(5-(5-chlorothiophen-2-yl)pyridin-2-yl)vinyl)-3-methyl-decahydronaphtho[2,3-c]furan-1(3H)-one 397768 (3R,3aS,4S,4aR,8aS,9aR,E)-3-methyl-4-(2-(5-(thiophen-3-yl)pyridin-2-yl)vinyl)-decahydronaphtho[2,3-c]furan-1(3H)-one 397769 (3R,3aS,4S,4aR,8aS,9aR,E)-3-methyl-4-(2-(5-(thiazol-2-yl)pyridin-2-yl)vinyl)-decahydronaphtho[2,3-c]furan-1(3H)-one 397770 (3R,3aS,4S,4aR,8aS,9aR,E)-4-(2-(5-(1H-imidazol-2-yl)pyridin-2-yl)vinyl)-3-methyl-decahydronaphtho[2,3-c]furan-1(3H)-one 397771 (3R,3aS,4S,4aR,8aS,9aR,E)-3-methyl-4-(2-(5-(1-methyl-1H-imidazol-5-yl)pyridin-2-yl)vinyl)-decahydronaphtho[2,3-c]furan-1(3H)-one 397772 (3R,3aS,4S,4aR,8aS,9aR,E)-3-methyl-4-(2-(5-(pyridin-2-yl)pyridin-2-yl)vinyl)-decahydronaphtho[2,3-c]furan-1(3H)-one 397773 (3R,3aS,4S,4aR,8aS,9aR,E)-3-methyl-4-(2-(5-(pyridin-3-yl)pyridin-2-yl)vinyl)-decahydronaphtho[2,3-c]furan-1(3H)-one 397774 (3R,3aS,4S,4aR,8aS,9aR,E)-3-methyl-4-(2-(5-(pyridin-4-yl)pyridin-2-yl)vinyl)-decahydronaphtho[2,3-c]furan-1(3H)-one 397775 (3R,3aS,4S,4aR,8aS,9aR)-3-methyl-4-[2-(1'-oxy-[3,3']bipyridinyl-6-yl)-vinyl]-decahydro-naphtho[2,3-c]furan-1-one 397776 (3R,3aS,4S,4aR,8aS,9aR,E)-3-methyl-4-(2-(5-(pyrazin-2-yl)pyridin-2-yl)vinyl)-decahydronaphtho[2,3-c]furan-1(3H)-one 397813 (3R,3aS,4S,4aR,8aS,9aR,E)-3-methyl-4-(2-(5-morpholinopyridin-2-yl)vinyl)-decahydronaphtho[2,3-c]furan-1(3H)-one 397820 (3aR,4R,9aS,E)-8-fluoro-4-(2-(5-(3-(trifluoromethyl)phenyl)pyridin-2-yl)vinyl)-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397822 (3aR,4R,9aS,E)-6,8-difluoro-4-(2-(5-(3-(trifluoromethyl)phenyl)pyridin-2-yl)vinyl)-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397825 (3aR,4R,9aS,E)-6-fluoro-4-(2-(5-(3-(trifluoromethyl)phenyl)pyridin-2-yl)vinyl)-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397828 (3aR,4R,9aS,E)-6-chloro-4-(2-(5-(3-(trifluoromethyl)phenyl)pyridin-2-yl)vinyl)-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397829 (3aR,4R,9aS,E)-8-chloro-4-(2-(5-(3-(trifluoromethyl)phenyl)pyridin-2-yl)vinyl)-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397830 (3aR,4R,9aS,E)-4-(2-(5-(3-chlorophenyl)pyridin-2-yl)vinyl)-6,8-difluoro-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397831 (3aR,4R,9aS,E)-4-(2-(5-(3-chlorophenyl)pyridin-2-yl)vinyl)-6-fluoro-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397832 (3aR,4R,9aS,E)-6-chloro-4-(2-(5-(3-chlorophenyl)pyridin-2-yl)vinyl)-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397834 (3aR,4R,9aS,E)-4-(2-(5-(3-chlorophenyl)pyridin-2-yl)vinyl)-8-fluoro-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397837 (3aR,4R,9aS,E)-8-chloro-4-(2-(5-(3-chlorophenyl)pyridin-2-yl)vinyl)-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397838 (3aR,4R,9aS,E)-4-(2-(5-(3-chlorophenyl)pyridin-2-yl)vinyl)-7-fluoro-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397842 (3aR,4R,9aS,E)-4-(2-(5-(3-chlorophenyl)pyridin-2-yl)vinyl)-7,8-difluoro-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397845 (3aR,4R,9aS,E)-4-(2-(5-(3-chlorophenyl)pyridin-2-yl)vinyl)-5-fluoro-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397849 (3aR,4R,9aS,E)-6-fluoro-4-(2-(5-(3-fluorophenyl)pyridin-2-yl)vinyl)-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397851 (3aR,4R,9aS,E)-8-fluoro-4-(2-(5-(3-fluorophenyl)pyridin-2-yl)vinyl)-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397855 (3aR,4R,9aS,E)-8-chloro-4-(2-(5-(3-fluorophenyl)pyridin-2-yl)vinyl)-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397858 (3aR,4R,9aS,E)-6-chloro-4-(2-(5-(3-fluorophenyl)pyridin-2-yl)vinyl)-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397861 (3aR,4R,9aS,E)-7-fluoro-4-(2-(5-(3-fluorophenyl)pyridin-2-yl)vinyl)-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397865 (3aR,4R,9aS,E)-7,8-difluoro-4-(2-(5-(3-fluorophenyl)pyridin-2-yl)vinyl)-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397868 (3aR,4R,9aS,E)-5-fluoro-4-(2-(5-(3-fluorophenyl)pyridin-2-yl)vinyl)-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397875 (R)-2-methoxy-6,10-dimethyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-ol 397876 (R)-2-methoxy-10-methyl-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-ol 397877 (R)-10-hydroxymethyl-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-ol 397878 (R)-10-hydroxymethyl-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-ol 397893 (3aR,4R,9aS,E)-4-(2-(5-(3-(trifluoromethyl)phenyl)pyridin-2-yl)vinyl)-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397894 (3aR,4R,9aS,E)-4-(2-(5-(3-fluorophenyl)pyridin-2-yl)vinyl)-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397897 (3aR,4R,9aS,E)-4-(2-(5-(3-chlorophenyl)pyridin-2-yl)vinyl)-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397912 (3aS,4S,9aR,E)-4-(2-(pyridin-2-yl)vinyl)-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397914 (3R,3aS,4S,9aR,E)-4-(2-(6-methoxyquinolin-2-yl)vinyl)-3-methyl-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397917 (3R,3aR,4R,9aS,E)-4-(2-(6-methoxyquinolin-2-yl)vinyl)-3-methyl-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397920 (3S,3aR,4R,9aS,E)-4-(2-(6-methoxyquinolin-2-yl)vinyl)-3-methyl-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397921 (3S,3aS,4S,9aR,E)-4-(2-(6-methoxyquinolin-2-yl)vinyl)-3-methyl-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397923 (3aS,4S,9aR,E)-4-(2-(6-methoxyquinolin-2-yl)vinyl)-3,3-dimethyl-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397924 (3aS,4S,9aR,E)-4-(2-(6-methoxyquinolin-2-yl)vinyl)-3a,4,9,9a-tetrahydronaphtho[2,3-c]furan-1(3H)-one 397943 SID24276280 397945 N-(4-methoxybenzyl)-2-(N-(2-ethylphenyl)-4-methylphenylsulfonamido)acetamide 397947 N-(3,4-dimethoxyphenethyl)-2-(N-(2-ethylphenyl)-4-methylphenylsulfonamido)acetamide 397949 4-methoxybenzyl 2-(N-(2-ethylphenyl)-4-methylphenylsulfonamido)acetate 397950 N-((5-benzyl-1,3,4-oxadiazol-2-yl)methyl)-N-(2-ethylphenyl)-4-methylbenzenesulfonamide 397952 N-((5-(4-chlorobenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(2-ethylphenyl)-4-methylbenzenesulfonamide 397953 N-((5-(4-methoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(2-ethylphenyl)-4-methylbenzenesulfonamide 397954 N-((5-(4-ethoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(2-ethylphenyl)-4-methylbenzenesulfonamide 397956 N-((5-(4-methoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-4-methyl-N-(2-methyl-3-(trifluoromethyl)phenyl)benzenesulfonamide 397959 N-((5-(4-methoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide 397960 N-((5-(4-ethoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide 397962 N-((5-(4-methoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(2,3-dichlorophenyl)-4-methylbenzenesulfonamide 397963 N-((5-(4-ethoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(2,3-dichlorophenyl)-4-methylbenzenesulfonamide 397967 N-((5-(4-(dimethylamino)benzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide 397969 3-(3-aminopropyl)-N,N-dibutyl-2-(3,4,5-trimethoxyphenylamino)-3H-benzo[d]imidazole-5-carboxamide 397970 N-((5-(4-(trifluoromethyl)benzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide 397972 N-((5-(4-fluorobenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide 397973 3-(3-aminopropyl)-N,N-diisopentyl-2-(3,4,5-trimethoxyphenylamino)-3H-benzo[d]imidazole-5-carboxamide 397975 N-((5-(2-fluorobenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide 397976 3-(3-aminopropyl)-N,N-dipropyl-2-(3,4,5-trimethoxyphenylamino)-3H-benzo[d]imidazole-5-carboxamide 397977 N-((5-(3-fluorobenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide 397980 3-(3-aminopropyl)-N,N-diisobutyl-2-(3,4,5-trimethoxyphenylamino)-3H-benzo[d]imidazole-5-carboxamide 397981 N-((5-(2-chlorobenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide 397982 3-(3-aminopropyl)-N,N-dipentyl-2-(3,4,5-trimethoxyphenylamino)-3H-benzo[d]imidazole-5-carboxamide 397983 2-(4-acetylphenylamino)-3-(3-aminopropyl)-N,N-diisopentyl-3H-benzo[d]imidazole-5-carboxamide 397984 2-(4-acetylphenylamino)-3-(2-aminoethyl)-N,N-diisopentyl-3H-benzo[d]imidazole-5-carboxamide 397985 2-(4-acetylphenylamino)-3-(4-aminobutyl)-N,N-diisopentyl-3H-benzo[d]imidazole-5-carboxamide 397987 2-(4-acetylphenylamino)-N,N-diisopentyl-3-(3-(methylamino)propyl)-3H-benzo[d]imidazole-5-carboxamide 397988 2-(4-acetylphenylamino)-3-(3-(dimethylamino)propyl)-N,N-diisopentyl-3H-benzo[d]imidazole-5-carboxamide 397990 N-((5-(3-chlorobenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide 397991 2-(4-acetylphenylamino)-3-(3-(diethylamino)propyl)-N,N-diisopentyl-3H-benzo[d]imidazole-5-carboxamide 397992 N-((5-(2,6-dichlorobenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide 397993 N-((5-(2,4-dichlorobenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide 397994 2-(4-acetylphenylamino)-N,N-diisopentyl-3-(3-(pyrrolidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 397995 N-((5-(4-methoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-4-chloro-N-(2,3-dichlorophenyl)benzenesulfonamide 397996 2-(4-acetylphenylamino)-N,N-diisopentyl-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 397998 N-((5-(4-ethoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(2,3-dichlorophenyl)-4-(trifluoromethyl)benzenesulfonamide 397999 N-((5-(4-methoxyphenoxy)-1,3,4-oxadiazol-2-yl)methyl)-N-(2-ethylphenyl)-4-methylbenzenesulfonamide 398000 2-(4-acetylphenylamino)-N,N-diisopentyl-3-(3-morpholinopropyl)-3H-benzo[d]imidazole-5-carboxamide 398002 2-(4-acetylphenylamino)-N,N-diisopentyl-3-(3-(4-methylpiperazin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398004 2-(4-acetylphenylamino)-3-(3-(dimethylamino)-2,2-dimethylpropyl)-N,N-diisopentyl-3H-benzo[d]imidazole-5-carboxamide 398005 2-(4-acetylphenylamino)-N,N-diisopentyl-3-(1-methylpiperidin-4-yl)-3H-benzo[d]imidazole-5-carboxamide 398006 tert-butyl 3-(2-(4-acetylphenylamino)-6-(diisopentylcarbamoyl)-1H-benzo[d]imidazol-1-yl)propylcarbamate 398007 N-(3-chloro-2-methylphenyl)-N-((5-(4-methoxyphenylamino)-1,3,4-oxadiazol-2-yl)methyl)-4-methylbenzenesulfonamide 398008 2-(4-acetylphenylamino)-3-(3-hydroxypropyl)-N,N-diisopentyl-3H-benzo[d]imidazole-5-carboxamide 398009 N-(2,3-dichlorophenyl)-N-((5-(4-methoxyphenylamino)-1,3,4-oxadiazol-2-yl)methyl)-4-methylbenzenesulfonamide 398010 N-(2,3-dichlorophenyl)-N-((5-(4-methoxyphenylamino)-1,3,4-oxadiazol-2-yl)methyl)-4-(trifluoromethyl)benzenesulfonamide 398011 N-(2-ethylphenyl)-N-((5-((4-methoxyphenoxy)methyl)-1,3,4-oxadiazol-2-yl)methyl)-4-methylbenzenesulfonamide 398012 2-(3-acetylphenylamino)-N,N-diisopentyl-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398013 N-(2-ethylphenyl)-N-((5-((4-methoxyphenylamino)methyl)-1,3,4-oxadiazol-2-yl)methyl)-4-methylbenzenesulfonamide 398014 N-(3-chloro-2-methylphenyl)-N-((5-((4-methoxyphenylamino)methyl)-1,3,4-oxadiazol-2-yl)methyl)-4-methylbenzenesulfonamide 398015 2-(2-acetylphenylamino)-N,N-diisopentyl-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398016 N,N-diisopentyl-2-(phenylamino)-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398018 N,N-diisopentyl-2-(4-methoxyphenylamino)-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398019 N,N-diisopentyl-3-(3-(piperidin-1-yl)propyl)-2-(4-propionylphenylamino)-3H-benzo[d]imidazole-5-carboxamide 398020 N,N-diisopentyl-2-(4-(methylcarbamoyl)phenylamino)-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398021 2-(4-carbamoylphenylamino)-N,N-diisopentyl-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398027 2-(4-acetamidophenylamino)-N,N-diisopentyl-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398029 methyl 4-(6-(diisopentylcarbamoyl)-1-(3-(piperidin-1-yl)propyl)-1H-benzo[d]imidazol-2-ylamino)benzoate 398032 N,N-diisopentyl-2-(4-nitrophenylamino)-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398034 2-(4-fluorophenylamino)-N,N-diisopentyl-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398035 2-(4-chlorophenylamino)-N,N-diisopentyl-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398036 2-(4-bromophenylamino)-N,N-diisopentyl-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398037 2-(biphenyl-4-ylamino)-3-(3-piperidin-1-yl-propyl)-3H-benzoimidazole-5-carboxylic acid bis-(3-methyl-butyl)-amide 398038 N,N-diisopentyl-2-(4-phenoxyphenylamino)-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398039 2-(4-benzoylphenylamino)-N,N-diisopentyl-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398040 N,N-diisopentyl-2-(4-(piperidin-1-yl)phenylamino)-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398041 N,N-diisopentyl-3-(3-(piperidin-1-yl)propyl)-2-(pyridin-3-ylamino)-3H-benzo[d]imidazole-5-carboxamide 398042 2-(1H-indol-4-ylamino)-N,N-diisopentyl-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398043 N,N-diisopentyl-3-(3-(piperidin-1-yl)propyl)-2-(thiophen-3-ylamino)-3H-benzo[d]imidazole-5-carboxamide 398044 2-(benzylamino)-N,N-diisopentyl-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398045 2-(4-acetylbenzylamino)-N,N-diisopentyl-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398046 2-(2-acetamidoethylamino)-N,N-diisopentyl-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398047 N,N-diisopentyl-2-(2-methoxyethylamino)-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398048 2-(4-acetylphenyl)-N,N-diisopentyl-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398049 N,N-diisopentyl-2-(4-methoxyphenyl)-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398050 methyl 4-(6-(diisopentylcarbamoyl)-1-(3-(piperidin-1-yl)propyl)-1H-benzo[d]imidazol-2-yl)benzoate 398051 2-(1H-indol-3-yl)-N,N-diisopentyl-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398052 N,N-diisopentyl-2-(1-methyl-1H-indol-3-yl)-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398053 2-(benzo[b]thiophen-2-yl)-N,N-diisopentyl-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398054 2-(4-acetylbenzyl)-N,N-diisopentyl-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398055 2-(4-methoxybenzyl)-N,N-diisopentyl-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398056 N,N-diisopentyl-2-(4-methoxybenzoyl)-3-(3-(piperidin-1-yl)propyl)-3H-benzo[d]imidazole-5-carboxamide 398066 (5R,8R,11S)-11-(3-aminopropyl)-5-[(4-hydroxyphenyl)methyl]-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14-dodecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione 398068 (5R,8R,11S)-11-(2-aminoethyl)-5-[(4-hydroxyphenyl)methyl]-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione 398070 (5R,8R,11S)-11-(aminomethyl)-5-[(4-hydroxyphenyl)methyl]-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione 398072 (5R,8R,11S)-5-[(4-hydroxyphenyl)methyl]-8-(propan-2-yl)-11-[(propan-2-ylamino)methyl]-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione 398073 N-{[(5R,8R,11S)-5-[(4-hydroxyphenyl)methyl]-6,9,12-trioxo-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecin-11-yl]methyl}acetamide 398075 (5R,8R,11S)-11-(aminomethyl)-5-[(3-chlorophenyl)methyl]-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione 398077 (5R,8R,11S)-11-(aminomethyl)-5-[(4-chlorophenyl)methyl]-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione 398080 (5R,8R,11S)-11-(aminomethyl)-8-(propan-2-yl)-5-{[3-(trifluoromethyl)phenyl]methyl}-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione 398081 (5R,8R,11S)-5-[(4-chlorophenyl)methyl]-11-[(methylamino)methyl]-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione 398082 (5R,8R,11S)-11-[(methylamino)methyl]-8-(propan-2-yl)-5-{[3-(trifluoromethyl)phenyl]methyl}-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione 398083 (5R,8R,11S)-5-[(3-chlorophenyl)methyl]-11-[(dimethylamino)methyl]-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione 398085 (5R,8R,11S)-5-[(4-chlorophenyl)methyl]-11-[(dimethylamino)methyl]-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione 398086 1-{[(5R,8R,11S)-5-[(4-chlorophenyl)methyl]-6,9,12-trioxo-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecin-11-yl]methyl}guanidine 398087 1-{[(5R,8R,11S)-6,9,12-trioxo-8-(propan-2-yl)-5-{[3-(trifluoromethyl)phenyl]methyl}-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecin-11-yl]methyl}guanidine 398089 {[(5R,8R,11S)-5-[(4-chlorophenyl)methyl]-6,9,12-trioxo-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecin-11-yl]methyl}urea 398090 (5R,8R,11S)-8-(propan-2-yl)-11-[(pyrimidin-2-ylamino)methyl]-5-{[3-(trifluoromethyl)phenyl]methyl}-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione 398092 (5R,8R,11S)-5-[(3-chlorophenyl)methyl]-8-(propan-2-yl)-11-[(1,3-thiazol-2-ylamino)methyl]-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione 398093 (5R,8R,11S)-5-[(3-chlorophenyl)methyl]-11-[(4,5-dihydro-1H-imidazol-2-ylamino)methyl]-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione 398095 (5R,8R,11S)-5-[(3-chlorophenyl)methyl]-8-(propan-2-yl)-11-[(1,4,5,6-tetrahydropyrimidin-2-ylamino)methyl]-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione 398096 1-{[(5R,8R,11S)-5-[(3-chlorophenyl)methyl]-6,9,12-trioxo-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecin-11-yl]methyl}-2-cyanoguanidine 398098 1-{[(5R,8R,11S)-5-[(3-chlorophenyl)methyl]-6,9,12-trioxo-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecin-11-yl]methyl}guanidine 398099 3-[(5R,8R,11S)-5-[(3-chlorophenyl)methyl]-6,9,12-trioxo-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecin-11-yl]propanimidamide 398100 1-{2-[(5R,8R,11S)-5-[(3-chlorophenyl)methyl]-6,9,12-trioxo-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecin-11-yl]ethyl}guanidine 398101 (5R,8R,11S)-8-(propan-2-yl)-11-(pyrrolidin-1-ylmethyl)-5-{[3-(trifluoromethyl)phenyl]methyl}-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione 398102 (5R,8R,11S)-11-[(5-methyl-1H-1,2,3-triazol-1-yl)methyl]-8-(propan-2-yl)-5-{[3-(trifluoromethyl)phenyl]methyl}-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione 398103 (5R,8R,11S)-11-[(4,5-dimethyl-1H-1,2,3-triazol-1-yl)methyl]-8-(propan-2-yl)-5-{[3-(trifluoromethyl)phenyl]methyl}-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione 398104 (5R,8R,11S)-11-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]-8-(propan-2-yl)-5-{[3-(trifluoromethyl)phenyl]methyl}-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione 398106 (5R,8R,11S)-5-[(3-chlorophenyl)methyl]-8-(propan-2-yl)-11-(1H-pyrazol-1-ylmethyl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione 398107 (5R,8R,11S)-5-[(3-chlorophenyl)methyl]-11-(1H-imidazol-1-ylmethyl)-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione 398108 (5R,8R,11S)-5-[(3-fluorophenyl)methyl]-8-(propan-2-yl)-11-(1,3-thiazol-4-ylmethyl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione 398335 2-(4-acetylphenylamino)-3-(3-aminopropyl)-N,N-diisobutyl-3H-benzo[d]imidazole-5-carboxamide 398336 4-[1-(1-methyl-pyridin-2-yl)-1H-imidazol-2-yl]-4-phenyl-piperidine-1-carboxylic acid ethyl ester 398812 3-propyl-1H-pyrazole-5-carboxylic acid 398813 SID14723313 398815 3-butyl-1H-pyrazole-5-carboxylic acid 399361 5-(((2R,3S)-2-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-3-(4-fluorophenyl)morpholino)methyl)-2H-1,2,4-triazol-3(4H)-one 400013 1-alpha-hydroxysalvinorin A 400492 Substance P 402579 1-(2-chloro-2-phenylethyl)-N-(3-fluorophenethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 402580 1-(2-chloro-2-phenylethyl)-N-(2-chlorophenethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 402582 1-(2-chloro-2-phenylethyl)-N-(3-chlorophenethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 402583 N-(4-chlorophenethyl)-7-(2-chloro-2-phenylethyl)-2-(methylthio)-7H-pyrrolo[2,3-d]pyrimidin-4-amine 402589 1-(2-chloro-2-phenylethyl)-N-(4-methylphenethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 402593 N-(4-methoxyphenethyl)-1-(2-chloro-2-phenylethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 402596 1-(2-chloro-2-(4-chlorophenyl)ethyl)-6-(methylthio)-N-phenethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 402599 1-(2-chloro-2-phenylethyl)-6-(ethylthio)-N-phenethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 402604 1-(2-chloro-2-phenylethyl)-N-(2-chlorobenzyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 402608 N-(4-chlorobenzyl)-1-(2-chloro-2-phenylethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 402613 1-(2-chloro-2-phenylethyl)-N-(2-fluorobenzyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 402614 1-(2-chloro-2-phenylethyl)-N-(3-fluorobenzyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 402616 1-(2-chloro-2-phenylethyl)-N-(4-fluorobenzyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 402620 N-benzyl-1-(2-chloro-2-(4-chlorophenyl)ethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 402622 N-benzyl-1-(2-chloro-2-(4-fluorophenyl)ethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 402623 1-(2-chloro-2-phenylethyl)-N-(3-chlorophenyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 402624 1-(2-chloro-2-phenylethyl)-N-(3-fluorophenyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 402626 N-(3-bromophenyl)-1-(2-chloro-2-phenylethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 402627 1-(2-chloro-2-phenylethyl)-6-(methylthio)-N-phenyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 402629 1-(2-chloro-2-phenylethyl)-N-(3-chlorophenyl)-6-(ethylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 402630 1-(2-chloro-2-phenylethyl)-N-(3-chlorophenyl)-6-(propylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 402631 1-(2-chloro-2-phenylethyl)-N-(3-chlorophenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 402632 N-(3-bromophenyl)-1-(2-chloro-2-(4-fluorophenyl)ethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 403900 (2R,3R,4S,5R)-2-(6-hydrazinyl-9H-purin-9-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol 405786 SID26752053 406850 1-(1-(3-(5-methoxy-2-methylphenoxy)-4-methylpentyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one 407384 oroidin 407549 SID26755702 408842 SID26748956 411582 1-(3-tert-butyl-1-p-tolyl-1H-pyrazol-5-yl)-3-(4-(6-(morpholinomethyl)pyridin-3-yl)naphthalen-1-yl)urea 412739 SID14723439 412741 3-benzyl-1H-pyrazole-5-carboxylic acid 412744 5-meta-chlorobenzyl-3-carboxyl-pyrazole 413905 SID29217517 415943 oxymorphindole 418977 BNTX 419205 4-(6-(2-chlorophenylamino)-1H-indazol-3-yl)-N-(2-(dimethylamino)ethyl)benzamide 419206 N-(2-methoxyphenyl)-3-phenyl-1H-indazol-6-amine 419596 SID26752060 420330 3-hydroxy-N-(2-hydroxy-1-methyl-ethyl)-5-(4-phenylamino-phenylamino)-isothiazole-4-carboxamidine 421066 SID26748950 421450 1-((1R,2S)-2-(((S)-3-(4-fluorobenzyl)piperidin-1-yl)methyl)cyclohexyl)-3-(3-acetylphenyl)urea 422410 8-(1-benzyl-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 422416 8-(1-(3-fluorobenzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 422417 8-(1-(3-(trifluoromethyl)benzyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 422925 8-(1-((5-phenyl-1,2,4-oxadiazol-3-yl)methyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 422926 8-(1-((5-phenylisoxazol-3-yl)methyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 423875 Dmt-Pro-Phe-D-2-Nal-NH2 424149 (2R,3R,4R,5R)-2-(6-(cyclopentylamino)-9H-purin-9-yl)-5-(hydroxymethyl)-3-methyl-tetrahydrofuran-3,4-diol 424150 (2R,3R,4R,5R)-2-(2-chloro-6-(cyclopentylamino)-9H-purin-9-yl)-5-(hydroxymethyl)-3-methyl-tetrahydrofuran-3,4-diol 424433 (S)-4-(2-(3-chlorophenyl)-2-hydroxyethylamino)-3-(4-methyl-6-morpholino-1H-benzo[d]imidazol-2-yl)pyridin-2(1H)-one 424776 (R)-3-(3,4-dioxo-2-(1-phenylpropylamino)cyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide 424777 (R)-3-(2-(1-(3-fluorophenyl)propylamino)-3,4-dioxocyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide 425061 (Z)-2-debromohymenialdisine 425386 4-amino-5-(4-chlorophenyl)-7-(t-butyl)pyrazolo[3,4-d]pyrimidine 426371 Phosphoric acid mono-[(1R,2S,4S,5S)-4-(2-iodo-6-methylamino-purin-9-yl)-1-phosphonooxymethyl-bicyclo[3.1.0]hex-2-yl] ester 428234 1-(1-(4-(3-phenylquinoxalin-2-yl)benzyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one 428237 SID29217482 428554 N'-(2-chloro-9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-6-yl)-3-methylthiophene-2-carbohydrazide 428706 5-(6-Amino-2-hex-1-ynyl-purin-9-yl)-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 428708 4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)quinoline 428882 SID26757060 428978 4-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-9H-purin-6-ylamino)benzenesulfonic acid 428980 N6-Phenyladenosine 429024 5'-(N-Cyclopropyl)carboxamidoadenosine 429062 (2R,3R,4S,5R)-2-(2-(2-(1H-indol-3-yl)ethoxy)-6-(ethylamino)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 429156 Angiotensin II 429662 SID26751818 430036 7-oxo-7H-benzimidazo[2,1-a]benz[de]isoquinoline-3-carboxylic acid acetate 430253 (S)-3-(4-chlorophenyl)-N'-(4-chlorophenylsulfonyl)-N-methyl-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboximidamide 430291 8-(1-(3-fluorobenzyl)-1H-pyrazol-4-yl)-1,3-dimethyl-1H-purine-2,6(3H,7H)-dione 430431 SID11113932 430577 (S)-4-methyl-5-(2-methyl-1,4-diazepan-1-ylsulfonyl)isoquinoline 430594 5-(2-Phenyl-pyrazolo[1,5-a]pyridin-3-yl)-1H-pyrazolo[3,4-c]pyridazin-3-ylamine 430613 4-(4-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-5-(pyridin-2-yl)-1H-imidazol-2-yl)benzamide 430646 1-tert-butyl-3-(naphthalen-1-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 431277 N-(benzo[d][1,3]dioxol-5-yl)-2-(5-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-1-methyl-1H-pyrazol-3-yloxy)acetamide 431309 2-(3,4-dimethoxyphenyl)-N-(5-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-1-methyl-1H-pyrazol-3-yl)acetamide 432077 (S)-7-(2-aminopropylamino)-2-(3,5-dimethoxyphenylamino)-5-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide 432112 (R)-7-(2-aminopropylamino)-2-(3,5-dimethoxyphenylamino)-5-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide 432143 7-(2-amino-2-methylpropylamino)-2-(3,5-dimethoxyphenylamino)-5-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide 432165 N-(2,5-dimethoxybenzyl)-4-phenoxy-1H-pyrazolo[4,3-c]pyridin-3-amine 432515 5-cyclopropyl-2-(3,5-dimethoxyphenylamino)-7-((S)-1-hydroxymethyl-2-pyridin-3-ylethylamino)pyrazolo[1,5-a]pyrimidine-3-carboxamide 432517 5-cyclopropyl-2-(3,5-dimethoxyphenylamino)-7-[(S)-2-hydroxy-1-(1H-indol-3-ylmethyl)ethylamino]pyrazolo[1,5-a]pyrimidine-3-carboxamide 432553 7-((R)-1-benzyl-2-hydroxyethylamino)-5-cyclopropyl-2-(3,5-dimethoxyphenylamino)pyrazolo[1,5-a]pyrimidine-3-carboxamide 432555 7-((S)-1-benzyl-2-hydroxyethylamino)-5-cyclopropyl-2-(3,5-dimethoxyphenylaminopyrazolo[1,5-a]pyrimidine-3-carboxamide 432591 5-cyclopropyl-2-(3,5-dimethoxyphenylamino)-7-((R)-2-hydroxymethylpyrrolidin-1-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide 432592 5-cyclopropyl-2-(3,5-dimethoxyphenylamino)-7-((S)-2-hydroxymethylpyrrolidin-1-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide 432622 5-cyclopropyl-2-(3,5-dimethoxyphenylamino)-7-((R)-1-hydroxymethyl-2-methylpropylamino)pyrazolo[1,5-a]pyrimidine-3-carboxamide 432623 7-amino-5-cyclopropyl-2-phenylaminopyrazolo[1,5-a]pyrimidine-3-carboxamide 432654 2-(3,5-dimethoxyphenylamino)-7-((R)-1-hydroxymethyl-2-methylpropylamino)-5-phenylpyrazolo[1,5-a]pyrimidine-3-carboxamide 432655 2-(3,5-dimethoxyphenylamino)-7-((R)-1-hydroxymethyl-2-methylpropylamino)-5-isopropylpyrazolo[1,5-a]pyrimidine-3-carboxamide 432690 2-(3,5-dimethoxyphenylamino)-7-((S)-1-hydroxymethyl-2-methylpropylamino)-5-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide 432691 2-(3,5-dimethoxyphenylamino)-7-((R)-1-hydroxymethyl-2-methylpropylamino)-5-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide 432726 2-(3,5-dimethoxyphenylamino)-7-((S)-2-hydroxypropylamino)-5-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide 432727 2-(3,5-dimethoxyphenylamino)-7-((S)-2-hydroxy-1-methylethylamino)-5-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide 432761 3,5-dimethoxyphenylamino)-7-((R)-2-hydroxypropylamino)-5-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide 433344 N6-cyclopentyl-5'-deoxy-5'-ethylthioadenosine 434258 (R)-N-(2-(1-(4-chlorobenzyl)pyrrolidin-3-ylamino)-2-oxoethyl)-3-(trifluoromethyl)benzamide 434488 1-(1-(4-(3-phenyl-5-(1H-tetrazol-5-yl)pyridin-2-yl)benzyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one 434539 6-(4-((4-(2-oxo-2,3-dihydrobenzo[d]imidazol-1-yl)piperidin-1-yl)methyl)phenyl)-5-phenylnicotinonitrile 436192 N-(5-(3-chlorobenzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide 436195 N-(5-(benzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide 436248 N-(5-(4-bromobenzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide 436277 N-(4-(4-(5-Methyl-1H-pyrazol-3-ylamino)-6-(4-methylpiperazin-1-yl)-pyrimidin-2-ylthio)phenyl)cyclopropanecarboxamide 436278 danusertib 436297 4-fluoro-N-(5-(4-fluorobenzylthio)-1,3,4-thiadiazol-2-yl)benzamide 436556 N-(5-(4-methoxybenzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide 436558 N-(5-(benzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide 436559 N-(5-(3-chlorobenzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide 436604 N-(5-(3-chlorobenzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide 436605 N-(5-(benzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide 436606 N-(5-(4-fluorobenzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide 436608 N-(5-(3-fluorobenzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide 436657 N-(5-(4-bromobenzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide 436659 N-(5-(4-nitrobenzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide 436660 N-(5-(3-fluorobenzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide 436662 N-(5-(4-methoxybenzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide 436702 N-(5-(3-fluorobenzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide 436704 N-(5-(4-methoxybenzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide 436851 N-(5-(4-fluorobenzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide 436853 N-(5-(4-nitrobenzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide 436899 N-(5-(4-bromobenzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide 436901 N-(5-(4-nitrobenzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide 438420 2-(4-((4-(2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)methyl)phenyl)-3-phenylquinoxaline-6-carboxylic acid 438421 3-(4-((4-(2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)methyl)phenyl)-2-phenylquinoxaline-6-carboxylic acid 438624 salvinorin A propyl ether 439021 metazocine 439124 1-(1-(4-(3-phenyl-6-(2H-tetrazol-5-yl)quinoxalin-2-yl)benzyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one 439125 1-(1-(4-(3-phenyl-7-(2H-tetrazol-5-yl)quinoxalin-2-yl)benzyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one 439814 3-(3-chloro-1H-pyrazol-5-yl)quinoxalin-2(1H)-one 440694 6-(cyclohexylmethoxy)-9H-purin-2-amine 442361 SID11111969 445395 atropine 446784 Buprenorphine 447055 5'-guanidinonaltrindole 448944 4-(1H-Indol-3-yl)-3-(3,4,5-trimethoxyphenyl)-1,5-dihydro-2H-pyrrole-2-one 449128 3-(1H-Indol-3-yl)-4-(3,4,5-trimethoxyphenyl)-1,5-dihydro-2Hpyrrole-2-one 449130 3-(3,4,5-Trimethoxyphenyl)-4-(1-{[2-(trimethylsilyl)ethoxy]-methyl}-1H-indol-3-yl)-1,5-dihydro-2H-pyrrole-2-one 449198 4-[1-(Ethoxymethyl)-1H-indol-3-yl]-3-(3,4,5-trimethoxyphenyl)-1,5-dihydro-2H-pyrrole-2-one 449199 4-[1-(Isopropoxymethyl)-1H-indol-3-yl]-3-(3,4,5-trimethoxyphenyl)-1,5-dihydro-2H-pyrrole-2-one 449200 4-[1-(tert-Butoxymethyl)-1H-indol-3-yl]-3-(3,4,5-trimethoxyphenyl)-1,5-dihydro-2H-pyrrole-2-one 449201 4-[1-(Phenoxymethyl)-1H-indol-3-yl]-3-(3,4,5-trimethoxyphenyl)-1,5-dihydro-2H-pyrrole-2-one 449267 4-{1-[(Benzyloxy)methyl]-1H-indol-3-yl}-3-(3,4,5-trimethoxyphenyl)-1,5-dihydro-2H-pyrrole-2-one 449342 3-(N-Methyl-1H-indol-3-yl)-4-(4-methoxyphenyl)-1,5-dihydro-2H-pyrrole-2-one 450003 9-(2,6-dimethylstyryl)-N-(4-(dipropylphosphoryl)phenyl)-2-isopropyl-9H-purin-6-amine 450004 9-(2,6-dimethylstyryl)-N-(4-(dipropylphosphoryl)phenyl)-2-isopropyl-9H-purin-6-amine 450005 N-(4-(dipropylphosphoryl)phenyl)-2-isopropyl-9-styryl-9H-purin-6-amine 450006 N-(4-(dipropylphosphoryl)phenyl)-2-isopropyl-9-styryl-9H-purin-6-amine 450078 9-(2,6-dimethylstyryl)-N-(4-(dimethylphosphoryl)phenyl)-9H-purin-6-amine 450249 9-(2-chloro-6-methylstyryl)-N-(4-(dimethylphosphoryl)phenyl)-9H-purin-6-amine 450250 9-(2-chlorostyryl)-N-(4-(dimethylphosphoryl)phenyl)-9H-purin-6-amine 450251 9-(2-(1H-indol-4-yl)vinyl)-N-(4-(dimethylphosphoryl)phenyl)-9H-purin-6-amine 450252 9-(2-(1H-indazol-4-yl)vinyl)-N-(4-(dimethylphosphoryl)phenyl)-9H-purin-6-amine 450331 9-(2,6-dimethylstyryl)-N-(4-(dipropylphosphoryl)phenyl)-9H-purin-6-amine 450332 9-(2,6-dimethylstyryl)-N6-(4-(dimethylphosphoryl)phenyl)-N2,N2-dimethyl-9H-purine-2,6-diamine 450333 9-(2,6-dimethylstyryl)-N-(4-(dimethylphosphoryl)phenyl)-2-(pyrrolidin-1-yl)-9H-purin-6-amine 450548 9-(2,6-dimethylstyryl)-N-(4-(dimethylphosphoryl)phenyl)-2-isopropyl-9H-purin-6-amine 450549 9-(2,6-dimethylstyryl)-2-cyclopentyl-N-(4-(dimethylphosphoryl)phenyl)-9H-purin-6-amine 450761 N-(2-aminoethyl)-1,8-dimethylimidazo[1,2-a]quinoxalin-4-amine hydrochloride 453859 3-(1,3-Dioxo-1,3-dihydro-2H-indolo[1',7':4,5,6]pyrrolo[3',4':2,3][1,4]diazepino[1,7-a]indol-2-yl)propyl Imidothiocarbamate 454702 4-(1-(2-chloro-2-(4-fluorophenyl)ethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-yl)morpholine 454703 1-(2-chloro-2-(4-fluorophenyl)ethyl)-N-(4-fluorobenzyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 454704 1-(2-chloro-2-(4-fluorophenyl)ethyl)-N-(2-fluorobenzyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 454705 1-(2-chloro-2-(4-fluorophenyl)ethyl)-6-(methylthio)-N-phenethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 454707 4-(1-(2-bromo-2-phenylethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-yl)morpholine 454708 N-benzyl-1-(2-bromo-2-phenylethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 454709 1-(2-bromo-2-phenylethyl)-6-(methylthio)-N-phenethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 454778 1-(2-chloro-2-(4-fluorophenyl)ethyl)-N-(3-fluorophenyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 454779 1-(2-chloro-2-(4-chlorophenyl)ethyl)-6-(methylthio)-N-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 454780 N-butyl-1-(2-chloro-2-(4-chlorophenyl)ethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 454781 1-(2-chloro-2-(4-chlorophenyl)ethyl)-N,N-diethyl-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 454782 4-(1-(2-chloro-2-(4-chlorophenyl)ethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-yl)morpholine 454783 N4-benzyl-1-(2-chloro-2-phenylethyl)-N6,N6-dimethyl-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine 454784 1-(2-chloro-2-phenylethyl)-N6,N6-dimethyl-N4-propyl-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine 454785 1-(2-chloro-2-phenylethyl)-N,N-dimethyl-4-morpholino-1H-pyrazolo[3,4-d]pyrimidin-6-amine 455131 1-(2-chloro-2-phenylethyl)-N-(2-fluorophenethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 455132 1-(2-chloro-2-(4-fluorophenyl)ethyl)-6-(methylthio)-N-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 455133 N-butyl-1-(2-chloro-2-(4-fluorophenyl)ethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 455134 1-(2-chloro-2-phenylethyl)-N,N-diethyl-6-(ethylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 455135 1-(2-chloro-2-phenylethyl)-N-propyl-6-(propylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 455136 N-butyl-1-(2-chloro-2-phenylethyl)-6-(propylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 455137 1-(2-chloro-2-phenylethyl)-N,N-diethyl-6-(propylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 455138 N-benzyl-1-(2-chloro-2-phenylethyl)-6-(propylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 455211 1-(2-bromo-2-phenylethyl)-6-(methylthio)-N-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 455212 1-(2-bromo-2-phenylethyl)-N-butyl-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 455213 1-(2-bromo-2-phenylethyl)-N-(2-ethoxyethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 455214 1-(2-bromo-2-phenylethyl)-6-(methylthio)-4-(pyrrolidin-1-yl)-1H-pyrazolo[3,4-d]pyrimidine 455215 1-(2-bromo-2-phenylethyl)-6-(methylthio)-4-(piperidin-1-yl)-1H-pyrazolo[3,4-d]pyrimidine 455950 N-(1-(3-fluorobenzyl)-1H-indazol-5-yl)-6-(4-(2-(methylsulfonyl)ethylamino)butoxy)quinazolin-4-amine 456386 6-(4-(2-(methylsulfonyl)ethylamino)butoxy)-N-(3-ethynylphenyl)quinazolin-4-amine 456444 6-(4-(2-(methylsulfonyl)ethylamino)butoxy)-N-(3-chloro-4-fluorophenyl)quinazolin-4-amine 458490 1-(4-amino-7-(3-hydroxypropyl)-5-p-tolyl-7H-pyrrolo[2,3-d]pyrimidin-6-yl)-2-fluoroethanone 458956 (2R,3R,4S,5R)-2-(6-amino-8-(methylamino)-9H-purin-9-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol 459149 (R)-3-cyclobutyl-2-((3S,4S)-3-(3-fluorophenyl)-4-((4-(imidazo[1,2-a]pyrimidin-3-yl)piperidin-1-yl)methyl)pyrrolidin-1-yl)propanoic acid 459150 (R)-3-cyclobutyl-2-((3S,4S)-3-(3-fluorophenyl)-4-((4-(imidazo[1,2-a]pyrazin-2-yl)piperidin-1-yl)methyl)pyrrolidin-1-yl)propanoic acid 459855 (R)-3-cyclobutyl-2-((3S,4S)-3-(3-fluorophenyl)-4-((4-(imidazo[1,2-b]pyridazin-3-yl)piperidin-1-yl)methyl)pyrrolidin-1-yl)propanoic acid 459856 (R)-3-cyclobutyl-2-((3S,4S)-3-(3-fluorophenyl)-4-((4-(imidazo[1,2-a]pyridin-2-yl)piperidin-1-yl)methyl)pyrrolidin-1-yl)propanoic acid 460058 (R)-2-(4-amino-5-phenyl-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2-phenylethanol 460059 (S)-2-(4-amino-5-phenyl-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2-phenylethanol 460094 (R)-3-cyclobutyl-2-((3S,4S)-3-(3-fluorophenyl)-4-((4-(imidazo[1,5-a]pyridin-3-yl)piperidin-1-yl)methyl)pyrrolidin-1-yl)propanoic acid 460266 (2S,3S)-N-(2-methoxy-5-(5-(trifluoromethyl)-1H-tetrazol-1-yl)benzyl)-2-phenylpiperidin-3-amine 466038 (R)-(-)-Apomorphine hydrochloride 466130 SID11532956 466506 ginkgolide B 467250 (2R,3S,4R,5R)-5-(2-chloro-6-(cyclopentylamino)-9H-purin-9-yl)-2-(hydroxymethyl)-3-methyl-tetrahydrofuran-3,4-diol 467452 (2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-2-(hydroxymethyl)-3-methyl-tetrahydrofuran-3,4-diol 469183 H-D-Phe-c[Cys-Tyr-DTrp-Orn-Thr-Pen]-Thr-NH2 470091 Naphthalene-2-carboxylic acid {4-[2-((R)-8-methoxy-1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-ethyl]-cyclohexyl}-amide 470598 3-({6,7-dimethyl-5-[(1-methylpyridin-1-ium-3-yl)carbonyl]-4-oxo-3,4,5,6,7,8-hexahydropteridin-2-yl}carbamoyl)-1-methylpyridin-1-ium 470599 7-(4-chlorobenzyl)-8-mercapto-3-methyl-1H-purine-2,6(3H,7H)-dione 470659 7-benzyl-3-methyl-8-(methylthio)-1H-purine-2,6(3H,7H)-dione 470660 1,7-dibenzyl-8-(3-chlorobut-2-enylthio)-3-methyl-1H-purine-2,6(3H,7H)-dione 470661 1,7-dibenzyl-8-(2-hydroxyethylthio)-3-methyl-1H-purine-2,6(3H,7H)-dione 470662 2-(7-(3-bromobenzyl)-3-methyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-ylthio)acetamide 470663 7-benzyl-3-methyl-8-(2-(1-(4-nitrophenyl)ethylidene)hydrazinyl)-1H-purine-2,6(3H,7H)-dione 470733 7-benzyl-8-(3,5-dimethyl-1H-pyrazol-1-yl)-1,3-dimethyl-1H-purine-2,6(3H,7H)-dione 470734 8-(3-chlorobut-2-enylthio)-7-(2-hydroxy-4-phenylbutyl)-3-methyl-1H-purine-2,6(3H,7H)-dione 470735 8-(2-(3-nitrobenzylidene)hydrazinyl)-7-allyl-3-methyl-1H-purine-2,6(3H,7H)-dione 470736 7-((Z)-3-chlorobut-2-enyl)-3-methyl-8-(2-(1-(4-nitrophenyl)ethylidene)hydrazinyl)-1H-purine-2,6(3H,7H)-dione 470830 8-(2-(4-nitrobenzylidene)hydrazinyl)-7-benzyl-3-methyl-1H-purine-2,6(3H,7H)-dione 470831 7-benzyl-3-methyl-8-(2-(1-phenylethylidene)hydrazinyl)-1H-purine-2,6(3H,7H)-dione 482056 2,7,8-Trihydroxy-3-phenyl-1,4-dibenzofurandione 482339 2,5-Dihydroxy-3-(4-hydroxyphenyl)-6-phenyl-1,4-benzoquinone 482340 2,5-Dihydroxy-3-(3,4-dihydroxyphenyl)-6-phenyl-1,4-benzoquinone 482341 2,5-Dihydroxy-3-phenyl-6-(3,4,5-trihydroxyphenyl)-1,4-benzoquinone 484626 SID11532953 485100 imatinib mesilate 485215 Ghrelin 487550 (4R,7S,10S,13S,16R,19S,22S,25R)-16-((1H-indol-3-yl)methyl)-25-amino-13-(4-aminobutyl)-7,19,22-tribenzyl-10-((R)-1-hydroxyethyl)-6,9,12,15,18,21,24-heptaoxo-1,2-dithia-5,8,11,14,17,20,23-heptaazacyclohexacosane-4-carboxylic acid 489669 5-(2-(4-(2-(dimethylamino)ethoxy)phenyl)-5-(pyridin-4-yl)-1H-imidazol-4-yl)-2,3-dihydroinden-1-one oxime 495699 H-Dmt-Tic-Gly-NH-Bzl 496153 3-(4-(N-(4-chlorophenyl)-N-(2-oxo-2-(2-(2-oxoindolin-3-ylidene)hydrazinyl)ethyl)sulfamoyl)phenyl)-N-(3-(dimethylamino)propyl)propanamide 496910 SID17389966 498812 N6-Cyclopentyl-9H-(5-chloro-5-deoxy-beta-D-ribofuranosyl)adenine 499059 N6-((+/-)-endo-norborn-2-yl)adenosine 506931 methyl 5-((3-(4,4-diphenylpiperidin-1-yl)propyl)carbamoyl)-2,6-dimethyl-4-(4-nitrophenyl)-1,4-dihydropyridine-3-carboxylate 509596 6-Methyl-7-[3-(4-methylpiperazin-1-yl)-propoxy]-4-(pyridin-2-ylamino)-quinoline-3-carbonitrile 509597 6-Methyl-7-(3-morpholinopropoxy)-4-(benzothiazol-2-ylamino)-quinoline-3-carbonitrile 509598 6-Methyl-7-[3-(piperidin-1-yl)-propoxy]-4-(benzothiazol-2-ylamino)-quinoline-3-carbonitrile 509599 6-Methyl-7-[3-(4-methylpiperazin-1-yl)-propoxy]-4-(6-methyl-benzothiazol-2-ylamino)-quinoline-3-carbonitrile 509681 6-methyl-4-(6-methylbenzo[d]thiazol-2-ylamino)-7-(3-(piperidin-1-yl)propoxy)quinoline-3-carbonitrile 509682 6-Methyl-7-[3-(4-methylpiperazin-1-yl)-propoxy]-4-[6-(trifluoromethoxy)-benzothiazol-2-ylamino]-quinoline-3-carbonitrile 509684 6-Methoxy-7-[3-(4-methylpiperazin-1-yl)-propoxy]-4-(benzothiazol-2-ylamino)-quinoline-3-carbonitrile 509685 6-Methoxy-7-[3-(4-methylpiperazin-1-yl)-propoxy]-4-[6-(trifluoromethoxy)-benzothiazol-2-ylamino]-quinoline-3-carbonitrile 509758 6-Methoxy-7-[2-(piperidin-1-yl)-ethoxyl]-4-(benzothiazol-2-ylamino)-quinoline-3-carbonitrile 509760 6-Methoxy-7-[2-(4-methylpiperazin-1-yl)-ethoxy]-4-(benzothiazol-2-ylamino)-quinoline-3-carbonitrile 509761 6-Methoxy-7-[3-(4-methylpiperazin-1-yl)-propoxy]-4-(1H-benzimidazol-2-ylamino)-quinoline-3-carbonitrile 510042 H-Dmt-Tic-Gly-NH-Ph 510194 (S)-3-((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamido)-3-(1H-benzo[d]imidazol-2-yl)propanoic acid 510514 5-(3-(pyridin-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510515 5-(1-methyl-3-(pyridin-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510516 5-(1-methyl-5-(pyridin-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510517 5-(1-ethyl-3-(pyridin-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510518 5-(1-cyclopentyl-3-(pyridin-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510604 cis-5-(1-(2-hydroxycyclopentyl)-3-(pyridin-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510605 trans-5-(1-(2-hydroxycyclopentyl)-3-(pyridin-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510606 cis-5-(1-(3-hydroxycyclohexyl)-3-(pyridin-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510607 trans-5-(1-(3-hydroxycyclohexyl)-3-(pyridin-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510608 5-(1-(2-methoxyethyl)-3-(pyridin-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510783 (E)-5-(1-(2-hydroxyethyl)-3-(pyridin-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510784 5-(1-(3-hydroxypropyl)-3-(pyridin-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510785 5-(1-(2,3-dihydroxypropyl)-3-(pyridin-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510786 5-(1-(1,3-dihydroxypropan-2-yl)-3-(pyridin-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510787 5-(1-(2-aminoethyl)-3-(pyridin-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510846 5-(1-(2-(dimethylamino)ethyl)-3-(pyridin-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510847 5-(1-(3-aminopropyl)-3-(pyridin-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510848 5-(1-(3-(dimethylamino)propyl)-3-(pyridin-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510849 5-(1-(piperidin-4-yl)-3-(pyridin-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510850 5-(1-(1-methylpiperidin-4-yl)-3-(pyridin-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510911 5-(1-(piperidin-4-ylmethyl)-3-(pyridin-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510912 5-(3-(pyridin-4-yl)-1-(tetrahydro-2H-pyran-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510913 5-(1-(piperidin-3-ylmethyl)-3-(pyridin-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510914 5-(1-(3-(methylamino)cyclohexyl)-3-(pyridin-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510915 5-(1-methyl-3-(1-methyl-1H-indazol-5-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510984 6-(1-methyl-3-(pyridin-4-yl)-1H-pyrazol-4-yl)-3,4-dihydroisoquinolin-1(2H)-one oxime 510985 5-(1-methyl-3-(pyridin-3-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510986 6-(1-methyl-3-(pyridin-4-yl)-1H-pyrazol-4-yl)isoindolin-1-one 510987 5-(1-methyl-3-(oxazol-5-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 510988 6-(1-methyl-3-(pyridin-4-yl)-1H-pyrazol-4-yl)-1H-indazole 510989 (E)-5-(3-(2-aminopyridin-4-yl)-1-methyl-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 511044 5-(3-(2-hydroxypyridin-4-yl)-1-methyl-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 511045 5-(1-methyl-3-(pyrimidin-4-yl)-1H-pyrazol-4-yl)-2,3-dihydroinden-1-one oxime 511046 N'-hydroxy-4-(1-methyl-3-(pyridin-4-yl)-1H-pyrazol-4-yl)benzamidine 511048 4-(4-(4-(1H-pyrazol-3-yl)phenyl)-1-methyl-1H-pyrazol-3-yl)pyridine 511049 4-(1-methyl-4-(4-(4-methyl-1H-pyrazol-3-yl)phenyl)-1H-pyrazol-3-yl)pyridine 511120 6-(1-methyl-3-pyridin-4-yl-1H-pyrazol-4-yl)-2,4-dihydro-indeno[1,2-c]pyrazole 511139 6-methoxy-5-(2-morpholinoethyl)-2-((1S,2S,4R)-1,3,3-trimethylbicyclo[2.2.1]heptan-2-yl)-2H-pyrido[4,3-b]indol-1(5H)-one 512926 TCMDC-135395 513787 (S)-1-(4-bromo-2,5-dimethoxyphenyl)propan-2-amine 517610 SID26751905 522679 3-(8-azabicyclo[3.2.1]octan-3-yl)-2-phenyl-1H-indole 522730 methyl 3-((4-(N-methyl-2-(4-methylpiperazin-1-yl)acetamido)phenylamino)(phenyl)methylene)-2-oxoindoline-6-carboxylate 530674 TCMDC-123476 543229 [5-(5-Amino-tetrazol-1-yl)-2-methoxy-benzyl]-((2S,3S)-2-phenyl-piperidin-3-yl)-amine dihydrochloride 543231 (2-Methoxy-5-tetrazol-1-yl-benzyl)-((2S,3S)-2-phenyl-piperidin-3-yl)-amine dihydrochloride 543232 [5-(5-Methanesulfonyl-tetrazol-1-yl)-2-methoxy-benzyl]-((2S,3S)-2-phenyl-piperidin-3-yl)-amine dihydrochloride 543234 [5-(5-Diethylamino-tetrazol-1-yl)-2-methoxy-benzyl]-((2S,3S)-2-phenyl-piperidin-3-yl)-amine dihydrochloride 543245 [5-(5-Ethyl-tetrazol-1-yl)-2-methoxy-benzyl]-((2S,3S)-2-phenyl-piperidin-3-yl)-amine dihydrochloride 543248 [2-Methoxy-5-(5-methylsulfanyl-tetrazol-1-yl)-benzyl]-((2S,3S)-2-phenyl-piperidin-3-yl)-amine dihydrochloride 543252 [2-Methoxy-5-(5-propyl-tetrazol-1-yl)-benzyl]-((2S,3S)-2-phenyl-piperidin-3-yl)-amine dihydrochloride 543383 (2-Chloro-4-{2-[2-hydroxy-2-(4-hydroxy-phenyl)-1-methyl-ethylamino]-ethyl}-phenoxy)-acetic acid ethyl ester hydrochloride 543635 1-(9-Ethylamino-2-furan-2-yl-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-methoxy-phenyl)-urea hydrochloride 543638 N*9*-Ethyl-2-furan-2-yl-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine-5,9-diamine hydrochloride 543650 2-Furan-2-yl-8-methyl-9-(4-methyl-piperazin-1-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine dihydrochloride 543678 1,4,5,6-Tetrahydro-pyrimidine-5-carboxylic acid but-2-ynyl ester hydrochloride 543680 1,4,5,6-Tetrahydro-pyrimidine-5-carboxylic acid prop-2-ynyl ester hydrochloride 543692 1,4,5,6-Tetrahydro-pyrimidine-5-carboxylic acid but-3-ynyl ester hydrochloride 544231 1-Propyl-3-m-tolyl-piperidine hydrochloride 544338 3-Phenyl-1-propyl-piperidine hydrochloride 544620 3-(4-Methyl-cyclohexyl)-1-propyl-piperidine hydrochloride 544623 3-(3-Methyl-cyclohexyl)-1-propyl-piperidine hydrochloride 544635 1-Propyl-3-o-tolyl-piperidine hydrochloride 544636 3-Cyclohexyl-1-propyl-piperidine hydrochloride 544740 1-Propyl-3-p-tolyl-piperidine hydrochloride 544960 6-[(2-Hydroxy-ethyl)-propyl-amino]-5,6,7,8-tetrahydro-naphthalene-2,3-diol hydrobromide 545010 6-(2-Chloro-ethylamino)-5,6,7,8-tetrahydro-naphthalene-2,3-diol hydrochloride 545023 6-[(2-Chloro-ethyl)-methyl-amino]-5,6,7,8-tetrahydro-naphthalene-2,3-diol hydrochloride 545026 N-[4-(7-Cyano-3,4-dihydro-1H-isoquinolin-2-yl)-butyl]-3-(1H-indol-3-yl)-acrylamide 545051 6-(2-Bromo-ethylamino)-5,6,7,8-tetrahydro-naphthalene-2,3-diol hydrobromide 545052 Trifluoro-methanesulfonic acid 2-[4-(3-1H-indol-3-yl-acryloylamino)-butyl]-1,2,3,4-tetrahydro-isoquinolin-7-yl ester 545083 6-[(2-Chloro-ethyl)-methyl-amino]-5,6,7,8-tetrahydro-naphthalene-1,2-diol hydrochloride 545098 6-(2-Bromo-propylamino)-5,6,7,8-tetrahydro-naphthalene-2,3-diol hydrobromide 545249 3-(4-tert-Butyl-benzyl)-1,2,3,4,4a,5,6,10b-octahydro-benzo[f]isoquinoline hydrochloride 545268 3-Butyl-2,3,4,5,6,7-hexahydro-1H-benzo[3,4]cyclohepta[1,2-c]pyridine hydrochloride 545271 3-[2-(4-Nitro-phenyl)-ethyl]-1,2,3,4,4a,5,6,10b-octahydro-benzo[f]isoquinoline hydrochloride 545278 2-Butyl-2,3,4,9-tetrahydro-1H-indeno[2,1-c]pyridine hydrochloride 545287 3-Cyclohexyl-1,2,3,4,4a,5,6,10b-octahydro-benzo[f]isoquinoline hydrochloride 545329 3-Butyl-1,2,3,4,4a,5,6,10b-octahydro-benzo[f]isoquinoline hydrochloride 545340 3-Butyl-2,3,4,4a,5,6,7,11b-octahydro-1H-benzo[3,4]cyclohepta[1,2-c]pyridine hydrochloride 545492 Benzyl-[2-(5-chloro-2-methoxy-phenyl)-3H-imidazol-4-ylmethyl]-methyl-amine dihydrochloride 545500 (4aS,9aR)-4a-Ethyl-2-(tetrahydro-furan-2-ylmethyl)-1,2,3,4,4a,9a-hexahydro-benzo[4,5]furo[2,3-c]pyridin-6-ol hydrochloride 545538 (4aS,9aR)-2-Cyclobutylmethyl-4a-ethyl-1,2,3,4,4a,9a-hexahydro-benzo[4,5]furo[2,3-c]pyridin-6-ol hydrochloride 545555 (4aS,9aR)-4a-Ethyl-2-furan-3-ylmethyl-1,2,3,4,4a,9a-hexahydro-benzo[4,5]furo[2,3-c]pyridin-6-ol hydrochloride 545558 (4aS,9aR)-4a-Ethyl-2-furan-2-ylmethyl-1,2,3,4,4a,9a-hexahydro-benzo[4,5]furo[2,3-c]pyridin-6-ol hydrochloride 545561 Benzyl-[2-(5-bromo-2-methoxy-phenyl)-3H-imidazol-4-ylmethyl]-methyl-amine dihydrochloride 545597 4-Naphthalen-1-ylmethyl-1H-imidazole hydrochloride 545614 Benzyl-[2-(3,4-dimethoxy-phenyl)-3H-imidazol-4-ylmethyl]-methyl-amine dihydrochloride 545615 (2E)-N'-[2-(3,4-dichlorophenyl)ethyl]-2-[(5-hydroxy-1H-indol-3-yl)methylene]hydrazinecarboximidamide hydrochloride 545627 (1H-Imidazol-4-yl)-naphthalen-1-yl-methanol hydrochloride 545633 (2E)-2-[(5-hydroxy-1H-indol-3-yl)methylene]hydrazinecarboximidamide hydrochloride 545674 (2H-Benzo[1,4]oxazin-3-yl)-[5-(4-quinolin-2-yl-piperazin-1-yl)-pentyl]-amine hydrobromide 545699 4-(Methoxy-naphthalen-1-yl-methyl)-1H-imidazole hydrochloride 545873 (1R,3S)Dimethyl-(2-methyl-4-phenyl-1,2,3,4-tetrahydro-naphthalen-2-yl)-amine hydrochloride 545946 trans-Allyl-(4-phenyl-1,2,3,4-tetrahydro-naphthalen-2-yl)-amine hydrochloride 546006 7-Fluoro-2-hexyl-10-(4-methyl-piperazin-1-yl)-2,4-dihydro-2,3,4,9-tetraaza-benzo[f]azulene hydrochloride 546009 3-Chloro-6-dimethylamino-6-methyl-8-phenyl-5,6,7,8-tetrahydro-naphthalen-2-ol hydrochloride 546082 3'-(4,5-Dihydro-1H-imidazol-2-ylamino)-2'-methyl-biphenyl-3-carbonitrile hydrochloride 546154 Biphenyl-2-carboxylic acid [3-chloro-4-((S)-3,4,11,11a-tetrahydro-1H,5H-2-oxa-4a,10-diaza-dibenzo[a,d]cycloheptene-10-carbonyl)-phenyl]-amide hydrochloride 546304 (S)-1-Phenoxy-3-[4-(4-phenoxy-phenyl)-piperidin-1-yl]-propan-2-ol hydrochloride 546306 1-Aminomethyl-3-cyclohexyl-6-methyl-isochroman-5-ol hydrobromide 546312 1-Aminomethyl-isochroman-5,6-diol hydrobromide 546313 1-(4-Pyrrolidin-1-yl-phenyl)-cyclopentanecarboxylic acid 2-diethylamino-ethyl ester hydrochloride 546314 1-(4-Tetrazol-1-yl-phenyl)-cyclopentanecarboxylic acid 2-diethylamino-ethyl ester hydrochloride 546323 1-(4-Nitro-phenyl)-cyclopentanecarboxylic acid 2-diethylamino-ethyl ester hydrochloride 546325 4-[4-(4-Fluoro-benzyl)-phenyl]-1-((E)-3-phenyl-allyl)-piperidine hydrochloride 546344 3-Cyclohexyl-6-methyl-1-methylaminomethyl-isochroman-5-ol hydrobromide 546361 1-Phenoxy-3-[4-(4-phenoxy-phenyl)-piperidin-1-yl]-propan-2-ol hydrochloride 546369 3-Cyclohexyl-1-dimethylaminomethyl-6-methyl-isochroman-5-ol hydrochloride 546370 1-Aminomethyl-6-methoxy-3-phenyl-isochroman-5-ol hydrochloride 546445 4-(4-Phenoxy-phenyl)-1-((E)-3-phenyl-allyl)-piperidine hydrochloride 546485 1-(4-Cyano-phenyl)-cyclopentanecarboxylic acid 2-diethylamino-ethyl ester hydrochloride 546488 3-Cyclohexyl-6-methyl-1-propylaminomethyl-isochroman-5-ol hydrochloride 546489 1-Aminomethyl-6-bromo-3-phenyl-isochroman-5-ol hydrochloride 546499 (R)-1-Phenoxy-3-[4-(4-phenoxy-phenyl)-piperidin-1-yl]-propan-2-ol hydrochloride 546508 1-(4-Iodo-phenyl)-cyclopentanecarboxylic acid 2-diethylamino-ethyl ester hydrochloride 546658 SID17405009 546730 SID26747513 547219 (3,5-Dimethoxy-phenyl)-(6,7-dimethoxy-quinazolin-4-yl)-amine hydrochloride 547305 (6,7-Dimethoxy-quinazolin-4-yl)-(3,4,5-trimethoxy-phenyl)-amine hydrochloride 547398 2-[2-(2-{2-[4-(1-Methyl-1,2,5,6-tetrahydro-pyridin-3-yl)-[1,2,5]thiadiazol-3-yloxy]-ethoxy}-ethoxy)-ethoxy]-ethanol hydrochloride 547404 12-[4-(1-Methyl-1,2,5,6-tetrahydro-pyridin-3-yl)-[1,2,5]thiadiazol-3-yloxy]-dodecan-1-ol hydrochloride 547426 5-(4-{2-[2-(2-Ethoxy-ethoxy)-ethoxy]-ethoxy}-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2,3,6-tetrahydro-pyridine hydrochloride 547428 (6,7-Dimethoxy-quinazolin-4-yl)-phenyl-amine hydrochloride 547448 (3-Chloro-phenyl)-quinazolin-4-yl-amine hydrochloride 547496 Canertinib dihydrochloride 547520 Acetic acid 2-[2-(2-{2-[4-(1-methyl-1,2,5,6-tetrahydro-pyridin-3-yl)-[1,2,5]thiadiazol-3-yloxy]-ethoxy}-ethoxy)-ethoxy]-ethyl ester hydrochloride 547527 5-{4-[2-(2-{2-[2-(4-Methoxy-[1,2,5]thiadiazol-3-yloxy)-ethoxy]-ethoxy}-ethoxy)-ethoxy]-[1,2,5]thiadiazol-3-yl}-1-methyl-1,2,3,6-tetrahydro-pyridine hydrochloride 547559 5-[4-(2-{2-[2-(2-Ethoxy-ethoxy)-ethoxy]-ethoxy}-ethoxy)-[1,2,5]thiadiazol-3-yl]-1-methyl-1,2,3,6-tetrahydro-pyridine hydrochloride 547567 6-Ethyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol hydrochloride 547602 SID47195871 547610 6-(2-Hydroxy-ethyl)-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol hydrochloride 548162 1N-{2-[2-hydroxy-(1R,2S,4aR,13bS,14aS)-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroisoquino[3,2-a]b-carbolin-1-ylcarboxamido]ethyl}-2-hydroxy-(1R,2S,4aR,13bS,14aS)-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroisoquino[3,2 dihydrochloride 548178 1N-{7-[2-hydroxy-(1R,2S,4aR,13bS,14aS)-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroisoquino[3,2-a]b-carbolin-1-ylcarboxamido]heptyl}-2-hydroxy-(1R,2S,4aR,13bS,14aS)-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroisoquino[3, dihydrochloride 548291 1N-{5-[2-hydroxy-(1R,2S,4aR,13bS,14aS)-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroisoquino[3,2-a]b-carbolin-1-ylcarboxamido]pentyl}-2-hydroxy-(1R,2S,4aR,13bS,14aS)-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroisoquino[3, dihydrochloride 548313 1N-{6-[2-hydroxy-(1R,2S,4aR,13bS,14aS)-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroisoquino[3,2-a]b-carbolin-1-ylcarboxamido]hexyl}-2-hydroxy-(1R,2S,4aR,13bS,14aS)-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroisoquino[3,2 dihydrochloride 548364 1-[(R)-5-(3-Aza-bicyclo[3.2.2]non-3-yl)-1-methyl-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl]-3-m-tolyl-urea hydrochloride 548492 1-((S)-5-Azepan-1-yl-1-methyl-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-m-tolyl-urea hydrochloride 548636 N-(5-Amino-pentyl)-2-(6-bromo-2-naphthalen-2-yl-4-oxo-4H-quinazolin-3-yl)-acetamide hydrochloride 548657 N-(6-Amino-hexyl)-2-(2-naphthalen-2-yl-4-oxo-6-phenyl-4H-quinazolin-3-yl)-acetamide hydrochloride 548663 N-(5-Amino-pentyl)-2-(4-oxo-2-phenethyl-6-phenyl-4H-quinazolin-3-yl)-acetamide hydrochloride 548667 N-[1-(8-Aza-spiro[4.5]decane-8-carbonyl)-3-(2-diethylamino-ethylcarbamoyl)-propyl]-3,5-dichloro-benzamide hydrochloride 548683 3-Chloro-N-[1-(3,3-dimethyl-butylcarbamoyl)-4-(4-methyl-piperazin-1-yl)-4-oxo-butyl]-benzamide hydrochloride 548685 3,4-Dichloro-N-[1-dipentylcarbamoyl-4-(4-methyl-piperazin-1-yl)-4-oxo-butyl]-benzamide hydrochloride 548743 SB-200646 hydrochloride 548769 N-[1-(3-Aza-spiro[5.5]undecane-3-carbonyl)-4-(4-methyl-piperazin-1-yl)-4-oxo-butyl]-3,5-dichloro-benzamide hydrochloride 548857 1-(4-Chloro-phenyl)-5-(2,4-dichloro-phenyl)-1H-[1,2,4]triazole-3-carboxylic acid piperidin-1-ylamide dihydrochloride 548900 5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-1H-[1,2,4]triazole-3-carboxylic acid piperidin-1-ylamide dihydrochloride 548957 N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-N-(pyridin-2-yl)cyclohexanecarboxamide, trihydrochloride 548966 4-Bromo-N-{4-[(4-dimethylamino-quinazolin-2-ylamino)-methyl]-cyclohexylmethyl}-2-trifluoromethoxy-benzenesulfonamide hydrochloride 549003 1-(3-Aminomethyl-4-chloro-2-hydroxy-phenyl)-3-(2-bromo-phenyl)-urea hydrochloride 549055 2-Amino-2-methyl-1-(1-methyl-1H-indol-3-yl)-propan-1-one hydrochloride 549111 (2S,5S)-5-Cyclopropyl-piperazine-2-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide dihydrochloride 549113 N-(4-Acetyl-phenyl)-2-[4-(6-methyl-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide 549116 (2S,5S)-5-tert-Butyl-piperazine-2-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide dihydrochloride 549119 N-(4-Acetyl-phenyl)-2-[4-(2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide 549121 2-[4-(5-Chloro-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(9-ethyl-9H-carbazol-3-yl)-acetamide 549140 (2S,5S)-5-Isopropyl-piperazine-2-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide dihydrochloride 549141 (2S,5S)-5-Ethyl-piperazine-2-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide dihydrochloride 549160 N-(9-Hydroxy-9H-fluoren-3-yl)-2-[4-(8-methyl-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide 549161 2-[4-(6-Chloro-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(4-cyclohexyl-phenyl)-acetamide 549164 2-[4-(2-Oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(4-phenoxy-phenyl)-acetamide 549166 2-[4-(2-Oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(9-oxo-9H-fluoren-4-yl)-acetamide 549167 N-(4-Benzoyl-phenyl)-2-[4-(8-methyl-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide 549169 2-[4-(6-Chloro-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(4-cyano-phenyl)-acetamide hydrochloride 549173 2-[4-(6-Chloro-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(9-hydroxy-9H-fluoren-3-yl)-acetamide 549182 N-(4-Acetyl-phenyl)-2-[4-(6-chloro-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide 549189 N-(4-Chloro-phenyl)-2-[4-(2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide 549194 2-[4-(6-Chloro-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(4-phenoxy-phenyl)-acetamide 549195 N-(9-Hydroxy-9H-fluoren-3-yl)-2-[4-(2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide 549205 (2S,5S)-5-Methyl-piperazine-2-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide dihydrochloride 549210 N-(9-Methyl-9H-carbazol-3-yl)-2-[4-(2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide 549212 (2S,5S)-5-(1-Methyl-cyclopropyl)-piperazine-2-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide dihydrochloride 549215 3-Chloro-4-[4-(4-hydroxy-4-pyrimidin-2-yl-piperidin-1-yl)-butyl]-4H-benzo[f][1,4]oxazepin-5-one hydrochloride 549216 3-Chloro-4-[4-(4-pyrimidin-2-yl-3,6-dihydro-2H-pyridin-1-yl)-butyl]-4H-benzo[f][1,4]oxazepin-5-one hydrochloride 549226 (R)-1-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethoxy)-5-chlorophenyl)urea hydrochloride 549353 5-[[(3-pyridyl)amino]carbonyl]amino-8-methyl-2-(2-furyl)-pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine hydrochloride 549360 5-[[(2-pyridyl)amino]carbonyl]amino-8-methyl-2-(2-furyl)-pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine hydrochloride 549420 rac-1-Butyl-3-isobutyl-9-(4-phenoxybenzyl)-1,4,9-triazaspiro[5.5]undecane-2,5-dione hydrochloride 549421 (3R)-3-cyclohexylmethyl-9-(6-phenylhexyl)-1-propyl-1,4,9-triazaspiro[5.5]undeca-2,5-dione hydrochloride 549432 rac-3-Isobutyl-9-(4-phenoxybenzyl)-1-propyl-1,4,9-triazaspiro[5.5]undecane-2,5-dione hydrochloride 549434 (R)-7-(4-chlorophenyl)-3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-4H-chromen-4-one hydrochloride 549451 (3R)-3-(2-methylpropyl)-9-(6-phenylhexyl)-1-propyl-1,4,9-triazaspiro[5.5]undeca-2,5-dione hydrochloride 549455 2-methyl-3-(1-(3-(piperidin-1-yl)propyl)piperidin-4-yl)-1H-indole dihydrochloride 549456 1-(1-(3-(piperidin-1-yl)propyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one dihydrochloride 549461 (3S)-3-(2-methylpropyl)-9-(6-phenylhexyl)-1-propyl-1,4,9-triazaspiro[5.5]undeca-2,5-dione hydrochloride 549462 rac-1-Butyl-3-isobutyl-9-(6-phenylhexyl)-1,4,9-triazaspiro[5.5]undecane-2,5-dione hydrochloride 549470 3-(1-(4-(piperidin-1-yl)butyl)piperidin-4-yl)-1H-indole dihydrochloride 549472 rac-1-Butyl-3-(cyclohexylmethyl)-9-(4-phenoxybenzyl)-1,4,9-triazaspiro[5.5]undecane-2,5-dione hydrochloride 549486 3-(1-(3-(piperidin-1-yl)propyl)piperidin-4-yl)-1H-indole dihydrochloride 549488 1-methyl-3-(1-(3-(piperidin-1-yl)propyl)piperidin-4-yl)-1H-indole dihydrochloride 549489 3-(1-(5-(piperidin-1-yl)pentyl)piperidin-4-yl)-1H-indole dihydrochloride 549495 S-(2-guanidylethyl)-isothiourea dihydrobromide 549496 2-{[amino(imino)methyl]thio}ethyl imidothiocarbamate dihydrobromide 549499 3-{[amino(imino)methyl]amino}propyl imidothiocarbamate dihydrobromide 549501 4-{[amino(imino)methyl]amino}butyl imidothiocarbamate dihydrobromide 549512 3-(1-(3-(piperidin-1-yl)propyl)piperidin-4-yl)benzo[d]isoxazole dihydrochloride 549513 1-(3-(4-(benzofuran-3-yl)piperidin-1-yl)propyl)piperidine dihydrochloride 549525 6-{[amino(imino)methyl]amino}hexyl imidothiocarbamate dihydrobromide 549562 (+/-)-1-[3-(3-fluorobiphenyl-2-yl)propyl]-4-[2-(4-fluorophenyl)-2-(1-isopropylpiperidin-4-yl)ethyl]piperazine trihydrochloride 549563 (+/-)-1-[3-(30-fluorobiphenyl-2-yl)propyl]-4-[2-(4-fluorophenyl)-2-(1-isopropylpiperidin-4-yl)ethyl]piperazine trihydrochloride 549564 (+/-)-1-[3-(40-fluorobiphenyl-2-yl)propyl]-4-[2-(4-fluorophenyl)-2-(1-isopropylpiperidin-4-yl)ethyl]piperazine trihydrochloride 549572 (+/-)-1-[3-(4-fluorobiphenyl-2-yl)propyl]-4-[2-(4-fluorophenyl)-2-(1-isopropylpiperidin-4-yl)ethyl]piperazine trihydrochloride 549580 (+/-)-1-[2-(4-fluorophenyl)-2-(1-methylpiperidin-4-yl)ethyl]-4-[4-(1-naphthyl)butyl]piperazine tri hydrochloride 549584 (+/-)-1-[2-(4-fluorophenyl)-2-(1-isopropylpiperidin-4-yl)ethyl]-4-[4-(2-methoxy-1-naphthyl)butyl]piperazine trihydrochloride 549585 (+/-)-1-[3-(6-fluorobiphenyl-2-yl)propyl]-4-[2-(4-fluorophenyl)-2-(1-isopropylpiperidin-4-yl)ethyl]piperazine trihydrochloride 549594 (+/-)-1-[3-(5-fluorobiphenyl-2-yl)propyl]-4-[2-(4-fluorophenyl)-2-(1-isopropylpiperidin-4-yl)ethyl]piperazinetrihydrochloride 549595 (3-(2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-phenylamino)-acetic acid hydrochloride 549601 N-(2,6-dimethylphenyl)-5-[3-(2-pyrrolidin-1-ylethoxy)phenyl]imidazo[1,5-a]pyrazin-8-amine hydrochloride 549603 N-(2,6-dimethylphenyl)-5-[4-(1-methylpiperidin-3-ylmethoxy)phenyl]imidazo[1,5-a]pyrazin-8-amine hydrochloride 549617 4-phenyl-1-(phenyl(o-tolyl)methyl)piperidin-4-ol 549630 N-methyl-N'-(1-methyl-3,5,11b-triaza-cyclopenta[a]anthracen-4-yl)-ethane-1,2-diamine hydrochloride 549648 1-(4-(4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl)-3-m-tolylurea hydrochloride 549668 1-butyl-3-(2-hydroxy-2-methyl-propyl)-9-(4-phenoxy-benzyl)-1,4,9-triaza-spiro[5.5]undecane-2,5-dione hydrochloride 549677 1-(4-(1-cyclohexyl-1-phenylprop-2-en-2-ylamino)piperidin-1-yl)-3-(pyridin-3-yl)propan-1-one 549679 2-cyclohexyl-2-phenyl-N-(1-(3-(pyridin-3-yl)propanoyl)piperidin-4-yl)acetamide 549680 2-(4-methoxy-3-(2-(piperidin-1-yl)ethoxy)phenyl)-4-methyl-2,3-dihydropyrrolo[3,4-b]indol-1(4H)-one 549692 (3R)-1-Butyl-3-isobutyl-9-(4-phenoxybenzyl)-1,4,9-triazaspiro[5.5]undecane-2,5-dione hydrochloride 549693 (R)-1-butyl-3-((R)-1-hydroxy-2-methyl-propyl)-9-(4-phenoxy-benzyl)-1,4,9-triaza-spiro[5.5]undecane-2,5-dione hydrochloride 549699 (R)-1-butyl-3-((S)-1-hydroxy-2-methyl-propyl)-9-(4-phenoxy-benzyl)-1,4,9-triaza-spiro[5.5]undecane-2,5-dione hydrochloride 549700 (S)-1-butyl-3-((R)-1-hydroxy-2-methyl-propyl)-9-(4-phenoxy-benzyl)-1,4,9-triaza-spiro[5.5]undecane-2,5-dione hydrochloride 549703 (R)-1-butyl-3-((R)-cyclohexyl-hydroxy-methyl)-9-(4-phenoxy-benzyl)-1,4,9-triaza-spiro[5.5]undecane-2,5-dione hydrochloride 550132 N-(6-Amino-hexyl)-2-(6-bromo-2-naphthalen-2-yl-4-oxo-4H-quinazolin-3-yl)-acetamide hydrochloride 550177 [2-Methoxy-5-(5-methyl-tetrazol-1-yl)-benzyl]-((2S,3S)-2-phenyl-piperidin-3-yl)-amine dihydrochloride 550182 [2-Methoxy-5-(5-phenyl-tetrazol-1-yl)-benzyl]-((2S,3S)-2-phenyl-piperidin-3-yl)-amine dihydrochloride 550214 N-(1-{4-Methoxy-3-[((2S,3S)-2-phenyl-piperidin-3-ylamino)-methyl]-phenyl}-1H-tetrazol-5-yl)-acetamide dihydrochloride 550227 [5-(5-Cyclopropyl-tetrazol-1-yl)-2-methoxy-benzyl]-((2S,3S)-2-phenyl-piperidin-3-yl)-amine dihydrochloride 550232 [2-Methoxy-5-(5-trifluoromethyl-tetrazol-1-yl)-benzyl]-((2S,3S)-2-phenyl-piperidin-3-yl)-amine dihydrochloride 550540 1,4,5,6-Tetrahydro-pyrimidine-5-carboxylic acid methyl ester hydrochloride 550544 3-((3aR,10aR)-2-Methyl-2,3,3a,4,10,10a-hexahydro-1H-2,4a-diaza-cyclopenta[b]fluoren-9-yl)-4-(1-methyl-1H-indol-3-yl)-pyrrole-2,5-dione hydrochloride 550887 3-(2-Methyl-cyclohexyl)-1-propyl-piperidine hydrochloride 550898 6-[Bis-(2-bromo-ethyl)-amino]-5,6,7,8-tetrahydro-naphthalene-2,3-diol hydrobromide 550920 6-[(2-Bromo-ethyl)-propyl-amino]-5,6,7,8-tetrahydro-naphthalene-2,3-diol hydrobromide 550922 3-Phenethyl-1,2,3,4,4a,5,6,10b-octahydro-benzo[f]isoquinoline hydrochloride 550961 6-[(2-Chloro-ethyl)-propyl-amino]-5,6,7,8-tetrahydro-naphthalene-2,3-diol hydrobromide 551097 3-(3,4-Dimethyl-phenyl)-1-propyl-piperidine hydrochloride 551141 6-[(2-Chloro-ethyl)-methyl-amino]-5,6,7,8-tetrahydro-naphthalen-2-ol hydrochloride 551223 11-(2-Dimethylamino-ethylsulfanyl)-6,11-dihydro-dibenzo[b,e]oxepine-2-carboxylic acid hydrochloride 551224 [11-(3-Dimethylamino-propylidene)-6,11-dihydro-dibenzo[b,e]oxepin-2-yl]-acetic acid hydrochloride 551254 Benzyl-[2-(3-methoxy-phenyl)-3H-imidazol-4-ylmethyl]-methyl-amine dihydrochloride 551269 3-(4-Methoxy-benzyl)-1,2,3,4,4a,5,6,10b-octahydro-benzo[f]isoquinoline hydrochloride 551275 3-Butyl-1,2,3,4,5,6-hexahydro-benzo[f]isoquinoline hydrochloride 551287 Benzyl-[2-(2,3-dimethoxy-phenyl)-3H-imidazol-4-ylmethyl]-methyl-amine dihydrochloride 551294 Benzyl-methyl-(2-phenyl-3H-imidazol-4-ylmethyl)-amine dihydrochloride 551299 (4aS,9aR)-2-Cyclopropylmethyl-4a-ethyl-1,2,3,4,4a,9a-hexahydro-benzo[4,5]furo[2,3-c]pyridin-6-ol hydrochloride 551303 Benzyl-[2-(5-bromo-2,3-dimethoxy-phenyl)-3H-imidazol-4-ylmethyl]-methyl-amine dihydrochloride 551308 Benzyl-[2-(2-fluoro-phenyl)-3H-imidazol-4-ylmethyl]-methyl-amine dihydrochloride 551329 Benzyl-[2-(4-fluoro-phenyl)-3H-imidazol-4-ylmethyl]-methyl-amine dihydrochloride 551375 Benzyl-[2-(2-methoxy-phenyl)-3H-imidazol-4-ylmethyl]-methyl-amine dihydrochloride 551444 Benzyl-[2-(4-methoxy-phenyl)-3H-imidazol-4-ylmethyl]-methyl-amine dihydrochloride 551459 (2H-Benzo[1,4]oxazin-3-yl)-[5-(4-phenyl-piperazin-1-yl)-pentyl]-amine hydrobromide 551501 1-Phenyl-4-((R)-2-phenyl-4,5-dihydro-1H-imidazol-4-ylmethyl)-piperazine hydrochloride 551570 trans-Diallyl-(4-phenyl-1,2,3,4-tetrahydro-naphthalen-2-yl)-amine hydrochloride 551643 Rimonabant. Hydrochloride 551644 1-(4-Amino-phenyl)-cyclopentanecarboxylic acid 2-diethylamino-ethyl ester hydrochloride 551721 1-Aminomethyl-3-phenyl-isochroman-5-ol hydrochloride 551738 1-Aminomethyl-6-bromo-3-phenyl-isochroman-5-ol hydrochloride 551811 6-(2-{2-[4-(4-Chloro-phenoxy)-piperidin-1-yl]-ethyl}-pyrrolidine-1-sulfonyl)-1H-indole hydrochloride 551830 Biphenyl-2-carboxylic acid [3-chloro-4-((S)-3,4,11,11a-tetrahydro-1H,5H-2-thia-4a,10-diaza-dibenzo[a,d]cycloheptene-10-carbonyl)-phenyl]-amide hydrochloride 551868 1-[3'-(4,5-Dihydro-1H-imidazol-2-ylamino)-2'-methyl-biphenyl-3-yl]-ethanone hydrochloride 551964 4-(3'-fluoroanilino)-6,7-dimethoxyquinazoline hydrochloride 552030 6-Isobutyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol hydrochloride 552106 SID26719789 552234 5,6,6a,7-Tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol hydrochloride 552251 SID46500370 552306 6-Isopropyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol hydrochloride 552320 6-Cyclopropylmethyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol hydrochloride 552335 Acetic acid 12-[4-(1-methyl-1,2,5,6-tetrahydro-pyridin-3-yl)-[1,2,5]thiadiazol-3-yloxy]-dodecyl ester hydrochloride 552361 1N-{4-[2-hydroxy-(1R,2S,4aR,13bS,14aS)-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroisoquino[3,2-a]b-carbolin-1-ylcarboxamido]butyl}-2-hydroxy-(1R,2S,4aR,13bS,14aS)-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroisoquino[3,2 dihydrochloride 552459 1N-{3-[2-hydroxy-(1R,2S,4aR,13bS,14aS)-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroisoquino[3,2-a]b-carbolin-1-ylcarboxamido]propyl}-2-hydroxy-(1R,2S,4aR,13bS,14aS)-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroisoquino[3, dihydrochloride 552521 N-(6-Amino-hexyl)-2-(6-bromo-4-oxo-2-phenethyl-4H-quinazolin-3-yl)-acetamide hydrochloride 552535 1-[(S)-5-(3-Aza-bicyclo[3.2.2]non-3-yl)-1-methyl-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl]-3-m-tolyl-urea hydrochloride 552582 1N-{8-[2-hydroxy-(1R,2S,4aR,13bS,14aS)-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroisoquino[3,2-a]b-carbolin-1-ylcarboxamido]octyl}-2-hydroxy-(1R,2S,4aR,13bS,14aS)-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroisoquino[3,2 dihydrochloride 552645 N-(5-Amino-pentyl)-2-(2-naphthalen-2-yl-4-oxo-6-phenyl-4H-quinazolin-3-yl)-acetamide hydrochloride 552670 Naphthalene-2-carboxylic acid [1-dipentylcarbamoyl-4-(4-methyl-piperazin-1-yl)-4-oxo-butyl]-amide hydrochloride 552674 N-[1-(8-Aza-spiro[4.5]decane-8-carbonyl)-4-(4-methyl-piperazin-1-yl)-4-oxo-butyl]-3,5-dichloro-benzamide hydrochloride 552687 6-Amino-2-[2-(6-chloro-2-naphthalen-2-yl-4-oxo-4H-quinazolin-3-yl)-acetylamino]-hexanoic acid methyl ester hydrochloride 552697 N-(5-Amino-pentyl)-2-(6-bromo-4-oxo-2-phenethyl-4H-quinazolin-3-yl)-acetamide hydrochloride 552698 N-(6-Amino-hexyl)-2-(4-oxo-2-phenethyl-6-phenyl-4H-quinazolin-3-yl)-acetamide hydrochloride 552851 2-{3-[3-(2,5-Dioxo-4-phenylamino-2,5-dihydro-1H-pyrrol-3-yl)-indol-1-yl]-propyl}-isothiourea hydrobromide 552855 (2S,5R)-5-Ethyl-4-methyl-piperazine-2-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide dihydrochloride 552856 Naphthalene-2-carboxylic acid {4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-amide hydrochloride 552868 N-(4-Benzoyl-phenyl)-2-[4-(6-chloro-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide hydrochloride 552879 2-[4-(6-Chloro-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(9-oxo-9H-fluoren-2-yl)-acetamide 552885 2-[4-(6-Chloro-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(9-oxo-9H-fluoren-3-yl)-acetamide 552900 N-(4-Cyano-phenyl)-2-[4-(2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide hydrochloride 552901 (2S,5S)-5-Ethyl-4-methyl-piperazine-2-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide dihydrochloride 552903 N-(9-Ethyl-9H-carbazol-3-yl)-2-[4-(8-methoxy-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide 552979 2-[4-(8-Methyl-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(9-oxo-9H-fluoren-3-yl)-acetamide 552994 3-Chloro-4-[4-(4-pyrimidin-2-yl-piperidin-1-yl)-butyl]-4H-benzo[f][1,4]oxazepin-5-one hydrochloride 552995 2-[4-(6-Methyl-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(9-oxo-9H-fluoren-2-yl)-acetamide 553000 N-(9-Ethyl-9H-carbazol-3-yl)-2-[4-(2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide 553004 2-[4-(6-Methyl-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(4-phenoxy-phenyl)-acetamide 553008 2-[4-(2-Oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(9-oxo-9H-fluoren-3-yl)-acetamide 553028 N-(9-Ethyl-9H-carbazol-3-yl)-2-[4-(8-methyl-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide 553043 6-fluoro-3-(1-(3-(piperidin-1-yl)propyl)piperidin-4-yl)-1H-indole dihydrochloride 553046 6-(furan-3-yl)-2-(3H-imidazo[4,5-c]pyridin-3-yl)-N-((S)-1-methoxypropan-2-yl)pyrimidin-4-amine 553054 4-phenyl-1-(phenyl(o-tolyl)methyl)piperidin-4-ol 553061 (+/-)-1-(3-biphenyl-2-ylpropyl)-4-[2-(4-fluorophenyl)-2-(1-isopropylpiperidin-4-yl)ethyl]piperazine tri hydrochloride 553066 (3S)-3-cyclohexylmethyl-9-(6-phenylhexyl)-1-propyl-1,4,9-triazaspiro[5.5]undeca-2,5-dione hydrochloride 553072 (RS)-1-butyl-3-(cyclohexylmethyl)-9-((2,3-dihydrobenzo[b][1,4]dioxin-6-yl)methyl)-1,4,9-triazaspiro[5.5]undecane-2,5-dione hydrochloride 553074 rac-9-Benzyl-1-butyl-3-isobutyl-1,4,9-triazaspiro[5.5]undecane-2,5-dione hydrochloride 553090 5-fluoro-3-(1-(3-(piperidin-1-yl)propyl)piperidin-4-yl)-1H-indole dihydrochloride 553097 (3S)-1,9-dibenzyl-3-(2-methylpropyl)-1,4,9-triazaspiro[5.5]-undeca-2,5-dione hydrochloride 553099 9-(4-allyloxyphenylmethyl)-1-butyl-3-cyclohexyl-1,4,9-triazaspiro[5.5]undeca-2,5-dione hydrochloride 553101 ethyl 3-(N-benzyl-N-methylaminomethyl)-7-(2,6-difluorobenzyl)-4,7-dihydro-2-(4-isobutyrylamidophenyl)-4-oxothieno[2,3-b]pyridine-5-carboxylate hydrochloride 553102 8-(1-phenyl-cyclohexyl)-4-propyl-2,8-diaza-spiro[4.5]decan-1-one 553103 1-butyl-9-((2,3-dihydrobenzo[b][1,4]dioxin-6-yl)methyl)-3-isobutyl-1,4,9-triazaspiro[5.5]undecane-2,5-dione hydrochloride 553104 rac-1-Butyl-3-(cyclohexylmethyl)-9-(4-methoxybenzyl)-1,4,9-triazaspiro[5.5]undecane-2,5-dione hydrochloride 553161 (3R)-1,9-dibenzyl-3-(2-methylpropyl)-1,4,9-triazaspiro[5.5]-undeca-2,5-dione hydrochloride 553162 N-(2-{[amino(imino)methyl]amino}ethyl)guanidine dihydrobromide 553167 1N-{9-[2-hydroxy-(1R,2S,4aR,13bS,14aS)-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroisoquino[3,2-a]b-carbolin-1-ylcarboxamido]nonyl}-2-hydroxy-(1R,2S,4aR,13bS,14aS)-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroisoquino[3,2 dihydrochloride 553172 22-hydroxy-12-methyl-15-oxa-8-thia-9,12,21,23-tetraazapentacyclo[14.6.2.1^{6,9}.0^{2,7}.0^{20,24}]pentacosa-1(23),2(7),3,5,16(24),17,19,21-octaen-25-one hydrochloride 553189 (+/-)-1-[3-(20-fluorobiphenyl-2-yl)propyl]-4-[2-(4-fluorophenyl)-2-(1-isopropylpiperidin-4-yl)ethyl]piperazinetri hydrochloride 553207 (S)-1-butyl-3-((S)-1-hydroxy-2-methyl-propyl)-9-(4-phenoxy-benzyl)-1,4,9-triaza-spiro[5.5]undecane-2,5-dione hydrochloride 553208 5-(1,4-diazepan-1-ylsulfonyl)isoquinoline 553212 2-(2-hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurine hydrochloride 553215 (4-(3-(2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-phenyl)-imidazol-1-yl)-acetic acid hydrochloride sals 553228 (3S)-1-Butyl-3-isobutyl-9-(4-phenoxybenzyl)-1,4,9-triazaspiro[5.5]undecane-2,5-dione hydrochloride 553314 (R)-N-(1-(3-(4-fluorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethyl)-N-(pyridin-3-ylmethyl)-2-(4-(trifluoromethyl)phenyl)acetamide 553424 1N-{12-[2-hydroxy-(1R,2S,4aR,13bS,14aS)-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroisoquino[3,2-a]b-carbolin-1-ylcarboxamido]dodecyl}-2-hydroxy-(1R,2S,4aR,13bS,14aS)-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroisoquino[ dihydrochloride 553476 1N-{10-[2-hydroxy-(1R,2S,4aR,13bS,14aS)-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroisoquino[3,2-a]b-carbolin-1-ylcarboxamido]decyl}-2-hydroxy-(1R,2S,4aR,13bS,14aS)-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroisoquino[3, dihydrochloride 553768 5-Methoxycarbonyl-1-methyl-3,6-dihydro-2H-thiopyranium 553777 3,5-Dichloro-N-(3-(3,4-dichloro-phenyl)-2-methoxyimino-5-{2-oxo-3-[2-oxo-2-(1lambda*4*-thiomorpholin-1-yl)-ethyl]-[1,4']bipiperidinyl-1'-yl}-pentyl)-N-ethyl-benzamide 553805 5-Ethoxycarbonyl-1-methyl-3,6-dihydro-2H-thiopyranium 554376 (E)-3-(2-(Purin-9-yl)vinyl)-4-methyl-N-(3-(4-methyl-1-imidazol-1-yl)-5-(trifluoromethyl)phenyl)benzamide 554672 ethyl 7-(3-(3-(3-(trifluoromethyl)phenyl)ureido)phenyl)pyrazolo[1,5-a]pyrimidine-3-carboxylate 554687 ethyl 7-(3-(3-(4-fluoro-3-(trifluoromethyl)phenyl)ureido)phenyl)pyrazolo[1,5-a]pyrimidine-3-carboxylate 554694 2,2,2-trifluoroethyl 7-(3-(3-(trifluoromethyl)benzamido)phenyl)pyrazolo[1,5-a]pyrimidine-3-carboxylate 556125 (E)-3-(2-(6-(Cyclopropylamino)-9H-purin-9-yl)vinyl)-4-methyl-N-(3-(iso-propyl)phenyl)benzamide 556324 salvinicin A 557741 Cisapride 558147 2-(dimethylamino)ethyl 7-(3-(3-(trifluoromethyl)benzamido)phenyl)pyrazolo[1,5-a]pyrimidine-3-carboxylate 558153 7-(3-(3-(4-chloro-3-(trifluoromethyl)phenyl)ureido)phenyl)-N-(2-(diethylamino)ethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide 559235 SID11110912 559593 (E)-3-(2-(6-(Cyclopropylamino)-9H-purin-9-yl)vinyl)-4-methyl-N-(3-(tert-butyl)phenyl)benzamide 559604 (E)-3-(2-(6-(Cyclopropylamino)-9H-purin-9-yl)vinyl)-4-methyl-N-(5-(tert-butyl)thiazo-2-yl)benzamide 559612 N-(3-(1H-imidazol-1-yl)-5-(trifluoromethyl)phenyl)-3-(2-(6-(cyclopropylamino)-9H-purin-9-yl)vinyl)-4-methylbenzamide 559905 ethyl 7-(3-(4-chloro-3-(trifluoromethyl)benzamido)phenyl)pyrazolo[1,5-a]pyrimidine-3-carboxylate 559919 ethyl 7-(3-(3-(4-(trifluoromethyl)phenyl)ureido)phenyl)pyrazolo[1,5-a]pyrimidine-3-carboxylate 559954 7-(3-(3-(4-chloro-3-(trifluoromethyl)phenyl)ureido)phenyl)-N-(2-morpholinoethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide 560592 (3R)-1-Azabicyclo[2.2.2]oct-3-yl9H-xanthene-9-carboxylate 561392 N-(4-Methyl-3-(2-(6-(methylamino)-9H-purin-9-yl)ethyl)phenyl)-3-(trifluoromethyl)-benzamide 561401 (E)-N-(4-Methyl-3-(2-(6-(pyridine-2-yl-amino)-9H-purin-9-yl)vinyl)phenyl)-3-(trifluoromethyl)-benzamide 561402 (E)-N-(4-Methyl-3-(2-(6-(pyrid-3-yl-amino)-9H-purin-9-yl)vinyl)phenyl)-3-(trifluoromethyl)-benzamide 561403 (E)-N-(4-Methyl-3-(2-(6-(pyrid-4-yl-amino)-9H-purin-9-yl)vinyl)phenyl)-3-(trifluoromethyl)-benzamide 561413 (E)-3-(2-(6-(Cyclopropylamino)-9H-purin-9-yl)vinyl)-4-methyl-N-(3-(trifluoromethyl)phenyl)benzamide 561421 (E)-3-(2-(6-(Cyclopropylamino)-9H-purin-9-yl)vinyl)-4-methyl-N-(2-fluoro-5-(trifluoromethyl)phenyl)benzamide 561422 (E)-3-(2-(6-(Cyclopropylamino)-9H-purin-9-yl)vinyl)-4-methyl-N-(4-chloro-3-(trifluoromethyl)phenyl)benzamide 561434 (E)-3-(2-(6-(cyclopropylamino)-9H-purin-9-yl)vinyl)-4-methyl-N-(3-(4-methyl-1H-imidazol-1-yl)-5-(trifluoromethyl)-phenyl)benzamide 561722 ethyl 7-(3-(3-(trifluoromethoxy)benzamido)phenyl)pyrazolo[1,5-a]pyrimidine-3-carboxylate 561724 ethyl 7-(3-(4-methyl-3-(trifluoromethyl)benzamido)phenyl)pyrazolo[1,5-a]pyrimidine-3-carboxylate 561725 ethyl 7-(3-(4-methoxy-3-(trifluoromethyl)benzamido)phenyl)pyrazolo[1,5-a]pyrimidine-3-carboxylate 561914 Solifenacin 562359 trans-4-((R)-1-aminoethyl)-N-(pyridin-4-yl)cyclohexanecarboxamide 563132 (E)-N-(3-(2-(6-(4-(Dimethylphosphoryl)phenylamino)-9H-purin-9-yl)-vinyl)-4-methylphenyl)-3-(trifluoromethyl)benzamide 563166 (E)-3-(2-(Purin-9-yl)vinyl)-4-methyl-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide 563381 ethyl 7-(3-(3-(trifluoromethyl)benzamido)phenyl)pyrazolo[1,5-a]pyrimidine-3-carboxylate 563409 ethyl 7-(3-(3-(4-methyl-3-(trifluoromethyl)phenyl)ureido)phenyl)pyrazolo[1,5-a]pyrimidine-3-carboxylate 563424 methyl 7-(3-(3-(trifluoromethyl)benzamido)phenyl)pyrazolo[1,5-a]pyrimidine-3-carboxylate 563448 N-(2-morpholinoethyl)-7-(3-(3-(trifluoromethyl)benzamido)phenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide 564602 1-(2-chloro-2-phenylethyl)-N-(4-methoxybenzyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 564882 (E)-N-(4-Methyl-3-(2-(6-(cyclopropylamino)-9H-purin-9-yl)vinyl)-phenyl)-3-(trifluoromethyl)benzamide 564893 (E)-N-(4-Methyl-3-(2-(6-(pyrimid-4-yl-amino)-9H-purin-9-yl)-vinyl)-phenyl)-3-(trifluoromethyl)-benzamide 565201 ethyl 7-(3-(3-(4-chloro-3-(trifluoromethyl)phenyl)ureido)phenyl)pyrazolo[1,5-a]pyrimidine-3-carboxylate 565217 N-(2-(dimethylamino)ethyl)-7-(3-(3-(trifluoromethyl)benzamido)phenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide 566385 1-(2-chloro-2-phenylethyl)-N-(4-chlorophenethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 566685 (E)-N-(4-Methyl-3-(2-(6-(methylamino)-9Hpurin-9-yl)vinyl)phenyl)-3-(trifluoromethyl)-benzamide 566697 (E)-N-(4-Methyl-3-(2-(6-(3-(N',N''-dimethylamino)propylamino)-9H-purin-9-yl)vinyl)phenyl)-3-(trifluoromethyl)benzamide 566698 (E)-1-(3-(2-(6-(Cyclopropylamino)-9H-purin-9-yl)vinyl)-4-methylphenyl)-3-(3-(trifluoromethyl)phenyl)urea 566719 (E)-3-(2-(6-(Cyclopropylamino)-9H-purin-9-yl)vinyl)-4-methyl-N-(5-(tert-butyl)oxazo-3-yl)benzamide 566720 (E)-3-(2-(6-(Cyclopropylamino)-9H-purin-9-yl)vinyl)-4-methyl-N-(1-methyl-3-(tert-butyl)pyrazo-5-yl)benzamide 566721 3-(2-(6-(cyclopropylamino)-9H-purin-9-yl)vinyl)-4-methyl-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide 566740 (E)-3-(2-(6-(Cyclopropylamino)-9H-purin-9-yl)vinyl)-4-methyl-N-[3-(morpholin-4-yl)-5-(trifluoromethyl)phenyl]benzamide 566741 (E)-3-(2-(6-(Cyclopropylamino)-9H-purin-9-yl)vinyl)-4-methyl-N-[3-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]benzamide 567055 7-(3-(3-(4-chloro-3-(trifluoromethyl)phenyl)ureido)phenyl)-N-(3-methoxypropyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide 567706 (3R)-1-Azabicyclo[2.2.2]oct-3-ylhydroxy(diphenyl)acetate 567991 (S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-ylamino)-1-oxo-3-phenylpropan-2-yl)-2-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 568329 1-tert-butyl-3-(naphthalen-1-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 568347 6-(2,6-dichlorophenyl)-2-((4-ethoxyphenyl)amino)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one 568348 N-(2-(4-((6-(2,6-dichlorophenyl)-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl)amino)phenoxy)ethyl)-N-ethylacetamide 568349 6-(2,6-dichlorophenyl)-2-((4-fluoro-3-methylphenyl)amino)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one 568350 6-(2,6-dichlorophenyl)-2-(4-fluorophenylamino)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one 570223 1-(1-(4-(6-oxo-3-phenyl-1,6-dihydropyrazin-2-yl)benzyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one 570225 1-(1-(4-(5-methyl-6-oxo-3-phenyl-1,6-dihydropyrazin-2-yl)benzyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one 570477 (1R,2R,3S,4R,5S)-4-(2-chloro-6-(cyclopentylamino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 571115 (2R,3S,4R,5R)-2-(hydroxymethyl)-5-(6-(methylamino)-2-(phenylethynyl)-9H-purin-9-yl)tetrahydrofuran-3,4-diol 572021 Naltrindole 572853 SID26751686 572872 (R)-7-hydroxy-N-((S)-1-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)-3-methylbutan-2-yl)-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 574645 6-Methyl-N5-(3-(pyrimidin-4-yl)pyridin-2-yl)-N1-(3-(trifluoromethyl)phenyl)isoquinoline-1,5-diamine 574646 6-Methyl-N5-(3-(6-(methylamino)pyrimidin-4-yl)pyridin-2-yl)-N1-(2-methylbenzo[d]thiazol-5-yl)isoquinoline-1,5-diamine 574647 6-(1-(4-Chlorophenylamino)-6-methylisoquinolin-5-yl)-N-methylquinazolin-2-amine 574663 6-(1-(3-tert-Butyl-1-methyl-1H-pyrazol-5-ylamino)-6-methylisoquinolin-5-yl)-N-methylquinazolin-2-amine 574682 N1-(4-chlorophenyl)-6-methyl-N5-(3-(pyrimidin-4-yl)pyridin-2-yl)isoquinoline-1,5-diamine 574683 N1-(4-chlorophenyl)-6-methyl-N5-(3-(6-(methylamino)pyrimidin-4-yl)pyridin-2-yl)isoquinoline-1,5-diamine 574692 3,3-Dimethyl-6-(6-methyl-5-(2-(methylamino)quinazolin-6-yl)isoquinolin-1-ylamino)indolin-2-one 574699 4-(6-Methyl-5-(3-(6-(methylamino)pyrimidin-4-yl)pyridin-2-ylamino)isoquinolin-1-ylamino)benzonitrile 574734 N1-(3-Ethynylphenyl)-6-methyl-N5-(3-(6-(methylamino)pyrimidin-4-yl)pyridin-2-yl)isoquinoline-1,5-diamine 574846 (S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid 580304 4-(2,4-dichloro-5-methoxyphenylamino)-7-(5-(morpholinomethyl)pyridin-3-yl)quinoline-3-carbonitrile 580311 4-(2,4-dichloro-5-methoxyphenylamino)-7-(6-(morpholinomethyl)pyridin-3-yl)quinoline-3-carbonitrile 580315 4-(2,4-dichloro-5-methoxyphenylamino)-7-(5-((4-methylpiperazin-1-yl)methyl)pyridin-2-yl)quinoline-3-carbonitrile 580316 4-(2,4-dichloro-5-methoxyphenylamino)-7-(5-(thiomorpholinomethyl)pyridin-2-yl)quinoline-3-carbonitrile 580317 4-(2,4-dichlorophenylamino)-7-(5-((4-methylpiperazin-1-yl)methyl)pyridin-2-yl)quinoline-3-carbonitrile 580327 4-(2,4-Dichloro-5-methoxy-phenylamino)-7-[5-(1-oxo-1lambda*4*-thiomorpholin-4-ylmethyl)-pyridin-2-yl]-quinoline-3-carbonitrile 580337 4-(2,4-dichloro-5-methoxyphenylamino)-7-(4-(morpholinomethyl)pyridin-2-yl)quinoline-3-carbonitrile 580349 4-(2,4-dichloro-5-methoxyphenylamino)-7-(5-(morpholinomethyl)pyridin-2-yl)quinoline-3-carbonitrile 580350 4-(2,4-dichloro-5-methoxyphenylamino)-6-(5-((4-methylpiperazin-1-yl)methyl)pyridin-2-yl)quinoline-3-carbonitrile 580370 4-(2,4-Dichloro-5-methoxy-phenylamino)-7-[5-(1,1-dioxo-1lambda*6*-thiomorpholin-4-ylmethyl)-pyridin-2-yl]quinoline-3-carbonitrile 580388 4-(2,4-dichloro-5-methoxyphenylamino)-7-(5-((dimethylamino)methyl)pyridin-2-yl)quinoline-3-carbonitrile 580398 7-(5-((4-methylpiperazin-1-yl)methyl)pyridin-2-yl)-4-(3,4,5-trimethoxyphenylamino)quinoline-3-carbonitrile 580428 4-(2,4-dichloro-5-methoxyphenylamino)-7-(6-(morpholinomethyl)pyridin-2-yl)quinoline-3-carbonitrile 580909 (2R,3R,4S,5R)-2-(6-(cyclobutylamino)-9H-purin-9-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol 583068 3-amino-N-(4-(6-(2,6-dichlorophenyl)-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-ylamino)phenyl)propanamide 583077 6-(2,6-dichlorophenyl)-2-(4-(2,3-dihydroxypropylamino)phenylamino)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one 583078 tert-butyl 3-(4-(6-(2,6-dichlorophenyl)-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-ylamino)phenylamino)-3-oxopropylcarbamate 583091 6-(2,6-dichlorophenyl)-2-(3-ethylphenylamino)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one 583099 6-(2,6-dichlorophenyl)-2-(3-((2,3-dihydroxypropoxy)methyl)phenylamino)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one 583100 2-(3-Aminophenylamino)-6-(2,6-dichlorophenyl)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one 583138 N-(3-(6-(2,6-dichlorophenyl)-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-ylamino)phenyl)acetamide 583139 6-(2,6-dichlorophenyl)-2-(4-(2-hydroxyethyl)phenylamino)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one 583144 2-(4-aminophenylamino)-6-(2,6-dichlorophenyl)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one 583145 N-(4-(6-(2,6-dichlorophenyl)-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-ylamino)phenyl)acetamide 583155 6-(2,6-dichlorophenyl)-8-methyl-2-(4-(3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yloxy)phenylamino)pyrido[2,3-d]pyrimidin-7(8H)-one 583160 6-(2,6-dichlorophenyl)-8-methyl-2-(4-(4-methylpiperazine-1-carbonyl)phenylamino)pyrido[2,3-d]pyrimidin-7(8H)-one 583165 6-(2,6-dichlorophenyl)-2-(4-iodophenylamino)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one 583166 2-chloro-N-(4-(6-(2,6-dichlorophenyl)-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-ylamino)phenyl)acetamide 594549 Tyr-D-Ala-Gly-Phe-Met-NH2 597216 SID11111835 604615 (E)-N-(4-(3-chloro-4-fluorophenylamino)-3-cyano-7-ethoxyquinolin-6-yl)-4-(dimethylamino)but-2-enamide 604689 2-[5-Chloro-7-(1-methyl-2-phenyl-ethylamino)-imidazo[4,5-b]pyridin-3-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 604745 5-Hydroxymethyl-3-methyl-2-[6-((S)-1-methyl-2-phenyl-ethylamino)-purin-9-yl]-tetrahydro-furan-3,4-diol 604916 2-(6-Ethylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 604972 5-[6-(1-Ethyl-propylamino)-purin-9-yl]-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid butyl-methyl-amide 604974 2-(6-Amino-2-chloro-purin-9-yl)-5-hydroxymethyl-3-methyl-tetrahydro-furan-3,4-diol 605045 5-[6-(1-Ethyl-propylamino)-purin-9-yl]-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid cyclopropylamide 605052 5-[6-(1-Ethyl-propylamino)-purin-9-yl]-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid isopropylamide 605170 2-Hydroxymethyl-5-(6-p-tolylamino-purin-9-yl)-tetrahydro-furan-3,4-diol 605243 6-Amino-9-(3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-1-methyl-1,9-dihydro-purin-2-one 605298 2-Hydroxymethyl-5-[6-(isopropyl-phenyl-amino)-purin-9-yl]-tetrahydro-furan-3,4-diol 605310 2-(3,4-Dihydroxy-5-{6-[N'-(4-sulfamoyl-phenyl)-hydrazino]-purin-9-yl}-tetrahydro-furan-2-yl)-N-ethyl-acetamide 605327 2-(6-Cyclodecylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 605364 2-(6-Cyclododecylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 605372 2-{3,4-Dihydroxy-5-[6-(3-iodo-benzylamino)-purin-9-yl]-tetrahydro-furan-2-yl}-N-methyl-acetamide 605384 2-(8-Butylamino-6-cyclopentylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 605385 (R)-2-[(R)-2-(6-{[5-(6-Amino-purin-9-yl)-3,4-dihydroxy-tetrahydro-furan-2-carbonyl]-amino}-hexanoylamino)-5-guanidino-pentanoylamino]-5-guanidino-pentanoic acid 605416 2-(8-Cyclopentylamino-6-propylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 605441 2-{5-[2-Chloro-6-(3-iodo-benzylamino)-purin-9-yl]-3,4-dihydroxy-tetrahydro-furan-2-yl}-N-methyl-acetamide 605491 2-(6-Amino-8-ethylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 605515 (2E)-3-{6-amino-9-[3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl]-9H-purin-2-yl}-N-(3-chlorophenyl)triaz-2-ene-1-carboxamide 605539 phenyl (2E)-3-{6-amino-9-[3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl]-9H-purin-2-yl}triaz-2-ene-1-carboxylate 605543 2-(6-Amino-8-propylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 605714 Sodium salt 4-[3-(2-{2-[4-(2-{4-[9-(3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-6-ylamino]-phenyl}-acetylamino)-phenyl]-acetylamino}-ethyl)-thioureido]-benzenesulfonate 605724 2-{4-[9-(3,4-Dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-6-ylamino]-phenyl}-N-{4-[(2-isothiocyanato-ethylcarbamoyl)-methyl]-phenyl}-acetamide 605726 2-{4-[9-(3,4-Dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-6-ylamino]-phenyl}-N-[4-({2-[3-(4-methoxy-phenyl)-thioureido]-ethylcarbamoyl}-methyl)-phenyl]-acetamide 605745 N-[4-({2-[3-(4-Cyano-phenyl)-thioureido]-ethylcarbamoyl}-methyl)-phenyl]-2-{4-[9-(3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-6-ylamino]-phenyl}-acetamide 605746 2-{4-[9-(3,4-Dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-6-ylamino]-phenyl}-N-(4-{[2-(3-pentafluorophenyl-thioureido)-ethylcarbamoyl]-methyl}-phenyl)-acetamide 605863 2-Hydroxymethyl-5-[7-(1-methyl-2-phenyl-ethylamino)-imidazo[4,5-b]pyridin-3-yl]-tetrahydro-furan-3,4-diol 605894 2-(6-Amino-purin-9-yl)-5-((S)-1-hydroxy-prop-2-ynyl)-tetrahydro-furan-3,4-diol 606143 2-(4-Cyclopentylamino-imidazo[4,5-c]pyridin-1-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 606297 5-(6-Amino-2-hept-1-ynyl-purin-9-yl)-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 606326 5-(6-Amino-2-oct-1-ynyl-purin-9-yl)-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 606419 2-(6-Amino-2-dodec-1-ynyl-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 606472 2-[6-(4-Amino-3-iodo-benzylamino)-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 606520 (N-Ac-ADAC) 2-(4-{Acetyl-[9-(3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-6-yl]-amino}-phenyl)-N-{4-[(2-amino-ethylcarbamoyl)-methyl]-phenyl}-acetamide 606538 5-[6-Amino-2-((Z)-hex-1-enyl)-purin-9-yl]-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 606602 2-Hydroxymethyl-5-[6-(3-hydroxy-propylamino)-purin-9-yl]-tetrahydro-furan-3,4-diol 606623 3,4-Dihydroxy-5-{6-[2-(7-nitro-benzo[1,2,5]oxadiazol-4-ylamino)-ethylamino]-purin-9-yl}-tetrahydro-furan-2-carboxylic acid ethylamide 606729 2-Hydroxymethyl-5-[6-((R)-1-hydroxymethyl-3-methyl-butylamino)-purin-9-yl]-tetrahydro-furan-3,4-diol 606761 3,4-Dihydroxy-5-{6-[3-(4-propoxy-phenyl)-ureido]-purin-9-yl}-tetrahydro-furan-2-carboxylic acid ethylamide 606774 2-Hydroxymethyl-5-[2-iodo-6-(piperidin-1-ylamino)-purin-9-yl]-tetrahydro-furan-3,4-diol 606775 2-[2-Chloro-6-((S)-1-hydroxymethyl-2-phenyl-ethylamino)-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 606780 5-{6-[8-(5-Dimethylamino-naphthalene-1-sulfonylamino)-octylamino]-purin-9-yl}-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 606781 3,4-Dihydroxy-5-{6-[6-(7-nitro-benzo[1,2,5]oxadiazol-4-ylamino)-hexylamino]-purin-9-yl}-tetrahydro-furan-2-carboxylic acid ethylamide 606782 3,4-Dihydroxy-5-{6-[4-(7-nitro-benzo[1,2,5]oxadiazol-4-ylamino)-butylamino]-purin-9-yl}-tetrahydro-furan-2-carboxylic acid ethylamide 606785 3,4-Dihydroxy-5-{6-[8-(7-nitro-benzo[1,2,5]oxadiazol-4-ylamino)-octylamino]-purin-9-yl}-tetrahydro-furan-2-carboxylic acid ethylamide 606786 3,4-Dihydroxy-5-{6-[10-(7-nitro-benzo[1,2,5]oxadiazol-4-ylamino)-decylamino]-purin-9-yl}-tetrahydro-furan-2-carboxylic acid ethylamide 606795 2-Hydroxymethyl-5-[6-((S)-1-hydroxymethyl-2-phenyl-ethylamino)-2-iodo-purin-9-yl]-tetrahydro-furan-3,4-diol 606800 2-[2-Chloro-6-((R)-1-hydroxymethyl-2-phenyl-ethylamino)-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 606804 2-Hydroxymethyl-5-[2-iodo-6-(morpholin-4-ylamino)-purin-9-yl]-tetrahydro-furan-3,4-diol 606810 5-{6-[12-(5-Dimethylamino-naphthalene-1-sulfonylamino)-dodecylamino]-purin-9-yl}-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 606832 5-{6-[3-(5-Dimethylamino-naphthalene-1-sulfonylamino)-propylamino]-purin-9-yl}-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 606836 5-{6-[4-(5-Dimethylamino-naphthalene-1-sulfonylamino)-butylamino]-purin-9-yl}-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 606846 5-{6-[10-(5-Dimethylamino-naphthalene-1-sulfonylamino)-decylamino]-purin-9-yl}-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 606879 5-{6-[6-(5-Dimethylamino-naphthalene-1-sulfonylamino)-hexylamino]-purin-9-yl}-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 606925 2-(2-Chloro-6-phenylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 606942 2-{6-Amino-2-[N'-(4-methyl-benzylidene)-hydrazino]-purin-9-yl}-5-hydroxymethyl-tetrahydro-furan-3,4-diol 606988 2-{6-[2-(4-Amino-3-iodo-phenyl)-ethylamino]-purin-9-yl}-5-hydroxymethyl-tetrahydro-furan-3,4-diol 607174 2-[6-(3-Fluoro-phenylamino)-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 607179 2-Hydroxymethyl-5-((7S,8S)-8-methyl-7-phenyl-7,8-dihydro-imidazo[2,1-i]purin-3-yl)-tetrahydro-furan-3,4-diol 607200 2-Hydroxymethyl-5-((7R,8R)-8-methyl-7-phenyl-7,8-dihydro-imidazo[2,1-i]purin-3-yl)-tetrahydro-furan-3,4-diol 607204 2-((R)-8-Benzyl-7,8-dihydro-imidazo[2,1-i]purin-3-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 607205 2-((S)-8-Benzyl-7,8-dihydro-imidazo[2,1-i]purin-3-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 607221 2-[6-(4-Fluoro-phenylamino)-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 607385 Sodium salt 2-[9-(3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-6-ylamino]-ethanesulfonate 607389 Octadecanoic acid (2-{2-[4-(2-{4-[9-(3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-6-ylamino]-phenyl}-acetylamino)-phenyl]-acetylamino}-ethyl)-amide 607529 2-(6-Cyclopentylamino-2-iodo-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 607537 2-(6-Cyclopentylamino-2-hydroxy-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 607538 2-(6-Cyclobutylamino-2-hydroxy-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 607562 2-[6-(Bicyclo[2.2.1]hept-2-ylamino)-2-hydroxy-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 607568 2-(6-Cycloheptylamino-2-hydroxy-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 607584 2-(6-Cyclohexylamino-2-hydroxy-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 607585 2-[6-(Decahydro-naphthalen-2-ylamino)-2-hydroxy-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 607638 (3R,4S,5R)-3,4-Dihydroxy-5-(6-{3-[4-(isopropyl-methyl-sulfamoyl)-phenyl]-ureido}-purin-9-yl)-tetrahydro-furan-2-carboxylic acid ethylamide 607646 3,4-Dihydroxy-5-(6-{3-[4-(pyrimidin-2-ylsulfamoyl)-phenyl]-ureido}-purin-9-yl)-tetrahydro-furan-2-carboxylic acid ethylamide 607647 5-[6-(2,4-Dichloro-benzoylamino)-purin-9-yl]-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 607711 2-Hydroxymethyl-5-((S)-8-phenyl-7,8-dihydro-imidazo[2,1-i]purin-3-yl)-tetrahydro-furan-3,4-diol 607712 2-Hydroxymethyl-5-((R)-8-phenyl-7,8-dihydro-imidazo[2,1-i]purin-3-yl)-tetrahydro-furan-3,4-diol 607751 (2S,5R)-2-(hydroxymethyl)-5-[(5E,8R)-5-imino-8-phenyl-5,7,8,9-tetrahydro-3H-imidazo[2,1-i]purin-3-yl]tetrahydrofuran-3,4-diol 607752 (2S,5R)-2-(hydroxymethyl)-5-[(5E,8S)-5-imino-8-phenyl-5,7,8,9-tetrahydro-3H-imidazo[2,1-i]purin-3-yl]tetrahydrofuran-3,4-diol 607852 2-[6-(3-aminoanilino)-9H-9-purinyl]-5-hydroxymethyltetrahydro-3,4-furandiol 607909 2-[6-(3-Ethyl-phenylamino)-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 607952 2-Hydroxymethyl-5-[6-(3-iodo-phenylamino)-purin-9-yl]-tetrahydro-furan-3,4-diol 608009 2-[6-(4-Ethyl-phenylamino)-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 608011 2-Hydroxymethyl-5-[6-(4-iodo-phenylamino)-purin-9-yl]-tetrahydro-furan-3,4-diol 608012 2-[6-(3-Amino-phenylamino)-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 608120 (3R,4S,5R)-3,4-Dihydroxy-5-(6-{3-[4-(piperidine-1-sulfonyl)-phenyl]-ureido}-purin-9-yl)-tetrahydro-furan-2-carboxylic acid ethylamide 608164 (3R,4S,5R)-5-(6-{3-[4-(Adamantan-1-ylsulfamoyl)-phenyl]-ureido}-purin-9-yl)-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 608165 (3R,4S,5R)-5-[6-(3-{4-[Bis-(2-chloro-ethyl)-sulfamoyl]-phenyl}-ureido)-purin-9-yl]-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 608171 (3R,4S,5R)-3,4-Dihydroxy-5-(6-{3-[4-(morpholine-4-sulfonyl)-phenyl]-ureido}-purin-9-yl)-tetrahydro-furan-2-carboxylic acid ethylamide 608172 (3R,4S,5R)-3,4-Dihydroxy-5-(6-{3-[4-(4-methoxy-phenylsulfamoyl)-phenyl]-ureido}-purin-9-yl)-tetrahydro-furan-2-carboxylic acid ethylamide 608179 (3R,4S,5R)-5-{6-[3-(4-Cyclopentylsulfamoyl-phenyl)-ureido]-purin-9-yl}-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 608180 (3R,4S,5R)-3,4-Dihydroxy-5-{6-[3-(4-pentylsulfamoyl-phenyl)-ureido]-purin-9-yl}-tetrahydro-furan-2-carboxylic acid ethylamide 608186 (3R,4S,5R)-5-{6-[3-(4-Ethylsulfamoyl-phenyl)-ureido]-purin-9-yl}-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 608187 (3R,4S,5R)-5-{6-[3-(4-Diethylsulfamoyl-phenyl)-ureido]-purin-9-yl}-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 608188 (3R,4S,5R)-5-{6-[3-(4-Benzylsulfamoyl-phenyl)-ureido]-purin-9-yl}-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 608191 (3R,4S,5R)-5-(6-{3-[4-(Allyl-methyl-sulfamoyl)-phenyl]-ureido}-purin-9-yl)-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 608195 3,4-Dihydroxy-5-(6-{3-[4-(pyridin-2-ylsulfamoyl)-phenyl]-ureido}-purin-9-yl)-tetrahydro-furan-2-carboxylic acid ethylamide 608200 (3R,4S,5R)-5-{6-[3-(4-Cyclohexylsulfamoyl-phenyl)-ureido]-purin-9-yl}-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 608213 (3R,4S,5R)-3,4-Dihydroxy-5-{6-[3-(4-propylsulfamoyl-phenyl)-ureido]-purin-9-yl}-tetrahydro-furan-2-carboxylic acid ethylamide 608215 (3R,4S,5R)-5-{6-[3-(4-tert-Butylsulfamoyl-phenyl)-ureido]-purin-9-yl}-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 608222 (3R,4S,5R)-5-{6-[3-(4-Dimethylsulfamoyl-phenyl)-ureido]-purin-9-yl}-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 608223 (3R,4S,5R)-5-(6-{3-[4-(2,5-Dihydro-pyrrole-1-sulfonyl)-phenyl]-ureido}-purin-9-yl)-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 608227 (3R,4S,5R)-5-{6-[3-(4-Diallylsulfamoyl-phenyl)-ureido]-purin-9-yl}-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 608234 (3R,4S,5R)-3,4-Dihydroxy-5-(6-{3-[4-(pyrrolidine-1-sulfonyl)-phenyl]-ureido}-purin-9-yl)-tetrahydro-furan-2-carboxylic acid ethylamide 608236 (3R,4S,5R)-5-{6-[3-(4-Dipropylsulfamoyl-phenyl)-ureido]-purin-9-yl}-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 608244 3,4-Dihydroxy-5-[6-[3-(4-methoxy-phenyl)-ureido]-2-(4-phenyl-but-1-ynyl)-purin-9-yl]-tetrahydro-furan-2-carboxylic acid ethylamide 608256 5-(6-Cyclopentylamino-purin-9-yl)-2-hydroxymethyl-3-methyl-tetrahydro-furan-3,4-diol 608270 1N-{2-[3',6'-dihydroxy-3-oxospiro[2,3-dihydro-1H-indene-1,9'-(9'H-xanthene)]-5-ylamino(thioxo)methylamino]ethyl}-2-(4-{4-[9-(3,4-dihydroxy-5-hydroxymethyltetrahydro-2-furanyl)-9H-6-purinylamino]benzylcarboxamido}phenyl)acetamide 608285 AdoC(Ahx)Arg6 608286 AdoC(beta-Ala)2AlaArg6 608287 AdoC(Aoc)Arg6 608288 (R)-2-((R)-2-{2-[(R)-2-(6-{[(R)-5-(6-Amino-purin-9-yl)-3,4-dihydroxy-tetrahydro-furan-2-carbonyl]-amino}-hexanoylamino)-5-guanidino-pentanoylamino]-5-guanidino-pentanoylamino}-5-guanidino-pentanoylamino)-5-guanidino-pentanoic acid 608290 AdoC(Dpr)2AlaArg6 608291 AdoC(Aun)Arg6 608292 AdoC(beta-Ala)Arg6 608293 AdoCGlyArg6 608295 AdoC(GABA)Arg6 608576 (S)2-Methanesulfinyl-10-[2-((S)-1-methyl-piperidin-2-yl)-ethyl]-10H-phenothiazine 608581 SID4253976 608677 isoelaeocarpicine 608678 isoelaeocarpine 608679 elaeocarpine 608680 habbemines B 608681 (R)-(1,2,3,5,6,8a-hexahydroindolizin-8-yl)(2-hydroxy-6-methylphenyl)methanone 608682 habbemines A 608868 (6,7-Dihydroxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-dimethyl-ammonium 608904 4-cyclopropylmethyl-10,17-dihydroxy-15-[1-(1-naphthyl)-(Z)-methylidene]-12-oxa-4-azoniapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10-trien-14-one 608905 4-cyclopropylmethyl-10,17-dihydroxy-15-[1-(4-phenylphenyl)-(Z)-methylidene]-12-oxa-4-azoniapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10-trien-14-one 608911 4-cyclopropylmethyl-10,17-dihydroxy-15-[1-(2-naphthyl)-(Z)-methylidene]-12-oxa-4-azoniapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10-trien-14-one 608912 4-cyclopropylmethyl-10,17-dihydroxy-15-[1-(1-naphthyl)-(E)-methylidene]-12-oxa-4-azoniapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10-trien-14-one 608913 15-[1-(9-anthryl)-(Z)-methylidene]-4-cyclopropylmethyl-10,17-dihydroxy-12-oxa-4-azoniapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10-trien-14-one 608914 4-cyclopropylmethyl-10,17-dihydroxy-15-[1-(2-naphthyl)-(E)-methylidene]-12-oxa-4-azoniapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10-trien-14-one 608915 15-[1-(9-anthryl)-(E)-methylidene]-4-cyclopropylmethyl-10,17-dihydroxy-12-oxa-4-azoniapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10-trien-14-one 608916 4-cyclopropylmethyl-10,17-dihydroxy-15-[1-(4-phenylphenyl)-(E)-methylidene]-12-oxa-4-azoniapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10-trien-14-one 609001 2-Chloro-N-(3-(R)-1-pyrrolidin-2-ylmethyl-1H-indol-5-yl)-benzenesulfonamide 609016 5'-(Chlorophenyl)-17-(cyclopropylmethyl)-6,7-didehydro-3,14-dihydroxy-4,5alpha-epoxypyrido-[2',3':6,7]morphinan 609017 6-(4-chlorophenyl)-19-cyclopropylmethyl-(2R,10R)-11-oxa-8,19-diazahexacyclo[10.9.1.01,10.02,18.04,9.016,22]docosa-4(9),5,7,12,14,16(22)-hexaen-13-ol 609054 17-cyclopropylmethyl-6-7-didehydro-3,14-dihydroxy-4,5alpha-epoxy-1'-methyl-4',5',6',7'-tetrahydroindolo[2',3';6,7]morphinan 609101 Naltrindole analogue 609140 Naltrindole analogue 609148 Naltrindole analogue 609149 Naltrindole analogue 609150 Naltrindole analogue 609151 Naltrindole analogue 609152 Naltrindole analogue 609153 Naltrindole analogue 609154 Naltrindole analogue 609155 Naltrindole analogue 609156 Naltrindole analogue 609157 Naltrindole analogue 609158 Naltrindole analogue 609159 Naltrindole analogue 609160 Naltrindole analogue 609161 Naltrindole analogue 609162 Naltrindole analogue 609163 Naltrindole analogue 609164 Naltrindole analogue 609165 Naltrindole analogue 609166 Naltrindole analogue 609170 N-cyclopropylmethyl-14beta-(2'-methylcinnamoylamino)-7,8-dihydronorcodeinone 609172 N-cyclopropylmethyl-14beta-(2'-chlorocinnamoylamino)-7,8-dihydronormorphinone 609173 N-cyclopropylmethyl-14beta-(2'-methylcinnamoylamino)-7,8-dihydronormorphinone 609178 N-cyclopropylmethyl-14beta-(2'-chlorocinnamoylamino)-7,8-dihydronorcodeinone 609201 3-butoxy-17-(cyclopropylmethyl)-10-methoxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-trien-13-one 609251 4-[(S)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-yl)-(3-methoxy-phenyl)-methyl]-N,N-diethyl-benzamide 609283 6-(4-bromophenyl)-19-methyl-(2R,10R)-11-oxa-8,19-diazahexacyclo[10.9.1.01,10.02,18.04,9.016,22]docosa-4(9),5,7,12,14,16(22)-hexaen-13-ol 609284 19-methyl-6-phenyl-(2R,10R)-11-oxa-8,19-diazahexacyclo[10.9.1.01,10.02,18.04,9.016,22]docosa-4(9),5,7,12,14,16(22)-hexaen-13-ol 609286 19-methyl-6-phenyl-(2S,10R)-11-oxa-8,19-diazahexacyclo[10.9.1.01,10.02,18.04,9.016,22]docosa-4(9),5,7,12,14,16(22)-hexaene-2,13-diol 609287 19-methyl-(2S,10R)-11-oxa-8,19-diazahexacyclo[10.9.1.01,10.02,18.04,9.016,22]docosa-4(9),5,7,12,14,16(22)-hexaene-2,13-diol 609289 6-(3,4-dichlorophenyl)-19-methyl-(2R,10R)-11-oxa-8,19-diazahexacyclo[10.9.1.01,10.02,18.04,9.016,22]docosa-4(9),5,7,12,14,16(22)-hexaen-13-ol 609291 6-(2,4-dichlorophenyl)-19-methyl-(2R,10R)-11-oxa-8,19-diazahexacyclo[10.9.1.01,10.02,18.04,9.016,22]docosa-4(9),5,7,12,14,16(22)-hexaen-13-ol 609293 19-methyl-(2R,10R)-11-oxa-8,19-diazahexacyclo[10.9.1.01,10.02,18.04,9.016,22]docosa-4(9),5,7,12,14,16(22)-hexaen-13-ol 609294 6-(4-chlorophenyl)-19-methyl-(2R,10R)-11-oxa-8,19-diazahexacyclo[10.9.1.01,10.02,18.04,9.016,22]docosa-4(9),5,7,12,14,16(22)-hexaen-13-ol 609301 17-propyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy-6,7:2',3'-indolomorphinan 609302 17-(3-methyl-2-butenyl)-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy-6,7:2',3'-indolomorphinan 609303 17-(2-methyl-2-propenyl)-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy-6,7:2',3'-indolomorphinan 609304 17-(1-methylethyl)-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy-6,7:2',3'-indolomorphinan 609305 17-hexyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy-6,7:2',3'-indolomorphinan 609306 17-butyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy-6,7:2',3'-indolomorphinan 609307 17-pentyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy-6,7:2',3'-indolomorphinan 609308 (E)-17-(2-butenyl)-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy-6,7:2',3'-indolomorphinan 609309 17-(3-methylbutyl)-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy-6,7:2',3'-indolomorphinan 609310 17-ethyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy-6,7:2',3'-indolomorphinan 609311 17-heptyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy-6,7:2',3'-indolomorphinan 609312 17-(2-methylpropyl)-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy-6,7:2',3'-indolomorphinan 609317 Naltrindole analogue 609323 3-hydroxy-4,10-dimethoxy-17-methyl-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-13-one 609329 10-hydroxy-3,4-dimethoxy-17-methyl-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-13-one 609376 6,11-Dimethyl-3-(3-phenyl-propyl)-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocin-8-ol 609384 4-(6-Amino-2-thiazol-2-ylethynyl-purin-9-yl)-2,3-dimethoxy-cyclopentanecarboxylic acid ethylamide 609385 4-[6-Amino-2-(4-formyl-phenylethynyl)-purin-9-yl]-2,3-dimethoxy-cyclopentanecarboxylic acid ethylamide 609429 22-Benzyl-19-(3-guanidino-propyl)-16-(1H-indol-3-ylmethyl)-4,7,15,18,21,24-hexaoxo-docosahydro-3a,8,14,17,20,23-hexaaza-cyclopentacyclotricosene-13-carboxylic acid amide 609762 2-({2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl}-amino)-3-(1H-benzoimidazol-2-yl)-propionic acid 609763 2-[2-Amino-3-((S)-4-hydroxy-2,6-dimethyl-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (1-carbamoyl-ethyl)-amide 609764 2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid [2-(1H-benzoimidazol-2-yl)-ethyl]-amide 609765 2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid [1-(1H-benzoimidazol-2-yl)-ethyl]-amide 609766 2-[({2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl}-amino)-methyl]-benzoimidazole-1-carboxylic acid 609767 (S)-2-({2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl}-amino)-succinamic acid 609768 2-[2-Amino-3-((R)-4-hydroxy-2,6-dimethyl-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (1-carbamoyl-ethyl)-amide 609769 (S)-3-({2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl}-amino)-succinamic acid 609770 2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid [1-(1H-benzoimidazol-2-yl)-ethyl]-amide 609781 2-Amino-1-[3-(1H-benzoimidazol-2-yl)-3,4-dihydro-1H-isoquinolin-2-yl]-3-(4-hydroxy-2,6-dimethyl-phenyl)-propan-1-one 609809 Norbinaltorphimine derivative 609810 17,17'-Dimethyl-3,3'-dimethoxy-6,6',7,7'-tetradehydro-4,5:4',5'-diepoxy-6,6'-(imino)[7,7'-bimorphinan] 609814 17,17'-Dimethyl-6,6',7,7'-tetradehydro-4,5:4',5'-diepoxy-6,6'-(imino)[7,7'-bimorphinan]-3,3'-diol 609823 Naltrindole analogue 609824 Naltrindole analogue 609826 (R)-3-{Methyl-[5-(4-trifluoromethyl-phenyl)-thiophene-2-carbonyl]-amino}-pyrrolidine-1-carboxylic acid (R)-[1-(4,4-dimethyl-cyclohexyl)-pyrrolidin-3-yl]-methyl-amide 609827 (S)-N-((R)-1-(4,4-dimethylcyclohexyl)pyrrolidin-3-yl)-N-methyl-3-(N-methyl-5-(4-(trifluoromethyl)phenyl)thiophene-2-carboxamido)pyrrolidine-1-carboxamide 609844 3-hydroxy-4,10-dimethoxy-17-methyl-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5,13-tetraen-13-yl cyanide 609845 3,10-dihydroxy-4-methoxy-17-methyl-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-13-one 609846 3,10-dihydroxy-4-methoxy-17-methyl-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5,13-tetraen-13-yl cyanide 609847 10-hydroxy-3,4-dimethoxy-17-methyl-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5,13-tetraen-13-yl cyanide 609848 17-benzyloxy-10-hydroxy-4-methyl-(13R,17S)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10-trien-14-one 609849 17-allyloxy-10-hydroxy-4-methyl-(13R,17S)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10-trien-14-one 609850 10-hydroxy-17-methoxy-4-methyl-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-14-one 609851 17-ethoxy-10-hydroxy-13-methyl-4-phenethyl-(13R,17S)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10-trien-14-one 609852 10-hydroxy-4-methyl-17-(1-naphthylmethoxy)-(13R,17S)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10-trien-14-one 609853 17-benzyloxy-10-hydroxy-4,13-dimethyl-(13R,17S)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10-trien-14-one 609854 17-(2,6-dichlorobenzyloxy)-10-hydroxy-4-methyl-(13R,17S)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10-trien-14-one 609855 Naltrindole analogue 609856 Naltrindole analogue 609857 Naltrindole analogue 609858 Naltrindole analogue 609859 Naltrindole analogue 609860 Naltrindole analogue 609861 Naltrindole analogue 609862 Naltrindole analogue 609863 Naltrindole analogue 609864 Naltrindole analogue 609865 Naltrindole analogue 609866 Naltrindole analogue 609867 Naltrindole analogue 609868 Naltrindole analogue 609869 Naltrindole analogue 609870 Naltrindole analogue 609871 Naltrindole analogue 609872 Naltrindole analogue 609873 Naltrindole analogue 609877 (R)-1-Phenyl-3,4-dihydro-1H-isoquinoline-2-carboxylic acid (S)-(1-aza-bicyclo[2.2.2]oct-3-yl) ester 609878 (S)-1-Phenyl-3,4-dihydro-1H-isoquinoline-2-carboxylic acid (S)-(1-aza-bicyclo[2.2.2]oct-3-yl) ester 609879 (S)-1-Thiophen-3-yl-3,4-dihydro-1H-isoquinoline-2-carboxylic acid (R)-(1-aza-bicyclo[2.2.2]oct-3-yl) ester 609880 (R)-1-Thiophen-3-yl-3,4-dihydro-1H-isoquinoline-2-carboxylic acid (R)-(1-aza-bicyclo[2.2.2]oct-3-yl) ester 609881 (2R,4R)-4-Hydroxy-1-phenyl-3,4-dihydro-1H-isoquinoline-2-carboxylic acid (R)-(1-aza-bicyclo[2.2.2]oct-3-yl) ester 609882 (2S,4S)-4-Hydroxy-1-phenyl-3,4-dihydro-1H-isoquinoline-2-carboxylic acid (S)-(1-aza-bicyclo[2.2.2]oct-3-yl) ester 609883 7-(4-fluorophenylamino)-1-((1S,3R)-3-hydroxycyclopentyl)-3-(4-methoxyphenyl)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one 609885 14beta-(2'-chlorocinnamoylamino)-7,8-dihydrocodeinone 609886 14beta-(2'-methylcinnamoylamino)-7,8-dihydrocodeinone 609887 17-methyl-4'-methyldihydromorphinone 609889 (2E)-N-[(1R,13R,17S)-10-hydroxy-4-methyl-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl]-3-(4-nitrophenyl)prop-2-enamide 609890 14beta-(4'-chlorocinnamoylamino)-7,8-dihydrocodeinone 609893 14beta-(2'-methylcinnamoylamino)-7,8-dihydromorphinone 609894 N-[(1R,13R,17S)-10-hydroxy-4-methyl-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl]-3-(4-methylphenyl)propanamide 609895 14beta-(4'-methylcinnamoylamino)-7,8-dihydrocodeinone 609985 4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-2,2,6,6-tetramethyl-1-oxo-piperidinium 609986 4-{2-[4-(5,7-Dioxo-6-propyl-4,5,6,7-tetrahydro-1H-imidazo[4,5-b]pyridin-2-yl)-phenoxy]-acetylamino}-2,2,6,6-tetramethyl-1-oxo-piperidinium 610017 3-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-2,2,5,5-tetramethyl-1-oxo-2,5-dihydro-1H-pyrrolium 610018 3-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tetrahydro-purin-3-ylmethyl)-2,2,5,5-tetramethyl-1-oxo-2,5-dihydro-1H-pyrrolium 610059 2-Chloro-N-[3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide 610060 3-Chloro-N-[3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide 612948 (S)-3-(4-chlorophenyl)-N-methyl-4-phenyl-N'-(piperidin-1-ylsulfonyl)-4,5-dihydro-1H-pyrazole-1-carboximidamide 623657 (2R,3S,4R,5R)-2-(hydroxymethyl)-5-(6-(4-methoxyphenylamino)-9H-purin-9-yl)tetrahydrofuran-3,4-diol 641792 4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1-(4-fluoro-phenyl)-butan-1-one;propionate HCl 641852 Phosphoric acid mono-[4-(3-carbamoyl-4-cyclohexylmethoxy-benzylcarbamoyl)-phenyl] ester 641856 Phosphoric acid mono-[4-(3-acetyl-4-cyclohexylmethoxy-benzylcarbamoyl)-phenyl] ester 641857 Phosphoric acid mono-[4-(4-cyclohexylmethoxy-3-methylcarbamoyl-benzylcarbamoyl)-phenyl] ester 642291 Phosphoric acid mono-{4-[1-(4-tert-butyl-benzyl)-2-oxo-azepan-3-ylcarbamoyl]-phenyl} ester 642293 Phosphoric acid mono-{4-[5-oxo-4-(3-phenyl-propyl)-[1,4]thiazepan-6-ylcarbamoyl]-phenyl} ester 642295 (Difluoro-p-tolyl-methyl)-phosphate 642299 [(4-{2-Acetylamino-2-[1-(3-cyclohexyl-propyl)-2-oxo-azepan-3-ylcarbamoyl]-ethyl}-phenyl)-difluoro-methyl]-phosphonic acid 642497 hydrogen (3-{[(4-nonylphenyl)methyl]amino}propyl)phosphonite 642597 3-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-benzylamine; succinate 642658 1-{3-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-benzyl}-pyrrolidine-2,5-dione with succinic acid 642665 N-{3-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-benzyl}-benzamide with succinic acid 642681 N-(1-Carbamoyl-2-phenyl-ethyl)-3-({2-[3-(1H-indol-3-yl)-2-(2-{2-[2-(4-sulfooxy-phenyl)-acetylamino]-hexanoylamino}-acetylamino)-propionylamino]-hexanoyl}-methyl-amino)-succinamic acid ammonium base (AR-R 15849) 642852 5-(2-Acetylamino-hexanoylamino)-19-[3-(diaminomethaniminium)-propyl]-24-hydroxy-16-(1H-indol-3-ylmethyl)-22-naphthalen-2-ylmethyl-4,7,15,18,21-pentaoxo-tetracosahydro-3a,8,14,17,20,23-hexaaza-cyclopentacyclotricosene-13-carboxylic acid amide 642855 8-(2-Acetylamino-hexanoylamino)-22-[3-(diaminomethaniminium)-propyl]-19-(1H-indol-3-ylmethyl)-25-naphthalen-2-ylmethyl-7,10,18,21,24,27-hexaoxo-6,11,17,20,23,26-hexaaza-spiro[4.22]heptacosane-16-carboxylic acid 642857 9-(2-Acetylamino-hexanoylamino)-23-[3-(diaminomethaniminium)-propyl]-20-(1H-indol-3-ylmethyl)-26-naphthalen-2-ylmethyl-8,11,19,22,25,28-hexaoxo-7,12,18,21,24,27-hexaaza-spiro[5.22]octacosane-17-carboxylic acid amide 642859 6-(2-Acetylamino-hexanoylamino)-20-[3-(diaminomethaniminium)-propyl]-17-(1H-indol-3-ylmethyl)-23-naphthalen-2-ylmethyl-5,8,16,19,22,25-hexaoxo-4,9,15,18,21,24-hexaaza-spiro[2.22]pentacosane-14-carboxylic acid amide 642860 1N-[12-carbamoyl-18-(3-diaminomethaniminiumpropyl)-15-(1H-3-indolylmethyl)-21-(2-naphthylmethyl)-3,6,14,17,20,23-hexaoxo-(4R,12S,15S,18R,21S)-spiro[2,7,13,16,19,22-hexaazacyclotricosane-1,2'-(2',3'-dihydro-1'H-indene)]-4-yl]-2-methyl 642861 5-(2-Acetylamino-hexanoylamino)-19-[3-(diaminomethaniminium)-propyl]-16-(1H-indol-3-ylmethyl)-22-naphthalen-2-ylmethyl-4,7,15,18,21,24-hexaoxo-tetracosahydro-3a,8,14,17,20,23-hexaaza-cyclopentacyclotricosene-13-carboxylic acid amide 642862 21-(2-Acetylamino-hexanoylamino)-7-[3-(diaminomethaniminium)-propyl]-10-(1H-indol-3-ylmethyl)-24,29-dimethyl-4-naphthalen-2-ylmethyl-2,5,8,11,19,22-hexaoxo-3,6,9,12,18,23-hexaaza-tricyclo[21.7.0.0*24,29*]triacontane-13-carboxylic acid amide 642951 (E)-(1S,2S,6R,7S)-7-((S)-1-Carbamoyl-2-phenyl-ethylcarbamoyl)-2,6-dihydroxy-1-(4-hydroxy-2,6-dimethyl-benzyl)-8-phenyl-oct-4-enyl-ammonium 642952 (E)-(1S,2R,6S,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-dimethyl-benzyl)-7-phenethylcarbamoyl-8-phenyl-oct-4-enyl-ammonium 642953 (E)-(1S,2S,6S,7R)-7-((S)-1-Carbamoyl-2-phenyl-ethylcarbamoyl)-2,6-dihydroxy-1-(4-hydroxy-2,6-dimethyl-benzyl)-8-phenyl-oct-4-enyl-ammonium 642954 (E)-(1S,2R,6S,7R)-7-((S)-1-Carbamoyl-2-phenyl-ethylcarbamoyl)-2,6-dihydroxy-1-(4-hydroxy-2,6-dimethyl-benzyl)-8-phenyl-oct-4-enyl-ammonium 642955 (E)-(1S,2S,6R,7R)-7-((S)-1-Carbamoyl-2-phenyl-ethylcarbamoyl)-2,6-dihydroxy-1-(4-hydroxy-2,6-dimethyl-benzyl)-8-phenyl-oct-4-enyl-ammonium 642956 (E)-(1S,2R,6R,7R)-7-((S)-1-Carbamoyl-2-phenyl-ethylcarbamoyl)-2,6-dihydroxy-1-(4-hydroxy-2,6-dimethyl-benzyl)-8-phenyl-oct-4-enyl-ammonium 642958 2-{(R)-2-[1-((S)-(S)-1-Carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-ethylcarbamoyl]-pyrrolidin-1-yl}-2-oxo-1-((S)-phenylmethyl)-ethyl-ammonium 642961 (E)-(1S,2R,6R,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-dimethyl-benzyl)-7-phenethylcarbamoyl-8-phenyl-oct-4-enyl-ammonium 642962 (E)-(1S,2S,6S,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-dimethyl-benzyl)-7-((S)-1-hydroxymethyl-2-phenyl-ethoxycarbonyl)-8-phenyl-oct-4-enyl-ammonium 642963 (E)-(1S,2S,6S,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-dimethyl-benzyl)-7-phenethyloxycarbonyl-8-phenyl-oct-4-enyl-ammonium 642964 (E)-(1S,2S,6S,7R)-7-((S)-1-Carbamoyl-2-phenyl-ethoxycarbonyl)-2,6-dihydroxy-1-(4-hydroxy-2,6-dimethyl-benzyl)-8-phenyl-oct-4-enyl-ammonium 642966 (E)-(1S,2S,6S,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-dimethyl-benzyl)-7-((S)-1-hydroxymethyl-2-phenyl-ethylcarbamoyl)-8-phenyl-oct-4-enyl-ammonium 642967 (E)-(1S,2S,6R,7S)-2,6-Dihydroxy-1-(4-hydroxy-2,6-dimethyl-benzyl)-7-phenethylcarbamoyl-8-phenyl-oct-4-enyl-ammonium 642968 (E)-(1S,2S,6R,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-dimethyl-benzyl)-7-phenethylcarbamoyl-8-phenyl-oct-4-enyl-ammonium 642969 (E)-(1S,2S,6S,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-dimethyl-benzyl)-7-phenethylcarbamoyl-8-phenyl-oct-4-enyl-ammonium 643230 3-(N-alkylamino) propylphosphonic acid derivative 643252 (2E)-2-[(2E)-3-[3,3-dimethyl-1-(5-{[2-(2-{2-[4-(2-oxo-2-{10-oxo-2,4,9-triazatricyclo[9.4.0.0^{3,8}]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}ethyl)piperazin-1-yl]ethoxy}ethoxy)ethyl]carbamoyl}pentyl)-5-sulfonato-2,3-dihydro-1H-indol-2-yl]prop-2-en-1-ylidene]-1-ethyl-3,3-dimethyl-2,3-dihydro-1H-indole-5-sulfonate 643319 Vasopressin Analogue 643321 Vasopressin Analogue 643322 Vasopressin Analogue 643330 (2S,4R)-4-Benzyl-1-[(S)-5-guanidino-2-(3-phenyl-propionylamino)-pentanoyl]-pyrrolidine-2-carboxylic acidbenzylamide acetylamino ion 643331 (2S,4R)-4-Benzyl-1-[(S)-5-guanidino-2-(3-1H-imidazol-4-yl-propionylamino)-pentanoyl]-pyrrolidine-2-carboxylic acid benzylamide acetylamino ion 643333 (2S,4R)-1-{(S)-2-[3-(2-Aminomethyl-phenyl)-propionylamino]-5-guanidino-pentanoyl}-4-benzyl-pyrrolidine-2-carboxylic acid benzylamide 643335 3-Chloro-4-[4-(5-pyrimidin-2-yl-3,6-dihydro-2H-pyridin-1-yl)-butyl]-4H-benzo[f][1,4]oxazepin-5-one fumarate 643336 4-(3-cyanophenyl)-5-(1H-1,2,4-triazol-1-yl)-1,3-thiazol-2-ylcarbamate 643337 3-Chloro-4-{4-[5-(4-methyl-pyrimidin-2-yl)-3,4-dihydro-2H-pyridin-1-yl]-butyl}-4H-benzo[f][1,4]oxazepin-5-one fumarate 643338 3-Chloro-4-[4-(3-pyrimidin-2-yl-piperidin-1-yl)-butyl]-4H-benzo[f][1,4]oxazepin-5-one fumarate 643489 (4-(2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetylamino)-indazol-1-yl)-acetic acid trifluoroacetate salt 643517 [Lys8(Alexa 488)]PVA 643518 [Lys8(Alexa 546)]PVA 643530 (S)-6-amino-5-((S)-2-((S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)pyrrolidine-2-carboxamido)-3-phenylpropanamido)-6-oxohexan-1-aminium 644124 2-(N',N''-Dicyclohexyl-guanidino)-3-phenyl-N-[4-(tributyl-lambda*5*-phosphanylmethyl)-phenyl]-propionamide; Chloride hydrochloride 644125 (S)-2-(N',N''-Dicyclohexyl-guanidino)-3-naphthalen-2-yl-N-[4-(tributyl-lambda*5*-phosphanylmethyl)-phenyl]-propionamide; dichloride 644128 2-(N',N''-Dicyclohexyl-guanidino)-3-naphthalen-1-yl-N-[4-(tributyl-lambda*5*-phosphanylmethyl)-phenyl]-propionamide; Chloride hydrochloride 644129 tributyl{4-[({[(E)-(cyclohexylamino)(cyclohexyliminio)1-(phenylmethyl)methyl]amino}acetyl)amino]benzyl}phosphonium; Chloride hydrochloride 644338 Quinapril analogue 644464 (+/-)-3-(cyclopropylmethyl)-1,2,3,4,5,6-hexahydro-cis-6,11-dimethyl-N-([1,1'-biphenyl]-4-ylmethyl)-2,6-methano-3-benzazocine-8-carboxamide 644466 (R)-3-(3,4-dioxo-2-(1-phenylethylamino)cyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide 644472 tert-butyl 2-({[(tert-butyl)oxycarbonyl]methyl}{2-[2-(2-{4-[2-(4-{2-[4-({[2-(hydroxymethyl)-4-(methylethylidene)-5-oxo(2-2,3-dihydrofuryl)]methyl}oxycarbonyl)phenyl]ethynyl}phenyl)ethynyl]phenoxy}ethoxy)ethoxy]ethyl}amino)acetate 644473 (2R,3S,4R)-5-((R)-6-amino-2-phenylethynyl-9H-purin-3-yl)-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid methylamide 644486 2-{4-[(4-{N-[3-(3-{3-[N-(3-{[(1-{2-[(4-amino-5-chloro-2-methoxyphenyl)carbonyloxy]ethyl}piperidin-4-yl)methyl]carbamoyl}propyl)-2,2-dimethylpropanamido]propyl}phenyl)propyl]-2,2-dimethylpropanamido}butanamido)methyl]piperidin-1-yl}ethyl 4-amino-5-chloro-2-methoxybenzoate 644489 4-((2-((4-chlorophenyl)-amino)-1,3-benzoxazol-5-yl)oxy)-N-methyl-2-pyridinecarboxamide 651776 4-Amino-5-chloro-N-[9-(4-fluoro-benzyl)-9-aza-bicyclo[3.3.1]non-3-yl]-2-methoxy-benzamide 651785 7-Methyl-8-oxo-5-p-tolyl-7,8-dihydro-[1,7]naphthyridine-6-carboxylic acid (R)-methyl-((S)-1-phenyl-ethyl)-amide 651794 (R)-1-Phenyl-3,4-dihydro-1H-isoquinoline-2-carboxylic acid (R)-(1-aza-bicyclo[2.2.2]oct-3-yl) ester 663451 9-methyl-8,9,10,11-tetrahydro-7H-16,18-(epiminomethano)-4,6-methanodibenzo[i,m][1,8,4,7,12]oxathiatriazacyclotetradecine-19,21-dione 675150 Leuprorelin 675154 SID29215426 675945 1,1,bis[[(5,11-di-hydro-6-oxo-6H-pyrido[2,3-b][1,4]benzodiazepin-11-yl)-carbonyl]methyl]-8,17-dimethyl-1,24-bis(2-methoybenzyl)-8,17-dimethyl-1,8,17,24-tetraazatetracosane tetraoxalate 675946 1,1-bis[[(5,11-di-hydro-6-oxo-6H-pyrido[2,3-b][1,4]benzodiazepin-11-yl)-carbonyl]methyl]-8,17-dimethyl-1,8,17,24-tetraazatetracosane tetraoxalate 675947 1,24-bis[[(5,11-di-hydro-6-oxo-6H-pyrido[2,3-b][1,4]benzodiazepin-11-yl)-carbonyl]methyl]-8,17-dimethyl-1-(2-methoybenzyl)-1,8,17,24-tetraazatetracosane tetraoxalate 675948 1,1,bis[[(5,11-di-hydro-6-oxo-6H-pyrido[2,3-b][1,4]benzodiazepin-11-yl)-carbonyl]methyl]-8,17-dimethyl-24-(2-methoybenzyl)-1,8,17,24-tetraazatetracosane tetraoxalate 675949 1,1,24,24-tetrakis[[(5,11-di-hydro-6-oxo-6H-pyrido[2,3-b][1,4]benzodiazepin-11-yl)-carbonyl]methyl]-8,17-dimethyl-1,8,17,24-tetraazatetracosane tetraoxalate 675951 N1,N1,N22,Tris[[(6,11-dihydro-5-oxo-5H-pyrido[2,3-b]-[1,4]benzodiazepin-11-yl)carbonyl]methyl]-7,16-dimethyl-7,16-diaza-1,22-docosanediamine Tetraoxalate 675952 N1,N22,Bis[[(6,11-dihydro-5-oxo-5H-pyrido[2,3-b]-[1,4]benzodiazepin-11-yl)carbonyl]methyl]-7,16-dimethyl-7,16-diaza-1,22-docosanediamine Tetraoxalate 675953 N1,N1,N22,N22-Tetrakis[[(6,11-dihydro-5-oxo-5H-pyrido[2,3-b]-[1,4]benzodiazepin-11-yl)carbonyl]methyl]-7,16-dimethyl-7,16-diaza-1,22-docosanediamine Tetraoxalate 675954 N1,N1,N22-Tris[[(5,10-dihydro-11-oxo-11H-dibenzo[b,e]-[1,4]diazepin-5-yl)carbonyl]methyl]-7,16-dimethyl-7,16-diaza-1,22-docosanediamine Tetraoxalate (C-tripinamide) 675955 N1,N22-Bis[[(5,10-dihydro-11-oxo-11H-dibenzo[b,e]-[1,4]diazepin-5-yl)carbonyl]methyl]-7,16-dimethyl-7,16-diaza-1,22-docosanediamine Tetraoxalate 675974 3-{2-[4-(4-Fluoro-benzyl)-piperidin-1-yl]-ethyl}-1H-quinazoline-2,4-dione hydrogen oxalate salt 675976 (1-Benzyl-piperidin-4-yl)-(4-fluoro-phenyl)-methanone hydrogen oxalate salt 675977 N-{2-[4-(4-Fluoro-benzoyl)-piperidin-1-yl]-ethyl}-benzamide hydrogen oxalate salt 675978 3-{2-[Methyl-(3-phenyl-propyl)-amino]-ethyl}-1H-quinazoline-2,4-dione hydrogen oxalate salt 675979 1-{2-[4-(4-Fluoro-benzoyl)-piperidin-1-yl]-ethyl}-3-phenyl-urea hydrogen oxalate salt 675980 (4-Fluoro-phenyl)-[1-(5-phenyl-pentyl)-piperidin-4-yl]-methanone hydrogen oxalate salt 675981 (4-Fluoro-phenyl)-[1-(3-phenyl-propyl)-piperidin-4-yl]-methanone hydrogen oxalate salt 676152 4-(1-Pentyl-1,2,5,6-tetrahydro-pyridin-3-yl)-thiazol-2-ylamine dihydrobromide 676249 7-methyl-2,3-dihydroxy-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine hydrobromide 676376 (-)-10-Keto-3-hydroxy-N-cyclopropylmethyl morphinan hydrochloride 676378 (-)-10-Keto-3-hydroxy-N-[(S)-tetrahydrofurfuryl] morphinan hydrochloride 676381 oxymorphone N-(Hydrazinocarbonyl)phenylalanyl-leucine hydrochloride 676383 oxymorphone semicarbazone hydrochloride 676384 Naltrexone N-(Hydrazinocarbonyl)phenylalanyl-leuine hydrochloride 676424 4-Fluoro-5-[6-methoxy-7-(1-methyl-piperidin-4-ylmethoxy)-quinazolin-4-ylamino]-2-methyl-phenol hydrochloride 676428 (4-Bromo-2-fluoro-phenyl)-{6-methoxy-7-[3-(4-methyl-piperazin-1-yl)-propoxy]-quinazolin-4-yl}-amine hydrochloride 676429 (4-Bromo-2-fluoro-phenyl)-[6-methoxy-7-(4-pyrrolidin-1-yl-but-2-enyloxy)-quinazolin-4-yl]-amine hydrochloride 676842 6-Methyl-1-naphthalen-1-ylmethyl-2,3,4,4a,9,9a-hexahydro-1H-beta-carboline hydrochloride 676875 (9-Methyl-9H-purin-6-yl)-(1-phenyl-propyl)-amine hydrochloride 676876 (9-Methyl-9H-purin-6-yl)-(1-phenyl-propyl)-amine hydrochloride 676952 4-(1-Phenethyl-1,2,5,6-tetrahydro-pyridin-3-yl)-thiazol-2-ylamine dihydrochloride 676953 4-[1-(3-Methyl-butyl)-1,2,5,6-tetrahydro-pyridin-3-yl]-thiazol-2-ylamine dihydrochloride 676954 4-(1-Hexyl-1,2,5,6-tetrahydro-pyridin-3-yl)-thiazol-2-ylamine dihydrochloride 676955 4-(1-Heptyl-1,2,5,6-tetrahydro-pyridin-3-yl)-thiazol-2-ylamine dihydrochloride 676958 4-(1-Butyl-1,2,5,6-tetrahydro-pyridin-3-yl)-thiazol-2-ylamine dihydrochloride 676959 4-(1-Methyl-1,2,5,6-tetrahydro-pyridin-3-yl)-thiazol-2-ylamine dihydrochloride 677167 N-[4-(4-{2-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-acetyl}-piperazin-1-yl)-phenyl]-methanesulfonamide hydrochloride hydrate 677326 4-[4-(4-Fluoro-benzoyl)-piperidin-1-yl]-1-phenyl-butan-1-one hydrochloride 677875 (+/-)-trans-2,3-dihydroxy-7-propyl-6a,7,8,12b-tetrahydro-6H-chromeno[3,4-c]isoquinoline hydrochloride 677885 4-(4'-fluoroanilino)-6,7-dimethoxyquinazoline hydrochloride 677886 4-[3'fluoro-5'-(trifluoromethyl)anilino)]-6,7-diethoxyquinazoline hydrochloride 677887 4-[3'-fluoro-5'-(trifluoromethyl)anilino]-6,7-dimethoxyquinazoline hydrochloride 677888 4-[(4'-fluorobenzyl)amino]-6,7-diethoxyquinazoline hydrochloride 677889 4-[(4'-fluorobenzyl)amino]-6,7-dimethoxyquinazoline hydrochloride 677890 4-(2'-fluoroanilino)-6,7-diethoxyquinazoline hydrochloride 677891 4-(4'-fluoroanilino)-6,7-diethoxyquinazoline hydrochloride 677897 7-{4-[4-(2-methoxyphenyl)-piperazin-1-yl]-butyl}-8-ethoxy-1,3-dimethyl-3,7-dihydropurine-2,6-dione hydrochloride 678073 3-hydroxy-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine hydrobromide 678119 4-(3'-bromoanilino)-6,7-dimethoxyquinazoline hydrochloride 678150 4-(3'-bromoanilino)-6,7-diethoxyquinazoline hydrochloride 678176 3-(4-(2-(6-amino-9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxytetrahydrofuran-2-yl)-9H-purin-2-ylamino)ethyl)phenyl)propanoic acid hydrochloride 678212 4-(3'-fluoroanilino)-6,7-diethoxyquinazoline hydrochloride 678213 4-(3'-iodoanilino)-6,7-diethoxyquinazoline hydrochloride 678256 4-(3'-iodoanilino)-6,7-dimethoxyquinazoline hydrochloride 678311 4-(2'-fluoroanilino)-6,7-dimethoxyquinazoline hydrochloride 678337 trans-2-(3-biphenyl-2-yl-oxiranyl)-4,5-dihydro-1H-imidazole hydrochloride 685651 3-(2-(4-bromophenyl)-2-oxoethylidene)indolin-2-one 690661 7-(2,6-difluorophenyl)-5-methyl-N-(4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)benzo[e][1,2,4]triazin-3-amine 695650 SID26755032 696004 5-(2-methylpiperazin-1-ylsulfonyl)isoquinoline 699395 Tramadol 699512 4-[(4-{4-[3-(pyridin-2-yl)-1H-pyrazol-4-yl]-2-pyridinyl}phenyl)-methyl]morpholine Hydrochloride 699515 Naltrindole hydrochloride 699646 (E)-3-{2-[(E)-3-(2-Benzyloxy-3-methyl-phenyl)-allyl]-phenyl}-acrylic acid; compound with (E)-3-{2-[(E)-3-(2-benzyloxy-3-methyl-phenyl)-propenyl]-phenyl}-acrylic acid 699647 (E)-3-{2-[(E)-3-(2-Benzyloxy-3-hydroxy-phenyl)-allyl]-phenyl}-acrylic acid; compound with (E)-3-{2-[(E)-3-(2-benzyloxy-3-hydroxy-phenyl)-propenyl]-phenyl}-acrylic acid 699648 (E)-3-{2-[(E)-3-(2-Benzyloxy-phenyl)-allyl]-phenyl}-acrylic acid; compound with (E)-3-{2-[(E)-3-(2-benzyloxy-phenyl)-propenyl]-phenyl}-acrylic acid 699649 (E)-3-{2-[(E)-3-(3-Benzyloxy-phenyl)-allyl]-phenyl}-acrylic acid; compound with (E)-3-{2-[(E)-3-(3-benzyloxy-phenyl)-propenyl]-phenyl}-acrylic acid 699650 (E)-3-{3-[(E)-3-(2-Benzyloxy-3-methyl-phenyl)-propenyl]-phenyl}-acrylic acid; compound with (E)-3-{3-[(E)-3-(2-benzyloxy-3-methyl-phenyl)-allyl]-phenyl}-acrylic acid 699651 (E)-3-{4-[(E)-3-(2-Benzyloxy-3-methyl-phenyl)-allyl]-phenyl}-acrylic acid; compound with (E)-3-{4-[(Z)-3-(2-benzyloxy-3-methyl-phenyl)-propenyl]-phenyl}-acrylic acid 699652 2-[(E)-3-(2-Benzyloxy-3-methyl-phenyl)-allyl]-benzoic acid; compound with 2-[(E)-3-(2-benzyloxy-3-methyl-phenyl)-propenyl]-benzoic acid 699653 {2-[(E)-3-(2-Benzyloxy-3-methyl-phenyl)-allyl]-phenyl}-acetic acid; compound with {2-[(E)-3-(2-benzyloxy-3-methyl-phenyl)-propenyl]-phenyl}-acetic acid 699654 (E)-3-{2-[(E)-3-(5-Acetyl-2-benzyloxy-phenyl)-allyl]-phenyl}-acrylic acid; compound with (E)-3-{2-[(E)-3-(5-acetyl-2-benzyloxy-phenyl)-propenyl]-phenyl}-acrylic acid 699655 (E)-3-{2-[(E)-3-(2-Phenoxy-phenyl)-allyl]-phenyl}-acrylic acid; compound with (E)-3-{2-[(E)-3-(2-phenoxy-phenyl)-propenyl]-phenyl}-acrylic acid 699656 (E)-3-(2-{(E)-3-[2-(2,6-Dichloro-benzyloxy)-3-hydroxymethyl-phenyl]-allyl}-phenyl)-acrylic acid; compound with (E)-3-(2-{(E)-3-[2-(2,6-dichloro-benzyloxy)-3-hydroxymethyl-phenyl]-propenyl}-phenyl)-acrylic acid 699666 3-(2-((E)-3-phenylprop-1-enyl)phenyl)acrylic acid 699667 3-(2-((E)-3-(4-methoxyphenyl)prop-1-enyl)phenyl)acrylic acid 699668 3-(2-((E)-3-(4-(benzyloxy)-3-methoxyphenyl)prop-1-enyl)phenyl)acrylic acid 700097 N3-(4-fluorophenyl)-1H-pyrazolo[3,4-d]pyrimidine-3,4-diamine 702208 (S)-methyl 4-hydroxy-2-(4-hydroxy-3-(3-methylbut-2-enyl)benzyl)-3-(4-hydroxyphenyl)-5-oxo-2,5-dihydrofuran-2-carboxylate 703576 N-(2-oxo-2-(2-(2-oxoindolin-3-ylidene)hydrazinyl)ethyl)-N-phenylbenzenesulfonamide 703577 4-ethoxy-N-(2-oxo-2-(2-(2-oxoindolin-3-ylidene)hydrazinyl)ethyl)-N-p-tolylbenzenesulfonamide 705778 Formoterol 705840 1,1'-(decane-1,10-diyl)bis(4-amino-2-methylquinolinium) iodide 706000 (+)-butaclamol 706008 SID46500333 739341 Dequalinium Analogue 840088 SID11113565 936429 SID26756649 957194 Histamine dihydrochloride 1049913 Sodium salt of N-{6-[2-(5-Bromo-pyrimidin-2-yloxy)-ethoxy]-5-p-tolyl-pyrimidin-4-yl}-4-(2-hydroxy-1,1-dimethyl-ethyl)-benzenesulfonamide 1049914 Sodium salt of 4-tert-Butyl-N-{6-[2-(5-hydroxymethyl-pyrimidin-2-yloxy)-ethoxy]-5-p-tolyl-pyrimidin-4-yl}-benzenesulfonamide 1051134 (-)-3-Hydroxy-N-methylmorphinan hydrochloride (levorphanol) 1077179 6-Amino-9-(3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-1,9-dihydro-purin-2-one 1077963 (7-chloro-2,3-dimethylquinolin-4-yl)-[4-(3,4-dimethylpiperazin-1-yl)phenyl]amine 1121348 4-Fluoro-N-{2-[4-((R)-2-hydroxymethyl-2,3-dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-ethyl}-benzamide 1122200 (trans)4-[4-(5-methoxy-2,3,4,4a,9,9a-hexahydro-1H-indeno[2,1-c]pyridin-2-yl)butyl]-4-azatetracyclo[5.4.2.02,6.08,11]trideca-9,12-diene-3,5-dione HCl 1122591 N-{4-[(3a,4,5,9b-Tetrahydro-1H-benzo[e]indol-2-ylamino)-methyl]-cyclohexylmethyl}-benzenesulfonamide 1122606 8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]indole-2-carbonitrile 1122607 8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]indole-2-carboxylic acid amide 1122608 8-{[4-(4,4-Dimethyl-2,6-dioxo-piperidin-1-yl)-butyl]-propyl-amino}-6,7,8,9-tetrahydro-3H-benzo[e]indole-2-carboxylic acid amide 1122615 3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-5-methylsulfanyl-2,3,5,6-tetrahydro-imidazo[1,2-c]quinazoline 1122643 2-(4-Methoxy-1H-indol-3-yl)-1-methyl-ethylamine 1122644 2-(6-Methoxy-1H-indol-3-yl)-1-methyl-ethylamine 1122645 3-(2-Amino-propyl)-1H-indol-4-ol 1122659 8-{[4-(4,4-Dimethyl-2,6-dioxo-piperidin-1-yl)-butyl]-propyl-amino}-6,7,8,9-tetrahydro-3H-benzo[e]indole-2-carbonitrile 1122660 8-Propylamino-6,7,8,9-tetrahydro-3H-benzo[e]indole-2-carboxylic acid amide 1122731 3-[2-(4-Benzyl-piperidin-1-yl)-ethyl]-1H-quinazoline-2,4-dione maleate 1122733 3-[2-(4-Benzoyl-piperidin-1-yl)-ethyl]-1H-quinazoline-2,4-dione maleate 1122918 (4-Chloro-2-fluoro-phenyl)-{6-methoxy-7-[3-(4-methyl-piperazin-1-yl)-propoxy]-quinazolin-4-yl}-amine hydrochloride 1122920 (4-Chloro-2-fluoro-phenyl)-[6-methoxy-7-(4-pyrrolidin-1-yl-but-2-enyloxy)-quinazolin-4-yl]-amine hydrochloride 1151780 1,3-Benzothiazol-2-yl(2-{[2-(3-pyridinyl)ethyl]amino}-4-pyrimidinyl)acetonitrile (Bis(trifluoroacetate)) 1151798 (4-Fluoro-phenyl)-(1-phenethyl-piperidin-4-yl)-methanone hydrogen oxalate salt 1151799 (4-Fluoro-phenyl)-[1-(4-phenyl-butyl)-piperidin-4-yl]-methanone hydrogen oxalate salt 1151855 8-{[4-(4,4-Dimethyl-2,6-dioxo-piperidin-1-yl)-butyl]-propyl-amino}-6,7,8,9-tetrahydro-3H-benzo[e]indole-2-carboxylic acid amide 1151856 8-(Cyclopropylmethyl-propyl-amino)-6,7,8,9-tetrahydro-3H-benzo[e]indole-2-carboxylic acid amide 1151863 Hydroxy-diphenyl-acetic acid 1-aza-bicyclo[2.2.2]oct-3-yl ester 1151886 3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-2,6-dihydro-3H-imidazo[1,2-c]quinazolin-5-one 1151887 3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-5-methylsulfanyl-2,3,5,6-tetrahydro-imidazo[1,2-c]quinazoline 1151903 3-(2-Amino-propyl)-1H-indol-5-ol 1151939 3,4-diarylpyrazoline derivative 1151940 (2-Iodo-phenyl)-[1-((S)-1-methyl-piperidin-2-ylmethyl)-1H-indol-3-yl]-methanone 1151944 2-(4-Methoxy-1H-indol-3-yl)-1-methyl-ethylamine 1151945 2-(5-Methoxy-1H-indol-3-yl)-1-methyl-ethylamine 1151946 2-(6-Methoxy-1H-indol-3-yl)-1-methyl-ethylamine 1151948 3-(2-Amino-propyl)-1H-indol-4-ol 1151949 2-(1H-Indol-3-yl)-1-methyl-ethylamine 1151950 9H-Xanthene-9-carboxylic acid 1-aza-bicyclo[2.2.2]oct-3-yl ester 1151951 2-(4-Iodo-phenyl)-1-methyl-ethylamine 1151986 6-Chloro-1-phenyl-1,2,3,4-tetrahydro-isoquinolin-7-ol 1153676 MCL-117 1154130 3-[8-sec-Butyl-14-(1H-indol-3-ylmethyl)-11-isobutyl-5-methyl-3,6,9,12,15-pentaoxo-1,4,7,10,13pentaaza-cyclopentadec-2-yl]-propionic acid 1154142 5-[3-amino(imino)methylaminopropyl]-3-[2-methyl-1-spiro[2,3-dihydro-1H-indene-1,4'-(hexahydropyridine)]-1-ylcarbonyl-(1R)-propyl]-(5R)-tetrahydro-1H-2,4-imidazoledione 1154150 3-{2-[2-Acetylamino-2-(10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5-yl)-acetylamino]-4-methyl-pentanoylamino}-N-[1-({1-[1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butyl}-methyl-carbamoyl)-2-methyl-butyl]-succinamic acid 1154173 16,24-dibenzyl-13-(sec-butyl)-25-methyl-1,3,4,6,6a,7,8,13,14,15,16,17,18,18a,19,20,21,23,24,25,26,26a-docosahydro-2H,12H-dipyridazino[1,6-a:1,6-d]pyrrolo[1,2-j][1,4,7,10,13,16]hexaazacyclooctadecine-3,6,12,15,18,23,26-heptaone (Oxytocin analogues) 1154174 16,24-dibenzyl-13-(sec-butyl)-25-methylperhydrodipyridazino[1,6-a:1,6-d]pyrrolo[1,2-j][1,4,7,10,13,16]hexaazacyclooctadecine-3,6,12,15,18,23,26-heptaone (Oxytocin analogues) 1154175 16,24-dibenzyl-13-(sec-butyl)-25-methyl-15-thioxo-1,6,6a,7,8,13,14,15,16,17,18,18a,19,20,21,23,24,25,26,26a-icosahydro-2H,12H-dipyridazino[1,6-a:1,6-d]pyrrolo[1,2-j][1,4,7,10,13,16]hexaazacyclooctadecine-6,12,18,23,26-pentaone (Oxytocin analogues) 1154177 16,24-dibenzyl-13-(sec-butyl)-25-methyl-1,6,6a,7,8,13,14,15,16,17,18,18a,19,20,21,23,24,25,26,26a-icosahydro-2H,12H-dipyridazino[1,6-a:1,6-d]pyrrolo[1,2-j][1,4,7,10,13,16]hexaazacyclooctadecine-6,12,15,18,23,26-hexaone (Oxytocin analogues) 1154178 16,24-dibenzyl-13-(sec-butyl)-25-methyl-(24R)-6,6a,7,8,13,14,15,16,17,18,18a,19,20,21,24,25,26,26a-octadecahydro-12H,23H-dipyridazino[1,6-a:1,6-d]pyrrolo[1,2-j][1,4,7,10,13,16]hexaazacyclooctadecine-6,12,15,18,23,26-hexaone (Oxytocin analogues) 1154179 16,24-dibenzyl-13-(sec-butyl)-25-methylperhydrodipyridazino[1,6-a:1,6-d]pyrrolo[1,2-j][1,4,7,10,13,16]hexaazacyclooctadecine-6,12,15,18,23,26-hexaone (Oxytocin analogues) 1154180 16,24-dibenzyl-13-(sec-butyl)-14-hydroxy-25-methylperhydrodipyridazino[1,6-a:1,6-d]pyrrolo[1,2-j][1,4,7,10,13,16]hexaazacyclooctadecine-6,12,15,18,23,26-hexaone (Oxytocin analogues) 1154181 16,24-dibenzyl-13-(sec-butyl)-25-methyl-1,6,6a,7,8,13,14,15,16,17,18,18a,19,20,21,23,24,25,26,26a-icosahydro-2H,12H-dipyridazino[1,6-a:1,6-d]pyrrolo[1,2-j][1,4,7,10,13,16]hexaazacyclooctadecine-6,12,18,23,26-pentaone (Oxytocin analogues) 1154182 16,24-dibenzyl-13-(sec-butyl)-2-N,N dimethylmethyl-25-methyl-1,6,6a,7,8,13,14,15,16,17,18,18a,19,20,21,23,24,25,26,26a-icosahydro-2H,12H-dipyridazino[1,6-a:1,6-d]pyrrolo[1,2-j][1,4,7,10,13,16]hexaazacyclooctadecine-6,12,15,18,23,26-hexaone (Oxytocin analogues) 1154183 16,24-dibenzyl-13-(sec-butyl)-4,10,25-trimethylperhydrodipyridazino[1,6-a:1,6-d]pyrrolo[1,2-j][1,4,7,10,13,16]hexaazacyclooctadecine-6,12,15,18,23,26-hexaone (Oxytocin analogues) 1154203 10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionylamino)-16-(4-hydroxy-benzyl)-13-(1-hydroxy-ethyl)-7-isopropyl-3,3-dimethyl-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentaaza-cycloicosane-4-carboxylic acid (1-carbamoyl-2-hydroxy-propyl)-amide (D-Phe-Cys-Tyr-D-Thr-Lys-Val-Pen-Thr-NH2) 1154342 d[Thr4,Orn8(5/6C-Flu)]VT 1154343 d(CH2)5[Tyr(Me)2,Thr4,Orn8,Tyr9-NH2]VT 1154344 d(CH2)5[Tyr(Me)2,Thr4,Orn8(5/6C-Flu),Tyr-NH29]VT 1154348 [HO1][Lys8(5/6C-Flu)]VT 1154349 d[Lys8(5/6-Flu)]VT 1154350 [HO1][Thr4,Orn8(5/6C-Flu)]VT 1154351 [HO1][Orn8(5/6C-Flu)]VT 1154352 d[Orn8(5/6C-Flu)]VT 1154353 desGly-NH2,d(CH2)5[D-Tyr2,Thr4,Orn8(5/6C-Flu)]VT 1154354 [HO1][Orn8(5/6C-Rhm)]VT 1154359 d[Thr4,Lys8(5/6C-Flu)]VT 1154360 [HO1][Thr4,Lys8(5/6C-Flu)]VT 1154409 Tyr-D-Ala-Phe-Gly-Tyr-Pro-Thr(Beta-D-Glc)-Gly-NH2 1154410 Tyr-D-Ala-Phe-Asp-Val-Val-Thr[Beta-D-Glc(OAc)4]-Gly-NH2 1154590 c(Cys-Ser-c(Cys-Ser-Ser-Leu-Met-Asp-Lys-Gln-Cys)-Val-Tyr-Phe-Cys)-His-Leu-Thr-Val-Ile-Trp 1154591 c(Cys-Ser-c(Cys-Ser-Ser-Leu-Met-Asp-Lys-Gln-Cys)-Val-Tyr-Phe-Cys)-His-Leu-Thr-Nva-Ile-Trp 1154593 c(Cys-Ser-c(Cys-Ser-Ser-Leu-Met-Asp-Lys-Gln-Cys)-Val-Tyr-Phe-Cys)-His-Leu-Thr-Leu-Ile-Trp 1154594 c(Cys-Ser-c(Cys-Ser-Ser-Leu-Met-Asp-Lys-Gln-Cys)-Val-Tyr-Phe-Cys)-His-Leu-Thr-Ile-Ile-Trp 1154633 (S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-({(S)-2-[(S)-3-(1H-indol-3-yl)-2-(2-{(S)-3-methyl-2-[2-(4-sulfooxy-phenyl)-acetylamino]-pentanoylamino}-acetylamino)-propionylamino]-3-methyl-pentanoyl}-methyl-amino)-succinamic acid 1154636 (S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-({(S)-2-[(S)-3-(1H-indol-3-yl)-2-(2-{(S)-2-[2-(4-sulfooxy-phenyl)-acetylamino]-hexanoylamino}-acetylamino)-propionylamino]-3-methyl-pentanoyl}-methyl-amino)-N-methyl-succinamic acid 1154902 (S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propionylamino)-4-methyl-pentanoylamino]-N-((S)-1-{(S)-1-[(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 1154908 (S)-3-{(S)-2-[(S)-2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-3-carboxy-propionylamino}-N-((S)-1-{(S)-1-[(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 1154910 (S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-4-methyl-pentanoylamino]-N-((S)-1-{(S)-1-[(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 1154911 (S)-2-{(S)-2-[(S)-2-((S)-2-{(S)-2-[(S)-2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-4-methyl-pentanoylamino}-3-carbamoyl-propionylamino)-3-methyl-pentanoylamino]-3-methyl-pentanoylamino}-3-(1H-indol-3-yl)-propionic acid 1154935 Pyz6-D-Trp8-SRIF 1154936 Pyz7-D-Trp8-SRIF 1154937 D-Trp8-SRIF-14 1154938 Ala11-SRIF-14-amide 1154943 Pyz11-D-Trp8-SRIF 1154944 GaIII-DOTATOC 1154945 YIII-DOTATOC 1154987 Ac-Cys-Ile-Tyr-Lys-Phe(4-Cl)-Tyr 1154989 (S)-2-((S)-2-((S)-2-((S)-2-((2S,3S)-2-((R)-2-acetamido-3-mercaptopropanamido)-3-methylpentanamido)-3-(4-hydroxyphenyl)propanamido)-6-aminohexanamido)-3-(4-nitrophenyl)propanamido)-3-(4-hydroxyphenyl)propanoic acid 1154990 Ac-Cys-Ile-Phe(4-NH2)-Lys-Tyr-Tyr 1154991 Ac-Cys-Ile-Tyr-Lys-Phe(4-F)-Tyr 1154992 Ac-Cys-Ile-Phe(4-NO2)-Lys-Phe(4-NO2)-Tyr 1154993 Ac-Cys-Ile-Tyr-Lys-Phe(4-I)-Tyr 1154995 Ac-Cys-Ile-Tyr-cyclo[Lys-Tyr-Tyr] 1154996 Cyclo[Ac-Cys-Ile-Tyr-Lys]-Tyr-Tyr 1154998 Ac-Cys-Ile-Tyr-Lys-Phe(4-NH2)-Tyr 1154999 Ac-Cys-Ile-Tyr-Lys-Phe(4-CN)-Tyr 1155000 Cyclo[Ac-Cys-Ile-Phe]-Lys-Tyr-Tyr 1155001 Ac-Cys-Ile-Tyr-Lys-Tyr-Tyr 1155002 Ac-Cys-Ile-Tyr-Lys-Tyr-Phe(4-NO2) 1155003 Ac-Cys-Ile-Phe(4-NO2)-Lys-Tyr-Phe(4-NO2) 1155004 Ac-Cys-Ile-Tyr-Lys-Phe(4-NO2)-Tyr-Phe 1155005 Ac-Cys-Ile-Phe(4-NO2)-Lys-Tyr-Tyr 1155006 Ac-Cys-Ile-Tyr-Lys-Phe(4-NO2)-Phe(4-NO2) 1155007 Ac-Cys-Ile-Tyr-Lys-Phe(4-N3)-Tyr 1155009 Cyclo[Ac-Cys-Ile-Tyr-Lys]-Phe(4-NO2)-Tyr 1155014 Demotensin 2 1155054 2-(6-Amino-purin-9-yl)-5-(1-hydroxy-prop-2-ynyl)-tetrahydro-furan-3,4-diol 1155074 3,4-Dihydroxy-5-(6-{3-[4-(5-methyl-isoxazol-3-ylsulfamoyl)-phenyl]-ureido}-purin-9-yl)-tetrahydro-furan-2-carboxylic acid ethylamide 1155078 Dynorphin(1-8) 1157462 (2S,5S)-2-(3-Methanesulfonyl-5-methoxy-4-propoxy-phenyl)-5-(3,4,5-trimethoxy-phenyl)-tetrahydro-furan 1157468 (S)-2-{(R)-2-[2-({1-[2-(2-Amino-5-guanidino-pentanoylamino)-5-guanidino-pentanoyl]-pyrrolidine-2-carbonyl}-amino)-3-(4-hydroxy-phenyl)-propionylamino]-3-methyl-pentylamino}-3-phenyl-propionic acid 1157469 (S)-2-{(R)-2-[2-({1-[2-(2-Amino-5-guanidino-pentanoylamino)-5-guanidino-pentanoyl]-pyrrolidine-2-carbonyl}-amino)-3-(4-hydroxy-phenyl)-propylamino]-3-methyl-pentanoylamino}-4-methyl-pentanoic acid 1157470 (S)-2-{(R)-2-[2-({1-[2-(2-Amino-5-guanidino-pentanoylamino)-5-guanidino-pentanoyl]-pyrrolidine-2-carbonyl}-amino)-3-(4-hydroxy-phenyl)-propionylamino]-3-methyl-pentanoylamino}-3-phenyl-propionic acid 1157496 (1S,2S,4S)-2-{2-[(S)-2-({1-[6-Amino-2-(2,6-diamino-hexylamino)-hexanoyl]-pyrrolidine-2-carbonyl}-amino)-3-(4-hydroxy-phenyl)-1-(S)-oxo-propylamino]-3-methyl-pentanoylamino}-4-methyl-pentanoic acid 1157555 N-[1-((S)-3-Acetylamino-2-oxo-4,4-diphenyl-butylcarbamoyl)-3-methyl-butyl]-3-(2-{2-[2-amino-3-(1H-indol-3-yl)-propionylamino]-3-methyl-pentanoylamino}-3-methyl-pentanoylamino)-succinamic acid 1157557 3-{2-[((S)-2-Acetylamino-3,3-diphenyl-propionyl)-methyl-amino]-4-methyl-pentanoylamino}-N-(1-{1-[1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 1157558 3-{2-[(S)-2-(Acetyl-methyl-amino)-3,3-diphenyl-propionylamino]-4-methyl-pentanoylamino}-N-(1-{1-[1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 1157563 3-[2-((S)-2-Acetylamino-3,3-diphenyl-propionylamino)-4-methyl-pentanoylamino]-5-(2-{2-[2-amino-3-(1H-indol-3-yl)-propionylamino]-3-methyl-pentanoylamino}-3-methyl-pentanoylamino)-4-oxo-pentanoic acid 1157565 3-{[2-((S)-2-Acetylamino-3,3-diphenyl-propionylamino)-4-methyl-pentanoyl]-methyl-amino}-N-(1-{1-[1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid 1157627 4-{2-[2-[(1-Acetyl-pyrrolidine-2-carbonyl)-amino]-3-(4-hydroxy-phenyl)-propionylamino]-4-carboxy-butyrylamino}-4-(1-carbamoyl-2-methyl-butylcarbamoyl)-butyric acid 1157682 3-(3,5-dibromo-4-hydroxybenzylidene)-5-iodoindolin-2-one 1157684 2-Methyl-furan-3-carboxylic acid [4-({2-[4-([1,4']bipiperidinyl-1'-carbonyl)-phenoxy]-phenyl}-methyl-carbamoyl)-phenyl]-amide 1157691 (3,4-Dimethoxy-phenyl)-(5-phenyl-oxazol-2-yl)-amine 1157692 3-(5-Phenyl-oxazol-2-ylamino)-benzonitrile 1157693 (2-Methoxy-phenyl)-(5-phenyl-oxazol-2-yl)-amine 1157694 N-(4-(3-fluorobenzyloxy)-3-(trifluoromethyl)phenyl)-6-(5-((2-(phenylsulfonyl)ethylamino)methyl)furan-2-yl)quinazolin-4-amine 1158139 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (1R,2S,4S)-4-hydroxy-2-(4-hydroxy-benzoylamino)-cyclopentyl ester; compound with 4-(2-carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (1R,2S,4R)-4-hydroxy-2-(4-hydroxy-benzoylamino)-cyclopentyl ester 1158145 Benzyl-[2-(3-fluoro-phenyl)-3H-imidazol-4-ylmethyl]-methyl-amine; dimaleate 1158250 8-chloro-11-(piperazin-1-yl)-dibenzo[b,f][1,4]oxazepin fumaric acid 1158373 8-chloro-11-(4-ethylpiperazin-1-yl)-dibenzo[b,f][1,4]oxazepine fumaric acid 1158374 8-[2-(3,4-Dimethoxy-phenyl)-vinyl]-7-methyl-1,3-dipropyl-3,7-dihydro-purine-2,6-dione; compound with 8-[2-(3,4-dimethoxy-phenyl)-vinyl]-7-methyl-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 1158759 H-D-Phe-c[Cys-Tyr-D-Trp-Arg-Thr-Pen]-Thr-NH2 (CTAP) 1173967 somatostatin 1209164 8-(tert-butyl)-6,9,12,17-tetrahydroxy-16-methyl-(6R,8R,9S,12R,16S,17R)-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,15,18-trione 1248202 (S)-1-[4-(4-benzhydrylthiosemicarbazido)-3-nitrobenzenesulfonyl]pyrrolidine-2-carboxylic acid{2-[(3-dimethylaminopropyl)methylamino]ethyl}amide 1248203 (S)-1-[4-(4-benzhydrylthiosemicarbazido)-3-nitrobenzenesulfonyl]pyrrolidine-2-carboxylic acid{3-[(3-dimethylaminopropyl)methylamino]propyl}amide 1248204 1-(3-Chloro-benzenesulfonyl,4-N-benzhydrylhydrazinecarboxamide)-pyrrolidine-2-carboxylic acid {2-[(2-dimethylamino-ethyl)-methyl-amino]-ethyl}-amide 1248205 (S)-1-(4-{4-bis-(2-chloro-phenyl)methyl]thiosemicarbazido)-3-nitrobenzenesulfonyl]pyrrolidine-2-carboxylic acid{2-[(2-dimethylaminoethyl)methylamino]ethyl}amide 1248206 (S)-1-(4-[4-(10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5-yl)thiosemicarbazido]-3-nitrobenzenesulfonyl)pyrrolidine-2-carboxylic acid amide 1248207 (S)-1-(4-[4-(10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5-yl)thiosemicarbazido]-3-nitrobenzenesulfonyl]pyrrolidine-2-carboxylic acid{2-[(2-dimethylaminoethyl)methylamino]ethyl}amide 1248208 (S)-1-(4-[4-(9H-fluoren-9-yl)thiosemicarbazido)-3-nitrobenzenesulfonyl]pyrrolidine-2-carboxylic acid{2-[(3-dimethylaminopropyl)methylamino]ethyl}amide 1248241 (S)-3-Bromo-N-(1-ethyl-pyrrolidin-2-ylmethyl)-6-hydroxy-2,5-dimethoxy-benzamide 1248243 (S)-3-Chloro-N-(1-ethyl-pyrrolidin-2-ylmethyl)-2-hydroxy-5,6-dimethoxy-benzamide; methanesulphite 1248246 (S)-N-(1-Ethyl-pyrrolidin-2-ylmethyl)-2-hydroxy-5,6-dimethoxy-3-propyl-benzamide; compound with 2,3-dihydroxy-but-2-enedioic acid 1248253 (S)-3-Ethyl-N-(1-ethyl-pyrrolidin-2-ylmethyl)-2-hydroxy-5,6-dimethoxy-benzamide; methanesulphite 1248259 (R)-(1H-Imidazo[4,5-c]quinolin-4-yl)-(1-methyl-2-phenyl-ethyl)-amine HCl 1248309 Ser-Ala-Asn-Ser-Asn-Pro-Ala-Met-Ala-Pro-Arg-Glu-Arg-Lys-Ala-Gly-Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-Ser-Cys 1248314 (R)-(4-Chloro-2-fluoro-phenyl)-[6-methoxy-7-(1-methyl-piperidin-3-ylmethoxy)-quinazolin-4-yl]-amine 1248315 (R)-(4-Bromo-2-fluoro-phenyl)-[6-methoxy-7-(1-methyl-piperidin-3-ylmethoxy)-quinazolin-4-yl]-amine 1248337 5-{(S)-3-[3-(1-{[2-(3,4-Dichloro-phenyl)-acetyl]-methyl-amino}-2-pyrrolidin-1-yl-ethyl)-phenyl]-thioureido}-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)-benzoic acid; compound with triethyl-amine 1248338 5-(3-{[({[({[(S)-3-(1-{[2-(3,4-Dichloro-phenyl)-acetyl]-methyl-amino}-2-pyrrolidin-1-yl-ethyl)-phenylcarbamoyl]-methyl}-carbamoyl)-methyl]-carbamoyl}-methyl)-carbamoyl]-methyl}-thioureido)-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)-benzoic acid; compoundwith triethyl-amine 1248339 5-(3-{[(S)-3-(1-{[2-(3,4-Dichloro-phenyl)-acetyl]-methyl-amino}-2-pyrrolidin-1-yl-ethyl)-phenylcarbamoyl]-methyl}-thioureido)-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)-benzoic acid; compound with triethyl-amine 1248340 5-{3-[({[(S)-3-(1-{[2-(3,4-Dichloro-phenyl)-acetyl]-methyl-amino}-2-pyrrolidin-1-yl-ethyl)-phenylcarbamoyl]-methyl}-carbamoyl)-methyl]-thioureido}-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)-benzoic acid; compound with triethyl-amine 1248403 4-Chloro-N-[5-(2-fluoro-phenyl)-1-methyl-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl]-benzamide 1248409 8-Acenaphthen-1-yl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 1248466 (R)-3-Bromo-N-(1-ethyl-pyrrolidin-2-ylmethyl)-2-hydroxy-5,6-dimethoxy-benzamide 1248475 (S)-(1H-Imidazo[4,5-c]quinolin-4-yl)-(1-methyl-2-phenyl-ethyl)-amine HCl 1248495 (S)-(4-Bromo-2-fluoro-phenyl)-[6-methoxy-7-(1-methyl-piperidin-3-ylmethoxy)-quinazolin-4-yl]-amine 1329859 8-[1-(3,4-Dichloro-phenyl)-meth-(E)-ylidene]-5-(3-hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]nonan-7-one 1336907 (R)-3-cyclopropylmethyl-19-(1-isothiocyanatoethyl)-15-methoxy-13-oxa-3-azahexacyclo[13.2.2.12,8.01,6.06,14.07,12]icosa-7,9,11,16-tetraen-11-ol 1336908 (R)-1-(3-cyclopropylmethyl-11,15-dimethoxy-13-oxa-3-azahexacyclo[13.2.2.12,8.01,6.06,14.07,12]icosa-7,9,11,18-tetraen-16-yl)ethyl isothiocyanate 1336910 (R)-19-(1-isothiocyanatoethyl)-15-methoxy-3-methyl-13-oxa-3-azahexacyclo[13.2.2.12,8.01,6.06,14.07,12]icosa-7,9,11,16-tetraen-11-ol 1337180 3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocin-8-ol 1341082 Icatibant 1341188 (2S,5R)-5-Ethyl-piperazine-2-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide; compound with ditrifluoroacetic acid 1341189 (2S,5R)-5-Isopropyl-piperazine-2-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide; compound with ditrifluoroacetic acid 1341190 (2S,5R)-5-Cyclopropyl-piperazine-2-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide; compound with ditrifluoroacetic acid 1341191 (2S,5R)-5-tert-Butyl-piperazine-2-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide; compound with ditrifluoroacetic acid 1341192 (2S,5R)-5-(1-Methyl-cyclopropyl)-piperazine-2-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide; compound with ditrifluoroacetic acid 1341193 (S)-4,7-Diaza-spiro[2.5]octane-6-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide; compound with ditrifluoroacetic acid 1341194 (S)-6-Isopropyl-piperazine-2-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide; compound with ditrifluoroacetic acid 1341199 H-Dmt-Tic-Lys(Z)-NH-CH2-Ph 1341200 H-Dmt-Tic-Lys(Ac)-NH-CH2-Ph 1341201 H-Dmt-Tic-Lys-NH-CH2-Ph 1341202 H-Dmt-Tic-Lys(Z)-NH-Ph 1341203 H-Dmt-Tic-Lys(Ac)-NH-Ph 1341204 H-Dmt-Tic-Lys-NH-Ph 1352714 isomer-13-(Octahydro-quinolizin-3-yl)-phenol 1352914 1-[3-(4,4-diphenylhexahydro-1-pyridinyl)propyl] 3-methyl 4,6-dimethyl-2-phenyl(3-nitro)-3,6-cyclohexadiene-1,3-dicarboxylate (niguldipine) 1352922 22-cyclopropylmethyl-14-oxa-11,22-diazaheptacyclo[13.9.1.01,13.02,21.04,12.05,10.019,25]pentacosa-4(12),5(10),6,8,15,17,19(25)-heptaene-2,16-diol 1352933 4-Methyl-1-{2-[(R)-1-(toluene-3-sulfonyl)-pyrrolidin-2-yl]-ethyl}-piperidine 1352971 (S)-2-((S)-2-{2-[(S)-2-Diallylamino-3-(4-hydroxy-phenyl)-propionylamino]-2-methyl-propionylamino}-3-phenyl-propionylamino)-4-methyl-pentanoic acid; compound with 4-[(S)-((2S,5R)-4-allyl-2,5-dimethyl-piperazin-1-yl)-(3-methoxy-phenyl)-methyl]-N,N-diethyl-benzamide 1352975 (5S,8R,11R,14R,17R,19aR)-11-(4-Amino-butyl)-17-benzyl-5-(4-hydroxy-benzyl)-14-(1-hydroxy-ethyl)-8-(1H-indol-3-ylmethyl)-tetradecahydro-3a,6,9,12,15,18-hexaaza-cyclopentacyclooctadecene-4,7,10,13,16,19-hexaone 1355735 N-{(R)-2-[(S)-2-(Adamantan-2-yloxycarbonylamino)-3-(1H-indol-3-yl)-2-methyl-propionylamino]-1-phenyl-ethyl}-succinamic acid 1355745 N-{(R)-2-[(R)-2-(adamantan-2-yloxycarbonylamino)-3-(1H-indol-3-yl)-2-methyl-propionylamino]-1-phenyl-ethyl}-succinamic acid 1358261 3-[(2-Adamantan-1-ylmethyl-5-phenyl-1H-pyrrole-3-carbonyl)-amino]-propionic acid; compound with 6-methylamino-hexane-1,2,3,4,5-pentaol 1358262 5-[(2-Cycloheptylmethyl-5-phenyl-1H-pyrrole-3-carbonyl)-amino]-isophthalic acid; compound with 6-methylamino-hexane-1,2,3,4,5-pentaol 1358263 5-[(S)-2-({6-[(Adamantan-1-ylmethyl)-carbamoyl]-1H-indole-5-carbonyl}-amino)-3-phenyl-propionylamino]-isophthalic acid; compound with 6-methylamino-hexane-1,2,3,4,5-pentaol 1358264 5-[(5-Cycloheptylmethyl-2-naphthalen-2-yl-1H-imidazole-4-carbonyl)-amino]-isophthalic acid; compound with 6-methylamino-hexane-1,2,3,4,5-pentaol 1358265 5-[(S)-2-({6-[(Adamantan-1-ylmethyl)-carbamoyl]-1H-benzoimidazole-5-carbonyl}-methyl-amino)-3-phenyl-propionylamino]-isophthalic acid; compound with 6-methylamino-hexane-1,2,3,4,5-pentaol 1358267 5-Cycloheptylmethyl-2-naphthalen-2-yl-1H-imidazole-4-carboxylic acid (3,5-bis-hydroxymethyl-phenyl)-amide; compound with 6-methylamino-hexane-1,2,3,4,5-pentaol 1358268 5-{[5-Cycloheptylmethyl-2-(1H-indol-5-yl)-1H-imidazole-4-carbonyl]-amino}-isophthalic acid; compound with 6-methylamino-hexane-1,2,3,4,5-pentaol 1358269 5-[(2-Adamantan-1-ylmethyl-5-phenyl-1H-pyrrole-3-carbonyl)-amino]-isophthalic acid; compound with 6-methylamino-hexane-1,2,3,4,5-pentaol 1358270 5-[(2-Cycloheptylmethyl-5-naphthalen-2-yl-1H-pyrrole-3-carbonyl)-amino]-isophthalic acid; compound with 6-methylamino-hexane-1,2,3,4,5-pentaol 1358271 5-[(5-Adamantan-1-ylmethyl-2-phenyl-1H-imidazole-4-carbonyl)-amino]-isophthalic acid; compound with 6-methylamino-hexane-1,2,3,4,5-pentaol 1358272 5-{[(S)-2-({6-[(Adamantan-1-ylmethyl)-carbamoyl]-1H-benzoimidazole-5-carbonyl}-amino)-3-phenyl-propionyl]-methyl-amino}-isophthalic acid; compound with 6-methylamino-hexane-1,2,3,4,5-pentaol 1358273 5-[(S)-2-({6-[(Adamantan-1-ylmethyl)-carbamoyl]-1H-benzoimidazole-5-carbonyl}-amino)-3-phenyl-propionylamino]-isophthalic acid; compound with 6-methylamino-hexane-1,2,3,4,5-pentaol 1358274 3-[(5-Cycloheptylmethyl-2-naphthalen-2-yl-1H-imidazole-4-carbonyl)-amino]-benzoic acid; compound with 6-methylamino-hexane-1,2,3,4,5-pentaol 1358275 5-{[2-(2-Adamantan-1-yl-ethyl)-5-phenyl-1H-pyrrole-3-carbonyl]-amino}-isophthalic acid; compound with 6-methylamino-hexane-1,2,3,4,5-pentaol 1358276 3-[(S)-2-({6-[(Adamantan-1-ylmethyl)-carbamoyl]-1H-benzoimidazole-5-carbonyl}-amino)-3-phenyl-propionylamino]-benzoic acid; compound with 6-methylamino-hexane-1,2,3,4,5-pentaol 1358277 5-((S)-2-{2-[(Adamantan-1-ylmethyl)-carbamoyl]-benzoylamino}-3-phenyl-propionylamino)-isophthalic acid; compound with 6-methylamino-hexane-1,2,3,4,5-pentaol 1358278 5-{[5-(2-Adamantan-1-yl-ethyl)-2-phenyl-1H-imidazole-4-carbonyl]-amino}-isophthalic acid; compound with 6-methylamino-hexane-1,2,3,4,5-pentaol 1358279 5-[(5-Cycloheptylmethyl-2-phenyl-1H-imidazole-4-carbonyl)-amino]-isophthalic acid; compound with 6-methylamino-hexane-1,2,3,4,5-pentaol 1358280 5-[(S)-2-({3-[(Adamantan-1-ylmethyl)-carbamoyl]-naphthalene-2-carbonyl}-amino)-3-phenyl-propionylamino]-isophthalic acid; compound with 6-methylamino-hexane-1,2,3,4,5-pentaol 1358281 5-((S)-2-{[6-(Adamantan-1-ylmethyl-methyl-carbamoyl)-1H-benzoimidazole-5-carbonyl]-amino}-3-phenyl-propionylamino)-isophthalic acid; compound with 6-methylamino-hexane-1,2,3,4,5-pentaol 1358283 1H-Benzoimidazole-5,6-dicarboxylic acid 6-[(adamantan-1-ylmethyl)-amide] 5-{[(S)-1-(3,5-bis-hydroxymethyl-phenylcarbamoyl)-2-phenyl-ethyl]-amide}; compound with 6-methylamino-hexane-1,2,3,4,5-pentaol 1358284 5-[1-[16-(1-adamantylmethylcarbamoyl)tetracyclo[6.6.2.02,7.09,14]hexadeca-2,4,6,9,11,13-hexaen-15-ylcarboxamido]-2-phenyl-(1S)-ethylcarboxamido]isophtalic acid 1358285 3-[(2-Cycloheptylmethyl-5-naphthalen-2-yl-1H-pyrrole-3-carbonyl)-amino]-benzoic acid; compound with 6-methylamino-hexane-1,2,3,4,5-pentaol 1363775 5-Methoxy-2-propyl-2,3,4,4a,9,9a-hexahydro-1H-indeno[2,1-c]pyridine 1363776 8-[4-(5-Methoxy-1,3,4,4a,9,9a-hexahydro-indeno[2,1-c]pyridin-2-yl)-butyl]-8-aza-spiro[4.5]decane-7,9-dione 1363777 8-[3-(5-Methoxy-1,3,4,4a,9,9a-hexahydro-indeno[2,1-c]pyridin-2-yl)-propyl]-8-aza-spiro[4.5]decane-7,9-dione 1363807 4,5-dihydroxy-6-[10-hydroxy-4-methyl-(5R,13R,14S,17R)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10,15-tetraen-14-yloxy]tetrahydro-2H-2-pyrancarboxylic acid 1363827 8-[3-(5-Methoxy-1,3,4,4a,9,9a-hexahydro-indeno[2,1-c]pyridin-2-yl)-propyl]-8-aza-spiro[4.5]decane-7,9-dione 1363828 5-Methoxy-2-propyl-2,3,4,4a,9,9a-hexahydro-1H-indeno[2,1-c]pyridine 1363829 8-[4-(5-Methoxy-1,3,4,4a,9,9a-hexahydro-indeno[2,1-c]pyridin-2-yl)-butyl]-8-aza-spiro[4.5]decane-7,9-dione 1363830 (alpha R,beta R)(2-Chloro-4-{2-[2-hydroxy-2-(4-hydroxy-phenyl)-1-methyl-ethylamino]-ethyl}-phenoxy)-acetic acid 1363890 2-hydroxymethyl-6-[10-hydroxy-4-methyl-(5R,13R,14S,17R)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10,15-tetraen-14-yloxy]tetrahydro-2H-3,4,5-pyrantriol 1367924 (S)-1,1-dimethyl-2-((2S,5S)-2-methyl-3lambda*4*-[1,3]oxathiolan-5-yl)-pyrrolidinium iodide 1367925 (2S,2'R,3'S,5'R)-1-methyl-2-(2-methyl-1,3-oxathiolan-5-yl)pyrrolidine 3-sulfoxide methyl iodide 1367926 (+)-(2S,2'S,3'S,5'S)-1-methyl-2-(2-methyl-1,3-oxathiolan-5-yl)pyrrolidine 3-oxide 1368009 (R)-1,1-dimethyl-2-((2R,5R)-2-methyl-3lambda*4*-[1,3]oxathiolan-5-yl)-pyrrolidinium iodide 1368057 (R)-4-Chloro-N-[5-(2-fluoro-phenyl)-1-methyl-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl]-benzamide 1368115 3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-2,6-dihydro-3H-imidazo[1,2-c]quinazolin-5-one 1368116 3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-5-methylsulfanyl-2,3,5,6-tetrahydro-imidazo[1,2-c]quinazoline 1368157 2-hydroxymethyl-6-[10-hydroxy-4-methyl-(5R,13R,14S,17R)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10,15-tetraen-14-yloxy]tetrahydro-2H-3,4,5-pyrantriol 1368162 (R-PIA)2-(4-Iodo-phenyl)-1-methyl-ethylamine 1368248 1-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-{3-[methyl-(1H-tetrazol-5-yl)-amino]-phenyl}-urea 1368269 (2-Iodo-phenyl)-[1-(1-methyl-piperidin-2-ylmethyl)-1H-indol-3-yl]-methanone 1368271 (S)-2-((2S,3R,5S)-3-hydroxy-2-methyl-3lambda*4*-[1,3]oxathiolan-5-yl)-1,1-dimethyl-pyrrolidinium iodide 1368273 (S)-2-((2R,3R,5R)-3-hydroxy-2-methyl-3lambda*4*-[1,3]oxathiolan-5-yl)-1,1-dimethyl-pyrrolidinium iodide 1368276 2-(1H-Indol-3-yl)-1-methyl-ethylamine 1368277 2-(5-Methoxy-1H-indol-3-yl)-1-methyl-ethylamine 1368333 3-Butyl-1,2,3,4,4a,5,6,10b-octahydro-benzo[f]isoquinoline hydrochloride 1368358 Biphenyl-2-carboxylic acid [3-chloro-4-((S)-3,4,11,11a-tetrahydro-1H,5H-2-oxa-4a,10-diaza-dibenzo[a,d]cycloheptene-10-carbonyl)-phenyl]-amide hydrochloride 1368548 2-{6-[2-(3,5-Dimethoxy-phenyl)-2-o-tolyl-ethylamino]-purin-9-yl}-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1369679 1-{(1R,2S)-2-[3-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-(3-methoxy-phenyl)-urea 1369680 1-(3-Cyano-phenyl)-3-{(1R,2S)-2-[3-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-urea 1369694 Tyr-Cys-Arg-Phe-Phe-Asn-Ala-Phe-Cys-Tyr 1369695 4S,10aS4-Methyl-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole 1369726 Ac-Nle-c[Asp-His-DNal(2')-Pro-Trp-Lys]-NH2 1369733 (R)N-(1-Benzyl-pyrrolidin-2-ylmethyl)-3-bromo-2-hydroxy-6-methoxy-benzamide 1369739 (Z)-7-(3-Hex-2-enylsulfanylmethyl-7-oxa-bicyclo[2.2.1]hept-2-yl)-hept-5-enoic acid 1369743 H-Tyr-Val-Nle-Gly-His-D-Phe-Arg-D-Trp-Asp-Arg-Phe-Gly-NH2 1369747 1-{(1R,2S)-2-[3-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-(3-methoxy-phenyl)-urea 1369748 1-(3-Cyano-phenyl)-3-{(1R,2S)-2-[3-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-urea 1369750 2-(4-Benzyloxy-benzylamino)-N-[3-(2-pyrrolidin-1-yl-ethyl)-3H-benzoimidazol-5-yl]-acetamide 1369762 1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benzoimidazole-5-sulfonic acid 4-fluoro-benzylamide 1369772 N-({[1-(4-Chloro-benzyl)-pyrrolidin-2-ylmethyl]-carbamoyl}-methyl)-3-trifluoromethyl-benzamide 1369773 N-{[(S)-1-(4-Chloro-benzyl)-pyrrolidin-3-ylcarbamoyl]-methyl}-3-trifluoromethyl-benzamide 1369782 (2R,3R,4S,5R)-2-{6-Amino-2-[(S)-1-hydroxymethyl-2-(4-methoxy-phenyl)-ethylamino]-purin-9-yl}-5-(2-ethyl-2H-tetrazol-5-yl)-tetrahydro-furan-3,4-diol 1369792 3-[4-({4-[3-(2-Fluoro-5-trifluoromethyl-phenyl)-ureido]-phenyl}-methyl-amino)-pyrimidin-2-ylamino]-benzenesulfonamide 1369793 4R,10aS4-Methyl-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole 1369821 4-phenyl-8-(2-phenyl-cyclohexyl)-2,8-diaza-spiro[4.5]decan-1-one 1369823 1-((5-(7-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-m-tolylurea 1369824 (1R,2R)-N-[2,3-bis(4-chlorophenyl)-1-methylpropyl]-2-(4-chlorophenyloxy)-2-methylpropanamide 1369825 N-[(1R,2R)-3-(4-chlorophenyl)-1-methyl-2-phenylpropyl]-2-(5-chloropyridyloxy)-2-methylpropanamide 1369834 (R)-2-furan-2-yl-5-(hexahydro-pyrrolo[1,2-a]pyrazin-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 1369835 (S)-2-furan-2-yl-7-(hexahydro-pyrrolo[1,2-a]pyrazin-2-yl)-[1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine 1369864 N-(2,6-dimethylphenyl)-6-(4-fluorophenyl)imidazo-[1,5-a]pyrazin-8-amine 1369867 {2-(hydroxymethyl)-5-[5-methyl-3-(2-methylpropyl)hexylidene]-4-oxo-1,3-dioxolan-2-yl}methyl 2,2-dimethylpropanoate 1369868 (2-(hydroxymethyl)-4-(3-methylbutylidene)-5-oxo-tetrahydrofuran-2-yl)methyl 3-isobutyl-5-methylhexanoate 1369873 (R)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-N-methyl-N-((R)-1-(tetrahydro-2H-pyran-4-yl)pyrrolidin-3-yl)pyrrolidine-1-carboxamide 1377956 TAK-652 1378043 azaline B 1382602 N-[5-(4-Chloro-phenyl)-1H-pyrazol-3-yl]-2-naphthalen-2-yl-acetamide 1382639 3,17,17,18,18-pentamethyl-13,16-dioxa-3-azaheptacyclo[13.5.2.12,8.01,6.06,14.07,12.015,19]tricosa-7,9,11-trien-11-ol 1382641 1-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-[4-methyl-3-(1H-tetrazol-5-ylamino)-phenyl]-urea 1382642 1-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-{3-[(1H-tetrazol-5-ylamino)-methyl]-phenyl}-urea 1382669 2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-N-methyl-N-[(R)-1-(3-phenyl-propylcarbamoyl)-ethyl]-propionamide 1382755 3,17,17,18,18-pentamethyl-13,16-dioxa-3-azaheptacyclo[13.5.2.12,8.01,6.06,14.07,12.015,19]tricosa-7,9,11-trien-11-ol 1382777 2-Amino-3-(4-benzyloxy-2,6-dimethyl-phenyl)-N-[(R)-1-(3-phenyl-propylcarbamoyl)-ethyl]-propionamide 1382800 N-(4-(2-(diethylamino)ethoxy)-3-methoxyphenyl)-N-methyl-4-(trifluoromethyl)benzamide 1382806 Quinoline-4-carboxylic acid {4-[2-(6-cyano-3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-cyclohexyl}-amide HCl (SB-277011) 1383498 sunepitron 1383775 (5E)-5-[(3aS,4S,5R,6aS)-5-hydroxy-4-((E)-{[(phenylamino)carbonyl]hydrazono}methyl)hexahydropentalen-2(1H)-ylidene]pentanoic acid 1383780 (-) 1,2,3,4,5,11-Hexahydro-6-(2-hydroxy)phenyl-3-methyl-2,6-methano-6H-azocino[4,5-b]indole 1383781 (-) 3(1,2,3,4,5,11-Hexahydro-3-methyl-2,6-methano-9-methoxy-6H-azocino[4,5-b]indol-6-yl)phenol methanesulfonate 1383872 11-(2-Octahydro-quinolizin-1-yl-acetyl)-5,11-dihydro-benzo[e]pyrido[3,2-b][1,4]diazepin-6-one 1383906 2-Methyl-6-phenyl-4-phenylethynyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid diethyl ester 1383932 2-Amino-3-(4-hydroxy-phenyl)-N-{1-[4-(3-hydroxy-phenyl)-3,4-dimethyl-piperidin-1-ylmethyl]-2-methyl-propyl}-propionamide 1383935 5-(3-Hydroxy-phenyl)-2-methyl-8-[1-phenyl-meth-(E)-ylidene]-2-aza-bicyclo[3.3.1]nonan-7-one 1383936 8-[1-(3,4-Dichloro-phenyl)-meth-(E)-ylidene]-5-(3-hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]nonan-7-one 1383937 5-(3-Methoxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]nonan-7-one 1383969 3-Phenyl-2-(1-phenyl-6-propoxy-1H-pyrazolo[3,4-d]pyrimidin-4-ylamino)-propan-1-ol 1384033 (S)-(+)9-(4-Methyl-piperazin-1-yl)-9,10-dihydro-4-thia-10a-aza-benzo[f]azulene(ST1622) 1384034 (R)-(-)7-Fluoro-9-(4-methyl-piperazin-1-yl)-9,10-dihydro-4-thia-10a-aza-benzo[f]azulene 1384035 4-{4-(4-Fluoro-phenyl)-5-[2-((S)-1-phenyl-ethylamino)-pyridin-4-yl]-thiazol-2-yl}-1-methyl-piperidin-4-ol 1384040 (R)-11-(4-tert-Butoxy-benzyl)-5-(1H-indol-3-ylmethyl)-17-isopropyl-hexadecahydro-3a,6,9,12,15,18,21-heptaaza-cyclopentacyclohenicosene-4,7,10,13,16,19,22-heptaone 1384058 Ac-c[Cys-Glu-His-D-Nal(2')-Arg-Trp-Cys]-Pro-Pro-Lys-Asp-NH2 1384059 Ac-c[Cys-Glu-His-D-Phe-Arg-Trp-D-Cys]-Pro-Pro-Lys-Asp-NH2 1384184 (4R,7S,10R)-10-[((S)-2-Amino-6-hydroxy-1,2,3,4-tetrahydro-naphthalene-2-carbonyl)-amino]-7-benzyl-3,3-dimethyl-6,9-dioxo-1,2-dithia-5,8-diaza-cycloundecane-4-carboxylic acid 1384185 (4R,7S,10R)-7-Benzyl-10-{[(2S,3R)-3-(4-hydroxy-phenyl)-pyrrolidine-2-carbonyl]-amino}-3,3-dimethyl-6,9-dioxo-1,2-dithia-5,8-diaza-cycloundecane-4-carboxylic acid 1384186 (4R,7S,10R)-7-Benzyl-10-{[(2S,3S)-3-(4-hydroxy-phenyl)-pyrrolidine-2-carbonyl]-amino}-3,3-dimethyl-6,9-dioxo-1,2-dithia-5,8-diaza-cycloundecane-4-carboxylic acid 1384187 (4R,7S,10R)-10-[((R)-2-Amino-5-hydroxy-indane-2-carbonyl)-amino]-7-benzyl-3,3-dimethyl-6,9-dioxo-1,2-dithia-5,8-diaza-cycloundecane-4-carboxylic acid 1384258 Phosphoric acid mono-[(1R,5S)-4-(2-hex-1-enyl-6-methylamino-purin-9-yl)-1-phosphonooxymethyl-bicyclo[3.1.0]hex-2-yl] ester 1384259 H-Tyr-DVal-Met-Gly-His-Phe-Arg-Trp-Asp-Arg-Phe-Gly-OH 1384300 1-(3-Acetyl-phenyl)-3-{2-[4-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-urea 1384301 1-{2-[4-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-(3-methoxy-phenyl)-urea 1384304 (3S)-8-(2,6-dimethoxyphenyl)-N,N-dimethyl-3,4-dihydro-2H-1-benzopyran-3-amine 1384306 4R,10aR4-Methyl-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole 1384316 (Z)-1-[10-(4-Amino-2-methyl-8,8a-dihydro-quinolinium-1-yl)-dec-5-enyl]-2-methyl-quinolin-4-ylamine;diiodide 1384329 TCMDC-139191 1384346 1-(6-Amino-purin-9-yl)-4-hydroxymethyl-bicyclo[3.1.0]hexane-2,3-diol 1384406 1N-methyl-4-[2-chloro-6-(3-fluorobenzylamino)-9H-9-purinyl]-2,3-dihydroxy-(1S,2R,3S,4R,5S)-bicyclo[3.1.0]hexane-1-carboxamide 1384407 1N-methyl-4-[2-chloro-6-(2,5-dichlorobenzylamino)-9H-9-purinyl]-2,3-dihydroxy-(1S,2R,3S,4R,5S)-bicyclo[3.1.0]hexane-1-carboxamide 1384408 (1S,2R,3S,4R,5S)-4-(6-(2,5-dimethoxybenzylamino)-2-chloro-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 1384409 1N-methyl-4-[2-chloro-6-(2-methylbenzylamino)-9H-9-purinyl]-2,3-dihydroxy-(1S,2R,3S,4R,5S)-bicyclo[3.1.0]hexane-1-carboxamide 1384410 (1S,2R,3S,4R,5S)-4-{2-chloro-6-[(pyridin-3-ylmethyl)amino]-9H-purin-9-yl}-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 1384411 1N-methyl-4-[2-chloro-6-(3-methylbenzylamino)-9H-9-purinyl]-2,3-dihydroxy-(1S,2R,3S,4R,5S)-bicyclo[3.1.0]hexane-1-carboxamide 1384412 (1S,2R,3S,4R,5S)-4-(6-(3-chlorobenzylamino)-2-(methylthio)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 1384413 (1S,2R,3S,4R,5S)-4-(6-(3-(3-hydroxyprop-1-ynyl)benzylamino)-2-chloro-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 1384414 (1S,2R,3S,4R,5S)-4-(2-chloro-6-(2-phenylcyclopropylamino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 1384415 1N-methyl-4-[6-(4-aminobenzylamino)-2-chloro-9H-9-purinyl]-2,3-dihydroxy-(1S,2R,3S,4R,5S)-bicyclo[3.1.0]hexane-1-carboxamide 1384426 1N-methyl-4-(2-amino-6-methylamino-9H-9-purinyl)-2,3-dihydroxy-(1S,2R,3S,4R,5S)-bicyclo[3.1.0]hexane-1-carboxamide 1384428 (1S,2R,3S,4R,5S)-4-(6-(cyclopentylamino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 1384429 (1S,2R,3S,4R,5S)-4-(6-(bicyclo[2.2.1]heptan-7-ylamino)-2-chloro-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 1384433 (3R,4S,5R)-2-(6-{[(2S,4S)-bicyclo[2.2.1]heptan-2-yl]amino}-9H-purin-9-yl)-5-(hydroxymethyl)oxolane-3,4-diol 1384434 (3R,4S,5R)-2-(6-{[(1R,4S)-bicyclo[2.2.1]heptan-2-yl]amino}-9H-purin-9-yl)-5-(hydroxymethyl)oxolane-3,4-diol 1384435 (3R,4S,5R)-2-(6-{[(1S,2R,4R)-bicyclo[2.2.1]heptan-2-yl]amino}-9H-purin-9-yl)-5-(hydroxymethyl)oxolane-3,4-diol 1384469 6-(2-Fluoro-benzenesulfonylamino)-2-methyl-hexanoic acid ((S)-7-fluoro-3a,4,5,9b-tetrahydro-1H-benzo[e]indol-2-yl)-amide 1384470 1-(3-chloro-4-[4-(10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5-yl)semicarbazido]benzenesulfonyl)-1H-pyrrole-2-carboxylic acid{2-[(3-dimethylaminopropyl)methylamino]ethyl}amide 1384471 1-(4-[4-(10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5-yl)thiosemicarbazido]-3-nitrobenzenesulfonyl]1H-pyrrole-2-carboxylic acid{2-[(3-dimethylaminopropyl)methylamino]ethyl}amide 1384472 1-(4-[4-(10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5-yl)thiosemicarbazido]-3-nitrobenzenesulfonyl]1H-pyrrole-2-carboxylic acid{2-[(2-dimethylaminoethyl)methylamino]ethyl}amide 1384473 1'N-[1-(5-amino-1-carbamoylpentylcarbamoyl)-2-(1H-3-indolyl)-(1S)-ethyl]spiro[1H-indene-1,4'-(hexahydropyridine)]-1'-carboxamide 1384474 1'N-[1-(5-aminopentylcarbamoyl)-2-(1H-3-indolyl)-(1S)-ethyl]spiro[1H-indene-1,4'-(hexahydropyridine)]-1'-carboxamide 1384534 (S)-1-(4-[4-(10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5-yl)thiosemicarbazido]-3-nitrobenzenesulfonyl]pyrrolidine-2-carboxylic acid{2-[(3-dimethylaminopropyl)methylamino]ethyl}amide 1384567 4,5-dihydroxy-6-[10-hydroxy-4-methyl-(5R,13R,14S,17R)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10,15-tetraen-14-yloxy]tetrahydro-2H-2-pyrancarboxylic acid 1384573 3-[Methyl-(4''-trifluoromethyl-biphenyl-4-carbonyl)-amino]-pyrrolidine-1-carboxylic acid [1-(4,4-dimethyl-cyclohexyl)-pyrrolidin-3-yl]-methyl-amide 1384588 2-(6-Amino-2-phenethylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1384592 4-{2-[1-(4-isopropylcyclohexyl)-2'-phenylspiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole]-5-yl]ethyl}-1,4-oxazinane 1384593 5'-butyl-1-(4-isopropylcyclohexyl)-2'-phenylspiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole] 1384594 5'-benzyl-1-(4-isopropylcyclohexyl)-2'-phenylspiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole] 1384595 1-(4-isopropylcyclohexyl)-2'-phenylspiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole] 1384596 1-(4-isopropylcyclohexyl)-5'-methyl-2'-phenylspiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole] 1384597 4-[5'-cyclopropylmethyl-1-(4-isopropylcyclohexyl)spiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole]-2-yl]phenyl fluoride 1384598 1-(4-isopropylcyclohexyl)-2',5'-diphenylspiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole] 1384599 2-[1-(4-isopropylcyclohexyl)-2'-phenylspiro[hexahydropyridine-4,1'-perhydropyrrolo[3,4-c]pyrrole]-5-yl]-1-ethanol 1384617 3-[2-Methoxy-5-(5-trifluoromethyl-tetrazol-1-yl)-phenyl]-6-phenyl-1-oxa-7-aza-spiro[4.5]dec-3-ene 1384618 3,6-Diphenyl-1-oxa-7-aza-spiro[4.5]decane 1384619 3-(2-Methoxy-5-trifluoromethoxy-phenyl)-6-phenyl-1-oxa-7-aza-spiro[4.5]decane 1384662 2,6-Dimethyl-4-((E)-styryl)-1,4-dihydro-pyridine-3,5-dicarboxylic acid 3-ethyl ester 5-methyl ester 1384687 2-Methyl-6-phenyl-4-styryl-1,4-dihydro-pyridine-3,5-dicarboxylic acid diethyl ester 1384723 2-Acetyl-7-hydroxy-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid {1-[4-(3-hydroxy-phenyl)-3,4-dimethyl-piperidin-1-ylmethyl]-2-methyl-propyl}-amide 1384724 3-({1-[4-(3-Hydroxy-phenyl)-3,4-dimethyl-piperidin-1-ylmethyl]-2-methyl-propylamino}-methyl)-1,2,3,4-tetrahydro-isoquinolin-7-ol 1384725 2-(2-Dimethylamino-acetyl)-7-hydroxy-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid {1-[4-(3-hydroxy-phenyl)-3,4-dimethyl-piperidin-1-ylmethyl]-2-methyl-propyl}-amide 1384726 7-Hydroxy-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid {1-[4-(3-hydroxy-phenyl)-3,4-dimethyl-piperidin-1-ylmethyl]-2-methyl-propyl}-amide 1384734 2-Cyclohexyl-6-methyl-4-phenylethynyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid 3-benzyl ester 5-ethyl ester 1384735 2-Cyclopentyl-6-methyl-4-phenylethynyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid 3-benzyl ester 5-ethyl ester 1384736 2-Cyclobutyl-6-methyl-4-phenylethynyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid 3-benzyl ester 5-ethyl ester 1384737 2-Cyclopropyl-6-methyl-4-phenylethynyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid 3-benzyl ester 5-ethyl ester 1384751 1-Phenyl-2-(1-phenyl-6-propoxy-1H-pyrazolo[3,4-d]pyrimidin-4-ylamino)-propan-1-ol 1384758 1-Phenyl-2-(1-phenyl-6-propoxy-1H-pyrazolo[3,4-d]pyrimidin-4-ylamino)-propan-1-ol 1384759 (S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-bicyclo[3.2.1]octane-6-carboxylic acid methyl ester 1384760 (S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-bicyclo[3.2.1]octane-6-carboxylic acid ethyl ester 1384761 (S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-bicyclo[3.2.1]octane-6-carboxylic acid isopropyl ester 1384762 (S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-bicyclo[3.2.1]octane-6-carboxylic acid benzyl ester 1384763 (S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-bicyclo[3.2.1]octane-6-carboxylic acid isobutyl ester 1384764 (S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-bicyclo[3.2.1]octane-6-carboxylic acid phenyl ester 1384765 (S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-bicyclo[3.2.1]octane-6-carboxylic acid phenethyl ester 1384766 (S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-bicyclo[3.2.1]octane-6-sulfonic acid methyl ester 1384767 (S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-aza-bicyclo[3.2.1]octane-6-carboxylic acid phenyl ester 1384815 (2R,3R,4S,5R)-2-{6-[(S)-2-(Benzothiazol-2-ylsulfanyl)-1-methyl-ethylamino]-2-chloro-purin-9-yl}-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1384819 Naltrindole analogue 1384821 Naltrindole analogue 1384824 Naltrindole analogue 1384828 Naltrindole analogue 1384829 Naltrindole analogue 1384843 (R)-11-(4-tert-Butoxy-benzyl)-5-(1H-indol-3-ylmethyl)-17-isopropyl-hexadecahydro-3a,6,9,12,15,18,21-heptaaza-cyclopentacyclohenicosene-4,7,10,13,16,19,22-heptaone 1384854 Ac-c[D-Cys-Glu-His-D-Nal(2')-Arg-Trp-Cys]-Pro-Pro-Lys-Asp-NH2 1384855 Ac-c[D-Cys-Glu-His-D-Phe-Arg-Trp-Cys]-Pro-Pro-Lys-Asp-NH2 1384856 (9-Benzyl-3,9-diaza-bicyclo[3.3.1]non-3-yl)-(2,3-dimethoxy-phenyl)-methanone 1384858 (2,3-Dimethoxy-phenyl)-[9-(4-fluoro-benzyl)-3,9-diaza-bicyclo[3.3.1]non-3-yl]-methanone 1384859 (5-Bromo-2,3-dimethoxy-phenyl)-[9-(4-fluoro-benzyl)-3,9-diaza-bicyclo[3.3.1]non-3-yl]-methanone 1384886 N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[2-(2-{2-[2-carboxyamino-3-(4-sulfo-phenyl)-propionylamino]-cyclohexyl}-acetylamino)-3-(1H-indol-3-yl)-propionylamino]-4-methylsulfanyl-butyrylamino}-succinamic acid 1384911 1-[4-(2-Ethynyl-phenyl)-piperazin-1-yl]-2-[8-(4-methyl-piperazin-1-yl)-naphthalen-2-yloxy]-ethanone 1384912 2-[8-(4-Methyl-piperazin-1-yl)-naphthalen-2-yloxy]-1-(4-naphthalen-2-yl-piperazin-1-yl)-ethanone 1384913 1-[4-(2,6-Dimethyl-phenyl)-piperazin-1-yl]-2-[8-(4-methyl-piperazin-1-yl)-naphthalen-2-yloxy]-ethanone 1384923 3-Methanesulfonyl-4-oxo-4,5,6,7-tetrahydro-benzo[c]thiophene-1-carboxylic acid ethyl ester 1384947 1-(5-Fluoro-benzo[b]thiophen-3-yl)-3-[4-(2-methyl-quinolin-8-yl)-piperazin-1-yl]-propan-1-ol 1384962 2-[(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-amino]-5-(2-methoxy-phenoxy)-cyclopentanol 1384964 2-[(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-amino]-5-(2,6-dimethoxy-phenoxy)-cyclopentanol 1385048 2-hydroxymethyl-6-[10-hydroxy-4-methyl-(5R,13R,14S,17R)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10-trien-14-yloxy]tetrahydro-2H-3,4,5-pyrantriol 1385056 9-(1-Phenyl-ethyl)-2-pyridin-4-yl-9H-1,3,9-triaza-fluoren-4-ylamine (APPPI) 1385057 3-[5,6-Dimethyl-7-(1-phenyl-ethyl)-2-pyridin-4-yl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino]-acrylic acid methyl ester 1385077 N*1*-[5,6-Dimethyl-2-phenyl-7-(1-phenyl-ethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-ethane-1,2-diamine 1385078 Cyclopentyl-[5,6-dimethyl-2-phenyl-7-(1-phenyl-ethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-amine 1385090 3,4,5-trihydroxy-6-[10-hydroxy-4-methyl-(5R,13R,14S,17R)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10-trien-14-yloxy]tetrahydro-2H-2-pyrancarboxylic acid 1385091 6-[4-cyclopropylmethyl-10-hydroxy-(5R,13R,14S,17R)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10,15-tetraen-14-yloxy]-3,4,5-trihydroxytetrahydro-2H-2-pyrancarboxylic acid 1385104 N-(9-Amino-6,7-dimethoxy-1,2,3,4-tetrahydro-acridin-3-ylmethyl)-3-trifluoromethyl-benzamide 1385110 5-Propyl-3,5-dihydro-2H-pyrrolo[2,3-f]indole-1-carboxylic acid (1,6-dihydro-pyridin-3-yl)-amide 1385112 Phosphoric acid mono-[(1R,5S)-4-(6-amino-2-methylsulfanyl-purin-9-yl)-1-phosphonooxymethyl-bicyclo[3.1.0]hex-2-yl] ester 1385114 Phosphoric acid mono-[(1R,5S)-4-(6-methylamino-purin-9-yl)-1-phosphonooxymethyl-bicyclo[3.1.0]hex-2-yl] ester 1385115 Phosphoric acid mono-[(1R,5S)-4-(2-chloro-6-methylamino-purin-9-yl)-1-phosphonooxymethyl-bicyclo[3.1.0]hex-2-yl] ester 1385116 Phosphoric acid mono-[(1R,5S)-4-(6-methylamino-2-methylsulfanyl-purin-9-yl)-1-phosphonooxymethyl-bicyclo[3.1.0]hex-2-yl] ester 1385117 Trans-Phosphoric acid mono-[(1R,5S)-4-(2-hex-1-enyl-6-methylamino-purin-9-yl)-1-phosphonooxymethyl-bicyclo[3.1.0]hex-2-yl] ester 1385118 Phosphoric acid mono-[(1R,5S)-4-(2-methyl-6-methylamino-purin-9-yl)-1-phosphonooxymethyl-bicyclo[3.1.0]hex-2-yl] ester 1385119 Phosphoric acid mono-[(1R,5S)-4-(2-fluoro-6-methylamino-purin-9-yl)-1-phosphonooxymethyl-bicyclo[3.1.0]hex-2-yl] ester 1385120 Phosphoric acid mono-[(1R,5S)-4-(2-hexyl-6-methylamino-purin-9-yl)-1-phosphonooxymethyl-bicyclo[3.1.0]hex-2-yl] ester 1385144 (S)-N-[(S)-7,7-Dimethyl-1-(4-o-tolyl-piperazine-1-sulfonylmethyl)-bicyclo[2.2.1]hept-2-yl]-2-(1,1-dioxo-hexahydro-1lambda*6*-thiopyran-4-ylamino)-4-methanesulfonyl-butyramide 1385145 (S)-2-Diethylamino-N-[(S)-7,7-dimethyl-1-(4-o-tolyl-piperazine-1-sulfonylmethyl)-bicyclo[2.2.1]hept-2-yl]-4-methanesulfonyl-butyramide 1385146 (S)-N-[(S)-7,7-Dimethyl-1-(4-o-tolyl-piperazine-1-sulfonylmethyl)-bicyclo[2.2.1]hept-2-yl]-4-methanesulfonyl-2-(piperidin-4-ylamino)-butyramide 1385147 (S)-2-Dimethylamino-N-[(S)-7,7-dimethyl-1-(4-o-tolyl-piperazine-1-sulfonylmethyl)-bicyclo[2.2.1]hept-2-yl]-4-methanesulfonyl-butyramide 1385148 (S)-N-[(S)-7,7-Dimethyl-1-(4-o-tolyl-piperazine-1-sulfonylmethyl)-bicyclo[2.2.1]hept-2-yl]-4-methanesulfonyl-2-(tetrahydro-pyran-4-ylamino)-butyramide 1385149 (S)-N-[(S)-7,7-Dimethyl-1-(4-o-tolyl-piperazine-1-sulfonylmethyl)-bicyclo[2.2.1]hept-2-yl]-4-methanesulfonyl-2-methylamino-butyramide 1385150 1-(((7,7-Dimethyl-2(s)-(2-(s)-amino-4-(carboxamide)-butyramido)bicyclo[2.2.1]heptan-1(S)-yl)methyl)sulfonyl)-4-(indan-1yl)piperidine 1385151 (S)-2-Cyclohexylamino-N-[(S)-7,7-dimethyl-1-(4-o-tolyl-piperazine-1-sulfonylmethyl)-bicyclo[2.2.1]hept-2-yl]-4-methanesulfonyl-butyramide 1385152 (S)-2-(Bis-hydroxymethyl-amino)-N-[(S)-7,7-dimethyl-1-(4-o-tolyl-piperazine-1-sulfonylmethyl)-bicyclo[2.2.1]hept-2-yl]-4-methanesulfonyl-butyramide 1385153 1-(((7,7-Dimethyl-2(s)-(2-(s)-amino-4-(methylsulfonyl)-butyramido)bicyclo[2.2.1]heptan-1(S)-yl)methyl)sulfonyl)-4-(indan-1yl)piperidine 1385154 (2S)-2-amino-N-((2S)-7,7-dimethyl-1-((4-o-tolylpiperazin-1-ylsulfonyl)methyl)bicyclo[2.2.1]heptan-2-yl)-4-(methylsulfonyl)butanamide 1385163 3-[2-(4-Phenyl-3,4-dihydro-2H-pyridin-1-yl)-ethyl]-1H-pyrrolo[2,3-b]pyridine 1385164 3-[2-(4-Styryl-3,4-dihydro-2H-pyridin-1-yl)-ethyl]-1H-pyrrolo[2,3-b]pyridine 1385173 (2S,5R,8R)-5,8-Dibenzyl-12-([1,4']bipiperidinyl-1'-carbonyl)-2-(1H-indol-3-ylmethyl)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 1385174 (2S,5R,8R,12S)-5,8-Dibenzyl-2-(1H-indol-3-ylmethyl)-12-(2-morpholin-4-yl-2-oxo-ethyl)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 1385175 2-[(2S,5R,8R,12S)-5,8-Dibenzyl-2-(1H-indol-3-ylmethyl)-3,6,11,14-tetraoxo-1,4,7,10tetraaza-cyclotetradec-12-yl]-N-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-acetamide 1385176 (2S,5R,8R)-5,8-Dibenzyl-2-(1H-indol-3-ylmethyl)-12-(morpholine-4-carbonyl)-1,4,7,10tetraaza-cyclotetradecane-3,6,11,14-tetraone 1385177 (2S,5R,8R)-5,8-Dibenzyl-2-(1H-indol-3-ylmethyl)-3,6,11,14-tetraoxo-1,4,7,10tetraaza-cyclotetradecane-12-carboxylic acid (2-hydroxy-1-hydroxymethyl-ethyl)-amide 1385182 3-Ethyl-10-oxo-1-propyl-10H-9-oxa-4-aza-phenanthrene-2-carbothioic acid S-(2,2,2-trifluoro-ethyl) ester 1385185 2-[8-(3-Amino-propyl)-6-phenethyl-imidazo[1,2-a]pyrazin-2-yl]-N-[2-(1H-indol-3-yl)-ethyl]-isobutyramide 1385186 3-[6-(1H-Indol-3-ylmethyl)-2-phenyl-imidazo[1,2-a]pyrazin-8-yl]-propylamine 1385187 8N-[2-amino-(1S,2S)-cyclohexyl]-15-oxo-(9aR,13aR)-11,12,13,15-tetrahydro-10H-benzo[7,8]quinazolino[5,4-ab]phenazine-8-carboxamide 1385199 N-{4-[2-(5-Amino-2-furan-2-yl-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)-ethyl]-phenyl}-hydroxylamine 1385206 N-({2-[(1-Cyclohexylmethyl-piperidin-3-ylmethyl)-carbamoyl]-ethylcarbamoyl}-methyl)-3,3,3-triphenyl-propionamide 1385207 6-(3,3,3-Triphenyl-propionylamino)-hexanoic acid (1-cyclohexylmethyl-piperidin-3-ylmethyl)-amide 1385208 1-[1-(3,3,3-Triphenyl-propionyl)-pyrrolidine-2-carbonyl]-pyrrolidine-2-carboxylic acid (1-cyclohexylmethyl-piperidin-3-ylmethyl)-amide 1385209 1-(3,3,3-Triphenyl-propionyl)-pyrrolidine-2-carboxylic acid {2-[(1-cyclohexylmethyl-piperidin-3-ylmethyl)-carbamoyl]-ethyl}-amide 1385210 N-(2-{2-[(1-Cyclohexylmethyl-piperidin-3-ylmethyl)-carbamoyl]-ethylcarbamoyl}-ethyl)-3,3,3-triphenyl-propionamide 1385212 1-(3,3,3-Triphenyl-propionyl)-pyrrolidine-2-carboxylic acid {[(1-cyclohexylmethyl-piperidin-3-ylmethyl)-carbamoyl]-methyl}-amide 1385213 (4-{2-[4-(6-Butyl-5,7-dioxo-4,5,6,7-tetrahydro-1H-imidazo[4,5-b]pyridin-2-yl)-phenoxy]-acetylamino}-phenyl)-acetic acid 1385219 2-Furan-2-yl-N*5*-methyl-N*5*-[(S)-1-(5-methyl-isoxazol-3-ylmethyl)-pyrrolidin-2-ylmethyl]-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine 1385220 (3R,3aR)-3-{4-[4-(4-Fluoro-phenoxy)-butyl]-piperazin-1-ylmethyl}-7,8-dimethoxy-3,3a,4,5-tetrahydro-isoxazolo[4,3-c]quinoline 1385221 (3R,3aR)-5-Methyl-3-[4-((E)-5-phenyl-pent-4-enyl)-piperazin-1-ylmethyl]-3,3a,4,5-tetrahydro-isoxazolo[4,3-c]quinoline 1385222 (3R,3aR)-7,8-Dimethoxy-3-[4-((Z)-5-phenyl-hex-4-enyl)-piperazin-1-ylmethyl]-3,3a,4,5-tetrahydro-isoxazolo[4,3-c]quinoline 1385223 (3R,3aR)-7-Methoxy-3-[4-(3-naphthalen-2-yl-propyl)-piperazin-1-ylmethyl]-3,3a-dihydro-naphtho[1,2-c]isoxazole 1385224 (3R,3aR)-3-[4-((E)-5-Phenyl-pent-4-enyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-isoxazolo[4,3-c]quinoline-5-carboxylic acid ethylamide 1385226 (R)-3-[4-(5-Phenyl-pent-4-enyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-isoxazolo[4,3-c]quinoline-5-carboxylic acid ethyl ester 1385227 (3R,3aR)-7,8-Dimethoxy-3-[4-(3-naphthalen-2-yl-propyl)-piperazin-1-ylmethyl]-3,3a,4,5-tetrahydro-isoxazolo[4,3-c]quinoline 1385228 (3R,3aR)-7,8-Dimethoxy-5-methyl-3-[4-((Z)-4-methyl-5-phenyl-pent-4-enyl)-piperazin-1-ylmethyl]-3,3a,4,5-tetrahydro-isoxazolo[4,3-c]quinoline 1385229 (3R,3aS)-3-[4-((E)-5-Phenyl-pent-4-enyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-chromeno[4,3-c]isoxazole 1385230 (3R,3aR)-3-[4-((E)-5-Phenyl-pent-4-enyl)-piperazin-1-ylmethyl]-3,3a-dihydro-naphtho[1,2-c]isoxazole 1385232 (3R,3aR)-3-[4-((E)-5-Phenyl-pent-4-enyl)-piperazin-1-ylmethyl]-3,3a,4,5-tetrahydro-isoxazolo[4,3-c]quinoline 1385233 (3R,3aR)-7-Methoxy-3-[4-((E)-5-phenyl-pent-4-enyl)-piperazin-1-ylmethyl]-3,3a-dihydro-naphtho[1,2-c]isoxazole 1385234 (3R,3aR)-7,8-Dimethoxy-3-[4-((E)-5-phenyl-pent-4-enyl)-piperazin-1-ylmethyl]-3,3a,4,5-tetrahydro-isoxazolo[4,3-c]quinoline 1385235 (3R,3aR)-3-[4-(3-Naphthalen-2-yl-propyl)-piperazin-1-ylmethyl]-3,3a,4,5-tetrahydro-isoxazolo[4,3-c]quinoline 1385236 (3R,3aR)-7,8-Dimethoxy-3-[4-((Z)-4-methyl-5-phenyl-pent-4-enyl)-piperazin-1-ylmethyl]-3,3a,4,5-tetrahydro-isoxazolo[4,3-c]quinoline 1385238 1-[(1R,2S)-2-(4-Benzyl-piperidin-1-ylmethyl)-cyclohexyl]-3-(3-methoxy-phenyl)-urea 1385239 1-[2-(3'-Cyano-biphenyl-4-yl)-4-(piperidin-1-ylamino)-butyl]-3-(3,5-dichloro-phenyl)-urea 1385240 1-(3,5-Dichloro-phenyl)-3-{4-[4-(3a,7a-dihydro-1H-indol-4-yl)-phenyl]-1-methyl-piperidin-4-ylmethyl}-urea 1385241 4-[N-Methyl-N''-((2R,3R,4R,5S)-2,3,4,5,6-pentahydroxy-hexyl)-hydrazino]-but-2-enoic acid [4-(4-benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-amide 1385255 1-Cyclohexyl-piperidine-4-carboxylic acid ((R)-1-(4-chloro-benzyl)-2-{4-[2-(cyclopropylmethyl-methanesulfonyl-amino)-phenyl]-piperazin-1-yl}-2-oxo-ethyl)-amide 1385257 1-Methyl-azocane-5-carboxylic acid ((R)-1-(4-chloro-benzyl)-2-{4-[2-(cyclopropylmethyl-methanesulfonyl-amino)-phenyl]-piperazin-1-yl}-2-oxo-ethyl)-amide 1385258 1-Ethyl-azocane-5-carboxylic acid ((R)-1-(4-chloro-benzyl)-2-{4-[2-(cyclopropylmethyl-methanesulfonyl-amino)-phenyl]-piperazin-1-yl}-2-oxo-ethyl)-amide 1385259 1-(3-Methyl-butyl)-piperidine-4-carboxylic acid ((R)-1-(4-chloro-benzyl)-2-{4-[2-(cyclopropylmethyl-methanesulfonyl-amino)-phenyl]-piperazin-1-yl}-2-oxo-ethyl)-amide 1385260 2-(4-Chloro-benzyloxy)-5-(4-chloro-phenyl)-6-(2,4-dichloro-phenyl)-nicotinonitrile 1385263 3-((S)-2-Amino-2-phenyl-ethyl)-1-(2,6-difluoro-benzyl)-5-(3-methoxy-phenyl)-[1,3,5]triazinane-2,4-dione 1385268 6-[3-(4-Chloro-3-fluoro-phenoxy)-prop-1-ynyl]-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-8-ylamine 1385269 2-Furan-2-yl-6-[3-(1-methyl-5-trifluoromethyl-4,5-dihydro-1H-pyrazol-3-yloxy)-prop-1-ynyl]-[1,2,4]triazolo[1,5-a]pyrazin-8-ylamine 1385270 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [(R)-2-(4-{2-[((S)-2-amino-cyclohexylamino)-methyl]-phenyl}-piperazin-1-yl)-1-(4-chloro-benzyl)-2-oxo-ethyl]-amide 1385271 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-[4-(2-{[(morpholin-4-ylmethyl)-amino]-methyl}-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-amide 1385272 6-{1-[2-(3a,7a-Dihydro-1H-indol-4-yloxy)-ethyl]-piperidin-4-yloxy}-4H-benzo[1,4]oxazin-3-one 1385273 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-[4-(2-{[(4-methyl-piperazin-1-ylmethyl)-amino]-methyl}-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-amide 1385274 (R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-[4-(2-{[([1,4]diazepan-1-ylmethyl)-amino]-methyl}-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-amide 1385275 5-[1-(2-Bromo-phenyl)-meth-(E)-ylidene]-3,3a,5,6,7,9a-hexahydro-pyrrolo[1,2-a]purin-(9Z)-ylideneamine 1385276 4-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-2-(4-dimethylamino-phenyl)-but-3-yn-2-ol 1385279 (S)-2-[(R)-2-(4-tert-Butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethylcarbamoyl]-4-methyl-piperazine-1-carboxylic acid tert-butyl ester 1385280 3-[3-(2-Benzyloxy-5-chloro-phenyl)-thiophen-2-yl]-benzenesulfonamide 1385281 3-{8-[2-(3,4-Dihydro-benzo[c][1,2]dioxin-8-yloxy)-ethyl]-8-aza-bicyclo[3.2.1]oct-2-en-3-yl}-1H-indole 1385282 (1R,4S,6S)-2-Aza-bicyclo[2.2.2]octane-6-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide 1385284 1,2-Dihydro-pyridine-4-carboxylic acid (1-{4-[(R)-2-(3-amino-propionylamino)-3-(2,4-dichloro-phenyl)-propionyl]-piperazin-1-yl}-cyclohexylmethyl)-amide 1385286 3-Amino-N-[(R)-1-(2,4-dichloro-benzyl)-2-oxo-2-(4-{1-[(2-thiazol-2-yl-ethylamino)-methyl]-cyclohexyl}-piperazin-1-yl)-ethyl]-propionamide 1385288 (4R,5S)-4-(4-Fluoro-phenyl)-piperidine-3-carboxylic acid {(R)-3-[(R)-6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3,4,5-tetrahydro-pyridazin-4-yl]-1-methyl-propyl}-amide 1385289 (2R,3R)-3-(4-Fluoro-phenyl)-piperidine-4-carboxylic acid {(R)-3-[(R)-6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3,4,5-tetrahydro-pyridazin-4-yl]-1-methyl-propyl}-amide 1385290 (S)-4-(4-Fluoro-phenyl)-pyrrolidine-3-carboxylic acid {(R)-3-[(R)-6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3,4,5-tetrahydro-pyridazin-4-yl]-1-methyl-propyl}-amide 1385291 (R)-4-(4-Fluoro-phenyl)-pyrrolidine-3-carboxylic acid {(R)-3-[(R)-6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3,4,5-tetrahydro-pyridazin-4-yl]-1-methyl-propyl}-amide 1385292 1-[2-[((R)-6-Amino-6,7,8,9-tetrahydro-5H-benzocycloheptene-7-carbonyl)-amino]-3-(4-chloro-phenyl)-propionyl]-4-cyclohexyl-piperidine-4-carboxylic acid tert-butylamide 1385293 (4S,5R)-4-(4-Fluoro-phenyl)-piperidine-3-carboxylic acid {(R)-3-[(R)-6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3,4,5-tetrahydro-pyridazin-4-yl]-1-methyl-propyl}-amide 1385294 (2S,3S)-3-(4-Fluoro-phenyl)-piperidine-4-carboxylic acid {(R)-3-[(R)-6-(4-chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3,4,5-tetrahydro-pyridazin-4-yl]-1-methyl-propyl}-amide 1385296 Bicyclo[2.2.1]hept-2-yl-(2-phenoxy-6,9-dihydro-1H-purin-6-yl)-amine 1385297 N*6*-Bicyclo[2.2.1]hept-2-yl-N*2*-phenyl-6,9-dihydro-1H-purine-2,6-diamine 1385307 3-{3-[4-(2-Chloro-phenyl)-piperazin-1-yl]-propyl}-6-(4-methoxy-phenyl)-1,5-dihydro-pyrrolo[3,2-d]pyrimidine-2,4-dione 1385308 2-[4-(3,4-Dihydro-benzo[c][1,2]dioxin-6-yl)-piperazin-1-ylmethyl]-tetrahydro-imidazo[1,5-a]pyridine-1,3-dione 1385309 (R)-2-[(S)-1-({(S)-1-[(S)-2-Amino-1-hydroxy-3-(4-hydroxy-phenyl)-propyl]-pyrrolidine-2-carbonyl}-amino)-2-phenyl-ethyl]-thiazolidine-4-carboxylic acid amide 1385310 (R)-2-[(R)-1-({(S)-1-[(S)-2-Amino-1-hydroxy-3-(4-hydroxy-phenyl)-propyl]-pyrrolidine-2-carbonyl}-amino)-2-phenyl-ethyl]-thiazolidine-4-carboxylic acid amide 1385311 (R)-2-[(S)-1-({1-[(S)-2-(S)-Amino-1-hydroxy-3-(4-hydroxy-phenyl)-propyl]-pyrrolidine-2-carbonyl}-amino)-2-(1H-indol-3-yl)-ethyl]-thiazolidine-4-carboxylic acid amide 1385312 5-{2-[4-(3a,7a-Dihydro-1H-indol-5-ylmethyl)-piperazin-1-yl]-ethoxy}-2-methyl-quinoline 1385313 K-252a analogue 1385314 K-252a analogue 1385316 K-252a analogue 1385317 N*4*-[2-(2-Chloro-phenoxymethyl)-pyrimidin-4-yl]-N*1*,N*1*-diethyl-pentane-1,4-diamine 1385319 N*4*-[2-(2,4-Dichloro-phenoxymethyl)-pyrimidin-4-yl]-N*1*,N*1*-diethyl-pentane-1,4-diamine 1385320 N*4*-[2-(3,4-Dichloro-phenoxymethyl)-pyrimidin-4-yl]-N*1*,N*1*-diethyl-pentane-1,4-diamine 1385323 N*4*-[2-(4-Chloro-phenoxymethyl)-pyrimidin-4-yl]-N*1*,N*1*-diethyl-pentane-1,4-diamine 1385324 Norbinaltorphimine derivative 1385325 1-(3a,7a-Dihydro-1H-indol-5-yl)-3-{(1R,2S)-2-[(S)-3-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-urea 1385326 N*1*,N*1*-Diethyl-N*4*-[2-(4-fluoro-phenoxymethyl)-pyrimidin-4-yl]-pentane-1,4-diamine 1385327 1-(3a,4-Dihydro-benzothiazol-6-yl)-3-{(1R,2S)-2-[(S)-3-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-urea 1385328 1-(3a,7a-Dihydro-1H-indazol-5-yl)-3-{(1R,2S)-2-[(S)-3-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-urea 1385329 Norbinaltorphimine derivative 1385330 1-(3-Chloro-3a,7a-dihydro-1H-indazol-5-yl)-3-{(1R,2S)-2-[(S)-3-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-urea 1385331 1-{(1R,2S)-2-[(S)-3-(4-Fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-3-(2,3,3a,7a-tetrahydro-1H-indol-5-yl)-urea 1385333 1-(4-Chloro-phenyl)-3-{(1R,2S)-2-[(S)-3-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-urea 1385335 (R)-3-Cyclobutyl-2-{(3S,4S)-3-[4-(5,7-dimethyl-pyrazolo[1,5-a]pyrimidin-3-yl)-piperidin-1-ylmethyl]-4-phenyl-pyrrolidin-1-yl}-propionic acid 1385337 (R)-3-Cyclobutyl-2-[(3S,4S)-3-(4-imidazo[1,2-a]pyridin-3-yl-piperidin-1-ylmethyl)-4-phenyl-pyrrolidin-1-yl]-propionic acid 1385339 (R)-3-Cyclobutyl-2-[(3S,4S)-3-(4-imidazo[1,2-a]pyrazin-3-yl-piperidin-1-ylmethyl)-4-phenyl-pyrrolidin-1-yl]-propionic acid 1385343 4-[6-Amino-5-(4-butoxy-2,6-difluoro-benzoyl)-pyridin-2-ylamino]-benzenesulfonamide 1385344 Dimethyl-[(2R,3aR,12bS)-1-(2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-yl)methyl]-amine 1385345 3-[2-(Pyrazin-2-ylamino)-5-[1,2,4]triazol-1-yl-thiazol-4-yl]-benzonitrile 1385346 3-[5-Imidazol-1-yl-2-(pyrazin-2-ylamino)-thiazol-4-yl]-benzonitrile 1385347 3-[5-(2-Methyl-imidazol-1-yl)-2-(3-methyl-pyridin-2-ylamino)-thiazol-4-yl]-benzonitrile 1385348 1-[5-Methoxy-6-(4-methyl-piperazin-1-yl)-2,3-dihydro-indol-1-yl]-2-(4-nitro-phenyl)-ethanone 1385349 1-[5-Methoxy-6-((3S,5R)-3,4,5-trimethyl-piperazin-1-yl)-2,3-dihydro-indol-1-yl]-2-(4-nitro-phenyl)-ethanone 1385352 (5E,8E,11E,14E)-20-Isothiocyanato-icosa-5,8,11,14-tetraenoic acid cyclopropylamide 1385353 (5E,8E,11E,14E)-20-Azido-icosa-5,8,11,14-tetraenoic acid cyclopropylamide 1385382 N-{1-[3-(4-tert-Butoxyamino-phenyl)-3-(3-fluoro-phenyl)-propyl]-piperidin-4-yl}-N-ethyl-2-(4-methanesulfonyl-phenyl)-acetamide 1385383 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {1-(4-chloro-benzyl)-2-oxo-2-[4-(1,2,3,4-tetrahydro-quinolin-8-yl)-piperazin-1-yl]-ethyl}-amide 1385384 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [2-[4-(1-acetyl-1,2,3,4-tetrahydro-quinolin-8-yl)-piperazin-1-yl]-1-(4-chloro-benzyl)-2-oxo-ethyl]-amide 1385385 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {1-(4-chloro-benzyl)-2-[4-(2,3-dihydro-1H-indol-7-yl)-piperazin-1-yl]-2-oxo-ethyl}-amide 1385386 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {1-(4-chloro-benzyl)-2-[4-(1H-indol-7-yl)-piperazin-1-yl]-2-oxo-ethyl}-amide 1385387 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [2-[4-(2-acetyl-1,2,3,4-tetrahydro-isoquinolin-8-yl)-piperazin-1-yl]-1-(4-chloro-benzyl)-2-oxo-ethyl]-amide 1385388 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {1-(4-chloro-benzyl)-2-[4-(2-methanesulfonyl-1,2,3,4-tetrahydro-isoquinolin-8-yl)-piperazin-1-yl]-2-oxo-ethyl}-amide 1385389 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid (1-(4-chloro-benzyl)-2-oxo-2-{4-[2-(propane-2-sulfonyl)-1,2,3,4-tetrahydro-isoquinolin-8-yl]-piperazin-1-yl}-ethyl)-amide 1385390 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [2-[4-(2-benzenesulfonyl-1,2,3,4-tetrahydro-isoquinolin-8-yl)-piperazin-1-yl]-1-(4-chloro-benzyl)-2-oxo-ethyl]-amide 1385391 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {1-(4-chloro-benzyl)-2-[4-(2-methyl-1,2,3,4-tetrahydro-isoquinolin-8-yl)-piperazin-1-yl]-2-oxo-ethyl}-amide 1385392 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {1-(4-chloro-benzyl)-2-[4-(2-ethyl-1,2,3,4-tetrahydro-isoquinolin-8-yl)-piperazin-1-yl]-2-oxo-ethyl}-amide 1385393 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {1-(4-chloro-benzyl)-2-[4-(2-ethyl-1,2,3,4-tetrahydro-isoquinolin-5-yl)-piperazin-1-yl]-2-oxo-ethyl}-amide 1385394 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {1-(4-chloro-benzyl)-2-[4-(2-methanesulfonyl-1,2,3,4-tetrahydro-isoquinolin-5-yl)-piperazin-1-yl]-2-oxo-ethyl}-amide 1385395 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {1-(4-chloro-benzyl)-2-oxo-2-[4-(5,6,7,8-tetrahydro-naphthalen-1-yl)-piperazin-1-yl]-ethyl}-amide 1385396 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [2-[4-(7-amino-5,6,7,8-tetrahydro-naphthalen-1-yl)-piperazin-1-yl]-1-(4-chloro-benzyl)-2-oxo-ethyl]-amide 1385397 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [2-[4-(7-acetylamino-5,6,7,8-tetrahydro-naphthalen-1-yl)-piperazin-1-yl]-1-(4-chloro-benzyl)-2-oxo-ethyl]-amide 1385398 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid (1-(4-chloro-benzyl)-2-{4-[7-(methanesulfonyl-methyl-amino)-5,6,7,8-tetrahydro-naphthalen-1-yl]-piperazin-1-yl}-2-oxo-ethyl)-amide 1385399 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {1-(4-chloro-benzyl)-2-[4-(7-methylamino-5,6,7,8-tetrahydro-naphthalen-1-yl)-piperazin-1-yl]-2-oxo-ethyl}-amide 1385400 (3R)-N-[3-(4-chlorophenyl)-1-{4-[7-(dimethylamino)-5,6,7,8-tetrahydronaphthalen-1-yl]piperazin-1-yl}-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 1385401 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {1-(4-chloro-benzyl)-2-[4-(7-diethylamino-5,6,7,8-tetrahydro-naphthalen-1-yl)-piperazin-1-yl]-2-oxo-ethyl}-amide 1385402 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {1-(4-chloro-benzyl)-2-[4-(7-dipropylamino-5,6,7,8-tetrahydro-naphthalen-1-yl)-piperazin-1-yl]-2-oxo-ethyl}-amide 1385403 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {1-(4-chloro-benzyl)-2-[4-(7-cyclobutylamino-5,6,7,8-tetrahydro-naphthalen-1-yl)-piperazin-1-yl]-2-oxo-ethyl}-amide 1385404 1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {1-(4-chloro-benzyl)-2-[4-(7-oxiranylamino-5,6,7,8-tetrahydro-naphthalen-1-yl)-piperazin-1-yl]-2-oxo-ethyl}-amide 1385405 (3R)-N-[3-(4-chlorophenyl)-1-{4-[(7S)-7-(dimethylamino)-5,6,7,8-tetrahydronaphthalen-1-yl]piperazin-1-yl}-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 1385406 (3R)-N-[3-(4-chlorophenyl)-1-{4-[(7R)-7-(dimethylamino)-5,6,7,8-tetrahydronaphthalen-1-yl]piperazin-1-yl}-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 1385407 N-(1-{4-[4-Methoxy-2-(4-methoxy-benzenesulfonyl)-benzoyl]-phenyl}-ethyl)-methanesulfonamide 1385408 1-[2-(4-amino-5-chloro-2-hydroxyphenylcarbonyloxy)ethyl]-4-(2-{1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydro-4-pyridinylcarboxamido}ethylcarboxamido)hexahydropyridine 1385409 1-[2-(4-amino-5-chloro-2-hydroxyphenylcarbonyloxy)ethyl]-4-(3-{1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydro-4-pyridinylcarboxamido}propylcarboxamido)hexahydropyridine 1385410 1-[2-(4-amino-5-chloro-2-hydroxyphenylcarbonyloxy)ethyl]-4-(2-{1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)ethyl]hexahydro-4-pyridinylcarboxamido}ethylcarbamoyl)hexahydropyridine 1385411 2-[4-(11-{[4-({10-[(1-{2-[(4-amino-5-chloro-2-methoxyphenyl)carbonyloxy]ethyl}piperidin-4-yl)carbamoyl]decyl}amino)-1,3,5-triazin-2-yl]amino}undecanamido)piperidin-1-yl]ethyl 4-amino-5-chloro-2-methoxybenzoate 1385413 (4-amino-1H-benzoimidazol-2-yl)(4-methylpiperazin-1-yl)methanone 1385414 2-(2-Furylmethoxy)-5-{[6-methoxy-7-(3-pyrrolidin-1-ylpropoxy)quinazolin-4-yl]amino} benzo-1,4-quinone 1385415 2-(2,2-Difluoroethoxy)-5-{[6-methoxy-7-(3-pyrrolidin-1-ylpropoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 1385416 2-(4-Benzylpiperidin-1-yl)-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 1385417 2-chloro-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 1385418 2-(dimethylamino)-5-{[6-methoxy-7-(2-methoxyethoxy)-quinazolin-4-yl]amino}benzo-1,4-quinone 1385419 2-{[-6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-5-morpholin-4-ylbenzo-1,4-quinone 1385420 2-Isopropoxy-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 1385421 2-(4-Benzylpiperazin-1-yl)-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 1385422 3-Chloro-2-[2-fluoro-1-(fluoromethyl)ethoxy]-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 1385423 3-chloro-2-methoxy-5-{[6-methoxy-7-(2-methoxyethoxy)-quinazolin-4-yl]amino}benzo-1,4-quinone 1385424 2-chloro-3-methoxy-6-{[6-methoxy-7-(2-methoxyethoxy)-quinazolin-4-yl]amino}-5-(methylthio)benzo-1,4-quinone 1385425 2-{[-6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-5-phenoxybenzo-1,4-quinone 1385426 2-[2-fluoro-1-(fluoromethyl)ethoxy]-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 1385427 2-{[6-Methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-5-(pyridin-3-ylmethoxy)benzo-1,4-quinone 1385428 N-(4-chlorophenyl)-4-{[2-(4-morpholinyl)ethyl]amino}-N-{2-oxo-2-[2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}benzenesulfonamide 1385429 2-{[6-Methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 1385430 N-(4-chlorophenyl)-4-(3-hydroxypropyl)-N-{2-oxo-2-[2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}benzenesulfonamide 1385431 2-{[6-Methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-5-piperidin-1-ylbenzo-1,4-quinone 1385432 3-{4-[(4-chloro{2-oxo-2-[2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}anilino)sulfonyl]phenyl}-N-(3-hydroxypropyl)propanamide 1385433 2-[(4-Fluorobenzyl)oxy]-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino} benzo-1,4-quinone 1385434 2-Methoxy-6-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 1385435 2-({6-methoxy-7-[(1-methylpiperidin-4-yl)methoxy]-quinazolin-4-yl}amino)-5-{2-[methyl(phenyl)amino]-ethoxy}benzo-1,4-quinone 1385436 N-(4-chlorophenyl)-4-[2-(4-morpholinyl)ethoxy]-N-{2-oxo-2-[2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}benzenesulfonamide 1385437 2-[4-(1H-imidazol-1-yl)phenoxy]-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 1385438 2-(3-Fluorophenoxy)-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 1385439 2-{[6-Methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-5-(2,2,2-trifluoro-1-phenylethoxy)benzo-1,4-quinone 1385440 N-(4-chlorophenyl)-4-[3-(dimethylamino)propoxy]-N-{2-[2-(1,3-dioxo-2,3-dihydro-4(1H)-isoquinolinylidene)hydrazino]-2-oxoethyl}benzenesulfonamide 1385441 2-[(2-Fluorobenzyl)oxy]-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 1385442 2-Chloro-3-(cyclopropylmethoxy)-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 1385443 2-[2-fluoro-1-(fluoromethyl)ethoxy]-3-methoxy-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-benzo-1,4-quinone 1385444 2-[2-fluoro-1-(fluoromethyl)ethoxy]-5-{[6-methoxy-7-(3-pyrrolidin-1-ylpropoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 1385445 4-ethoxy-N-{1-methyl-2-oxo-2-[(2Z)-2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}-N-(4-methylphenyl)-benzene-sulfonamide 1385446 methyl-3-({[4-chloro({4-[3-(dimethylamino)propoxy]phenyl}sulfonyl)anilino]acetyl}hydrazono)-2-oxo-2,3-dihydro-1H-indole-7-carboxylate 1385447 2-[3-({[4-chloro({4-[3-(dimethylamino)propoxy]phenyl}sulfonyl)anilino]acetyl}hydrazono)-2-oxo-2,3-dihydro-1H-indole-1-yl]acetamide 1385448 4-ethoxy-N-{1-(hydroxymethyl)-2-oxo-2-[(2Z)-2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}-N-(4-methylphenyl)benzenesulfonamide 1385449 N-(4-chlorophenyl)-4-ethoxy-N-{2-oxo-2-[(2Z)-2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}benzenesulfonamide 1385450 2-{[6-Methoxy-7-(3-pyrrolidin-1-ylpropoxy)quinazolin-4-yl]amino}-5-(pyridin-2-ylmethoxy)benzo-1,4-quinone 1385451 N-(4-chlorophenyl)-4-[3-(dimethylamino)propoxy]-N-{2-oxo-2-[(2Z)-2-(2-oxo-1,2-dihydro-3H-pyrrolo[3,2-c]pyridin-3-ylidene)hydrazino]ethyl}benzenesulfonamide 1385452 N-(4-chlorophenyl)-4-[3-(dimethylamino)propoxy]-N-{2-oxo-2-[(2Z)-2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}benzenesulfonamide 1385453 N-(4-chlorophenyl)-4-ethoxy-N-{2-oxo-2-[(2Z)-2-(2-oxo-1,2-dihydro-3H-pyrrolo[3,2-c]pyridin-3-ylidene)hydrazino]ethyl}benzenesulfonamide 1385454 N-(4-chlorophenyl)-4-[2-(dimethylamino)ethoxy]-N-{2-oxo-2-[(2Z)-2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}benzenesulfonamide 1385455 N-(4-chlorophenyl)-N-{2-oxo-2-[(2Z)-2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}-2-thiophenesulfonamide 1385456 4-cyano-N-(4-methylphenyl)-N-{2-oxo-2-[2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}benzenesulfonamide 1385457 N-(4-methylphenyl)-N-{2-oxo-2-[2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}-1-naphthalenesulfonamide 1385458 N-(4-chlorophenyl)-N-{2-oxo-2-[(2Z)-2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}benzenesulfonamide 1385459 N-(4-chlorophenyl)-4-[2-(2-methoxyethoxy)ethoxy]-N-{2-oxo-2-[(2Z)-2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}benzenesulfonamide 1385460 N-(4-chlorophenyl)-N-{2-oxo-2-[(2Z)-2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}-4-propoxybenzenesulfonamide 1385461 4-butoxy-N-(4-chlorophenyl)-N-{2-oxo-2-[(2Z)-2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}benzenesulfonamide 1385462 N-(4-chlorophenyl)-4-(2-methoxyethoxy)-N-{2-oxo-2-[(2Z)-2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}benzenesulfonamide 1385463 N-(4-chlorophenyl)-N-{2-oxo-2-[(2Z)-2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}-4-propylbenzenesulfonamide 1385464 4-tert-butyl-N-(4-chlorophenyl)-N-{2-oxo-2-[(2E)-2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}benzenesulfonamide 1385465 N-(4-chlorophenyl)-N-{2-oxo-2-[(2Z)-2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}-4-tert-pentylbenzenesulfonamide 1385466 4-methoxy-N-(4-methylphenyl)-N-{2-oxo-2-[2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}benzenesulfonamide 1385467 N-(4-methylphenyl)-N-{2-oxo-2-[(2Z)-2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}-4-methoxy-benzenesulfonamide 1385469 rac-N-(2-(2,5-dimethylpiperazin-1-yl)-4-methylquinolin-6-yl)-2-(4-(trifluoromethoxy)phenoxy)acetamide 1385471 7-((S)-2-(3-hydroxy-5-phenylpentyl)-5-oxopyrrolidin-1-yl)heptanoic acid 1385472 (2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-(azidomethyl)-tetrahydrothiophene-3,4-diol 1385496 N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-5,6-dichloro-4-oxo-4H-chromene-2-carboxamide 1385497 (R)-8-((S)-sec-butyl)-2-(4-hydroxybicyclo[2.2.2]octan-1-yl)-4-propyl-7,8-dihydro-1H-imidazo[1,2-g]purin-5(4H)-one 1385500 N-[3-(4-chlorophenyl-2-(4-fluorophenyl)-1-methylpropyl]-2-(4-chlorophenyloxy)-2-methylpropanamide 1385501 N-[3-(4-chlorophenyl)-2-(3-fluorophenyl)-1-methylpropyl]-2-(4-chlorophenyloxy)-2-methylpropanamide 1385502 N-[3-(4-chlorophenyl)-2-(2-fluorophenyl)-1-methylpropyl]-2-(4-chlorophenyloxy)-2-methylpropanamide 1385503 N-[3-(2-chlorophenyl)-1-methyl-2-phenylpropyl]-2-(4-chlorophenyloxy)-2-methylpropanamide 1385504 N-[1-methyl-2-phenyl-3-(4-trifluoromethylphenyl)propyl]-2-(4-chlorophenyloxy)-2-methylpropanamide 1385505 N-[1-methyl-2-phenyl-3-(4-fluorophenyl)propyl]-2-(4-chlorophenyloxy)-2-methylpropanamide 1385506 N-[2,3-bis(phenyl)-1-methylpropyl]-2-(4-chlorophenyloxy)-2-methylpropanamide 1385507 N-[3-(4-chlorophenyl)-1-methyl-2-phenylpropyl]-2-(2-chlorophenyloxy)-2-methylpropanamide 1385508 N-3-(4-chlorophenyl)-1-methyl-2-phenyl-propyl]-2-(3-pyridyloxy)-2-methylpropanamide 1385509 N-(4-(4-chlorophenyl)-3-phenylbutan-2-yl)-2-methyl-2-(pyridin-4-yloxy)propanamide 1385511 5-{N'-[(1E)-[3-(hexadecyloxy)-2-methoxyphenyl](piperidin-1-yl)methylidene]hydrazinesulfonyl}benzene-1,3-dicarboxylic acid 1385515 (4S,10bR)-4-isopropyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino[2,1-a]isoindol-6(2H)-one 1385521 6-guanidino-2-(3''-(1''-(p-toluenesulfonyl)indolyl)ethyloxy)adenosine 1385522 6-guanidino-2-(3''-indolylethyloxy)adenosine 1385526 (5alpha)-17-allylllyl-14-hydroxy-6-oxo-4,5-epoxymorphinan-3-yl-17-(cyclobutylmethyl)morphinan-3-yl sebacoylate 1385528 1-[(4-oxo-2-pentyl-4,5,6,7-tetrahydrobenzothiophen-5-yl)ethyl]-4-(6-fluorobenzisoxazol-3-yl)piperidine 1385529 (2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 9-acetoxy-2-(2-bromo-5-methoxy-tetrahydrofuran-3-yl)-6a,10b-dimethyl-4,10-dioxo-dodecahydro-1H-benzo[f]isochromene-7-carboxylate 1385532 17-(cyclopropylmethyl)-7'(3,4-diformylnaphthoylamino)-6,7-didehydro-4,5R-epoxy-14-hydroxyindolo[2',3':6,7]-morphinan 1385533 (1S,5S)-(-)-5-(3-hydroxyphenyl)-9-oxo-2-phenylethyl-2-azabicyclo[3.3.1]nonane 1385534 2-{4-[(2-{N-[3-(4-{3-[N-({[(1-{2-[(4-amino-5-chloro-2-methoxyphenyl)carbonyloxy]ethyl}piperidin-4-yl)methyl]carbamoyl}methyl)-2,2-dimethylpropanamido]prop-1-yn-1-yl}phenyl)prop-2-yn-1-yl]-2,2-dimethylpropanamido}acetamido)methyl]piperidin-1-yl}ethyl 4-amino-5-chloro-2-methoxybenzoate 1385535 2-(4-{4-[N-(3-{3-[3-(N-{3-[(1-{2-[(4-amino-2-methoxyphenyl)carbonyloxy]ethyl}piperidin-4-yl)carbamoyl]propyl}-2,2-dimethylpropanamido)prop-1-yn-1-yl]phenyl}prop-2-yn-1-yl)-2,2-dimethylpropanamido]butanamido}piperidin-1-yl)ethyl 4-amino-5-chloro-2-methoxybenzoate 1385536 2-(4-{4-[N-(3-{4-[3-(N-{3-[(1-{2-[(4-amino-5-chloro-2-methoxyphenyl)carbonyloxy]ethyl}piperidin-4-yl)carbamoyl]propyl}-2,2-dimethylpropanamido)prop-1-yn-1-yl]phenyl}prop-2-yn-1-yl)-2,2-dimethylpropanamido]butanamido}piperidin-1-yl)ethyl 4-amino-5-chloro-2-methoxybenzoate 1385537 2-{4-[(4-{N-[3-(3-{3-[N-(3-{[(1-{2-[(4-amino-2-methoxyphenyl)carbonyloxy]ethyl}piperidin-4-yl)methyl]carbamoyl}propyl)-2,2-dimethylpropanamido]prop-1-yn-1-yl}phenyl)prop-2-yn-1-yl]-2,2-dimethylpropanamido}butanamido)methyl]piperidin-1-yl}ethyl 4-amino-5-chloro-2-methoxybenzoate 1385538 2-{4-[(4-{N-[3-(4-{3-[N-(3-{[(1-{2-[(4-amino-5-chloro-2-methoxyphenyl)carbonyloxy]ethyl}piperidin-4-yl)methyl]carbamoyl}propyl)-2,2-dimethylpropanamido]prop-1-yn-1-yl}phenyl)prop-2-yn-1-yl]-2,2-dimethylpropanamido}butanamido)methyl]piperidin-1-yl}ethyl 4-amino-5-chloro-2-methoxybenzoate 1385539 2-{4-[(2-{N-[3-(4-{3-[N-({[(1-{2-[(4-amino-5-chloro-2-methoxyphenyl)carbonyloxy]ethyl}piperidin-4-yl)methyl]carbamoyl}methyl)-2,2-dimethylpropanamido]propyl}phenyl)propyl]-2,2-dimethylpropanamido}acetamido)methyl]piperidin-1-yl}ethyl 4-amino-5-chloro-2-methoxybenzoate 1385540 2-(4-{4-[N-(3-{4-[3-(N-{3-[(1-{2-[(4-amino-5-chloro-2-methoxyphenyl)carbonyloxy]ethyl}piperidin-4-yl)carbamoyl]propyl}-2,2-dimethylpropanamido)propyl]phenyl}propyl)-2,2-dimethylpropanamido]butanamido}piperidin-1-yl)ethyl 4-amino-5-chloro-2-methoxybenzoate 1385541 2-{4-[(4-{N-[3-(3-{3-[N-(3-{[(1-{2-[(4-amino-5-chloro-2-methoxyphenyl)carbonyloxy]ethyl}piperidin-4-yl)methyl]carbamoyl}propyl)-2,2-dimethylpropanamido]propyl}phenyl)propyl]-2,2-dimethylpropanamido}butanamido)methyl]piperidin-1-yl}ethyl 4-amino-5-chloro-2-methoxybenzoate 1385542 2-(4-(4-(tert-butoxycarbonyl(3-(4-(3-(tert-butoxycarbonyl(4-(cyclohexylamino)-4-oxobutyl)amino)propyl)phenyl)propyl)-amino)butanamido)piperidin-1-yl)ethyl 4-Amino-5-chloro-2-methoxybenzoate 1385543 benzo[b]thiophene-2-carboxylic acid (1-{1-(R)-[3-(3,5-dimethyl-piperazin-1-yl)-propylcarbamoyl]-2-phenyl-ethylcarbamoyl}-cyclopentyl)-amide 1385545 7alpha-[(cinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine 1385546 7alpha-[(2'-methylcinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine 1385547 7alpha-[(2'-chlorocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine 1385548 7alpha-[(4'-Methylcinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine 1385549 7alpha-[(4'-chlorocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine 1385550 7alpha-[(4'-nitrocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine 1385551 3-butoxy-N-(4-(3,4-diethoxyphenyl)-1,2,5-oxadiazol-3-yl)benzamide 1385552 7alpha-[(2'-methoxycinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine 1385553 7alpha-[(4'-methoxycinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine 1385554 7alpha-[(cinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 1385555 7alpha-[(2'-methylcinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 1385556 7alpha-[(2'-chlorocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 1385557 7alpha-[(4'-methylcinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 1385558 7alpha-[(4'-chlorocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 1385559 7alpha-[(4'-nitrocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 1385560 7alpha-[(cinnamyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine 1385561 7alpha-[(4'-chlorocinnamyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine 1385562 7alpha-[(cinnamyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 1385563 7alpha-[(4'-chlorocinnamyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 1385564 1'-(o-methylcinnamoyl)-[7alpha,8alpha:3',4']-pyrrolidino-6,14-endoethenotetrahydrooripavine 1385565 1'-(p-methylcinnamoyl)-[7alpha,8alpha:3',4']-pyrrolidino-6,14-endoethenotetrahydrooripavine 1385581 Dequalinium Analogue 1385582 (E)-1-[10-(4-Amino-2-methyl-8,8a-dihydro-quinolinium-1-yl)-dec-5-enyl]-2-methyl-quinolin-4-ylamine;diiodide 1385583 Dequalinium Analogue 1385584 4-Amino-1-dec-5-enyl-2-methyl-8,8a-dihydro-quinolinium 1385585 4-Amino-1-decyl-2-methyl-8,8a-dihydro-quinolinium iodide 1385586 4-Amino-1,2-dimethyl-8,8a-dihydro-quinolinium iodide 1385589 Dequalinium Analogue 1385592 Dequalinium Analogue 1385598 1H-Indole-2-carboxylic acid {4-[2-(7-cyano-3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-cyclohexyl}-amide 1385599 Naphthalene-2-carboxylic acid {4-[2-(6-cyano-3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-cyclohexyl}-amide 1385600 1H-Indole-2-carboxylic acid {4-[2-(6-cyano-3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-cyclohexyl}-amide 1385601 N-{4-[2-(7-Cyano-3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-cyclohexyl}-3-phenyl-acrylamide 1385602 Naphthalene-1-carboxylic acid {4-[2-(6-cyano-3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-cyclohexyl}-amide 1385603 N-{4-[2-(6-Cyano-3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-cyclohexyl}-3-(3-methanesulfonyl-phenyl)-acrylamide 1385620 salvinicin B 1385637 (R)-2-iodo-N-(3-(pyrrolidin-2-ylmethyl)-1H-indol-5-yl)benzenesulfonamide 1385638 2-(7-Cyclohexylamino-imidazo[4,5-b]pyridin-3-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385639 5-Hydroxymethyl-3-methyl-2-[6-((R)-1-methyl-2-phenyl-ethylamino)-purin-9-yl]-tetrahydro-furan-3,4-diol 1385640 2-(7-Cyclopentylamino-imidazo[4,5-b]pyridin-3-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385641 2-(5-Chloro-7-cyclopentylamino-imidazo[4,5-b]pyridin-3-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385642 2-(5-Chloro-7-cyclohexylamino-imidazo[4,5-b]pyridin-3-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385644 3,4-dihydroxy-5-[10-hydroxy-4-methyl-(5R,13R,14S,17R)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10,15-tetraen-14-yloxy]tetrahydro-2-furancarboxylic acid 1385647 5-(7-Amino-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 1385657 2-Hydroxymethyl-5-[6-(4-phenyl-butylamino)-purin-9-yl]-tetrahydro-furan-3,4-diol 1385660 5-[6-Amino-2-(3-hydroxy-pent-1-ynyl)-purin-9-yl]-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 1385669 5-(6-Amino-purin-9-yl)-3,4-dihydroxy-4-methyl-tetrahydro-furan-2-carboxylic acid ethylamide 1385673 2-Chloromethyl-5-[6-(3-iodo-benzylamino)-purin-9-yl]-tetrahydro-furan-3,4-diol 1385674 (2R,3S,5R)-2-(6-Cyclopropylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385675 2-(6-Cyclooctylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385676 2-(6-Cyclopentylamino-purin-9-yl)-5-isopropylsulfanylmethyl-tetrahydro-furan-3,4-diol 1385678 2-[6-(3-Iodo-benzylamino)-purin-9-yl]-5-methylsulfanylmethyl-tetrahydro-furan-3,4-diol 1385679 2-Ethylsulfanylmethyl-5-[6-(3-iodo-benzylamino)-purin-9-yl]-tetrahydro-furan-3,4-diol 1385680 2-(6-Benzylamino-purin-9-yl)-5-propylsulfanylmethyl-tetrahydro-furan-3,4-diol 1385681 2-(6-Cycloheptylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385684 2-(6-Benzylamino-purin-9-yl)-5-chloromethyl-tetrahydro-furan-3,4-diol 1385689 2-(6-Cyclopentylamino-8-propylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385690 2-(6-Cyclopentylamino-8-ethylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385691 2-(6,8-Bis-cyclopentylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385693 2-(8-Cyclopentylamino-6-ethylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385694 2-(6-Cyclopentylamino-8-methylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385695 (2E)-3-{6-amino-9-[3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl]-9H-purin-2-yl}-N-ethyltriaz-2-ene-1-carboxamide 1385696 (2E)-3-{6-amino-9-[3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl]-9H-purin-2-yl}-N-(2-chlorophenyl)triaz-2-ene-1-carboxamide 1385697 2-{6-amino-2-(E)-N-benzylurea)-diazenyl]-9H-purin-9-yl}-5-(hydroxymethyl)tetrahydrofuran-3,4-diol 1385698 (2E)-3-{6-anilino-9-[3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl]-9H-purin-2-yl}triaz-2-ene-1-carboxamide 1385699 2-(6-Butylamino-8-cyclopentylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385701 5-[6-Amino-2-(5-phenyl-pent-1-ynyl)-purin-9-yl]-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 1385702 (2E)-3-{6-amino-9-[3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl]-9H-purin-2-yl}triaz-2-ene-1-carboxamide 1385703 2-{6-amino-2-[(E)-(N-cyclohexylurea)diazenyl]-9H-purin-9-yl}-5-(hydroxymethyl)tetrahydrofuran-3,4-diol 1385704 2-{6-amino-2-[(1E)-3-benzoyltriaz-1-enyl]-9H-purin-9-yl}-5-(hydroxymethyl)tetrahydrofuran-3,4-diol 1385705 (2E)-3-{6-amino-9-[3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl]-9H-purin-2-yl}-N-1,3-thiazol-2-yltriaz-2-ene-1-carboxamide 1385706 2-{6-amino-2-[(E)-N-(4-methoxyphenyl)urea]diazenyl]-9H-purin-9-yl}-5-(hydroxymethyl)tetrahydrofuran-3,4-diol 1385707 2-{6-N-(ethyl-2,2-diphenyl)-2-[(E)-(N-phenylurea)diazenyl]-9H-purin-9-yl}-5-(hydroxymethyl)tetrahydrofuran-3,4-diol 1385708 2-{6-N-cyclopentyl-2-[(E)-(N-phenylurea)diazenyl]-9H-purin-9-yl}-5-(hydroxymethyl)tetrahydrofuran-3,4-diol 1385709 2-{6-amino-2-[(E)-N-(2-methoxyphenyl)urea]diazenyl]-9H-purin-9-yl}-5-(hydroxymethyl)tetrahydrofuran-3,4-diol 1385710 (2E)-3-{6-amino-9-[3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl]-9H-purin-2-yl}-N-(4-chlorophenyl)triaz-2-ene-1-carboxamide 1385711 (2E)-3-{6-amino-9-[3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl]-9H-purin-2-yl}-N-phenyltriaz-2-ene-1-carboxamide 1385712 2-{6-anilino-2-[(E)-(N-phenylurea)diazenyl]-9H-purin-9-yl}-5-(hydroxymethyl)tetrahydrofuran-3,4-diol 1385713 2-(8-Cyclopentylamino-6-methylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385714 2-(6-Amino-2-phenylazo-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385715 2-(6-Amino-2-nitroso-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385717 2-(6-Cyclopentylamino-purin-9-yl)-5-ethylaminomethyl-tetrahydro-furan-3,4-diol 1385718 2-(6-Cyclopentylamino-purin-9-yl)-5-propylsulfanylmethyl-tetrahydro-furan-3,4-diol 1385719 2-(6-Cyclopentylamino-purin-9-yl)-5-methylsulfanylmethyl-tetrahydro-furan-3,4-diol 1385720 2-(6-Cyclopentylamino-purin-9-yl)-5-isobutylsulfanylmethyl-tetrahydro-furan-3,4-diol 1385721 2-(6-Cyclopentylamino-purin-9-yl)-5-methylaminomethyl-tetrahydro-furan-3,4-diol 1385722 2-(6-Cyclopentylamino-purin-9-yl)-5-methylselanylmethyl-tetrahydro-furan-3,4-diol 1385723 2-(6-Cyclopentylamino-purin-9-yl)-5-propylaminomethyl-tetrahydro-furan-3,4-diol 1385724 2-(6-Amino-8-butylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385735 2-Hydroxymethyl-5-[6-(3-phenyl-propylamino)-purin-9-yl]-tetrahydro-furan-3,4-diol 1385738 2-(6-Benzylamino-2-nitro-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385739 2-Hydroxymethyl-5-[6-(3-iodo-benzylamino)-2-nitro-purin-9-yl]-tetrahydro-furan-3,4-diol 1385740 5-(6-Amino-purin-9-yl)-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid cyclohexylamide 1385741 2-(6-Cyclopentylamino-2-nitro-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385742 2-Hydroxymethyl-5-[7-(3-iodo-benzylamino)-5-nitro-imidazo[4,5-b]pyridin-3-yl]-tetrahydro-furan-3,4-diol 1385743 5-(6-Amino-purin-9-yl)-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid pentylamide 1385744 2-(6-Amino-2-nitro-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385745 2-(7-Cyclopentylamino-5-nitro-imidazo[4,5-b]pyridin-3-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385746 2-Hydroxymethyl-5-(6-methoxyamino-2-nitro-purin-9-yl)-tetrahydro-furan-3,4-diol 1385747 2-(6-Amino-2-oct-1-ynyl-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385753 2-(7-Amino-5-nitro-imidazo[4,5-b]pyridin-3-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385758 2-(6-Amino-2-hept-1-ynyl-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385760 5-(6-Amino-2-pent-1-ynyl-purin-9-yl)-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 1385761 2-(6-Amino-2-pent-1-ynyl-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385776 5-[6-Amino-2-((Z)-5-phenyl-pent-1-enyl)-purin-9-yl]-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 1385777 5-[6-Amino-2-((E)-styryl)-purin-9-yl]-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 1385778 2-[6-Amino-2-((Z)-hex-1-enyl)-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385779 5-[6-Amino-2-((E)-hex-1-enyl)-purin-9-yl]-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 1385780 5-(6-Amino-2-hexyl-purin-9-yl)-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 1385803 2-(6-Amino-2-{N'-[3,3-diphenyl-prop-2-en-(E)-ylidene]-hydrazino}-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385804 2-(6-Amino-2-{N'-[(E)-3-(4-dimethylamino-phenyl)-prop-2-en-(E)-ylidene]-hydrazino}-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385805 2-(6-Amino-2-{N'-[(E)-3-(2-methoxy-phenyl)-prop-2-en-(E)-ylidene]-hydrazino}-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385806 2-(6-Amino-2-{N'-[(E)-3-furan-2-yl-prop-2-en-(E)-ylidene]-hydrazino}-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385807 2-(6-Amino-2-{N'-[(E)-3-(4-nitro-phenyl)-prop-2-en-(E)-ylidene]-hydrazino}-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385809 2-(6-Amino-2-{N'-[(E)-3-(2-nitro-phenyl)-prop-2-en-(E)-ylidene]-hydrazino}-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385810 2-(6-Amino-2-{N'-[(E)-3-(4-hydroxy-3-methoxy-phenyl)-prop-2-en-(E)-ylidene]-hydrazino}-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385811 2-(6-Amino-2-{N'-[(E)-3-(4-methoxy-phenyl)-prop-2-en-(E)-ylidene]-hydrazino}-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385814 2-(6-Amino-2-{N'-[(E)-3-phenyl-prop-2-en-(E)-ylidene]-hydrazino}-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385815 2-(6-Amino-2-{N'-[1-furan-2-yl-meth-(E)-ylidene]-hydrazino}-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385825 Ammonium; 4-{4-[9-(3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-6-ylamino]-butyl}-benzenesulfonate 1385826 2-(6-Decylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1385827 Sodium salt 4-{3-[9-(3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-6-ylamino]-propyl}-benzenesulfonate 1385828 Sodium salt 10-[9-(3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-6-ylamino]-decane-1-sulfonate 1385845 3,4-Dihydroxy-5-{6-[2-(1-naphthalen-1-ylmethyl-1H-indol-3-yl)-ethylamino]-purin-9-yl}-tetrahydro-furan-2-carboxylic acid cyclopropylamide 1385849 3,4-Dihydroxy-5-{6-[2-(1H-indol-3-yl)-ethylamino]-purin-9-yl}-tetrahydro-furan-2-carboxylic acid cyclopropylamide 1385858 5-[2-Chloro-6-(3-iodo-benzylamino)-purin-9-yl]-3,4-dihydroxy-3-methyl-tetrahydro-furan-2-carboxylic acid methylamide 1385859 5-[2-Chloro-6-(3-iodo-benzylamino)-purin-9-yl]-3,4-dihydroxy-4-methyl-tetrahydro-furan-2-carboxylic acid methylamide 1385860 2-(6-Cyclohexylamino-purin-9-yl)-5-hydroxymethyl-3-methyl-tetrahydro-furan-3,4-diol 1385891 3,4-Dihydroxy-5-[6-(3-iodo-benzylamino)-2-methylamino-purin-9-yl]-3-methyl-tetrahydro-furan-2-carboxylic acid methylamide 1385892 2-(6-Benzylamino-purin-9-yl)-5-hydroxymethyl-3-methyl-tetrahydro-furan-3,4-diol 1385893 5-[2-Chloro-6-(3-iodo-benzylamino)-purin-9-yl]-2-hydroxymethyl-3-methyl-tetrahydro-furan-3,4-diol 1385894 3,4-Dihydroxy-5-[6-(3-iodo-benzylamino)-purin-9-yl]-3-methyl-tetrahydro-furan-2-carboxylic acid methylamide 1385917 14beta-(2'-chlorocinnamoylamino)-7,8-dihydromorphinone 1385924 3-Methoxy-2-phenyl-quinoline-4-carboxylic acid ((R)-1-phenyl-propyl)-amide 1385926 (-)-3-Hydroxy-N-(S)-tetrahydrofurfuryl]morphinan hydrochloride 1385964 7-Chloro-3-(3,5-dimethyl-phenyl)-6-nitro-4-{2-[(S)-6-(3-phenyl-propyl)-piperidin-2-yl]-ethoxy}-1H-quinolin-2-one 1385967 7-Chloro-3-(3,5-dimethyl-phenyl)-4-[2-((S)-6-ethyl-piperidin-2-yl)-ethoxy]-6-nitro-1H-quinolin-2-one 1385968 7-Chloro-3-(3,5-dimethyl-phenyl)-4-[2-((S)-6-methyl-piperidin-2-yl)-ethoxy]-6-nitro-1H-quinolin-2-one 1385971 (+/-)-trans-2-[3-methoxy-4-(4-chlorophenylthioethoxy)-5-(N-methyl-N-hydroxyureidyl)methylphenyl]-5-(3,4,5-trimethoxyphenyl)tetrahydrofuran 1385972 (+/-)-trans-2-[3-methoxy-4-(2-bromorophenylthioethoxy)-5-(N-butyl-N-hydroxyureidyl)phenyl]-5-(3,4,5-trimethoxyphenyl)tetrahydrofuran 1385973 (+/-)-trans-2-[3-methoxy-4-(3-bromorophenylthioethoxy)-5-(N-butyl-N-hydroxyureidyl)phenyl]-5-(3,4,5-trimethoxyphenyl)tetrahydrofuran 1385974 (+/-)-trans-2-[3-methoxy-4-(4-bromophenylthioethoxy)-5-(N-butyl-N-hydroxyureidyl)phenyl]-5-(3,4,5-trimethoxyphenyl)tetrahydrofuran 1385975 (+/-)-trans-2-[3-methoxy-4-(3,4-dichlorophenylthioethoxy)-5-(N-butyl-N-hydroxyureidyl)phenyl]-5-(3,4,5-trimethoxyphenyl)tetrahydrofuran 1385976 (+/-)-trans-2-[3-methoxy-4-(2,3,5,6tetrafluorophenylthioethoxy)-5-(N-butyl-N-hydroxyureidyl)phenyl]-5-(3,4,5-trimethoxyphenyl)tetrahydrofuran 1385977 (+/-)-trans-2-[3-methoxy-4-(4-bromophenylsulphonylethoxy)-5-(N-butyl-N-hydroxyureidyl)phenyl]-5-(3,4,5-trimethoxyphenyl)tetrahydrofuran 1385978 (+/-)-trans-2-[3-methoxy-4-(4-chlorophenylthioethoxy)-5-(N-butyl-N-hydroxyureidyl)phenyl]-5-(3,4,5-trimethoxyphenyl)tetrahydrofuran 1385979 {(S)-2-[(R)-6-Oxo-3-(2-phenyl-pyrazolo[1,5-a]pyridin-3-yl)-6H-pyridazin-1-yl]-cyclohexyl}-acetic acid 1385980 {(R)-2-[(R)-6-Oxo-3-(2-phenyl-pyrazolo[1,5-a]pyridin-3-yl)-6H-pyridazin-1-yl]-cyclohexyl}-acetic acid 1385981 (+/-)-trans-2-[3-methoxy-4-(4-methoxyphenylthioethoxy)-5-(N-butyl-N-hydroxyureidyl)phenyl]-5-(3,4,5-trimethoxyphenyl)tetrahydrofuran 1385982 (+/-)-trans-2-[3-methoxy-4-(4-chlorophenylthioethoxy)-5-(N-butyl-N-hydroxyureidyl)methylphenyl]-5-(3,4,5-trimethoxyphenyl)tetrahydrofuran 1385983 (+/-)-trans-2-[3-methoxy-4-(2,3,5,6tetrafluoro-phenylsulphonylethoxy)-5-(N-butyl-N-hydroxyureidyl)phenyl]-5-(3,4,5-trimethoxyphenyl)tetrahydrofuran 1385984 (+/-)-trans-2-[3-methoxy-4-(2-bromophenylsulphonylethoxy)-5-(N-butyl-N-hydroxyureidyl)phenyl]-5-(3,4,5-trimethoxyphenyl)tetrahydrofuran 1385985 3-[(3R,4R)-3,4-Dimethyl-1-((S)-2-phenyl-cyclopropylmethyl)-piperidin-4-yl]-phenol 1385986 3-[(3R,4R)-3,4-Dimethyl-1-((R)-2-phenyl-cyclopropylmethyl)-piperidin-4-yl]-phenol 1386449 Acetic acid 2-methyl-2-aza-bicyclo[2.2.1]hept-5-yl ester 1386450 Acetic acid 2-benzyl-2-aza-bicyclo[2.2.1]hept-6-yl ester 1386451 2,2-Diphenyl-propionic acid 2-methyl-2-aza-bicyclo[2.2.1]hept-5-yl ester 1386452 2,2-Diphenyl-propionic acid 2-methyl-2-aza-bicyclo[2.2.1]hept-6-yl ester 1386471 (4aS,9aR)-4a-Ethyl-2-propyl-1,2,3,4,4a,9a-hexahydro-benzo[4,5]furo[2,3-c]pyridin-6-ol 1386786 2-Hydroxy-2-phenyl-propionic acid 1-aza-bicyclo[2.2.2]oct-3-yl ester 1386787 2-Hydroxy-2-phenyl-propionic acid 1-aza-bicyclo[2.2.2]oct-3-yl ester 1386860 (R)-2-{(R)-2-[2-({1-[(R)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-hydroxy-cyclopentanecarbonyl}-amino)-acetylamino]-3-phenyl-propionylamino}-4-methyl-pentanoic acid 1386861 (R)-2-{(R)-2-[2-({1-[(R)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-hydroxy-cyclohexanecarbonyl}-amino)-acetylamino]-3-phenyl-propionylamino}-4-methyl-pentanoic acid 1387073 Acetic acid 2-methyl-2-aza-bicyclo[2.2.1]hept-5-yl ester 1387074 Acetic acid 2-benzyl-2-aza-bicyclo[2.2.1]hept-6-yl ester 1387075 2,2-Diphenyl-propionic acid 2-methyl-2-aza-bicyclo[2.2.1]hept-5-yl ester 1387076 2,2-Diphenyl-propionic acid 2-methyl-2-aza-bicyclo[2.2.1]hept-6-yl ester 1387128 3-[2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-6-(3-o-tolyl-ureido)-hexanoylamino]-N-(1-carbamoyl-2-phenyl-ethyl)-N-methyl-succinamic acid 1387253 3-[5-Imidazol-1-yl-2-(3-methyl-pyridin-2-ylamino)-thiazol-4-yl]-benzonitrile 1387292 2-Hydroxy-2-phenyl-propionic acid 1-aza-bicyclo[2.2.2]oct-3-yl ester 1387293 (RR)-2-Hydroxy-2-phenyl-propionic acid 1-aza-bicyclo[2.2.2]oct-3-yl ester (RR-QNA) 1387443 (R)-2-{(R)-2-[2-({1-[(R)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-hydroxy-cyclopentanecarbonyl}-amino)-acetylamino]-3-phenyl-propionylamino}-4-methyl-pentanoic acid 1387444 (R)-2-{(R)-2-[2-({1-[(R)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-hydroxy-cyclohexanecarbonyl}-amino)-acetylamino]-3-phenyl-propionylamino}-4-methyl-pentanoic acid 1387445 2-Hydroxy-8-aza-bicyclo[3.2.1]octane-6-carboxylic acid methyl ester 1387479 [(2S,3S)-2-(3-Chloro-phenyl)-1-aza-bicyclo[2.2.2]oct-3-yl]-(2,4-dimethoxy-benzyl)-amine 1417391 Isobutyl-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with maleic acid 1417392 4-(3-Isobutoxy-propyl)-1H-imidazole; compound with maleic acid 1417393 4-[3-(4-Methyl-pentyloxy)-propyl]-1H-imidazole; compound with maleic acid 1417394 4-[3-(3,3-Dimethyl-butoxy)-propyl]-1H-imidazole; compound with maleic acid 1417395 4-[3-(3-Methyl-butoxy)-propyl]-1H-imidazole; compound with maleic acid 1417404 (S)-4-Ethyl-piperazine-2-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide; compound with 2 TFA 1417405 (S)-4-(2,2-Difluoro-ethyl)-piperazine-2-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide; compound with 2 TFA 1417406 (S)-4-Isobutyl-piperazine-2-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide; compound with 2 TFA 1417407 (S)-4-(2-Amino-propionyl)-piperazine-2-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide; compound with 2 TFA 1442025 6-Amino-2-((S)-2-{(R)-2-[2-amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionylamino]-5-guanidino-1-oxo-pentylamino}-3-phenyl-propionylamino)-hexanoic acid amide 1442796 (3S,4R,5R)-2-(6-Amino-8-hex-1-ynyl-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1503098 2,7-Dimethyl-8-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-deca-2,4-dienedioic acid 1503213 2-[4-(6,7-Dihydroxy-1,2,3,4-tetrahydro-isoquinolin-1-ylmethyl)-phenoxy]-6-hydroxymethyl-tetrahydro-pyran-3,4,5-triol 1503480 N-alpha-Z-Arg-D-Pro-N-Epsolon-Z-Lys-D-Pro-Gln-Gln-D-Phe-D-Phe-GlyPsi(CH2S)D-Leu-D-Met-OMe 1503483 N-alpha-Z-Arg-D-Pro-N-Epsolon-Z-Lys-D-Pro-Gln-Gln-D-Phe-D-Phe-GlyPsi(CH2S)Leu-D-Met-OMe 1503566 N-alpha-Z-Arg-D-Pro-N-Epsolon-Z-Lys-Pro-Asn-Arg-D-Phe-Phe-D-Trp-Leu-Met-OMe 1503569 N-alpha-Z-Arg-Pro-N-Epsolon-Z-Lys-Pro-Gln-Gln-D-Trp-D-Trp-D-Trp-D-Leu-D-Met 1503577 N-alpha-Z-Arg-D-Pro-N-Epsolon-Z-Lys-D-Pro-Gln-Gln-D-Phe-D-Phe-Sar-MeLeu-D-Met-OMe 1503580 N-alpha-Z-Arg-D-Pro-N-Epsolon-Z-Lys-D-Pro-Gln-Gln-D-Phe-D-Phe-Sar-Leu-D-Met-OMe 1503581 N-alpha-Z-Arg-D-Pro-N-Epsolon-Z-Lys-Pro-Asn-Arg-D-Phe-Phe-D-Trp-Leu-Met 1503609 (3S,4R)-5-[6-Amino-2-((E)-5-phenyl-pent-1-enyl)-purin-9-yl]-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid ethylamide 1510266 1-{7-[3-(4-Nitro-phenyl)-allyl]-2,7-diaza-tricyclo[4.4.0.0*3,8*]dec-2-yl}-propan-1-one 1510267 1-{7-[3-(3-Chloro-phenyl)-allyl]-2,7-diaza-tricyclo[4.4.0.0*3,8*]dec-2-yl}-propan-1-one 1510268 1-[7-(3-Phenyl-allyl)-2,7-diaza-tricyclo[4.4.0.0*3,8*]dec-2-yl]-propan-1-one 1510269 1-{7-[3-(3-Nitro-phenyl)-allyl]-2,7-diaza-tricyclo[4.4.0.0*3,8*]dec-2-yl}-propan-1-one 1510331 H-Tyr-Val-Nle-Gly-Pro-Phe-Arg-D-Nal(2'')-Asp-Arg-Phe-Gly-NH2 1510453 H-Tyr-Gly-Gly*-Phe*-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Lys-Trp-Asp-Asn-Gln-OH 1510454 H-Tyr-Gly-Gly-Phe*-Leu*-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Lys-Trp-Asp-Asn-Gln-OH 1510455 H-Tyr*-Gly*-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Lys-Trp-Asp-Asn-Gln-OH 1510456 H-Tyr-Gly-Gly-Phe-Leu*-Arg*-Arg-Ile-Arg-Pro-Lys-Leu-Lys-Trp-Asp-Asn-Gln-OH 1510460 3-(dimethylamino)propyl imidothiocarbamate dihydrobromide 1510557 8-Cyclopentyl-3-(3-fluoro-propyl)-1-propyl-3,7-dihydro-purine-2,6-dione 1510561 8-[2-(3,4-Dimethoxy-phenyl)-vinyl]-7-methyl-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 1510562 8-[2-(3-Chloro-phenyl)-vinyl]-1,3,7-trimethyl-3,7-dihydro-purine-2,6-dione 1510568 carfentanil 1540439 Sodium salt 4-hydroxy-5-hydroxymethyl-2-[6-(4-sulfo-phenylamino)-purin-9-yl]-tetrahydro-furan-3-olate 1542001 3-[2-((S)-2-Acetylamino-3,3-diphenyl-propionylamino)-4-methyl-pentanoylamino]-N-[1-(1-{[1-carboxy-2-(1H-indol-3-yl)-ethyl]-methyl-carbamoyl}-2-methyl-butylcarbamoyl)-2-methyl-butyl]-succinamic acid 1542054 6,11-Dimethyl-3-(tetrahydro-furan-2-ylmethyl)-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocin-8-ol 1542055 (2S,6S,11S)-6,11-Dimethyl-3-[(S)-1-(tetrahydro-furan-2-yl)methyl]-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocin-8-ol 1542096 6,11-Diethyl-3-furan-3-ylmethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocin-8-ol 1542170 N-{(R)-2-[(R)-3-(2,3-Dihydro-1H-indol-3-yl)-2-methyl-2-((1S,4S)-1,7,7-trimethyl-bicyclo[2.2.1]hept-2-yloxycarbonylamino)-propionylamino]-1-phenyl-ethyl}-succinamic acid; compound with (2R,3R,4R,5S)-6-methylamino-hexane-1,2,3,4,5-pentaol 1542209 5-(8-Hydroxy-6,11-dimethyl-1,2,5,6-tetrahydro-4H-2,6-methano-benzo[d]azocin-3-ylmethyl)-5H-furan-2-one 1542211 5-(8-Hydroxy-6,11-dimethyl-1,2,5,6-tetrahydro-4H-2,6-methano-benzo[d]azocin-3-ylmethyl)-dihydro-furan-2-one 1542212 5-(8-Hydroxy-6,11-dimethyl-1,2,5,6-tetrahydro-4H-2,6-methano-benzo[d]azocin-3-ylmethyl)-3-methylene-dihydro-furan-2-one 1542213 5-(8-Hydroxy-6,11-dimethyl-1,2,5,6-tetrahydro-4H-2,6-methano-benzo[d]azocin-3-ylmethyl)-5H-furan-2-one 1542215 5-(8-Hydroxy-6,11-dimethyl-1,2,5,6-tetrahydro-4H-2,6-methano-benzo[d]azocin-3-ylmethyl)-dihydro-furan-2-one 1542669 (1S,9R,13R)-10-(cyclopropylmethyl)-1,13-dimethyl-10-azatricyclo[7.3.1.0^{2,7}]trideca-2(7),3,5-triene-4-carboxamide 1542814 1N-methyl-4-[2-chloro-6-(2-chloro-5-iodobenzylamino)-9H-9-purinyl]-2,3-dihydroxy-(1S,2R,3S,4R,5S)-bicyclo[3.1.0]hexane-1-carboxamide 1542815 1N-methyl-4-[2-chloro-6-(5-iodo-2-methoxybenzylamino)-9H-9-purinyl]-2,3-dihydroxy-(1S,2R,3S,4R,5S)-bicyclo[3.1.0]hexane-1-carboxamide 1542816 1N-methyl-4-[6-(4-amino-3-iodobenzylamino)-2-chloro-9H-9-purinyl]-2,3-dihydroxy-(1S,2R,3S,4R,5S)-bicyclo[3.1.0]hexane-1-carboxamide 1542817 (1S,2R,3S,4R,5S)-4-(2-chloro-6-(2,2-diphenylethylamino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 1542818 (1S,2R,3S,4R,5S)-4-(6-(3-chlorobenzylamino)-2-iodo-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 1542819 1N-methyl-4-[6-(2-carbamoylmethoxy-5-chlorobenzylamino)-2-chloro-9H-9-purinyl]-2,3-dihydroxy-(1S,2R,3S,4R,5S)-bicyclo[3.1.0]hexane-1-carboxamide 1542820 1N-methyl-4-[6-(2-benzyloxy-5-chlorobenzylamino)-2-chloro-9H-9-purinyl]-2,3-dihydroxy-(1S,2R,3S,4R,5S)-bicyclo[3.1.0]hexane-1-carboxamide 1542821 1N-methyl-4-{2-chloro-6-[2-chloro-5-(3-hydroxy-1-propynyl)benzylamino]-9H-9-purinyl}-2,3-dihydroxy-(1S,2R,3S,4R,5S)-bicyclo[3.1.0]hexane-1-carboxamide 1542841 difluoro(2-{[(2Z)-1-methyl-5-(2-{[2-(2-{2-[4-(2-oxo-2-{10-oxo-2,4,9-triazatricyclo[9.4.0.0^{3,8}]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}ethyl)piperazin-1-yl]ethoxy}ethoxy)ethyl]carbamoyl}ethyl)-2H-pyrrol-1-ium-2-ylidene]methyl}-5-(thiophen-2-yl)-1H-pyrrol-1-yl)boranuide 1542842 difluoro(2-{[(2Z)-1-methyl-5-{2-[(5-{[5-({4-[4-(2-oxo-2-{10-oxo-2,4,9-triazatricyclo[9.4.0.0^{3,8}]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}ethyl)piperazin-1-yl]butyl}carbamoyl)pentyl]carbamoyl}pentyl)carbamoyl]ethyl}-2H-pyrrol-1-ium-2-ylidene]methyl}-5-(thiophen-2-yl)-1H-pyrrol-1-yl)boranuide 1542843 difluoro(2-{[(2Z)-1-methyl-5-[2-({20-[4-(2-oxo-2-{10-oxo-2,4,9-triazatricyclo[9.4.0.0^{3,8}]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}ethyl)piperazin-1-yl]-3,6,9,12,15,18-hexaoxaicosan-1-yl}carbamoyl)ethyl]-2H-pyrrol-1-ium-2-ylidene]methyl}-5-(thiophen-2-yl)-1H-pyrrol-1-yl)boranuide 1542844 difluoro(2-{[(2Z)-1-methyl-5-[2-({6-[4-(2-oxo-2-{10-oxo-2,4,9-triazatricyclo[9.4.0.0^{3,8}]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}ethyl)piperazin-1-yl]hexyl}carbamoyl)ethyl]-2H-pyrrol-1-ium-2-ylidene]methyl}-5-(thiophen-2-yl)-1H-pyrrol-1-yl)boranuide 1542906 (1S,2R,3S,4R,5S)-4-(6-(3-bromobenzylamino)-2-chloro-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 1543062 N-{4-[2-(6-Cyano-3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-cyclohexyl}-3-(4-fluoro-phenyl)-acrylamide 1543063 N-{4-[2-(6-Cyano-3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-cyclohexyl}-3-phenyl-acrylamide 1543126 2-{6-[2-(4-Hydroxy-3-iodo-phenyl)-1-methyl-ethylamino]-purin-9-yl}-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1543814 2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-3-(1H-indol-3-yl)-propionylamino]-propionylamino}-N-{[1-(1-hydroxymethyl-3-methyl-butylcarbamoyl)-2-(3H-imidazol-4-yl)-ethylcarbamoyl]-methyl}-3-methyl-butyramide 1543823 2-[2-[2-(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-3-(1H-indol-3-yl)-propionylamino]-propionylamino}-3-methyl-butyrylamino)-acetylamino]-3-(3H-imidazol-4-yl)-propionylamino]-4-methyl-pentanoic acid ethyl ester 1543826 2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-3-(1H-indol-3-yl)-propionylamino]-propionylamino}-N-{1-[1-(1-ethoxymethyl-3-methyl-butylcarbamoyl)-2-(3H-imidazol-4-yl)-ethylcarbamoyl]-ethyl}-3-methyl-butyramide 1543827 2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-3-(1H-indol-3-yl)-propionylamino]-propionylamino}-N-{1-[1-(1-ethoxymethyl-3-methyl-butylcarbamoyl)-2-(3H-imidazol-4-yl)-ethylcarbamoyl]-ethyl}-3-methyl-butyramide 1543828 2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-3-(1H-indol-3-yl)-propionylamino]-propionylamino}-N-{[2-(3H-imidazol-4-yl)-1-(1-isobutyl-pentylcarbamoyl)-ethylcarbamoyl]-methyl}-3-methyl-butyramide 1543835 2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-3-(1H-indol-3-yl)-propionylamino]-propionylamino}-N-{[2-(3H-imidazol-4-yl)-1-(3-methyl-1-propoxymethyl-butylcarbamoyl)-ethylcarbamoyl]-methyl}-3-methyl-butyramide 1543836 2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-3-(1H-indol-3-yl)-propionylamino]-propionylamino}-N-{[2-(3H-imidazol-4-yl)-1-(1-methoxymethyl-3-methyl-butylcarbamoyl)-ethylcarbamoyl]-methyl}-3-methyl-butyramide 1543838 2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-3-(1H-indol-3-yl)-propionylamino]-propionylamino}-N-{[1-(1-ethoxymethyl-3-methyl-butylcarbamoyl)-2-(3H-imidazol-4-yl)-ethylcarbamoyl]-methyl}-3-methyl-butyramide 1543839 2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-3-(1H-indol-3-yl)-propionylamino]-propionylamino}-N-({2-(3H-imidazol-4-yl)-1-[3-methyl-1-(3-methyl-butoxymethyl)-butylcarbamoyl]-ethylcarbamoyl}-methyl)-3-methyl-butyramide 1543944 2-[2-(2-{2-[2-(2-{2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-6-amino-hexanoylamino}-3-carboxy-propionylamino)-3-cyclohexyl-propionylamino]-3-cyclohexyl-propionylamino}-3-cyclohexyl-propionylamino)-acetylamino]-5-guanidino-pentanoic acid 1543945 2-[2-(2-{2-[2-(2-{2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-6-amino-hexanoylamino}-3-carboxy-propionylamino)-hexanoylamino]-hexanoylamino}-hexanoylamino)-acetylamino]-5-guanidino-pentanoic acid 1543952 2-[2-(2-{2-[2-(2-{2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-6-amino-hexanoylamino}-3-carboxy-propionylamino)-4-methylsulfanyl-butyrylamino]-4-carbamoyl-butyrylamino}-4-methyl-pentanoylamino)-acetylamino]-5-guanidino-pentanoic acid 1544077 Tyr-D-Ala-Phe-Gly-Tyr-Pro-Thr[Beta-D-Glc(OAc)4]-Gly-NH2 1544160 (S)-2-{(S)-2-[(1-{(S)-2-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-4-methyl-pentanoylamino]-3-carbamoyl-propionyl}-pyrrolidine-2-carbonyl)-amino]-3-methyl-pentanoylamino}-3-(1H-indol-3-yl)-propionic acid 1544161 (S)-2-{(S)-2-[(1-{(S)-2-[(S)-2-((S)-2-Acetylamino-3-phenyl-propionylamino)-4-methyl-pentanoylamino]-3-carbamoyl-propionyl}-pyrrolidine-2-carbonyl)-amino]-3-methyl-pentanoylamino}-3-(1H-indol-3-yl)-propionic acid 1544162 (S)-3-{(S)-2-[(S)-2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-4-methyl-pentanoylamino}-4-(2-{(S)-1-[(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-pyrrolidin-1-yl)-4-oxo-butyric acid 1544164 (S)-2-{(S)-2-[(1-{(S)-2-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propionylamino)-4-methyl-pentanoylamino]-3-carbamoyl-propionyl}-pyrrolidine-2-carbonyl)-amino]-3-methyl-pentanoylamino}-3-(1H-indol-3-yl)-propionic acid 1544165 (S)-2-((S)-2-{[1-((S)-2-{(S)-2-[(S)-2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-4-methyl-pentanoylamino}-3-carbamoyl-propionyl)-pyrrolidine-2-carbonyl]-amino}-3-methyl-pentanoylamino)-3-(1H-indol-3-yl)-propionic acid 1544170 Ala6-SRIF-14-amide 1544171 Ala7-SRIF-14-amide 1544173 Demotensin 1 1544187 3-[2-((S)-2-Acetylamino-3,3-diphenyl-propionylamino)-4-methyl-pentanoylamino]-N-[1-({1-[1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butyl}-methyl-carbamoyl)-2-methyl-butyl]-succinamic acid 1544266 N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[3-(1H-indol-3-yl)-2-(2-{4-methylsulfanyl-2-[2-(4-sulfooxy-phenyl)-acetylamino]-butyrylamino}-acetylamino)-propionylamino]-4-methylsulfanyl-butyrylamino}-N-methyl-succinamic acid 1544267 N-(1-Carbamoyl-2-phenyl-ethyl)-3-({2-[2-(2-{2-[2-(4-hydroxy-phenyl)-acetylamino]-hexanoylamino}-acetylamino)-3-(1H-indol-3-yl)-propionylamino]-hexanoyl}-methyl-amino)-succinamic acid 1544268 N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[3-(1H-indol-3-yl)-2-(2-{4-methylsulfanyl-2-[2-(4-sulfooxy-phenyl)-acetylamino]-butyrylamino}-acetylamino)-propionylamino]-4-methylsulfanyl-butyrylamino}-succinamic acid 1544269 N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[2-(2-{2-[2-(4-hydroxy-phenyl)-acetylamino]-hexanoylamino}-acetylamino)-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-N-methyl-succinamic acid 1544409 H-Dmt-Tic-Glu-NH2 1544521 (S)-3-[2-((R)-2-Acetylamino-3-phenyl-propionylamino)-5-amino-pentanoylamino]-N-{(S)-1-[(S)-1-((S)-carboxy-2-(S)-1-1H-indol-3-yl-ethylcarbamoyl)-2-(S)-methyl-butylcarbamoyl]-2-methyl-butyl}-succinamic acid 1544605 alpha-melanotropin-II(MT-II) peptide 1544650 (S)-2-Amino-N-((5S,8S)-5-benzyl-4,7,13,16-tetraoxo-hexadecahydro-3a,6,12,15-tetraaza-cyclopentacyclopentadecen-8-yl)-3-(4-hydroxy-phenyl)-propionamide 1544658 (S)-2-Amino-3-(4-hydroxy-phenyl)-N-((5S,8S)-5-naphthalen-2-ylmethyl-4,7,13,16-tetraoxo-hexadecahydro-3a,6,12,15-tetraaza-cyclopentacyclopentadecen-8-yl)-propionamide 1544700 2-{2-[2-[2-[2-(2-Amino-3-methyl-pentanoylamino)-3-methyl-pentanoylamino]-3-(1H-indol-3-yl)-propionylamino]-3-(1H-imidazol-4-yl)-propionylamino]-4-methyl-pentanoylamino}-succinic acid 1544702 2-{2-[2-[2-[2-(2-Amino-3-methyl-pentanoylamino)-3-methyl-pentanoylamino]-3-(1H-indol-3-yl)-propionylamino]-3-(1H-indol-3-yl)-propionylamino]-4-methyl-pentanoylamino}-succinic acid 1544710 2-{2-[2-[2-[2-(2-Amino-3-methyl-pentanoylamino)-3-methyl-pentanoylamino]-3-(1H-indol-3-yl)-propionylamino]-3-(1H-indol-3-yl)-propionylamino]-4-methyl-pentanoylamino}-succinic acid 1544712 2-(2-{2-[2-[2-(2-Amino-3-methyl-pentanoylamino)-3-methyl-pentanoylamino]-3-(1H-indol-3-yl)-propionylamino]-3-phenyl-propionylamino}-4-methyl-pentanoylamino)-succinic acid 1544779 Tyr-D-Ala-Phe-Asp-Val-Val-Thr[Beta-D-Glc]-Gly-NH2 1544780 Tyr-D-Ala-Phe-Thr(-D-Glc)-Tyr-Pro-Ser-NH2 1544782 Tyr-D-Ala-Phe-Thr[Beta-D-Glc(OAc)4]-Val-ValGly-NH2 1544783 2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-3-phenyl-propionylamino)-N-{1-[1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-3-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-butyramide 1544784 Tyr-D-Ala-Phe-Thr[-D-Glc(OAc)4]-Tyr-Pro-Ser-NH2 1544945 H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys*-Ile*-Arg-Pro-Lys-Leu-Lys-Trp-Asp-Asn-Gln-OH 1544946 H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys-Ile*-Lys*-Pro-Lys-Leu-Lys-Trp-Asp-Asn-Gln-OH 1544947 H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys-Ile*-Arg*-Pro-Lys-Leu-Lys-Trp-Asp-Asn-Gln-OH 1544948 H-Tyr-Gly-Gly-Phe-Leu-Lys*-Arg*-Ile-Arg-Pro-Lys-Leu-Lys-Trp-Asp-Asn-Gln-OH 1544958 (R)-11-{Hydroxy-[4-hydroxy-3-(3-methyl-but-2-enyl)-phenyl]-methyl}-5-(1H-indol-3-ylmethyl)-17-isopropyl-hexadecahydro-3a,6,9,12,15,18,21-heptaaza-cyclopentacyclohenicosene-4,7,10,13,16,19,22-heptaone 1544960 (R)-11-[Hydroxy-(4-methoxy-phenyl)-methyl]-5-(1H-indol-3-ylmethyl)-17-isopropyl-hexadecahydro-3a,6,9,12,15,18,21-heptaaza-cyclopentacyclohenicosene-4,7,10,13,16,19,22-heptaone 1544961 (R)-11-{Hydroxy-[4-methoxy-3-(2-methyl-butyl)-phenyl]-methyl}-5-(1H-indol-3-ylmethyl)-17-isopropyl-hexadecahydro-3a,6,9,12,15,18,21-heptaaza-cyclopentacyclohenicosene-4,7,10,13,16,19,22-heptaone 1544962 (R)-5-(1H-Indol-3-ylmethyl)-17-isopropyl-11-(4-methoxy-benzyl)-hexadecahydro-3a,6,9,12,15,18,21-heptaaza-cyclopentacyclohenicosene-4,7,10,13,16,19,22-heptaone 1544964 (R)-11-{Hydroxy-[4-methoxy-3-(3-methyl-but-2-enyl)-phenyl]-methyl}-5-(1H-indol-3-ylmethyl)-17-isopropyl-hexadecahydro-3a,6,9,12,15,18,21-heptaaza-cyclopentacyclohenicosene-4,7,10,13,16,19,22-heptaone 1544965 (R)-5-(1H-Indol-3-ylmethyl)-17-isopropyl-11-[4-methoxy-3-(2-methyl-butyl)-benzyl]-hexadecahydro-3a,6,9,12,15,18,21-heptaaza-cyclopentacyclohenicosene-4,7,10,13,16,19,22-heptaone 1545039 Boc-cyclo-(D-Asp-Tyr(SO3H)-Nle-D-Lys)-Trp-Nle-Asp-Phe-NH2 1545049 Boc-cyclo-(Asp-Tyr(SO3H)-Nle-D-Lys)-Trp-Nle-Asp-Phe-NH2 1545054 2-[2-({2-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl}-amino)-3-phenyl-propionylamino]-3-(4-amino-phenyl)-propionic acid 1545057 2-[2-({2-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl}-amino)-3-(4-amino-phenyl)-propionylamino]-3-phenyl-propionic acid 1545071 3-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrrolidine-4-carboxylic acid [1-benzyl-2-(2-carbamoyl-pyrrolidin-1-yl)-2-oxo-ethyl]-amide 1545122 (S)-3-[2-({(S)-2-[(S)-2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-4-methylsulfanyl-butyrylamino}-3-phenyl-propionylamino)-3-(3H-imidazol-4-yl)-propionylamino]-4-methyl-pentanoyl}-sec-butyl-amino)-acetylamino]-succinamic acid 1545124 1-(1-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-3-methyl-pentanoyl}-pyrrolidine-2-carbonyl)-pyrrolidine-2-carboxylic acid 1545142 Ac-Phe-Lys-AspMet-GIn-Leu-Gly-Arg-OH 1545626 H-(2R,3S)beta-MePhe-c[Cys-Tyr-D-Trp-Arg-Thr-Pen]-Thr-NH2 1545627 H-(2R,3R)beta-MePhe-c[Cys-Tyr-D-Trp-Arg-Thr-Pen]-Thr-NH2 1545727 (S)-2-{(R)-2-[2-({1-[2-(2-Amino-5-guanidino-pentanoylamino)-5-guanidino-pentanoyl]-pyrrolidine-2-carbonyl}-amino)-3-(4-hydroxy-phenyl)-propionylamino]-3-phenyl-propionylamino}-4-methyl-pentanoic acid 1545787 Tyr-Pro-D-(NMe)Phe-D-Pro-NH2 1545790 Tyr-Pro-L-(NMe)Phe-Pro-NH2 1545791 Tyr-Pro-D-Phe-D-Pro-NH2 1545810 Tyr-Pro-D-Phe-Pro-NH2 1545811 Tyr-(NMe)Ala-L-Phe-D-Pro-NH2 1545812 Tyr-Ala-L-Phe-D-Pro-NH2 1545894 Tyr-Gly-Gly-(L-Tic)-c(Cys-Arg-Arg-Ile-Arg-Pro-Cys) 1546131 13-(2-Amino-ethyl)-19-benzyl-22-(4-ethoxy-benzyl)-16-isopropyl-12,15,18,21,24-pentaoxo-7,8-dithia-11,14,17,20,23-pentaaza-spiro[5.19]pentacosane-10-carboxylic acid (5-amino-1-carbamoyl-pentyl)-amide 1546163 H-Tyr-Val-Nle-Gly-Pro-D-Nal(2'')-Arg-D-Nal-Asp-Arg-Phe-Gly-NH2 1546164 (S)-1-[2-Amino-3-(4-hydroxy-2-methyl-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid [(S)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-ethyl]-amide 1546165 (S)-1-[2-Amino-3-(2-ethyl-4-hydroxy-6-methyl-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid [(S)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-ethyl]-amide 1546168 (S)-1-[2-Amino-3-(4-hydroxy-2-isopropyl-6-methyl-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid [(S)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-ethyl]-amide 1546169 (S)-1-[2-Amino-3-(2,6-diethyl-4-hydroxy-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid [(S)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-ethyl]-amide 1546170 (S)-1-[2-Amino-3-(4-hydroxy-2,6-diisopropyl-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid [(S)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-ethyl]-amide 1546171 (S)-1-[2-Amino-3-(4-hydroxy-2,3,6-trimethyl-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid [(S)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-ethyl]-amide 1546173 5N-[1-[1-carbamoyl-2-phenyl-(1S)-ethylcarbamoyl]-2-phenyl-(1S)-ethyl]-1-[2-amino-3-(4-hydroxy-2,5-dimethylphenyl)-(2S)-propanoyl]-(5S)-dihydro-1H-5-pyrrolecarboxamide 1546175 [N40,Pro1,Tyr4,Nle 14]BB 1546176 [N40,Pro1,Tyr4]BB 1546177 [Tyr4]Bombesin 1546229 2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid ((R)-5-amino-1-carbamoyl-pentyl)-amide 1546272 Degarelix analogue 1546273 Degarelix analogue 1546279 2-{2-[(S)-2-(Acetyl-butyl-amino)-acetylamino]-acetylamino}-6-amino-hexanoic acid benzyl-({1-[1-((S)-carbamoylmethyl-carbamoyl)-2-(1H-indol-3-yl)-ethylcarbamoyl]-4-guanidino-butylcarbamoyl}-methyl)-amide 1546284 2-{2-[{2-[2-(Acetyl-butyl-amino)-acetylamino]-acetyl}-(4-amino-butyl)-amino]-acetylamino}-N-{[1-(carbamoylmethyl-carbamoyl)-2-(1H-indol-3-yl)-ethylcarbamoyl]-methyl}-N-(3-guanidino-propyl)-3-phenyl-propionamide 1546286 2-[(S)-2-((S)-2-Acetylamino-hexanoylamino)-1-oxo-ethylamino]-6-amino-hexanoic acid {1-[{[1-(carbamoylmethyl-carbamoyl)-2-(1H-indol-3-yl)-ethylcarbamoyl]-methyl}-(4-guanidino-butyl)-carbamoyl]-2-phenyl-ethyl}-amide 1546316 7-Hydroxy-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-[(S)-1-({[(S)-2-[(S)-2-((S)-1-carbamoyl-2-hydroxy-ethylcarbamoyl)-pyrrolidin-1-yl]-1-(4-hydroxy-benzyl)-2-oxo-ethylcarbamoyl]-methyl}-carbamoyl)-2-phenyl-ethylcarbamoyl]-ethyl}-amide 1546317 6-Hydroxy-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-[(S)-1-({[(S)-2-[(S)-2-((S)-1-carbamoyl-2-hydroxy-ethylcarbamoyl)-pyrrolidin-1-yl]-1-(4-hydroxy-benzyl)-2-oxo-ethylcarbamoyl]-methyl}-carbamoyl)-2-phenyl-ethylcarbamoyl]-ethyl}-amide 1546318 6-Hydroxy-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-[(S)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-ethylcarbamoyl]-ethyl}-amide 1546319 (S)-N-{(S)-1-[(S)-1-(Carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-3-((S)-2-{(R)-2-[(7-hydroxy-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl)-amino]-propionylamino}-3-phenyl-propionylamino)-succinamic acid 1546359 Sub[-Tyr-Arg-Leu-Arg-Tyr-NH2]2 1546360 Adp[-Trp-Arg-Nva-Arg-Tyr-NH2]2 1546361 Pim[-Trp-Arg-Nva-Arg-Tyr-NH2]2 1546362 Sub[-Trp-Arg-Nva-Arg-Tyr-NH2]2 1546367 2-[2-(2-{2-[2-(2-Amino-4-carbamoyl-butyrylamino)-4-carbamoyl-butyrylamino]-3-phenyl-propionylamino}-3-phenyl-propionylamino)-acetylamino]-4-methyl-pentanoic acid (1-carbamoyl-3-methylsulfanyl-propyl)-amide 1546373 Cyclo[Ac-Cys-Ile-Tyr-Lys-Tyr-Phe] 1546378 2-(2-(2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamido)acetic acid 1546379 Hoo-Phe-Orn-Pro-hle-Pff-Phe-NH2 1546384 [pGlu4]U-II(4-11) 1546386 H-Tyr-Tic-Cha-Phe-OH 1546413 Ac-Nle4-cyclo(Asp5-His6-D-4,4'-Bip7-Pip8-Trp9-Lys10)-NH2 1546414 Ac-Nle4-cyclo(Asp5-Pro6-D-4,4'-Bip7-Pro8-Trp9-Lys10)-NH2 1546415 Ac-Nle4-cyclo(Asp5-His6-D-4-Dip-Pro8-Trp9-Lys10)-NH2 1546416 Ac-Nle4-cyclo(Asp5-Oic6-D-4,4'-Bip7-Pro8-Trp9-Lys10)-NH2 1546417 Ac-Nle4-cyclo(Asp5-Pro6-D-4,4'-Bip7-Pip8-Trp9-Lys10)-NH2 1546418 c-Nle4-cyclo(Asp5-Tic6-D-4,4'-Bip7-Pip8-Trp9-Lys10)-NH2 1546419 Ac-Nle4-cyclo(Asp5-Oic6-D-4,4'-Bip7-Pip8-Trp9-Lys10)-NH2 1546420 Ac-Nle4-cyclo(Asp5-Val6-D-4,4'-Bip7-Pip8-Trp9-Lys10)-NH2 1546421 Ac-Nle4-cyclo(Asp5-Chg6-D-4,4'-Bip7-Pip8-Trp9-Lys10)-NH2 1546422 Ac-Nle4-cyclo(Asp5-Phg6-D-4,4'-Bip7-Pip8-Trp9-Lys10)-NH2 1546423 Ac-Nle4-cyclo(Asp5-Oic6-D-4,4'-Bic7-Pip8-Trp9-Lys10)-NH2 1546424 Ac-Nle4-cyclo(Asp5-Oic6-D-D-pBzlPhe7-Pip8-Trp9-Lys10)-NH2 1546428 H-Tyr-D-Ala-Gly-Phe-Phe-Pro-Leu-Trp-O-3,5-Bzl(CF3)2 1546429 H-Tyr-D-Ala-Gly-Phe-D-Phe-Pro-Leu-Trp-O-3,5-Bzl(CF3)2 1546503 [Phe1psi(CH2-NH)Gly2(pF)Phe4Aib7Arg14Lys15]N/OFQ-NH2 1546557 (S)-2-{(S)-2-[(S)-2-[(1-{(S)-2-[(Adamantane-1-carbonyl)-amino]-6-amino-1-(S)-oxo-hexyl}-pyrrolidine-2-carbonyl)-amino]-3-(4-hydroxy-phenyl)-propionylamino]-3-methyl-pentanoylamino}-4-methyl-pentanoic acid 1546636 (+)-8-Hydroxy-3,6,11-trimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-4-carboxylic acid [({[1-(1-carbamoyl-3-methylsulfanyl-propylcarbamoyl)-2-phenyl-ethylcarbamoyl]-methyl}-carbamoyl)-methyl]-amide 1546647 Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,4,7,10tetraaza-cyclohexadec-12-ylcarbamoyl)-2-(4-hydroxy-phenyl)-ethyl-ammonium 1546648 Acetate1-[1-({[1-(1-carbamoyl-3-methyl-butylcarbamoyl)-2-phenyl-ethylcarbamoyl]-methyl}-carbamoyl)-ethylcarbamoyl]-2-(4-hydroxy-phenyl)-ethyl-ammonium 1546649 Acetate1-[1-({[1-(1-carbamoyl-3-methyl-butylcarbamoyl)-2-phenyl-ethylcarbamoyl]-methyl}-carbamoyl)-propylcarbamoyl]-2-(4-hydroxy-phenyl)-ethyl-ammonium 1546650 Acetate1-[1-({[1-(1-carbamoyl-3-methyl-butylcarbamoyl)-2-phenyl-ethylcarbamoyl]-methyl}-carbamoyl)-butylcarbamoyl]-2-(4-hydroxy-phenyl)-ethyl-ammonium 1546651 Acetate1-(3-benzyl-2,5,8-trioxo-1,4,7triaza-cyclotridec-9-ylcarbamoyl)-2-(4-hydroxy-phenyl)-ethyl-ammonium 1546652 Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,4,7,10tetraaza-cyclopentadec-12-ylcarbamoyl)-2-(4-hydroxy-phenyl)-ethyl-ammonium 1546653 Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,4,7,10tetraaza-cyclotridec-12-ylcarbamoyl)-2-(4-hydroxy-phenyl)-ethyl-ammonium 1546654 Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,4,7,10tetraaza-cyclotetradec-12-ylcarbamoyl)-2-(4-hydroxy-phenyl)-ethyl-ammonium 1546658 Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,4,7,10tetraaza-cyclohexadec-12-ylcarbamoyl)-2-(4-hydroxy-phenyl)-ethyl-ammonium 1546659 3-{(4R,10R,13S)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-10-benzyl-4-[(R)-1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-3,3,14,14-tetramethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradec-7-yl}-propionic acid 1546660 2-(2-{[(4R,10R,13S)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-10-benzyl-7-(3H-imidazol-4-ylmethyl)-3,3,14,14-tetramethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradecane-4-carbonyl]-amino}-hexanoylamino)-succinic acid 1546661 Acetate1-[1-({[1-(1-carbamoyl-3-methyl-butylcarbamoyl)-2-phenyl-ethylcarbamoyl]-methyl}-carbamoyl)-pentylcarbamoyl]-2-(4-hydroxy-phenyl)-ethyl-ammonium 1546663 {(4R,10R,13S)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-10-benzyl-4-[1-(carbamoylmethyl-carbamoyl)-pentylcarbamoyl]-3,3,14,14-tetramethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradec-7-yl}-acetic acid 1546664 (4R,10R,13S)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-10-benzyl-7-hydroxymethyl-3,3,14,14-tetramethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradecane-4-carboxylic acid [(R)-1-(carbamoylmethyl-carbamoyl)-2-methyl-propyl]-amide 1546665 3-(2-{[(4R,10R,13S)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-10-benzyl-7-(3H-imidazol-4-ylmethyl)-3,3,14,14-tetramethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradecane-4-carbonyl]-amino}-hexanoylamino)-succinamic acid 1546761 (S)-2-{[(4R,7S)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7-(4-iodo-benzyl)-14,14-dimethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradecane-4-carbonyl]-amino}-3-phenyl-propionic acid 1546765 (S)-2-{[(4R,7S)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7-(4-bromo-benzyl)-14,14-dimethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradecane-4-carbonyl]-amino}-3-phenyl-propionic acid 1546778 (S)-2-{[(4R,7S)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7-(4-fluoro-benzyl)-14,14-dimethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradecane-4-carbonyl]-amino}-3-phenyl-propionic acid 1546779 (S)-2-{[(4R,7S)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7-(4-chloro-benzyl)-14,14-dimethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradecane-4-carbonyl]-amino}-3-phenyl-propionic acid 1546780 (4R,7S)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7-benzyl-14,14-dimethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradecane-4-carboxylic acid 1546790 2-Amino-pentanedioic acid 5-amide 1-({1-[1-({[1-(1-carbamoyl-3-methylsulfanyl-propylcarbamoyl)-3-methyl-butylcarbamoyl]-methyl}-carbamoyl)-2-phenyl-ethylcarbamoyl]-2-phenyl-ethyl}-amide) 1547039 21-(2-Acetylamino-hexanoylamino)-7-[3-(diaminomethaniminium)-propyl]-10-(1H-indol-3-ylmethyl)-4-naphthalen-2-ylmethyl-2,5,8,11,19,22-hexaoxo-3,6,9,12,18,23-hexaaza-tricyclo[21.7.0.0*24,29*]triaconta-24(29),25,27 1547040 3-(2-Acetylamino-hexanoylamino)-17-[3-(diaminomethaniminium)-propyl]-14-(1H-indol-3-ylmethyl)-20-naphthalen-2-ylmethyl-2,5,13,16,19,22-hexaoxo-1,6,12,15,18,21-hexaaza-tricyclo[21.8.0.0*25,30*]hentriaconta-25(30),26,28-triene-11-carboxylic acid amide 1547054 Radiolabeled octreotide derivative 1547055 Radiolabeled octreotide derivative 1547058 Radiolabeled octreotide derivative 1547059 Radiolabeled octreotide derivative 1547218 Motilin 1547267 2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-N*1*-[1-(1-carbamoyl-2-methyl-propylcarbamoyl)-2-phenyl-ethyl]-succinamide 1547268 14-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-benzyl-3,8,15-trioxo-1,4,9triaza-cyclopentadecane-5-carboxylic acid amide 1547269 12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-isobutyl-3,7,13-trioxo-1,4,8triaza-cyclotridecane-5-carboxylic acid amide 1547270 14-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-benzyl-3,11,15-trioxo-1,4,10triaza-cyclopentadecane-5-carboxylic acid amide 1547271 2-{2-[2-(2-Amino-3-phenyl-propionylamino)-pentanoylamino]-3-phenyl-propionylamino}-succinamide 1547272 12,25-Bis-[2-amino-3-(4-hydroxy-phenyl)-propionylamino]-2,15-dibenzyl-3,10,13,16,23,26-hexaoxo-1,4,9,14,17,22hexaaza-cyclohexacosane-5,18-dicarboxylic acid diamide 1547282 12,25-Bis-[2-amino-3-(4-hydroxy-phenyl)-propionylamino]-2,15-dibenzyl-3,7,13,16,20,26-hexaoxo-1,4,8,14,17,21hexaaza-cyclohexacosane-5,18-dicarboxylic acid diamide 1547284 12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-benzyl-3,10,13-trioxo-1,4,9triaza-cyclotridecane-5-carboxylic acid amide 1547285 13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-3,8,14-trioxo-1,4,9triaza-cyclotetradecane-5-carboxylic acid amide 1547377 24-benzyl-16-(4-ethoxybenzyl)-25-methyl-13-[1-methyl-(1S)-propyl]perhydrodipyrido[1,2-a:1,2-d]pyrrolo[1,2-j][1,4,7,10,13,16]hexaazacyclooctadecine-6,12,15,18,23,26-hexaone 1547378 24-(1H-5-imidazolylmethyl)-13-[1-methyl-(1S)-propyl]-16-(2-naphthylmethyl)perhydrodipyrido[1,2-a:1,2-d]pyrrolo[1,2-j][1,4,7,10,13,16]hexaazacyclooctadecine-6,12,15,18,23,26-hexaone 1547379 18-(3-Amino-propyl)-15-benzyl-3-sec-butyl-6-(1H-indol-3-ylmethyl)-16-methyl-1,4,7,13,16,19-hexaaza-tricyclo[19.4.0.0*9,13*]pentacosane-2,5,8,14,17,20-hexaone 1547383 16,24-dibenzyl-13,25-dimethylperhydrodipyrido[1,2-a:1,2-d]pyrrolo[1,2-j][1,4,7,10,13,16]hexaazacyclooctadecine-6,12,15,18,23,26-hexaone 1547535 (R)-2-[(R)-2-(2-{2-[(R)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-methyl-propionylamino}-acetylamino)-3-phenyl-propionylamino]-4-methyl-pentanoic acid 1547707 cyclo(7-12) Des-AA1,5-[Tyr2,Glu7,D-Trp8,IAmp9,Lys12]-CbmSRIF 1547742 c(Cys-Ser-c(Cys-Ser-Ser-Leu-Met-Asp-Lys-Gln-Cys)-Val-Tyr-Phe-Cys)-His-Leu-Thr-Cha-Ile-Trp 1547743 c(Cys-Ser-c(Cys-Ser-Ser-Leu-Met-Asp-Lys-Gln-Cys)-Val-Tyr-Phe-Cys)-His-Leu-Thr-gamma MeLeu-Ile-Trp 1547755 (7RS,9aRS)-2-furan-2-yl-5-[7-(1H-pyrazolo[3,4-d]pyrimidin-4-yloxymethyl)-octahydropyrido[1,2-a]pyrazin-2-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-ylamine 1547860 6,10,13,14-tetramethyl-(1S,4R,13S,14R,17S)-3,18-dioxatetracyclo[11.5.0.01,17.04,17]octadeca-5,9-dien-4-ol 1547861 Sodium salt {3-[(1R,2S,6S)-1-(4,5-diphenyl-oxazol-2-yl)-7-oxa-bicyclo[4.1.0]hept-2-ylmethyl]-phenoxy}-acetate 1547867 3,4,7,11-tetramethyl-(1R,3R,4S,11S,12S,13S)-14,18-dioxatetracyclo[9.6.1.04,16.013,17]octadeca-7,16-diene-12,13-diol 1547966 Ac-YR[CEHdFRWC]SPPKD-NH2 1548442 CUDPUATUYCRFFNAFCYCRKL 1548695 cyclo(6-12) Des-AA1,5-[Tyr2,Glu6,D-Trp8,IAmp9,Dab12]SRIF 1549608 H-Dmt-Tic-Gly-NH-CH2-Bid 1590098 4-(3'-chloroanilino)-6,7-diethoxyquinazoline hydrochloride 1590212 (4-Chloro-2-fluoro-phenyl)-[6-methoxy-7-(piperidin-4-ylmethoxy)-quinazolin-4-yl]-amine hydrochloride 1590213 (4-Chloro-2-fluoro-phenyl)-[6-methoxy-7-(1-methyl-piperidin-4-ylmethoxy)-quinazolin-4-yl]-amine hydrochloride 1590214 2-Chloro-4-fluoro-5-[6-methoxy-7-(1-methyl-piperidin-4-ylmethoxy)-quinazolin-4-ylamino]-phenol hydrochloride 1590215 (4-Chloro-2-fluoro-phenyl)-[6-methoxy-7-(3-pyrrolidin-1-yl-propoxy)-quinazolin-4-yl]-amine hydrochloride 1590216 7-{4-[4-(3-chlorophenyl)-piperazin-1-yl]-butyl}-8-ethoxy-1,3-dimethyl-3,7-dihydropurine-2,6-dione hydrochloride 1590268 N-({[1-(4-Chloro-benzyl)-pyrrolidin-2-ylmethyl]-carbamoyl}-methyl)-3-trifluoromethyl-benzamide 1590313 4-amino-N-1-azatricyclo[3.3.1.0~3,7~]non-4-yl-5-chloro-2-methoxybenzamide 1591426 H-Tyr-c[D-Orn-(D or L)Atc-Glu]-NH2 1591744 3-O-(tert-Butyldimethylsilyl)-6,14-endo-etheno-7alpha-(3-carboxy-3-n-butenyl) tetrahydrooripavine gama-Lactone 1591745 (R)-1-(3-cyclopropylmethyl-11,15-dimethoxy-13-oxa-3-azahexacyclo[13.2.2.12,8.01,6.06,14.07,12]icosa-7,9,11,18-tetraen-16-yl)ethyl isothiocyanate 1591746 (S)-1-(11,15-dimethoxy-3-methyl-13-oxa-3-azahexacyclo[13.2.2.12,8.01,6.06,14.07,12]icosa-7,9,11,18-tetraen-16-yl)ethyl isothiocyanate 1591747 (R)-1-(11,15-dimethoxy-3-methyl-13-oxa-3-azahexacyclo[13.2.2.12,8.01,6.06,14.07,12]icosa-7,9,11,18-tetraen-16-yl)ethyl isothiocyanate 1591748 (S)-19-(1-isothiocyanatoethyl)-15-methoxy-3-methyl-13-oxa-3-azahexacyclo[13.2.2.12,8.01,6.06,14.07,12]icosa-7,9,11,16-tetraen-11-ol 1591749 (S)-1-(3-cyclopropylmethyl-11,15-dimethoxy-13-oxa-3-azahexacyclo[13.2.2.12,8.01,6.06,14.07,12]icosa-7,9,11,18-tetraen-16-yl)ethyl isothiocyanate 1591750 5-(3-cyclopropylmethyl-11-hydroxy-15-methoxy-13-oxa-3-azahexacyclo[13.2.2.12,8.01,6.06,14.07,12]icosa-7,9,11,18-tetraen-16-yl)-3-methylenetetrahydro-2-furanone 1591807 (3R,4S,5S)-2-(6-{[(4S)-bicyclo[2.2.1]heptan-2-yl]amino}-9H-purin-9-yl)-5-(chloromethyl)oxolane-3,4-diol 1591810 (3R,4S,5S)-2-(6-{[(1S,2R,4R)-bicyclo[2.2.1]heptan-2-yl]amino}-9H-purin-9-yl)-5-(chloromethyl)oxolane-3,4-diol 1591811 (3R,4S,5S)-2-(6-{[(2S,4S)-bicyclo[2.2.1]heptan-2-yl]amino}-9H-purin-9-yl)-5-(chloromethyl)oxolane-3,4-diol 1594201 H-Tyr-c[D-Orn-(D or L)Atc-Glu]-NH2 1594214 (R)1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-3-methoxy-propan-2-ol 1594698 3-[1-(8-Methyl-8-aza-bicyclo[3.2.1]oct-3-yl)-piperidin-4-yl]-2-phenyl-1H-indole 1594760 3-[(2-Fluoro-phenyl)-phenyl-methoxy]-8-methyl-8-aza-bicyclo[3.2.1]octane 1594761 3-[(3-Chloro-phenyl)-phenyl-methoxy]-8-methyl-8-aza-bicyclo[3.2.1]octane 1594769 8-Methyl-3-(phenyl-o-tolyl-methoxy)-8-aza-bicyclo[3.2.1]octane 1594775 3alpha-(bis-chloro-phenylmethoxy)tropane 1594782 Aminobenztropine 1594792 8-Methyl-3-[phenyl-(3-trifluoromethyl-phenyl)-methoxy]-8-aza-bicyclo[3.2.1]octane 1594798 3-[(3-Fluoro-phenyl)-phenyl-methoxy]-8-methyl-8-aza-bicyclo[3.2.1]octane 1594800 3-[Bis-(3-fluoro-phenyl)-methoxy]-8-methyl-8-aza-bicyclo[3.2.1]octane 1594801 3-[(2-Chloro-phenyl)-phenyl-methoxy]-8-methyl-8-aza-bicyclo[3.2.1]octane 1594906 4-Amino-N-(1-aza-tricyclo[3.3.1.1*3,7*]dec-4-ylmethyl)-5-chloro-2-methoxy-benzamide 1594909 8-(2-(1H-indol-3-yl)ethyl)-N-(bis(4-fluorophenyl)methyl)-8-aza-bicyclo[3.2.1]octan-3-amine 1594910 N-(bis(4-fluorophenyl)methyl)-8-methyl-8-aza-bicyclo[3.2.1]octan-3-amine 1594914 8-(2-aminoethyl)-N-(bis(4-fluorophenyl)methyl)-8-aza-bicyclo[3.2.1]octan-3-amine 1594915 N-(bis(4-chlorophenyl)methyl)-8-methyl-8-aza-bicyclo[3.2.1]octan-3-amine 1594916 N-((4-chlorophenyl)(phenyl)methyl)-8-methyl-8-aza-bicyclo[3.2.1]octan-3-amine 1594918 N-(bis(4-fluorophenyl)methyl)-8-aza-bicyclo[3.2.1]octan-3-amine 1594919 8-allyl-N-(bis(4-fluorophenyl)methyl)-8-aza-bicyclo[3.2.1]octan-3-amine 1594920 N-(bis(4-fluorophenyl)methyl)-8-butyl-8-aza-bicyclo[3.2.1]octan-3-amine 1594921 N-(bis(4-fluorophenyl)methyl)-8-(4-phenylbutyl)-8-aza-bicyclo[3.2.1]octan-3-amine 1594922 3-(3-(bis(4-fluorophenyl)methylamino)-8-aza-bicyclo[3.2.1]octan-8-yl)-N-phenylpropanamide 1594923 N-(bis(3,4-dichlorophenyl)methyl)-8-methyl-8-aza-bicyclo[3.2.1]octan-3-amine 1594924 N-(bis(4-fluorophenyl)methyl)-N,8-dimethyl-8-aza-bicyclo[3.2.1]octan-3-amine 1595151 3,4,5-trihydroxy-6-[10-methoxy-4-methyl-(5R,13R,14S,17R)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10,15-tetraen-14-yloxy]tetrahydro-2H-2-pyrancarboxylic acid 1595152 3,4,5-trihydroxy-6-[10-hydroxy-(5R,13R,14S,17R)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10,15-tetraen-14-yloxy]tetrahydro-2H-2-pyrancarboxylic acid 1595158 6-[4-allyl-10-hydroxy-(5R,13R,14S,17R)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10,15-tetraen-14-yloxy]-3,4,5-trihydroxytetrahydro-2H-2-pyrancarboxylic acid 1595166 2-[14-(6-carboxy-3,4,5-trihydroxytetrahydro-2H-2-pyranyloxy)-10-hydroxy-(5R,13R,14S,17R)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10,15-tetraen-4-yl]acetic acid 1595186 1-{(S)-1-[4-(4-Fluoro-phenyl)-butyl]-piperidin-3-ylmethyl}-3-[3-(1-methyl-1H-tetrazol-5-yl)-phenyl]-urea 1595187 1-[(S)-1-(4-Fluoro-benzyl)-piperidin-3-ylmethyl]-3-[3-(1-methyl-1H-tetrazol-5-yl)-phenyl]-urea 1595188 2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid ((R)-1-carbamoyl-4-guanidino-butyl)-amide 1595189 (R)-2-({2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl}-amino)-3-(1H-indol-3-yl)-propionic acid 1595191 (1R,6S)-5-Methyl-6-((S)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-yl)-cyclohexa-2,4-dienecarbonitrile 1595192 (5R,6R)-5-Methyl-6-((R)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-yl)-cyclohexa-1,3-dienecarbonitrile 1595195 (S)1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol-2-yl]-piperidin-1-yl}-3-methoxy-propan-2-ol 1595196 (S)-(-)-10-{4-[2-(butoxy)ethoxy]phenyl}-1-isobutyl-N-(4-{[(1-propyl-1H-imidazol-5-yl)methyl]sulfinyl}phenyl)-1,2,3,4,5,6-hexahydro-1-benzazecine-7-carboxamide 1595198 (S)-(-)-8-{4-[2-(butoxy)ethoxy]phenyl}-1-propyl-N-(4-{[(1-propyl-1H-imidazol-5-yl)methyl]sulfinyl}phenyl)-1,2,3,4-tetrahydro-1-benzazocine-5-carboxamide 1595199 (S)-(-)-8-{4-[2-(butoxy)ethoxy]phenyl}-1-isobutyl-N-(4-{[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]sulfinyl}phenyl)-1,2,3,4-tetrahydro-1-benzazocine-5-carboxamide 1595200 (S)-(-)-8-{4-[2-(butoxy)ethoxy]phenyl}-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(4-{[(1-propyl-1H-imidazol-5-yl)methyl]-sulfinyl}phenyl)-1,2,3,4-tetrahydro-1-benzazocine-5-carboxamide 1595201 (S)-(-)-8-{4-[2-(butoxy)ethoxy]phenyl}-1-propyl-N-(4-{[(4-propyl-4H-1,2,4-tri azol-3-yl)methyl]sulfinyl}phenyl)-1,2,3,4-tetrahydro-1-benzazocine-5-carboxamide 1595202 (S)-(-)-9-{4-[2-(butoxy)ethoxy]phenyl}-1-isobutyl-N-(4-{[(1-propyl-1H-imidazol-5-yl)methyl]sulfinyl}phenyl)-2,3,4,5-tetrahydro-1H-1-benzazonine-6-carboxamide 1595203 (S)-(-)-10-{4-[2-(butoxy)ethoxy]phenyl}-1-propyl-N-(4-{[(1-propyl-1H-imidazol-5-yl)methyl]sulfinyl}phenyl)-1,2,3,4,5,6-hexahydro-1-benzazecine-7-carboxamide 1595204 (S)-(-)-9-{4-[2-(butoxy)ethoxy]phenyl}-1-propyl-N-(4-{[(1-propyl-1H-imidazol-5-yl)methyl]sulfinyl}phenyl)-2,3,4,5-tetrahydro-1H-1-benzazonine-6-carboxamide 1595295 3-[2-((S)-Cyclobutylamino)-propyl]-1-(2,6-difluoro-benzyl)-5-(2-fluoro-3-methoxy-phenyl)-6-methyl-1H-pyrimidine-2,4-dione hydrochloride 1595349 H-Lys-Arg-Pro-Hyp-Gly-Igl-Ser-D-BT-OH (JMV1645) 1595399 pGlu-His-Trp-Ser-Tyr-Gly-Leu-Arg-Pro-Gly-NH2 1595419 (6S,11R)-3-cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocin-8-ol 1627140 Sulfuric acid mono-[10,13-dimethyl-3,6-bis-sulfooxy-17-(1,4,5,5-tetramethyl-hexyl)-hexadecahydro-cyclopenta[a]phenanthren-2-yl] ester with trisodium salt 1627179 (5-{1-[3-(Carboxymethyl-carbamoyl)-5-chloro-4-hydroxy-phenyl]-4-[17-(1,5-dimethyl-hexyl)-10,13-dimethyl-hexadecahydro-cyclopenta[a]phenanthren-3-yl]-but-1-enyl}-3-chloro-2-hydroxy-benzoylamino)-acetic acid 1627446 Cosalane derivative 1627449 5-{1-{3-carboxylato-4-[4-(3-carboxyphenyl)benzyloxy]-5-chlorophenyl}-4-[1-(1,5-dimethylhexyl)-9a,11a-dimethylperhydrocyclopenta[a]phenanthren-7-yl]-1-butenyl}-2-[4-(3-carboxyphenyl)benzyloxy]-3-chlorobenzoate 1627454 2-(5-{1-[3-(1-carboxy-3-methylsulfanylpropylcarbamoyl)-5-chloro-4-hydroxyphenyl]-4-[1-(1,5-dimethylhexyl)-9a,11a-dimethylperhydrocyclopenta[a]phenanthren-7-yl]-1-butenyl}-3-chloro-2-hydroxyphenylcarboxamido)-4-methylsulfanylbutanoic acid 1627461 2-(3-carboxylatobenzyloxy)-5-{1-[3-carboxylato-4-(3-carboxylatobenzyloxy)-5-chlorophenyl]-4-[1-(1,5-dimethylhexyl)-9a,11a-dimethylperhydrocyclopenta[a]phenanthren-7-yl]-1-butenyl}-3-chlorobenzoate 1627465 2-(2-carboxylatobenzyloxy)-5-{1-[3-carboxylato-4-(2-carboxylatobenzyloxy)-5-chlorophenyl]-4-[1-(1,5-dimethylhexyl)-9a,11a-dimethylperhydrocyclopenta[a]phenanthren-7-yl]-1-butenyl}-3-chlorobenzoate 1627518 Cosalane 1627768 5-{1-[3-carboxylato-5-chloro-4-(3-nitrobenzyloxy)phenyl]-4-[1-(1,5-dimethylhexyl)-9a,11a-dimethylperhydrocyclopenta[a]phenanthren-7-yl]-1-butenyl}-3-chloro-2-(3-nitrobenzyloxy)benzoate 1631657 N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[2-(2-{2-[2-(4-hydroxy-phenyl)-acetylamino]-hexanoylamino}-acetylamino)-3-(1H-indol-3-yl)-propionylamino]-6-[3-(2-methyl-benzoyl)-ureido]-hexanoylamino}-N-methyl-succinamic acid 1631664 N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[2-(2-{2-[2-(4-hydroxy-phenyl)-acetylamino]-hexanoylamino}-acetylamino)-3-(1H-indol-3-yl)-propionylamino]-6-[3-(4-hydroxy-phenyl)-acryloylamino]-hexanoylamino}-N-methyl-succinamic acid 1631682 H-Lys-Lys-Arg-Pro-Hyp-Gly-Igl-Ser-D-BT-OH (JMV1639) 1631687 H-DArg-Arg-Pro-Hyp-Gly-Thi-Ser-DTic-Oic-Arg-OH (HOE-140) 1631827 (R)-6-Acetylamino-2-({2-[2-amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl}-amino)-hexanoic acid 1632189 3-{(S)-6-[3-(4-Acetyl-phenyl)-ureido]-2-[2-tert-butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-N-(1-carbamoyl-2-phenyl-ethyl)-succinamic acid 1632190 3-{6-[3-(3-Acetyl-phenyl)-ureido]-2-[2-tert-butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-N-(1-carbamoyl-2-phenyl-ethyl)-succinamic acid 1632194 3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-6-[3-(2-nitro-phenyl)-ureido]-hexanoylamino}-N-(1-carbamoyl-2-phenyl-ethyl)-succinamic acid 1632195 4-(3-{(S)-5-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-5-[1-(1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-carboxy-ethylcarbamoyl]-pentyl}-ureido)-benzoic acid methyl ester 1632196 3-(3-{5-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-5-[1-(1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-carboxy-ethylcarbamoyl]-pentyl}-ureido)-benzoic acid methyl ester 1632197 2-(3-{5-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-5-[1-(1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-carboxy-ethylcarbamoyl]-pentyl}-ureido)-benzoic acid methyl ester 1632203 3-{(S)-2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-6-[3-(3-nitro-phenyl)-ureido]-hexanoylamino}-N-(1-carbamoyl-2-phenyl-ethyl)-succinamic acid 1632214 3-{(S)-2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-6-[3-(3-methoxy-phenyl)-ureido]-hexanoylamino}-N-(1-carbamoyl-2-phenyl-ethyl)-succinamic acid 1632215 3-{(S)-2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-6-[3-(4-methoxy-phenyl)-ureido]-hexanoylamino}-N-(1-carbamoyl-2-phenyl-ethyl)-succinamic acid 1632303 2-[2-({2-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl}-amino)-3-phenyl-propionylamino]-3-[4-(2-bromo-acetylamino)-phenyl]-propionic acid 1632306 2-{2-({2-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl}-amino)-3-[4-(2-bromo-acetylamino)-phenyl]-propionylamino}-3-phenyl-propionic acid 1632316 3-{(S)-2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-6-[3-(4-nitro-phenyl)-ureido]-hexanoylamino}-N-(1-carbamoyl-2-phenyl-ethyl)-succinamic acid 1632523 (R,R)5-[1-{1-[2-[1-amino-4-amino(imino)methylaminobutylcarboxamido]-5-amino(imino)methylaminopentanoyl]tetrahydro-1H-2-pyrrolylcarboxamido}-2-(4-hydroxyphenyl)ethylcarboxamido]-2-benzyl-6-methyl-4-oxooctanoic acid 1632535 (S,S)2-{1-[2-{1-[2-[1-amino-4-amino(imino)methylaminobutylcarboxamido]-5-amino(imino)methylaminopentanoyl]tetrahydro-1H-2-pyrrolylcarboxamido}-1-cyano-3-(4-hydroxyphenyl)propylamino]-2-methylbutylcarboxamido}-4-methylpentanoic acid 1632625 (S)-2-[(R)-5-({1-[2-(2-Amino-5-guanidino-pentanoylamino)-5-guanidino-pentanoyl]-pyrrolidine-2-carbonyl}-amino)-2-benzyl-6-(4-hydroxy-phenyl)-4-oxo-hexanoylamino]-4-methyl-pentanoic acid 1632764 Sodium salt 2-[2-{2-[(2,6-dimethyl-piperidine-1-carbonyl)-amino]-4,4-dimethyl-pentanoylamino}-3-(1-methoxymethyl-1H-indol-3-yl)-propionylamino]-hexanoate 1632766 (S,S)2-{1-[2-{1-[2-[1-amino-4-amino(imino)methylaminobutylcarboxamido]-5-amino(imino)methylaminopentanoyl]tetrahydro-1H-2-pyrrolylcarboxamido}-1-cyano-3-(4-hydroxyphenyl)propylamino]-2-methylbutylcarboxamido}-4-methylpentanoic acid 1632963 N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[3-(1H-indol-3-yl)-2-(2-{2-[2-(4-sulfooxy-phenyl)-acetylamino]-hexanoylamino}-acetylamino)-propionylamino]-6-[3-(2-methyl-benzoyl)-ureido]-hexanoylamino}-N-methyl-succinamic acid 1633012 1-{1-[4-(5-sec-Butyl-6-hydroxy-3-phenyl-1,6-dihydro-pyrazin-2-yl)-benzyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 1633013 1-{1-[4-(5-Benzyl-6-hydroxy-3-phenyl-1,6-dihydro-pyrazin-2-yl)-benzyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one 1633014 1-(1-{4-[6-Hydroxy-5-(4-hydroxy-benzyl)-3-phenyl-1,6-dihydro-pyrazin-2-yl]-benzyl}-piperidin-4-yl)-1,3-dihydro-benzoimidazol-2-one 1633047 {(S)-5-[(S)-2-({2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl}-amino)-3-phenyl-propionylamino]-5-carbamoyl-pentyl}-carbamic acid benzyl ester 1633109 H-Dmt-Tic-NH-CH[(CH2)4-NH-Z]-Bid 1633110 H-Dmt-Tic-NH-(D)-CH[(CH2)4-NH-Z]-Bid 1633111 H-Dmt-Tic-NH-CH[(CH2)4-NH-Ac]-Bid 1633112 H-Dmt-Tic-NH-CH[(CH2)4-NH2]-Bid 1633237 2-Amino-N*4*-[1-(1-{[(1-carbamoyl-3-methyl-butylcarbamoyl)-methyl]-carbamoyl}-2-phenyl-ethylcarbamoyl)-2-phenyl-ethyl]-N*1*-(2-{2-[4-(2,6-dioxo-1,3-dipropyl-2,3,4,5,6,7-hexahydro-1H-purin-8-yl)-phenoxy]-acetylamino}-ethyl)-succinamide-4-Methylsulfanyl-butyramide 1633273 5-Hydroxymethyl-2-methyl-2-[6-(1-methyl-2-phenyl-ethylamino)-purin-9-yl]-tetrahydro-furan-3,4-diol 1633274 xv5-Hydroxymethyl-2-methyl-2-[6-(1-methyl-2-phenyl-ethylamino)-purin-9-yl]-tetrahydro-furan-3,4-diol 1633275 (2R,3S,5R)-2-(6-Amino-purin-9-yl)-5-hydroxymethyl-2-methyl-tetrahydro-furan-3,4-diol 1633276 2-(6-Cyclopentylamino-purin-9-yl)-5-hydroxymethyl-2-methyl-tetrahydro-furan-3,4-diol 1633382 2-(2-{2-[2-(2-{4-[9-(3,4-Dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-6-ylamino]-phenyl}-acetylamino)-3-phenyl-propionylamino]-3-phenyl-propionylamino}-acetylamino)-4-methyl-pentanoic acid (1-carbamoyl-3-methylsulfanyl-propyl)-amide 1633570 Radiolabeled octreotide derivative 1633571 Radiolabeled octreotide derivative 1633572 Radiolabeled octreotide derivative 1633575 Radiolabeled octreotide derivative 1633576 Radiolabeled octreotide derivative 1633577 Radiolabeled octreotide derivative 1633578 Radiolabeled octreotide derivative 1633646 oxymorphone N-(Hydrazinocarbonyl)phenylalanyl-leucylarginylarginylisoleucine methyl ester hydrochloride 1633647 Naltrexone N-(Hydrazinocarbonyl)phenylalanyl-leucylarginylarginylisoleucine methyl ester hydrochloride 1633859 [2-{2-[1-{[2-(2,4-Dichloro-phenyl)-2-imidazol-1-ylmethyl-[1,3]dioxolan-4-ylmethyl]-carbamoyl}-2-(2,3-dihydro-1H-imidazol-4-yl)-ethylcarbamoyl]-pyrrolidin-1-yl}-1-(1H-indol-3-ylmethyl)-2-oxo-ethyl]-carbamic acid tert-butyl ester 1633860 2-[1-{[2-(2,4-Dichloro-phenyl)-2-imidazol-1-ylmethyl-[1,3]dioxolan-4-ylmethyl]-carbamoyl}-2-(2,3-dihydro-1H-imidazol-4-yl)-ethylcarbamoyl]-pyrrolidine-1-carboxylic acid 2,2-diphenyl-ethyl ester 1633861 2-[1-{[2-(2,4-Dichloro-phenyl)-2-imidazol-1-ylmethyl-[1,3]dioxolan-4-ylmethyl]-carbamoyl}-2-(1H-imidazol-4-yl)-ethylcarbamoyl]-5-oxo-pyrrolidine-1-carboxylic acid benzyl ester 1704319 (S)-4-Methyl-piperazine-2-carboxylic acid [(S)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide dihydrochloride 1704359 N5-(3-(9H-Purin-6-yl)pyridin-2-yl)-N1-(4-chlorophenyl)-6-methylisoquinoline-1,5-diamine dihydrochloride 1704526 1-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-4-(3-phenyl-allyl)-piperazine; Dihydrochloride 1704956 (R)-4-Methyl-piperazine-2-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide dihydrochloride 1705170 (S)-1-Methyl-piperazine-2-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide dihydrochloride 1726337 (3S,4aR,6S,8R,8aR)-6-Ethylcarbamoyloxy-3-furan-3-yl-4a,8a-dimethyl-1,5-dioxo-dodecahydro-2-oxa-phenanthrene-8-carboxylic acid methyl ester 1797172 (2R)-5-carbamimidamido-N-[(1S)-1-carbamoyl-2-(1H-indol-3-yl)ethyl]-2-[(2S)-2-[(2S)-3-(4H-imidazol-4-yl)-2-[4-(1-{6-[(3,7,14,18,22-pentahydroxy-2,6,10,15,19,23-hexamethyltetracosan-11-yl)oxy]hexyl}-1H-1,2,3-triazol-4-yl)butanamido]propanamido]-3-phenylpropanamido]pentanamide 1797641 H-Tyr-Val-DMet-Gly-His-Phe-Arg-Trp-Asp-Arg-Phe-Gly-OH 1797653 7-(3-Hexylsulfanylmethyl-7-oxa-bicyclo[2.2.1]hept-2-yl)-hept-5-enoic acid 1798072 3-[14-(1H-Indol-3-ylmethyl)-11-isobutyl-8-isopropyl-5-methyl-3,6,9,12,15-pentaoxo-1,4,7,10,13pentaaza-cyclopentadec-2-yl]-propionic acid 1798506 8-(tert-butyl)-6,9,12,17-tetrahydroxy-16-methyl-(6R,8R,9R,12R,16S,17R)-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,15,18-trione 1798590 (3S,4aR,6S,8R,8aR)-6-Carbamoyloxy-3-furan-3-yl-4a,8a-dimethyl-1,5-dioxo-dodecahydro-2-oxa-phenanthrene-8-carboxylic acid methyl ester 1798591 (3S,4aR,6S,8R,8aR)-6-Butoxy-3-furan-3-yl-4a,8a-dimethyl-1,5-dioxo-dodecahydro-2-oxa-phenanthrene-8-carboxylic acid methyl ester 1798594 (3S,4aR,6S,8R,8aR)-3-Furan-3-yl-4a,8a-dimethyl-6-methylcarbamoyloxy-1,5-dioxo-dodecahydro-2-oxa-phenanthrene-8-carboxylic acid methyl ester 1798595 (3S,4aR,6S,8R,8aR)-6-Allyloxy-3-furan-3-yl-4a,8a-dimethyl-1,5-dioxo-dodecahydro-2-oxa-phenanthrene-8-carboxylic acid methyl ester 1798598 (3S,4aR,6S,8R,8aR)-6-Benzyloxy-3-furan-3-yl-4a,8a-dimethyl-1,5-dioxo-dodecahydro-2-oxa-phenanthrene-8-carboxylic acid methyl ester 1798648 Octreotide 1798871 5-(3-Hydroxy-phenyl)-2-methyl-8-[1-phenyl-meth-(E)-ylidene]-2-aza-bicyclo[3.3.1]nonan-7-one 1798942 3-(2-Amino-3-phenyl-propionylamino)-N-{1-[1-tert-butoxycarbonyl-2-(1H-indol-3-yl)-ethylcarbamoyl]-pentyl}-succinamic acid 1798973 2-[2-(2-{2-[2-(2-{2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-6-amino-hexanoylamino}-3-carboxy-propionylamino)-3-cyclohexyl-propionylamino]-3-cyclohexyl-propionylamino}-3-methyl-butyrylamino)-propionylamino]-5-guanidino-pentanoic acid 1798998 N-(bis(4-fluorophenyl)methyl)-8-methyl-8-aza-bicyclo[3.2.1]octan-3-amine 1799103 (E)-3-[6-Amino-9-((3S,4R,5R)-3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-8-yl]-1-phenyl-propenone 1799104 (3S,4R,5R)-2-(6-Amino-8-phenylethynyl-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol 1799319 2-(2-{2-[(2R)-2-[(2S)-2-(2-{6-amino-2-[2-acetamido-3-(1H-imidazol-4-yl)propanamido]hexanamido}-3-carboxypropanamido)-3-cyclohexylpropanamido]-3-cyclohexylpropanamido]-4-methylpentanamido}propanamido)-5-[(diaminomethylidene)amino]pentanoic acid 1799321 2-[2-(2-{2-[2-(2-{2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-6-amino-hexanoylamino}-3-carboxy-propionylamino)-3-cyclohexyl-propionylamino]-3-cyclohexyl-propionylamino}-pentanoylamino)-propionylamino]-5-guanidino-pentanoic acid 1799322 2-[2-(2-{2-[2-(2-{2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-6-amino-hexanoylamino}-3-carboxy-propionylamino)-3-cyclohexyl-propionylamino]-3-cyclohexyl-propionylamino}-3-methyl-pentanoylamino)-propionylamino]-5-guanidino-pentanoic acid 1799324 2-[2-(2-{2-[2-(2-{2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-6-amino-hexanoylamino}-3-carboxy-propionylamino)-3-cyclohexyl-propionylamino]-3-cyclohexyl-propionylamino}-3-cyclohexyl-propionylamino)-propionylamino]-5-guanidino-pentanoic acid 1799325 2-[2-(2-{2-[2-(2-{2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-6-amino-hexanoylamino}-3-carboxy-propionylamino)-3-cyclohexyl-propionylamino]-3-cyclohexyl-propionylamino}-4-methyl-pentanoylamino)-propionylamino]-5-guanidino-pentanoic acid 1799326 2-[2-(2-{2-[2-(2-{2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-6-amino-hexanoylamino}-3-carboxy-propionylamino)-3-phenyl-propionylamino]-3-phenyl-propionylamino}-3-phenyl-propionylamino)-propionylamino]-5-guanidino-pentanoic acid 1799456 [1-(2-Benzyl-1-oxo-3-thioxo-octahydro-4a(R)-pyrido[1,2-c]pyrimidin-5(S)-ylcarbamoyl)-2-(1H-indol-3-yl)-ethyl]-carbamic acid tert-butyl ester 1799459 [1-(2-Benzyl-1,3-dithioxo-octahydro-4a(R)-pyrido[1,2-c]pyrimidin-5(S)-ylcarbamoyl)-2-(1H-indol-3-yl)-ethyl]-carbamic acid tert-butyl ester 1799460 [1-(2-Benzyl-1,3-dithioxo-octahydro-4a(S)-pyrido[1,2-c]pyrimidin-5(R)-ylcarbamoyl)-2-(1H-indol-3-yl)-ethyl]-carbamic acid tert-butyl ester 1799462 [1-(2-Benzyl-1-oxo-3-thioxo-octahydro-4a(S)-pyrido[1,2-c]pyrimidin-5(R)-ylcarbamoyl)-2-(1H-indol-3-yl)-ethyl]-carbamic acid tert-butyl ester 1799463 [1-(2-Benzyl-3-methoxy-1-oxo-octahydro-4a(S)-pyrido[1,2-c]pyrimidin-5(R)-ylcarbamoyl)-2-(1H-indol-3-yl)-ethyl]-carbamic acid tert-butyl ester 1799465 [1-(2-Benzyl-3-oxo-1-thioxo-octahydro-4a(S)-pyrido[1,2-c]pyrimidin-5(R)-ylcarbamoyl)-2-(1H-indol-3-yl)-ethyl]-carbamic acid tert-butyl ester 1799466 [1-(2-Benzyl-3-oxo-1-thioxo-octahydro-4a(R)-pyrido[1,2-c]pyrimidin-5(S)-ylcarbamoyl)-2-(1H-indol-3-yl)-ethyl]-carbamic acid tert-butyl ester 1799525 7-(3-Hexylsulfanylmethyl-7-oxa-bicyclo[2.2.1]hept-2-yl)-hept-5-enoic acid 1799657 3-(2-Amino-3-naphthalen-1-yl-propionylamino)-N-{1-[1-tert-butoxycarbonyl-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-phenyl-ethyl}-succinamic acid 1799658 N-(1-{[1-tert-Butoxycarbonyl-2-(1H-indol-3-yl)-ethyl]-methyl-carbamoyl}-pentyl)-3-(2-methylamino-3-naphthalen-1-yl-propionylamino)-succinamic acid 1799660 3-(2-Amino-3-naphthalen-1-yl-propionylamino)-N-(1-{[1-tert-butoxycarbonyl-2-(1H-indol-3-yl)-ethyl]-methyl-carbamoyl}-pentyl)-succinamic acid 1799661 3-(2-Amino-3-naphthalen-2-yl-propionylamino)-N-(1-{[1-tert-butoxycarbonyl-2-(1H-indol-3-yl)-ethyl]-methyl-carbamoyl}-pentyl)-succinamic acid 1799662 3-(2-Amino-3-naphthalen-1-yl-propionylamino)-N-{[1-tert-butoxycarbonyl-2-(1H-indol-3-yl)-ethylcarbamoyl]-phenyl-methyl}-succinamic acid 1799663 N-{[1-tert-Butoxycarbonyl-2-(1H-indol-3-yl)-ethylcarbamoyl]-cyclohexyl-methyl}-3-(2-dimethylamino-3-naphthalen-1-yl-propionylamino)-succinamic acid 1799664 N-{[1-tert-Butoxycarbonyl-2-(1H-indol-3-yl)-ethylcarbamoyl]-phenyl-methyl}-3-(2-dimethylamino-3-naphthalen-1-yl-propionylamino)-succinamic acid 1799665 3-(2-Amino-3-naphthalen-1-yl-propionylamino)-N-{[1-tert-butoxycarbonyl-2-(1H-indol-3-yl)-ethylcarbamoyl]-cyclohexyl-methyl}-succinamic acid 1799666 N-(1-{[1-tert-Butoxycarbonyl-2-(1H-indol-3-yl)-ethyl]-methyl-carbamoyl}-pentyl)-3-(2-dimethylamino-3-naphthalen-1-yl-propionylamino)-succinamic acid 1799667 3-(2-Amino-3-naphthalen-1-yl-propionylamino)-N-({[1-tert-butoxycarbonyl-2-(1H-indol-3-yl)-ethyl]-methyl-carbamoyl}-phenyl-methyl)-succinamic acid 1799668 3-(2-Amino-3-naphthalen-1-yl-propionylamino)-N-(1-{[1-tert-butoxycarbonyl-2-(1H-indol-3-yl)-ethyl]-methyl-carbamoyl}-2-phenyl-ethyl)-succinamic acid 1799669 3-(2-Amino-3-naphthalen-1-yl-propionylamino)-N-(1-{[1-tert-butoxycarbonyl-2-(1H-indol-3-yl)-ethyl]-methyl-carbamoyl}-pentyl)-succinamic acid 1799712 (-)-(2S,2'R,3'S,5'R)-1-methyl-2-(2-methyl-1,3-oxathiolan-5-yl)pyrrolidine 3-oxide 1826117 N-(2,6-dimethylphenyl)-5-[5-(4-methylpiperazin-1-ylmethyl)thiophen-2-yl]imidazo[1,5-a]pyrazin-8-amine hydrochloride 1826138 N-(2,6-dimethylphenyl)-5-(5-pyrrolidin-1-ylmethylthiophen-2-yl)imidazo[1,5-a]pyrazin-8-amine 1826197 2,6-Dimethyl-4-(4-nitro-phenyl)-pyridine-3,5-dicarboxylic acid 3-[3-(4,4-diphenyl-piperidin-1-yl)-propyl] ester 5-methyl ester 1826198 5-[3-(4,4-Diphenyl-piperidin-1-yl)-propylcarbamoyl]-2,6-dimethyl-4-(3-nitro-phenyl)-nicotinic acid methyl ester 2038609 3-(5-Trifluoromethyl-cyclohexa-1,3-dienyl)-pyrrolidine 2038747 (Z)-7-[(1R,2S,5R)-2-(4a,5-Dihydro-quinoline-8-sulfonylamino)-5-fluoro-cyclopentyl]-hept-5-enoic acid 2038772 1,3-Diamino-6-hydroxy-9,9a-dihydro-4aH-xanthene-2-carbonitrile 2038773 1,3-Diamino-7-hydroxy-9,9a-dihydro-4aH-xanthene-2-carbonitrile 2038774 3-Amino-6,7-dihydroxy-1-propylamino-9,9a-dihydro-4aH-xanthene-2-carbonitrile 2038775 3-Amino-1-ethylamino-6,7-dihydroxy-9,9a-dihydro-4aH-xanthene-2-carbonitrile 2038776 1,3-Diamino-6,7-dimethoxy-9,9a-dihydro-4aH-xanthene-2-carbonitrile 2038777 1,3-Diamino-5-hydroxy-9,9a-dihydro-4aH-xanthene-2-carbonitrile 2038779 8,10-Diamino-2,3,10a,11-tetrahydro-6aH-1,4,6-trioxa-naphthacene-9-carbonitrile 2038780 1,3,7-Triamino-9,9a-dihydro-4aH-xanthene-2-carbonitrile 2038781 1,3-Diamino-9,9a-dihydro-4aH-xanthene-2-carbonitrile 2038782 1,3-Diamino-6-[1,4]dioxan-2-yl-7-hydroxy-9,9a-dihydro-4aH-xanthene-2-carbonitrile 2038783 1,3-Diamino-6,8-dihydroxy-9,9a-dihydro-4aH-xanthene-2-carbonitrile 2038784 1,3-Diamino-6-ethoxy-7-hydroxy-9,9a-dihydro-4aH-xanthene-2-carbonitrile 2038785 1,3-Diamino-5,6-dihydroxy-9,9a-dihydro-4aH-xanthene-2-carbonitrile 2038787 1,3-Diamino-6,7-dihydroxy-9,9a-dihydro-4aH-xanthene-2-carbonitrile 2038788 1,3-Diamino-6-(pyrrolidin-1-ylmethoxy)-9,9a-dihydro-4aH-xanthene-2-carbonitrile 2038789 3-Amino-6,7-dihydroxy-1-(2-hydroxy-ethylamino)-9,9a-dihydro-4aH-xanthene-2-carbonitrile 2038790 2-(1,3-Diamino-2-cyano-7-methoxy-9,9a-dihydro-4aH-xanthen-9-yl)-malononitrile 2038791 2-(1,3-Diamino-7-bromo-2-cyano-9,9a-dihydro-4aH-xanthen-9-yl)-malononitrile 2038792 2-(1,3-Diamino-2-cyano-7-hydroxy-9,9a-dihydro-4aH-xanthen-9-yl)-malononitrile 2038794 2-(1,3-Diamino-2-cyano-6-methoxy-9,9a-dihydro-4aH-xanthen-9-yl)-malononitrile 2038795 2-(1,3-Diamino-2-cyano-6-hydroxy-9,9a-dihydro-4aH-xanthen-9-yl)-malononitrile 2038803 4-{2-[4-(3-Oxo-3,4-dihydro-2H-benzo[1,4]oxazin-6-yloxy)-piperidin-1-yl]-ethoxy}-3a,7a-dihydro-1H-indole-2-carbonitrile 2038816 1-(3a,7a-Dihydro-1H-indazol-6-yl)-3-{(1R,2S)-2-[(S)-3-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-urea 2038817 1-(2,3-Dimethyl-3a,7a-dihydro-1H-indol-6-yl)-3-{(1R,2S)-2-[(S)-3-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-urea 2038818 1-(3a,4-Dihydro-1H-benzoimidazol-5-yl)-3-{(1R,2S)-2-[(S)-3-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-urea 2038819 1-(3a,7a-Dihydro-1H-indol-6-yl)-3-{(1R,2S)-2-[(S)-3-(4-fluoro-benzyl)-piperidin-1-ylmethyl]-cyclohexyl}-urea 2038820 2-(Allyloxy)-5-{[6-methoxy-7-(3-pyrrolidin-1-ylpropoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 2038821 2-{[6-Methoxy-7-(3-pyrrolidin-1-ylpropoxy)quinazolin-4-yl]amino}-5-[(1-methylprop-2-yn-1-yl)oxy]benzo-1,4-quinone 2038822 2-{[6-Methoxy-7-(3-pyrrolidin-1-ylpropoxy)quinazolin-4-yl]amino}-5-[(1-phenylprop-2-yn-1-yl)oxy]benzo-1,4-quinone 2038823 2-{[6-Methoxy-7-(3-pyrrolidin-1-ylpropoxy)quinazolin-4-yl]amino}-5-(prop-2-yn-1-yloxy)benzo-1,4-quinone 2038824 2-Bromo-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 2038825 2-{[6-Methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-5-(2-phenoxyethoxy)benzo-1,4-quinone 2038826 2-{[6-Methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-5-pyrrolidin-1-ylbenzo-1,4-quinone 2038827 2,3-Dichloro-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 2038828 2-Chloro-3-methoxy-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 2038829 3-Chloro-2-[(3-fluorobenzyl)oxy]-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 2038830 2-{[6-Methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-5-[methyl(phenyl) amino] benzo-1,4-quinon 2038831 2-methoxy-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 2038832 2-[2-Fluoro-1-(fluoromethyl)ethoxy]-5-({6-methoxy-7-[(1-methylpiperidin-4-yl)methoxy]quinazolin-4-yl}amino)benzo-1,4-quinone 2038833 2-chloro-5-methoxy-3-{[6-methoxy-7-(2-methoxyethoxy)-quinazolin-4-yl]amino}benzo-1,4-quinone 2038835 2-Bromo-6-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 2038836 2-{[6-Methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-5-(methylthio)benzo-1,4-quinone 2038837 2-{[6-Methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-5-(2-methylaziridin-1-yl)benzo-1,4-quinone 2038838 2-Chloro-3-isopropoxy-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 2038839 2-{[6-Methoxy-7-(2-methoxyethoxy)-4-quinazolinyl]amino}-5-methylbenzo-1,4-quinone 2038840 2,3-dimethoxy-5-{[6-methoxy-7-(2-methoxyethoxy)-quinazolin-4-yl]amino}benzo-1,4-quinone 2038841 2-(2,2-Difluoroethoxy)-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 2038842 2-(Benzyloxy)-5-{[6-methoxy-7-(3-pyrrolidin-1-ylpropoxy)quinazolin-4-yl]amino}benzo-1,4-quinone 2038843 2-{[6-Methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-5-[(3-phenylprop-2-yn-1-yl)oxy]benzo-1,4-quinone 2038845 2-{[-6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-5-(5-methyl-2-oxo-1,3-oxazolidin-3-yl)benzo-1,4-quinone 2038846 2-{[6-Methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-5-[(pentafluorobenzyl)oxy]benzo-1,4-quinone 2038847 2-{[6-Methoxy-7-(3-pyrrolidin-1-ylpropoxy)quinazolin-4-yl]amino}-5-[(penta fluorobenzyl)oxy]benzo-1,4-quinone 2038848 2-{[6-Methoxy-7-(3-pyrrolidin-1-ylpropoxy)quinazolin-4-yl]amino}-5-[(3-phenylprop-2-yn-1-yl)oxy]benzo-1,4-quinone 2038849 2-(Benzyloxy)-5-({6-methoxy-7-[(1-methylpiperidin-4-yl)methoxy]quinazolin-4-yl}amino)benzo-1,4-quinone 2038929 (1S)-1-(2-((S)-4-(6-fluoronaphthalen-1-yl)-2-methylpiperazin-1-yl)ethyl)-1,3,7,7a-tetrahydroisobenzofuran-5-carboxamide 2038930 (1R)-1-(2-((S)-4-(6-fluoronaphthalen-1-yl)-2-methylpiperazin-1-yl)ethyl)-1,3,7,7a-tetrahydroisobenzofuran-5-carboxamide 2038931 (1R)-1-(2-((S)-4-(6-cyanonaphthalen-1-yl)-2-methylpiperazin-1-yl)ethyl)-1,3,7,7a-tetrahydroisobenzofuran-5-carboxamide 2486446 cyclo(7-12) Des-AA1,5-[Tyr2,Glu7,D-Trp8,IAmp9,Dab(Gaba)12]SRIF 2486448 cyclo(7-12) Des-AA1,5-[Tyr2,Glu7,D-Trp8,IAmp9,D-hhLys12]SRIF